Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1Lig 7.189082030
21x39 3.62867507
31x43 4.68563406
41x55 3.975424174
51x58 1.99667404
62x39 3.41729407
72x43 4.79417468
82x46 3.99396469
92x50 5.81433569
102x53 8.03813437
112x56 2.96833407
12E1x50 9.47833539
13E1x52 7.59556607
143x29 4.27833436
153x33 7.30063435
163x37 6.42597637
173x40 3.25583437
183x41 4.48104406
193x43 6.34771468
203x46 4.67729469
213x50 6.1495569
223x53 4.589384188
23I2x57 8.571464187
244x61 3.5325434
25E2 14.11641334
26E2x50 5.98333439
27E2x52 7.26187434
285x43 7.85067535
295x47 8.05521409
305x51 4.65417406
315x58 5.70278608
325x64 2.90042405
335x68 3.50938405
34I3 4.765605
356x32 2.53813407
366x48 5.69944639
376x49 6.86479406
386x51 5.07896437
39E3 8.78204933
407x32 2.97771402
417x42 6.12896437
427x47 3.839384168
437x49 6.20533569
447x53 4.95903669
458x50 5.30958408
468x52 1.33875404
47G.HN.30 3.14104407
48G.S1.02 4.659575
49G.S1.06 4.761044219
50G.H1.01 4.0165219
51G.S2.01 4.80854428
52G.S2.08 8.84688475
53G.S3.01 4.81437474
54G.S3.03 8.06217577
55G.S3.04 7.2925427
56G.S3.06 6.89944626
57G.S3.07 3.506254219
58G.s3h2.03 5.07708419
59G.H2.04 4.71083409
60G.H2.06 5.5157619
61G.h2s4.01 7.06687429
62G.S4.02 5.03271427
63G.s4h3.15 2.10854409
64G.H3.09 5.1325709
65G.H3.17 7.97639625
66G.H3.18 6.58021429
67G.S5.03 3.43542408
68G.S5.05 3.8225149
69G.S5.07 5.68562409
70G.HG.08 3.15979406
71G.hgh4.02 6.82455238
72G.hgh4.05 8.13333406
73G.H4.03 5.89504
74G.H4.15 5.34667408
75G.h4s6.02 5.036674247
76G.S6.02 7.87792408
77G.H5.03 4.97555148
78G.H5.08 6.37708478
79G.H5.26 6.12271407
80b.1x4 2.57896408
81b.1x11 3.02937408
82b.1x15 2.63646407
83b.lhb1x6 3.994153
84b.lhb1x11 4.14404
85b.b1x4 4.74396497
86b.l1x3 8.66097649
87b.b2x1 8.65417528
88b.b2x5 6.10583607
89b.b3x3 3.6125408
90b.l3x2 5.88133549
91b.b4x3 4.566254107
92b.b4x6 8.91238749
93b.b5x2 5.98979407
94b.b5x3 6.42403649
95b.b5x5 5.14205
96b.b5x7 5.65333407
97b.l5x1 4.359174108
98b.l5x5 8.01012729
99b.b6x5 4.012226106
100b.l6x5 6.182924124
101b.b7x1 5.896335124
102b.l7x4 4.07438409
103b.b8x3 3.6354126
104b.b8x4 5.104036106
105b.l8x3 3.25708403
106b.b9x3 5.56479406
107b.b9x4 7.46479409
108b.l9x3 7.33861689
109b.l9x6 5.25917718
110b.b10x5 4.85083509
111b.b11x4 5.57062489
112b.l11x2 7.1589
113b.b12x6 8.39536788
114b.b12x7 6.694174289
115b.b13x7 7.86183557
116b.l13x3 7.84083659
117b.l13x6 3.83667619
118b.b15x1 6.61783559
119b.b15x2 6.66292416
120b.l15x1 4.6775417
121b.l15x2 6.33667459
122b.b16x4 8.88667556
123b.b16x5 5.18437415
124b.b16x6 8.76639658
125b.b17x5 6.22361617
126b.b17x7 8.11625418
127b.l17x3 8.96556619
128b.l17x6 5.823519
129b.l17x7 4.37104417
130b.b18x3 5.06063418
131b.l18x1 5.995487136
132b.l18x2 5.780424137
133b.b19x2 6.98867516
134b.b19x4 5.69771418
135b.l19x2 5.66667519
136b.b20x2 5.78958416
137b.b20x4 10.6793518
138b.b20x6 7.76883516
139b.b21x1 6.40708617
140b.b21x2 3.18104406
141b.b21x7 5.79111605
142b.b22x5 5.921674137
143b.l22x5 7.68655159
144b.b23x2 4.77375406
145b.b23x6 6.23345727
146b.l23x1 7.495426
147b.b24x4 7.12063426
148b.b24x6 5.88146428
149b.l24x3 5.83187405
150b.l25x3 8.776835119
151b.l25x6 10.926428
152b.l27x1 10.3164729
153b.l27x2 7.980424119
154b.b28x3 3.97817547
155b.b28x4 8.282294116
156b.b28x6 8.61855119
157b.b28x7 5.78687499
158g.h2x11 9.987924136
159g.ctx3 6.72817509
160g.ctx6 3.873336156
161g.ctx14 5.75875499
162g.ctx15 6.86604499
163g.ctx16 5.22042898
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
11x39 7x42 12.80783.70833YesYes077
22x50 7x46 19.17835.88917YesNo099
32x53 7x46 18.72576.38833YesNo079
42x50 7x49 14.81496.3975YesYes699
57x45 7x49 31.29559.65083NoYes099
66x48 7x45 30.86429.79333YesNo099
76x48 Lig 44.97493.2525YesYes390
82x43 7x54 99.95995.68083YesNo087
92x43 3x46 43.38473.52917YesYes689
103x46 7x53 43.26174.13083YesYes699
113x43 7x53 35.3128.05667YesYes689
123x43 6x44 35.1926.805YesNo089
136x44 6x48 30.79968.18583NoYes099
142x43 3x50 56.51254.97333YesYes689
153x50 7x53 48.42036.00333YesYes699
167x49 7x53 45.98423.1025YesYes699
177x54 8x50 99.997.5375NoYes078
181x61 8x50 99.99995.18333NoYes058
191x61 8x53 10010.1325NoNo055
203x40 3x41 10.14943.16583YesYes076
21E2 Lig 11.15863.88YesYes340
225x68 I3 16.6134.395YesYes055
23G.H5.26 I3 17.70349.00167YesYes075
24G.H5.20 G.H5.26 21.63946.29083NoYes087
25G.H5.20 G.H5.25 21.8164.38417NoNo087
266x37 G.H5.25 21.99245.19167NoNo087
275x58 6x37 22.520510.9408YesNo088
283x50 5x58 18.33677.28583YesYes098
29b.b3x2 b.b4x6 10.32785.50583NoYes459
30b.b2x5 b.b3x2 11.69157.69YesNo075
31b.b2x5 b.l4x1 11.48465.35333YesNo075
32b.l4x1 g.ctx16 11.62855.28083NoYes058
33b.b28x7 g.ctx16 16.74023.92417YesYes998
34b.b28x7 b.lhb1x11 19.80673.6225YesYes094
35b.b25x7 b.lhb1x11 32.38884.71167NoYes074
36b.b25x7 b.b28x6 32.894215.185NoYes079
37b.b27x3 b.b28x6 17.29110.0083NoYes089
38b.b27x3 b.l25x3 83.47627.19083NoYes089
39b.l25x3 b.l27x2 99.76218.92583YesYes1199
40b.l25x4 b.l27x2 1004.43417NoYes059
418x53 b.l25x4 99.99667.045NoNo055
42b.b28x4 b.b28x6 16.55558.12YesYes1169
43b.b28x4 b.l25x3 16.777210.3708YesYes1169
44G.H5.10 G.S5.03 12.55343.52NoYes078
45G.H5.10 G.S6.02 12.74016.33667NoYes078
46G.H5.13 G.S6.02 13.67025.75NoYes078
475x68 G.H5.13 13.85573.18917YesNo057
48b.b8x2 b.b8x4 13.95296.36NoYes086
49b.b8x2 b.b9x3 14.10084.79083NoYes086
50b.b9x3 b.l7x5 14.71696.83333YesNo066
51b.l7x3 b.l7x5 15.02084.66667NoNo096
52b.l5x3 b.l7x3 15.17649.07667NoNo089
53b.l5x3 b.l5x5 15.33212.98833NoYes089
54b.l3x1 b.l5x5 15.86266.39083NoYes299
55b.b2x1 b.l3x1 15.88617.2842YesNo289
56b.b2x1 b.l27x1 15.99616.34833YesYes289
57b.l25x6 b.l27x1 15.835418.825YesYes289
58b.b22x1 b.l25x6 60.87513.7725NoYes288
59b.b22x1 b.b22x2 69.10473.46667NoNo088
60b.b22x2 b.b26x3 69.14375.755NoNo086
61b.b26x3 b.b27x3 68.16493.68583NoNo068
62G.H3.18 G.S4.02 12.83948.375YesYes297
63G.H3.15 G.H3.18 12.96646.44333NoYes289
64G.H3.15 G.H3.17 54.52866.59167NoYes285
65G.H3.17 b.l25x6 50.01113.83333YesYes258
66G.H2.04 G.H2.08 41.55633.8625YesNo098
67G.H2.08 G.H3.15 41.47263.18417NoNo288
68G.s3h2.03 b.l7x4 15.37483.41YesYes099
69G.H2.07 G.s3h2.03 45.89526.66417NoYes099
70G.H2.04 G.H2.07 44.326.08333YesNo099
71G.s3h2.03 b.l9x6 34.56014.69833YesYes198
72G.H2.06 b.l9x6 32.94165.0775YesYes198
73G.H2.06 b.l17x6 32.19437.14417YesYes199
74G.S4.02 G.S5.02 13.01354.53917YesNo076
75G.H3.09 G.S5.02 12.88243.2425YesNo096
76G.H3.09 G.H4.15 11.62253.66083YesYes098
77b.l17x5 b.l17x6 32.08475.03083NoYes169
78b.l17x5 b.l19x2 31.9872.4525NoYes169
79b.l17x3 b.l19x2 21.40614.305YesYes199
80b.b19x4 b.l17x3 11.60037.645YesYes189
81b.b17x7 b.b20x6 25.28511.6108YesYes186
82b.b17x7 b.b21x1 21.50333.9825YesYes187
83b.1x19 b.b21x1 17.28662.38083NoYes067
84b.1x15 b.1x19 16.8082.9225YesNo076
85b.b20x4 b.b20x6 17.79444.36583YesYes186
86b.l21x7 b.l23x1 12.88325.70333NoYes256
87b.b23x6 b.l21x7 12.19384.1425YesNo275
88b.lhb1x11 g.ctx5 12.08515.065YesNo049
89b.l22x1 g.ctx5 11.80094.00167NoNo099
90b.l7x4 b.l9x5 14.61634.2425YesNo098
91b.l11x2 b.l9x5 14.46383.07333YesNo098
92b.l11x2 b.l9x3 13.53728.40167YesYes899
93b.b10x2 b.b14x3 12.52464.62667NoNo065
942x46 7x53 14.85663.51667YesYes699
952x46 2x50 14.67613.50417YesYes699
963x40 6x48 11.25924.595YesYes379
972x53 7x42 13.116912.86YesYes377
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x33Lig13.73673YesYes5010
3x36Lig5.295833NoYes8010
3x37Lig14.74423YesYes7010
3x40Lig3.0553YesYes7010
5x39Lig12.83173NoYes5010
5x43Lig21.55423YesYes5010
6x48Lig3.25253YesYes9010
6x51Lig5.078333YesYes7010
7x34Lig6.605830NoYes5010
E3Lig4.83253YesYes3010
E1Lig4.131673NoYes4010
E2Lig3.883YesYes4010
E2x52Lig4.115833YesYes4010
2x533x368.426673YesNo7821
2x537x4212.863YesYes7722
2x603x324.113NoNo6612
E1x49E215.71170NoYes4421
3x22E28.4953NoYes4421
3x253x294.145833NoYes9621
3x25E2x506.8253NoYes9922
3x294x653.6553YesNo6512
3x29E2x503.23YesYes6912
3x333x375.07753YesYes5711
3x334x577.346673YesNo5712
3x334x613.041673YesYes5412
3x367x423.656673NoYes8712
3x373x415.538333YesYes7612
3x374x5610.04673YesNo7512
3x403x413.165833YesYes7612
4x574x613.834173NoYes7422
4x614x654.515833YesNo4522
4x64E213.85923NoYes5421
4x645x353.420833NoNo5122
4x65E2x527.18250NoYes5421
E2E247.81583YesYes4411
E2E2x504.2253YesYes4912
5x39E2x529.443333NoYes5411
5x31E25.410830NoYes4421
5x35E210.26253NoYes1421
5x27E29.033NoYes3421
5x28E25.928333NoYes5421
5x29E36.66750NoYes1321
5x33E310.84673NoYes1321
5x36E35.39250NoYes4321
5x395x436.929173NoYes5511
5x405x433.250NoYes4521
5x436x524.873YesNo5812
6x446x488.185830NoYes9921
6x486x523.833333YesNo9812
6x487x414.536673YesNo9812
6x487x459.793333YesNo9912
6x517x376.663333YesNo7712
6x517x413.964173YesNo7812
E3E319.19423YesYes3311
7x27E37.495833NoYes3321
7x30E33.0050NoYes4321
7x387x424.290830NoYes6722
2x60Lig3.154173NoYes6010
3x29Lig6.11253YesYes6010
2x533x324.47753YesNo7622
3x406x484.5953YesYes7911
E2E2x528.305833YesYes4411
6x517x384.613YesNo7612
E2x51Lig3.141670NoYes3010
5x32E22.773330NoYes3421
5x436x552.653YesNo5512
5x30E32.413NoYes5321
3x405x502.20753YesNo7912
6x58Lig1.870NoYes4010
3x375x4611.759173YesNo7612
2x67E11.738330NoNo3421
7x31Lig1.69250NoYes4010
3x374x531.393YesNo7812

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
88.89Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
80.95Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
76.19Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
72.73Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
65.00Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
64.00Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
61.90Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
60.87Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
60.00Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
59.09Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
59.09Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
58.33Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
57.89Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
57.89Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
57.89Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
56.52Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
56.52Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
55.56Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
55.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
54.17Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
54.17Consensusangiotensin_onOrthosteric Ligandat1_on
54.17Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
54.17Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
53.85Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
52.63Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
52.00Single6JODAngiotensin II6JOD-AT2-Angiotensin II
52.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
52.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
52.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
52.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
51.85Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
51.85Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
51.85Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
50.00Single6IGLIRL16206IGL-ETB-IRL1620
50.00Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
50.00Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
48.28Single5GLHEndothelin-15GLH-ETB-Endothelin-1
47.83Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
47.62Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
47.37Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
46.43Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
46.15Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
46.15Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
46.15Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
45.83Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
45.83Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
45.83Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
45.83Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
45.83Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
45.83Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
45.83Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
45.45Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
45.16Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
44.44Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
44.44Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
44.44Single8ZRTET-18ZRT-ETB-ET-1
44.44Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
44.00Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
44.00Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
44.00Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
43.48Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
43.48Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
43.48Single7EZCUKA7EZC-A2A-UKA
43.48Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
43.48Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
43.48Consensuschemerin_onOrthosteric Ligandcml1_on
43.48Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
43.33Single6IGKEndothelin-36IGK-ETB-Endothelin-3
42.86Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
42.86Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
42.86Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.86Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
42.86Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
42.86Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
42.86Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
42.86Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
42.31Single5WF5UK-4320975WF5-A2A-UK-432097
42.31Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
42.31Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
42.31Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.31Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
42.31Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
42.31Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
42.31Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
42.31Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
42.11Single6ME9Ramelteon6ME9-MT2-Ramelteon
42.11Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
41.94Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
41.67Single5WF6UK-4320975WF6-A2A-UK-432097
41.67Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
41.67Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
41.67Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
41.67Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
41.67Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
41.67Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
41.67Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
41.38Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
41.38Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
40.91Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
40.91Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
40.91Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
40.91Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.91Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
40.91Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
40.91Consensusrelaxin_onOrthosteric Ligandrxfp4_on
40.91Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
40.91Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
40.91Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
40.74Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
40.74Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
40.74Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
40.00Single4IARErgotamine4IAR-5-HT1B-Ergotamine
40.00Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
40.00Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
40.00Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
40.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
40.00Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
40.00Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
40.00Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
40.00Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
40.00Single8IY6Endothelin-18IY6-ETB-Endothelin-1
40.00Single8WDTphotoNECA8WDT-A2A-photoNECA
40.00Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
40.00Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
40.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
40.00Consensusendothelin_onOrthosteric Ligandetb_on eta_on
40.00Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
40.00Consensuslpl_onOrthosteric Ligands1p_on lpa_on
40.00Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
40.00Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
40.00Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
40.00Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
39.29Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
39.29Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
39.29Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
39.29Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
39.29Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
39.29Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
39.29Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
39.29Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
39.13Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
39.13Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
39.13Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
39.13Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
39.13Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
39.13Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
39.13Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
39.13Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
39.13Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
39.13Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
39.13Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
39.13Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
39.13Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
39.13Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
39.13Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
39.13Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
39.13Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
39.13Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
38.89Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
38.89Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
38.89Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
38.71Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
38.71Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
38.46Single3QAKUK-4320973QAK-A2A-UK-432097
38.46Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
38.46Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
38.46Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
38.46Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
38.46Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
38.46Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
38.46Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
38.46Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
38.10Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
38.10Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
38.10Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
38.10Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
38.10Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
38.10Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
38.10Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
38.10Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
38.10Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
37.93Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
37.93Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
37.93Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
37.93Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
37.50Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
37.50Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
37.50Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
37.50Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
37.50Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
37.50Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
37.50Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
37.50Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
37.50Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
37.50Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.50Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.50Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
37.50Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
37.04Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
37.04Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
37.04Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
37.04Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
37.04Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
37.04Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
36.67Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
36.67Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
36.67Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
36.67Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
36.67Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
36.67Single9KDFRES-701-39KDF-ETB-RES-701-3
36.67Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
36.67Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
36.36Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
36.36Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
36.36Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
36.36Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
36.36Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
36.36Single8JXSPF-61428JXS-D1-PF-6142
36.36Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
36.36Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
36.36Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
36.36Consensusa3_on_gpOrthosteric Liganda3a_on_gp
36.36Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
36.36Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
36.36Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
36.36Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
36.36Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
36.00Single4UG2CGS216804UG2-A2A-CGS21680
36.00Single5ZTYAM102575ZTY-CB2-AM10257
36.00Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
36.00Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
36.00Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
36.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
36.00Single7XN9L-054,5227XN9-SST2-L-054,522
36.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
36.00Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
36.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
36.00Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
36.00Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
36.00Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
36.00Consensuskisspeptin_onOrthosteric Ligandkiss1_on
36.00Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
36.00Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
35.71Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
35.71Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
35.71Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
35.71Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
35.71Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
35.48Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
35.48Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
35.48Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
35.48Consensusbradykinin_onOrthosteric Ligandbk2_on
35.48Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
35.48Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
35.00Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
35.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
35.00Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
35.00Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
34.78Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
34.78Single5V54Methiothepin5V54-5-HT1B-Methiothepin
34.78Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
34.78Single6OS1TRV0266OS1-AT1-TRV026
34.78Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
34.78Single7B6WCyclazosin7B6W-α1b-Cyclazosin
34.78Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
34.78Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
34.78Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
34.78Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
34.78Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
34.78Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
34.78Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
34.78Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
34.78Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
34.78Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
34.78Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
34.78Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
34.78Consensus5ht1_offOrthosteric Ligand5ht1b_off
34.78Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
34.78Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
34.78Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
34.78Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
34.78Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.78Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
34.62Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
34.62Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
34.62Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
34.62Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
34.62Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
34.62Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
34.62Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
34.62Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
34.62Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
34.62Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
34.62Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
34.62Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
34.48Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
34.48Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
34.48Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
34.48Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
34.48Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
34.48Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
34.48Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
34.48Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
34.48Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
34.38Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
34.38Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.38Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.38Consensusbombesin_onOrthosteric Ligandbb2_on
34.38Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
34.38Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
34.38Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.38Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
34.38Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
33.33Single3D4STimolol3D4S-β2-Timolol
33.33Single4RWADIPP-NH24RWA-δ-DIPP-NH2
33.33Single4XEENeurotensin4XEE-NTS1-Neurotensin
33.33Single4XESNeurotensin4XES-NTS1-Neurotensin
33.33Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
33.33Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
33.33Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
33.33Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
33.33Single5UVIZM-2413855UVI-A2A-ZM-241385
33.33Single6A93Risperidone6A93-5-HT2A-Risperidone
33.33Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
33.33Single6MH8ZM-2413856MH8-A2A-ZM-241385
33.33Single6MXTSalmeterol6MXT-β2-Salmeterol
33.33Single6OS2TRV0266OS2-AT1-TRV026
33.33Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
33.33Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
33.33Single6YVRNTS8-136YVR-NTS1-NTS8-13
33.33Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
33.33Single7DFPSpiperone7DFP-D2-Spiperone
33.33Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
33.33Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
33.33Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
33.33Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
33.33Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
33.33Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
33.33Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
33.33Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
33.33Single7T32ZM-2413857T32-A2A-ZM-241385
33.33Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
33.33Single7UL3Famotidine7UL3-H2-Famotidine
33.33Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
33.33Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
33.33Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
33.33Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
33.33Single7XNACYN1548067XNA-SST2-CYN154806
33.33Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
33.33Single7YITNalfurafine7YIT-κ-Nalfurafine
33.33Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
33.33Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
33.33Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
33.33Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
33.33Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
33.33Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
33.33Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
33.33Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
33.33Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
33.33Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
33.33Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
33.33Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
33.33Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
33.33Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
33.33Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
33.33Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
33.33Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
33.33Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
33.33Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
33.33Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
33.33Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
33.33Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
33.33Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
33.33Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
33.33Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
33.33Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
33.33Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
33.33Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
33.33Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
33.33Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
33.33Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
33.33Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
33.33Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
33.33Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
33.33Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
33.33Consensuslpa_offOrthosteric Ligandlpa1_off
33.33Consensuslpl_offOrthosteric Ligands1p_off lpa_off
33.33Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
33.33Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
33.33Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
33.33Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
33.33Consensusorexin_onOrthosteric Ligandox2_on
33.33Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
33.33Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
33.33Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
33.33Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
33.33Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
33.33Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
32.26Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
32.26Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
32.14Single6PT2KGCHM076PT2-δ-KGCHM07
32.14Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
32.14Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
32.14Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
32.14Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
32.14Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
32.00Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
32.00Single4BUONeurotensin4BUO-NTS1-Neurotensin
32.00Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
32.00Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
32.00Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
32.00Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
32.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
32.00Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
32.00Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
32.00Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
32.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
32.00Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
32.00Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
32.00Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
32.00Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
32.00Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
32.00Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
32.00Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
32.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
32.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
32.00Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
32.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
31.82Single3EMLZM-2413853EML-A2A-ZM-241385
31.82Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
31.82Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
31.82Single6DRXLisuride6DRX-5-HT2B-Lisuride
31.82Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
31.82Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
31.82Single6S0LZM-2413856S0L-A2A-ZM-241385
31.82Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
31.82Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
31.82Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
31.82Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
31.82Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
31.82Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
31.82Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
31.82Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
31.82Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
31.82Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
31.82Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
31.82Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
31.82Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
31.82Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
31.82Single9CHXS-Carazolol9CHX-β2-S-Carazolol
31.82Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
31.82Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
31.82Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
31.82Consensusa3_onOrthosteric Liganda3a_on
31.82Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
31.82Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
31.82Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
31.82Consensushca_on_gpOrthosteric Ligandhca2_on_gp
31.82Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
31.82Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
31.58Single6ME5Agomelatine6ME5-MT1-Agomelatine
31.58Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
31.58Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
31.43Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
31.43Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
31.25Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
31.25Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
31.03Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
31.03Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
31.03Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
31.03Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
31.03Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
31.03Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
30.77Single3NY9ICI118-5513NY9-β2-ICI118-551
30.77Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
30.77Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
30.77Single7SK9CCX6627SK9-ACKR3-CCX662
30.77Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
30.77Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
30.77Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
30.77Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single8QJ2pN1628QJ2-MC4-pN162-Gs
30.77Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
30.77Single8XQJJN2418XQJ-Apelin-JN241
30.77Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
30.77Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
30.77Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single2YCWS-Carazolol2YCW-β1-S-Carazolol
30.43Single4NTJAZD12834NTJ-P2Y12-AZD1283
30.43Single5D6LS-Carazolol5D6L-β2-S-Carazolol
30.43Single5IUAQ274563485IUA-A2A-Q27456348-Na
30.43Single5N2RPSB-365N2R-A2A-PSB-36-Na
30.43Single5N2SPSB365N2S-A1-PSB36
30.43Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
30.43Single6D26Fevipiprant6D26-DP2-Fevipiprant
30.43Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
30.43Single6S0QZM-2413856S0Q-A2A-ZM-241385
30.43Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
30.43Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
30.43Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
30.43Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.43Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
30.43Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
30.43Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
30.43Single8GNEKW-63568GNE-A2A-KW-6356-Na
30.43Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
30.43Single8QOTNanobody-E8QOT-μ-Nanobody-E
30.43Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
30.43Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
30.43Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
30.43Single8ZMFA1L108ZMF-5-HT2C-A1L10
30.43Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
30.43Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
30.43Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
30.43Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
30.43Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
30.43Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
30.43Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
30.43Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
30.43Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
30.43Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
30.43Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
30.43Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
30.43Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
30.43Consensusdp_offOrthosteric Liganddp2_off
30.43Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
30.43Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
30.43Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
30.43Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
30.43Consensustrace-amine_onOrthosteric Ligandta1_on
30.30Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
30.00Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
30.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
30.00Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
30.00Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
30.00Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
30.00Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
30.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
30.00Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
30.00Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
30.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
30.00Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
30.00Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
30.00Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
30.00Consensuspac_onOrthosteric Ligandpac1_on
29.63Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
29.63Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
29.63Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
29.63Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
29.63Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
29.63Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.63Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
29.63Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
29.63Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
29.63Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensussomatostatin_offOrthosteric Ligandsst2_off
29.17Single2YDVNECA2YDV-A2A-NECA
29.17Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
29.17Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
29.17Single4UHRCGS216804UHR-A2A-CGS21680
29.17Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
29.17Single5D5AS-Carazolol5D5A-β2-S-Carazolol
29.17Single5D5BS-Carazolol5D5B-β2-S-Carazolol
29.17Single5G53NECA5G53-A2A-NECA-Gs
29.17Single5TZRMK86665TZR-FFA1-MK8666
29.17Single5XR8AM8415XR8-CB1-AM841
29.17Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
29.17Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
29.17Single6J21Aprepitant6J21-NK1-Aprepitant
29.17Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
29.17Single7FEECP559407FEE-CB1-CP55940-ZCZ011
29.17Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
29.17Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
29.17Single7PX4PSB-21137PX4-A2A-PSB-2113
29.17Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
29.17Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
29.17Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
29.17Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
29.17Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
29.17Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.17Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
29.17Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
29.17Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
29.17Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
29.17Single8E0GBU728E0G-μ-BU72
29.17Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
29.17Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
29.17Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
29.17Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
29.17Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
29.17Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
29.17Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
29.17Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
29.17Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
29.17Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
29.17Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
29.17Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
29.17Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
29.17Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
29.17Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
29.17Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
29.17Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
29.17Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
29.17Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
29.17Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
29.17Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Consensusa2_onOrthosteric Liganda2b_on
29.17Consensusa2_on_gpOrthosteric Liganda2b_on_gp
29.17Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
29.17Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
29.17Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
29.17Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
29.17Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
29.17Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
29.17Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
29.17Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
29.17Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
29.17Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
29.17Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
29.17Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Consensusneurotensin_onOrthosteric Ligandnts1_on
29.17Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
29.03Single4XT3Fractalkine4XT3-US28-Fractalkine
29.03Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
29.03Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
29.03Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
29.03Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
29.03Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
29.03Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
29.03Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
28.95Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
28.57Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
28.57Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
28.57Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
28.57Single6B73MP11046B73-κ-MP1104
28.57Single6ME2Ramelteon6ME2-MT1-Ramelteon
28.57Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
28.57Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
28.57Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
28.57Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
28.57Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
28.57Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
28.57Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
28.57Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8GNGIstradefylline8GNG-A2A-Istradefylline
28.57Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
28.57Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
28.57Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
28.57Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
28.57Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
28.57Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
28.57Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
28.57Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
28.57Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
28.57Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
28.57Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
28.57Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
28.57Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
28.57Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
28.57Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
28.57Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
28.57Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
28.57Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
28.57Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
28.57Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
28.12Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
28.12Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
28.12Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
28.00Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
28.00Single4AMIBucindolol4AMI-β1-Bucindolol
28.00Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
28.00Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
28.00Single4PY02MeSATP4PY0-P2Y12-2MeSATP
28.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
28.00Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
28.00Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
28.00Single6KQICP559406KQI-CB1-CP55940-Org27569
28.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
28.00Single6ZG4HTL00099366ZG4-M1-HTL0009936
28.00Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
28.00Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
28.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
28.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
28.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
28.00Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
28.00Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
28.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single8JJLOlodaterol8JJL-β2-Olodaterol
28.00Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.00Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
28.00Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
28.00Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
28.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
28.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
28.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
28.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
28.00Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
28.00Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
28.00Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
28.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
28.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
28.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
28.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
27.59Single3OE0CVX153OE0-CXCR4-CVX15
27.59Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
27.59Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
27.59Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
27.59Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
27.59Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
27.27Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
27.27Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
27.27Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
27.27Single5IU7Q274563465IU7-A2A-Q27456346-Na
27.27Single5JTBZM-2413855JTB-A2A-ZM-241385
27.27Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
27.27Single6A94Zotepine6A94-5-HT2A-Zotepine
27.27Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
27.27Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
27.27Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
27.27Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
27.27Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
27.27Single6TPNHTL66416TPN-OX2-HTL6641
27.27Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
27.27Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
27.27Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
27.27Single7F61PF-036547467F61-H3-PF-03654746
27.27Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
27.27Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
27.27Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
27.27Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
27.27Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
27.27Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
27.27Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
27.27Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
27.27Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
27.27Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
27.27Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
27.27Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
27.27Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
27.27Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
27.27Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
27.27Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
27.27Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
27.27Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.27Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
27.27Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
27.27Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
27.27Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
27.27Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
27.27Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
27.27Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
27.27Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
27.27Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
27.27Consensusa2_offOrthosteric Liganda2a_off
27.27Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
27.27Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
27.27Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
27.27Consensushca_onOrthosteric Ligandhca2_on
27.27Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
27.27Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
27.27Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
26.92Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
26.92Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
26.92Single5X93K-87945X93-ETB-K-8794
26.92Single6IBLArformoterol6IBL-β1-Arformoterol
26.92Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
26.92Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
26.92Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
26.92Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
26.92Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
26.92Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single7UM4AS26747237UM4-5-HT5A-AS2674723
26.92Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
26.92Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
26.92Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
26.92Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
26.92Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
26.92Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
26.92Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
26.92Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
26.92Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
26.92Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
26.92Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
26.92Single8ZPLHF511168ZPL-CXCR4-HF51116
26.92Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
26.92Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
26.92Consensuscck_onOrthosteric Ligandccka_on cckb_on
26.92Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
26.92Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
26.92Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
26.92Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
26.92Consensusendothelin_offOrthosteric Ligandetb_off
26.92Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
26.92Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Consensusprostanoid_offOrthosteric Ligandep_off dp_off
26.67Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.67Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
26.67Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
26.67Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.67Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
26.67Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.67Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
26.67Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.67Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.67Consensusvasop-oxy_onOrthosteric Ligandv2_on
26.67Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
26.47Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
26.47Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
26.32Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
26.32Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
26.09Single2Y04Salbutamol2Y04-β1-Salbutamol
26.09Single3NY8ICI118-5513NY8-β2-ICI118-551
26.09Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
26.09Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
26.09Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
26.09Single4EJ4Naltrindole4EJ4-δ-Naltrindole
26.09Single4GBRS-Carazolol4GBR-β2-S-Carazolol
26.09Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
26.09Single5IU8Q274563475IU8-A2A-Q27456347-Na
26.09Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
26.09Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
26.09Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
26.09Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
26.09Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
26.09Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
26.09Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
26.09Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
26.09Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
26.09Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
26.09Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
26.09Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
26.09Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
26.09Single7PYRPSB-21157PYR-A2A-PSB-2115
26.09Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
26.09Single7UL4Alvimopan7UL4-μ-Alvimopan
26.09Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
26.09Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
26.09Single7V3ZCP559407V3Z-CB1-CP55940
26.09Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
26.09Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
26.09Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
26.09Single7WC7Lisuride7WC7-5-HT2A-Lisuride
26.09Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
26.09Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
26.09Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
26.09Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
26.09Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.09Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
26.09Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
26.09Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
26.09Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
26.09Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
26.09Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
26.09Single8JXRLSD8JXR-D1-LSD
26.09Single8K5DGSK2560738K5D-HCA2-GSK256073
26.09Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
26.09Single8T1WCVN4248T1W-GPR6-CVN424
26.09Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
26.09Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
26.09Single8X64Desloratadine8X64-H1-Desloratadine
26.09Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
26.09Single9AS1DMT9AS1-5-HT2A-DMT
26.09Single9H37A1IR09H37-A2A-A1IR0-Na
26.09Single9IYAONO-97105319IYA-GPR55-ONO-9710531
26.09Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
26.09Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
26.09Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
26.09Consensus5ht5_onOrthosteric Ligand5ht5a_on
26.09Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
26.09Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
26.09Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
26.09Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
26.09Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
26.09Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
26.09Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
26.09Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
26.09Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
26.09Consensusblt_onOrthosteric Ligandblt1_on
26.09Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
26.09Consensuscck_offOrthosteric Ligandccka_off
26.09Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
26.09Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
26.09Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
26.09Consensusdopamine_offOrthosteric Ligandd2_off d3_off
26.09Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
26.09Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
26.09Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
26.09Consensusleukotriene_onOrthosteric Ligandblt_on
26.09Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
25.93Single6KNMJN241-96KNM-Apelin-JN241-9
25.93Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
25.93Single6PT3DPI-2876PT3-δ-DPI-287
25.93Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
25.93Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
25.93Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
25.93Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
25.93Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
25.93Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
25.93Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
25.93Single8X5YAstemizole8X5Y-H1-Astemizole
25.93Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
25.93Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
25.93Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
25.93Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
25.93Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
25.93Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
25.93Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
25.93Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
25.93Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
25.81Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
25.81Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
25.81Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
25.81Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
25.81Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
25.81Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
25.81Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
25.81Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
25.81Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
25.71Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
25.71Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
25.71Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
25.71Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
25.71Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
25.64Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
25.00Single2RH1S-Carazolol2RH1-β2-S-Carazolol
25.00Single2Y03Isoprenaline2Y03-β1-Isoprenaline
25.00Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
25.00Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
25.00Single4XNWMRS25004XNW-P2Y1-MRS2500
25.00Single4XT1Fractalkine4XT1-US28-Fractalkine
25.00Single5C1MBU725C1M-μ-BU72
25.00Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
25.00Single5TVNLSD5TVN-5-HT2B-LSD
25.00Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
25.00Single5WIUNemonapride5WIU-D4-Nemonapride
25.00Single5WIVNemonapride5WIV-D4-Nemonapride-Na
25.00Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
25.00Single5XPRBosentan5XPR-ETB-Bosentan
25.00Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
25.00Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
25.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
25.00Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
25.00Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
25.00Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
25.00Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
25.00Single6PS6Timolol6PS6-β2-Timolol
25.00Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
25.00Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
25.00Single7C61Ergotamine7C61-5-HT1B-Ergotamine
25.00Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
25.00Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
25.00Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
25.00Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
25.00Single7F8XNN90567F8X-CCKA-NN9056
25.00Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
25.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7QA8Peptide7QA8-STE2-Peptide
25.00Single7QA8Peptide7QA8-STE2-Peptide
25.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
25.00Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
25.00Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
25.00Single7W41PD1762527W41-BB2-PD176252
25.00Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
25.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
25.00Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
25.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
25.00Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
25.00Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
25.00Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
25.00Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
25.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
25.00Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
25.00Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
25.00Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
25.00Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
25.00Single8S4DCMF-0198S4D-Apelin-CMF-019
25.00Single8TF5Oleic acid8TF5-GPR6-Oleic acid
25.00Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
25.00Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
25.00Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
25.00Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
25.00Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
25.00Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
25.00Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
25.00Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
25.00Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
25.00Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
25.00Consensusadenosine_offOrthosteric Liganda1_off a2_off
25.00Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
25.00Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
25.00Consensusamine_offonOrthosteric Ligandamine_off amine_on
25.00Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
25.00Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
25.00Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
25.00Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
25.00Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
25.00Consensusbombesin_offOrthosteric Ligandbb2_off
25.00Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
25.00Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
25.00Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
25.00Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
25.00Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
25.00Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
25.00Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
25.00Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
25.00Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
25.00Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
25.00Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
25.00Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
25.00Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
25.00Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
25.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
25.00Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
25.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
24.39Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
24.32Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
24.24Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
24.24Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
24.24Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
24.24Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
24.14Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
24.14Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
24.14Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
24.14Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
24.14Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
24.14Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
24.00Single3P0GBI1671073P0G-β2-BI167107
24.00Single4BV0Neurotensin4BV0-NTS1-Neurotensin
24.00Single4DJHJDTic4DJH-κ-JDTic
24.00Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
24.00Single4U15Tiotropium4U15-M3-Tiotropium
24.00Single6H7JIsoprenaline6H7J-β1-Isoprenaline
24.00Single6J20Aprepitant6J20-NK1-Aprepitant
24.00Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
24.00Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
24.00Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
24.00Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
24.00Single6OL9Tiotropium6OL9-M5-Tiotropium
24.00Single6TQ7SB-3348676TQ7-OX1-SB-334867
24.00Single6WGTLSD6WGT-5-HT2A-LSD
24.00Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
24.00Single7F1TMIP-1a7F1T-CCR5-MIP-1a
24.00Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
24.00Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
24.00Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
24.00Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
24.00Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
24.00Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
24.00Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
24.00Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
24.00Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.00Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
24.00Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
24.00Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
24.00Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
24.00Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.00Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
24.00Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
24.00Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
24.00Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
24.00Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
24.00Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
24.00Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
24.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
24.00Single9BJKNaloxone9BJK-μ-Naloxone-NAM
24.00Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
24.00Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
24.00Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.00Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
24.00Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
24.00Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
24.00Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
24.00Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
24.00Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
24.00Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
24.00Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
24.00Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
24.00Consensuslpa_onOrthosteric Ligandlpa1_on
24.00Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
24.00Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
24.00Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
24.00Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
24.00Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
23.81Single3OE9IT1t3OE9-CXCR4-IT1t
23.81Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
23.81Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
23.81Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
23.81Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
23.81Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
23.81Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
23.81Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
23.81Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
23.81Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
23.81Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
23.81Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
23.81Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
23.81Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
23.81Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
23.81Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.81Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
23.81Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
23.81Consensusgq_nucleotideOrthosteric Ligandgq_p2y
23.81Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
23.68Consensuspth_onOrthosteric Ligandpth1_on pth2_on
23.53Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
23.53Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
23.53Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
23.53Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
23.53Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
23.53Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
23.53Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
23.53Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
23.33Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
23.33Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
23.33Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
23.33Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
23.33Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
23.33Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
23.33Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
23.33Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
23.33Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
23.33Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
23.08Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
23.08Single4LDEBI1671074LDE-β2-BI167107
23.08Single5CXVTiotropium5CXV-M1-Tiotropium
23.08Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
23.08Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
23.08Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
23.08Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
23.08Single7K15MKD0467K15-BLT1-MKD046-Na
23.08Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
23.08Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
23.08Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
23.08Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
23.08Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
23.08Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
23.08Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
23.08Single8JJ8Formoterol8JJ8-β2-Formoterol
23.08Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
23.08Single8JWY2-1188JWY-A2A-2-118
23.08Single8JWZAB9288JWZ-A2A-AB928-Na
23.08Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
23.08Single8XQJJN2418XQJ-Apelin-JN241
23.08Single8XWACXCL18XWA-CXCR2-CXCL1
23.08Single8XWMCXCL68XWM-CXCR2-CXCL6
23.08Single8XWSCXCL58XWS-CXCR2-CXCL5
23.08Single8XYIVUF106618XYI-CXCR3-VUF10661
23.08Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Single9DGIZ85267113509DGI-CB1-Z8526711350
23.08Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
23.08Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
23.08Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
23.08Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
23.08Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
23.08Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
23.08Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
23.08Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
23.08Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
23.08Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
23.08Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
23.08Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
22.86Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
22.86Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
22.86Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
22.73Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
22.73Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
22.73Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
22.73Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
22.73Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
22.73Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
22.73Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
22.73Single4BWBNeurotensin4BWB-NTS1-Neurotensin
22.73Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
22.73Single6AKXA4R6AKX-CCR5-A4R
22.73Single6AKYMaraviroc6AKY-CCR5-Maraviroc
22.73Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
22.73Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
22.73Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
22.73Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
22.73Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
22.73Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
22.73Single7F8YDevazepide7F8Y-CCKA-Devazepide
22.73Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
22.73Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
22.73Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
22.73Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
22.73Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
22.73Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
22.73Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
22.73Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
22.73Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
22.73Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
22.73Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
22.73Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
22.73Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
22.73Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
22.73Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
22.73Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
22.73Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
22.73Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
22.73Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
22.73Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
22.73Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
22.73Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
22.73Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
22.73Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
22.73Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
22.73Single8Y0HVUF114188Y0H-CXCR3-VUF11418
22.73Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
22.73Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
22.73Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
22.73Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
22.73Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
22.73Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
22.73Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
22.73Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
22.73Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
22.73Consensusorexin_offOrthosteric Ligandox2_off ox1_off
22.73Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
22.73Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
22.73Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
22.58Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
22.58Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
22.58Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
22.58Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
22.58Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
22.58Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
22.58Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
22.58Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
22.58Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
22.22Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
22.22Single6K1QIRL25006K1Q-ETB-IRL2500
22.22Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
22.22Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
22.22Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
22.22Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
22.22Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
22.22Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
22.22Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
22.22Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
22.22Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
22.22Single8XVUCXCL28XVU-CXCR2-CXCL2
22.22Single8XWFCXCL38XWF-CXCR2-CXCL3
22.22Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
22.22Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
22.22Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
22.22Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
22.22Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
22.22Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
22.22Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
22.22Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
21.88Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
21.88Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
21.88Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
21.88Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
21.88Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
21.88Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
21.74Single2YDOAdenosine2YDO-A2A-Adenosine
21.74Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
21.74Single3RZECidoxepin3RZE-H1-Cidoxepin
21.74Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
21.74Single4MBSMaraviroc4MBS-CCR5-Maraviroc
21.74Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
21.74Single4ZJCSB-6740424ZJC-OX1-SB-674042
21.74Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
21.74Single5IUBQ274563445IUB-A2A-Q27456344-Na
21.74Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
21.74Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
21.74Single6AQFZM-2413856AQF-A2A-ZM-241385
21.74Single6KUXRS-799486KUX-α2a-RS-79948
21.74Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
21.74Single6PS0S-Carazolol6PS0-β2-S-Carazolol
21.74Single6PS4ICI118-5516PS4-β2-ICI118-551
21.74Single6PS5S-Propranolol6PS5-β2-S-Propranolol
21.74Single6TPGEMPA6TPG-OX2-EMPA
21.74Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
21.74Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
21.74Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
21.74Single7AROLUF58337ARO-A2A-LUF5833-Na
21.74Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
21.74Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
21.74Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
21.74Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
21.74Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
21.74Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
21.74Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
21.74Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
21.74Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
21.74Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
21.74Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
21.74Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
21.74Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
21.74Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
21.74Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
21.74Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
21.74Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
21.74Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
21.74Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
21.74Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
21.74Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
21.74Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
21.74Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
21.74Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
21.74Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
21.74Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
21.74Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
21.74Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
21.74Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
21.74Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
21.74Single8IHKAcifran8IHK-HCA3-Acifran
21.74Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
21.74Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
21.74Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
21.74Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
21.74Single8K5CAcipimox8K5C-HCA2-Acipimox
21.74Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
21.74Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
21.74Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
21.74Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
21.74Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
21.74Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
21.74Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
21.74Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
21.74Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
21.74Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
21.74Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
21.74Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
21.74Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
21.74Consensusalpha1_onOrthosteric Ligandalpha1a_on
21.74Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
21.74Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
21.74Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
21.74Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
21.74Consensusgrh_offOrthosteric Ligandgnrh1_off
21.74Consensusopsins_offOrthosteric Ligandrhodopsin_off
21.74Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
21.74Consensussensory_offOrthosteric Ligandopsins_off
21.62Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
21.62Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
21.43Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
21.43Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
21.43Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
21.43Single9IPYJR14a9IPY-C3aB-JR14a
21.43Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
21.43Single9JF4PD1683689JF4-BB1-PD168368
21.43Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
21.43Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Single6FJ3PTH6FJ3-PTH1-PTH
21.21Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
21.21Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
21.21Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
21.21Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
21.21Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
21.21Single7SK3CXCL127SK3-ACKR3-CXCL12
21.21Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
21.21Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
21.21Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
21.21Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
21.05Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
21.05Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
21.05Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
21.05Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
21.05Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
21.05Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
21.05Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.83Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
20.83Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
20.83Single2Y02Carmoterol2Y02-β1-Carmoterol
20.83Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
20.83Single4MQSIperoxo4MQS-M2-Iperoxo
20.83Single4QKX35V4QKX-β2-35V
20.83Single4U14Tiotropium4U14-M3-Tiotropium
20.83Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
20.83Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
20.83Single5T04Neurotensin5T04-NTS1-Neurotensin
20.83Single6D27CAY104716D27-DP2-CAY10471
20.83Single6H7MSalbutamol6H7M-β1-Salbutamol
20.83Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
20.83Single6PS1Timolol6PS1-β2-Timolol
20.83Single6TOTLemborexant6TOT-OX1-Lemborexant
20.83Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
20.83Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
20.83Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
20.83Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
20.83Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
20.83Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
20.83Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
20.83Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
20.83Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
20.83Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
20.83Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
20.83Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
20.83Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
20.83Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
20.83Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
20.83Single8CU6LJ-45178CU6-A2A-LJ-4517
20.83Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
20.83Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
20.83Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
20.83Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
20.83Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
20.83Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
20.83Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
20.83Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
20.83Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
20.83Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
20.83Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
20.83Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
20.83Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
20.83Single8JJOAlprenolol8JJO-β2-Alprenolol
20.83Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
20.83Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
20.83Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
20.83Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
20.83Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
20.83Single8X63Mepyramine8X63-H1-Mepyramine
20.83Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
20.83Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
20.83Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
20.83Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
20.83Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
20.83Single9JEAAtropine9JEA-M1-Atropine
20.83Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
20.83Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
20.83Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
20.83Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
20.83Consensusalpha2_onOrthosteric Ligandalpha2b_on
20.83Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
20.83Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
20.83Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
20.83Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
20.83Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
20.83Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
20.83Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
20.83Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
20.83Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
20.83Consensushistamine_offOrthosteric Ligandh1_off
20.83Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
20.83Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
20.83Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
20.69Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
20.69Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
20.69Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
20.69Single8IEBA1LYA8IEB-GPR156-A1LYA
20.69Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
20.69Single8WKYPG-9348WKY-MC4-PG-934
20.69Single8XWNCXCL88XWN-CXCR2-CXCL8
20.69Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
20.69Single9M4TSilodosin9M4T-Alpha1A-Silodosin
20.69Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
20.69Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
20.59Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
20.59Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
20.59Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
20.59Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
20.59Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
20.59Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
20.59Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
20.59Consensusglp_onOrthosteric Ligandglp1_on glp2_on
20.59Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
20.00Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
20.00Single5JQHS-Carazolol5JQH-β2-S-Carazolol
20.00Single5WQCEMPA5WQC-OX2-EMPA
20.00Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
20.00Single6E67BI1671076E67-β2-BI167107-Gs(CT)
20.00Single6HLOAprepitant6HLO-NK1-Aprepitant
20.00Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
20.00Single6LUQHaloperidol6LUQ-D2-Haloperidol
20.00Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
20.00Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
20.00Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
20.00Single6TP6Filorexant6TP6-OX1-Filorexant
20.00Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
20.00Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
20.00Single7C4SS1P7C4S-S1P3-S1P
20.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
20.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
20.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
20.00Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
20.00Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.00Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
20.00Single7SK5CXCL127SK5-ACKR3-CXCL12
20.00Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
20.00Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
20.00Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
20.00Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
20.00Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
20.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
20.00Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
20.00Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
20.00Single8IEBA1LYA8IEB-GPR156-A1LYA
20.00Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
20.00Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
20.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
20.00Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
20.00Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
20.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
20.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
20.00Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
20.00Single9EHSLUF76029EHS-A3A-LUF7602
20.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
20.00Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
20.00Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
20.00Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
20.00Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
20.00Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
20.00Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
20.00Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
20.00Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
20.00Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
20.00Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
20.00Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
20.00Consensusp2y_offOrthosteric Ligandp2y1_off
20.00Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
20.00Consensussensory_onOrthosteric Ligandopsins_on
20.00Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
20.00Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
19.51Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
19.44Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
19.44Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
19.44Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
19.35Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
19.35Single6W25SHU91196W25-MC4-SHU9119-Ca
19.35Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
19.35Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
19.35Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
19.23Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
19.23Single5XRAAM115425XRA-CB1-AM11542
19.23Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
19.23Single6E59L-7607356E59-NK1-L-760735
19.23Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
19.23Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
19.23Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
19.23Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
19.23Single7TUYGSK682753A7TUY-GPR183-GSK682753A
19.23Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
19.23Single8EA0Iperoxo8EA0-M3-Iperoxo
19.23Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
19.23Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
19.23Single8XVLZibotentan8XVL-ETA-Zibotentan
19.23Single8ZWFJR14a8ZWF-C3aB-JR14a
19.23Single9AS9RS130-1809AS9-5-HT2A-RS130-180
19.23Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
19.23Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.23Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
19.23Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
19.23Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
19.23Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
19.23Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
19.23Consensustachykinin_offOrthosteric Ligandnk1_off
19.05Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
19.05Single3OE6IT1t3OE6-CXCR4-IT1t
19.05Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
19.05Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
19.05Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
19.05Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
19.05Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
19.05Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
19.05Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
19.05Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
19.05Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
19.05Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
19.05Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
19.05Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
19.05Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
19.05Consensus5ht2_onOrthosteric Ligand5ht2b_on
19.05Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.05Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
19.05Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
18.92Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
18.92Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
18.75Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
18.75Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
18.75Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
18.75Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
18.60Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
18.52Single4N4WSANT-14N4W-SMO-SANT-1
18.52Single6CM4Risperidone6CM4-D2-Risperidone
18.52Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
18.52Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
18.52Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
18.52Consensusalpha1_offOrthosteric Ligandalpha1a_off
18.52Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
18.52Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
18.42Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
18.42Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
18.18Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
18.18Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
18.18Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
18.18Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
18.18Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
18.18Single3PBLEticlopride3PBL-D3-Eticlopride
18.18Single4O9RCyclopamine4O9R-SMO-Cyclopamine
18.18Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
18.18Single6HLLCP999946HLL-NK1-CP99994
18.18Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
18.18Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
18.18Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
18.18Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
18.18Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
18.18Single7SRQLSD7SRQ-5-HT2B-LSD
18.18Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
18.18Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
18.18Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
18.18Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
18.18Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
18.18Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
18.18Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
18.18Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
18.18Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
18.18Single8K5BNiacin8K5B-HCA2-Niacin
18.18Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
18.18Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
18.18Single9AS7Psilocin9AS7-5-HT2A-Psilocin
18.18Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
18.18Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
18.18Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
18.18Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
18.18Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
18.18Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
17.95Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
17.95Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
17.86Single6H7LDobutamine6H7L-β1-Dobutamine
17.86Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
17.86Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
17.86Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
17.86Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8XVJMacitentan8XVJ-ETA-Macitentan
17.86Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
17.86Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
17.86Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
17.78Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
17.65Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
17.65Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
17.65Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
17.65Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
17.50Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.50Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
17.50Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
17.39Single3ODUIT1t3ODU-CXCR4-IT1t
17.39Single3PWHZM-2413853PWH-A2A-ZM-241385
17.39Single4QINSAG1.54QIN-SMO-SAG1.5
17.39Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
17.39Single5WS3EMPA5WS3-OX2-EMPA
17.39Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
17.39Single6DS0Ly2660976DS0-5-HT2B-Ly266097
17.39Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
17.39Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
17.39Single6TODEMPA6TOD-OX1-EMPA-Na
17.39Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
17.39Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
17.39Single7BR3Elagolix7BR3-GnRH1-Elagolix
17.39Single7F8ULintitript7F8U-CCKA-Lintitript
17.39Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
17.39Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
17.39Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
17.39Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
17.39Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
17.39Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
17.39Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
17.39Single7XRRLemborexant7XRR-OX2-Lemborexant
17.39Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
17.39Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
17.39Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
17.39Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
17.39Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
17.39Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
17.39Single8IWESpermidine8IWE-TA9-Spermidine
17.39Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
17.39Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
17.39Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
17.39Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
17.39Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
17.39Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
17.39Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
17.39Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
17.39Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
17.39Single9H2XA1IR19H2X-A2A-A1IR1-Na
17.39Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
17.39Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
17.39Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
17.39Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Consensusalpha2_offOrthosteric Ligandalpha2c_off
17.39Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
17.39Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
17.39Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
17.39Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
17.39Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
17.39Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
17.39Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
17.39Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
17.39Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
17.39Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
17.39Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
17.39Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
17.39Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
17.24Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
17.24Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
17.24Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
17.24Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
17.14Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
17.14Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
17.14Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
17.14Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
17.14Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
17.14Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
17.14Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
17.14Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
17.14Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
17.07Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
16.67Single3REYXAC3REY-A2A-XAC
16.67Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
16.67Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
16.67Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
16.67Single6FFIMMPEP6FFI-mGlu5-MMPEP
16.67Single6IQLL7458706IQL-D4-L745870
16.67Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
16.67Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
16.67Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
16.67Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
16.67Single6TPKRetosiban6TPK-OT-Retosiban
16.67Single6V9SGTPL114036V9S-OX1-GTPL11403
16.67Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
16.67Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
16.67Single6ZG9GSK10347026ZG9-M1-GSK1034702
16.67Single6ZINSR486926ZIN-NTS1-SR48692
16.67Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
16.67Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
16.67Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
16.67Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
16.67Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
16.67Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
16.67Single7VODCariprazine7VOD-5-HT2A-Cariprazine
16.67Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
16.67Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
16.67Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
16.67Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
16.67Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
16.67Single8IEIA1LYA8IEI-GPR156-A1LYA
16.67Single8IEIA1LYA8IEI-GPR156-A1LYA
16.67Single8IEPA1LYA8IEP-GPR156-A1LYA
16.67Single8IEPA1LYA8IEP-GPR156-A1LYA
16.67Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.67Single8KIGSHU91198KIG-MC3-SHU9119-Ca
16.67Single8RLNLUF58348RLN-A2A-LUF5834
16.67Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
16.67Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
16.67Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8ZPMAMD0708ZPM-CXCR4-AMD070
16.67Single8ZPNAMD31008ZPN-CXCR4-AMD3100
16.67Single9ARXSerotonin9ARX-5-HT2A-Serotonin
16.67Single9AS3LSD9AS3-5-HT2A-LSD
16.67Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9AS5Mescaline9AS5-5-HT2A-Mescaline
16.67Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
16.67Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
16.67Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
16.67Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
16.67Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
16.67Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
16.67Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
16.67Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
16.67Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
16.67Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
16.67Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
16.67Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
16.67Consensusvasop-oxy_offOrthosteric Ligandot_off
16.13Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
16.13Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
16.13Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
16.00Single2Y01Dobutamine2Y01-β1-Dobutamine
16.00Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
16.00Single4DAJTiotropium4DAJ-M3-Tiotropium
16.00Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
16.00Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
16.00Single4YAYZD-71554YAY-AT1-ZD-7155
16.00Single5DHGC-355DHG-NOP-C-35
16.00Single5DSGTiotropium5DSG-M4-Tiotropium
16.00Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
16.00Single5TGZAM65385TGZ-CB1-AM6538
16.00Single5UENDU1725UEN-A1-DU172
16.00Single5UIGCmpd-15UIG-A2A-Cmpd-1
16.00Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
16.00Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
16.00Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
16.00Single6FFHFenobam6FFH-mGlu5-Fenobam
16.00Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
16.00Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
16.00Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
16.00Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single7BU7BI1671077BU7-β1-BI167107
16.00Single7F83PF-051904577F83-Ghrelin-PF-05190457
16.00Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
16.00Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
16.00Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
16.00Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
16.00Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
16.00Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
16.00Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
16.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
16.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
16.00Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
16.00Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
16.00Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
16.00Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
15.79Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
15.79Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
15.79Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
15.79Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
15.62Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
15.62Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
15.62Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
15.62Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.62Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.38Single2Y00Dobutamine2Y00-β1-Dobutamine
15.38Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
15.38Single6HLPNetupitant6HLP-NK1-Netupitant
15.38Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
15.38Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
15.38Single6Z4SSR486926Z4S-NTS1-SR48692
15.38Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
15.38Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
15.38Single7SINNPS-21437SIN-CaS-NPS-2143
15.38Single7SINNPS-21437SIN-CaS-NPS-2143
15.38Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
15.38Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
15.38Single7WC6LSD7WC6-5-HT2A-LSD
15.38Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
15.38Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
15.38Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
15.38Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
15.38Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
15.38Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
15.38Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
15.38Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
15.38Single9HAPTolvaptan9HAP-V2-Tolvaptan
15.38Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
15.38Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
15.38Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
15.38Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
15.38Consensusblt_offOrthosteric Ligandblt1_off
15.38Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
15.15Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
15.15Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
15.15Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
15.15Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
15.15Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
15.15Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
15.15Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
15.00Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
15.00Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
15.00Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
15.00Single7WC4Serotonin7WC4-5-HT2A-Serotonin
15.00Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
15.00Single8PWNTheophylline8PWN-A2A-Theophylline
14.81Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
14.81Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
14.81Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
14.81Single7R0CAVP7R0C-V2-AVP-Arrestin2
14.81Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
14.81Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
14.81Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
14.81Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
14.81Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
14.81Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
14.81Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
14.71Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
14.71Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
14.71Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
14.71Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
14.71Consensuscalcitonin_onOrthosteric Ligandctlike_on
14.29Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
14.29Single3RFMCaffeine3RFM-A2A-Caffeine
14.29Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
14.29Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
14.29Single6TQ9SB-4081246TQ9-OX1-SB-408124
14.29Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
14.29Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
14.29Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
14.29Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
14.29Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
14.29Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
14.29Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
14.29Single9CHUNoradrenaline9CHU-β2-Noradrenaline
14.29Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
13.79Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
13.79Single5CGDHTL142425CGD-mGlu5-HTL14242
13.79Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
13.64Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
13.64Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
13.64Single7WC5Psilocin7WC5-5-HT2A-Psilocin
13.64Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
13.64Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
13.64Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
13.64Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
13.64Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
13.64Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
13.64Single9LRCHistamine9LRC-H4-Histamine
13.64Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
13.64Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
13.64Consensusgi_sensoryOrthosteric Ligandgi_opsins
13.64Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
13.64Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
13.64Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
13.64Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
13.51Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
13.33Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
13.33Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
13.04Single5L7IVismodegib5L7I-SMO-Vismodegib
13.04Single6TP4ACT-4622066TP4-OX1-ACT-462206
13.04Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
13.04Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
13.04Single7UL2SR486927UL2-NTS1-SR48692-Na
13.04Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
13.04Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
13.04Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
13.04Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
13.04Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
13.04Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
13.04Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
13.04Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
13.04Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
13.04Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
13.04Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
13.04Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.04Consensusneurotensin_offOrthosteric Ligandnts1_off
13.04Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
12.90Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
12.90Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
12.90Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
12.90Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
12.90Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
12.50Single4S0VSuvorexant4S0V-OX2-Suvorexant
12.50Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
12.50Single5ZKQABT-4915ZKQ-PAF-ABT-491
12.50Single6TPJSuvorexant6TPJ-OX2-Suvorexant
12.50Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
12.50Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
12.50Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
12.50Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
12.50Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
12.50Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
12.50Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
12.50Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
12.50Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
12.50Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
12.50Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
12.50Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
12.50Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
12.50Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
12.50Consensusangiotensin_offOrthosteric Ligandat1_off
12.50Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
12.50Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
12.50Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
12.20Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
12.00Single6TP3Nemorexant6TP3-OX1-Nemorexant
12.00Single6VI4JDTic6VI4-κ-JDTic
12.00Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
12.00Single8K2WAMG4878K2W-CXCR3-AMG487
12.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
12.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
12.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
12.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
11.76Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
11.76Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
11.76Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
11.54Single4QIMANTA XV4QIM-SMO-ANTA XV
11.54Single5DHHSB-6121115DHH-NOP-SB-612111
11.54Single6GPSMK08126GPS-CCR2-MK0812
11.54Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
11.54Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
11.54Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
11.54Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
11.54Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
11.11Single4JKVTaladegib4JKV-SMO-Taladegib
11.11Single5CGCHTL142425CGC-mGlu5-HTL14242
11.11Single6GPXMK08126GPX-CCR2-MK0812
11.11Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
11.11Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
11.11Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
11.11Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
11.11Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
11.11Single9HC04YI9HC0-mGlu5-4YI
11.11Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
10.81Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
10.71Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
10.71Single5V56TC1145V56-SMO-TC114
10.71Single5V57TC1145V57-SMO-TC114
10.71Single7P2L4YI7P2L-mGlu5-4YI
10.71Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
10.71Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
10.53Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
10.34Single5X33BIIL2605X33-BLT1-BIIL260
10.34Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single5MZPCaffeine5MZP-A2A-Caffeine-Na
10.00Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
10.00Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
10.00Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
10.00Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
10.00Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
10.00Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
9.52Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
9.38Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
9.38Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
9.09Single3OE8IT1t3OE8-CXCR4-IT1t
9.09Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
9.09Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
9.09Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
9.09Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
8.70Single3UZAGTPL92363UZA-A2A-GTPL9236
8.70Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
8.70Single8JPSCCL78JPS-ACKR1-CCL7
8.70Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
8.70Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
8.70Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
8.33Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
8.33Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
8.33Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.33Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
8.33Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
8.33Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single9B9Y7DY9B9Y-CB1-7DY
8.33Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
8.33Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
8.33Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
8.00Single4K5YCP-3763954K5Y-CRF1-CP-376395
8.00Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
8.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
8.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
8.00Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
8.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
8.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
8.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
8.00Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
7.69Single7VV6C48/807VV6-MRGPRX2-C48/80
7.69Single8IYXYL-3658IYX-GPR34-YL-365
7.69Single9BA0A1AKN9BA0-CB1-A1AKN
7.69Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
7.41Single4Z9GCP-3763954Z9G-CRF1-CP-376395
7.41Single6IIVDaltroban6IIV-TXA2-Daltroban
7.41Single7YXAONO-54306087YXA-S1P5-ONO-5430608
7.41Single8GTIBMK-C2058GTI-CRF1-BMK-C205
7.41Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
7.41Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
7.41Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
7.14Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
7.14Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
7.14Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
7.14Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
7.14Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
7.14Single8GTGBMK-I1528GTG-CRF1-BMK-I152
7.14Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
7.14Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
7.14Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
7.14Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
7.14Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
7.14Single9B9ZA1AKO9B9Z-CB1-A1AKO
7.14Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
7.14Consensusep_offOrthosteric Ligandep4_off
6.90Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
6.67Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
6.67Single6IIURamatroban6IIU-TXA2-Ramatroban
6.67Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
6.67Single8GTMBMK-C2038GTM-CRF1-BMK-C203
6.67Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
6.67Single9BJKNAM9BJK-μ-Naloxone-NAM
6.45Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
6.25Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
6.25Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
5.26Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
5.26Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
5.00Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.55Single8HS2Fab0468HS2-GPR20-Fab046
4.55Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
4.35Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
4.35Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
4.35Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.17Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.17Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
4.00Single6LI0C176LI0-GPR52-C17
4.00Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.00Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
4.00Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
4.00Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.00Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
4.00Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.00Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
3.85Single5U09Taranabant5U09-CB1-Taranabant
3.85Single6C1QNDT95137276C1Q-C5a1-PMX53-NDT9513727
3.85Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
3.70Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
3.57Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
3.57Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
3.33Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
3.33Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
3.12Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
2.94Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2

Consensus Members
Id Members
fpr2-alx_on_gp 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
fpr1-alx_on_gp 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
Net Summary
Imin 2.96917
Number of Linked Nodes 890
Number of Links 1058
Number of Hubs 163
Number of Links mediated by Hubs 638
Number of Communities 28
Number of Nodes involved in Communities 218
Number of Links involved in Communities 308
Path Summary
Number Of Nodes in MetaPath 98
Number Of Links MetaPath 97
Number of Shortest Paths 1461414
Length Of Smallest Path 3
Average Path Length 29.2031
Length of Longest Path 59
Minimum Path Strength 0.4975
Average Path Strength 5.96003
Maximum Path Strength 21.9358
Minimum Path Correlation 0.7
Average Path Correlation 0.977584
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.88679
Average % Of Corr. Nodes 42.2391
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 52.2799
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
peptide_on_gpcck_on_gp
angiotensin_on_gp
apelin_on_gp
bombesin_on_gp
bradykinin_on_gp
compl-peptide_on_gp
endothelin_on_gp
formylpeptide_on_gp
galanin_on_gp
ghrelin_on_gp
kisspeptin_on_gp
melanocortin_on_gp
motilin_on_gp
neuromedin-u_on_gp
npy_on_gp
neurotensin_on_gp
opioid_on_gp
orexin_on_gp
relaxin_on_gp
somatostatin_on_gp
tachykinin_on_gp
trh_on_gp
vasop-oxy_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download formylpeptide_on_gp.zip



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