| 5ht1_off | 5ht1b_off |
| 5ht1_on | 5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on |
| 5ht1_on_gp | 5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp |
| 5ht1a_on | 8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 |
| 5ht1a_on_gp | 8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 |
| 5ht1b_off | 5V54-5-HT1B-Methiothepin |
| 5ht1d_on | 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 |
| 5ht1d_on_gp | 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 |
| 5ht1e_on | 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 |
| 5ht1e_on_gp | 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 |
| 5ht1f_on | 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 |
| 5ht1f_on_gp | 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 |
| 5ht2_off | 5ht2a_off 5ht2b_off 5ht2c_off |
| 5ht2_on | 5ht2b_on |
| 5ht2_on_gp | 5ht2b_on_gp |
| 5ht2a_off | 6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179 |
| 5ht2b_off | 6DRZ-5-HT2B-Methysergide |
| 5ht2b_on | 7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2 |
| 5ht2b_on_gp | 7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2 |
| 5ht2c_off | 6BQH-5-HT2C-Ritanserin |
| 5ht4_on | 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 |
| 5ht4_on_gp | 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 |
| 5ht5_on | 5ht5a_on |
| 5ht5_on_gp | 5ht5a_on_gp |
| 5ht5a_on | 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 |
| 5ht5a_on_gp | 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 |
| 5ht6_on | 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 |
| 5ht6_on_gp | 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 |
| 5ht7_on | 7XTC-5-HT7-5-CT-Gs/β1/γ2 |
| 5ht7_on_gp | 7XTC-5-HT7-5-CT-Gs/β1/γ2 |
| 5ht_off | 5ht2_off 5ht1_off |
| 5ht_on | 5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on |
| 5ht_on_gp | 5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp |
| a1_off | 5UEN-A1-DU172 5N2S-A1-PSB36 |
| a1_on | 7LD4-A1-Adenosine-Gi2/β1/γ2 |
| a1_on_gp | 7LD4-A1-Adenosine-Gi2/β1/γ2 |
| a2_off | a2a_off |
| a2_on | a2b_on |
| a2_on_gp | a2b_on_gp |
| a2a_off | 3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na |
| a2b_on | 8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 |
| a2b_on_gp | 8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 |
| a3_on | a3a_on |
| a3_on_gp | a3a_on_gp |
| a3a_on | 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2 |
| a3a_on_gp | 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2 |
| adenosine_off | a1_off a2_off |
| adenosine_on | a1_on a2_on a3_on |
| adenosine_on_gp | a1_on_gp a2_on_gp a3_on_gp |
| adrenergic_off | alpha_off beta_off |
| adrenergic_on | alpha_on beta_on |
| adrenergic_on_gp | alpha_on_gp beta_on_gp |
| alicarboxylic_off | succinate_off |
| alicarboxylic_on | succinate_on hca_on |
| alicarboxylic_on_gp | succinate_on_gp hca_on_gp |
| alpha1_off | alpha1a_off |
| alpha1_on | alpha1a_on |
| alpha1_on_gp | alpha1a_on_gp |
| alpha1a_off | 7YMJ-Alpha1A-Tamsulosin |
| alpha1a_on | 7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 |
| alpha1a_on_gp | 7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 |
| alpha2_off | alpha2c_off |
| alpha2_on | alpha2b_on |
| alpha2_on_gp | alpha2b_on_gp |
| alpha2b_on | 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 |
| alpha2b_on_gp | 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 |
| alpha2c_off | 6KUW-α2c-PubChem 57213234 |
| alpha_off | alpha1_off alpha2_off |
| alpha_on | alpha1_on alpha2_on |
| alpha_on_gp | alpha1_on_gp alpha2_on_gp |
| amine_off | 5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off |
| amine_offon | amine_off amine_on |
| amine_offon_gp | amine_on_gp amine_off |
| amine_on | 5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on |
| amine_on_gp | 5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp |
| angiotensin_off | at1_off |
| angiotensin_on | at1_on |
| angiotensin_on_gp | at1_on_gp |
| apelin_on | 8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2 |
| apelin_on_gp | 8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2 |
| at1_off | 4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan |
| at1_on | 7F6G-AT1-SAR1-AngII-Gq/β1/γ2 |
| at1_on_gp | 7F6G-AT1-SAR1-AngII-Gq/β1/γ2 |
| bb2_off | 7W41-BB2-PD176252 |
| bb2_on | 7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2 |
| bb2_on_gp | 7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2 |
| beta1_off | 2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na |
| beta1_on | 8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2 |
| beta1_on_gp | 8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2 |
| beta2_off | 2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol |
| beta2_on | 7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 |
| beta2_on_gp | 7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 |
| beta3_on | 7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 |
| beta3_on_gp | 7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 |
| beta_off | beta1_off beta2_off |
| beta_on | beta1_on beta2_on beta3_on |
| beta_on_gp | beta1_on_gp beta2_on_gp beta3_on_gp |
| bk2_on | 7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2 |
| bk2_on_gp | 7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2 |
| blt1_off | 5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na |
| blt1_on | 7VKT-BLT1-LTB4-Gi1/β1/γ2 |
| blt1_on_gp | 7VKT-BLT1-LTB4-Gi1/β1/γ2 |
| blt_off | blt1_off |
| blt_on | blt1_on |
| blt_on_gp | blt1_on_gp |
| bombesin_off | bb2_off |
| bombesin_on | bb2_on |
| bombesin_on_gp | bb2_on_gp |
| bradykinin_on | bk2_on |
| bradykinin_on_gp | bk2_on_gp |
| c3a_on | 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 |
| c3a_on_gp | 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 |
| c5a1_on | 8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2 |
| c5a1_on_gp | 8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2 |
| cannabinoid_off | cb2_off cb1_off |
| cannabinoid_on | cb2_on cb1_on |
| cannabinoid_on_gp | cb2_on_gp cb1_on_gp |
| cb1_off | 5U09-CB1-Taranabant 5TGZ-CB1-AM6538 |
| cb1_on | 6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2 |
| cb1_on_gp | 6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2 |
| cb2_off | 5ZTY-CB2-AM10257 |
| cb2_on | 8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 |
| cb2_on_gp | 8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 |
| cck_off | ccka_off |
| cck_on | ccka_on cckb_on |
| cck_on_gp | ccka_on_gp cckb_on_gp |
| ccka_off | 7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript |
| ccka_on | 7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 |
| ccka_on_gp | 7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 |
| cckb_on | 8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2 |
| cckb_on_gp | 8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2 |
| ccr1_on | 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 |
| ccr1_on_gp | 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 |
| ccr2_off | 6GPS-CCR2-MK0812 |
| ccr2_on | 7XA3-CCR2-CCL2-Gi1/β1/γ2 |
| ccr2_on_gp | 7XA3-CCR2-CCL2-Gi1/β1/γ2 |
| ccr5_off | 5UIW-CCR5-5P7-CCL5 |
| ccr5_on | 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 |
| ccr5_on_gp | 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 |
| ccr6_on | 6WWZ-CCR6-CCL20-Go/β1/γ2 |
| ccr6_on_gp | 6WWZ-CCR6-CCL20-Go/β1/γ2 |
| ccr8_on | 8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2 |
| ccr8_on_gp | 8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2 |
| ccr_off | ccr2_off ccr5_off |
| ccr_on | ccr6_on ccr8_on ccr2_on ccr1_on ccr5_on |
| ccr_on_gp | ccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp |
| chemerin_on | cml1_on |
| chemerin_on_gp | cml1_on_gp |
| chemokine_off | ccr_off cxcr_off |
| chemokine_on | ccr_on cxcr_on |
| chemokine_on_gp | ccr_on_gp cxcr_on_gp |
| class-a_off | sensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off |
| class-a_on | sensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on |
| class-a_on_gp | sensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp |
| cml1_on | 7YKD-CML1-Chemerin-9-Gi1/β1/γ2 |
| cml1_on_gp | 7YKD-CML1-Chemerin-9-Gi1/β1/γ2 |
| compl-peptide_on | c5a1_on c3a_on |
| compl-peptide_on_gp | c5a1_on_gp c3a_on_gp |
| cxcr1_on | 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 |
| cxcr1_on_gp | 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 |
| cxcr2_on | 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 |
| cxcr2_on_gp | 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 |
| cxcr3_off | 8K2W-CXCR3-AMG487 |
| cxcr3_on | 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 |
| cxcr3_on_gp | 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 |
| cxcr4_off | 4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t |
| cxcr4_on | 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 |
| cxcr4_on_gp | 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 |
| cxcr_off | cxcr3_off cxcr4_off |
| cxcr_on | cxcr3_on cxcr4_on cxcr1_on cxcr2_on |
| cxcr_on_gp | cxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp |
| cyslt1_off | 6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na |
| cyslt2_off | 6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372 |
| cyslt_off | cyslt2_off cyslt1_off |
| d1_on | 7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 |
| d1_on_gp | 7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 |
| d2_off | 6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone |
| d2_on | 7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 |
| d2_on_gp | 7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 |
| d3_off | 3PBL-D3-Eticlopride |
| d3_on | 7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 |
| d3_on_gp | 7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 |
| d4_on | 8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2 |
| d4_on_gp | 8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2 |
| d5_on | 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 |
| d5_on_gp | 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 |
| dop_off | 4EJ4-δ-Naltrindole |
| dop_on | 8F7S-δ-Deltorphin-Gi1/β1/γ2 |
| dop_on_gp | 8F7S-δ-Deltorphin-Gi1/β1/γ2 |
| dopamine_off | d2_off d3_off |
| dopamine_on | d2_on d1_on d3_on d4_on d5_on |
| dopamine_on_gp | d2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp |
| dp2_off | 6D26-DP2-Fevipiprant |
| dp_off | dp2_off |
| endothelin_off | etb_off |
| endothelin_on | etb_on eta_on |
| endothelin_on_gp | etb_on_gp eta_on_gp |
| ep4_off | 5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352 |
| ep_off | ep4_off |
| eta_on | 8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| eta_on_gp | 8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| etb_off | 5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500 |
| etb_on | 8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2 |
| etb_on_gp | 8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2 |
| ffa2_on | 8J22-FFA2-TUG-1375-Gi1/β1/γ2 |
| ffa2_on_gp | 8J22-FFA2-TUG-1375-Gi1/β1/γ2 |
| ffa3_on | 8J21-FFA3-Butyric acid-Gi1/β1/γ2 |
| ffa3_on_gp | 8J21-FFA3-Butyric acid-Gi1/β1/γ2 |
| ffa_on | ffa2_on ffa3_on |
| ffa_on_gp | ffa2_on_gp ffa3_on_gp |
| formylpeptide_on | fpr2-alx_on fpr1-alx_on |
| formylpeptide_on_gp | fpr2-alx_on_gp fpr1-alx_on_gp |
| fp-alpha_on | 8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| fp-alpha_on_gp | 8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| fpr1-alx_on | 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 |
| fpr1-alx_on_gp | 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 |
| fpr2-alx_on | 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2 |
| fpr2-alx_on_gp | 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2 |
| gal1_on | 7WQ3-GAL1-Galanin-Gi1/β1/γ2 |
| gal1_on_gp | 7WQ3-GAL1-Galanin-Gi1/β1/γ2 |
| gal2_on | 7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2 |
| gal2_on_gp | 7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2 |
| galanin_on | gal2_on gal1_on |
| galanin_on_gp | gal2_on_gp gal1_on_gp |
| ghrelin_off | 6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457 |
| ghrelin_on | 7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2 |
| ghrelin_on_gp | 7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2 |
| gi_5ht | 8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 |
| gi_adenosine | 7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2 |
| gi_adrenergic | 7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2 |
| gi_alicarboxylic | gi_hca gi_succinate |
| gi_amine | gi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine |
| gi_apelin | 8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2 |
| gi_cannabinoid | 8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2 |
| gi_cck | 7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2 |
| gi_chemerin | 7YKD-CML1-Chemerin-9-Gi1/β1/γ2 |
| gi_chemokine | 6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2 |
| gi_class-a | gi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein |
| gi_compl-pept | 8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2 |
| gi_dopamine | 7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 |
| gi_endothelin | 8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2 |
| gi_ffa | 8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2 |
| gi_formylpeptide | 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2 |
| gi_galanin | 7WQ3-GAL1-Galanin-Gi1/β1/γ2 |
| gi_ghrelin | 7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2 |
| gi_hca | 8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 |
| gi_histamine | 8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 |
| gi_leukotriene | 7VKT-BLT1-LTB4-Gi1/β1/γ2 |
| gi_lipid | gi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p |
| gi_lpa | 7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2 |
| gi_muscarinic | 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 |
| gi_neurotensin | 6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1 |
| gi_npy | 8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2 |
| gi_nucleotide | gi_adenosine gi_p2y |
| gi_opioid | 8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2 |
| gi_opsins | 8IU2-Opsin1LW-Retinal-Gi1/β1/γ2 |
| gi_orexin | 7SQO-OX2-TAK-925-Gi1/β1/γ2 |
| gi_p2y | 7XXI-P2Y12-2MeSADP-Gi2/β1/γ2 |
| gi_peptide | gi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin |
| gi_protein | gi_chemokine gi_chemerin |
| gi_relaxin | 7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2 |
| gi_s1p | 7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2 |
| gi_sensory | gi_opsins |
| gi_somatostatin | 7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2 |
| gi_succinate | 8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1 |
| gnrh1_off | 7BR3-GnRH1-Elagolix |
| gq_amine | gq_muscarinic gq_histamine |
| gq_angiotensin | 7F6G-AT1-SAR1-AngII-Gq/β1/γ2 |
| gq_bombesin | 7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2 |
| gq_bradykinin | 7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2 |
| gq_cck | 8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2 |
| gq_class-a | gq_peptide gq_amine gq_nucleotide |
| gq_histamine | 7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2 |
| gq_kisspeptin | 8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1 |
| gq_muscarinic | 6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2 |
| gq_nucleotide | gq_p2y |
| gq_p2y | 7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2 |
| gq_peptide | gq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin |
| grh_off | gnrh1_off |
| gs_5ht | 7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2 |
| gs_adenosine | 8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 |
| gs_adrenergic | 7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2 |
| gs_amine | gs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine |
| gs_cck | 7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1 |
| gs_class-a | gs_peptide gs_nucleotide gs_amine |
| gs_dopamine | 7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 |
| gs_histamine | 8POK-H2-Histamine-Gs/β1/γ2 |
| gs_melanocortin | 7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 |
| gs_nucleotide | gs_adenosine |
| gs_peptide | gs_cck gs_melanocortin gs_vasop-oxy |
| gs_trace-amine | 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 |
| gs_vasop-oxy | 7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2 |
| h1_off | 8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole |
| h1_on | 7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2 |
| h1_on_gp | 7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2 |
| h2_on | 8POK-H2-Histamine-Gs/β1/γ2 |
| h2_on_gp | 8POK-H2-Histamine-Gs/β1/γ2 |
| h3_on | 8YUU-H3-Histamine-Gi1/β1/γ1 |
| h3_on_gp | 8YUU-H3-Histamine-Gi1/β1/γ1 |
| h4_on | 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2 |
| h4_on_gp | 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2 |
| hca2_on | 8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 |
| hca2_on_gp | 8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 |
| hca_on | hca2_on |
| hca_on_gp | hca2_on_gp |
| histamine_off | h1_off |
| histamine_on | h1_on h2_on h3_on h4_on |
| histamine_on_gp | h1_on_gp h2_on_gp h3_on_gp h4_on_gp |
| kiss1_on | 8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1 |
| kiss1_on_gp | 8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1 |
| kisspeptin_on | kiss1_on |
| kisspeptin_on_gp | kiss1_on_gp |
| kop_off | 4DJH-κ-JDTic |
| kop_on | 8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 |
| kop_on_gp | 8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 |
| leukotriene_off | blt_off cyslt_off |
| leukotriene_on | blt_on |
| leukotriene_on_gp | blt_on_gp |
| lipid_off | cannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off |
| lipid_offon | lipid_off lipid_on |
| lipid_offon_gp | lipid_on_gp lipid_off |
| lipid_on | cannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on |
| lipid_on_gp | cannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp |
| lpa1_off | 4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307 |
| lpa1_on | 7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2 |
| lpa1_on_gp | 7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2 |
| lpa_off | lpa1_off |
| lpa_on | lpa1_on |
| lpa_on_gp | lpa1_on_gp |
| lpl_off | s1p_off lpa_off |
| lpl_on | s1p_on lpa_on |
| lpl_on_gp | s1p_on_gp lpa_on_gp |
| m1_off | 5CXV-M1-Tiotropium |
| m1_on | 6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2 |
| m1_on_gp | 6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2 |
| m2_off | 5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384 |
| m2_on | 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 |
| m2_on_gp | 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 |
| m3_off | 4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589 |
| m3_on | 8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2 |
| m3_on_gp | 8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2 |
| m4_off | 5DSG-M4-Tiotropium |
| m4_on | 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 |
| m4_on_gp | 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 |
| m5_off | 6OL9-M5-Tiotropium |
| mc1_on | 7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 |
| mc1_on_gp | 7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 |
| mc2_on | 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 |
| mc2_on_gp | 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 |
| mc3_on | 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 |
| mc3_on_gp | 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 |
| mc4_on | 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 |
| mc4_on_gp | 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 |
| mc5_on | 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 |
| mc5_on_gp | 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 |
| melanocortin_on | mc1_on mc4_on mc2_on mc3_on mc5_on |
| melanocortin_on_gp | mc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp |
| mop_off | 4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan |
| mop_on | 8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 |
| mop_on_gp | 8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 |
| motilin_on | 8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| motilin_on_gp | 8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| muscarinic_off | m2_off m3_off m4_off m5_off m1_off |
| muscarinic_on | m2_on m3_on m4_on m1_on |
| muscarinic_on_gp | m2_on_gp m3_on_gp m4_on_gp m1_on_gp |
| neuromedin-u_on | nmur1_on nmur2_on |
| neuromedin-u_on_gp | nmur1_on_gp nmur2_on_gp |
| neurotensin_off | nts1_off |
| neurotensin_on | nts1_on |
| neurotensin_on_gp | nts1_on_gp |
| nk1_off | 6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735 |
| nk1_on | 7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| nk1_on_gp | 7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| nk2_on | 7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| nk2_on_gp | 7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| nk3_on | 8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| nk3_on_gp | 8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| nmur1_on | 7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| nmur1_on_gp | 7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| nmur2_on | 7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| nmur2_on_gp | 7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| nop_off | 4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111 |
| nop_on | 8F7X-NOP-Nociceptin-Gi1/β1/γ2 |
| nop_on_gp | 8F7X-NOP-Nociceptin-Gi1/β1/γ2 |
| npy1_off | 5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299 |
| npy1_on | 8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 |
| npy1_on_gp | 8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 |
| npy2_off | 7DDZ-Y2-JNJ-31020028 |
| npy2_on | 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2 |
| npy2_on_gp | 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2 |
| npy4_on | 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 |
| npy4_on_gp | 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 |
| npy_off | npy1_off npy2_off |
| npy_on | npy1_on npy2_on npy4_on |
| npy_on_gp | npy1_on_gp npy2_on_gp npy4_on_gp |
| nts1_off | 7UL2-NTS1-SR48692-Na |
| nts1_on | 6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1 |
| nts1_on_gp | 6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1 |
| nucleotide_off | adenosine_off p2y_off |
| nucleotide_offon | nucleotide_off nucleotide_on |
| nucleotide_offon_gp | nucleotide_on_gp nucleotide_off |
| nucleotide_on | adenosine_on p2y_on |
| nucleotide_on_gp | adenosine_on_gp p2y_on_gp |
| opioid_off | mop_off nop_off dop_off kop_off |
| opioid_on | mop_on nop_on dop_on kop_on |
| opioid_on_gp | mop_on_gp nop_on_gp dop_on_gp kop_on_gp |
| opsin1lw_on | 8IU2-Opsin1LW-Retinal-Gi1/β1/γ2 |
| opsin1lw_on_gp | 8IU2-Opsin1LW-Retinal-Gi1/β1/γ2 |
| opsins_off | rhodopsin_off |
| opsins_on | rhodopsin_on opsin1lw_on |
| opsins_on_gp | rhodopsin_on_gp opsin1lw_on_gp |
| orexin_off | ox2_off ox1_off |
| orexin_on | ox2_on |
| orexin_on_gp | ox2_on_gp |
| ot_off | 6TPK-OT-Retosiban |
| ox1_off | 6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na |
| ox2_off | 5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant |
| ox2_on | 7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| ox2_on_gp | 7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| p2y10_on | 8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2 |
| p2y10_on_gp | 8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2 |
| p2y12_on | 7XXI-P2Y12-2MeSADP-Gi2/β1/γ2 |
| p2y12_on_gp | 7XXI-P2Y12-2MeSADP-Gi2/β1/γ2 |
| p2y1_off | 4XNW-P2Y1-MRS2500 |
| p2y1_on | 7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2 |
| p2y1_on_gp | 7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2 |
| p2y_off | p2y1_off |
| p2y_on | p2y1_on p2y10_on p2y12_on |
| p2y_on_gp | p2y1_on_gp p2y10_on_gp p2y12_on_gp |
| paf_off | 5ZKQ-PAF-ABT-491 |
| peptide_off | cck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off |
| peptide_offon | peptide_off peptide_on |
| peptide_offon_gp | peptide_on_gp peptide_off |
| peptide_on | cck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on |
| peptide_on_gp | cck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp |
| prostanoid_off | ep_off dp_off |
| prostanoid_on | tp_on fp-alpha_on |
| prostanoid_on_gp | tp_on_gp fp-alpha_on_gp |
| protein_off | chemokine_off grh_off |
| protein_offon | protein_off protein_on |
| protein_offon_gp | protein_on_gp protein_off |
| protein_on | chemokine_on chemerin_on |
| protein_on_gp | chemokine_on_gp chemerin_on_gp |
| relaxin_on | rxfp4_on |
| relaxin_on_gp | rxfp4_on_gp |
| rhodopsin_off | 1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal |
| rhodopsin_on | 6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1 |
| rhodopsin_on_gp | 6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1 |
| rxfp4_on | 7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2 |
| rxfp4_on_gp | 7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2 |
| s1p1_off | 3V2W-S1P1-PubChem 51892645 |
| s1p1_on | 7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2 |
| s1p1_on_gp | 7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2 |
| s1p3_on | 7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 |
| s1p3_on_gp | 7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 |
| s1p5_off | 7YXA-S1P5-ONO-5430608 |
| s1p5_on | 7EW1-S1P5-Siponimod-Gi1/β1/γ2 |
| s1p5_on_gp | 7EW1-S1P5-Siponimod-Gi1/β1/γ2 |
| s1p_off | s1p1_off s1p5_off |
| s1p_on | s1p1_on s1p3_on s1p5_on |
| s1p_on_gp | s1p1_on_gp s1p3_on_gp s1p5_on_gp |
| sensory_off | opsins_off |
| sensory_offon | sensory_off sensory_on |
| sensory_offon_gp | sensory_on_gp sensory_on |
| sensory_on | opsins_on |
| sensory_on_gp | opsins_on_gp |
| somatostatin_off | sst2_off |
| somatostatin_on | sst2_on sst4_on sst5_on |
| somatostatin_on_gp | sst2_on_gp sst4_on_gp sst5_on_gp |
| sst2_off | 7XNA-SST2-CYN154806 |
| sst2_on | 7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2 |
| sst2_on_gp | 7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2 |
| sst4_on | 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 |
| sst4_on_gp | 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 |
| sst5_on | 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 |
| sst5_on_gp | 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 |
| succinate_off | 6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554 |
| succinate_on | 8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1 |
| succinate_on_gp | 8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1 |
| ta1_on | 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2 |
| ta1_on_gp | 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2 |
| tachykinin_off | nk1_off |
| tachykinin_on | nk1_on nk2_on nk3_on |
| tachykinin_on_gp | nk1_on_gp nk2_on_gp nk3_on_gp |
| tp_on | 8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| tp_on_gp | 8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2 |
| trace-amine_on | ta1_on |
| trace-amine_on_gp | ta1_on_gp |
| trh_on | 7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2 |
| trh_on_gp | 7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2 |
| v2_on | 7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2 |
| v2_on_gp | 7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2 |
| vasop-oxy_off | ot_off |
| vasop-oxy_on | v2_on |
| vasop-oxy_on_gp | v2_on_gp |