Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.43 3.5125429
2G.HN.47 3.1875426
3G.S1.03 2.71409
4G.S1.05 7.23439
5G.S1.06 3.645168
6G.S2.08 9.305405
7G.S3.03 6.406676157
8G.S3.04 7.274536
9G.S3.06 9.57536
10G.H2.06 4.088336179
11G.H2.07 7.2475409
12G.H2.09 4.4625408
13G.h2s4.01 7.572539
14G.S4.02 6.6375437
15G.S4.04 6.1725439
16G.S4.05 3.4925467
17G.s4h3.04 6.5578
18G.s4h3.05 7.1775479
19G.H3.01 7.7525409
20G.H3.09 6.606539
21G.H3.17 4.45404
22G.H3.18 5.2975439
23G.S5.03 3.618568
24G.S5.05 4.32769
25G.HG.04 4.782578
26G.hgh4.01 4.114574
27G.hgh4.02 4.56578
28G.H4.03 3.2325403
29G.H4.11 2.68478
30G.H4.15 5.496508
31G.S6.02 4.945668
32G.S6.04 6.825468
33G.s6h5.01 5.5975469
34G.H5.03 5.385468
35G.H5.08 9.315158
36G.H5.14 4.8025466
37G.H5.26 5.2075465
38b.1x1 3.7325404
39b.1x15 3.3625407
40b.lhb1x6 5.3483
41b.b1x3 4.3725427
42b.b1x6 8.915429
43b.l1x3 7.68333629
44b.l1x6 8.7175409
45b.b2x5 5.85833627
46b.b3x3 4.5685128
47b.l3x1 7.722539
48b.l3x2 5.1075409
49b.b4x2 5.2425428
50b.b4x3 4.1085127
51b.b4x4 5.245628
52b.b4x6 8.25875829
53b.l4x2 8.805424
54b.b5x3 5.82333629
55b.b5x5 4.70754125
56b.b5x7 5.7075407
57b.l5x1 3.865408
58b.l5x5 10.1986739
59b.b6x5 3.6545126
60b.b7x1 6.225454
61b.b7x2 3.6954128
62b.b8x3 4.0325456
63b.b8x4 5.686506
64b.b9x4 5.918559
65b.l9x3 6.07429759
66b.l9x6 4.8175408
67b.b10x5 4.676559
68b.l10x1 3.6665273
69b.b11x4 5.3775459
70b.l11x2 7.738559
71b.b12x6 9.01333658
72b.l12x1 4.5125456
73b.b13x7 7.77597
74b.l13x3 6.93833699
75b.b15x1 6.245499
76b.l15x1 4.463336177
77b.l15x2 5.38499
78b.b16x4 6.5525496
79b.b16x6 8.01429798
80b.b17x5 5.622547
81b.l17x3 7.42428749
82b.b18x3 4.01448
83b.b18x5 3.326505
84b.l18x1 6.6556286
85b.l18x3 10.92254285
86b.b19x2 5.14286746
87b.b19x4 6.058548
88b.l19x2 5.924549
89b.b20x2 7.354546
90b.b20x4 9.07833648
91b.b20x6 7.14667646
92b.l20x2 7.7225409
93b.b21x1 8.69447
94b.b21x3 3.7375446
95b.b21x5 5.9254254
96b.b21x7 5.291676255
97b.l21x5 4.8854104
98b.b22x5 6.99407
99b.l22x5 7.44667689
100b.b23x6 7.6456107
101b.b24x3 3.845405
102b.b24x4 7.075106
103b.b24x6 4.65754108
104b.b24x7 7.825489
105b.l24x3 4.6975485
106b.b25x3 9.7965105
107b.b25x6 3.24754103
108b.l25x3 9.1145199
109b.l25x6 10.4354218
110b.b26x3 3.25586
111b.l26x5 4.486525
112b.b27x1 3.7825486
113b.l27x1 10.575219
114b.l27x2 7.88254199
115b.b28x3 4.75427
116b.b28x6 10.11409
117b.b28x7 5.3275429
118g.h1x8 3.73254247
119g.h1x11 4.2525409
120g.l1x4 7.266548
121g.ctx3 6.04689
122g.ctx5 4.345489
123g.ctx6 3.46667686
124g.ctx14 4.815629
125g.ctx16 5.67571728
126Lig 11.69932910
127NT.F68 6.895416
128NT.Y73 5.065414
1291x44 7.485415
1301x47 12.0675416
1311x58 5.56254135
1321x61 3.15507
1332x45 5.376516
1342x49 5.08833618
1352x51 8.3285136
1362x54 3.60254137
1372x57 8.18419
1382x58 3.494137
1392x63 4.105415
1402x64 12.4717
1412x67 3.675416
142E1.V176 4.8945182
1433x36 5.102516
1443x38 8.01667618
1453x39 5.89416
1463x41 3.478516
1473x43 8.102518
1483x44 6.72167618
1493x45 4.01515
1503x46 7.27571719
1513x47 3.556519
1523x48 6.145407
1533x49 4.7625417
1543x50 8.19419
1553x53 6.61417
1563x54 3.00254118
1573x58 4.1345117
1584x42 3.7775405
1594x46 4.76417
1604x52 4.15413
1614x53 4.712519
1624x60 8.8418
163E2.Q253 7.1725414
164E2x51 8.9785149
165E2x52 7.525417
166E2.E259 5.35413
1675x36 3.994144
1685x39 8.36667618
1695x40 8.034516
1706x34 5.5775405
1716x51 3.874516
1726x53 6.302519
1736x54 4.0175415
174E3.N329 7.955415
1757x37 6.74667617
1767x47 5.08506
1777x51 4.084505
1787x58 4.14407
1798x67 5.0825104
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b2x5 b.l4x1 15.18284.94YesNo275
2b.b2x3 b.b2x5 24.88696.98NoYes267
3b.b26x2 b.b2x3 25.22384.86NoNo076
4b.b26x1 b.b26x2 25.54233.44NoNo097
5b.b26x1 b.l27x1 25.70664.94NoYes099
6G.H2.09 b.l27x1 43.28547.41YesYes089
7G.H2.09 G.H2.10 74.50334.42YesNo086
8G.H2.10 b.l5x5 71.37055.22NoYes069
9G.h2s4.01 b.l5x5 71.025311.02YesYes399
10G.H2.07 G.h2s4.01 61.50054.01YesYes099
11G.H2.07 G.S3.08 57.01348.58YesNo099
12G.S3.08 G.s3h2.01 56.9281.84NoNo099
13G.S3.07 G.s3h2.01 56.84241.68NoNo099
14G.S1.06 G.S3.07 56.49794.07YesNo1689
15G.S1.06 G.S4.03 55.97512.85YesNo087
16b.l1x5 b.l3x2 10.73196.18NoYes079
17b.l1x5 b.l3x1 10.93313.03NoYes079
18G.S1.05 G.h2s4.01 11.325114.61YesYes399
19G.S1.05 G.S1.07 13.6652.77YesNo099
20G.H2.09 G.H3.17 27.53983.39YesYes084
21G.H3.15 G.H3.17 27.18633.62NoYes084
22G.H3.15 G.H3.18 27.01726.04NoYes389
23G.H3.18 G.S4.02 26.96827.54YesYes397
24G.H2.05 G.H2.07 16.8573NoYes079
25G.H3.12 G.S1.07 13.57352.85NoNo089
26G.H3.01 G.s4h3.06 15.874411.68YesNo098
27G.s4h3.05 G.s4h3.06 17.62933.92YesNo798
28G.s4h3.04 G.s4h3.05 33.488314.94YesYes789
29G.HG.04 G.s4h3.04 11.90726.19YesYes788
30G.H4.11 G.HG.04 15.47112.51YesYes788
31G.H4.11 G.H4.15 30.4192.51YesYes088
32G.H4.15 G.S4.06 37.43977.87YesNo087
33G.S4.04 G.S4.06 38.23433.93YesNo097
34G.H3.08 G.S4.04 16.44086.09NoYes399
35G.H2.05 G.H3.08 16.6274.86NoNo079
36G.HG.15 G.s4h3.04 11.86253.52NoYes778
37G.H4.11 G.HG.15 12.38222.85YesNo787
38G.hgh4.01 G.s4h3.04 16.80264.03YesYes748
39G.H3.02 G.hgh4.01 12.87273.24NoYes084
40G.H3.02 G.H4.15 13.38512.49NoYes088
41G.H3.12 G.S4.04 13.39555.02NoYes389
42G.H3.09 G.S4.04 10.74569.65YesYes399
43G.H3.09 G.S5.02 26.43655.02YesNo396
44G.S4.02 G.S5.02 27.26915.89YesNo376
45G.H3.06 G.H4.15 10.05499.74NoYes078
46G.H3.06 G.h4s6.01 16.72287.05NoNo074
47G.H3.09 G.h4s6.01 16.87414.96YesNo094
48G.S4.03 G.S5.05 54.22382.51NoYes079
49G.H2.09 b.b6x1 99.11532.63YesNo089
50b.b6x1 b.l9x6 99.07463.59NoYes098
51b.l11x1 b.l9x6 19.71352.9NoYes098
52b.b11x6 b.l11x1 19.53233.71NoNo099
53b.b10x3 b.b11x4 11.05753.38NoYes089
54b.b11x4 b.l9x3 11.86825.48YesYes599
55G.H2.06 b.l9x6 1003.58YesYes098
56G.H2.06 b.b18x1 99.5162.8YesNo099
57G.S5.03 G.S5.05 51.43975.02YesYes689
58G.HG.07 G.s4h3.05 14.10346.91NoYes799
59G.HG.07 G.s4h3.02 12.34816.12NoNo799
60G.H3.01 G.s4h3.08 10.58471.21YesNo098
61G.S5.03 G.S6.02 50.33473.63YesYes688
62G.H5.13 G.S6.02 49.18274.6NoYes078
635x64 G.H5.13 49.08054.15NoNo077
645x64 G.H5.20 48.87572.82NoNo078
65G.H5.20 G.H5.25 38.72122.77NoNo086
663x58 G.H5.20 10.06694.28YesNo078
676x45 G.H5.25 38.39555.54NoNo096
68b.b18x1 b.l19x1 99.448113.46NoNo099
69b.l17x5 b.l19x1 99.37695.89NoNo069
70b.b19x6 b.l17x5 57.83413.26NoNo496
71b.b19x6 b.l17x3 57.73556.97NoYes499
72b.b20x6 b.l17x3 40.35034.53YesYes469
73b.b17x7 b.b20x6 48.79988.57NoYes486
74b.b17x5 b.b17x7 48.62158.2YesNo478
75b.b17x5 b.b21x1 13.35756.53YesYes477
76b.1x15 g.h1x11 15.1571.43YesYes079
77b.1x8 g.h1x11 11.59581.58NoYes059
78b.1x8 g.h1x8 10.7051.7NoYes057
79b.l17x5 b.l19x2 41.47132.94NoYes469
80b.b20x4 b.l19x2 40.82563.57YesYes489
81b.b20x4 b.b20x6 40.37264.28YesYes486
82b.1x15 g.l1x4 11.293.76YesYes078
83b.l26x5 g.ctx4 17.91715.03YesNo057
84g.ctx3 g.ctx4 17.54634.83YesNo097
85b.l25x5 b.l27x1 20.60486.78NoYes2179
86b.b24x1 b.l25x5 20.46984.83NoNo047
878x56 b.b24x1 20.29644.96NoNo064
888x56 8x60 12.06742.48NoNo065
898x60 b.l25x1 11.09682.77NoNo053
90b.b24x2 b.l25x1 10.90293.13NoNo053
91b.b19x4 b.l17x3 17.130512.32YesYes489
92b.b19x2 b.b19x4 15.90342.59YesYes468
93b.b19x2 b.l20x1 44.01163.65YesNo466
94b.b16x5 b.l20x1 43.50654.15NoNo456
95b.b16x5 b.l14x6 72.43196.92NoNo453
96b.b16x7 b.l14x6 35.86235.43NoNo493
97b.b16x7 b.l16x3 35.149912.99NoNo493
98b.b17x2 b.l16x3 68.86995.41NoNo033
99b.b17x2 g.h1x13 67.43987.22NoNo031
100g.h1x10 g.h1x13 66.00942.72NoNo091
101b.b17x3 g.h1x10 61.71124.58NoNo059
102b.b16x6 b.b17x3 47.36347.84YesNo985
103b.b15x1 b.b16x6 20.11199.02YesYes998
104b.b11x3 b.b15x1 12.93682.62NoYes059
105b.b19x2 b.b20x6 31.764710.72YesYes466
106b.b16x5 b.b17x5 29.63246.65NoYes457
107b.b17x4 b.l14x6 35.86238.5NoNo453
108b.b17x4 b.l16x3 35.14995.82NoNo453
109b.b13x7 b.b16x6 11.491117.04YesYes978
110b.b16x4 b.b17x3 12.91674.85YesNo965
111b.b16x4 b.l13x3 11.48416.55YesYes969
112b.b16x6 b.l13x3 11.49737.41YesYes989
113b.l13x3 b.l15x2 11.49363.78YesYes999
1145x54 6x45 38.28714.15NoNo079
1155x54 6x51 38.17942.85NoYes076
1166x51 6x54 37.67034.37YesYes165
1175x47 6x54 37.47362.83NoYes175
1183x44 5x47 32.04427.31YesNo187
1193x44 Lig 18.89833.77YesYes180
1203x44 3x47 10.60632.49YesYes189
121b.l4x1 g.ctx16 10.89752.64NoYes258
122b.b11x6 b.l9x3 17.58813.95NoYes599
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
7x37Lig7.611YesYes7010
5x40Lig16.051YesYes6010
6x57Lig4.871NoYes5010
6x53Lig6.171YesYes9010
7x41Lig13.061NoYes8010
3x44Lig3.771YesYes8010
E2.K258Lig13.911NoYes5010
5x39Lig3.211YesYes8010
7x38Lig5.611NoYes6010
7x42Lig4.51NoYes6010
7x45Lig6.821NoYes8010
2x64Lig3.641YesYes7010
3x36Lig6.881YesYes6010
2x67Lig3.821YesYes6010
3x37Lig8.461NoYes8010
E2x52Lig17.591YesYes7010
1x36Lig17.160NoYes4010
2x68Lig6.651NoYes6010
E1.H177Lig5.141NoYes2010
E1.H174Lig8.11NoYes2010
LigNT.V718.311YesNo0401
1x25Lig7.141NoYes1010
LigNT.F684.561YesYes0601
LigNT.N696.811YesNo0301
LigNT.Y733.491YesYes0401
NT.F68NT.P655.781YesNo6812
NT.F68NT.N6912.081YesNo6311
NT.F68NT.Y735.161YesYes6411
NT.V71NT.Y738.831NoYes4411
1x23NT.Y732.780NoYes1421
1x251x272.711NoNo1112
1x301x334.761NoNo1312
1x431x477.651NoYes7622
1x432x649.041NoYes7721
1x442x648.681YesYes5721
1x442x654.131YesNo5622
1x442x6811.271YesNo5621
1x472x6427.511YesYes6721
2x633x324.371YesNo5622
2x633x363.731YesYes5621
2x642x6510.021YesNo7612
2x642x6821.91YesNo7611
2x643x366.011YesYes7611
2x673x324.281YesNo6612
2x673x332.951YesNo6712
2x673x363.651YesYes6611
E1.E175E1.H1749.850NoNo1221
E1.H177E2.Q25314.841NoYes2412
E1.H177E2x524.531NoYes2711
3x33E2x525.190NoYes7721
3x363x405.241YesNo6612
3x374x606.781NoYes8812
3x375x395.811NoYes8811
3x403x442.620NoYes6821
3x415x393.791YesYes6821
3x415x433.071YesNo6722
3x443x472.491YesYes8912
3x445x4313.821YesNo8712
3x445x477.311YesNo8712
3x446x5310.321YesYes8911
3x477x495.441YesNo9922
4x605x376.71YesNo8622
4x605x3913.51YesYes8821
E2x50E2x522.790NoYes9721
E2.D262E2.K2582.770NoNo4521
5x375x3911.491NoYes6821
5x375x407.831NoYes6621
5x395x4012.41YesYes8611
5x435x472.851NoNo7722
5x446x578.790NoNo4521
6x526x533.751NoYes8921
6x527x494.251NoNo8922
6x537x453.381YesNo9811
6x537x497.891YesNo9912
6x56E3.N3299.671NoYes8522
6x567x377.51NoYes8721
6x576x585.241NoNo5512
7x37E3.N3299.671YesYes7512
7x347x374.681NoYes4721
7x347x382.741NoNo4621
7x377x383.771YesNo7611
7x377x417.251YesNo7811
1x30Lig2.431NoYes1010
5x385x402.250NoYes6621
1x397x421.710NoNo7621
5x405x411.641YesNo6512
E1.E178Lig1.160NoYes3010

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
90.91Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
58.06Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
51.61Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
43.24Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
41.94Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
41.94Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
40.00Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
40.00Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
39.39Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
39.39Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
39.39Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
38.89Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
38.24Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
38.24Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
37.50Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
37.50Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
36.36Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
35.29Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
34.48Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
34.38Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
33.33Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
32.35Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
32.35Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
32.35Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
32.35Consensusglp_onOrthosteric Ligandglp1_on glp2_on
32.35Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
31.43Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
31.25Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.25Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
30.77Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
30.30Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
30.30Consensuscalcitonin_onOrthosteric Ligandctlike_on
30.00Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
29.41Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
29.41Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
29.41Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
28.95Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
28.95Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
28.95Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
28.57Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
28.57Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
28.57Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
28.12Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
28.12Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
27.78Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
27.78Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
27.78Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
27.59Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
27.59Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
27.50Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
27.50Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
27.27Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
27.27Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
27.27Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
27.27Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
27.27Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
27.27Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
27.27Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
27.27Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
27.03Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
26.92Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
26.92Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
26.92Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
26.92Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
26.92Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
26.92Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
26.92Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
26.92Consensushca_on_gpOrthosteric Ligandhca2_on_gp
26.83Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
26.67Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
26.67Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
26.47Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
26.47Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
26.47Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
26.32Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
26.32Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
26.19Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
25.93Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
25.93Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
25.93Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
25.93Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
25.93Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
25.93Consensusa3_on_gpOrthosteric Liganda3a_on_gp
25.93Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
25.93Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
25.93Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.93Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.81Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
25.81Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
25.81Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
25.81Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.71Single6FJ3PTH6FJ3-PTH1-PTH
25.71Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
25.71Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
25.71Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
25.71Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
25.71Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
25.00Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
25.00Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
25.00Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
25.00Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
25.00Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
25.00Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
25.00Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
25.00Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
25.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
25.00Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
25.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
25.00Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
25.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
25.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
25.00Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
25.00Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
25.00Single8K5BNiacin8K5B-HCA2-Niacin
25.00Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
25.00Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
25.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
25.00Consensusa2_onOrthosteric Liganda2b_on
25.00Consensusa2_on_gpOrthosteric Liganda2b_on_gp
25.00Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
25.00Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
25.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.00Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
25.00Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
25.00Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
25.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
25.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
24.39Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
24.32Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
24.32Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
24.32Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
24.32Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
24.32Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
24.32Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
24.24Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
24.24Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
24.24Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.24Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
24.14Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
24.14Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
24.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
24.00Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
24.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
23.68Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
23.68Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
23.68Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
23.68Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
23.68Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
23.53Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
23.53Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
23.53Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
23.53Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
23.53Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
23.53Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
23.53Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
23.33Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
23.33Single7UM4AS26747237UM4-5-HT5A-AS2674723
23.33Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
23.33Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
23.33Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
23.26Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
23.08Single2YDOAdenosine2YDO-A2A-Adenosine
23.08Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
23.08Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
23.08Single8K5CAcipimox8K5C-HCA2-Acipimox
23.08Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
23.08Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.08Consensushca_onOrthosteric Ligandhca2_on
22.86Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
22.86Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
22.86Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
22.86Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
22.86Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
22.86Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
22.86Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
22.86Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
22.86Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
22.86Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
22.86Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
22.73Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
22.58Single4UG2CGS216804UG2-A2A-CGS21680
22.58Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
22.58Single7SK9CCX6627SK9-ACKR3-CCX662
22.58Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
22.58Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
22.58Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
22.58Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
22.58Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
22.50Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
22.50Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
22.22Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
22.22Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
22.22Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
22.22Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
22.22Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
22.22Single8K5DGSK2560738K5D-HCA2-GSK256073
22.22Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
22.22Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
22.22Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
22.22Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
22.22Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
22.22Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
22.22Consensusa3_onOrthosteric Liganda3a_on
22.22Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
22.22Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
22.22Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
22.22Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
22.22Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
21.95Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
21.95Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
21.88Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
21.88Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
21.88Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
21.88Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
21.88Single9M4TSilodosin9M4T-Alpha1A-Silodosin
21.88Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
21.88Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
21.88Consensuslpl_onOrthosteric Ligands1p_on lpa_on
21.88Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
21.62Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
21.62Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.62Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
21.62Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
21.62Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
21.62Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
21.62Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
21.62Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.62Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
21.62Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
21.62Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
21.62Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.62Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.62Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
21.62Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
21.43Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
21.43Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
21.43Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
21.43Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
21.43Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
21.43Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
21.43Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
21.43Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
21.43Consensuspth_onOrthosteric Ligandpth1_on pth2_on
21.21Single3QAKUK-4320973QAK-A2A-UK-432097
21.21Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
21.21Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
21.21Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
21.21Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
21.21Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
21.05Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
21.05Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
21.05Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
21.05Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
21.05Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
21.05Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
21.05Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
21.05Consensusbradykinin_onOrthosteric Ligandbk2_on
21.05Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
21.05Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
21.05Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
21.05Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
20.83Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
20.83Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
20.69Single2YDVNECA2YDV-A2A-NECA
20.69Single4UHRCGS216804UHR-A2A-CGS21680
20.69Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
20.69Single5G53NECA5G53-A2A-NECA-Gs
20.69Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
20.69Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
20.69Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
20.69Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
20.69Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
20.69Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
20.69Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.69Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
20.69Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
20.69Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.69Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
20.59Single5WF5UK-4320975WF5-A2A-UK-432097
20.59Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
20.59Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
20.59Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
20.59Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
20.59Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
20.59Consensusangiotensin_onOrthosteric Ligandat1_on
20.59Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
20.59Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
20.59Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
20.59Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
20.51Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
20.51Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
20.00Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
20.00Single3D4STimolol3D4S-β2-Timolol
20.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
20.00Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
20.00Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
20.00Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
20.00Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
20.00Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.00Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
20.00Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
20.00Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
20.00Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
20.00Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
20.00Single8JWY2-1188JWY-A2A-2-118
20.00Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.00Single8XYIVUF106618XYI-CXCR3-VUF10661
20.00Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
20.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.00Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.00Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
20.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
20.00Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
20.00Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
20.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
20.00Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
20.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
20.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
19.57Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
19.51Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
19.44Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
19.44Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
19.44Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
19.44Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
19.44Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
19.44Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
19.44Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
19.44Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
19.44Consensuspac_onOrthosteric Ligandpac1_on
19.35Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
19.35Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
19.35Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
19.35Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
19.35Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
19.35Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
19.35Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
19.35Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
19.35Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
19.35Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
19.35Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
19.23Single3PWHZM-2413853PWH-A2A-ZM-241385
19.23Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
19.23Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
19.23Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
19.23Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
19.23Single8IWESpermidine8IWE-TA9-Spermidine
19.23Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
19.23Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
19.23Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
19.23Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
19.23Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
19.05Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.92Single4XT3Fractalkine4XT3-US28-Fractalkine
18.92Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
18.92Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
18.92Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
18.92Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
18.92Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.92Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
18.92Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
18.92Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
18.92Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
18.92Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
18.92Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
18.75Single3NY9ICI118-5513NY9-β2-ICI118-551
18.75Single5WF6UK-4320975WF6-A2A-UK-432097
18.75Single5ZTYAM102575ZTY-CB2-AM10257
18.75Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
18.75Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
18.75Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
18.75Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
18.75Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
18.75Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
18.75Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
18.75Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
18.75Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
18.75Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
18.75Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
18.52Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
18.52Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
18.52Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
18.52Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
18.52Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
18.52Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
18.52Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
18.52Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
18.52Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
18.52Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
18.52Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
18.52Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
18.52Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
18.52Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
18.52Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
18.52Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
18.42Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
18.42Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
18.42Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
18.42Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
18.18Single4XT1Fractalkine4XT1-US28-Fractalkine
18.18Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
18.18Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
18.18Single7F8XNN90567F8X-CCKA-NN9056
18.18Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
18.18Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
18.18Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
18.18Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
18.18Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
18.18Single8WDTphotoNECA8WDT-A2A-photoNECA
18.18Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
18.18Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
18.18Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
17.95Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
17.95Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
17.86Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
17.86Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
17.86Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
17.86Single5TGZAM65385TGZ-CB1-AM6538
17.86Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
17.86Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
17.86Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
17.86Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
17.86Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
17.86Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
17.86Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
17.86Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
17.86Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
17.86Single9JEAAtropine9JEA-M1-Atropine
17.86Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
17.86Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
17.86Consensusblt_onOrthosteric Ligandblt1_on
17.86Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
17.86Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
17.86Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
17.86Consensusleukotriene_onOrthosteric Ligandblt_on
17.86Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
17.86Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
17.86Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
17.65Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
17.65Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
17.65Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
17.65Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
17.65Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
17.65Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
17.65Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
17.65Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
17.65Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
17.65Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
17.65Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
17.65Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.65Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
17.65Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
17.50Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.50Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.50Consensusbombesin_onOrthosteric Ligandbb2_on
17.50Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
17.50Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.24Single2YCWS-Carazolol2YCW-β1-S-Carazolol
17.24Single5D6LS-Carazolol5D6L-β2-S-Carazolol
17.24Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
17.24Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
17.24Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
17.24Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
17.24Single6PS6Timolol6PS6-β2-Timolol
17.24Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
17.24Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
17.24Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
17.24Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
17.24Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
17.24Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.24Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
17.24Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
17.24Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
17.24Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
17.24Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
17.24Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
17.24Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
17.24Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
17.24Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
17.24Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
17.24Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.24Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
17.24Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
17.24Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
17.24Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.24Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.24Consensustrace-amine_onOrthosteric Ligandta1_on
17.14Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.14Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
17.14Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.14Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
17.14Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
17.07Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
17.07Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
16.67Single4U15Tiotropium4U15-M3-Tiotropium
16.67Single5D5AS-Carazolol5D5A-β2-S-Carazolol
16.67Single5D5BS-Carazolol5D5B-β2-S-Carazolol
16.67Single5V54Methiothepin5V54-5-HT1B-Methiothepin
16.67Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
16.67Single5XR8AM8415XR8-CB1-AM841
16.67Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
16.67Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
16.67Single6J21Aprepitant6J21-NK1-Aprepitant
16.67Single6JODAngiotensin II6JOD-AT2-Angiotensin II
16.67Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
16.67Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.67Single6OL9Tiotropium6OL9-M5-Tiotropium
16.67Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
16.67Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
16.67Single7P2L4YI7P2L-mGlu5-4YI
16.67Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
16.67Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
16.67Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
16.67Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
16.67Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
16.67Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
16.67Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
16.67Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
16.67Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
16.67Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
16.67Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
16.67Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
16.67Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
16.67Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
16.67Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
16.67Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
16.67Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
16.67Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
16.67Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
16.67Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
16.67Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
16.67Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
16.67Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
16.67Single9AS9RS130-1809AS9-5-HT2A-RS130-180
16.67Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
16.67Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
16.67Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
16.67Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
16.67Consensus5ht1_offOrthosteric Ligand5ht1b_off
16.67Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
16.67Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
16.67Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
16.67Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
16.67Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
16.67Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
16.67Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
16.67Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
16.67Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
16.67Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
16.67Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
16.67Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
16.67Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
16.67Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
16.67Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
16.67Consensuslpa_onOrthosteric Ligandlpa1_on
16.67Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
16.67Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.67Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
16.67Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
16.67Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
16.28Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
16.28Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
16.28Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
16.22Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
16.22Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
16.22Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
16.22Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
16.22Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
16.22Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
16.22Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
16.22Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
16.22Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
16.13Single4N4WSANT-14N4W-SMO-SANT-1
16.13Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
16.13Single4XEENeurotensin4XEE-NTS1-Neurotensin
16.13Single4XESNeurotensin4XES-NTS1-Neurotensin
16.13Single5CXVTiotropium5CXV-M1-Tiotropium
16.13Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
16.13Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
16.13Single6OS2TRV0266OS2-AT1-TRV026
16.13Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
16.13Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
16.13Single6YVRNTS8-136YVR-NTS1-NTS8-13
16.13Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
16.13Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
16.13Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
16.13Single7K15MKD0467K15-BLT1-MKD046-Na
16.13Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
16.13Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
16.13Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
16.13Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
16.13Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
16.13Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
16.13Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
16.13Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
16.13Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
16.13Single8JWZAB9288JWZ-A2A-AB928-Na
16.13Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
16.13Single9DGIZ85267113509DGI-CB1-Z8526711350
16.13Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
16.13Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
16.13Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
16.13Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
16.13Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
16.13Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
16.13Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
16.13Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
16.13Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
16.13Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
16.13Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
16.13Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
16.13Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
16.13Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
16.00Single3UZAGTPL92363UZA-A2A-GTPL9236
16.00Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
16.00Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
16.00Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
16.00Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
16.00Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
16.00Single9LRCHistamine9LRC-H4-Histamine
16.00Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
16.00Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
16.00Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
15.79Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
15.79Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
15.79Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
15.79Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
15.79Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
15.79Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
15.79Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
15.79Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
15.62Single4BUONeurotensin4BUO-NTS1-Neurotensin
15.62Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
15.62Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
15.62Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
15.62Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
15.62Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
15.62Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
15.62Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
15.62Single7EZCUKA7EZC-A2A-UKA
15.62Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
15.62Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
15.62Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
15.62Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
15.62Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
15.62Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
15.62Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
15.62Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
15.62Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
15.62Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
15.62Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
15.62Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
15.62Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
15.62Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
15.62Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
15.62Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.62Single8XVJMacitentan8XVJ-ETA-Macitentan
15.62Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
15.62Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
15.62Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
15.62Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
15.62Consensuscck_onOrthosteric Ligandccka_on cckb_on
15.62Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
15.62Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
15.62Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
15.62Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusprostanoid_offOrthosteric Ligandep_off dp_off
15.38Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
15.38Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
15.38Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
15.38Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
15.38Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
15.38Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
15.38Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
15.38Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
15.38Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
15.38Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
15.38Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
15.38Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
15.38Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
15.38Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
15.38Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
15.38Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
15.15Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
15.15Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
15.15Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
15.15Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
15.15Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
15.15Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
15.15Single7XN9L-054,5227XN9-SST2-L-054,522
15.15Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
15.15Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
15.15Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
15.15Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
15.15Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
15.15Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
15.15Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
15.15Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
15.00Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
15.00Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
15.00Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
14.81Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
14.81Single4BWBNeurotensin4BWB-NTS1-Neurotensin
14.81Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
14.81Single5U09Taranabant5U09-CB1-Taranabant
14.81Single5ZKQABT-4915ZKQ-PAF-ABT-491
14.81Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
14.81Single6ME9Ramelteon6ME9-MT2-Ramelteon
14.81Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
14.81Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
14.81Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
14.81Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
14.81Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.81Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.81Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
14.81Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
14.81Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
14.81Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
14.81Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
14.81Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
14.81Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
14.81Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
14.81Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
14.81Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
14.81Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
14.81Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
14.81Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
14.81Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
14.81Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
14.81Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
14.81Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
14.81Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
14.81Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
14.81Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
14.81Single8Y0HVUF114188Y0H-CXCR3-VUF11418
14.81Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
14.81Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
14.81Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
14.81Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
14.81Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
14.81Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
14.81Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
14.81Single9H2XA1IR19H2X-A2A-A1IR1-Na
14.81Consensusalpha2_offOrthosteric Ligandalpha2c_off
14.81Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
14.81Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
14.81Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
14.81Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
14.81Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
14.81Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.81Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.81Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.81Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
14.81Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
14.81Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
14.81Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
14.71Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
14.71Single4IARErgotamine4IAR-5-HT1B-Ergotamine
14.71Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
14.71Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
14.71Single7QA8Peptide7QA8-STE2-Peptide
14.71Single7QA8Peptide7QA8-STE2-Peptide
14.71Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
14.71Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
14.71Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
14.71Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
14.71Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
14.71Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.71Single8XWNCXCL88XWN-CXCR2-CXCL8
14.71Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
14.71Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
14.71Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
14.71Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
14.71Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
14.71Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
14.71Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
14.71Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
14.71Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
14.63Single5GLHEndothelin-15GLH-ETB-Endothelin-1
14.63Single6IGKEndothelin-36IGK-ETB-Endothelin-3
14.63Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
14.29Single3REYXAC3REY-A2A-XAC
14.29Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
14.29Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
14.29Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
14.29Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
14.29Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
14.29Single5IU7Q274563465IU7-A2A-Q27456346-Na
14.29Single5IUBQ274563445IUB-A2A-Q27456344-Na
14.29Single5JTBZM-2413855JTB-A2A-ZM-241385
14.29Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
14.29Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
14.29Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
14.29Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
14.29Single6AQFZM-2413856AQF-A2A-ZM-241385
14.29Single6FFIMMPEP6FFI-mGlu5-MMPEP
14.29Single6HLOAprepitant6HLO-NK1-Aprepitant
14.29Single6MH8ZM-2413856MH8-A2A-ZM-241385
14.29Single6PS0S-Carazolol6PS0-β2-S-Carazolol
14.29Single6PS4ICI118-5516PS4-β2-ICI118-551
14.29Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
14.29Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
14.29Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
14.29Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
14.29Single7AROLUF58337ARO-A2A-LUF5833-Na
14.29Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
14.29Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
14.29Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
14.29Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
14.29Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
14.29Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
14.29Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
14.29Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
14.29Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
14.29Single7UL3Famotidine7UL3-H2-Famotidine
14.29Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
14.29Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
14.29Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
14.29Single7XNACYN1548067XNA-SST2-CYN154806
14.29Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
14.29Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
14.29Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
14.29Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
14.29Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
14.29Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
14.29Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
14.29Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
14.29Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
14.29Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8IHKAcifran8IHK-HCA3-Acifran
14.29Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
14.29Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
14.29Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
14.29Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
14.29Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
14.29Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
14.29Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
14.29Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
14.29Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
14.29Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
14.29Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
14.29Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
14.29Single9AS5Mescaline9AS5-5-HT2A-Mescaline
14.29Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
14.29Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
14.29Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
14.29Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
14.29Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
14.29Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
14.29Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
14.29Consensusa2_offOrthosteric Liganda2a_off
14.29Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
14.29Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
14.29Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
14.29Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
14.29Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
14.29Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
14.29Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
14.29Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
14.29Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
14.29Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
14.29Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
13.95Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
13.95Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.89Single3OE0CVX153OE0-CXCR4-CVX15
13.89Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
13.89Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
13.89Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
13.89Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
13.89Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
13.89Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
13.89Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
13.89Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
13.89Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
13.89Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
13.89Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.89Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
13.89Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
13.89Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
13.89Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
13.89Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
13.89Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
13.89Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
13.79Single2Y04Salbutamol2Y04-β1-Salbutamol
13.79Single3EMLZM-2413853EML-A2A-ZM-241385
13.79Single3NY8ICI118-5513NY8-β2-ICI118-551
13.79Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
13.79Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
13.79Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
13.79Single4EJ4Naltrindole4EJ4-δ-Naltrindole
13.79Single4GBRS-Carazolol4GBR-β2-S-Carazolol
13.79Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
13.79Single4MQSIperoxo4MQS-M2-Iperoxo
13.79Single4QIMANTA XV4QIM-SMO-ANTA XV
13.79Single4QKX35V4QKX-β2-35V
13.79Single4U14Tiotropium4U14-M3-Tiotropium
13.79Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
13.79Single4YAYZD-71554YAY-AT1-ZD-7155
13.79Single5DSGTiotropium5DSG-M4-Tiotropium
13.79Single5IU8Q274563475IU8-A2A-Q27456347-Na
13.79Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
13.79Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
13.79Single5T04Neurotensin5T04-NTS1-Neurotensin
13.79Single5UENDU1725UEN-A1-DU172
13.79Single5UIGCmpd-15UIG-A2A-Cmpd-1
13.79Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
13.79Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
13.79Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
13.79Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
13.79Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
13.79Single6DRXLisuride6DRX-5-HT2B-Lisuride
13.79Single6FFHFenobam6FFH-mGlu5-Fenobam
13.79Single6H7MSalbutamol6H7M-β1-Salbutamol
13.79Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
13.79Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
13.79Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
13.79Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
13.79Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
13.79Single6PS1Timolol6PS1-β2-Timolol
13.79Single6S0LZM-2413856S0L-A2A-ZM-241385
13.79Single6TOTLemborexant6TOT-OX1-Lemborexant
13.79Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
13.79Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
13.79Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
13.79Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
13.79Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
13.79Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
13.79Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
13.79Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
13.79Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
13.79Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
13.79Single7PYRPSB-21157PYR-A2A-PSB-2115
13.79Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
13.79Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
13.79Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
13.79Single7UL4Alvimopan7UL4-μ-Alvimopan
13.79Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
13.79Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
13.79Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
13.79Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
13.79Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
13.79Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
13.79Single8CU6LJ-45178CU6-A2A-LJ-4517
13.79Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
13.79Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
13.79Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
13.79Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
13.79Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
13.79Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
13.79Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
13.79Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
13.79Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
13.79Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
13.79Single8JJOAlprenolol8JJO-β2-Alprenolol
13.79Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
13.79Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
13.79Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
13.79Single8T1WCVN4248T1W-GPR6-CVN424
13.79Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
13.79Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
13.79Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
13.79Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
13.79Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
13.79Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
13.79Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
13.79Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
13.79Single9AS1DMT9AS1-5-HT2A-DMT
13.79Single9CHXS-Carazolol9CHX-β2-S-Carazolol
13.79Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
13.79Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
13.79Single9H37A1IR09H37-A2A-A1IR0-Na
13.79Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
13.79Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
13.79Consensus5ht5_onOrthosteric Ligand5ht5a_on
13.79Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
13.79Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
13.79Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
13.79Consensusalpha2_onOrthosteric Ligandalpha2b_on
13.79Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
13.79Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
13.79Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
13.79Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
13.79Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
13.79Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
13.79Consensusdopamine_offOrthosteric Ligandd2_off d3_off
13.79Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
13.79Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
13.79Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
13.79Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
13.79Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
13.79Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
13.79Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
13.79Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
13.79Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
13.51Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
13.51Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
13.51Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
13.51Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
13.51Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
13.51Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
13.51Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
13.51Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
13.51Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
13.51Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
13.51Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
13.51Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
13.51Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
13.51Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
13.51Consensusvasop-oxy_onOrthosteric Ligandv2_on
13.51Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
13.33Single2RH1S-Carazolol2RH1-β2-S-Carazolol
13.33Single2Y03Isoprenaline2Y03-β1-Isoprenaline
13.33Single4JKVTaladegib4JKV-SMO-Taladegib
13.33Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
13.33Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
13.33Single5C1MBU725C1M-μ-BU72
13.33Single5CGCHTL142425CGC-mGlu5-HTL14242
13.33Single5IUAQ274563485IUA-A2A-Q27456348-Na
13.33Single5JQHS-Carazolol5JQH-β2-S-Carazolol
13.33Single5N2SPSB365N2S-A1-PSB36
13.33Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
13.33Single5TVNLSD5TVN-5-HT2B-LSD
13.33Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
13.33Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
13.33Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
13.33Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
13.33Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
13.33Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
13.33Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
13.33Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
13.33Single6S0QZM-2413856S0Q-A2A-ZM-241385
13.33Single6TP6Filorexant6TP6-OX1-Filorexant
13.33Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
13.33Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
13.33Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
13.33Single7C4SS1P7C4S-S1P3-S1P
13.33Single7C61Ergotamine7C61-5-HT1B-Ergotamine
13.33Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
13.33Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
13.33Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
13.33Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.33Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
13.33Single7SINNPS-21437SIN-CaS-NPS-2143
13.33Single7SINNPS-21437SIN-CaS-NPS-2143
13.33Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
13.33Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
13.33Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
13.33Single7W41PD1762527W41-BB2-PD176252
13.33Single7WC6LSD7WC6-5-HT2A-LSD
13.33Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
13.33Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
13.33Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
13.33Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
13.33Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
13.33Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
13.33Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
13.33Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
13.33Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
13.33Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.33Single8GNEKW-63568GNE-A2A-KW-6356-Na
13.33Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
13.33Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
13.33Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
13.33Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.33Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.33Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
13.33Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
13.33Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
13.33Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
13.33Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
13.33Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9B9ZA1AKO9B9Z-CB1-A1AKO
13.33Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
13.33Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
13.33Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
13.33Single9EHSLUF76029EHS-A3A-LUF7602
13.33Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
13.33Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
13.33Single9HC04YI9HC0-mGlu5-4YI
13.33Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
13.33Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
13.33Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
13.33Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
13.33Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
13.33Consensusadenosine_offOrthosteric Liganda1_off a2_off
13.33Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.33Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.33Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
13.33Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
13.33Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
13.33Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
13.33Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
13.33Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
13.33Consensusamine_offonOrthosteric Ligandamine_off amine_on
13.33Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
13.33Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
13.33Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
13.33Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
13.33Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
13.33Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
13.33Consensusblt_offOrthosteric Ligandblt1_off
13.33Consensusbombesin_offOrthosteric Ligandbb2_off
13.33Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
13.33Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
13.33Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
13.33Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
13.33Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
13.33Consensusep_offOrthosteric Ligandep4_off
13.33Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
13.33Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
13.33Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.33Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
13.33Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
13.33Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
13.33Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
13.33Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
13.16Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
13.16Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
13.16Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
13.16Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.16Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
13.16Single8ZRTET-18ZRT-ETB-ET-1
13.16Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
13.16Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
13.16Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
13.04Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
13.04Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
13.04Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
12.90Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
12.90Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
12.90Single4BV0Neurotensin4BV0-NTS1-Neurotensin
12.90Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
12.90Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
12.90Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
12.90Single5V56TC1145V56-SMO-TC114
12.90Single5V57TC1145V57-SMO-TC114
12.90Single5XRAAM115425XRA-CB1-AM11542
12.90Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
12.90Single6H7JIsoprenaline6H7J-β1-Isoprenaline
12.90Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
12.90Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
12.90Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
12.90Single7B6WCyclazosin7B6W-α1b-Cyclazosin
12.90Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
12.90Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.90Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
12.90Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
12.90Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
12.90Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
12.90Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
12.90Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
12.90Single7PX4PSB-21137PX4-A2A-PSB-2113
12.90Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
12.90Single7TUYGSK682753A7TUY-GPR183-GSK682753A
12.90Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
12.90Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
12.90Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
12.90Single8E0GBU728E0G-μ-BU72
12.90Single8EA0Iperoxo8EA0-M3-Iperoxo
12.90Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
12.90Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
12.90Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
12.90Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
12.90Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
12.90Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
12.90Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
12.90Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
12.90Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
12.90Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
12.90Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
12.90Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
12.90Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
12.90Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
12.90Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
12.90Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
12.90Single9BJKNaloxone9BJK-μ-Naloxone-NAM
12.90Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
12.90Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
12.90Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
12.90Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
12.90Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
12.90Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.90Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
12.90Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
12.90Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
12.90Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
12.90Consensusneurotensin_onOrthosteric Ligandnts1_on
12.90Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.90Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
12.90Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.90Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.82Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
12.82Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
12.82Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
12.82Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
12.82Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
12.82Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
12.50Single4AMIBucindolol4AMI-β1-Bucindolol
12.50Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
12.50Single4LDEBI1671074LDE-β2-BI167107
12.50Single4RWADIPP-NH24RWA-δ-DIPP-NH2
12.50Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
12.50Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
12.50Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
12.50Single5X33BIIL2605X33-BLT1-BIIL260
12.50Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
12.50Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
12.50Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
12.50Single6ZG4HTL00099366ZG4-M1-HTL0009936
12.50Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
12.50Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
12.50Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
12.50Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
12.50Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.50Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
12.50Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
12.50Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
12.50Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
12.50Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
12.50Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
12.50Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
12.50Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
12.50Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single7YITNalfurafine7YIT-κ-Nalfurafine
12.50Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
12.50Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
12.50Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
12.50Single8HS2Fab0468HS2-GPR20-Fab046
12.50Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
12.50Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
12.50Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
12.50Single8JJ8Formoterol8JJ8-β2-Formoterol
12.50Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
12.50Single8PWNTheophylline8PWN-A2A-Theophylline
12.50Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
12.50Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
12.50Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.50Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
12.50Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
12.50Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
12.50Consensusalpha1_offOrthosteric Ligandalpha1a_off
12.50Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
12.50Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
12.50Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
12.50Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
12.50Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.50Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.50Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
12.50Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
12.50Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
12.50Consensuslpa_offOrthosteric Ligandlpa1_off
12.50Consensuslpl_offOrthosteric Ligands1p_off lpa_off
12.50Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
12.50Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
12.50Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
12.50Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
12.50Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
12.50Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
12.50Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.50Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.20Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
12.20Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
12.20Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
12.20Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Consensusendothelin_onOrthosteric Ligandetb_on eta_on
12.20Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
12.12Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
12.12Single5CGDHTL142425CGD-mGlu5-HTL14242
12.12Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
12.12Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
12.12Single6H7LDobutamine6H7L-β1-Dobutamine
12.12Single6IBLArformoterol6IBL-β1-Arformoterol
12.12Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
12.12Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
12.12Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
12.12Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.12Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
12.12Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
12.12Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
12.12Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
12.12Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
12.12Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
12.12Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
12.12Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
12.12Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8XVUCXCL28XVU-CXCR2-CXCL2
12.12Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
12.12Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
12.12Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
12.12Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
12.12Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
12.12Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
12.12Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
12.12Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
12.12Consensuschemerin_onOrthosteric Ligandcml1_on
12.12Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
12.12Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
12.12Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
12.12Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
12.12Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single3RFMCaffeine3RFM-A2A-Caffeine
12.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
12.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
12.00Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
12.00Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
11.76Single6PT3DPI-2876PT3-δ-DPI-287
11.76Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
11.76Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
11.76Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
11.76Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
11.76Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
11.76Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
11.76Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
11.76Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
11.76Single8QJ2pN1628QJ2-MC4-pN162-Gs
11.76Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
11.76Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
11.76Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
11.76Single9JF4PD1683689JF4-BB1-PD168368
11.76Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
11.76Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.63Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
11.63Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
11.63Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
11.63Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
11.54Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
11.54Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
11.54Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
11.54Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
11.54Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
11.54Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.54Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
11.54Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
11.54Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
11.54Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
11.54Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
11.54Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
11.54Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
11.54Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
11.54Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
11.54Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
11.54Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.54Consensus5ht2_onOrthosteric Ligand5ht2b_on
11.54Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
11.54Consensusgi_sensoryOrthosteric Ligandgi_opsins
11.54Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
11.54Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
11.54Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
11.54Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
11.54Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
11.43Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
11.43Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
11.43Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.43Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
11.43Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
11.43Single8IEBA1LYA8IEB-GPR156-A1LYA
11.43Single8IEIA1LYA8IEI-GPR156-A1LYA
11.43Single8IEPA1LYA8IEP-GPR156-A1LYA
11.43Single8IEPA1LYA8IEP-GPR156-A1LYA
11.43Single8KIGSHU91198KIG-MC3-SHU9119-Ca
11.43Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
11.43Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
11.43Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
11.43Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.43Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.43Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
11.43Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
11.43Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Consensussomatostatin_offOrthosteric Ligandsst2_off
11.11Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
11.11Single3OE9IT1t3OE9-CXCR4-IT1t
11.11Single4O9RCyclopamine4O9R-SMO-Cyclopamine
11.11Single5L7IVismodegib5L7I-SMO-Vismodegib
11.11Single6LI0C176LI0-GPR52-C17
11.11Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
11.11Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
11.11Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
11.11Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.11Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
11.11Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
11.11Single7SRQLSD7SRQ-5-HT2B-LSD
11.11Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
11.11Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.11Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
11.11Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
11.11Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
11.11Single8IEBA1LYA8IEB-GPR156-A1LYA
11.11Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
11.11Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
11.11Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
11.11Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
11.11Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
11.11Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
11.11Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
11.11Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
11.11Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
11.11Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
11.11Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
11.11Single9B9Y7DY9B9Y-CB1-7DY
11.11Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
11.11Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
11.11Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
11.11Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
11.11Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
11.11Consensusgq_nucleotideOrthosteric Ligandgq_p2y
11.11Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
11.11Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.11Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
11.11Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
10.81Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
10.81Single6PT2KGCHM076PT2-δ-KGCHM07
10.81Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
10.81Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
10.81Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
10.81Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
10.81Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
10.81Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
10.71Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
10.71Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
10.71Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
10.71Single4QINSAG1.54QIN-SMO-SAG1.5
10.71Single4S0VSuvorexant4S0V-OX2-Suvorexant
10.71Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
10.71Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
10.71Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
10.71Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
10.71Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
10.71Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
10.71Single6ME2Ramelteon6ME2-MT1-Ramelteon
10.71Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
10.71Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
10.71Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
10.71Single6TODEMPA6TOD-OX1-EMPA-Na
10.71Single6TPJSuvorexant6TPJ-OX2-Suvorexant
10.71Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
10.71Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
10.71Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
10.71Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
10.71Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
10.71Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
10.71Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
10.71Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
10.71Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
10.71Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
10.71Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
10.71Single8GNGIstradefylline8GNG-A2A-Istradefylline
10.71Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
10.71Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
10.71Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
10.71Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
10.71Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
10.71Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
10.71Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
10.71Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
10.71Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
10.71Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
10.71Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
10.71Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Consensusangiotensin_offOrthosteric Ligandat1_off
10.71Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.71Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
10.71Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
10.71Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
10.53Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
10.53Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
10.53Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
10.53Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
10.53Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
10.34Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
10.34Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
10.34Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
10.34Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
10.34Single4ZJCSB-6740424ZJC-OX1-SB-674042
10.34Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
10.34Single5UVIZM-2413855UVI-A2A-ZM-241385
10.34Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
10.34Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
10.34Single6KUXRS-799486KUX-α2a-RS-79948
10.34Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
10.34Single6PS5S-Propranolol6PS5-β2-S-Propranolol
10.34Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
10.34Single6TP3Nemorexant6TP3-OX1-Nemorexant
10.34Single6TPGEMPA6TPG-OX2-EMPA
10.34Single6V9SGTPL114036V9S-OX1-GTPL11403
10.34Single6VI4JDTic6VI4-κ-JDTic
10.34Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
10.34Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
10.34Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
10.34Single6ZG9GSK10347026ZG9-M1-GSK1034702
10.34Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
10.34Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
10.34Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
10.34Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
10.34Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
10.34Single7F61PF-036547467F61-H3-PF-03654746
10.34Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single7T32ZM-2413857T32-A2A-ZM-241385
10.34Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
10.34Single7VV6C48/807VV6-MRGPRX2-C48/80
10.34Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
10.34Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
10.34Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
10.34Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
10.34Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
10.34Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
10.34Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
10.34Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
10.34Single8RLNLUF58348RLN-A2A-LUF5834
10.34Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
10.34Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
10.34Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
10.34Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
10.34Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
10.34Single8ZPNAMD31008ZPN-CXCR4-AMD3100
10.34Single9AS3LSD9AS3-5-HT2A-LSD
10.34Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9BA0A1AKN9BA0-CB1-A1AKN
10.34Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
10.34Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
10.34Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
10.34Consensusalpha1_onOrthosteric Ligandalpha1a_on
10.34Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
10.34Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
10.34Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
10.34Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
10.34Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
10.34Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
10.34Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
10.34Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
10.34Consensusopsins_offOrthosteric Ligandrhodopsin_off
10.34Consensussensory_offOrthosteric Ligandopsins_off
10.26Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
10.26Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
10.26Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
10.00Single2Y01Dobutamine2Y01-β1-Dobutamine
10.00Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
10.00Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
10.00Single4DAJTiotropium4DAJ-M3-Tiotropium
10.00Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
10.00Single5DHHSB-6121115DHH-NOP-SB-612111
10.00Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
10.00Single6D27CAY104716D27-DP2-CAY10471
10.00Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
10.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
10.00Single6GPSMK08126GPS-CCR2-MK0812
10.00Single6IIVDaltroban6IIV-TXA2-Daltroban
10.00Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
10.00Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
10.00Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
10.00Single7BU7BI1671077BU7-β1-BI167107
10.00Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.00Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
10.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
10.00Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
10.00Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
10.00Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
10.00Single7V3ZCP559407V3Z-CB1-CP55940
10.00Single7WC7Lisuride7WC7-5-HT2A-Lisuride
10.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
10.00Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
10.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
10.00Single7YXAONO-54306087YXA-S1P5-ONO-5430608
10.00Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.00Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
10.00Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
10.00Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
10.00Single8JXRLSD8JXR-D1-LSD
10.00Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
10.00Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
10.00Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
10.00Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
10.00Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
10.00Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
10.00Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
10.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
10.00Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
10.00Single9IYAONO-97105319IYA-GPR55-ONO-9710531
10.00Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
10.00Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
10.00Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
10.00Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.00Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.00Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
10.00Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
10.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
10.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
10.00Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
10.00Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
9.76Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
9.76Single9KDFRES-701-39KDF-ETB-RES-701-3
9.76Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
9.68Single2Y00Dobutamine2Y00-β1-Dobutamine
9.68Single4NTJAZD12834NTJ-P2Y12-AZD1283
9.68Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
9.68Single5N2RPSB-365N2R-A2A-PSB-36-Na
9.68Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
9.68Single5WIUNemonapride5WIU-D4-Nemonapride
9.68Single5WIVNemonapride5WIV-D4-Nemonapride-Na
9.68Single5WQCEMPA5WQC-OX2-EMPA
9.68Single6D26Fevipiprant6D26-DP2-Fevipiprant
9.68Single6E67BI1671076E67-β2-BI167107-Gs(CT)
9.68Single6GPXMK08126GPX-CCR2-MK0812
9.68Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
9.68Single6LUQHaloperidol6LUQ-D2-Haloperidol
9.68Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
9.68Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
9.68Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
9.68Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
9.68Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
9.68Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
9.68Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
9.68Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.68Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
9.68Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
9.68Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
9.68Single8QOTNanobody-E8QOT-μ-Nanobody-E
9.68Single8S4DCMF-0198S4D-Apelin-CMF-019
9.68Single8TF5Oleic acid8TF5-GPR6-Oleic acid
9.68Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
9.68Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
9.68Single8ZMFA1L108ZMF-5-HT2C-A1L10
9.68Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
9.68Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
9.68Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
9.68Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
9.68Single9HAPTolvaptan9HAP-V2-Tolvaptan
9.68Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
9.68Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
9.68Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
9.68Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
9.68Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
9.68Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
9.68Consensusdp_offOrthosteric Liganddp2_off
9.52Single6IGLIRL16206IGL-ETB-IRL1620
9.52Single8IY6Endothelin-18IY6-ETB-Endothelin-1
9.52Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
9.38Single3P0GBI1671073P0G-β2-BI167107
9.38Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
9.38Single4DJHJDTic4DJH-κ-JDTic
9.38Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
9.38Single5TZRMK86665TZR-FFA1-MK8666
9.38Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
9.38Single6J20Aprepitant6J20-NK1-Aprepitant
9.38Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
9.38Single6OS1TRV0266OS1-AT1-TRV026
9.38Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
9.38Single6TQ7SB-3348676TQ7-OX1-SB-334867
9.38Single6WGTLSD6WGT-5-HT2A-LSD
9.38Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
9.38Single7F1TMIP-1a7F1T-CCR5-MIP-1a
9.38Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
9.38Single7FEECP559407FEE-CB1-CP55940-ZCZ011
9.38Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
9.38Single7R0CAVP7R0C-V2-AVP-Arrestin2
9.38Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
9.38Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
9.38Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
9.38Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
9.38Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
9.38Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
9.38Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
9.38Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
9.38Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
9.38Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
9.38Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
9.38Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
9.38Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
9.38Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
9.38Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
9.38Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
9.38Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
9.38Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
9.38Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
9.38Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
9.38Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
9.38Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
9.38Consensustachykinin_offOrthosteric Ligandnk1_off
9.30Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
9.30Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
9.09Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
9.09Single4PY02MeSATP4PY0-P2Y12-2MeSATP
9.09Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
9.09Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
9.09Single6A93Risperidone6A93-5-HT2A-Risperidone
9.09Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
9.09Single6CM4Risperidone6CM4-D2-Risperidone
9.09Single6IIURamatroban6IIU-TXA2-Ramatroban
9.09Single6KQICP559406KQI-CB1-CP55940-Org27569
9.09Single6MXTSalmeterol6MXT-β2-Salmeterol
9.09Single7DFPSpiperone7DFP-D2-Spiperone
9.09Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
9.09Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
9.09Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
9.09Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
9.09Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
9.09Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
9.09Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8JJLOlodaterol8JJL-β2-Olodaterol
9.09Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
9.09Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
9.09Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
9.09Single8XQJJN2418XQJ-Apelin-JN241
9.09Single8XWACXCL18XWA-CXCR2-CXCL1
9.09Single8XWMCXCL68XWM-CXCR2-CXCL6
9.09Single8XWSCXCL58XWS-CXCR2-CXCL5
9.09Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
9.09Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
9.09Single9BJKNAM9BJK-μ-Naloxone-NAM
9.09Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
9.09Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
9.09Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
9.09Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
9.09Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
9.09Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
9.09Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
9.09Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
9.09Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
9.09Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
8.82Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
8.82Single5X93K-87945X93-ETB-K-8794
8.82Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.82Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
8.82Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
8.82Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
8.82Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
8.82Single8XWFCXCL38XWF-CXCR2-CXCL3
8.82Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
8.82Single8ZPLHF511168ZPL-CXCR4-HF51116
8.82Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
8.82Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.82Consensusendothelin_offOrthosteric Ligandetb_off
8.82Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
8.82Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
8.82Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
8.57Single6KNMJN241-96KNM-Apelin-JN241-9
8.57Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
8.57Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.57Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
8.57Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
8.57Single8X5YAstemizole8X5Y-H1-Astemizole
8.57Single8XQJJN2418XQJ-Apelin-JN241
8.57Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
8.57Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
8.57Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
8.57Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
8.57Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.57Consensuskisspeptin_onOrthosteric Ligandkiss1_on
8.57Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
8.57Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
8.57Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
8.57Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
8.33Single5MZPCaffeine5MZP-A2A-Caffeine-Na
8.33Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
8.33Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
8.33Single8IEIA1LYA8IEI-GPR156-A1LYA
8.33Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.33Single8WKYPG-9348WKY-MC4-PG-934
8.33Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.33Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
8.33Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.33Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.33Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
8.33Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
8.33Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
8.11Single7SK5CXCL127SK5-ACKR3-CXCL12
8.11Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.11Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
8.11Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
8.11Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
8.11Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
8.11Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
8.00Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.00Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.00Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
7.89Single6W25SHU91196W25-MC4-SHU9119-Ca
7.89Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
7.89Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
7.89Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
7.89Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
7.89Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
7.69Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
7.69Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
7.69Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
7.69Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
7.69Single9CHUNoradrenaline9CHU-β2-Noradrenaline
7.69Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
7.69Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
7.69Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
7.69Consensusp2y_offOrthosteric Ligandp2y1_off
7.69Consensussensory_onOrthosteric Ligandopsins_on
7.50Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
7.50Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
7.41Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
7.41Single3OE6IT1t3OE6-CXCR4-IT1t
7.41Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
7.41Single4XNWMRS25004XNW-P2Y1-MRS2500
7.41Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
7.41Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
7.41Single6ME5Agomelatine6ME5-MT1-Agomelatine
7.41Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
7.41Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
7.41Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
7.41Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.41Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.41Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
7.32Single7SK3CXCL127SK3-ACKR3-CXCL12
7.14Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
7.14Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
7.14Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
7.14Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
7.14Single3PBLEticlopride3PBL-D3-Eticlopride
7.14Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
7.14Single6HLLCP999946HLL-NK1-CP99994
7.14Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
7.14Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
7.14Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
7.14Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
7.14Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
7.14Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
7.14Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
7.14Single7UL2SR486927UL2-NTS1-SR48692-Na
7.14Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
7.14Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
7.14Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
7.14Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
7.14Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
7.14Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
7.14Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
7.14Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
7.14Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
7.14Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9AS7Psilocin9AS7-5-HT2A-Psilocin
7.14Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.14Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
7.14Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
7.14Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
7.14Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
7.14Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
7.14Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
7.14Consensusneurotensin_offOrthosteric Ligandnts1_off
7.14Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
6.98Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
6.90Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
6.90Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
6.90Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
6.90Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
6.90Single3ODUIT1t3ODU-CXCR4-IT1t
6.90Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
6.90Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
6.90Single5WS3EMPA5WS3-OX2-EMPA
6.90Single6AKXA4R6AKX-CCR5-A4R
6.90Single6AKYMaraviroc6AKY-CCR5-Maraviroc
6.90Single6B73MP11046B73-κ-MP1104
6.90Single6DS0Ly2660976DS0-5-HT2B-Ly266097
6.90Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
6.90Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
6.90Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
6.90Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.90Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.90Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
6.90Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
6.90Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
6.90Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
6.90Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
6.90Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
6.90Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
6.90Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
6.90Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
6.90Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
6.90Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
6.90Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
6.90Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
6.90Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
6.90Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
6.90Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
6.90Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
6.90Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
6.90Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
6.90Consensusorexin_offOrthosteric Ligandox2_off ox1_off
6.90Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
6.90Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
6.90Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
6.82Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
6.67Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
6.67Single3RZECidoxepin3RZE-H1-Cidoxepin
6.67Single4MBSMaraviroc4MBS-CCR5-Maraviroc
6.67Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
6.67Single6A94Zotepine6A94-5-HT2A-Zotepine
6.67Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
6.67Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
6.67Single6TPKRetosiban6TPK-OT-Retosiban
6.67Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
6.67Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
6.67Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
6.67Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
6.67Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
6.67Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.67Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
6.67Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
6.67Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
6.67Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
6.67Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
6.67Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
6.67Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
6.67Single8K2WAMG4878K2W-CXCR3-AMG487
6.67Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
6.67Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
6.67Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
6.67Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
6.67Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
6.67Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
6.67Single8ZPMAMD0708ZPM-CXCR4-AMD070
6.67Single9ARXSerotonin9ARX-5-HT2A-Serotonin
6.67Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
6.67Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
6.67Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
6.67Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
6.67Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
6.67Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
6.67Consensusvasop-oxy_offOrthosteric Ligandot_off
6.45Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
6.45Single2Y02Carmoterol2Y02-β1-Carmoterol
6.45Single5DHGC-355DHG-NOP-C-35
6.45Single7F83PF-051904577F83-Ghrelin-PF-05190457
6.45Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
6.45Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
6.45Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
6.45Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
6.45Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
6.45Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
6.45Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
6.45Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
6.45Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
6.45Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
6.45Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
6.45Single8X63Mepyramine8X63-H1-Mepyramine
6.45Single8X64Desloratadine8X64-H1-Desloratadine
6.45Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
6.45Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
6.45Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
6.45Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
6.45Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
6.45Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
6.45Consensushistamine_offOrthosteric Ligandh1_off
6.25Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
6.25Single5XPRBosentan5XPR-ETB-Bosentan
6.25Single6HLPNetupitant6HLP-NK1-Netupitant
6.25Single6Z4SSR486926Z4S-NTS1-SR48692
6.25Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
6.25Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
6.25Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
6.25Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
6.25Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
6.25Single8JXSPF-61428JXS-D1-PF-6142
6.25Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
6.25Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
6.25Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
6.25Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
6.25Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
6.25Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
6.25Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
6.06Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
6.06Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
6.06Single6E59L-7607356E59-NK1-L-760735
6.06Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
6.06Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
6.06Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
6.06Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
6.06Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
6.06Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
6.06Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
6.06Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
6.06Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
6.06Single8XVLZibotentan8XVL-ETA-Zibotentan
6.06Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
6.06Single8ZWFJR14a8ZWF-C3aB-JR14a
6.06Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.88Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
5.88Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
5.88Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
5.88Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
5.88Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.88Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.88Consensusorexin_onOrthosteric Ligandox2_on
5.71Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
5.71Single6K1QIRL25006K1Q-ETB-IRL2500
5.71Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
5.71Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
5.71Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
5.71Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.71Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.71Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
5.56Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
5.56Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
5.56Single9IPYJR14a9IPY-C3aB-JR14a
5.56Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
5.41Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
5.41Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.41Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
5.41Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
5.26Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
4.55Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.55Single6D35Cholesterol6D35-SMO-Cholesterol
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.55Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.55Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.55Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
4.55Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.55Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.55Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.55Single7XW7K1-707XW7-TSH-K1-70
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.55Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.55Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.55Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WVXNorrin8WVX-LGR4-Norrin
4.55Single8WVYNorrin8WVY-LGR4-Norrin
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.55Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9KHHNorrin9KHH-LGR4-Norrin
4.55Single9S37NB219S37-LGR4-NB21
4.55Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.35Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.17Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.17Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.17Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.00Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
4.00Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
4.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.00Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.00Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.00Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.00Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.00Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
3.85Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
3.85Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
3.85Single5L7DCholesterol5L7D-SMO-Cholesterol
3.85Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
3.85Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.85Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
3.85Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.70Single3OE8IT1t3OE8-CXCR4-IT1t
3.70Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
3.70Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.70Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
3.70Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.70Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
3.70Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
3.57Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
3.57Single6OBAGTPL110746OBA-β2-S-Alprenolol-GTPL11074
3.57Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
3.57Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.57Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.57Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
3.57Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
3.57Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
3.57Single8JPSCCL78JPS-ACKR1-CCL7
3.57Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
3.57Single8XQPAristolochic acid A8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
3.57Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
3.57Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
3.57Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
3.45Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
3.45Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
3.45Single7CKZMevidalen7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
3.45Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.45Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
3.45Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
3.45Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
3.45Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.45Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
3.45Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.45Single8K9LBMS-9861228K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
3.45Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.45Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.45Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
3.33Single6C1QNDT95137276C1Q-C5a1-PMX53-NDT9513727
3.33Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
3.33Single7BR3Elagolix7BR3-GnRH1-Elagolix
3.33Single7F8ULintitript7F8U-CCKA-Lintitript
3.33Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.33Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.33Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
3.33Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
3.33Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
3.33Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
3.33Single7XRRLemborexant7XRR-OX2-Lemborexant
3.33Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.33Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.33Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
3.33Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.33Single8Y72BMS-9861228Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
3.33Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.33Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.33Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
3.33Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
3.23Single5O9HNDT95137275O9H-C5a1-NDT9513727
3.23Single6IQLL7458706IQL-D4-L745870
3.23Single6TPNHTL66416TPN-OX2-HTL6641
3.23Single6ZINSR486926ZIN-NTS1-SR48692
3.23Single7VODCariprazine7VOD-5-HT2A-Cariprazine
3.23Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Single8IYXYL-3658IYX-GPR34-YL-365
3.23Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.23Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
3.23Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.23Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.23Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.23Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
3.23Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
3.23Consensusgrh_offOrthosteric Ligandgnrh1_off
3.12Single6C1RAvacopan; Na6C1R-C5a1-PMX53-Avacopan; Na
3.12Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
3.12Single7RBTLSN35566727RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
3.12Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
3.12Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
3.12Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
3.12Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
3.03Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
3.03Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
3.03Single8YYXLeukotriene e48YYX-Oxoglutarate-Leukotriene e4-chim(Gi1-CtGq)/β1/γ2
3.03Single9CM7AZ-17299CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
3.03Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
3.03Single9IYBA1D5Q9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
2.94Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
2.94Single8XXVA1D5Q8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
2.86Single8GTMBMK-C2038GTM-CRF1-BMK-C203
2.70Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
2.63Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.63Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.50Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.50Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.44Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.27Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
7TS0 7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
Net Summary
Imin 2.47
Number of Linked Nodes 841
Number of Links 1070
Number of Hubs 179
Number of Links mediated by Hubs 685
Number of Communities 29
Number of Nodes involved in Communities 313
Number of Links involved in Communities 464
Path Summary
Number Of Nodes in MetaPath 123
Number Of Links MetaPath 122
Number of Shortest Paths 1689676
Length Of Smallest Path 3
Average Path Length 31.9929
Length of Longest Path 64
Minimum Path Strength 1.34
Average Path Strength 5.43553
Maximum Path Strength 24.705
Minimum Path Correlation 0.71
Average Path Correlation 0.987947
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.77778
Average % Of Corr. Nodes 47.3127
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 44.953
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
crf_on_gpcrf2_on_gp
crf1_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download crf2_on_gp.zip



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