Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg Int. Strength Num Of Links Community ConSurf
1A:A:V34 4.91615
2A:A:L36 4.09417
3A:A:L37 4.442519
4A:A:K46 5.862519
5A:A:I184 4.5475419
6A:A:F189 6.91419
7A:A:F191 6.685415
8A:A:F196 6.88333617
9A:A:K197 7.58416
10A:A:M198 4.1825417
11A:A:F199 7.962515
12A:A:D200 3.205419
13A:A:V201 4.912519
14A:A:Q204 3.90667619
15A:A:S206 3.195418
16A:A:E207 8.8875419
17A:A:R208 4.8525419
18A:A:K210 6.248519
19A:A:W211 4.87719
20A:A:I212 3.246518
21A:A:H213 7.4025418
22A:A:C214 3.6375417
23A:A:F215 5.24819
24A:A:E216 4.3425417
25A:A:A220 2.055418
26A:A:I221 3.832518
27A:A:F223 4.146519
28A:A:L227 6.5375417
29A:A:Y230 5.37875818
30A:A:D231 7.955419
31A:A:M243 3.1225418
32A:A:H244 4.0125414
33A:A:M247 3.8475416
34A:A:F250 6.51333619
35A:A:C254 4.095615
36A:A:W258 4.915615
37A:A:F259 4.59714719
38A:A:T262 3.1425417
39A:A:S263 3.2125417
40A:A:I264 3.324516
41A:A:I265 2.705618
42A:A:L266 3.132519
43A:A:F267 3.53429719
44A:A:F274 5.156519
45A:A:S281 4.375417
46A:A:P282 4.2725415
47A:A:L283 4.4975407
48A:A:C286 4.09516
49A:A:Y287 6.37143717
50A:A:Y290 7.525407
51A:A:I303 4.426517
52A:A:Q304 6.68415
53A:A:F307 4.45333618
54A:A:N311 5.7875418
55A:A:I319 4.192515
56A:A:Y320 5.555817
57A:A:F323 3.954514
58A:A:N331 7.4725418
59A:A:F334 5.44513
60A:A:F336 5.25518
61A:A:V339 3.894518
62A:A:V342 2.5225417
63A:A:I344 2.9925426
64A:A:L348 3.25429
65A:A:C351 2.88833624
66A:A:L353 4.138527
67B:B:L14 4.5525408
68B:B:L30 4.305405
69B:B:T34 4.45415
70B:B:I37 3.92502
71B:B:V40 3.83143713
72B:B:I43 3.38413
73B:B:M45 4.152514
74B:B:R48 5.10667617
75B:B:L51 7.7419
76B:B:H54 7.98857719
77B:B:I58 3.436519
78B:B:Y59 7.445618
79B:B:M61 3.98833616
80B:B:W63 6.04143717
81B:B:L70 5.748515
82B:B:V71 4.22518
83B:B:S72 5.4975419
84B:B:S74 6.57419
85B:B:D76 5.602519
86B:B:L79 3.28714717
87B:B:I80 9.63418
88B:B:I81 4.8617
89B:B:W82 10.4067619
90B:B:S84 3.6725415
91B:B:N88 4.34754107
92B:B:K89 5.60667619
93B:B:H91 6.295415
94B:B:I93 6.036517
95B:B:L95 4.874518
96B:B:W99 8.37429719
97B:B:C103 2.6075418
98B:B:Y105 4.46429716
99B:B:A106 3.36416
100B:B:S108 4.59416
101B:B:N110 6.8575414
102B:B:Y111 7.074514
103B:B:V112 3.28418
104B:B:A113 2.135619
105B:B:C114 3.505618
106B:B:G115 2.8175419
107B:B:G116 1.8125419
108B:B:L117 3.41429719
109B:B:I120 3.625416
110B:B:C121 2.80167618
111B:B:S122 3.456518
112B:B:I123 3.39716
113B:B:Y124 5.49429716
114B:B:E130 2.8775473
115B:B:L139 4.766509
116B:B:H142 5.98125819
117B:B:G144 2.5675418
118B:B:Y145 4.25875818
119B:B:L146 2.99667617
120B:B:C148 3.065416
121B:B:C149 2.855618
122B:B:F151 4.865619
123B:B:L152 3.134513
124B:B:D154 6.24416
125B:B:Q156 5.16405
126B:B:I157 3.29429717
127B:B:V158 3.3515
128B:B:T159 4.42571719
129B:B:S160 3.536516
130B:B:S161 7.69419
131B:B:D163 6.358519
132B:B:T165 4.184517
133B:B:C166 3.09167618
134B:B:A167 3.965414
135B:B:L168 4.99667616
136B:B:W169 10.252518
137B:B:I171 4.46416
138B:B:Q176 6.866514
139B:B:T178 5.745414
140B:B:F180 6.33286717
141B:B:H183 7.10714719
142B:B:G185 1.705415
143B:B:D186 6.48667619
144B:B:V187 3.808519
145B:B:L190 3.35515
146B:B:L192 3.33415
147B:B:F199 6.47333619
148B:B:V200 5.25536
149B:B:S201 3.68519
150B:B:C204 7.2517
151B:B:D205 5.936519
152B:B:S207 4.0575415
153B:B:A208 2.005436
154B:B:K209 9.375616
155B:B:L210 5.114505
156B:B:W211 8.225618
157B:B:D212 6.8625419
158B:B:V213 4.375614
159B:B:R214 4.4375409
160B:B:E215 5.6325413
161B:B:C218 4.51415
162B:B:R219 6.015415
163B:B:Q220 6.914537
164B:B:F222 5.63538
165B:B:H225 7.025839
166B:B:I229 5.11437
167B:B:I232 3.48167638
168B:B:F234 6.1975435
169B:B:F235 6.44429716
170B:B:P236 5.6675417
171B:B:N237 5.74415
172B:B:F241 4.98375836
173B:B:T243 5.15638
174B:B:S245 6.565439
175B:B:D247 6.536539
176B:B:T249 5.09636
177B:B:C250 2.93167618
178B:B:R251 11.338538
179B:B:F253 6.82167636
180B:B:D254 5.1975409
181B:B:R256 9.955409
182B:B:D258 8.9225437
183B:B:Q259 4.3475456
184B:B:E260 9.5525436
185B:B:L261 3.136555
186B:B:T263 5.6431
187B:B:Y264 5.16667615
188B:B:H266 3.5025414
189B:B:I269 3.092514
190B:B:C271 3.83415
191B:B:I273 5.9575416
192B:B:S275 3.9225418
193B:B:V276 1.7716
194B:B:F278 5.84667617
195B:B:S279 3.7475419
196B:B:R283 5.75857719
197B:B:L284 3.386515
198B:B:L285 5.1516
199B:B:L286 4.81417
200B:B:A287 2.07516
201B:B:G288 2.7925417
202B:B:Y289 6.41286717
203B:B:D290 6.9825416
204B:B:D291 6.0975418
205B:B:N293 5.2125415
206B:B:C294 3.03515
207B:B:N295 6.462516
208B:B:W297 6.16571718
209B:B:D298 6.082519
210B:B:L300 3.98833616
211B:B:K301 5.315405
212B:B:R304 8.3525415
213B:B:V307 3.99413
214B:B:H311 7.255619
215B:B:R314 12.348518
216B:B:V315 3.132517
217B:B:C317 2.545417
218B:B:L318 3.77833616
219B:B:T321 8.415417
220B:B:D323 6.89417
221B:B:M325 4.792515
222B:B:V327 5.01516
223B:B:W332 11.08819
224B:B:D333 6.485419
225B:B:L336 3.776517
226B:B:K337 8.125416
227B:B:I338 2.88571715
228B:B:W339 7.19625819
229G:G:R27 4.955408
230G:G:V30 3.0425458
231G:G:Y40 6.5475416
232G:G:D48 6.372519
233G:G:L50 3.428519
234G:G:L51 3.614516
235G:G:N59 6.08619
236G:G:P60 8.1425419
237G:G:F61 4.97778918
238L:L:V21 4.74420
239L:L:Q25 5.85167620
240L:L:S26 3.58400
241L:L:I39 4.368520
242L:L:C41 5.05420
243L:L:Y46 7.57520
244L:L:F48 6.358520
245L:L:Y51 9.5925420
246L:L:Y52 7.934520
247L:L:I53 3.044520
248L:L:W55 5.865820
249L:L:K57 6.272520
250L:L:Q62 3.9775420
251L:L:L64 8.7525420
252L:L:I67 4.395420
253L:L:F69 4.874520
254L:L:N71 6.138520
255L:L:P72 5.632520
256L:L:G73 3.1375420
257L:L:S74 4.725420
258L:L:H76 3.9075420
259L:L:N80 3.3425420
260L:L:F83 5.452520
261L:L:V91 2.7875420
262L:L:A98 2.3375420
263L:L:F99 4.7154130
264L:L:M100 8.3925420
265L:L:L102 3.028520
266L:L:I112 2.7420
267L:L:Y113 5.675620
268L:L:Y114 7.4125420
269L:L:C115 5.182520
270L:L:R117 14.536520
271L:L:L123 3.4375420
272L:L:R124 10.57420
273L:L:I125 4.9425420
274L:L:I126 5.1975420
275L:L:K128 7.8825420
276L:L:F129 5.856520
277L:L:W132 5.45429720
278L:L:V136 4.175400
279L:L:V140 3.76754120
280N:N:T289 5.798520
281N:N:L291 3.31833620
282N:N:Q293 4.87667620
283N:N:V305 3.1490
284N:N:I307 5.2775400
285N:N:C309 4.425420
286N:N:Y318 6.758520
287N:N:I319 4.914520
288N:N:H320 4.112520
289N:N:W321 5.44667620
290N:N:Y322 6.182520
291N:N:Q323 5.514520
292N:N:Q329 4.8725420
293N:N:P330 6.135420
294N:N:Y335 9.615420
295N:N:L340 2.955400
296N:N:E341 7.5975420
297N:N:V344 2.9475420
298N:N:F348 4.2325420
299N:N:L359 5.83520
300N:N:I361 4.52400
301N:N:N371 5.16420
302N:N:Y372 4.83620
303N:N:Y373 5.466520
304N:N:C374 4.505620
305N:N:Q375 8.7525420
306N:N:Q376 6.2420
307N:N:E379 5.1575420
308N:N:P381 2.4075400
309N:N:Y382 8.63420
310N:N:F384 6.445420
311N:N:G387 3.645420
312R:R:P33 9.0925445
313R:R:F35 6.266545
314R:R:H36 11.51548
315R:R:F38 4.0775425
316R:R:D42 5.42527
317R:R:E44 4.4975424
318R:R:H46 7.708524
319R:R:W53 7.85857722
320R:R:M57 3.4425425
321R:R:H60 7.182528
322R:R:F64 5.57407
323R:R:N71 5.778509
324R:R:L75 1.8625407
325R:R:F78 6.572506
326R:R:Y91 6.048527
327R:R:L95 5.18429
328R:R:T98 4.76628
329R:R:V102 4.23426
330R:R:L106 5.7125428
331R:R:R109 7.61526
332R:R:F110 10.01527
333R:R:Y113 6.986526
334R:R:Y114 7.395422
335R:R:H126 5.444526
336R:R:Y130 5.472526
337R:R:F131 5.06333625
338R:R:L132 4.216505
339R:R:N133 4.846528
340R:R:M134 5.90167627
341R:R:H135 7.425428
342R:R:C136 4.305426
343R:R:I138 6.95428
344R:R:F140 6.49857727
345R:R:T142 2.7525408
346R:R:D147 5.032528
347R:R:R148 4.898529
348R:R:Y149 10.21628
349R:R:L150 6.355426
350R:R:I152 2.57427
351R:R:R159 4.772525
352R:R:R160 6.5575424
353R:R:W175 4.822529
354R:R:T182 3.944526
355R:R:L200 5.75425
356R:R:E204 6.135425
357R:R:F205 7.388529
358R:R:P208 2.9275409
359R:R:I219 3.61527
360R:R:M220 4.0325424
361R:R:L229 2.2675412
362R:R:R235 6.17833615
363R:R:L243 4.435427
364R:R:F250 6.152529
365R:R:C253 2.6425427
366R:R:F254 4.96857729
367R:R:F257 6.498526
368R:R:H258 7.854528
369R:R:R260 6.33404
370R:R:Q261 4.2275406
371R:R:W267 4.2975402
372R:R:M270 3.3925163
373R:R:L276 4.3525424
374R:R:Y279 6.16143725
375R:R:H280 6.774525
376R:R:T284 4.41425
377R:R:S287 3.4075427
378R:R:D293 5.555629
379R:R:P294 2.97429
380R:R:Y297 5.77667629
381R:R:F304 4.96408
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Int. Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.

Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1B:B:S316 B:B:W332 13.56554.94NoYes099
2B:B:C317 B:B:S316 13.48851.72YesNo079
3A:A:W258 B:B:W332 13.52484.69YesYes159
4A:A:I212 A:A:W258 37.63552.35YesYes185
5A:A:I212 A:A:W211 29.14983.52YesYes189
6A:A:V201 A:A:W211 67.34658.58YesYes199
7A:A:G202 A:A:V201 95.19511.84NoYes199
8A:A:G202 A:A:K46 94.40233.49NoYes199
9A:A:F267 A:A:I49 94.38652.51YesNo097
10A:A:C224 A:A:I49 94.05891.64NoNo077
11A:A:C224 A:A:G40 94.02031.96NoNo079
12A:A:G40 A:A:K46 93.98245.23NoYes099
13A:A:F250 A:A:F307 11.34636.43YesYes198
14A:A:I221 A:A:I264 19.36312.94YesYes186
15A:A:F307 A:A:L266 11.33262.44YesYes189
16B:B:D186 B:B:Y145 27.50615.75YesYes198
17B:B:D186 B:B:G185 27.41431.68YesYes195
18B:B:D205 B:B:H183 15.46168.82YesYes199
19B:B:D205 B:B:G185 27.32491.68YesYes195
20A:A:F267 A:A:F334 94.77963.22YesYes193
21A:A:F334 A:A:Y320 95.98352.06YesYes137
22A:A:E298 A:A:Y290 11.89153.37NoYes047
23A:A:E318 A:A:Y320 49.98725.61NoYes147
24A:A:E318 R:R:R235 50.02348.14NoYes145
25A:A:D341 A:A:Y320 50.009610.34NoYes187
26A:A:D341 R:R:R235 49.99413.57NoYes185
27A:A:F354 R:R:R235 1008.55NoYes055
28A:A:F354 A:A:K349 99.98446.2NoNo055
29A:A:K349 R:R:G303 99.96881.74NoNo056
30R:R:F304 R:R:G303 99.95311.51YesNo086
31R:R:F304 R:R:F78 96.34115.36YesYes086
32R:R:C298 R:R:F78 92.67235.59NoYes076
33R:R:C298 R:R:P294 92.5641.88NoYes279
34R:R:D293 R:R:P294 74.78161.61YesYes299
35B:B:C218 G:G:Q18 18.18493.05YesNo059
36G:G:E22 G:G:Q18 17.78127.65NoNo099
37B:B:Q220 G:G:E22 17.5812.55YesNo079
38B:B:D258 B:B:Q220 11.504613.05YesYes377
39B:B:I18 G:G:A23 20.15143.25NoNo078
40B:B:L14 G:G:A23 18.53991.58YesNo088
41B:B:L14 G:G:L19 13.70476.92YesNo089
42B:B:I18 G:G:R27 12.63373.76NoYes078
43B:B:D290 B:B:R314 10.808720.25YesYes168
44B:B:S275 B:B:T274 13.47763.2YesNo188
45R:R:N71 R:R:P294 17.85946.52YesYes099
46R:R:D99 R:R:N71 17.526812.12NoYes099
47R:R:D99 R:R:S290 34.977210.31NoNo098
48R:R:G103 R:R:S290 34.42361.86NoNo258
49R:R:G103 R:R:L106 34.39761.71NoYes258
50R:R:H60 R:R:L106 33.267811.57YesYes288
51R:R:H60 R:R:R109 15.86153.39YesYes286
52R:R:D42 R:R:Y113 22.37948.05YesYes276
53L:L:S74 R:R:Y113 30.67765.09YesYes206
54L:L:N71 L:L:S74 30.06397.45YesYes200
55L:L:N71 L:L:P72 28.37696.52YesYes200
56R:R:D293 R:R:D99 17.58876.65YesNo099
57R:R:F110 R:R:H60 16.914411.31YesYes278
58R:R:D293 R:R:N289 55.909810.77YesNo299
59R:R:F254 R:R:N289 54.95879.67YesNo299
60R:R:F254 R:R:M134 54.10563.73YesYes297
61R:R:M134 R:R:Y130 29.0227.18YesYes276
62R:R:Y130 R:R:Y279 24.22772.98YesYes265
63R:R:F257 R:R:M134 25.02247.46YesYes267
64R:R:F257 R:R:Y279 24.41764.13YesYes265
65R:R:H126 R:R:Y113 11.21485.44YesYes266
66L:L:I53 L:L:P72 16.71253.39YesYes200
67L:L:C115 L:L:I53 15.45763.27YesYes200
68L:L:C115 L:L:Q25 13.76473.05YesYes200
69R:R:L41 R:R:Y279 39.71814.69NoYes255
70R:R:E44 R:R:L41 39.53513.98YesNo245
71L:L:H76 R:R:E44 39.20116.15YesYes204
72L:L:F69 L:L:H76 19.48613.39YesYes200
73L:L:F69 L:L:Y66 13.85795.16YesNo000
74L:L:Q25 L:L:V136 10.10215.73YesYes000
75L:L:I126 L:L:Y52 11.06974.84YesYes200
76L:L:F129 L:L:I126 10.6838.79YesYes200
77L:L:F129 N:N:Y322 11.78493.09YesYes200
78L:L:H76 L:L:N78 19.44823.83YesNo200
79L:L:N78 N:N:L380 19.382313.73NoNo000
80N:N:L380 N:N:P381 19.4591.64NoYes000
81N:N:E379 N:N:P381 18.18853.14YesYes000
82N:N:E379 N:N:Q376 17.60735.1YesYes200
83N:N:L291 N:N:Q376 13.16612.66YesYes200
84A:A:I221 A:A:L37 17.05682.85YesYes189
85A:A:W211 B:B:Y145 38.12332.89YesYes198
86B:B:R314 B:B:T274 13.3223.88YesNo188
87B:B:D205 B:B:S207 11.396510.31YesYes195
88A:A:W258 B:B:R314 23.70334YesYes158
89B:B:C218 B:B:K209 12.09978.08YesYes156
90A:A:L37 A:A:V201 17.87982.98YesYes199
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1 Node2 LinkStrength Comm IsNode1Hub? IsNode2Hub? Node1Cons Node2Cons Node1Shell Node2Shell
L:L:Y52 R:R:R117 12.35 2 Yes No 0 6 0 1
L:L:N71 R:R:G118 1.7 2 Yes No 0 7 0 1
L:L:S74 R:R:Y113 5.09 2 Yes Yes 0 6 0 1
L:L:S74 R:R:G118 1.86 2 Yes No 0 7 0 1
L:L:S74 R:R:L120 4.5 2 Yes No 0 1 0 1
L:L:H76 R:R:R40 2.26 2 Yes No 0 6 0 1
L:L:H76 R:R:E44 6.15 2 Yes Yes 0 4 0 1
L:L:K84 R:R:H272 6.55 0 No No 0 3 0 1
L:L:G120 R:R:R117 4.5 0 No No 0 6 0 1
L:L:F122 R:R:Y114 8.25 0 No Yes 0 2 0 1
L:L:L123 R:R:L54 4.15 2 Yes No 0 5 0 1
L:L:R124 R:R:P50 14.41 2 Yes No 0 5 0 1
L:L:I125 R:R:H46 10.61 2 Yes Yes 0 4 0 1
L:L:I125 R:R:G47 1.76 2 Yes No 0 2 0 1
N:N:N378 R:R:P50 1.63 2 No No 0 5 0 1
N:N:L380 R:R:G47 5.13 0 No No 0 2 0 1
R:R:H36 R:R:L120 11.57 4 Yes No 8 1 2 1
R:R:A39 R:R:Y113 4 2 No Yes 8 6 2 1
R:R:A39 R:R:L120 3.15 2 No No 8 1 2 1
R:R:A39 R:R:H126 2.93 2 No Yes 8 6 2 2
R:R:E44 R:R:L41 3.98 2 Yes No 4 5 1 2
R:R:L276 R:R:L41 2.77 2 Yes No 4 5 2 2
R:R:D42 R:R:W53 2.23 2 Yes Yes 7 2 2 2
R:R:D42 R:R:Y113 8.05 2 Yes Yes 7 6 2 1
R:R:E43 R:R:H46 6.15 0 No Yes 5 4 2 1
R:R:E43 R:R:Y113 12.35 0 No Yes 5 6 2 1
R:R:E43 R:R:R117 9.3 0 No No 5 6 2 1
R:R:E44 R:R:L276 6.63 2 Yes Yes 4 4 1 2
R:R:H46 R:R:P50 1.53 2 Yes No 4 5 1 1
R:R:H46 R:R:W53 14.81 2 Yes Yes 4 2 1 2
R:R:H46 R:R:Y114 5.44 2 Yes Yes 4 2 1 1
R:R:L54 R:R:W53 2.28 2 No Yes 5 2 1 2
R:R:M57 R:R:W53 2.33 2 Yes Yes 5 2 2 2
R:R:W53 R:R:Y114 13.5 2 Yes Yes 2 2 2 1
R:R:L54 R:R:M57 2.83 2 No Yes 5 5 1 2
R:R:M57 R:R:Y114 2.39 2 Yes Yes 5 2 2 1
R:R:H126 R:R:Y113 5.44 2 Yes Yes 6 6 2 1
R:R:C119 R:R:G118 1.96 0 No No 3 7 2 1
R:R:H272 R:R:H273 9.55 0 No No 3 3 1 2
L:L:G75 R:R:R40 1.5 0 No No 0 6 0 1
R:R:E44 R:R:H272 1.23 2 Yes No 4 3 1 1

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
62.50Single8HS2Fab0468HS2-GPR20-Fab046
46.15Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
37.50Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
36.36Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
33.33Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
31.58Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
31.58Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
30.77Single4BWBNeurotensin4BWB-NTS1-Neurotensin
30.00Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
26.67Single5T04Neurotensin5T04-NTS1-Neurotensin
26.67Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
25.93Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
25.00Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
25.00Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
25.00Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
24.00Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
23.53Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
23.53Single4BV0Neurotensin4BV0-NTS1-Neurotensin
23.53Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
23.53Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
23.53Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
23.53Consensusneurotensin_onOrthosteric Ligandnts1_on
23.53Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
23.08Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
22.73Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
22.22Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
22.22Single4XEENeurotensin4XEE-NTS1-Neurotensin
22.22Single4XESNeurotensin4XES-NTS1-Neurotensin
22.22Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
22.22Single6YVRNTS8-136YVR-NTS1-NTS8-13
22.22Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
22.22Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
22.22Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
22.22Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
22.22Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
21.74Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
21.43Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
21.43Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
21.05Single4BUONeurotensin4BUO-NTS1-Neurotensin
21.05Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
21.05Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
21.05Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
20.83Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
20.83Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
20.83Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
20.00Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
20.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
20.00Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
20.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
20.00Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
20.00Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
20.00Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
19.23Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
19.23Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
19.05Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
18.75Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
18.75Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
18.75Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
18.75Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
18.52Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
18.52Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
18.18Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
18.18Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
18.18Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
18.18Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
18.18Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
18.18Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
17.86Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
17.39Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
16.67Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
16.67Single6OS1TRV0266OS1-AT1-TRV026
16.67Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
16.67Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
16.67Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
16.67Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
16.67Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
16.67Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
16.67Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
16.67Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
16.67Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
16.67Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
16.67Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
16.00Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
16.00Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
15.79Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
15.79Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
15.79Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
15.79Single8XQJJN2418XQJ-Apelin-JN241
15.38Single6FJ3PTH6FJ3-PTH1-PTH
15.38Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
15.38Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
15.38Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
15.38Single8JPSCCL78JPS-ACKR1-CCL7
15.38Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
15.00Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
15.00Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
15.00Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
14.81Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
14.81Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
14.81Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
14.81Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
14.81Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
14.81Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
14.29Single4O9RCyclopamine4O9R-SMO-Cyclopamine
14.29Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
14.29Single6KNMJN241-96KNM-Apelin-JN241-9
14.29Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
14.29Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
14.29Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
14.29Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
14.29Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
14.29Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
14.29Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
14.29Single8XQJJN2418XQJ-Apelin-JN241
14.29Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
14.29Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
13.79Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
13.79Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
13.64Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
13.64Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
13.64Single8XWNCXCL88XWN-CXCR2-CXCL8
13.64Consensuslpl_onOrthosteric Ligands1p_on lpa_on
13.64Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
13.33Single4QINSAG1.54QIN-SMO-SAG1.5
13.33Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
13.33Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
13.33Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
13.33Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
13.33Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
13.33Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
13.33Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
13.33Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
13.33Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
13.04Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
13.04Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
13.04Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
13.04Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
13.04Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
13.04Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
12.90Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
12.50Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
12.50Single6D35Cholesterol6D35-SMO-Cholesterol
12.50Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
12.50Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
12.50Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
12.50Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
12.50Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
12.50Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
12.50Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
12.50Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
12.50Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
12.50Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
12.50Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
12.50Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
12.50Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.50Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.50Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.50Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.50Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
12.50Single7DTTCa7DTT-CaS-Ca-Ca
12.50Single7DTTCa7DTT-CaS-Ca-Ca
12.50Single7DTUTryptophan7DTU-CaS-Tryptophan
12.50Single7DTUTryptophan7DTU-CaS-Tryptophan
12.50Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
12.50Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
12.50Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
12.50Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
12.50Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
12.50Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
12.50Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
12.50Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
12.50Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
12.50Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
12.50Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
12.50Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
12.50Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
12.50Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
12.50Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
12.50Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
12.50Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
12.50Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
12.50Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
12.50Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
12.50Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
12.50Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
12.50Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
12.50Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
12.50Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
12.50Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
12.50Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
12.50Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
12.50Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
12.50Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
12.50Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
12.50Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
12.50Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
12.50Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
12.50Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
12.50Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.50Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.50Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.50Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.50Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
12.50Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
12.50Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
12.50Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
12.50Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
12.50Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
12.50Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
12.50Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
12.50Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
12.50Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
12.50Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
12.50Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
12.50Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
12.50Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
12.50Single7XW7K1-707XW7-TSH-K1-70
12.50Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
12.50Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
12.50Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
12.50Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
12.50Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
12.50Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
12.50Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
12.50Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
12.50Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
12.50Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
12.50Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
12.50Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
12.50Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
12.50Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
12.50Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
12.50Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
12.50Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
12.50Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
12.50Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
12.50Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
12.50Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
12.50Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
12.50Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
12.50Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
12.50Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
12.50Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
12.50Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
12.50Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
12.50Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
12.50Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
12.50Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
12.50Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
12.50Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
12.50Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
12.50Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
12.50Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
12.50Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
12.50Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
12.50Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
12.50Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
12.50Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
12.50Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
12.50Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
12.50Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
12.50Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
12.50Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
12.50Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
12.50Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
12.50Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
12.50Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
12.50Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
12.50Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
12.50Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
12.50Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
12.50Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
12.50Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
12.50Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
12.50Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
12.50Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
12.50Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
12.50Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
12.50Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8WVXNorrin8WVX-LGR4-Norrin
12.50Single8WVYNorrin8WVY-LGR4-Norrin
12.50Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
12.50Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
12.50Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
12.50Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
12.50Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
12.50Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
12.50Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
12.50Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
12.50Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
12.50Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
12.50Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
12.50Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
12.50Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
12.50Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
12.50Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
12.50Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
12.50Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
12.50Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
12.50Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
12.50Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
12.50Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
12.50Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
12.50Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
12.50Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
12.50Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
12.50Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
12.50Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
12.50Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
12.50Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
12.12Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
12.00Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
12.00Single6JODAngiotensin II6JOD-AT2-Angiotensin II
12.00Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
12.00Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
12.00Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
12.00Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
12.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
12.00Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
12.00Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
12.00Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
12.00Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
11.76Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
11.76Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
11.76Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
11.76Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
11.76Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
11.76Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
11.76Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.76Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
11.76Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
11.76Single8K5DGSK2560738K5D-HCA2-GSK256073
11.76Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.76Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
11.76Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
11.76Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
11.76Consensushca_on_gpOrthosteric Ligandhca2_on_gp
11.76Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
11.54Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
11.54Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
11.54Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
11.54Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
11.54Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
11.54Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
11.54Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
11.54Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
11.54Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
11.54Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
11.54Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single4XT3Fractalkine4XT3-US28-Fractalkine
11.11Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
11.11Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
11.11Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
11.11Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
11.11Single7C4SS1P7C4S-S1P3-S1P
11.11Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
11.11Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
11.11Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
11.11Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
11.11Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.11Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.11Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.11Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.11Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
11.11Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
11.11Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
11.11Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
11.11Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
11.11Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
11.11Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
11.11Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
11.11Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
11.11Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
11.11Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
11.11Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
11.11Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
11.11Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
11.11Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
11.11Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
11.11Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
11.11Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
11.11Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
11.11Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
11.11Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
11.11Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
11.11Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
11.11Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
10.81Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
10.71Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
10.71Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
10.71Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
10.71Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
10.71Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
10.71Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
10.71Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
10.71Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
10.71Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
10.53Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
10.53Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
10.53Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
10.53Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
10.53Single7F1TMIP-1a7F1T-CCR5-MIP-1a
10.53Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
10.53Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
10.53Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
10.53Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
10.53Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
10.53Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
10.53Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
10.53Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
10.53Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
10.53Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
10.53Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
10.53Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
10.53Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
10.53Consensuslpa_onOrthosteric Ligandlpa1_on
10.53Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
10.53Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
10.34Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
10.34Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
10.34Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
10.34Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
10.34Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
10.34Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
10.34Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
10.34Single8IY6Endothelin-18IY6-ETB-Endothelin-1
10.34Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
10.34Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
10.34Consensusbradykinin_onOrthosteric Ligandbk2_on
10.34Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
10.34Consensusendothelin_onOrthosteric Ligandetb_on eta_on
10.34Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
10.00Single5GLHEndothelin-15GLH-ETB-Endothelin-1
10.00Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
10.00Single6IGKEndothelin-36IGK-ETB-Endothelin-3
10.00Single6KQICP559406KQI-CB1-CP55940-Org27569
10.00Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
10.00Single6OS2TRV0266OS2-AT1-TRV026
10.00Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
10.00Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
10.00Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
10.00Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
10.00Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
10.00Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
10.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8XWACXCL18XWA-CXCR2-CXCL1
10.00Single8XWMCXCL68XWM-CXCR2-CXCL6
10.00Single8XWSCXCL58XWS-CXCR2-CXCL5
10.00Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
10.00Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
10.00Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
10.00Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
10.00Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
10.00Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
10.00Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
10.00Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
10.00Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
10.00Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
10.00Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
10.00Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
10.00Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
10.00Consensuslpa_offOrthosteric Ligandlpa1_off
10.00Consensuslpl_offOrthosteric Ligands1p_off lpa_off
10.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
10.00Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
10.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
10.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
10.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
9.68Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
9.68Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
9.68Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
9.68Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
9.68Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
9.68Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
9.52Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
9.52Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
9.52Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
9.52Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
9.52Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
9.52Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
9.52Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
9.52Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
9.52Single8XVUCXCL28XVU-CXCR2-CXCL2
9.52Single8XWFCXCL38XWF-CXCR2-CXCL3
9.52Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
9.52Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
9.52Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
9.52Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
9.52Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
9.52Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
9.38Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
9.38Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
9.09Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
9.09Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
9.09Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
9.09Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
9.09Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
9.09Single7SK9CCX6627SK9-ACKR3-CCX662
9.09Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
9.09Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
9.09Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
9.09Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
9.09Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
9.09Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
9.09Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
9.09Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
9.09Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
9.09Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
9.09Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
9.09Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
8.70Single4XT1Fractalkine4XT1-US28-Fractalkine
8.70Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
8.70Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
8.70Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
8.70Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.70Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
8.70Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
8.70Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.70Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
8.70Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
8.70Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
8.70Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.70Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
8.70Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.70Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.70Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
8.70Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
8.70Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
8.70Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
8.70Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
8.70Consensussomatostatin_offOrthosteric Ligandsst2_off
8.70Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
8.33Single5L7DCholesterol5L7D-SMO-Cholesterol
8.33Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
8.33Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
8.33Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
8.33Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
8.33Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
8.33Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
8.33Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
8.33Single7XNACYN1548067XNA-SST2-CYN154806
8.33Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
8.33Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
8.33Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.33Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
8.33Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.33Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.33Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
8.33Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
8.33Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
8.33Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
8.33Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
8.33Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
8.33Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
8.33Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
8.00Single3OE0CVX153OE0-CXCR4-CVX15
8.00Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
8.00Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
8.00Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
8.00Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
8.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
8.00Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
8.00Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
8.00Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
8.00Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
8.00Consensusangiotensin_onOrthosteric Ligandat1_on
8.00Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
8.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
8.00Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
8.00Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
8.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
8.00Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
8.00Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.00Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.00Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
7.69Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
7.69Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
7.69Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
7.69Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
7.69Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
7.69Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
7.69Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
7.69Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
7.69Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
7.69Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
7.69Consensusp2y_offOrthosteric Ligandp2y1_off
7.69Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
7.41Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
7.41Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
7.41Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
7.41Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
7.41Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
7.41Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
7.41Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
7.41Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
7.41Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
7.41Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
7.41Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
7.41Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
7.41Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
7.14Single4XNWMRS25004XNW-P2Y1-MRS2500
7.14Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
7.14Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
7.14Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
7.14Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
7.14Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
7.14Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
7.14Single7SK3CXCL127SK3-ACKR3-CXCL12
7.14Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
7.14Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
7.14Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
7.14Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
7.14Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
7.14Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
7.14Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
7.14Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
7.14Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
7.14Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
6.90Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
6.90Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
6.90Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
6.90Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
6.90Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
6.90Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
6.90Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
6.67Single6IGLIRL16206IGL-ETB-IRL1620
6.67Single6LI0C176LI0-GPR52-C17
6.67Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
6.67Single7UL2SR486927UL2-NTS1-SR48692-Na
6.67Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
6.67Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
6.67Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
6.67Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
6.67Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
6.67Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
6.67Single8K5BNiacin8K5B-HCA2-Niacin
6.67Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
6.67Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
6.67Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
6.67Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
6.67Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9B9Y7DY9B9Y-CB1-7DY
6.67Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
6.67Consensusgq_nucleotideOrthosteric Ligandgq_p2y
6.67Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
6.67Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
6.67Consensusneurotensin_offOrthosteric Ligandnts1_off
6.67Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
6.45Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
6.45Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
6.45Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
6.45Consensusbombesin_onOrthosteric Ligandbb2_on
6.45Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
6.45Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
6.45Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
6.45Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
6.25Single3PWHZM-2413853PWH-A2A-ZM-241385
6.25Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
6.25Single5U09Taranabant5U09-CB1-Taranabant
6.25Single5ZKQABT-4915ZKQ-PAF-ABT-491
6.25Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
6.25Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
6.25Single7BR3Elagolix7BR3-GnRH1-Elagolix
6.25Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
6.25Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
6.25Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
6.25Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
6.25Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
6.25Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
6.25Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
6.25Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
6.25Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
6.25Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
6.25Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
6.25Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
6.25Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
6.25Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
6.25Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
6.25Single9BA0A1AKN9BA0-CB1-A1AKN
6.25Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
6.25Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
6.25Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
6.25Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
6.25Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
6.25Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
6.25Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
6.25Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
6.25Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
6.25Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
6.25Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
5.88Single3REYXAC3REY-A2A-XAC
5.88Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
5.88Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
5.88Single6ZINSR486926ZIN-NTS1-SR48692
5.88Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
5.88Single7VV6C48/807VV6-MRGPRX2-C48/80
5.88Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
5.88Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
5.88Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
5.88Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
5.88Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
5.88Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
5.88Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
5.88Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
5.88Single8K5CAcipimox8K5C-HCA2-Acipimox
5.88Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
5.88Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
5.88Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
5.88Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
5.88Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
5.88Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
5.88Consensusgrh_offOrthosteric Ligandgnrh1_off
5.88Consensushca_onOrthosteric Ligandhca2_on
5.88Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
5.56Single4QIMANTA XV4QIM-SMO-ANTA XV
5.56Single4YAYZD-71554YAY-AT1-ZD-7155
5.56Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
5.56Single5TGZAM65385TGZ-CB1-AM6538
5.56Single5UIGCmpd-15UIG-A2A-Cmpd-1
5.56Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
5.56Single6D27CAY104716D27-DP2-CAY10471
5.56Single6IIVDaltroban6IIV-TP-Daltroban
5.56Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
5.56Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
5.56Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
5.56Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
5.56Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
5.56Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
5.56Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
5.56Single7V3ZCP559407V3Z-CB1-CP55940
5.56Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
5.56Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
5.56Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
5.56Single7YXAONO-54306087YXA-S1P5-ONO-5430608
5.56Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
5.56Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
5.56Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
5.56Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
5.56Single8RLNLUF58348RLN-A2A-LUF5834
5.56Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
5.56Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
5.56Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
5.56Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
5.56Single9B9ZA1AKO9B9Z-CB1-A1AKO
5.56Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
5.56Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
5.56Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
5.56Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
5.56Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
5.56Consensusblt_onOrthosteric Ligandblt1_on
5.56Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
5.56Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
5.56Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
5.56Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
5.56Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
5.56Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
5.56Consensusleukotriene_onOrthosteric Ligandblt_on
5.56Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
5.56Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
5.56Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
5.56Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
5.56Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
5.56Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
5.26Single4JKVTaladegib4JKV-SMO-Taladegib
5.26Single5C1MBU725C1M-μ-BU72
5.26Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
5.26Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
5.26Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
5.26Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
5.26Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
5.26Single6Z4SSR486926Z4S-NTS1-SR48692
5.26Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
5.26Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
5.26Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
5.26Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
5.26Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
5.26Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
5.26Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
5.26Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
5.26Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
5.26Consensusblt_offOrthosteric Ligandblt1_off
5.26Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
5.26Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
5.26Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
5.26Consensusep_offOrthosteric Ligandep4_off
5.26Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
5.26Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
5.26Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
5.26Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
5.26Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
5.26Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
5.00Single5V56TC1145V56-SMO-TC114
5.00Single5V57TC1145V57-SMO-TC114
5.00Single5XR8AM8415XR8-CB1-AM841
5.00Single5XRAAM115425XRA-CB1-AM11542
5.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
5.00Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
5.00Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
5.00Single7FEECP559407FEE-CB1-CP55940-ZCZ011
5.00Single7R0CAVP7R0C-V2-AVP-Arrestin2
5.00Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
5.00Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
5.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
5.00Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
5.00Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single8E0GBU728E0G-μ-BU72
5.00Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
5.00Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
5.00Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
5.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
5.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
5.00Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
5.00Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
5.00Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
5.00Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
5.00Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
5.00Consensusa2_onOrthosteric Liganda2b_on
5.00Consensusa2_on_gpOrthosteric Liganda2b_on_gp
5.00Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
5.00Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
5.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
5.00Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
5.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
5.00Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
5.00Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
5.00Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
5.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
5.00Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
5.00Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
4.76Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
4.76Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
4.76Single5X33BIIL2605X33-BLT1-BIIL260
4.76Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
4.76Single6IIURamatroban6IIU-TP-Ramatroban
4.76Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
4.76Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
4.76Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
4.76Single7K15MKD0467K15-BLT1-MKD046-Na
4.76Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
4.76Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
4.76Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
4.76Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
4.76Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
4.76Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
4.76Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
4.76Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
4.76Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
4.76Single8JWY2-1188JWY-A2A-2-118
4.76Single8JWZAB9288JWZ-A2A-AB928-Na
4.76Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
4.76Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
4.76Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
4.76Single8XYIVUF106618XYI-CXCR3-VUF10661
4.76Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
4.76Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
4.76Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
4.76Consensusalpha1_offOrthosteric Ligandalpha1a_off
4.76Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
4.76Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
4.76Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
4.76Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
4.76Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
4.76Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
4.76Consensusorexin_onOrthosteric Ligandox2_on
4.55Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
4.55Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
4.55Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
4.55Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
4.55Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
4.55Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
4.55Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
4.55Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
4.55Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
4.55Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
4.55Single7UM4AS26747237UM4-5-HT5A-AS2674723
4.55Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
4.55Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
4.55Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
4.55Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
4.55Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
4.55Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
4.55Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
4.55Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
4.55Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
4.55Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
4.55Consensuscck_onOrthosteric Ligandccka_on cckb_on
4.55Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
4.55Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
4.55Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
4.55Consensuschemerin_onOrthosteric Ligandcml1_on
4.55Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
4.55Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
4.55Consensusprostanoid_offOrthosteric Ligandep_off dp_off
4.55Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
4.55Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
4.55Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single4UG2CGS216804UG2-A2A-CGS21680
4.35Single5EE7MK08935EE7-Glucagon-MK0893
4.35Single5ZTYAM102575ZTY-CB2-AM10257
4.35Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
4.35Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
4.35Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
4.35Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
4.35Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
4.35Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
4.35Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
4.35Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
4.35Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
4.35Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single8QJ2pN1628QJ2-MC4-pN162-Gs
4.35Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
4.35Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
4.35Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
4.35Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
4.35Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
4.35Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
4.35Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
4.35Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
4.35Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
4.17Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
4.17Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
4.17Single7F8XNN90567F8X-CCKA-NN9056
4.17Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
4.17Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
4.17Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
4.17Single8KIGSHU91198KIG-MC3-SHU9119-Ca
4.17Single8WKYPG-9348WKY-MC4-PG-934
4.17Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
4.17Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
4.17Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
4.17Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
4.17Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
4.17Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
4.17Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
4.00Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
4.00Single7SK5CXCL127SK5-ACKR3-CXCL12
4.00Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
4.00Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
4.00Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
4.00Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
4.00Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
4.00Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
4.00Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
4.00Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
4.00Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
4.00Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
4.00Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
4.00Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
3.85Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
3.85Single6W25SHU91196W25-MC4-SHU9119-Ca
3.85Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
3.85Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.85Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
3.85Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
3.85Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
3.85Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
3.85Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
3.85Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
3.85Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
3.70Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
3.70Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
3.70Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
3.70Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
3.70Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
3.70Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
3.70Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
3.70Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
3.70Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
3.70Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
3.70Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
3.70Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
3.70Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
3.70Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
3.70Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
3.70Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
3.70Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
3.70Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
3.70Consensusvasop-oxy_onOrthosteric Ligandv2_on
3.70Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
3.57Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
3.57Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
3.57Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
3.57Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
3.57Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
3.57Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
3.57Single8ZRTET-18ZRT-ETB-ET-1
3.57Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
3.57Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
3.57Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
3.57Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
3.57Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
3.57Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
3.45Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
3.45Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
3.45Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
3.45Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
3.45Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
3.33Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
3.33Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
3.33Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
3.33Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3
3.33Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
3.23Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
3.23Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
2.94Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy

PDB Summary
PDB 8HSC
Class A
SubFamily Orphan
Type Orphan
SubType GPR20
Species Homo Sapiens
Ligand Fab046
Other Ligand(s) -
Protein Partners Gi1/Beta1/Gamma2
PDB Resolution 3.22
Date 2023-03-08 
D.O.I. 10.1038/s41421-023-00520-8
Net Summary
Imin 1.53
Number of Linked Nodes 1034
Number of Links 1597
Number of Hubs 381
Number of Links mediated by Hubs 1242
Number of Communities 16
Number of Nodes involved in Communities 534
Number of Links involved in Communities 962
Path Summary
Number Of Nodes in MetaPath 91
Number Of Links MetaPath 90
Number of Shortest Paths 9623153
Length Of Smallest Path 3
Average Path Length 38.2253
Length of Longest Path 69
Minimum Path Strength 1.12
Average Path Strength 4.61429
Maximum Path Strength 25.44
Minimum Path Correlation 0.7
Average Path Correlation 0.997533
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.85714
Average % Of Corr. Nodes 44.4533
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 63.6023
Maximum Path Hubs % 100
AnnotationTypeLinks
Gene OntologyMolecular Function
Gene OntologyBiological Process
Gene OntologyCellular Component
SCOP2Domain Identifier• Ras-like P-loop GTPases   • Transducin (heterotrimeric G protein), gamma chain
SCOP2Family Identifier• Ras-like P-loop GTPases   • Transducin (heterotrimeric G protein), gamma chain
Membrane Protein Annotations-• Orientations of Proteins in Membranes database (OPM)   • Protein Data Bank of Transmembrane Proteins (PDBTM)   • MemProtMD


Details about the values in these tables can be found in the corresponding documentation page .
PDBsumOpen PDBsum Page
ChainA
ProteinG Protein α Sub unit
UniProtP63096
Sequence
>8HSC_Chain_A
CTLSAEDKA AVERSKMID RNLREDGEK AAREVKLLL LGAGESGKN 
TIVKQMKTG IVETHFTFK DLHFKMFDV GAQRSERKK WIHCFEGVT 
AIIFCVALS DYDLMNRMH ESMKLFDSI CNNKWFTDT SIILFLNKK 
DLFEEKIKK SPLTICYPE YAGSNTYEE AAAYIQCQF EDLNKRKDT 
KEIYTHFTC STDTKNVQF VFDAVTDVI IKNNLKDCG LF


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainB
ProteinG Protein β Sub unit
UniProtP62873
Sequence
>8HSC_Chain_B
ELDQLRQEA EQLKNQIRD ARKACADAT LSQITNNID PVGRIQMRT 
RRTLRGHLA KIYAMHWGT DSRLLVSAS QDGKLIIWD SYTTNKVHA 
IPLRSSWVM TCAYAPSGN YVACGGLDN ICSIYNLKT REGNVRVSR 
ELAGHTGYL SCCRFLDDN QIVTSSGDT TCALWDIET GQQTTTFTG 
HTGDVMSLS LAPDTRLFV SGACDASAK LWDVREGMC RQTFTGHES 
DINAICFFP NGNAFATGS DDATCRLFD LRADQELMT YSHDNIICG 
ITSVSFSKS GRLLLAGYD DFNCNVWDA LKADRAGVL AGHDNRVSC 
LGVTDDGMA VATGSWDSF LKIWN


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainG
ProteinG Protein γ Sub unit
UniProtP59768
Sequence
>8HSC_Chain_G
ASIAQARKL VEQLKMEAN IDRIKVSKA AADLMAYCE AHAKEDPLL 
TPVPASENP FRE


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainR
ProteinReceptor
UniProtQ99678
Sequence
>8HSC_Chain_R
VPLFHLFAR LDEELHGTF PGLWLALMA VHGAIFLAG LVLNGLALY 
VFCCRTRAK TPSVIYTIN LVVTDLLVG LSLPTRFAV YYGARGCLR 
CAFPHVLGY FLNMHCSIL FLTCICVDR YLAIVRPEG SRRCRQPAC 
ARAVCAFVW LAAGAVTLS VLGVRVFAL TVLEFLLPL LVISVFTGR 
IMCALSRPG LLHQGRQRR VRAMQLLLT VLIIFLVCF TPFHARQVA 
VALWPDMPH HTSLVVYHV AVTLSSLNS CMDPIVYCF VTSGFQATV 
RGL


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  




This receptor, from the same or other species and bound to the same or other ligands, is also present in the following networks:
Show PDB Class SubFamily Type SubType Species Orthosteric Ligand Other Ligand(s) Protein Partners Resolution Date DOI
8HS2AOrphanOrphanGPR20Homo sapiensFab046--3.082023-03-0810.1038/s41421-023-00520-8
8HSCAOrphanOrphanGPR20Homo sapiensFab046-Gi1/β1/γ23.222023-03-0810.1038/s41421-023-00520-8
8HSC (No Gprot) AOrphanOrphanGPR20Homo sapiensFab046-3.222023-03-0810.1038/s41421-023-00520-8
8HS3AOrphanOrphanGPR20Homo sapiens--Gi1/β1/γ23.142023-03-0810.1038/s41421-023-00520-8
8HS3 (No Gprot) AOrphanOrphanGPR20Homo sapiens--3.142023-03-0810.1038/s41421-023-00520-8




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