Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.33 2.70125404
2G.HN.37 2.04875403
3G.HN.52 2.81469404
4G.S1.02 4.92275585
5G.S1.05 4.79188409
6G.S1.06 3.64754208
7G.H1.01 4.774374209
8G.S2.05 8.34281423
9G.S2.08 6.50125485
10G.S3.02 6.14906424
11G.S3.03 7.46825587
12G.S3.04 8.54875526
13G.S3.06 8.24475525
14G.s3h2.03 5.27812429
15G.H2.02 3.3975428
16G.H2.06 4.70062829
17G.H2.07 4.43078829
18G.h2s4.01 5.425629
19G.S4.04 5.44719409
20G.s4h3.03 5.052194168
21G.H3.09 5.62271679
22G.H3.13 4.77813475
23G.H3.17 5.87042625
24G.H3.18 5.729064199
25G.S5.04 3.56313479
26G.S5.05 3.85758149
27G.HG.03 3.799384106
28G.HG.04 5.868124109
29G.HG.07 3.251755109
30G.HG.14 2.76405
31G.hgh4.02 5.005187217
32G.hgh4.05 6.4405507
33G.H4.03 5.19575504
34G.H4.12 5.9275475
35G.H4.15 4.53531478
36G.h4s6.02 5.14478
37G.S6.02 7.27938407
38G.s6h5.01 5.1995149
39G.s6h5.05 3.30813409
40G.H5.08 4.69344488
41G.H5.20 2.96313609
42G.H5.25 4.94812407
43b.1x15 2.61469407
44b.lhb1x11 4.3475404
45b.b1x3 5.13062437
46b.b1x4 3.92594437
47b.b1x6 8.06656409
48b.l1x3 7.37214799
49b.b2x1 7.6925528
50b.b2x5 5.80125737
51b.l3x2 4.47275599
52b.b4x2 4.35125408
53b.b4x3 4.26719467
54b.b4x5 3.97344467
55b.b4x6 9.98896699
56b.l4x2 11.7663434
57b.b5x2 4.98906407
58b.b5x3 5.99268799
59b.b5x5 5.12938465
60b.b5x7 5.69563407
61b.l5x1 4.39925568
62b.l5x5 7.574529
63b.b6x5 4.04571766
64b.l6x5 5.569064174
65b.b7x1 5.172755174
66b.b7x4 3.04375568
67b.l7x2 3.18425529
68b.b8x3 3.74594406
69b.b8x4 5.20312666
70b.l8x1 3.805465
71b.b9x4 6.07125409
72b.l9x3 5.6775729
73b.l9x6 4.215131028
74b.b10x3 2.82281428
75b.b10x4 5.81594406
76b.b10x5 4.684509
77b.l10x1 4.5775403
78b.b11x4 5.20425529
79b.b11x6 7.43594429
80b.l11x2 8.54313429
81b.b12x2 5.15313427
82b.b12x3 3.77906448
83b.b12x5 3.97656446
84b.b12x6 7.5275728
85b.b13x7 7.394547
86b.l13x3 7.11583649
87b.l13x6 3.9475629
88b.l13x7 4.18875449
89b.b15x1 6.00521649
90b.b15x2 6.93437456
91b.b15x3 4.50563449
92b.l15x2 5.95625449
93b.b16x4 9.9925446
94b.b16x5 4.94594405
95b.b16x6 7.9425648
96b.b17x7 7.15031458
97b.l17x3 8.92688659
98b.l17x6 6.1175529
99b.b18x3 4.65688458
100b.b18x5 5.14125405
101b.l18x1 6.722327136
102b.l18x2 5.176874137
103b.b19x2 6.53312656
104b.b19x4 6.3775458
105b.l19x2 5.3475409
106b.b20x2 5.23975556
107b.b20x4 10.6055558
108b.b20x6 6.92225556
109b.b21x1 8.43594457
110b.b21x5 4.6695504
111b.b21x7 5.8185505
112b.b22x5 4.636256137
113b.l22x5 6.580636119
114b.b23x1 3.45688405
115b.b23x6 7.355426187
116b.l23x1 7.70219406
117b.b24x4 9.360944186
118b.b24x5 3.22562405
119b.b24x6 7.414384188
120b.b24x7 7.403124119
121b.l24x3 3.226115
122b.l25x3 8.2645129
123b.l25x4 3.62406405
124b.b26x3 4.48406406
125b.l27x1 10.088729
126b.l27x2 5.966884129
127b.b28x3 4.47281407
128b.b28x4 8.251254126
129b.b28x5 3.4775535
130b.b28x6 9.734384129
131b.b28x7 5.91188439
132g.h1x1 0.934062402
133g.h1x8 2.8915507
134g.l1x4 4.77575508
135g.h2x11 9.948444136
136g.ctx3 5.765216239
137g.ctx5 4.427814239
138g.ctx6 3.11506
139g.ctx14 5.18344439
140g.ctx15 7.10625439
141g.ctx16 4.86766838
142NT 14.0287815
1431x32 2.56325513
1441x39 5.06719418
1451x47 2.52406406
1461x53 3.693134259
1471x59 2.95875405
1482x38 4.618444266
1492x40 3.86094408
1502x42 4.96925507
1512x46 4.64219409
1522x53 4.87937416
1532x57 3.22156418
1542x60 7.16875415
155E1x50 6.9645519
156E1x52 4.76042607
1573x32 5.52542615
1583x33 4.404514
1593x35 5.13408
1603x37 4.39225516
1613x49 6.319064268
1623x50 6.63625519
1633x51 7.2854278
1643x56 3.655836276
165I2x52 3.48156404
1664x42 3.78063408
1674x56 3.56625505
1684x61 6.56031414
1694x65 6.23625415
170E2 11.98421513
171E2x52 7.07281413
1725x58 6.90479618
173I3 4.245636153
1746x44 3.95419
1756x48 5.87518719
1766x51 5.39771616
1776x52 5.766518
1786x58 4.14075515
1796x62 4.51812412
180E3 5.24104612
1817x27 5.59688411
1827x42 4.75646616
1837x49 5.58675509
1847x50 4.00062409
1857x52 2.57938418
1867x53 5.06146619
1878x50 5.844255258
1888x54 2.22406406
189Lig 50.54441810
190G.s4h3.04 5.798754100
191G.s4h3.11 2.06875400
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1G.HN.47 b.b5x3 19.16322.82NoYes069
2G.HN.47 b.b4x2 19.3714.40625NoYes068
3b.b4x2 b.b5x8 37.39124.185YesNo085
4b.b5x7 b.b5x8 37.57133.39YesNo075
5b.b5x7 b.l8x8 18.97347.87125YesNo074
6b.b5x7 b.b8x4 19.26656.3475YesYes076
7b.b7x2 b.b8x4 21.71113.79NoYes686
8b.b6x5 b.b7x2 21.80373.79YesNo668
9b.b2x4 b.b6x5 42.44613.27NoYes066
10b.b10x4 b.b2x4 42.518214.1038YesNo066
11b.b10x2 b.b10x4 38.92515.04875NoYes066
12b.b10x2 b.b14x3 37.14062.7775NoNo065
13b.b11x5 b.b14x3 40.43243.94NoNo065
14b.b10x1 b.b11x5 47.48633.26NoNo096
15b.b10x1 b.l9x6 47.57583.975NoYes098
16G.H2.07 b.l9x6 61.41382.7725YesYes298
17b.l8x1 b.l8x8 19.15542.79375YesNo054
18b.b6x5 b.l8x1 19.69682.93125YesYes665
19G.H2.04 G.H2.07 62.15014.125NoYes099
20G.H2.04 G.H3.08 62.23624.09625NoNo099
21G.H3.08 G.S4.04 62.28385.175NoYes099
22G.H3.09 G.S4.04 99.841610.3138YesYes099
23G.H3.09 G.S5.04 97.90293.19625YesYes799
24G.S5.04 G.S5.06 98.05683.6325YesNo098
25G.S5.06 G.s4h3.01 49.86134.32375NoNo087
26G.HG.04 G.s4h3.01 50.998612.025YesNo097
27G.H4.03 G.HG.04 50.79072.96625YesYes049
28G.H4.03 G.HG.01 1008.5075YesNo045
29G.HG.01 G.s6h5.02 99.94683.63625NoNo057
30G.s6h5.02 G.s6h5.05 99.843.89NoYes079
31G.s6h5.01 G.s6h5.05 99.67922.8925YesYes099
32G.S5.05 G.s6h5.01 99.00525.835YesYes1499
33G.S4.03 G.S5.05 97.75153.14NoYes079
34G.S1.04 G.S4.03 97.69456.24375NoNo077
35G.S1.02 G.S1.04 48.11453.16625YesNo857
36G.S5.06 G.S6.05 48.26726.6975NoNo084
37G.H4.07 G.S6.05 48.64963.465NoNo054
38G.H4.03 G.H4.07 48.65113.00125YesNo045
39G.S1.02 G.S3.01 47.87373.3525YesNo854
40G.S1.04 G.S3.03 49.5232.895NoYes877
41G.S3.01 G.S3.03 48.16557.46125NoYes847
42G.S1.05 G.S1.07 38.76315.02YesNo099
43G.H3.18 G.S4.02 35.02617.8475YesNo1998
44G.S1.05 G.S4.02 35.21343.3875YesNo098
45G.H5.08 G.S3.01 95.85563.6525YesNo884
46G.H2.06 b.l9x6 18.49462.9825YesYes298
47G.H2.06 b.l17x6 17.97146.57YesYes299
48G.H3.15 G.H3.17 35.04413.53125NoYes085
49G.H3.15 G.H3.18 35.14844.23NoYes089
50G.H5.08 G.H5.12 94.38283.2425YesNo086
513x50 5x58 21.73457.58875YesYes198
523x47 5x58 40.24713.035NoYes198
533x47 5x57 88.82515.1625NoNo097
543x51 5x57 89.19965.8825YesNo087
553x51 3x56 90.09275.85YesYes2786
563x56 I2x52 91.25233.86875YesYes064
57I2x51 I2x52 94.01374.3725NoYes054
58G.H5.12 I2x51 94.19832.355NoNo065
597x49 7x50 11.9573.26YesYes099
607x49 7x53 21.7493.49YesYes099
613x50 7x53 11.89175.01375YesYes199
626x40 7x53 11.67695.86NoYes189
635x58 6x40 12.50593.965YesNo188
64b.l17x5 b.l17x6 18.00294.78375NoYes269
65b.l17x5 b.l19x2 17.87112.575NoYes069
66b.b20x2 b.l19x2 13.85915.7825YesYes069
67g.ctx3 g.ctx6 15.92835.59875YesYes096
68b.l22x5 g.ctx6 29.17773.79375YesYes096
69b.l22x5 b.lhb1x3 14.79415.47875YesNo092
70b.l24x3 b.lhb1x3 14.8765.45375YesNo052
71b.h2x5 b.l24x3 30.37693.0025NoYes055
72b.h2x1 b.h2x5 30.53573.31875NoNo055
73b.b24x7 b.l22x5 14.830714.29YesYes1199
74b.b24x7 b.l24x3 15.11976.2225YesYes1195
75b.b21x5 b.h2x1 30.91627.245YesNo045
76b.lhb1x11 b.lhb1x9 11.46773.10125YesNo043
77b.b23x1 b.lhb1x9 11.65223.0325YesNo053
78b.b25x7 b.lhb1x11 23.78477.24375NoYes074
79b.lhb1x11 g.ctx5 11.69934.24YesYes049
80b.b25x7 b.b28x6 21.70314.5225NoYes079
81b.b28x4 b.b28x6 11.10826.525YesYes1269
82b.b4x6 b.b5x3 14.26810.585YesYes999
83b.b1x6 b.b4x6 21.861818.0788YesYes099
84b.b1x6 b.b28x5 21.05623.92625YesYes095
85b.l25x3 b.l27x2 14.06874.725YesYes1299
86b.b4x6 b.l1x3 14.29144.36625YesYes999
87b.b4x2 b.l3x2 17.67926.9125YesYes089
88b.l1x3 b.l3x2 16.3952.835YesYes999
89b.b21x5 b.b21x7 31.31328.3825YesYes045
90b.b21x7 b.b24x6 34.32518.07875YesYes058
91b.b23x6 b.b24x6 34.24647.7175YesYes1878
92b.b23x6 b.l23x2 35.57684.45625YesNo078
93b.l21x7 b.l23x2 36.065.055NoNo058
94b.l21x7 b.l23x1 36.1535.055NoYes056
95b.l25x4 b.l27x2 12.03034.48875YesYes059
963x47 5x54 48.39075.7725NoNo198
975x54 6x44 48.52974.19875NoYes189
986x44 6x48 47.93325.76625YesYes199
996x48 6x51 36.40183.49375YesYes196
1006x51 Lig 27.05224.485YesYes160
1013x34 3x35 10.14893.295NoYes068
1022x53 3x35 16.49466.72125YesYes068
103b.b28x5 g.ctx16 18.2023.92375YesYes358
104b.b23x1 g.ctx6 12.86692.7675YesYes056
105g.ctx3 g.ctx5 12.79025.4275YesYes2399
106b.l23x1 b.l25x6 36.445418.6138YesNo068
107G.S1.07 G.S4.04 38.86993.3525NoYes099
108G.H3.17 b.l25x6 34.18543.625YesNo258
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
NTNT24.84621YesYes5511
LigNT41.12751YesYes0501
7x24NT7.05250NoYes8521
1x392x574.688751YesYes8822
1x397x425.91751YesYes8621
2x533x326.1651YesYes6521
2x562x603.486251NoYes7521
2x577x423.868751YesYes8621
2x603x282.811YesNo5512
2x603x329.213751YesYes5511
2x60Lig13.1651YesYes5010
2x63E1x506.74751NoYes5922
2x63E24.44751NoYes5321
E1x49E23.91751NoYes3321
E1x50E24.15251YesYes9321
3x22E26.676250NoYes3321
3x323x333.466251YesYes5412
3x327x423.741YesYes5611
3x32Lig7.578751YesYes5010
3x333x374.148751YesYes4622
3x375x435.248751YesNo6521
4x64E28.246251NoYes5321
E2E240.9751YesYes3311
E2E2x518.39251YesNo3311
E2Lig31.74251YesYes3010
E2E2x526.386251YesYes3312
5x39E2x523.881251NoYes5322
5x32E23.823750NoYes4321
5x35E211.82371NoYes4321
5x39E23.703751NoYes5321
5x36Lig6.058751NoYes4010
5x406x557.70NoNo3522
5x406x586.5150NoYes3521
5x43Lig3.016251NoYes5010
6x486x513.493751YesYes9621
6x486x523.528751YesYes9822
6x516x525.631251YesYes6812
6x516x557.5351YesNo6512
6x517x374.9951YesNo6712
6x51Lig4.4851YesYes6010
6x547x343.061250NoNo4521
6x587x302.67751YesNo5412
6x587x342.951251YesNo5511
6x58Lig4.453751YesYes5010
6x62Lig5.573751YesYes2010
7x27E33.343751YesYes1212
7x27Lig13.37621YesYes1010
7x387x427.738751NoYes5611
7x42Lig3.406251YesYes6010
E2NT3.13751YesYes3511
1x317x352.86750NoNo5421
2x537x423.86751YesYes6621
2x563x322.988751NoYes7521
6x517x386.246251YesNo6511
6x586x624.106251YesYes5211
E3E33.833751YesYes2222
7x34Lig4.278751NoYes5010
7x35Lig3.5451NoYes4010
7x38Lig9.27751NoYes5010
E2x51Lig11.5451NoYes3010
7x27NT2.7351YesYes1511
7x28NT6.12251NoYes3521
5x36E2x516.9451NoNo4311
5x376x625.460NoYes1221
6x627x272.93251YesYes2111
6x64Lig2.91250NoYes1010
5x436x522.72251NoYes5812
1x32NT2.36251YesYes3521
5x335x362.336250NoNo2421
5x31E21.36251NoYes0321

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
87.50Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
70.00Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
65.00Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
61.90Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
60.00Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
60.00Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
60.00Consensusbradykinin_onOrthosteric Ligandbk2_on
60.00Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
60.00Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
59.09Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
58.82Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
58.82Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
57.14Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
56.52Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
56.52Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
56.25Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
54.55Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
54.17Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
54.17Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
53.85Consensusendothelin_onOrthosteric Ligandetb_on eta_on
52.63Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
52.00Single7SK3CXCL127SK3-ACKR3-CXCL12
52.00Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
52.00Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
50.00Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
50.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
50.00Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
50.00Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
50.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
50.00Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
50.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
50.00Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
48.15Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
48.15Single8IY6Endothelin-18IY6-ETB-Endothelin-1
48.00Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
48.00Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
48.00Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
48.00Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
47.83Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
47.83Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
47.62Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
47.62Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
47.62Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
47.37Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
47.37Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
47.06Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
46.43Single5GLHEndothelin-15GLH-ETB-Endothelin-1
46.15Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
45.83Single3OE0CVX153OE0-CXCR4-CVX15
45.83Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
45.83Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
45.83Consensusangiotensin_onOrthosteric Ligandat1_on
45.83Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
45.83Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
45.45Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
45.45Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
45.45Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
45.45Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
45.00Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
44.44Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
44.44Single8ZPNAMD31008ZPN-CXCR4-AMD3100
44.00Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
44.00Single6JODAngiotensin II6JOD-AT2-Angiotensin II
44.00Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
44.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
44.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
44.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
44.00Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
44.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
43.75Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
43.48Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
43.48Single8XWNCXCL88XWN-CXCR2-CXCL8
43.48Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
43.33Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
42.86Single6IGLIRL16206IGL-ETB-IRL1620
42.86Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
42.31Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
42.31Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
42.31Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.31Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
42.31Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
42.31Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
42.31Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
42.11Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
42.11Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
41.67Single7SK5CXCL127SK5-ACKR3-CXCL12
41.67Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
41.67Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
41.67Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
41.67Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
41.67Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
41.38Single6IGKEndothelin-36IGK-ETB-Endothelin-3
41.38Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
41.38Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
41.18Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
41.18Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
40.91Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
40.91Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
40.91Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
40.91Single8XVUCXCL28XVU-CXCR2-CXCL2
40.91Single8XWFCXCL38XWF-CXCR2-CXCL3
40.91Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
40.91Single8ZPLHF511168ZPL-CXCR4-HF51116
40.74Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
40.74Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
40.74Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
40.74Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
40.00Single5C1MBU725C1M-μ-BU72
40.00Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
40.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
40.00Single8S4DCMF-0198S4D-Apelin-CMF-019
40.00Single8TF5Oleic acid8TF5-GPR6-Oleic acid
40.00Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
40.00Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
40.00Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
40.00Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
40.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
40.00Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
40.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
40.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
40.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
39.29Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
39.29Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
39.29Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
39.29Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
39.29Single9KDFRES-701-39KDF-ETB-RES-701-3
39.29Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
39.29Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
39.29Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
39.13Single5WF6UK-4320975WF6-A2A-UK-432097
39.13Single6KNMJN241-96KNM-Apelin-JN241-9
39.13Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
39.13Single7XN9L-054,5227XN9-SST2-L-054,522
39.13Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
39.13Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
39.13Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
39.13Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
38.89Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
38.89Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
38.46Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
38.46Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
38.46Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
38.46Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
38.46Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
38.46Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
38.46Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
38.10Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
38.10Single6OS1TRV0266OS1-AT1-TRV026
38.10Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
38.10Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
38.10Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
38.10Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
38.10Single8E0GBU728E0G-μ-BU72
38.10Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
38.10Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
38.10Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
38.10Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
38.10Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
38.10Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
37.93Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
37.50Single4IARErgotamine4IAR-5-HT1B-Ergotamine
37.50Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
37.50Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
37.50Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
37.50Single8WDTphotoNECA8WDT-A2A-photoNECA
37.50Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
37.50Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
37.50Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
37.50Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
37.50Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
37.50Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
37.04Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
37.04Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
37.04Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
37.04Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
37.04Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
37.04Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
37.04Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
37.04Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
37.04Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
36.84Single7F61PF-036547467F61-H3-PF-03654746
36.84Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
36.84Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
36.84Single8ZPMAMD0708ZPM-CXCR4-AMD070
36.84Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
36.84Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
36.84Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
36.67Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
36.67Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
36.67Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
36.67Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
36.36Single4RWADIPP-NH24RWA-δ-DIPP-NH2
36.36Single6A93Risperidone6A93-5-HT2A-Risperidone
36.36Single6MXTSalmeterol6MXT-β2-Salmeterol
36.36Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
36.36Single6OS2TRV0266OS2-AT1-TRV026
36.36Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
36.36Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
36.36Single8XWACXCL18XWA-CXCR2-CXCL1
36.36Single8XWMCXCL68XWM-CXCR2-CXCL6
36.36Single8XWSCXCL58XWS-CXCR2-CXCL5
36.36Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
36.36Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
36.36Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
36.36Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
36.36Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
36.36Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
36.36Consensuslpa_offOrthosteric Ligandlpa1_off
36.36Consensuslpl_offOrthosteric Ligands1p_off lpa_off
36.00Single3QAKUK-4320973QAK-A2A-UK-432097
36.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
36.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
36.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
36.00Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
36.00Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
36.00Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
35.71Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
35.71Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
35.71Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
35.71Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
35.48Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
35.00Single4QIMANTA XV4QIM-SMO-ANTA XV
35.00Single6D27CAY104716D27-DP2-CAY10471
35.00Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
35.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
35.00Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
35.00Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
35.00Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
35.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
35.00Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
35.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
35.00Single8T1WCVN4248T1W-GPR6-CVN424
35.00Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
35.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
35.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
34.78Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
34.78Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
34.78Single7EZCUKA7EZC-A2A-UKA
34.78Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
34.78Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
34.78Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
34.78Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
34.78Consensusprostanoid_offOrthosteric Ligandep_off dp_off
34.62Single5WF5UK-4320975WF5-A2A-UK-432097
34.62Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
34.62Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
34.62Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
34.62Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.62Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
34.62Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
34.48Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
34.48Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
34.38Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
33.33Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
33.33Single5L7IVismodegib5L7I-SMO-Vismodegib
33.33Single5N2RPSB-365N2R-A2A-PSB-36-Na
33.33Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
33.33Single6D26Fevipiprant6D26-DP2-Fevipiprant
33.33Single7C61Ergotamine7C61-5-HT1B-Ergotamine
33.33Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
33.33Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
33.33Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
33.33Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
33.33Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
33.33Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
33.33Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
33.33Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
33.33Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
33.33Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
33.33Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
33.33Single8QJ2pN1628QJ2-MC4-pN162-Gs
33.33Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
33.33Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
33.33Single8XQJJN2418XQJ-Apelin-JN241
33.33Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
33.33Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
33.33Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
33.33Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
33.33Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
33.33Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
33.33Consensusdp_offOrthosteric Liganddp2_off
33.33Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
33.33Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
33.33Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
33.33Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
33.33Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
33.33Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Consensusvasop-oxy_onOrthosteric Ligandv2_on
33.33Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
32.14Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
32.14Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
32.14Single8ZRTET-18ZRT-ETB-ET-1
32.14Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
32.00Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
32.00Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
32.00Single7F8XNN90567F8X-CCKA-NN9056
32.00Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
32.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
32.00Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
32.00Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
32.00Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
32.00Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
32.00Consensuslpl_onOrthosteric Ligands1p_on lpa_on
32.00Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
32.00Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
32.00Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.82Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
31.82Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
31.82Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
31.82Single7R0CAVP7R0C-V2-AVP-Arrestin2
31.82Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
31.82Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
31.82Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
31.82Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
31.82Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
31.82Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
31.82Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
31.82Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
31.82Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.82Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
31.82Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
31.82Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
31.82Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
31.82Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
31.82Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
31.58Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
31.58Single5WS3EMPA5WS3-OX2-EMPA
31.58Single6AKYMaraviroc6AKY-CCR5-Maraviroc
31.58Single7BR3Elagolix7BR3-GnRH1-Elagolix
31.58Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
31.58Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.58Single8GNGIstradefylline8GNG-A2A-Istradefylline
31.58Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
31.58Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
31.58Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
31.58Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
31.58Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
31.58Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
31.58Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
31.58Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
31.58Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
31.25Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
31.25Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
31.03Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
31.03Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
31.03Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
31.03Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
31.03Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
31.03Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
30.77Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
30.77Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
30.77Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
30.77Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
30.77Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
30.77Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
30.77Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
30.77Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
30.77Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
30.77Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
30.77Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
30.77Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
30.77Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
30.43Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
30.43Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
30.43Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
30.43Single7K15MKD0467K15-BLT1-MKD046-Na
30.43Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
30.43Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
30.43Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
30.43Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
30.43Single7YITNalfurafine7YIT-κ-Nalfurafine
30.43Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
30.43Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
30.43Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
30.43Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
30.43Single8JJ8Formoterol8JJ8-β2-Formoterol
30.43Single8JJLOlodaterol8JJL-β2-Olodaterol
30.43Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
30.43Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
30.43Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.43Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
30.43Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.43Single8XQJJN2418XQJ-Apelin-JN241
30.43Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
30.43Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
30.43Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
30.43Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
30.43Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
30.43Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
30.43Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
30.43Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
30.43Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
30.43Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
30.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
30.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
30.00Single6KUXRS-799486KUX-α2a-RS-79948
30.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
30.00Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
30.00Single6TPGEMPA6TPG-OX2-EMPA
30.00Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
30.00Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
30.00Single7AROLUF58337ARO-A2A-LUF5833-Na
30.00Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
30.00Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
30.00Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
30.00Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
30.00Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.00Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
30.00Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
30.00Single8IHKAcifran8IHK-HCA3-Acifran
30.00Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
30.00Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
30.00Single8K5CAcipimox8K5C-HCA2-Acipimox
30.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
30.00Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
30.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
30.00Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
30.00Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
30.00Single9BA0A1AKN9BA0-CB1-A1AKN
30.00Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
30.00Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
30.00Consensusgrh_offOrthosteric Ligandgnrh1_off
30.00Consensushca_onOrthosteric Ligandhca2_on
29.63Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
29.63Single6PT2KGCHM076PT2-δ-KGCHM07
29.63Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
29.63Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
29.63Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
29.63Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
29.63Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
29.63Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
29.63Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
29.63Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
29.63Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
29.63Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
29.41Consensusp2y_offOrthosteric Ligandp2y1_off
29.17Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
29.17Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
29.17Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
29.17Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
29.17Single6IBLArformoterol6IBL-β1-Arformoterol
29.17Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
29.17Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
29.17Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
29.17Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
29.17Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.17Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
29.17Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
29.17Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
29.17Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
29.17Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
29.17Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
29.17Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
29.17Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
29.17Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
29.17Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
29.17Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
29.03Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
28.57Single2Y01Dobutamine2Y01-β1-Dobutamine
28.57Single4EJ4Naltrindole4EJ4-δ-Naltrindole
28.57Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
28.57Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
28.57Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
28.57Single5TGZAM65385TGZ-CB1-AM6538
28.57Single5UENDU1725UEN-A1-DU172
28.57Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
28.57Single6TOTLemborexant6TOT-OX1-Lemborexant
28.57Single7BU7BI1671077BU7-β1-BI167107
28.57Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
28.57Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
28.57Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
28.57Single7UL4Alvimopan7UL4-μ-Alvimopan
28.57Single7V3ZCP559407V3Z-CB1-CP55940
28.57Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
28.57Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
28.57Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
28.57Single7YXAONO-54306087YXA-S1P5-ONO-5430608
28.57Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
28.57Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
28.57Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
28.57Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
28.57Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
28.57Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
28.57Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
28.57Single8JXRLSD8JXR-D1-LSD
28.57Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
28.57Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
28.57Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
28.57Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
28.57Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
28.57Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
28.57Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
28.57Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
28.57Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
28.57Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
28.57Consensusa3_onOrthosteric Liganda3a_on
28.57Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
28.57Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
28.57Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
28.57Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
28.57Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
28.57Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
28.57Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
28.57Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
28.57Consensushca_on_gpOrthosteric Ligandhca2_on_gp
28.57Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
28.57Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
28.00Single3NY9ICI118-5513NY9-β2-ICI118-551
28.00Single4UG2CGS216804UG2-A2A-CGS21680
28.00Single6PT3DPI-2876PT3-δ-DPI-287
28.00Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
28.00Single7SK9CCX6627SK9-ACKR3-CCX662
28.00Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
28.00Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
28.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
28.00Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
28.00Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
28.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
28.00Single8X5YAstemizole8X5Y-H1-Astemizole
28.00Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
28.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
28.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
28.00Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
28.00Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
28.00Single9IPYJR14a9IPY-C3aB-JR14a
28.00Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
28.00Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
28.00Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
27.78Single3OE6IT1t3OE6-CXCR4-IT1t
27.78Single4XNWMRS25004XNW-P2Y1-MRS2500
27.78Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
27.78Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
27.78Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
27.78Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
27.78Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
27.59Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
27.59Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
27.59Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
27.59Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
27.59Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
27.59Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
27.27Single2Y00Dobutamine2Y00-β1-Dobutamine
27.27Single4JKVTaladegib4JKV-SMO-Taladegib
27.27Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
27.27Single5N2SPSB365N2S-A1-PSB36
27.27Single5WQCEMPA5WQC-OX2-EMPA
27.27Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
27.27Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
27.27Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
27.27Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
27.27Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
27.27Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
27.27Single6TP6Filorexant6TP6-OX1-Filorexant
27.27Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
27.27Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
27.27Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
27.27Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
27.27Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
27.27Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
27.27Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
27.27Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
27.27Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.27Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
27.27Single8JXSPF-61428JXS-D1-PF-6142
27.27Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.27Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.27Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
27.27Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
27.27Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
27.27Single9B9ZA1AKO9B9Z-CB1-A1AKO
27.27Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
27.27Single9EHSLUF76029EHS-A3A-LUF7602
27.27Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
27.27Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
27.27Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
27.27Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
27.27Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
27.27Consensusa3_on_gpOrthosteric Liganda3a_on_gp
27.27Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
27.27Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
27.27Consensusadenosine_offOrthosteric Liganda1_off a2_off
27.27Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
27.27Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
27.27Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
27.27Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
27.27Consensusep_offOrthosteric Ligandep4_off
27.27Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
27.27Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
27.27Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
27.27Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
27.27Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
27.27Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Consensustrace-amine_onOrthosteric Ligandta1_on
26.92Single4XT1Fractalkine4XT1-US28-Fractalkine
26.92Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
26.92Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
26.92Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
26.92Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
26.92Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
26.92Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
26.92Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
26.92Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
26.92Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
26.67Single4XT3Fractalkine4XT3-US28-Fractalkine
26.32Single3OE9IT1t3OE9-CXCR4-IT1t
26.32Single4O9RCyclopamine4O9R-SMO-Cyclopamine
26.32Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
26.32Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
26.32Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
26.32Single8K5BNiacin8K5B-HCA2-Niacin
26.32Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
26.32Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
26.32Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
26.32Single9B9Y7DY9B9Y-CB1-7DY
26.32Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
26.32Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
26.32Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
26.32Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
26.09Single2YDVNECA2YDV-A2A-NECA
26.09Single3P0GBI1671073P0G-β2-BI167107
26.09Single4UHRCGS216804UHR-A2A-CGS21680
26.09Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
26.09Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
26.09Single5G53NECA5G53-A2A-NECA-Gs
26.09Single5V56TC1145V56-SMO-TC114
26.09Single5V57TC1145V57-SMO-TC114
26.09Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
26.09Single6J21Aprepitant6J21-NK1-Aprepitant
26.09Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
26.09Single7F1TMIP-1a7F1T-CCR5-MIP-1a
26.09Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
26.09Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
26.09Single7PX4PSB-21137PX4-A2A-PSB-2113
26.09Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
26.09Single7TUYGSK682753A7TUY-GPR183-GSK682753A
26.09Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
26.09Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
26.09Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
26.09Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
26.09Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
26.09Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
26.09Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
26.09Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
26.09Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
26.09Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
26.09Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
26.09Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
26.09Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
26.09Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
26.09Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
26.09Single8ZWFJR14a8ZWF-C3aB-JR14a
26.09Single9BJKNaloxone9BJK-μ-Naloxone-NAM
26.09Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
26.09Consensusa2_onOrthosteric Liganda2b_on
26.09Consensusa2_on_gpOrthosteric Liganda2b_on_gp
26.09Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
26.09Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
26.09Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
26.09Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
26.09Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
26.09Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
26.09Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
26.09Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
26.09Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
26.09Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
26.09Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
26.09Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
26.09Consensuslpa_onOrthosteric Ligandlpa1_on
26.09Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
26.09Consensusrelaxin_onOrthosteric Ligandrxfp4_on
26.09Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
26.09Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.09Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
25.93Single6HLOAprepitant6HLO-NK1-Aprepitant
25.93Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
25.93Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
25.93Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
25.93Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
25.93Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
25.93Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
25.93Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
25.93Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
25.93Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
25.81Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
25.81Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
25.81Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
25.81Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
25.81Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
25.81Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
25.81Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
25.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
25.00Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
25.00Single3ODUIT1t3ODU-CXCR4-IT1t
25.00Single3PWHZM-2413853PWH-A2A-ZM-241385
25.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
25.00Single4AMIBucindolol4AMI-β1-Bucindolol
25.00Single4LDEBI1671074LDE-β2-BI167107
25.00Single4N4WSANT-14N4W-SMO-SANT-1
25.00Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
25.00Single4PY02MeSATP4PY0-P2Y12-2MeSATP
25.00Single4QINSAG1.54QIN-SMO-SAG1.5
25.00Single4S0VSuvorexant4S0V-OX2-Suvorexant
25.00Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
25.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
25.00Single6AKXA4R6AKX-CCR5-A4R
25.00Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
25.00Single6CM4Risperidone6CM4-D2-Risperidone
25.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
25.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
25.00Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
25.00Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
25.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
25.00Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
25.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
25.00Single6TODEMPA6TOD-OX1-EMPA-Na
25.00Single6TPJSuvorexant6TPJ-OX2-Suvorexant
25.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
25.00Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
25.00Single7DFPSpiperone7DFP-D2-Spiperone
25.00Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
25.00Single7F8ULintitript7F8U-CCKA-Lintitript
25.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
25.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
25.00Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
25.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
25.00Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
25.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
25.00Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
25.00Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
25.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
25.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
25.00Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
25.00Single7XRRLemborexant7XRR-OX2-Lemborexant
25.00Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
25.00Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
25.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
25.00Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
25.00Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
25.00Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
25.00Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
25.00Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
25.00Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
25.00Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
25.00Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
25.00Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
25.00Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
25.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
25.00Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
25.00Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
25.00Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
25.00Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
25.00Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
25.00Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Single8XYIVUF106618XYI-CXCR3-VUF10661
25.00Single8Y0HVUF114188Y0H-CXCR3-VUF11418
25.00Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
25.00Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
25.00Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
25.00Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
25.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
25.00Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
25.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
25.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
25.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
25.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
25.00Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
25.00Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
25.00Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
25.00Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
25.00Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
25.00Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
25.00Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
25.00Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
25.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
25.00Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
25.00Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
25.00Consensusorexin_offOrthosteric Ligandox2_off ox1_off
25.00Consensusorexin_onOrthosteric Ligandox2_on
25.00Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
25.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
25.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
25.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
25.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
24.14Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
24.14Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
24.14Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
24.00Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
24.00Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
24.00Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
24.00Single5X93K-87945X93-ETB-K-8794
24.00Single6H7LDobutamine6H7L-β1-Dobutamine
24.00Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
24.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
24.00Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
24.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
24.00Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
24.00Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
24.00Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
24.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
24.00Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
24.00Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
24.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
24.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
24.00Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
24.00Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
24.00Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
24.00Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
24.00Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
24.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
24.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
24.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
24.00Consensuscck_onOrthosteric Ligandccka_on cckb_on
24.00Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
24.00Consensuschemerin_onOrthosteric Ligandcml1_on
24.00Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
24.00Consensusendothelin_offOrthosteric Ligandetb_off
24.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
24.00Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
24.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
24.00Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
23.81Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
23.81Single2YDOAdenosine2YDO-A2A-Adenosine
23.81Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
23.81Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
23.81Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
23.81Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
23.81Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
23.81Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
23.81Single5IUBQ274563445IUB-A2A-Q27456344-Na
23.81Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
23.81Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
23.81Single6AQFZM-2413856AQF-A2A-ZM-241385
23.81Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
23.81Single6MH8ZM-2413856MH8-A2A-ZM-241385
23.81Single6PS0S-Carazolol6PS0-β2-S-Carazolol
23.81Single6PS4ICI118-5516PS4-β2-ICI118-551
23.81Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
23.81Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
23.81Single6TP3Nemorexant6TP3-OX1-Nemorexant
23.81Single6V9SGTPL114036V9S-OX1-GTPL11403
23.81Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
23.81Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
23.81Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
23.81Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
23.81Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
23.81Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
23.81Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
23.81Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.81Single7T32ZM-2413857T32-A2A-ZM-241385
23.81Single7UL3Famotidine7UL3-H2-Famotidine
23.81Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
23.81Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
23.81Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
23.81Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
23.81Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
23.81Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
23.81Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
23.81Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
23.81Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
23.81Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
23.81Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
23.81Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
23.81Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
23.81Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
23.81Single8K2WAMG4878K2W-CXCR3-AMG487
23.81Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
23.81Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
23.81Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
23.81Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
23.81Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
23.81Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
23.81Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
23.81Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
23.81Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
23.81Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
23.81Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
23.81Consensusalpha1_onOrthosteric Ligandalpha1a_on
23.81Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
23.81Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
23.81Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
23.81Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
23.81Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
23.81Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
23.81Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
23.81Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.81Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
23.53Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
23.53Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
23.33Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
23.08Single5ZTYAM102575ZTY-CB2-AM10257
23.08Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
23.08Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
23.08Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
23.08Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
23.08Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
23.08Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
23.08Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
23.08Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
23.08Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
23.08Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
23.08Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
22.73Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
22.73Single2Y02Carmoterol2Y02-β1-Carmoterol
22.73Single2Y04Salbutamol2Y04-β1-Salbutamol
22.73Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
22.73Single3NY8ICI118-5513NY8-β2-ICI118-551
22.73Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
22.73Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
22.73Single4GBRS-Carazolol4GBR-β2-S-Carazolol
22.73Single4QKX35V4QKX-β2-35V
22.73Single5IU8Q274563475IU8-A2A-Q27456347-Na
22.73Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
22.73Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
22.73Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
22.73Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
22.73Single6GPSMK08126GPS-CCR2-MK0812
22.73Single6H7MSalbutamol6H7M-β1-Salbutamol
22.73Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
22.73Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
22.73Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
22.73Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
22.73Single6PS1Timolol6PS1-β2-Timolol
22.73Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
22.73Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
22.73Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
22.73Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
22.73Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
22.73Single7PYRPSB-21157PYR-A2A-PSB-2115
22.73Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
22.73Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
22.73Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
22.73Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
22.73Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
22.73Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
22.73Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
22.73Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.73Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
22.73Single8CU6LJ-45178CU6-A2A-LJ-4517
22.73Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
22.73Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
22.73Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
22.73Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
22.73Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
22.73Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
22.73Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
22.73Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
22.73Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
22.73Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
22.73Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
22.73Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
22.73Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
22.73Single8K5DGSK2560738K5D-HCA2-GSK256073
22.73Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
22.73Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
22.73Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
22.73Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
22.73Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
22.73Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
22.73Single9CHXS-Carazolol9CHX-β2-S-Carazolol
22.73Single9H37A1IR09H37-A2A-A1IR0-Na
22.73Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
22.73Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
22.73Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
22.73Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
22.73Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
22.73Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
22.73Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
22.73Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.73Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.73Consensusblt_onOrthosteric Ligandblt1_on
22.73Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
22.73Consensuscck_offOrthosteric Ligandccka_off
22.73Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
22.73Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
22.73Consensusdopamine_offOrthosteric Ligandd2_off d3_off
22.73Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
22.73Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
22.73Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.73Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.73Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
22.73Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.73Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.73Consensusleukotriene_onOrthosteric Ligandblt_on
22.73Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
22.58Single6FJ3PTH6FJ3-PTH1-PTH
22.58Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
22.58Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
22.58Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
22.22Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
22.22Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
22.22Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
22.22Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
22.22Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
22.22Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
22.22Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
22.22Single8A2OTheophylline8A2O-A2A-Theophylline-Na
22.22Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
22.22Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
22.22Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
22.22Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
22.22Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
22.22Single8WKYPG-9348WKY-MC4-PG-934
22.22Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.22Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
22.22Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
22.22Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
22.22Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
22.22Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
22.22Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
22.22Consensussensory_onOrthosteric Ligandopsins_on
21.88Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
21.88Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
21.74Single2RH1S-Carazolol2RH1-β2-S-Carazolol
21.74Single2Y03Isoprenaline2Y03-β1-Isoprenaline
21.74Single2YCWS-Carazolol2YCW-β1-S-Carazolol
21.74Single5D6LS-Carazolol5D6L-β2-S-Carazolol
21.74Single5IUAQ274563485IUA-A2A-Q27456348-Na
21.74Single5JQHS-Carazolol5JQH-β2-S-Carazolol
21.74Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
21.74Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
21.74Single5WIUNemonapride5WIU-D4-Nemonapride
21.74Single5WIVNemonapride5WIV-D4-Nemonapride-Na
21.74Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
21.74Single6E67BI1671076E67-β2-BI167107-Gs(CT)
21.74Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
21.74Single6GPXMK08126GPX-CCR2-MK0812
21.74Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
21.74Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
21.74Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
21.74Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
21.74Single6S0QZM-2413856S0Q-A2A-ZM-241385
21.74Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
21.74Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
21.74Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
21.74Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
21.74Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
21.74Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
21.74Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
21.74Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
21.74Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
21.74Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
21.74Single7W41PD1762527W41-BB2-PD176252
21.74Single7WC6LSD7WC6-5-HT2A-LSD
21.74Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
21.74Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
21.74Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
21.74Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
21.74Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8GNEKW-63568GNE-A2A-KW-6356-Na
21.74Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
21.74Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
21.74Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
21.74Single8QOTNanobody-E8QOT-μ-Nanobody-E
21.74Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
21.74Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
21.74Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
21.74Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
21.74Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
21.74Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
21.74Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
21.74Single9HAPTolvaptan9HAP-V2-Tolvaptan
21.74Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
21.74Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
21.74Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
21.74Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
21.74Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
21.74Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
21.74Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
21.74Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
21.74Consensusamine_offonOrthosteric Ligandamine_off amine_on
21.74Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
21.74Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
21.74Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
21.74Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
21.74Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
21.74Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
21.74Consensusblt_offOrthosteric Ligandblt1_off
21.74Consensusbombesin_offOrthosteric Ligandbb2_off
21.74Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
21.74Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
21.74Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
21.74Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
21.74Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.74Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.74Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
21.43Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
21.43Single7XNACYN1548067XNA-SST2-CYN154806
21.43Single8IEBA1LYA8IEB-GPR156-A1LYA
21.43Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
21.43Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
21.43Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
21.43Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
21.43Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
21.21Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
21.21Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
21.21Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
21.21Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
21.05Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
21.05Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
21.05Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
21.05Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
21.05Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
21.05Single6ME5Agomelatine6ME5-MT1-Agomelatine
21.05Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
21.05Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
21.05Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
21.05Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
21.05Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
21.05Single7WC5Psilocin7WC5-5-HT2A-Psilocin
21.05Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
21.05Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
21.05Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
21.05Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
21.05Single8JPSCCL78JPS-ACKR1-CCL7
21.05Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
21.05Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
21.05Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
21.05Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
21.05Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
21.05Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
21.05Single9LRCHistamine9LRC-H4-Histamine
21.05Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
21.05Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
21.05Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
21.05Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
21.05Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
21.05Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
20.83Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
20.83Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
20.83Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
20.83Single4BV0Neurotensin4BV0-NTS1-Neurotensin
20.83Single4DJHJDTic4DJH-κ-JDTic
20.83Single4U15Tiotropium4U15-M3-Tiotropium
20.83Single5D5AS-Carazolol5D5A-β2-S-Carazolol
20.83Single5D5BS-Carazolol5D5B-β2-S-Carazolol
20.83Single5XR8AM8415XR8-CB1-AM841
20.83Single5XRAAM115425XRA-CB1-AM11542
20.83Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
20.83Single6H7JIsoprenaline6H7J-β1-Isoprenaline
20.83Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
20.83Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
20.83Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
20.83Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
20.83Single6OL9Tiotropium6OL9-M5-Tiotropium
20.83Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
20.83Single6TQ7SB-3348676TQ7-OX1-SB-334867
20.83Single6WGTLSD6WGT-5-HT2A-LSD
20.83Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
20.83Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
20.83Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
20.83Single7FEECP559407FEE-CB1-CP55940-ZCZ011
20.83Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
20.83Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
20.83Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
20.83Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
20.83Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
20.83Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
20.83Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
20.83Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
20.83Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
20.83Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
20.83Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
20.83Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
20.83Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
20.83Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
20.83Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
20.83Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
20.83Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
20.83Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
20.83Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.83Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
20.83Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
20.83Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
20.83Single8XVLZibotentan8XVL-ETA-Zibotentan
20.83Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
20.83Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
20.83Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
20.83Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
20.83Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
20.83Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
20.83Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
20.83Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
20.83Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
20.83Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
20.83Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
20.83Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
20.83Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
20.83Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
20.83Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
20.83Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
20.83Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
20.83Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.83Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
20.83Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
20.83Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
20.83Consensusneurotensin_onOrthosteric Ligandnts1_on
20.83Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
20.83Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.83Consensustachykinin_offOrthosteric Ligandnk1_off
20.69Single6W25SHU91196W25-MC4-SHU9119-Ca
20.69Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
20.69Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
20.69Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
20.59Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
20.59Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
20.00Single3D4STimolol3D4S-β2-Timolol
20.00Single3PBLEticlopride3PBL-D3-Eticlopride
20.00Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
20.00Single4XEENeurotensin4XEE-NTS1-Neurotensin
20.00Single4XESNeurotensin4XES-NTS1-Neurotensin
20.00Single5CXVTiotropium5CXV-M1-Tiotropium
20.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
20.00Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
20.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
20.00Single5X33BIIL2605X33-BLT1-BIIL260
20.00Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
20.00Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
20.00Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
20.00Single6KQICP559406KQI-CB1-CP55940-Org27569
20.00Single6LI0C176LI0-GPR52-C17
20.00Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
20.00Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
20.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
20.00Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
20.00Single6YVRNTS8-136YVR-NTS1-NTS8-13
20.00Single6ZG4HTL00099366ZG4-M1-HTL0009936
20.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
20.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
20.00Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
20.00Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
20.00Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.00Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.00Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
20.00Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
20.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
20.00Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
20.00Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
20.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
20.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
20.00Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
20.00Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
20.00Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
20.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
20.00Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
20.00Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
20.00Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
20.00Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
20.00Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
20.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
20.00Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
20.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
20.00Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
20.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
20.00Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
20.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
20.00Single9BJKNAM9BJK-μ-Naloxone-NAM
20.00Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single9DGIZ85267113509DGI-CB1-Z8526711350
20.00Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
20.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
20.00Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
20.00Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
20.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
20.00Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
20.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.00Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.00Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
20.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
20.00Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
20.00Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
20.00Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
20.00Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
20.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
20.00Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
20.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
20.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
20.00Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
20.00Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.44Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
19.44Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
19.44Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
19.35Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
19.35Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
19.35Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
19.35Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
19.35Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
19.35Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
19.35Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
19.35Consensuspac_onOrthosteric Ligandpac1_on
19.23Single4BUONeurotensin4BUO-NTS1-Neurotensin
19.23Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
19.23Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
19.23Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
19.23Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
19.23Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
19.23Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
19.23Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
19.23Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
19.23Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
19.23Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
19.23Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
19.23Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
19.23Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
19.23Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
19.23Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
19.23Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
19.23Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
19.23Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
19.05Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
19.05Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
19.05Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
19.05Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
19.05Single4BWBNeurotensin4BWB-NTS1-Neurotensin
19.05Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
19.05Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
19.05Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
19.05Single5U09Taranabant5U09-CB1-Taranabant
19.05Single6B73MP11046B73-κ-MP1104
19.05Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
19.05Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
19.05Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
19.05Single6ME9Ramelteon6ME9-MT2-Ramelteon
19.05Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
19.05Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
19.05Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
19.05Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
19.05Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
19.05Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
19.05Single7F8YDevazepide7F8Y-CCKA-Devazepide
19.05Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
19.05Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
19.05Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.05Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.05Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
19.05Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
19.05Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
19.05Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
19.05Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
19.05Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
19.05Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
19.05Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
19.05Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
19.05Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
19.05Single8IWESpermidine8IWE-TA9-Spermidine
19.05Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
19.05Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
19.05Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
19.05Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
19.05Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
19.05Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
19.05Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
19.05Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.05Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
19.05Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
19.05Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
19.05Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
19.05Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
19.05Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
19.05Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
19.05Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
19.05Consensusalpha2_offOrthosteric Ligandalpha2c_off
19.05Consensusangiotensin_offOrthosteric Ligandat1_off
19.05Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.05Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
19.05Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
19.05Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
19.05Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
19.05Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.05Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.05Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
19.05Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
19.05Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
19.05Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.05Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
18.75Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
18.75Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
18.75Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
18.75Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
18.75Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
18.75Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
18.52Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
18.52Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
18.52Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
18.52Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
18.52Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
18.52Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
18.52Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
18.52Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
18.52Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
18.42Consensuspth_onOrthosteric Ligandpth1_on pth2_on
18.18Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
18.18Single3REYXAC3REY-A2A-XAC
18.18Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
18.18Single5IU7Q274563465IU7-A2A-Q27456346-Na
18.18Single5JTBZM-2413855JTB-A2A-ZM-241385
18.18Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
18.18Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
18.18Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
18.18Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
18.18Single6IQLL7458706IQL-D4-L745870
18.18Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
18.18Single6PS5S-Propranolol6PS5-β2-S-Propranolol
18.18Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
18.18Single6VI4JDTic6VI4-κ-JDTic
18.18Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
18.18Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
18.18Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
18.18Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
18.18Single6ZG9GSK10347026ZG9-M1-GSK1034702
18.18Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
18.18Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
18.18Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
18.18Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
18.18Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
18.18Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
18.18Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
18.18Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
18.18Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
18.18Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
18.18Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
18.18Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
18.18Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
18.18Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
18.18Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
18.18Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
18.18Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
18.18Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
18.18Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
18.18Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
18.18Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
18.18Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
18.18Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
18.18Single8RLNLUF58348RLN-A2A-LUF5834
18.18Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
18.18Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
18.18Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
18.18Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
18.18Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
18.18Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
18.18Single9AS5Mescaline9AS5-5-HT2A-Mescaline
18.18Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
18.18Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
18.18Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
18.18Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
18.18Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
18.18Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
18.18Consensusa2_offOrthosteric Liganda2a_off
18.18Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
18.18Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
18.18Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
18.18Consensusglp_onOrthosteric Ligandglp1_on glp2_on
18.18Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
18.18Consensusopsins_offOrthosteric Ligandrhodopsin_off
18.18Consensussensory_offOrthosteric Ligandopsins_off
17.86Single7QA8Peptide7QA8-STE2-Peptide
17.86Single7QA8Peptide7QA8-STE2-Peptide
17.86Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
17.86Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
17.86Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
17.86Single8IEBA1LYA8IEB-GPR156-A1LYA
17.86Single8IEIA1LYA8IEI-GPR156-A1LYA
17.86Single8IEIA1LYA8IEI-GPR156-A1LYA
17.86Single8IEPA1LYA8IEP-GPR156-A1LYA
17.86Single8IEPA1LYA8IEP-GPR156-A1LYA
17.86Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.86Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
17.86Single8KIGSHU91198KIG-MC3-SHU9119-Ca
17.86Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
17.86Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensussomatostatin_offOrthosteric Ligandsst2_off
17.65Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
17.65Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
17.65Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
17.65Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
17.65Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
17.65Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
17.65Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
17.65Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
17.65Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
17.65Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
17.65Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
17.65Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
17.65Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
17.50Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
17.50Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
17.39Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
17.39Single3EMLZM-2413853EML-A2A-ZM-241385
17.39Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
17.39Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
17.39Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
17.39Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
17.39Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
17.39Single4YAYZD-71554YAY-AT1-ZD-7155
17.39Single5DHHSB-6121115DHH-NOP-SB-612111
17.39Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
17.39Single5T04Neurotensin5T04-NTS1-Neurotensin
17.39Single5UIGCmpd-15UIG-A2A-Cmpd-1
17.39Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
17.39Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
17.39Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
17.39Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
17.39Single6DRXLisuride6DRX-5-HT2B-Lisuride
17.39Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
17.39Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
17.39Single6IIVDaltroban6IIV-TXA2-Daltroban
17.39Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
17.39Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
17.39Single6S0LZM-2413856S0L-A2A-ZM-241385
17.39Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
17.39Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
17.39Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
17.39Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
17.39Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
17.39Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
17.39Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
17.39Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
17.39Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
17.39Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
17.39Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
17.39Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
17.39Single7WC7Lisuride7WC7-5-HT2A-Lisuride
17.39Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
17.39Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
17.39Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
17.39Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
17.39Single8JJOAlprenolol8JJO-β2-Alprenolol
17.39Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
17.39Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
17.39Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
17.39Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
17.39Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
17.39Single8X64Desloratadine8X64-H1-Desloratadine
17.39Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
17.39Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
17.39Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
17.39Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
17.39Single9JEAAtropine9JEA-M1-Atropine
17.39Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
17.39Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
17.39Consensus5ht5_onOrthosteric Ligand5ht5a_on
17.39Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
17.39Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
17.39Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
17.39Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
17.39Consensusalpha2_onOrthosteric Ligandalpha2b_on
17.39Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
17.39Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
17.39Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
17.39Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
17.39Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
17.39Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
17.39Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
17.39Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
17.39Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
17.24Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
17.24Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.24Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
17.24Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.24Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
17.14Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
17.14Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.14Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.14Consensusbombesin_onOrthosteric Ligandbb2_on
17.14Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
17.14Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
17.14Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
17.14Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
16.67Single4NTJAZD12834NTJ-P2Y12-AZD1283
16.67Single5CGCHTL142425CGC-mGlu5-HTL14242
16.67Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
16.67Single5TVNLSD5TVN-5-HT2B-LSD
16.67Single5XPRBosentan5XPR-ETB-Bosentan
16.67Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
16.67Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
16.67Single6HLPNetupitant6HLP-NK1-Netupitant
16.67Single6LUQHaloperidol6LUQ-D2-Haloperidol
16.67Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
16.67Single6PS6Timolol6PS6-β2-Timolol
16.67Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
16.67Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
16.67Single7C4SS1P7C4S-S1P3-S1P
16.67Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
16.67Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
16.67Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
16.67Single7SINNPS-21437SIN-CaS-NPS-2143
16.67Single7SINNPS-21437SIN-CaS-NPS-2143
16.67Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
16.67Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
16.67Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
16.67Single7WC4Serotonin7WC4-5-HT2A-Serotonin
16.67Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
16.67Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
16.67Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
16.67Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
16.67Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
16.67Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
16.67Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
16.67Single8PWNTheophylline8PWN-A2A-Theophylline
16.67Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
16.67Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
16.67Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
16.67Single8ZMFA1L108ZMF-5-HT2C-A1L10
16.67Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
16.67Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
16.67Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
16.67Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
16.67Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
16.67Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
16.67Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
16.67Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
16.67Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
16.67Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
16.67Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
16.67Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
16.67Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
16.67Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
16.67Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
16.67Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
16.67Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
16.67Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.67Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
16.67Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.67Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
16.67Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.67Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.67Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
16.22Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
16.22Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.13Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
16.13Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
16.13Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
16.13Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
16.13Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
16.13Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
16.13Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
16.13Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
16.13Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
16.13Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
16.00Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
16.00Single5TZRMK86665TZR-FFA1-MK8666
16.00Single5V54Methiothepin5V54-5-HT1B-Methiothepin
16.00Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
16.00Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.00Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
16.00Single7B6WCyclazosin7B6W-α1b-Cyclazosin
16.00Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
16.00Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
16.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
16.00Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
16.00Single8EA0Iperoxo8EA0-M3-Iperoxo
16.00Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
16.00Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
16.00Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
16.00Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
16.00Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
16.00Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.00Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Consensus5ht1_offOrthosteric Ligand5ht1b_off
16.00Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
16.00Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
16.00Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.00Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
16.00Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
15.79Single3OE8IT1t3OE8-CXCR4-IT1t
15.79Single3RFMCaffeine3RFM-A2A-Caffeine
15.79Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
15.79Single6TQ9SB-4081246TQ9-OX1-SB-408124
15.79Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
15.79Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
15.79Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
15.79Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
15.79Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
15.79Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
15.79Single9CHUNoradrenaline9CHU-β2-Noradrenaline
15.79Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.79Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
15.79Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
15.79Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
15.79Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
15.62Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
15.62Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
15.62Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
15.62Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
15.62Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
15.62Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
15.38Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
15.38Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
15.38Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
15.38Single6IIURamatroban6IIU-TXA2-Ramatroban
15.38Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
15.38Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
15.38Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8JWY2-1188JWY-A2A-2-118
15.38Single8JWZAB9288JWZ-A2A-AB928-Na
15.38Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
15.38Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
15.38Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
15.38Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
15.38Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
15.38Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
15.38Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
15.38Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
15.15Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
15.15Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
15.15Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
15.15Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
15.15Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
15.15Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
15.15Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
15.15Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
15.00Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
15.00Single3UZAGTPL92363UZA-A2A-GTPL9236
15.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
15.00Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
15.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
15.00Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
15.00Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
15.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
15.00Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
15.00Consensus5ht2_onOrthosteric Ligand5ht2b_on
15.00Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
15.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
15.00Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.00Consensusgi_sensoryOrthosteric Ligandgi_opsins
15.00Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
15.00Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
15.00Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.00Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
14.81Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
14.81Single5CGDHTL142425CGD-mGlu5-HTL14242
14.81Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
14.81Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.81Single7UM4AS26747237UM4-5-HT5A-AS2674723
14.81Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
14.81Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
14.81Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single8XVJMacitentan8XVJ-ETA-Macitentan
14.81Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
14.81Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
14.81Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
14.81Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
14.71Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
14.71Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
14.71Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
14.71Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
14.71Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
14.71Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
14.71Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
14.63Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
14.29Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
14.29Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
14.29Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
14.29Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
14.29Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
14.29Single6HLLCP999946HLL-NK1-CP99994
14.29Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
14.29Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
14.29Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
14.29Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
14.29Single6TP4ACT-4622066TP4-OX1-ACT-462206
14.29Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
14.29Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
14.29Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
14.29Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
14.29Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
14.29Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
14.29Single7SRQLSD7SRQ-5-HT2B-LSD
14.29Single7UL2SR486927UL2-NTS1-SR48692-Na
14.29Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
14.29Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
14.29Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
14.29Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
14.29Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
14.29Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
14.29Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
14.29Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
14.29Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
14.29Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
14.29Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
14.29Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
14.29Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
14.29Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
14.29Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
14.29Consensusgq_nucleotideOrthosteric Ligandgq_p2y
14.29Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.29Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
14.29Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
14.29Consensusneurotensin_offOrthosteric Ligandnts1_off
14.29Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
13.95Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
13.89Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
13.89Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
13.89Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
13.79Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
13.79Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
13.79Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
13.79Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
13.79Single9M4TSilodosin9M4T-Alpha1A-Silodosin
13.64Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
13.64Single6ME2Ramelteon6ME2-MT1-Ramelteon
13.64Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
13.64Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
13.64Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
13.64Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
13.64Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
13.64Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
13.64Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
13.64Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
13.64Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
13.64Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
13.64Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
13.64Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
13.64Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
13.64Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
13.64Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
13.64Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
13.64Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
13.64Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
13.64Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
13.64Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
13.64Single9H2XA1IR19H2X-A2A-A1IR1-Na
13.64Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
13.64Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
13.64Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
13.64Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
13.64Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
13.64Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
13.51Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
13.51Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
13.51Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
13.33Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
13.33Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
13.33Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
13.33Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
13.16Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
13.16Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
13.16Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
13.16Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
13.04Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
13.04Single5UVIZM-2413855UVI-A2A-ZM-241385
13.04Single6A94Zotepine6A94-5-HT2A-Zotepine
13.04Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
13.04Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
13.04Single6TPNHTL66416TPN-OX2-HTL6641
13.04Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
13.04Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
13.04Single6ZINSR486926ZIN-NTS1-SR48692
13.04Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
13.04Single7VODCariprazine7VOD-5-HT2A-Cariprazine
13.04Single7VV6C48/807VV6-MRGPRX2-C48/80
13.04Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
13.04Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
13.04Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
13.04Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
13.04Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
13.04Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
13.04Single9ARXSerotonin9ARX-5-HT2A-Serotonin
13.04Single9AS3LSD9AS3-5-HT2A-LSD
13.04Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
13.04Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
13.04Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
13.04Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
12.90Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
12.90Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
12.90Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
12.82Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
12.50Single4DAJTiotropium4DAJ-M3-Tiotropium
12.50Single4MQSIperoxo4MQS-M2-Iperoxo
12.50Single4U14Tiotropium4U14-M3-Tiotropium
12.50Single5DHGC-355DHG-NOP-C-35
12.50Single5DSGTiotropium5DSG-M4-Tiotropium
12.50Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
12.50Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
12.50Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
12.50Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
12.50Single7F83PF-051904577F83-Ghrelin-PF-05190457
12.50Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
12.50Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
12.50Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
12.50Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
12.50Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
12.50Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
12.50Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
12.50Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
12.50Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
12.50Single8X63Mepyramine8X63-H1-Mepyramine
12.50Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
12.50Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
12.50Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
12.50Single9AS1DMT9AS1-5-HT2A-DMT
12.50Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
12.50Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
12.50Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
12.50Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
12.50Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
12.50Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
12.50Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
12.50Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
12.50Consensushistamine_offOrthosteric Ligandh1_off
12.50Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
12.12Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
12.12Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
12.12Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
12.12Consensuscalcitonin_onOrthosteric Ligandctlike_on
12.00Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
12.00Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
12.00Single6Z4SSR486926Z4S-NTS1-SR48692
12.00Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
12.00Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
12.00Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
12.00Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
12.00Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
12.00Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
12.00Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
12.00Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
11.76Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
11.76Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
11.76Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
11.76Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
11.76Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
11.76Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
11.76Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
11.76Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
11.76Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
11.76Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
11.54Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
11.54Single6E59L-7607356E59-NK1-L-760735
11.54Single6J20Aprepitant6J20-NK1-Aprepitant
11.54Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
11.54Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
11.54Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
11.54Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
11.54Single9AS9RS130-1809AS9-5-HT2A-RS130-180
11.54Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
11.43Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
11.43Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
11.43Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
11.43Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
11.43Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
11.43Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
11.43Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
11.11Single5MZPCaffeine5MZP-A2A-Caffeine-Na
11.11Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
11.11Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
11.11Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
11.11Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
11.11Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
11.11Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
11.11Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
11.11Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
11.11Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
11.11Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
11.11Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
10.81Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
10.71Single6K1QIRL25006K1Q-ETB-IRL2500
10.71Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
10.71Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
10.71Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
10.71Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.53Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
10.53Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
10.34Single9JF4PD1683689JF4-BB1-PD168368
10.34Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.34Consensuskisspeptin_onOrthosteric Ligandkiss1_on
10.26Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
10.00Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
10.00Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
10.00Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
10.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
10.00Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
10.00Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
10.00Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
10.00Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
10.00Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.00Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
10.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
10.00Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.00Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.00Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
9.68Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
9.52Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
9.52Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
9.52Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
9.52Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
9.52Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
9.52Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
9.09Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
9.09Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
9.09Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
9.09Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
9.09Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
9.09Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
9.09Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
9.09Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
9.09Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
9.09Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
9.09Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
9.09Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
9.09Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.09Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
9.09Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9AS7Psilocin9AS7-5-HT2A-Psilocin
9.09Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
9.09Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
9.09Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
8.82Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
8.70Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
8.70Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
8.70Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
8.70Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
8.70Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
8.70Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
8.70Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
8.70Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
8.70Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
8.70Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
8.70Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
8.57Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
8.33Single3RZECidoxepin3RZE-H1-Cidoxepin
8.33Single6FFIMMPEP6FFI-mGlu5-MMPEP
8.33Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
8.33Single6TPKRetosiban6TPK-OT-Retosiban
8.33Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.33Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
8.33Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
8.33Consensusvasop-oxy_offOrthosteric Ligandot_off
8.00Single6FFHFenobam6FFH-mGlu5-Fenobam
8.00Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
8.00Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
8.00Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
8.00Single9IYAONO-97105319IYA-GPR55-ONO-9710531
7.69Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
7.69Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
7.69Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
7.69Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
7.69Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
7.69Single9HC04YI9HC0-mGlu5-4YI
7.41Single7P2L4YI7P2L-mGlu5-4YI
7.41Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
7.41Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
6.25Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
6.25Single6D35Cholesterol6D35-SMO-Cholesterol
6.25Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
6.25Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
6.25Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
6.25Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
6.25Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
6.25Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
6.25Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
6.25Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
6.25Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
6.25Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
6.25Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
6.25Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
6.25Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
6.25Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
6.25Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
6.25Single7DTTCa7DTT-CaS-Ca-Ca
6.25Single7DTTCa7DTT-CaS-Ca-Ca
6.25Single7DTUTryptophan7DTU-CaS-Tryptophan
6.25Single7DTUTryptophan7DTU-CaS-Tryptophan
6.25Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
6.25Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
6.25Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
6.25Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
6.25Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.25Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.25Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.25Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.25Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
6.25Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
6.25Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
6.25Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
6.25Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
6.25Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
6.25Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
6.25Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
6.25Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
6.25Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
6.25Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
6.25Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
6.25Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
6.25Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
6.25Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
6.25Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
6.25Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
6.25Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.25Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.25Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.25Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.25Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
6.25Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
6.25Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
6.25Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
6.25Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
6.25Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
6.25Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.25Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.25Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.25Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.25Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.25Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.25Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.25Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.25Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
6.25Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
6.25Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
6.25Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
6.25Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
6.25Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
6.25Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
6.25Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
6.25Single7XW7K1-707XW7-TSH-K1-70
6.25Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
6.25Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
6.25Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
6.25Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
6.25Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
6.25Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
6.25Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
6.25Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
6.25Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
6.25Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
6.25Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
6.25Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
6.25Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
6.25Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
6.25Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
6.25Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
6.25Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
6.25Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
6.25Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
6.25Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
6.25Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
6.25Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
6.25Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
6.25Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
6.25Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
6.25Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
6.25Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
6.25Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
6.25Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
6.25Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
6.25Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
6.25Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
6.25Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.25Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.25Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
6.25Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
6.25Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
6.25Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
6.25Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
6.25Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
6.25Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
6.25Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
6.25Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
6.25Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
6.25Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
6.25Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
6.25Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
6.25Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
6.25Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
6.25Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
6.25Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
6.25Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
6.25Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single8WVXNorrin8WVX-LGR4-Norrin
6.25Single8WVYNorrin8WVY-LGR4-Norrin
6.25Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
6.25Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
6.25Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
6.25Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
6.25Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
6.25Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
6.25Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
6.25Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.25Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.25Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.25Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.25Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.25Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.25Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
6.25Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
6.25Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.25Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.25Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.25Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.25Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
6.25Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
6.25Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
6.25Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
6.25Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
6.25Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
6.25Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
6.25Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
6.25Single9KHHNorrin9KHH-LGR4-Norrin
6.25Single9S37NB219S37-LGR4-NB21
6.25Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
5.88Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.88Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.88Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.88Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.88Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.88Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.88Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.88Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.88Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.88Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.88Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.88Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.88Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.88Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.88Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
5.88Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
5.56Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
5.56Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
5.56Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
5.56Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
5.26Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
5.26Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
5.26Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
5.26Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
5.26Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
5.00Single5L7DCholesterol5L7D-SMO-Cholesterol
5.00Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
5.00Single8HS2Fab0468HS2-GPR20-Fab046
5.00Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
5.00Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.55Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
4.17Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.00Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.70Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
3.70Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.70Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.70Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
3.57Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.57Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
3.12Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
3.12Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.94Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.94Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.86Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.63Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
cxcr3_on_gp 8HNK-CXCR3-CXCL11-Gi1/β1/γ2
8HNL-CXCR3-PS372424-Gi1/β1/γ2
cxcr4_on_gp 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
cxcr1_on_gp 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
cxcr2_on_gp 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
Net Summary
Imin 2.6475
Number of Linked Nodes 901
Number of Links 1123
Number of Hubs 191
Number of Links mediated by Hubs 735
Number of Communities 27
Number of Nodes involved in Communities 253
Number of Links involved in Communities 379
Path Summary
Number Of Nodes in MetaPath 109
Number Of Links MetaPath 108
Number of Shortest Paths 2855600
Length Of Smallest Path 3
Average Path Length 41.0457
Length of Longest Path 71
Minimum Path Strength 0.520833
Average Path Strength 5.23392
Maximum Path Strength 24.09
Minimum Path Correlation 0.7
Average Path Correlation 0.989945
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.51515
Average % Of Corr. Nodes 36.3317
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 54.2182
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following differences:
Id1st Network2nd Network
cxcr_off_on_gpcxcr_on_gpcxcr_off
This network is also present in following consensuses:
IdComponents
chemokine_on_gpccr_on_gp
cxcr_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download cxcr_on_gp.zip



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