Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg Int. Strength Num Of Links Community ConSurf
1A:A:L42 7.2125476
2A:A:L43 5.1825409
3A:A:K52 5.62609
4A:A:S53 5.7475499
5A:A:I56 7.005476
6A:A:I62 6.354238
7A:A:Y67 10.238507
8A:A:T76 6.194115
9A:A:Q81 6.6325405
10A:A:F84 8.93404
11A:A:M87 5.7575406
12A:A:I91 4.0825405
13A:A:M94 8.8975407
14A:A:N106 10.245405
15A:A:Y128 6.27254254
16A:A:D138 6.4554248
17A:A:I141 7.1825406
18A:A:R148 7.8875466
19A:A:Y159 12.1585119
20A:A:Y160 6.364506
21A:A:D163 7.82754114
22A:A:Y172 12.3285118
23A:A:P174 7.01254119
24A:A:D178 6.1385119
25A:A:R181 10.35754116
26A:A:R183 6.398599
27A:A:F194 8.665478
28A:A:F201 9.71833677
29A:A:R213 6.024509
30A:A:R214 7.3225447
31A:A:W216 9.134509
32A:A:M227 6.56477
33A:A:E234 10.102567
34A:A:Y235 6.83333668
35A:A:R247 10.055469
36A:A:M248 6.98468
37A:A:E250 6.5409
38A:A:F255 6.815669
39A:A:Y261 9.417128
40A:A:W263 16.17754125
41A:A:F264 10.835129
42A:A:F272 7.05579
43A:A:N274 6.09499
44A:A:K275 8.9225499
45A:A:D277 5.525409
46A:A:Y291 13.842565
47A:A:F292 9.17568
48A:A:Y295 8.906506
49A:A:F313 4.904569
50A:A:C330 5.12254207
51A:A:T334 8.1754239
52I:I:?2 7.69590
53I:I:?1 8.8725490
54K:K:D3 5.4025409
55K:K:V7 4.7525409
56K:K:Y13 5.99714739
57K:K:L34 7.246588
58K:K:Y46 8.6725134
59K:K:F55 8.73547
60K:K:F59 9.99447
61K:K:Y65 6.025445
62K:K:F68 8.4775408
63K:K:F71 5.7145285
64K:K:L76 4.194502
65K:K:F85 8.18748
66K:K:Y86 6.94547
67K:K:Y92 6.916545
68K:K:R101 7.434547
69K:K:I108 4.76445
70K:K:F109 6.588503
71K:K:I113 7.855445
72K:K:H122 7.01714743
73K:K:F124 9.14333643
74K:K:I129 3.9625442
75K:K:Q133 6.0525403
76K:K:L145 5.8875444
77K:K:F146 6.67333648
78K:K:Y149 7.90714744
79K:K:F162 6.6925408
80K:K:F171 6.39254275
81K:K:R173 7.13714789
82K:K:F174 5.015407
83K:K:W177 7.69429789
84K:K:N179 7.1985176
85K:K:E181 8.9775489
86K:K:L186 6.4525458
87K:K:F191 7.05659
88K:K:H194 5.775409
89K:K:R195 6.3725439
90K:K:I196 4.784299
91K:K:R199 5.3125409
92K:K:F202 4.864509
93K:K:E204 5.5445299
94K:K:Y206 6.86754298
95K:K:R209 5.0175409
96K:K:K210 8.76167658
97K:K:T213 8.42459
98K:K:Y217 8.42333659
99K:K:M219 5.242558
100K:K:K220 6.0775439
101K:K:K224 8.2025439
102K:K:R226 7.0625409
103K:K:E239 5.905439
104K:K:R240 5.6575439
105K:K:L243 6.43439
106K:K:P252 5.4125427
107K:K:F253 8.498529
108K:K:Y259 6.21375859
109K:K:H262 5.445438
110K:K:L267 7.4725439
111K:K:F269 5.926538
112K:K:I270 7.5325458
113K:K:L279 5.0225409
114K:K:H280 4.015409
115K:K:Y281 9.26754219
116K:K:H282 7.0725219
117K:K:F289 5.6075408
118K:K:M294 5.8375428
119K:K:F296 8.91529
120K:K:Y297 6.504529
121K:K:E300 9.032529
122K:K:L303 6.3375427
123K:K:V313 2.71408
124K:K:Y315 6.09667639
125K:K:D317 7.275439
126K:K:N322 6.175439
127K:K:H330 9.94529
128K:K:F342 9.315406
129K:K:Y356 6.994539
130K:K:P359 5.75149
131K:K:E360 5.338577149
132K:K:L362 6.2925406
133K:K:Y368 9.555409
134K:K:S371 5.73254148
135K:K:D373 6.5425409
136K:K:F375 6.9456148
137K:K:F382 8.27526
138K:K:K383 5.5075439
139K:K:R386 6.758525
140K:K:L413 4.9075427
141K:K:F417 5.32286727
142K:K:L421 7.995425
143K:K:L424 4.5975425
144K:K:R436 7.211437149
145K:K:K448 7.648527
146K:K:F452 8.81526
147K:K:F453 7.04428
148K:K:W458 7.916527
149K:K:Q464 6.5025425
150K:K:Y466 6.955403
151K:K:P472 4.614219
152K:K:V477 5.7175438
153K:K:N478 4.68254219
154K:K:Y506 6.148539
155K:K:F509 6.652539
156K:K:R516 8.228559
157K:K:W517 9.62409
158K:K:Q518 7.8875489
159K:K:E520 9.698559
160K:K:F526 7.83167688
161K:K:I529 3.635485
162K:K:L555 8.75754104
163K:K:M561 5.65254134
164K:K:H562 11.0145107
165K:K:M565 10.215405
166K:K:W576 7.9725408
167K:K:Y580 9.246676108
168K:K:F581 7.694316
169K:K:Y582 6.7954105
170K:K:R591 9.034105
171K:K:L601 4.55754154
172K:K:M603 2.22407
173K:K:I606 6.98254154
174K:K:I624 4.274153
175K:K:Q633 6.9125407
176K:K:E639 6.774176
177K:K:Q642 7.18754138
178K:K:R648 8.6154154
179K:K:Y651 6.5725155
180K:K:?701 9.1751030
181L:L:P10 9.6525410
182L:L:Y11 5.455400
183L:L:I12 7.355610
184L:L:L13 7.492510
185O:O:?1 11.76171290
186R:R:E53 6.22412
187R:R:V56 6.5175412
188R:R:T58 5.7975411
189R:R:Y70 6.074517
190R:R:F74 5.9175407
191R:R:L108 5.43254169
192R:R:T115 4.625407
193R:R:M120 6.165418
194R:R:E123 7.264516
195R:R:F127 5.418514
196R:R:H132 5.8665184
197R:R:P133 4.33254185
198R:R:W134 6.743336198
199R:R:Y144 9.0225416
200R:R:Y145 9.685414
201R:R:R148 7.4125417
202R:R:D149 8.724225
203R:R:L157 6.955406
204R:R:E165 8.71408
205R:R:Y167 5.77408
206R:R:F174 5.55407
207R:R:V201 6.9475405
208R:R:L204 7.64254225
209R:R:F205 10.51414
210R:R:M207 7.1406
211R:R:E209 6.16754195
212R:R:C224 6.82254199
213R:R:P226 5.67515
214R:R:N240 9.334226
215R:R:W316 10.1875418
216R:R:R322 6.55333615
217R:R:F326 4.645414
218R:R:Y342 5.83833614
219R:R:H343 7.9375414
220R:R:Y344 5.815411
221R:R:Y346 8.888514
222R:R:N350 5.79516
223R:R:F353 7.086517
224R:R:Y354 7.54125817
225R:R:F371 4.7425408
226R:R:F375 7.5425407
227W:W:?1 9.8127311160
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Int. Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.

Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1A:A:R213 A:A:W216 64.710310YesYes099
2A:A:R213 A:A:T47 60.30963.88YesNo098
3A:A:R247 A:A:T47 51.70456.47YesNo098
4A:A:E49 A:A:R247 33.91538.14NoYes099
5A:A:E49 A:A:R183 33.33486.98NoYes099
6A:A:R183 O:O:?1 25.78978.57YesYes990
7A:A:K52 O:O:?1 12.177410.71YesYes090
8A:A:M248 A:A:Y291 11.53288.38YesYes685
9A:A:E234 A:A:M248 14.003810.83YesYes678
10A:A:F220 A:A:W216 66.6085.01NoYes099
11A:A:W263 A:A:Y261 35.156112.54YesYes1258
12A:A:W263 K:K:F109 35.72887.02YesYes053
13A:A:Y261 K:K:M114 35.15629.58YesNo084
14K:K:F109 K:K:M114 35.24244.98YesNo034
15K:K:F109 K:K:I113 72.044312.56YesYes035
16K:K:F85 K:K:I113 71.82053.77YesYes485
17K:K:F85 K:K:I153 75.46526.28YesNo485
18K:K:I153 K:K:Y86 81.38993.63NoYes457
19K:K:F59 K:K:Y86 84.092810.32YesYes477
20K:K:F55 K:K:F59 86.660615YesYes477
21K:K:F162 K:K:F55 89.942611.79YesYes087
22K:K:F162 K:K:I58 90.13475.02YesNo087
23K:K:F174 K:K:I58 90.19867.54YesNo077
24K:K:F174 K:K:Q61 85.9555.86YesNo079
25K:K:K178 K:K:Q61 45.13446.78NoNo099
26K:K:E181 K:K:K178 49.13329.45YesNo099
27K:K:E181 K:K:W517 90.026214.17YesYes099
28K:K:W517 K:K:Y259 1008.68YesYes099
29K:K:K210 K:K:Y259 31.71299.55YesYes589
30K:K:D212 K:K:K210 43.663812.44NoYes588
31K:K:D212 K:K:K30 43.65466.91NoNo089
32K:K:A211 K:K:K30 43.56774.82NoNo089
33K:K:A211 R:R:F174 43.48062.77NoYes087
34R:R:F174 R:R:H172 41.6392.26YesNo076
35R:R:H172 R:R:K175 41.462213.1NoNo064
36R:R:K175 R:R:L168 41.28522.82NoNo044
37R:R:A176 R:R:L168 41.1084.73NoNo064
38R:R:A176 R:R:M180 41.01933.22NoNo067
39R:R:E165 R:R:M180 40.752813.53YesNo087
40R:R:E165 R:R:H104 40.485811.08YesNo088
41R:R:H104 R:R:S161 40.39678.37NoNo087
42R:R:N158 R:R:S161 40.30752.98NoNo087
43R:R:L108 R:R:N158 39.77126.87YesNo098
44K:K:Q518 K:K:Q61 41.072212.8YesNo099
45K:K:E181 K:K:Q518 41.06975.1YesYes899
46K:K:L186 K:K:Y259 33.77724.69YesYes589
47K:K:F261 K:K:L186 33.35249.74NoYes588
48K:K:F261 K:K:S268 39.447913.21NoNo088
49K:K:C221 K:K:S268 78.9063.44NoNo098
50K:K:C221 K:K:Y206 78.75054.03NoYes098
51K:K:I196 K:K:Y206 75.05096.04YesYes2998
52K:K:I196 K:K:I485 74.99937.36YesNo099
53K:K:G198 K:K:I485 74.37083.53NoNo099
54K:K:?701 K:K:G198 74.21357.4YesNo009
55K:K:?701 K:K:I197 12.561919.41YesNo309
56K:K:I197 K:K:Y13 12.50483.63NoYes399
57K:K:I270 K:K:Y259 33.80827.25YesYes589
58K:K:I270 K:K:M219 33.74914.37YesYes588
59K:K:M219 K:K:S268 39.61387.67YesNo088
60K:K:P35 K:K:Q176 11.8254.74NoNo059
61K:K:D635 K:K:E639 13.39167.8NoYes046
62K:K:D635 K:K:R578 13.1149.53NoNo046
63K:K:E52 K:K:K178 12.42135.4NoNo059
64K:K:E52 K:K:R50 10.24793.49NoNo053
65K:K:R50 K:K:Y46 10.17718.52NoYes034
66K:K:V521 K:K:W177 10.16613.68NoYes089
67K:K:F191 K:K:K210 12.57878.69YesYes598
68K:K:?701 K:K:K220 10.34018.72YesYes309
69K:K:?701 K:K:D335 51.48716.71YesNo309
70K:K:D317 K:K:D335 22.54123.99YesNo399
71K:K:D317 K:K:Y315 15.8313.45YesYes399
72K:K:M308 K:K:Y315 12.54428.38NoYes099
73K:K:I254 K:K:M308 12.19474.37NoNo099
74K:K:H307 K:K:I254 11.84766.63NoNo089
75K:K:D335 K:K:N322 28.78225.39NoYes399
76K:K:N322 K:K:Y315 15.82146.98YesYes399
77K:K:K319 K:K:N322 12.9155.6NoYes399
78K:K:K319 K:K:Y356 12.56665.97NoYes399
79K:K:D373 K:K:Y315 17.45243.45YesYes099
80K:K:D373 K:K:L305 12.54594.07YesNo099
81K:K:L305 K:K:L377 11.5024.15NoNo096
82K:K:L377 K:K:L381 11.15866.92NoNo065
83K:K:L381 K:K:M294 10.47794.24NoYes058
84R:R:L108 R:R:N360 34.53016.87YesNo1699
85R:R:D112 R:R:N360 34.87376.73NoNo099
86R:R:D112 R:R:S357 34.307510.31NoNo099
87R:R:S357 R:R:T115 34.21296.4NoYes097
88R:R:F353 R:R:T115 33.14433.89YesYes077
89R:R:F353 R:R:Y319 17.51636.19YesNo076
90R:R:R322 R:R:Y319 11.39776.17YesNo056
91R:R:F353 R:R:Y354 13.430614.44YesYes177
92A:A:F220 A:A:Y261 66.75165.16NoYes1298
93K:K:V521 K:K:W517 10.14738.58NoYes089
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1 Node2 LinkStrength Comm IsNode1Hub? IsNode2Hub? Node1Cons Node2Cons Node1Shell Node2Shell
L:L:R8 R:R:E53 4.65 1 No Yes 0 2 0 1
L:L:R8 R:R:R212 5.33 1 No No 0 1 0 1
L:L:R8 R:R:Y339 11.32 1 No No 0 2 0 1
L:L:R9 R:R:F326 6.41 0 No Yes 0 4 0 1
L:L:P10 R:R:W334 16.21 1 Yes No 0 4 0 1
L:L:P10 R:R:Y339 6.95 1 Yes No 0 2 0 1
L:L:P10 R:R:Y342 11.13 1 Yes Yes 0 4 0 1
L:L:Y11 R:R:E53 5.61 0 Yes Yes 0 2 0 1
L:L:Y11 R:R:V223 8.83 0 Yes No 0 4 0 1
L:L:Y11 R:R:T225 3.75 0 Yes No 0 4 0 1
L:L:I12 R:R:F127 5.02 1 Yes Yes 0 4 0 1
L:L:I12 R:R:H131 11.93 1 Yes No 0 3 0 1
L:L:I12 R:R:Y342 6.04 1 Yes Yes 0 4 0 1
L:L:I12 R:R:H343 6.63 1 Yes Yes 0 4 0 1
L:L:I12 R:R:Y346 10.88 1 Yes Yes 0 4 0 1
L:L:L13 R:R:Y145 15.24 1 Yes Yes 0 4 0 1
L:L:L13 R:R:F205 7.31 1 Yes Yes 0 4 0 1
L:L:L13 R:R:P226 6.57 1 Yes Yes 0 5 0 1
L:L:L13 R:R:F326 3.65 1 Yes Yes 0 4 0 1
L:L:L13 R:R:Y346 4.69 1 Yes Yes 0 4 0 1
R:R:E53 R:R:N57 7.89 1 Yes No 2 2 1 2
R:R:E53 R:R:Y339 6.73 1 Yes No 2 2 1 1
R:R:H131 R:R:V56 11.07 1 No Yes 3 2 1 2
R:R:H343 R:R:V56 4.15 1 Yes Yes 4 2 1 2
R:R:E123 R:R:F127 3.5 1 Yes Yes 6 4 2 1
R:R:E123 R:R:N350 7.89 1 Yes Yes 6 6 2 2
R:R:F127 R:R:Y144 5.16 1 Yes Yes 4 6 1 2
R:R:F127 R:R:Y145 5.16 1 Yes Yes 4 4 1 1
R:R:F127 R:R:Y346 8.25 1 Yes Yes 4 4 1 1
R:R:H131 R:R:H343 15.53 1 No Yes 3 4 1 1
R:R:Y144 R:R:Y145 5.96 1 Yes Yes 6 4 2 1
R:R:F205 R:R:Y145 12.38 1 Yes Yes 4 4 1 1
R:R:F205 R:R:M207 13.68 1 Yes Yes 4 6 1 2
R:R:F205 R:R:P226 8.67 1 Yes Yes 4 5 1 1
R:R:Q210 R:R:R212 5.84 0 No No 1 1 2 1
R:R:Q210 R:R:T225 5.67 0 No No 1 4 2 1
R:R:P226 R:R:T225 5.25 1 Yes No 5 4 1 1
R:R:P226 R:R:V233 3.53 1 Yes No 5 5 1 2
R:R:F326 R:R:P226 4.33 1 Yes Yes 4 5 1 1
R:R:R322 R:R:Y342 6.17 1 Yes Yes 5 4 2 1
R:R:R322 R:R:Y346 11.32 1 Yes Yes 5 4 2 1
R:R:N350 R:R:R322 3.62 1 Yes Yes 6 5 2 2
R:R:C327 R:R:F326 4.19 0 No Yes 3 4 2 1
R:R:I329 R:R:W334 4.7 0 No No 3 4 2 1
R:R:W334 R:R:Y342 3.86 1 No Yes 4 4 1 1
R:R:H343 R:R:Y342 5.44 1 Yes Yes 4 4 1 1
R:R:N350 R:R:Y346 9.3 1 Yes Yes 6 4 2 1
R:R:S213 R:R:V223 3.23 0 No No 1 4 2 1
R:R:M325 R:R:Y342 2.39 0 No Yes 4 4 2 1

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
75.00Single4XEENeurotensin4XEE-NTS1-Neurotensin
75.00Single4XESNeurotensin4XES-NTS1-Neurotensin
75.00Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
75.00Single6YVRNTS8-136YVR-NTS1-NTS8-13
75.00Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
75.00Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
75.00Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
72.22Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
70.59Single4BUONeurotensin4BUO-NTS1-Neurotensin
68.75Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
68.75Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
68.75Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
68.75Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
68.75Consensusneurotensin_onOrthosteric Ligandnts1_on
68.75Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
66.67Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
64.71Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
64.29Single4BWBNeurotensin4BWB-NTS1-Neurotensin
61.11Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
61.11Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
61.11Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
58.82Single4BV0Neurotensin4BV0-NTS1-Neurotensin
58.82Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
57.89Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
56.25Single5T04Neurotensin5T04-NTS1-Neurotensin
55.56Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
55.56Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
55.56Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
55.56Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
55.56Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
52.63Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
52.63Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
52.38Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
50.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
50.00Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
50.00Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
50.00Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
48.00Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
48.00Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
47.37Single6OS2TRV0266OS2-AT1-TRV026
47.37Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
47.37Single8XWSCXCL58XWS-CXCR2-CXCL5
47.37Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
47.06Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
47.06Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
47.06Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
47.06Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
47.06Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
47.06Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
45.45Single7XNACYN1548067XNA-SST2-CYN154806
45.45Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
44.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
43.75Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
43.75Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
43.75Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
43.75Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
43.75Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
43.48Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
42.86Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
42.86Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
42.86Single8XQJJN2418XQJ-Apelin-JN241
42.86Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
42.86Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
42.31Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
42.11Single6OS1TRV0266OS1-AT1-TRV026
42.11Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
42.11Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
42.11Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
41.67Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
41.67Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
41.18Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
41.18Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
41.18Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
41.18Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
40.91Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
40.91Single8XWNCXCL88XWN-CXCR2-CXCL8
40.91Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
40.91Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
40.91Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
40.91Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
40.91Consensussomatostatin_offOrthosteric Ligandsst2_off
40.00Single4XNWMRS25004XNW-P2Y1-MRS2500
40.00Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
40.00Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
40.00Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
40.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
40.00Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
40.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8XQJJN2418XQJ-Apelin-JN241
40.00Single8XWACXCL18XWA-CXCR2-CXCL1
40.00Single8XWMCXCL68XWM-CXCR2-CXCL6
40.00Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
40.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
39.29Single5GLHEndothelin-15GLH-ETB-Endothelin-1
39.29Single6IGKEndothelin-36IGK-ETB-Endothelin-3
39.29Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
39.29Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
39.29Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
39.13Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
39.13Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
39.13Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
39.13Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
39.13Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
39.13Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
39.13Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
39.13Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
39.13Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
39.13Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
38.89Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
38.89Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
38.89Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
38.89Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
38.46Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
38.46Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
38.46Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
38.46Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
38.46Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
38.10Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
38.10Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
38.10Single8XVUCXCL28XVU-CXCR2-CXCL2
38.10Single8XWFCXCL38XWF-CXCR2-CXCL3
38.10Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
38.10Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
38.10Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
37.93Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
37.50Single3OE0CVX153OE0-CXCR4-CVX15
37.50Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
37.50Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
37.50Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
37.50Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
37.50Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
37.50Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
37.50Consensusgq_nucleotideOrthosteric Ligandgq_p2y
37.50Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
37.04Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
37.04Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
37.04Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
37.04Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
36.84Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
36.84Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
36.84Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
36.84Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
36.67Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
36.36Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
36.36Single6KNMJN241-96KNM-Apelin-JN241-9
36.36Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
36.36Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
36.36Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
36.36Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
36.00Single6JODAngiotensin II6JOD-AT2-Angiotensin II
36.00Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
36.00Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
36.00Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
36.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
36.00Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
36.00Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
36.00Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
35.71Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
35.71Single8IY6Endothelin-18IY6-ETB-Endothelin-1
35.29Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
35.29Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
35.29Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
35.29Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
35.00Single7F1TMIP-1a7F1T-CCR5-MIP-1a
35.00Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
35.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
35.00Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
34.78Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
34.78Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
34.78Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
34.78Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.62Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
34.62Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
34.62Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
34.62Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
34.62Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
34.62Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
34.62Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
34.62Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.48Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
33.33Single4XT3Fractalkine4XT3-US28-Fractalkine
33.33Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
33.33Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
33.33Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
33.33Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
33.33Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
33.33Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
33.33Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
33.33Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
33.33Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
33.33Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
33.33Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
33.33Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
33.33Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
33.33Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
33.33Consensusp2y_offOrthosteric Ligandp2y1_off
33.33Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
33.33Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
32.14Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
32.14Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
32.14Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
32.14Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
32.00Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
32.00Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
32.00Consensusangiotensin_onOrthosteric Ligandat1_on
32.00Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
32.00Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
32.00Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
31.82Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
31.82Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
31.82Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
31.82Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
31.82Consensuscck_onOrthosteric Ligandccka_on cckb_on
31.82Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
31.82Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
31.82Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
31.82Consensuschemerin_onOrthosteric Ligandcml1_on
31.82Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
31.82Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
31.58Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
31.58Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
31.58Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
31.58Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
31.58Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
31.58Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
31.58Consensushca_on_gpOrthosteric Ligandhca2_on_gp
31.58Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
31.58Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
31.25Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
31.25Single7V6A-7V6A-M4-PubChem 9864275-Gi1/β1/γ2
31.25Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
31.03Single6IGLIRL16206IGL-ETB-IRL1620
31.03Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
31.03Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
31.03Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
31.03Consensusbradykinin_onOrthosteric Ligandbk2_on
31.03Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
31.03Consensusendothelin_onOrthosteric Ligandetb_on eta_on
31.03Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
30.77Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
30.77Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
30.77Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
30.77Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.77Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
30.77Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
30.77Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
30.77Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
30.77Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
30.43Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
30.43Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
30.43Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
30.43Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
30.43Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
30.43Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
30.43Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
30.00Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
30.00Single6Z4SSR486926Z4S-NTS1-SR48692
30.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
30.00Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
29.63Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
29.63Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
29.63Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
29.63Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.63Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
29.63Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
29.63Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
29.63Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
29.63Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
29.63Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.41Single4O9RCyclopamine4O9R-SMO-Cyclopamine
29.41Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
29.41Single7UL2SR486927UL2-NTS1-SR48692-Na
29.41Consensusneurotensin_offOrthosteric Ligandnts1_off
29.41Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
29.17Single4XT1Fractalkine4XT1-US28-Fractalkine
29.17Single7F8XNN90567F8X-CCKA-NN9056
29.17Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
29.17Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
29.17Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
29.17Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
29.17Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
29.17Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
29.17Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
29.03Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
29.03Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
28.57Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
28.57Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
28.57Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
28.57Single7SK3CXCL127SK3-ACKR3-CXCL12
28.57Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
28.57Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.57Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
28.57Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
28.57Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
28.57Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
28.57Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
28.57Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
28.57Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
28.57Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
28.57Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
28.57Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
28.57Consensusrelaxin_onOrthosteric Ligandrxfp4_on
28.57Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
28.00Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
28.00Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
28.00Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
28.00Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
28.00Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
28.00Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
28.00Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
27.78Single4QINSAG1.54QIN-SMO-SAG1.5
27.78Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
27.78Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
27.78Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
27.78Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
27.78Single8GNGIstradefylline8GNG-A2A-Istradefylline
27.78Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
27.78Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
27.78Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
27.78Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
27.78Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
27.78Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
27.59Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
27.59Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
27.27Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
27.27Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
27.27Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
27.27Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
27.27Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
27.27Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
27.27Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
27.27Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
27.27Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
26.92Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
26.92Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
26.92Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
26.92Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
26.92Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
26.92Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
26.92Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
26.92Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
26.92Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
26.67Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
26.67Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
26.67Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
26.67Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
26.67Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
26.67Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
26.32Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
26.32Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
26.32Single5UVIZM-2413855UVI-A2A-ZM-241385
26.32Single6MH8ZM-2413856MH8-A2A-ZM-241385
26.32Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
26.32Single6ZINSR486926ZIN-NTS1-SR48692
26.32Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
26.32Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
26.32Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
26.32Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
26.32Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
26.32Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
26.32Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
26.32Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
26.32Consensushca_onOrthosteric Ligandhca2_on
26.09Single7EZCUKA7EZC-A2A-UKA
26.09Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
26.09Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
26.09Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
26.09Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
25.93Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
25.93Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
25.93Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
25.93Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
25.93Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
25.81Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
25.81Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.81Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.81Consensusbombesin_onOrthosteric Ligandbb2_on
25.81Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
25.81Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
25.81Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.00Single3EMLZM-2413853EML-A2A-ZM-241385
25.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
25.00Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
25.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
25.00Single5WF6UK-4320975WF6-A2A-UK-432097
25.00Single6D27CAY104716D27-DP2-CAY10471
25.00Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
25.00Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
25.00Single6S0LZM-2413856S0L-A2A-ZM-241385
25.00Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
25.00Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
25.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
25.00Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
25.00Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
25.00Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
25.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
25.00Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
25.00Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
25.00Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
25.00Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
25.00Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
25.00Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
25.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
25.00Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
25.00Single8K5DGSK2560738K5D-HCA2-GSK256073
25.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
25.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
25.00Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
25.00Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
25.00Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
25.00Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
25.00Single8ZRTET-18ZRT-ETB-ET-1
25.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
25.00Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
25.00Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
25.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
25.00Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
25.00Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
25.00Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
24.24Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
24.14Single6FJ3PTH6FJ3-PTH1-PTH
24.14Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
24.14Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
24.14Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
24.14Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
24.14Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
24.00Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
24.00Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
24.00Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
24.00Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
24.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.00Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
24.00Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
24.00Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
24.00Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
24.00Consensuslpl_onOrthosteric Ligands1p_on lpa_on
24.00Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
24.00Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
24.00Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
23.81Single5IUAQ274563485IUA-A2A-Q27456348-Na
23.81Single5N2RPSB-365N2R-A2A-PSB-36-Na
23.81Single5N2SPSB365N2S-A1-PSB36
23.81Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
23.81Single6S0QZM-2413856S0Q-A2A-ZM-241385
23.81Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
23.81Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
23.81Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
23.81Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
23.81Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.81Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
23.81Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
23.81Single8GNEKW-63568GNE-A2A-KW-6356-Na
23.81Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
23.81Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
23.81Single8QOTNanobody-E8QOT-μ-Nanobody-E
23.81Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
23.81Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
23.81Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
23.81Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
23.53Single8JPSCCL78JPS-ACKR1-CCL7
23.53Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
23.33Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
23.33Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
23.33Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
23.33Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
23.33Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
23.08Single3QAKUK-4320973QAK-A2A-UK-432097
23.08Single7SK5CXCL127SK5-ACKR3-CXCL12
23.08Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
23.08Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
23.08Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
23.08Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
23.08Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
22.73Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
22.73Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
22.73Single7PX4PSB-21137PX4-A2A-PSB-2113
22.73Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
22.73Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
22.73Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
22.73Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
22.73Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
22.73Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
22.73Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
22.73Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
22.73Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.73Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
22.73Consensuslpa_onOrthosteric Ligandlpa1_on
22.73Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
22.58Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
22.58Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
22.58Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
22.22Single3OE9IT1t3OE9-CXCR4-IT1t
22.22Single5WF5UK-4320975WF5-A2A-UK-432097
22.22Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
22.22Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
22.22Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
22.22Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
22.22Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
22.22Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
22.22Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
22.22Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
22.22Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.22Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
22.22Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
22.22Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
22.22Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
22.22Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
22.22Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
22.22Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
21.88Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
21.74Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
21.74Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
21.74Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
21.74Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
21.74Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
21.74Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
21.74Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
21.74Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
21.74Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
21.74Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
21.74Consensuslpa_offOrthosteric Ligandlpa1_off
21.74Consensuslpl_offOrthosteric Ligands1p_off lpa_off
21.62Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
21.43Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
21.43Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
21.43Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
21.43Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
21.43Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
21.43Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
21.43Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
21.21Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
21.21Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
21.21Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
21.05Single3PWHZM-2413853PWH-A2A-ZM-241385
21.05Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
21.05Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
21.05Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
21.05Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
21.05Single7F8YDevazepide7F8Y-CCKA-Devazepide
21.05Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
21.05Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
21.05Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
21.05Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
21.05Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
21.05Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
21.05Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
20.83Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
20.83Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
20.83Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
20.83Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
20.83Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
20.83Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.83Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
20.83Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
20.83Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
20.83Consensusprostanoid_offOrthosteric Ligandep_off dp_off
20.69Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
20.69Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
20.69Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
20.69Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
20.59Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
20.59Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
20.59Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
20.00Single3REYXAC3REY-A2A-XAC
20.00Single4UG2CGS216804UG2-A2A-CGS21680
20.00Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
20.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
20.00Single5IUBQ274563445IUB-A2A-Q27456344-Na
20.00Single5JTBZM-2413855JTB-A2A-ZM-241385
20.00Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
20.00Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
20.00Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
20.00Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
20.00Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
20.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
20.00Single7AROLUF58337ARO-A2A-LUF5833-Na
20.00Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
20.00Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
20.00Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
20.00Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
20.00Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
20.00Single7T32ZM-2413857T32-A2A-ZM-241385
20.00Single7XN9L-054,5227XN9-SST2-L-054,522
20.00Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
20.00Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
20.00Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
20.00Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
20.00Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
20.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
20.00Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
20.00Single8K5CAcipimox8K5C-HCA2-Acipimox
20.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
20.00Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
20.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
20.00Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Consensusa2_offOrthosteric Liganda2a_off
20.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
20.00Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
20.00Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
20.00Consensusgrh_offOrthosteric Ligandgnrh1_off
20.00Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
20.00Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
19.35Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
19.35Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
19.35Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
19.35Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
19.35Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
19.23Single4IARErgotamine4IAR-5-HT1B-Ergotamine
19.23Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
19.23Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
19.23Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
19.23Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
19.23Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
19.23Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
19.23Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
19.23Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
19.23Single8WDTphotoNECA8WDT-A2A-photoNECA
19.23Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
19.23Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.23Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
19.23Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
19.05Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
19.05Single4QIMANTA XV4QIM-SMO-ANTA XV
19.05Single5IU8Q274563475IU8-A2A-Q27456347-Na
19.05Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
19.05Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
19.05Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
19.05Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
19.05Single7PYRPSB-21157PYR-A2A-PSB-2115
19.05Single7V3ZCP559407V3Z-CB1-CP55940
19.05Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
19.05Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
19.05Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
19.05Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
19.05Consensusa3_onOrthosteric Liganda3a_on
19.05Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
19.05Consensuscck_offOrthosteric Ligandccka_off
19.05Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
19.05Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
18.75Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
18.75Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
18.75Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
18.75Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
18.75Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
18.75Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
18.75Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
18.52Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
18.52Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
18.52Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
18.52Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
18.52Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
18.52Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
18.52Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
18.52Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
18.52Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
18.52Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
18.18Single4JKVTaladegib4JKV-SMO-Taladegib
18.18Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
18.18Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
18.18Single6D26Fevipiprant6D26-DP2-Fevipiprant
18.18Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
18.18Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
18.18Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
18.18Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
18.18Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
18.18Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
18.18Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
18.18Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
18.18Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
18.18Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
18.18Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
18.18Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
18.18Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
18.18Consensusa3_on_gpOrthosteric Liganda3a_on_gp
18.18Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
18.18Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
18.18Consensusadenosine_offOrthosteric Liganda1_off a2_off
18.18Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
18.18Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
18.18Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
18.18Consensusdp_offOrthosteric Liganddp2_off
18.18Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
18.18Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
18.18Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
18.18Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
17.86Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
17.86Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
17.86Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
17.86Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
17.86Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
17.86Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
17.86Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
17.86Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.86Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.65Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
17.65Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
17.65Single8A2OTheophylline8A2O-A2A-Theophylline-Na
17.65Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
17.65Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
17.39Single5TZRMK86665TZR-FFA1-MK8666
17.39Single5V56TC1145V56-SMO-TC114
17.39Single5V57TC1145V57-SMO-TC114
17.39Single5XR8AM8415XR8-CB1-AM841
17.39Single5XRAAM115425XRA-CB1-AM11542
17.39Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
17.39Single7B6WCyclazosin7B6W-α1b-Cyclazosin
17.39Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
17.39Single7FEECP559407FEE-CB1-CP55940-ZCZ011
17.39Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
17.39Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
17.39Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
17.39Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
17.39Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
17.39Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
17.39Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
17.39Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
17.39Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
17.39Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
17.39Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
17.39Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.39Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
17.39Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
17.39Consensusa2_onOrthosteric Liganda2b_on
17.39Consensusa2_on_gpOrthosteric Liganda2b_on_gp
17.39Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.39Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.39Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
17.39Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
17.39Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
17.39Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
17.39Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
17.39Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
17.24Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
17.24Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
17.24Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
17.24Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
17.24Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.24Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
17.24Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
17.24Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
17.24Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
17.14Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
17.14Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
17.14Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single3OE6IT1t3OE6-CXCR4-IT1t
16.67Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
16.67Single4PY02MeSATP4PY0-P2Y12-2MeSATP
16.67Single4RWADIPP-NH24RWA-δ-DIPP-NH2
16.67Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
16.67Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
16.67Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
16.67Single6KQICP559406KQI-CB1-CP55940-Org27569
16.67Single6ME5Agomelatine6ME5-MT1-Agomelatine
16.67Single6MXTSalmeterol6MXT-β2-Salmeterol
16.67Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
16.67Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
16.67Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
16.67Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
16.67Single7K15MKD0467K15-BLT1-MKD046-Na
16.67Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
16.67Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
16.67Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
16.67Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
16.67Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
16.67Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
16.67Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
16.67Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
16.67Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
16.67Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
16.67Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
16.67Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
16.67Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
16.67Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
16.67Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
16.67Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
16.67Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
16.67Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
16.67Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
16.67Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.67Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.67Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
16.67Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
16.67Consensusorexin_onOrthosteric Ligandox2_on
16.67Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.67Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
16.67Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
16.67Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.22Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
16.13Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
16.13Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
16.13Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
16.13Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
16.00Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
16.00Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
16.00Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
16.00Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
16.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
16.00Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
16.00Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
16.00Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
16.00Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
16.00Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
16.00Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
16.00Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
16.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
16.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
16.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
16.00Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
15.79Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
15.79Single5L7IVismodegib5L7I-SMO-Vismodegib
15.79Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
15.79Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
15.79Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
15.79Single8K5BNiacin8K5B-HCA2-Niacin
15.79Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
15.79Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
15.79Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
15.79Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
15.62Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
15.62Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
15.62Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
15.62Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
15.62Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
15.62Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
15.38Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
15.38Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
15.38Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
15.38Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
15.38Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
15.38Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
15.38Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
15.38Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
15.38Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
15.38Consensuskisspeptin_onOrthosteric Ligandkiss1_on
15.38Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
15.38Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
15.15Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
15.15Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
15.15Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
15.15Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
15.15Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
15.15Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
15.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
15.00Single3ODUIT1t3ODU-CXCR4-IT1t
15.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
15.00Single6ME9Ramelteon6ME9-MT2-Ramelteon
15.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
15.00Single7BR3Elagolix7BR3-GnRH1-Elagolix
15.00Single7F8ULintitript7F8U-CCKA-Lintitript
15.00Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
15.00Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
15.00Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
15.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
15.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
15.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
15.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
15.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
15.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
15.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
15.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
15.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.00Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
15.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
15.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
14.81Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
14.81Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
14.81Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
14.81Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
14.81Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.81Single8WKYPG-9348WKY-MC4-PG-934
14.81Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
14.81Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
14.81Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
14.81Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
14.81Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
14.81Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
14.71Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
14.71Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
14.29Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
14.29Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
14.29Single6AQFZM-2413856AQF-A2A-ZM-241385
14.29Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
14.29Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
14.29Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
14.29Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
14.29Single7VV6C48/807VV6-MRGPRX2-C48/80
14.29Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
14.29Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
14.29Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
14.29Single8IEBA1LYA8IEB-GPR156-A1LYA
14.29Single8IHKAcifran8IHK-HCA3-Acifran
14.29Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
14.29Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
14.29Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
14.29Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
14.29Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
14.29Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
14.29Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
14.29Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
14.29Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
14.29Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.29Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
13.79Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
13.79Single6W25SHU91196W25-MC4-SHU9119-Ca
13.79Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.64Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
13.64Single4YAYZD-71554YAY-AT1-ZD-7155
13.64Single5TGZAM65385TGZ-CB1-AM6538
13.64Single5UENDU1725UEN-A1-DU172
13.64Single5UIGCmpd-15UIG-A2A-Cmpd-1
13.64Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
13.64Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
13.64Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
13.64Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
13.64Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
13.64Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
13.64Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
13.64Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
13.64Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
13.64Single8CU6LJ-45178CU6-A2A-LJ-4517
13.64Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
13.64Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.64Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
13.64Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
13.64Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
13.64Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
13.64Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
13.64Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
13.64Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
13.64Single9IYAONO-97105319IYA-GPR55-ONO-9710531
13.64Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
13.51Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.33Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
13.33Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
13.33Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
13.33Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
13.33Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
13.33Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
13.33Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
13.33Consensusvasop-oxy_onOrthosteric Ligandv2_on
13.33Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
13.04Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
13.04Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
13.04Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
13.04Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
13.04Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
13.04Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
13.04Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
13.04Single7C4SS1P7C4S-S1P3-S1P
13.04Single7C61Ergotamine7C61-5-HT1B-Ergotamine
13.04Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
13.04Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
13.04Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
13.04Single7W41PD1762527W41-BB2-PD176252
13.04Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.04Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
13.04Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
13.04Single8JXSPF-61428JXS-D1-PF-6142
13.04Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
13.04Single8S4DCMF-0198S4D-Apelin-CMF-019
13.04Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
13.04Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
13.04Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
13.04Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
13.04Consensusblt_offOrthosteric Ligandblt1_off
13.04Consensusbombesin_offOrthosteric Ligandbb2_off
13.04Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
13.04Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
13.04Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
13.04Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
13.04Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
12.90Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
12.90Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
12.50Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
12.50Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
12.50Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
12.50Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
12.50Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
12.50Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
12.50Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.50Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
12.50Single7R0CAVP7R0C-V2-AVP-Arrestin2
12.50Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
12.50Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
12.50Single8E0GBU728E0G-μ-BU72
12.50Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
12.50Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
12.50Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
12.50Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
12.50Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
12.50Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
12.50Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
12.50Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
12.50Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
12.50Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
12.50Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.50Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
12.50Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
12.50Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
12.50Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.50Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
12.50Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.50Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.50Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.20Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
12.12Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
12.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
12.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
12.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
12.00Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
12.00Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
12.00Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
12.00Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
12.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
12.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
12.00Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.00Single8JJLOlodaterol8JJL-β2-Olodaterol
12.00Single8JWY2-1188JWY-A2A-2-118
12.00Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
12.00Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
12.00Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.00Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
12.00Single8XYIVUF106618XYI-CXCR3-VUF10661
12.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
12.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
12.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
12.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
12.00Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
12.00Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.00Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
12.00Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.00Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
12.00Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
11.90Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
11.76Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
11.76Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
11.76Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.76Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
11.76Single8HS2Fab0468HS2-GPR20-Fab046
11.76Single8PWNTheophylline8PWN-A2A-Theophylline
11.76Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.76Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.54Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
11.54Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
11.54Single6IBLArformoterol6IBL-β1-Arformoterol
11.54Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
11.54Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
11.54Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
11.54Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
11.54Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
11.54Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
11.54Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
11.54Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
11.54Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
11.54Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
11.54Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
11.11Single3NY9ICI118-5513NY9-β2-ICI118-551
11.11Single3RFMCaffeine3RFM-A2A-Caffeine
11.11Single5ZTYAM102575ZTY-CB2-AM10257
11.11Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
11.11Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
11.11Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
11.11Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
11.11Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
11.11Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
10.71Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
10.71Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
10.71Single7QA8Peptide7QA8-STE2-Peptide
10.71Single7QA8Peptide7QA8-STE2-Peptide
10.71Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
10.71Single8IEBA1LYA8IEB-GPR156-A1LYA
10.71Single8IEIA1LYA8IEI-GPR156-A1LYA
10.71Single8IEPA1LYA8IEP-GPR156-A1LYA
10.71Single8IEPA1LYA8IEP-GPR156-A1LYA
10.71Single8KIGSHU91198KIG-MC3-SHU9119-Ca
10.53Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
10.53Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
10.53Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
10.53Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
10.53Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
10.53Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.53Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
10.53Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
10.34Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
10.34Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
10.34Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
10.00Single6LI0C176LI0-GPR52-C17
10.00Single6PT2KGCHM076PT2-δ-KGCHM07
10.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
10.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
10.00Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
10.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
10.00Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
10.00Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
10.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
10.00Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
10.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
10.00Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
10.00Single9B9Y7DY9B9Y-CB1-7DY
10.00Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
10.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
9.68Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
9.68Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
9.68Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
9.52Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
9.52Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
9.52Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
9.52Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
9.52Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
9.52Single5U09Taranabant5U09-CB1-Taranabant
9.52Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
9.52Single6ME2Ramelteon6ME2-MT1-Ramelteon
9.52Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
9.52Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
9.52Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
9.52Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
9.52Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
9.52Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
9.52Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.52Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
9.52Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
9.52Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Single9BA0A1AKN9BA0-CB1-A1AKN
9.52Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
9.52Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
9.52Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
9.52Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
9.38Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
9.09Single2YDOAdenosine2YDO-A2A-Adenosine
9.09Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
9.09Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
9.09Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
9.09Single6KUXRS-799486KUX-α2a-RS-79948
9.09Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
9.09Single6V9SGTPL114036V9S-OX1-GTPL11403
9.09Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
9.09Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
9.09Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
9.09Single7UL3Famotidine7UL3-H2-Famotidine
9.09Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
9.09Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
9.09Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
9.09Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
9.09Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
9.09Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8K2WAMG4878K2W-CXCR3-AMG487
9.09Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
9.09Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
9.09Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
9.09Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
9.09Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
9.09Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
9.09Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
9.09Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
9.09Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
9.09Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
9.09Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
9.09Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
8.82Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
8.82Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
8.70Single2Y02Carmoterol2Y02-β1-Carmoterol
8.70Single2Y04Salbutamol2Y04-β1-Salbutamol
8.70Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
8.70Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
8.70Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
8.70Single6DRXLisuride6DRX-5-HT2B-Lisuride
8.70Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
8.70Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
8.70Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
8.70Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
8.70Single6PS1Timolol6PS1-β2-Timolol
8.70Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
8.70Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
8.70Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
8.70Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
8.70Single7UL4Alvimopan7UL4-μ-Alvimopan
8.70Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
8.70Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
8.70Single7YXAONO-54306087YXA-S1P5-ONO-5430608
8.70Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
8.70Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
8.70Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
8.70Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
8.70Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
8.70Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
8.70Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
8.70Single8RLNLUF58348RLN-A2A-LUF5834
8.70Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
8.70Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
8.70Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.70Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
8.70Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
8.70Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
8.70Single9B9ZA1AKO9B9Z-CB1-A1AKO
8.70Single9CHXS-Carazolol9CHX-β2-S-Carazolol
8.70Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
8.70Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
8.70Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
8.70Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
8.57Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
8.33Single2Y03Isoprenaline2Y03-β1-Isoprenaline
8.33Single4NTJAZD12834NTJ-P2Y12-AZD1283
8.33Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
8.33Single5C1MBU725C1M-μ-BU72
8.33Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
8.33Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
8.33Single6LUQHaloperidol6LUQ-D2-Haloperidol
8.33Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
8.33Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
8.33Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
8.33Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
8.33Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
8.33Single7SINNPS-21437SIN-CaS-NPS-2143
8.33Single7SINNPS-21437SIN-CaS-NPS-2143
8.33Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
8.33Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
8.33Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
8.33Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
8.33Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
8.33Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
8.33Single8TF5Oleic acid8TF5-GPR6-Oleic acid
8.33Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
8.33Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
8.33Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
8.33Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
8.33Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
8.33Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
8.33Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
8.33Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
8.33Consensusep_offOrthosteric Ligandep4_off
8.33Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
8.33Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.33Consensustrace-amine_onOrthosteric Ligandta1_on
8.11Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
8.00Single2YDVNECA2YDV-A2A-NECA
8.00Single3P0GBI1671073P0G-β2-BI167107
8.00Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
8.00Single4UHRCGS216804UHR-A2A-CGS21680
8.00Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
8.00Single5G53NECA5G53-A2A-NECA-Gs
8.00Single6H7JIsoprenaline6H7J-β1-Isoprenaline
8.00Single6J20Aprepitant6J20-NK1-Aprepitant
8.00Single6J21Aprepitant6J21-NK1-Aprepitant
8.00Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
8.00Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
8.00Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
8.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
8.00Single6WGTLSD6WGT-5-HT2A-LSD
8.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
8.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
8.00Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
8.00Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
8.00Single7TUYGSK682753A7TUY-GPR183-GSK682753A
8.00Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
8.00Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
8.00Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
8.00Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
8.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
8.00Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
8.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
8.00Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
8.00Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
8.00Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
8.00Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
8.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
8.00Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.00Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
7.69Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
7.69Single4AMIBucindolol4AMI-β1-Bucindolol
7.69Single4LDEBI1671074LDE-β2-BI167107
7.69Single4N4WSANT-14N4W-SMO-SANT-1
7.69Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
7.69Single5X33BIIL2605X33-BLT1-BIIL260
7.69Single6A93Risperidone6A93-5-HT2A-Risperidone
7.69Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
7.69Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
7.69Single7DFPSpiperone7DFP-D2-Spiperone
7.69Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
7.69Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
7.69Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
7.69Single7YITNalfurafine7YIT-κ-Nalfurafine
7.69Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
7.69Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
7.69Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
7.69Single8JJ8Formoterol8JJ8-β2-Formoterol
7.69Single8JWZAB9288JWZ-A2A-AB928-Na
7.69Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
7.69Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
7.69Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
7.69Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
7.69Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
7.69Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
7.69Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
7.69Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
7.69Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
7.69Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
7.41Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
7.41Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
7.41Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
7.41Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
7.41Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
7.41Single7UM4AS26747237UM4-5-HT5A-AS2674723
7.41Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
7.41Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
7.41Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
7.41Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
7.41Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
7.41Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
7.41Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
7.14Single5EE7MK08935EE7-Glucagon-MK0893
7.14Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
7.14Single6D35Cholesterol6D35-SMO-Cholesterol
7.14Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
7.14Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
7.14Single6PT3DPI-2876PT3-δ-DPI-287
7.14Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
7.14Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
7.14Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
7.14Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
7.14Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
7.14Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
7.14Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
7.14Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
7.14Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
7.14Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
7.14Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.14Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.14Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.14Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.14Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
7.14Single7DTTCa7DTT-CaS-Ca-Ca
7.14Single7DTTCa7DTT-CaS-Ca-Ca
7.14Single7DTUTryptophan7DTU-CaS-Tryptophan
7.14Single7DTUTryptophan7DTU-CaS-Tryptophan
7.14Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
7.14Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
7.14Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
7.14Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
7.14Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
7.14Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
7.14Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
7.14Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
7.14Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
7.14Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
7.14Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
7.14Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
7.14Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
7.14Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
7.14Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
7.14Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
7.14Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
7.14Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
7.14Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
7.14Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.14Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.14Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.14Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.14Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.14Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.14Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
7.14Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
7.14Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
7.14Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
7.14Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
7.14Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
7.14Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.14Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.14Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.14Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.14Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.14Single7SK9CCX6627SK9-ACKR3-CCX662
7.14Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
7.14Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
7.14Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
7.14Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
7.14Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
7.14Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
7.14Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
7.14Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
7.14Single7XW7K1-707XW7-TSH-K1-70
7.14Single8IEIA1LYA8IEI-GPR156-A1LYA
7.14Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
7.14Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
7.14Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
7.14Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
7.14Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
7.14Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
7.14Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
7.14Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
7.14Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
7.14Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
7.14Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
7.14Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
7.14Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
7.14Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
7.14Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
7.14Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
7.14Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
7.14Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
7.14Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
7.14Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
7.14Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
7.14Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
7.14Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
7.14Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
7.14Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
7.14Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
7.14Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
7.14Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
7.14Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
7.14Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
7.14Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
7.14Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
7.14Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
7.14Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
7.14Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
7.14Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
7.14Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
7.14Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
7.14Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
7.14Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
7.14Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
7.14Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
7.14Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
7.14Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
7.14Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
7.14Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
7.14Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
7.14Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
7.14Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
7.14Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
7.14Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
7.14Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
7.14Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
7.14Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
7.14Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
7.14Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
7.14Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
7.14Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
7.14Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8WVXNorrin8WVX-LGR4-Norrin
7.14Single8WVYNorrin8WVY-LGR4-Norrin
7.14Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
7.14Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
7.14Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
7.14Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
7.14Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
7.14Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
7.14Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
7.14Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
7.14Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
7.14Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.14Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.14Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.14Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.14Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.14Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.14Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.14Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.14Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.14Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.14Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
7.14Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
7.14Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
7.14Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
7.14Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
7.14Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
7.14Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
7.14Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
6.90Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
6.90Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
6.90Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
6.90Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
6.90Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
6.67Single6HLOAprepitant6HLO-NK1-Aprepitant
6.67Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
6.67Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
6.67Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
6.67Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
6.67Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
6.67Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
6.67Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
6.67Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
6.67Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.67Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.67Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
6.67Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
6.25Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
6.25Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
6.25Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
6.25Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
6.25Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
6.25Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
5.88Single5MZPCaffeine5MZP-A2A-Caffeine-Na
5.88Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
5.88Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
5.88Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
5.88Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
5.88Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
5.88Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
5.88Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
5.88Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
5.88Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single5L7DCholesterol5L7D-SMO-Cholesterol
5.56Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
5.56Single7WC4Serotonin7WC4-5-HT2A-Serotonin
5.56Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
5.56Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.26Single3OE8IT1t3OE8-CXCR4-IT1t
5.26Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
5.26Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
5.26Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
5.26Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.26Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
5.26Consensussensory_onOrthosteric Ligandopsins_on
5.00Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
5.00Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
5.00Single3UZAGTPL92363UZA-A2A-GTPL9236
5.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
5.00Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
5.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
5.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
5.00Single7WC5Psilocin7WC5-5-HT2A-Psilocin
5.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.00Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
5.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
5.00Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.00Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.00Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
5.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.00Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.00Consensusgi_sensoryOrthosteric Ligandgi_opsins
5.00Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.00Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
5.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
5.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
4.76Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
4.76Single3PBLEticlopride3PBL-D3-Eticlopride
4.76Single5NDZAZ3451; Na5NDZ-PAR2-AZ3451; Na
4.76Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
4.76Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
4.76Single6HLLCP999946HLL-NK1-CP99994
4.76Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
4.76Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
4.76Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
4.76Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
4.76Single6TP4ACT-4622066TP4-OX1-ACT-462206
4.76Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
4.76Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
4.76Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
4.76Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
4.76Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
4.76Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
4.76Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
4.76Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.76Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
4.76Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.76Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.76Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
4.76Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
4.76Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
4.76Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
4.76Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
4.76Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
4.76Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
4.76Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
4.55Single4S0VSuvorexant4S0V-OX2-Suvorexant
4.55Single5WS3EMPA5WS3-OX2-EMPA
4.55Single6B73MP11046B73-κ-MP1104
4.55Single6DS0Ly2660976DS0-5-HT2B-Ly266097
4.55Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
4.55Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
4.55Single6TODEMPA6TOD-OX1-EMPA-Na
4.55Single6TPJSuvorexant6TPJ-OX2-Suvorexant
4.55Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
4.55Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
4.55Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
4.55Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
4.55Single7XRRLemborexant7XRR-OX2-Lemborexant
4.55Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
4.55Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
4.55Single8G94CD698G94-S1P1-CD69-Gi1/β1/γ2
4.55Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.55Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
4.55Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
4.55Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
4.55Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
4.55Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
4.55Single8IWESpermidine8IWE-TA9-Spermidine
4.55Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
4.55Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
4.55Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
4.55Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
4.55Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.55Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.55Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.55Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
4.55Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8Y0HVUF114188Y0H-CXCR3-VUF11418
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
4.55Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.55Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
4.55Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
4.55Consensusalpha2_offOrthosteric Ligandalpha2c_off
4.55Consensusangiotensin_offOrthosteric Ligandat1_off
4.55Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
4.55Consensusorexin_offOrthosteric Ligandox2_off ox1_off
4.55Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
4.55Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
4.55Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
4.55Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
4.35Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
4.35Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
4.35Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
4.35Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
4.35Single4ZJCSB-6740424ZJC-OX1-SB-674042
4.35Single6A94Zotepine6A94-5-HT2A-Zotepine
4.35Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
4.35Single6IQLL7458706IQL-D4-L745870
4.35Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
4.35Single6PS0S-Carazolol6PS0-β2-S-Carazolol
4.35Single6PS4ICI118-5516PS4-β2-ICI118-551
4.35Single6PS5S-Propranolol6PS5-β2-S-Propranolol
4.35Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
4.35Single6TP3Nemorexant6TP3-OX1-Nemorexant
4.35Single6TPGEMPA6TPG-OX2-EMPA
4.35Single6TPKRetosiban6TPK-OT-Retosiban
4.35Single6TPNHTL66416TPN-OX2-HTL6641
4.35Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
4.35Single6ZG9GSK10347026ZG9-M1-GSK1034702
4.35Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
4.35Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
4.35Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
4.35Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
4.35Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
4.35Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.35Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.35Single7VODCariprazine7VOD-5-HT2A-Cariprazine
4.35Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
4.35Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.35Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.35Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
4.35Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
4.35Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
4.35Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
4.35Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
4.35Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
4.35Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
4.35Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
4.35Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
4.35Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
4.35Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.35Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.35Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.35Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.35Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
4.35Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
4.35Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
4.35Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.35Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
4.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9BJKNaloxone9BJK-μ-Naloxone-NAM
4.35Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
4.35Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
4.35Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
4.35Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
4.35Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
4.35Consensusopsins_offOrthosteric Ligandrhodopsin_off
4.35Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
4.35Consensussensory_offOrthosteric Ligandopsins_off
4.35Consensusvasop-oxy_offOrthosteric Ligandot_off
4.17Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
4.17Single2Y01Dobutamine2Y01-β1-Dobutamine
4.17Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
4.17Single3NY8ICI118-5513NY8-β2-ICI118-551
4.17Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
4.17Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
4.17Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
4.17Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
4.17Single4EJ4Naltrindole4EJ4-δ-Naltrindole
4.17Single4GBRS-Carazolol4GBR-β2-S-Carazolol
4.17Single4QKX35V4QKX-β2-35V
4.17Single5DHGC-355DHG-NOP-C-35
4.17Single6GPSMK08126GPS-CCR2-MK0812
4.17Single6H7MSalbutamol6H7M-β1-Salbutamol
4.17Single6IIVDaltroban6IIV-TP-Daltroban
4.17Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
4.17Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
4.17Single6TOTLemborexant6TOT-OX1-Lemborexant
4.17Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
4.17Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
4.17Single7BU7BI1671077BU7-β1-BI167107
4.17Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
4.17Single7F83PF-051904577F83-Ghrelin-PF-05190457
4.17Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
4.17Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
4.17Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
4.17Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
4.17Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
4.17Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
4.17Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
4.17Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
4.17Single7WC7Lisuride7WC7-5-HT2A-Lisuride
4.17Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
4.17Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
4.17Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
4.17Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
4.17Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
4.17Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
4.17Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
4.17Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
4.17Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
4.17Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
4.17Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
4.17Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
4.17Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
4.17Single8JJOAlprenolol8JJO-β2-Alprenolol
4.17Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
4.17Single8JXRLSD8JXR-D1-LSD
4.17Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
4.17Single8T1WCVN4248T1W-GPR6-CVN424
4.17Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.17Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
4.17Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
4.17Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
4.17Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
4.17Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
4.17Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
4.17Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
4.17Consensus5ht5_onOrthosteric Ligand5ht5a_on
4.17Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
4.17Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
4.17Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
4.17Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
4.17Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
4.17Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
4.17Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
4.17Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
4.17Consensusblt_onOrthosteric Ligandblt1_on
4.17Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
4.17Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
4.17Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
4.17Consensusdopamine_offOrthosteric Ligandd2_off d3_off
4.17Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
4.17Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
4.17Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
4.17Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
4.17Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
4.17Consensusleukotriene_onOrthosteric Ligandblt_on
4.17Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
4.00Single2RH1S-Carazolol2RH1-β2-S-Carazolol
4.00Single2Y00Dobutamine2Y00-β1-Dobutamine
4.00Single2YCWS-Carazolol2YCW-β1-S-Carazolol
4.00Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
4.00Single5D6LS-Carazolol5D6L-β2-S-Carazolol
4.00Single5JQHS-Carazolol5JQH-β2-S-Carazolol
4.00Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
4.00Single5TVNLSD5TVN-5-HT2B-LSD
4.00Single5WIUNemonapride5WIU-D4-Nemonapride
4.00Single5WIVNemonapride5WIV-D4-Nemonapride-Na
4.00Single5WQCEMPA5WQC-OX2-EMPA
4.00Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
4.00Single5XPRBosentan5XPR-ETB-Bosentan
4.00Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
4.00Single6E67BI1671076E67-β2-BI167107-Gs (fused)
4.00Single6GPXMK08126GPX-CCR2-MK0812
4.00Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
4.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
4.00Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
4.00Single6PS6Timolol6PS6-β2-Timolol
4.00Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
4.00Single6TP6Filorexant6TP6-OX1-Filorexant
4.00Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
4.00Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
4.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
4.00Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
4.00Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
4.00Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
4.00Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
4.00Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
4.00Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
4.00Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
4.00Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.00Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
4.00Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
4.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
4.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
4.00Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
4.00Single8ZMFA1L108ZMF-5-HT2C-A1L10
4.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.00Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
4.00Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
4.00Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
4.00Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
4.00Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
4.00Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
4.00Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
4.00Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
4.00Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
4.00Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
4.00Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
4.00Consensusamine_offonOrthosteric Ligandamine_off amine_on
4.00Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
4.00Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
4.00Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
4.00Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
4.00Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
4.00Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
3.85Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
3.85Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
3.85Single4DJHJDTic4DJH-κ-JDTic
3.85Single5D5AS-Carazolol5D5A-β2-S-Carazolol
3.85Single5D5BS-Carazolol5D5B-β2-S-Carazolol
3.85Single5V54Methiothepin5V54-5-HT1B-Methiothepin
3.85Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
3.85Single6E59L-7607356E59-NK1-L-760735
3.85Single6TQ7SB-3348676TQ7-OX1-SB-334867
3.85Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
3.85Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
3.85Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
3.85Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
3.85Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
3.85Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
3.85Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
3.85Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
3.85Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
3.85Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
3.85Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
3.85Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
3.85Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
3.85Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
3.85Single8XVLZibotentan8XVL-ETA-Zibotentan
3.85Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
3.85Single9BJKNAM9BJK-μ-Naloxone-NAM
3.85Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
3.85Consensus5ht1_offOrthosteric Ligand5ht1b_off
3.85Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
3.85Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
3.85Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
3.85Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
3.85Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
3.85Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
3.85Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
3.85Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
3.85Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
3.85Consensustachykinin_offOrthosteric Ligandnk1_off
3.70Single3D4STimolol3D4S-β2-Timolol
3.70Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
3.70Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
3.70Single6CM4Risperidone6CM4-D2-Risperidone
3.70Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
3.70Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
3.70Single6IIURamatroban6IIU-TP-Ramatroban
3.70Single6ZG4HTL00099366ZG4-M1-HTL0009936
3.70Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
3.70Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
3.70Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
3.70Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
3.70Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
3.70Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
3.70Consensusalpha1_offOrthosteric Ligandalpha1a_off
3.70Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
3.70Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
3.57Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
3.57Single5X93K-87945X93-ETB-K-8794
3.57Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
3.57Single6H7LDobutamine6H7L-β1-Dobutamine
3.57Single6K1QIRL25006K1Q-ETB-IRL2500
3.57Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
3.57Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
3.57Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
3.57Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
3.57Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
3.57Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
3.57Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
3.57Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
3.57Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
3.57Consensusendothelin_offOrthosteric Ligandetb_off
3.57Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
3.57Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
3.57Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
3.57Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
3.45Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
3.45Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
3.33Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
3.33Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
3.23Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
3.23Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
3.12Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
3.12Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
3.03Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.78Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1 Node2 LinkStrength Comm IsNode1Hub? IsNode2Hub? Node1Cons Node2Cons Node1Shell Node2Shell
K:K:D3 R:R:S368 7.36 0 Yes No 9 8 2 1
K:K:L4 K:K:L8 6.92 0 No No 9 9 1 2
K:K:L4 W:W:?1 8.51 0 No Yes 9 0 1 0
K:K:E5 R:R:H102 4.92 0 No No 9 8 1 2
K:K:E5 W:W:?1 11.77 0 No Yes 9 0 1 0
K:K:L8 R:R:R166 3.64 0 No No 9 9 2 1
R:R:F371 R:R:T84 3.89 0 Yes No 8 9 1 2
R:R:F371 R:R:T87 3.89 0 Yes No 8 7 1 2
R:R:L105 R:R:L162 4.15 16 No No 8 9 1 1
R:R:L105 R:R:Y364 10.55 16 No No 8 9 1 2
R:R:L105 W:W:?1 6.62 16 No Yes 8 0 1 0
R:R:L108 R:R:V159 4.47 16 Yes No 9 8 2 1
R:R:L108 R:R:Y364 3.52 16 Yes No 9 9 2 2
R:R:I252 R:R:V159 4.61 0 No No 8 8 2 1
R:R:V159 W:W:?1 4.07 0 No Yes 8 0 1 0
R:R:L162 W:W:?1 9.46 16 No Yes 9 0 1 0
R:R:R166 W:W:?1 27.39 0 No Yes 9 0 1 0
R:R:I252 R:R:N256 4.25 0 No No 8 9 2 2
R:R:L305 R:R:N256 5.49 0 No No 8 9 1 2
R:R:V304 R:R:V367 8.02 0 No No 8 7 2 1
R:R:L305 W:W:?1 4.73 0 No Yes 8 0 1 0
R:R:V308 W:W:?1 19.34 0 No Yes 8 0 1 0
R:R:V367 W:W:?1 5.09 0 No Yes 7 0 1 0
R:R:S368 W:W:?1 5.13 0 No Yes 8 0 1 0
R:R:F371 R:R:F375 5.36 0 Yes Yes 8 7 1 2
R:R:F371 W:W:?1 5.83 0 Yes Yes 8 0 1 0
K:K:L4 R:R:G301 3.42 0 No No 9 8 1 2

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
71.43Single8JPBPubChem 118610427; GDP; Mg8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
69.23Single8JPFPubChem 1186104278JPF-NTS1-Neurotensin-PubChem 118610427
31.58Single5LWEVercirnon5LWE-CCR9-Vercirnon
27.27Single8FN0PubChem 1186104278FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
25.00Single8JR9PCO3718JR9-PTH1-PCO371-chim(NtGi1-Gs)/β1/γ2
25.00Single8PJKt7m8PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
21.05Single6LFLPubChem 1534669966LFL-CXCR2-PubChem 153466996
21.05Single8GW8KHF8GW8-PTH1-KHF-Gs/β1/γ2
19.05Single8TB7PubChem 1685102188TB7-GPR61-PubChem 168510218
18.75Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
15.79Single6QZHHY-133073; Na6QZH-CCR7-HY-133073; Na
15.38Single4PXFOctyl-Beta-D-Glucopyranoside4PXF-Rhodopsin-Octyl-β-D-Glucopyranoside-Arrestin1 Finger Loop
13.33Single8PKMt7m8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
12.50Single8XQPAristolochic acid A8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
11.76Single5VEXNNC06405VEX-GLP-1-NNC0640
11.76Single6KK7PubChem 681786306KK7-GLP-1-PubChem 68178630
11.11Single4K5YCP-3763954K5Y-CRF1-CP-376395
11.11Single5VEWPF-063722225VEW-GLP-1-PF-06372222
11.11Single6KJVPubChem 681786306KJV-GLP-1-PubChem 68178630
11.11Single6KK1PubChem 681786306KK1-GLP-1-PubChem 68178630
11.11Single8XQRFlufenamic acid8XQR-TAS2R14-Flufenamic acid-Gt3/β1/γ1
11.11Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
10.53Single5X7DPubChem 1293189635X7D-β2-S-Carazolol-PubChem 129318963
10.53Single5XEZNNC06405XEZ-Glucagon-NNC0640
10.53Single8XQOAristolochic acid A8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
10.53Single8XQSFlufenamic acid8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
10.00Single4Z9GCP-3763954Z9G-CRF1-CP-376395
10.00Single5XF1NNC06405XF1-Glucagon-NNC0640
10.00Single8GTIBMK-C2058GTI-CRF1-BMK-C205
10.00Single8XQLAristolochic acid A8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
9.52Single8GTGBMK-I1528GTG-CRF1-BMK-I152
9.09Single8J20AR4206268J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
8.70Single8GTMBMK-C2038GTM-CRF1-BMK-C203
8.33Single6LN2PubChem 681786306LN2-GLP-1-PubChem 68178630
5.88Single8Y69Cholesterol8Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
5.56Single8Y69Cholesterol8Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
5.26Single7EJX(1R;2R)-2-PCCA7EJX-GPR88-(1R;2R)-2-PCCA-Gi1/β1/γ2
5.26Single8XQNAristolochic acid A8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
5.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
4.17Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
3.85Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
3.12Single3VG9Antibody3VG9-A2A-ZM-241385-Antibody
2.86Single3VGAAntibody3VGA-A2A-ZM-241385-Antibody

PDB Summary
PDB 8JPC
Class A
SubFamily Peptide
Type Neurotensin
SubType NTS1
Species Homo Sapiens
Ligand Neurotensin-(8-13)
Other Ligand(s) PubChem 118610427; GDP; Mg
Protein Partners Gq; GRK2
PDB Resolution 3.07
Date 2023-08-09
D.O.I. 10.1038/s41586-023-06395-9
Net Summary
Imin 3.44
Number of Linked Nodes 1204
Number of Links 1435
Number of Hubs 227
Number of Links mediated by Hubs 821
Number of Communities 31
Number of Nodes involved in Communities 289
Number of Links involved in Communities 420
Path Summary
Number Of Nodes in MetaPath 94
Number Of Links MetaPath 93
Number of Shortest Paths 4539327
Length Of Smallest Path 3
Average Path Length 38.3681
Length of Longest Path 74
Minimum Path Strength 1.225
Average Path Strength 7.39046
Maximum Path Strength 25.295
Minimum Path Correlation 0.7
Average Path Correlation 0.997889
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.63158
Average % Of Corr. Nodes 57.5223
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 52.5769
Maximum Path Hubs % 100
AnnotationTypeLinks
Gene OntologyMolecular Function
Gene OntologyBiological Process
Gene OntologyCellular Component
SCOP2Domain Identifier• G protein-coupled receptor-like   • Protein kinase-like (PK-like)   • PH domain-like   • Regulator of G-protein signaling, RGS
SCOP2Family Identifier• G protein-coupled receptor-like   • Protein kinase-like (PK-like)   • PH domain-like   • Regulator of G-protein signaling, RGS
Membrane Protein Annotations-• Orientations of Proteins in Membranes database (OPM)   • Protein Data Bank of Transmembrane Proteins (PDBTM)   • MemProtMD


Details about the values in these tables can be found in the corresponding documentation page .
CodeALF
PDB ResiduesI:I:?2
Environment DetailsOpen EMBL-EBI Page
CodeALF
NameTetrafluoroaluminate Ion
Synonyms
  • tetrafluoroaluminate(1−)
  • Tetrafluoroaluminate Ion
  • Tetrafluoroaluminate anion
Identifier
FormulaAl F4
Molecular Weight102.975
SMILES
PubChem91866986
Formal Charge-1
Total Atoms5
Total Chiral Atoms0
Total Bonds4
Total Aromatic Bonds0

CodeMG
PDB ResiduesI:I:?1
Environment DetailsOpen EMBL-EBI Page
CodeMG
NameMAGNESIUM ION
Synonyms
Identifier
FormulaMg
Molecular Weight24.305
SMILES
PubChem
Formal Charge2
Total Atoms1
Total Chiral Atoms0
Total Bonds0
Total Aromatic Bonds0

CodeSTU
PDB ResiduesK:K:?701
Environment DetailsOpen EMBL-EBI Page
CodeSTU
NameStaurosporine
SynonymsStaurosporine
Identifier
FormulaC28 H26 N4 O3
Molecular Weight466.531
SMILES
PubChem44259
Formal Charge0
Total Atoms61
Total Chiral Atoms4
Total Bonds68
Total Aromatic Bonds24

CodeGDP
PDB ResiduesO:O:?1
Environment DetailsOpen EMBL-EBI Page
CodeGDP
NameGuanosine-5'-Diphosphate
SynonymsGuanosine-5'-Diphosphate
Identifier
FormulaC10 H15 N5 O11 P2
Molecular Weight443.201
SMILES
PubChem135398619
Formal Charge0
Total Atoms43
Total Chiral Atoms4
Total Bonds45
Total Aromatic Bonds5

CodeSRW
PDB ResiduesW:W:?1
Environment DetailsOpen EMBL-EBI Page
CodeSRW
Name2-[{2-(1-fluorocyclopropyl)-4-[4-(2-methoxyphenyl)piperidin-1-yl]quinazolin-6-yl}(methyl)amino]ethan-1-ol
Synonyms
Identifier
FormulaC26 H31 F N4 O2
Molecular Weight450.548
SMILES
PubChem118610427
Formal Charge0
Total Atoms64
Total Chiral Atoms0
Total Bonds68
Total Aromatic Bonds17

PDBsumOpen PDBsum Page
ChainA
ProteinG Protein α Sub unit
UniProtP50148
Sequence
>8JPC_Chain_A
RELKLLLLG TGESGKSTF IKQMRIIHG SGYSDEDKR GFTKLVYQN 
IFTAMQAMI RAMDTLKIP YKYEHNKAH AQLVREVDV EKVSAFENP 
YVDAIKSLW NDPGIQECY DRRREYQLS DSTKYYLND LDRVADPAY 
LPTQQDVLR VRVPTTGII EYPFDLQSV IFRMVDVGG QRSERRKWI 
HCFENVTSI MFLVALSEY DQVLVESDN ENRMEESKA LFRTIITYP 
WFQNSSVIL FLNKKDLLE EKIMYSHLV DYFPEYDGP QRDAQAARE 
FILKMFVDL NPDSDKIIY SHFTCATDT ENIRFVFAA VKDTILQLN 
LK


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainK
ProteinKinase
UniProtP21146
Sequence
>8JPC_Chain_K
ADLEAVLAD VSYLMAMEK SKATPAARA SKKILLPEP SIRSVMQKY 
LEDRGEVTF EKIFSQKLG YLLFRDFCL KHLEEAKPL VEFYEEIKK 
YEKLETEEE RLVCSREIF DTYIMKELL ACSHPFSKS AIEHVQGHL 
VKKQVPPDL FQPYIEEIC QNLRGDVFQ KFIESDKFT RFCQWKNVE 
LNIHLTMND FSVHRIIGR GGFGEVYGC RKADTGKMY AMKCLDKKR 
IKMKQGETL ALNERIMLS LVSTGDCPF IVCMSYAFH TPDKLSFIL 
DLMNGGDLH YHLSQHGVF SEPDMIFYA AEIILGLEH MHNRFVVYR 
DLKPANILL DEHGHVRIS DLGLACDFS KKKPHASVG THGYMAPEV 
LQKGVAYDS SADWFSLGC MLFKLLRGH SPFRQHKTK DKHEIDRMT 
LTMAVELPD SFSPELRSL LEGLLQRDV NRRLGCLGR GAQEVKESP 
FFRDLDWQM VFLQKYPPP LIPPRGEVN AADAFDIGS FDEEDTKGI 
KLLDSDQEL YRNFPLTIS ERWQQEVAE TVFDTINAE TDRLEARKK 
TKNKQLGHE EDYALGKDC IMHGYMSKM GNPFLTQWQ RRYFYLFPN 
RLEWRGEGE APQSLLTME EIQSVEETQ IKERKCLLL KIRGGKQFV 
LQCDSDPEL VQWKKELRD AYREAQQLV Q


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainR
ProteinReceptor
UniProtP30989
Sequence
>8JPC_Chain_R
SELDVNTDI YSKVLVTAV YLALFVVGT VGNTVTAFT LTVHYHLGS 
LALSDLLTL LLAMPVELY NFIWVHHPW AFGDAGCRG YYFLRDACT 
YATALNVAS LSVERYLAI CHPFKAKTL MSRSRTKKF ISAIWLASA 
LLAVPMLFT MGEQNRSAD GQHAGGLVC TPTIHTATV KVVIQVNTF 
MSFIFPMVV ISVLNTIIA NKLTVMVRQ AAEPGRVQA LRHGVRVLR 
AVVIAFVVC WLPYHVRRL MFCYISDEQ WTPFLYDFY HYFYMVTNA 
LFYVSSTIN PILYNLVSA NFRHIFLAT


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  




This receptor, from the same or other species and bound to the same or other ligands, is also present in the following networks:
Show PDB Class SubFamily Type SubType Species Orthosteric Ligand Other Ligand(s) Protein Partners Resolution Date DOI
8JPFAPeptideNeurotensinNTS1Homo sapiensNeurotensinPubChem 118610427-3.022023-08-0910.1038/s41586-023-06395-9
8JPC (No Gprot) APeptideNeurotensinNTS1Homo sapiensNeurotensin-(8-13)PubChem 118610427; GDP; Mg3.072023-08-0910.1038/s41586-023-06395-9
8JPBAPeptideNeurotensinNTS1Homo sapiensNeurotensin-(8-13)PubChem 118610427; GDP; MgGq; GRK23.072023-08-0910.1038/s41586-023-06395-9
8JPB (No Gprot) APeptideNeurotensinNTS1Homo sapiensNeurotensin-(8-13)PubChem 118610427; GDP; Mg3.072023-08-0910.1038/s41586-023-06395-9
8FN1APeptideNeurotensinNTS1Rattus norvegicusNeurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ22.882023-03-2910.1021/acs.biochem.3c00029
8FN1 (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin/Neuromedin-N-2.882023-03-2910.1021/acs.biochem.3c00029
8FN0APeptideNeurotensinNTS1Rattus norvegicusNeurotensin/Neuromedin-NPubChem 118610427chim(NtGi1-Go)/β1/γ22.892023-03-2910.1021/acs.biochem.3c00029
8FN0 (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin/Neuromedin-NPubChem 1186104272.892023-03-2910.1021/acs.biochem.3c00029
8FMZAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ22.592023-03-2910.1021/acs.biochem.3c00029
8FMZ (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin/Neuromedin-N-2.592023-03-2910.1021/acs.biochem.3c00029
7UL2APeptideNeurotensinNTS1Homo sapiensSR48692Na-2.42022-06-2910.1038/s41594-022-00859-8
6ZINAPeptideNeurotensinNTS1Rattus norvegicusSR48692--2.642021-02-1010.1126/sciadv.abe5504
6ZA8APeptideNeurotensinNTS1Rattus norvegicusRTI-3a--2.722021-02-1010.1126/sciadv.abe5504
6Z8NAPeptideNeurotensinNTS1Rattus norvegicusSRI-9829--2.82021-02-1010.1126/sciadv.abe5504
6Z66APeptideNeurotensinNTS1Rattus norvegicus---3.192021-02-1010.1126/sciadv.abe5504
6Z4VAPeptideNeurotensinNTS1Rattus norvegicusNTS8-13--2.62021-02-1010.1126/sciadv.abe5504
6Z4SAPeptideNeurotensinNTS1Rattus norvegicusSR48692--2.712021-02-1010.1126/sciadv.abe5504
6Z4QAPeptideNeurotensinNTS1Rattus norvegicusSR142948A--2.922021-02-1010.1126/sciadv.abe5504
6YVRAPeptideNeurotensinNTS1Rattus norvegicusNTS8-13--2.462021-02-1010.1126/sciadv.abe5504
7L0SAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin-Gi1/β1/γ14.52021-01-0610.1038/s41594-020-00554-6
7L0S (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin-4.52021-01-0610.1038/s41594-020-00554-6
7L0RAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin-Gi1/β1/γ14.22021-01-0610.1038/s41594-020-00554-6
7L0R (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin-4.22021-01-0610.1038/s41594-020-00554-6
7L0QAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin-Gi1/β1/γ14.32021-01-0610.1038/s41594-020-00554-6
7L0Q (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin-4.32021-01-0610.1038/s41594-020-00554-6
7L0PAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin-Gi1/β1/γ14.12021-01-0610.1038/s41594-020-00554-6
7L0P (No Gprot) APeptideNeurotensinNTS1Rattus norvegicusNeurotensin-4.12021-01-0610.1038/s41594-020-00554-6
6UP7APeptideNeurotensinNTS1Homo sapiensNeurotensin-Arrestin24.22020-02-2610.1038/s41586-020-1953-1
6PWCAPeptideNeurotensinNTS1Homo sapiensNeurotensin-Arrestin24.92019-12-0410.1038/s41422-019-0256-2
6OSAAPeptideNeurotensinNTS1Homo sapiensJMV449-Gi1/β1/γ232019-07-1010.1038/s41586-019-1337-6
6OSA (No Gprot) APeptideNeurotensinNTS1Homo sapiensJMV449-32019-07-1010.1038/s41586-019-1337-6
6OS9APeptideNeurotensinNTS1Homo sapiensJMV449-Gi1/β1/γ232019-07-1010.1038/s41586-019-1337-6
6OS9 (No Gprot) APeptideNeurotensinNTS1Homo sapiensJMV449-32019-07-1010.1038/s41586-019-1337-6
5T04APeptideNeurotensinNTS1Rattus norvegicusNeurotensin--3.32016-12-2110.1038/srep38564
4XESAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin--2.62015-07-2910.1038/ncomms8895
4XEEAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin--2.92015-07-2910.1038/ncomms8895
4BWBAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin--3.572014-01-2910.1073/pnas.1317903111
4BV0APeptideNeurotensinNTS1Rattus norvegicusNeurotensin--3.12014-01-2910.1073/pnas.1317903111
4BUOAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin--2.752014-01-2910.1073/pnas.1317903111
3ZEVAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin--32014-01-2910.1073/pnas.1317903111
4GRVAPeptideNeurotensinNTS1Rattus norvegicusNeurotensin-(8-13)--2.82012-10-1710.1038/nature11558




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