Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.43 3.99583479
2G.HN.47 3.165475
3G.S2.01 3.15667419
4G.S3.03 6.34889608
5G.S3.04 8.58333417
6G.S3.06 8.01133517
7G.H2.05 8.69667418
8G.H2.06 6.05333619
9G.H2.07 8.42167419
10G.h2s4.01 7.57667519
11G.S4.02 5.17583418
12G.S4.03 4.12333467
13G.S4.04 4.43917459
14G.S4.07 7.11754178
15G.s4h3.04 7.44583408
16G.H3.01 6.52167409
17G.H3.08 7.68167408
18G.H3.09 4.81067559
19G.H3.13 8.75833656
20G.H3.17 9.72611645
21G.S5.03 5.32733569
22G.S5.04 5.53917459
23G.S5.05 6.73533569
24G.S5.06 3.66733558
25G.s5hg.01 6.82917409
26G.HG.03 4.3225406
27G.HG.15 6.041335187
28G.hgh4.05 10.57084186
29G.hgh4.20 7.26917403
30G.H4.03 4.47417404
31G.H4.10 10.87424187
32G.H4.12 3.825404
33G.H4.15 6.58083458
34G.S6.01 3.535455
35G.S6.02 7.31111668
36G.S6.05 6.24917455
37G.s6h5.05 5.08167409
38G.H5.03 6.00167469
39G.H5.08 4.33533508
40G.H5.23 7.94754114
41b.1x3 1.50833401
42b.1x4 1.978508
43b.lhb1x3 2.92583402
44b.l1x3 8.50667679
45b.b2x1 6.26667418
46b.b2x5 9.2825407
47b.l3x2 7.29917409
48b.b4x2 6.45833408
49b.b4x6 12.8573579
50b.b5x2 6.30833407
51b.b5x3 6.27679
52b.b5x7 7.59083487
53b.l5x1 5.45733588
54b.l5x5 10.4125419
55b.b6x1 4.58733519
56b.b6x5 3.86817226
57b.b7x1 6.42667404
58b.b8x4 5.33278686
59b.l9x3 7.66917419
60b.l9x6 4.74917418
61b.b10x5 6.4175409
62b.l10x1 3.47533503
63b.b11x4 5.06333419
64b.b11x6 6.81167419
65b.l11x2 7.53933519
66b.b12x6 12.745418
67b.b12x7 6.1454149
68b.l12x3 3.94145
69b.l13x3 8.31667599
70b.l13x6 8.6025419
71b.b15x2 8.16436
72b.l15x1 4.915417
73b.l15x2 6.44667499
74b.b16x6 8.75524798
75b.b17x5 7.57167437
76b.b17x7 9.51417438
77b.l17x3 9.40778639
78b.b18x3 4.77133538
79b.b18x5 7.73417435
80b.l18x1 7.359335246
81b.b19x2 7.19619736
82b.b19x4 6.11083438
83b.b20x4 9.11667438
84b.b20x6 7.00143736
85b.b20x7 3.998509
86b.l20x1 5.68833436
87b.l20x2 5.912675159
88b.b21x1 10.3308437
89b.b21x2 3.32533506
90b.b21x5 6.1725404
91b.b21x7 5.00111605
92b.l21x5 4.201335104
93b.b22x5 5.236675247
94b.l22x5 6.47067509
95b.b23x6 7.447335107
96b.l23x1 8.18333546
97b.b24x4 5.6125106
98b.b24x6 5.414174108
99b.b25x3 4.3625105
100b.l25x3 6.64417449
101b.l25x5 7.325447
102b.l25x6 11.582548
103b.l27x1 9.60444649
104b.l27x2 5.64333549
105b.b28x4 5.514174136
106b.b28x6 9.248675139
107g.h1x11 3.3575409
108g.ctx3 6.374509
109g.ctx4 3.72407
110g.ctx9 4.32167406
111Lig 6.899331520
1121x56 4.4654258
1131x61 5.36917406
1142x39 6.585834117
1152x40 3.525834208
1162x42 3.4654167
1172x50 6.2425429
1182x51 5.59417407
1192x54 6.95417428
1202x65 6.51867528
121E1x50 7.646674125
122E1.F101 6.559335124
1233x32 5.70667428
1243x33 5.62083428
1253x50 6.755119
1264x60 6.26667429
127E2.Y177 6.68627
128E2.T184 5.99933529
129E2.W185 6.17111628
130E2x51 5.84222628
131E2x52 7.46944626
1325x37 3.53867526
1335x53 3.326674285
1345x56 4.419335119
1355x59 3.172508
1366x29 5.15083405
1376x30 7.44167408
1386x48 7.87167629
1397x39 8.22583428
1407x45 6.33167429
1417x46 5.27111628
1427x47 5.12667408
1437x53 7.041674269
1448x53 1.06667405
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1G.HN.40 b.b5x2 39.88417.94667NoYes077
2G.HN.40 b.b5x3 40.00876.12NoYes779
3G.HN.47 b.b5x3 42.07412.82YesYes759
4G.HN.47 b.l1x4 47.40183.23YesNo056
5G.HN.51 b.l1x4 54.98248.46NoNo046
6G.HN.51 G.hns1.02 55.24914.12667NoNo044
7G.hns1.02 I1.K63 55.38185.77667NoNo046
8I1.K63 I2x57 55.77742.91NoNo065
9I2x53 I2x57 59.52785.74333NoNo085
103x49 I2x53 59.764510.26NoNo098
112x42 3x49 59.74773.09333YesNo1679
122x42 3x46 60.16513.29667YesNo079
132x39 3x46 72.00715.80667YesNo079
142x39 G.H5.23 66.95588.94YesYes1174
156x33 G.H5.23 70.60845.98667NoYes084
166x33 G.H5.24 70.60376.07667NoNo087
176x29 G.H5.24 1006.80333YesNo057
186x29 G.H5.21 99.81756.39333YesNo055
19G.H5.21 G.h3s5.02 99.75583.01667NoNo054
20G.h3s5.02 G.h3s5.03 99.56833.04NoNo047
21G.S4.02 G.h3s5.03 99.50493.43333YesNo087
22G.S1.05 G.S4.02 99.197612.37NoYes198
23G.S1.05 G.h2s4.01 99.247411.3667NoYes199
24G.H2.07 G.h2s4.01 72.45024.67667YesYes199
25G.H2.04 G.H2.07 71.95999.33333NoYes099
26G.H2.04 G.H3.08 71.793415.0867NoYes098
27G.H3.08 G.S4.04 71.30067.16667YesYes089
28G.H3.09 G.S4.04 35.25134.28333YesYes599
29G.H3.09 G.S6.01 29.3163.25667YesYes595
30G.S6.01 G.S6.03 27.31744.39667YesNo055
31G.H4.12 G.S6.03 27.11032.88YesNo045
32G.H4.08 G.H4.12 52.60227.54333NoYes034
33G.H4.08 G.hgh4.11 51.71445.09667NoNo035
34G.hgh4.08 G.hgh4.11 47.97624.17NoNo065
35G.H4.10 G.hgh4.08 46.626215.82YesNo076
36G.H4.10 G.HG.15 42.91372.93333YesYes1877
37G.HG.15 G.s4h3.04 40.24447.65333YesYes078
38G.hgh4.01 G.s4h3.04 37.95912.2433NoYes068
39G.hgh4.01 G.s4h3.15 37.09067.36333NoNo069
40G.s4h3.03 G.s4h3.15 36.6313.14NoNo089
41G.S4.07 G.s4h3.03 33.79123.99YesNo1788
42G.S4.07 G.s5hg.01 31.506610.6YesYes089
43G.S5.07 G.s5hg.01 29.19617.45667NoYes099
44G.H1.04 G.S5.07 27.32884.72NoNo079
45G.H1.04 G.H5.03 24.48752.83333NoYes079
46G.H5.03 G.S5.05 15.388711.2767YesYes699
47G.S4.04 G.S5.04 35.44673.25YesYes599
48G.S5.04 G.S5.06 34.15134.15333YesYes598
49G.S5.06 G.S6.05 30.41244.05667YesYes585
50G.H4.12 G.S6.05 27.34673.56667YesYes045
51G.h2s4.01 b.l7x2 50.64014.46333YesNo199
52b.b6x1 b.l7x2 51.19792.83YesNo199
53b.b6x1 b.l9x6 37.22513.59YesYes198
54b.l11x1 b.l9x6 34.25825.31NoYes198
55b.b11x6 b.l11x1 34.17873.71YesNo199
56b.b26x1 b.l27x1 15.47614.94NoYes099
57b.b26x1 b.b2x1 15.74585.93667NoYes098
58b.b2x1 b.b6x1 16.84547.58333YesYes189
59G.S5.03 G.S5.05 10.10615.44YesYes699
606x32 G.H5.24 29.886414.4567NoNo077
616x32 8x47 29.90956.97667NoNo079
626x36 8x47 31.115622.9767NoNo089
636x36 6x40 31.20975.49NoNo088
646x40 7x53 30.80712.0867NoYes2689
653x46 7x53 46.19092.79NoYes099
66b.b11x6 b.l9x3 31.313910.2267YesYes199
67b.b11x4 b.l9x3 26.14163.65333YesYes199
68b.b10x3 b.b11x4 24.48425.07NoYes089
69b.b10x3 b.b6x2 24.22735.63333NoNo088
70b.b10x2 b.b6x2 23.972.81667NoNo068
71b.b10x2 b.b10x4 22.41756.96NoNo066
72b.b10x4 b.b14x5 19.00224.85667NoNo065
73b.b14x5 b.b15x1 14.43053.24667NoNo059
74b.b15x1 b.b16x6 13.59138.68333NoYes998
75b.b5x2 b.l4x3 38.37958.77333YesNo076
76b.b4x7 b.l4x3 38.210311.08NoNo086
77b.b4x7 b.l2x5 38.040613.1033NoNo085
78b.l2x5 b.l4x2 37.870616.12NoNo054
79b.l4x1 b.l4x2 37.70016.36NoNo054
80b.b2x5 b.l4x1 37.52914.94YesNo075
81b.b2x5 b.l26x1 37.01399.7YesNo077
82b.l26x1 b.l26x3 36.6326.26333NoNo2177
83b.l26x3 b.l26x5 36.49510.1633NoNo075
84b.l26x5 g.ctx4 36.32126.15NoYes057
85g.ctx3 g.ctx4 34.91573.75667YesYes097
86b.l22x3 g.ctx3 31.285710.31NoYes099
87b.l22x3 b.l22x5 31.09982.64NoYes099
88b.l22x5 b.l24x2 28.45428.09667YesNo096
89b.h2x5 b.l24x2 28.26217.86NoNo056
90b.h2x1 b.h2x5 28.06963.93NoNo055
91b.b21x5 b.h2x1 27.29544.71YesNo045
92b.b21x5 b.b21x7 25.924611.5733YesYes045
93b.b21x7 b.b23x2 21.48393.51667YesNo056
94b.b22x5 b.b23x2 20.86276.49667YesNo076
95b.b22x5 b.l18x1 18.87357.5YesYes2476
96b.l18x1 b.l18x3 18.260913.6933YesNo065
97b.l18x3 b.l18x5 18.144414.98NoNo052
98b.l18x5 b.l20x2 17.93097.63667NoYes029
99b.l20x2 g.l1x5 13.38846.26YesNo1594
100g.l1x3 g.l1x5 13.20320.466667NoNo014
101g.l1x2 g.l1x3 12.98310.466667NoNo021
102b.b17x5 g.l1x2 12.76381.82667YesNo072
103b.b4x2 b.b5x8 10.84515.01667YesNo085
104b.b5x7 b.b5x8 10.41633.39YesNo075
1057x46 Lig 58.87996.03YesYes280
1067x45 7x46 67.60775.72YesYes298
1077x45 7x49 73.51435.38667YesNo099
1087x49 7x53 73.790910.3467NoYes099
1093x32 Lig 35.8288.2YesYes280
110E1.D102 E1x50 10.76832.60667NoYes045
1113x22 E1.D102 11.48294.04333NoNo014
1123x22 E2.D176 12.1973.14NoNo013
1133x26 E2.D176 12.91082.45NoNo043
1143x26 4x61 13.62413.1NoNo044
1154x61 E2.Y177 14.32463.63NoYes247
1163x32 E2x51 33.24733.73333YesYes288
117E2x51 E2x52 16.620512.38YesYes286
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
1x39Lig10.20670NoYes7010
2x54Lig17.81672YesYes8010
2x57Lig11.19672NoYes6010
2x58Lig3.053330NoYes7010
2x65Lig3.893332YesYes8010
3x32Lig8.22YesYes8010
3x35Lig4.370NoYes7010
3x36Lig3.463330NoYes7010
E2.T184Lig5.216672YesYes0010
7x35Lig3.726672NoYes6010
7x38Lig6.846670NoYes7010
7x39Lig5.792YesYes8010
7x42Lig10.722NoYes9010
7x46Lig6.032YesYes8010
2x65NT.S294.666672YesNo8012
1x362x659.250NoYes6821
1x387x3912.11330NoYes4821
1x427x392.853330NoYes8821
1x427x425.623330NoNo8921
1x432x582.910NoNo7721
2x503x3911.80672YesNo9922
2x547x423.196672YesNo8911
2x547x463.712YesYes8811
2x547x473.093332YesYes8812
2x573x287.252NoNo6612
2x573x324.673332NoYes6811
2x65E1.K964.382YesNo8012
2x65E2.T18410.40332YesYes8011
E1.K96E2.T18432NoYes0021
3x283x326.222NoYes6821
3x32E2x513.733332YesYes8812
3x366x482.810NoYes7912
E2.S182E2.T1846.932NoYes0021
E2.S182E2.W1854.942NoYes0022
E2.T184E2.W1854.446672YesYes0012
E2.W185E2x516.352YesYes0822
7x38E2.W1856.450NoYes7012
6x487x4510.54672YesYes9922
6x487x465.843332YesYes9821
6x516x557.876670NoNo8712
6x517x374.160NoNo8712
7x357x3912.14672NoYes6811
7x457x465.722YesYes9821
6x51Lig2.960NoYes8010
2x507x463.483332YesYes9821
3x397x466.842NoYes9821
2x533x352.476670NoNo8721
1x392x612.280NoNo7812

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
82.35Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
82.35Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
82.35Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
81.25Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
76.47Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
76.47Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
73.33Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
68.75Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
66.67Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
66.67Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
66.67Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
66.67Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
66.67Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
64.71Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
64.71Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
64.71Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
61.11Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
61.11Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
61.11Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
60.00Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
58.82Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
57.89Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
55.56Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
55.00Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
52.94Single6IIVDaltroban6IIV-TP-Daltroban
52.63Single6IIURamatroban6IIU-TP-Ramatroban
50.00Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
50.00Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
47.06Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
38.89Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
38.89Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
38.10Single4N4WSANT-14N4W-SMO-SANT-1
36.84Single5TGZAM65385TGZ-CB1-AM6538
36.84Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
36.84Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
36.84Single9B9ZA1AKO9B9Z-CB1-A1AKO
35.29Single9B9Y7DY9B9Y-CB1-7DY
35.00Single5CGCHTL142425CGC-mGlu5-HTL14242
35.00Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
35.00Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
35.00Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
35.00Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
35.00Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
35.00Consensusep_offOrthosteric Ligandep4_off
35.00Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
34.78Single5EE7MK08935EE7-Glucagon-MK0893
33.33Single5U09Taranabant5U09-CB1-Taranabant
33.33Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
33.33Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
33.33Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
33.33Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
33.33Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
33.33Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
33.33Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
33.33Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
33.33Single9BA0A1AKN9BA0-CB1-A1AKN
33.33Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
33.33Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
31.82Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
31.82Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
31.82Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
31.82Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
31.58Single2YDOAdenosine2YDO-A2A-Adenosine
31.58Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
31.58Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
31.58Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
31.58Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
31.58Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
31.58Single8K5CAcipimox8K5C-HCA2-Acipimox
31.58Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
31.58Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
31.25Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
31.25Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
30.43Single5CGDHTL142425CGD-mGlu5-HTL14242
30.43Single6H7LDobutamine6H7L-β1-Dobutamine
30.43Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
30.43Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
30.43Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
30.43Consensusprostanoid_offOrthosteric Ligandep_off dp_off
30.00Single2Y01Dobutamine2Y01-β1-Dobutamine
30.00Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
30.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
30.00Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
30.00Single7YXAONO-54306087YXA-S1P5-ONO-5430608
30.00Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
30.00Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
30.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
30.00Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
30.00Single8T1WCVN4248T1W-GPR6-CVN424
30.00Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
30.00Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
30.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
30.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
30.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
30.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
30.00Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
29.63Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
29.41Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
29.41Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
29.41Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
29.41Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
29.41Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
29.41Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
29.41Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
29.41Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
29.41Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
29.17Single6PT3DPI-2876PT3-δ-DPI-287
29.17Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
29.17Single7SK9CCX6627SK9-ACKR3-CCX662
29.17Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
29.17Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
28.57Single2Y00Dobutamine2Y00-β1-Dobutamine
28.57Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
28.57Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
28.57Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
28.57Single7C61Ergotamine7C61-5-HT1B-Ergotamine
28.57Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
28.57Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
28.57Single8TF5Oleic acid8TF5-GPR6-Oleic acid
28.57Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
28.57Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
28.57Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
28.57Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
28.57Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
28.57Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Consensustrace-amine_onOrthosteric Ligandta1_on
28.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
28.00Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
28.00Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
28.00Single8WDTphotoNECA8WDT-A2A-photoNECA
28.00Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
27.78Single5L7IVismodegib5L7I-SMO-Vismodegib
27.78Single6LI0C176LI0-GPR52-C17
27.78Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
27.78Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
27.78Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
27.78Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
27.78Single8K5BNiacin8K5B-HCA2-Niacin
27.78Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
27.78Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
27.78Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
27.78Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
27.78Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
27.78Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
27.78Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
27.78Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
27.27Single2YDVNECA2YDV-A2A-NECA
27.27Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
27.27Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
27.27Single4UHRCGS216804UHR-A2A-CGS21680
27.27Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
27.27Single5G53NECA5G53-A2A-NECA-Gs
27.27Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
27.27Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
27.27Single7TUYGSK682753A7TUY-GPR183-GSK682753A
27.27Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
27.27Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
27.27Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
27.27Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
27.27Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
27.27Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
27.27Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
27.27Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
27.27Single9BJKNAM9BJK-μ-Naloxone-NAM
27.27Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
27.27Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
27.27Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
27.27Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
27.27Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
26.92Single3QAKUK-4320973QAK-A2A-UK-432097
26.92Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
26.92Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
26.67Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Single6AKXA4R6AKX-CCR5-A4R
26.32Single6AKYMaraviroc6AKY-CCR5-Maraviroc
26.32Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
26.32Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
26.32Single6TODEMPA6TOD-OX1-EMPA-Na
26.32Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
26.32Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.32Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.32Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
26.32Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
26.32Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
26.32Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
26.32Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
26.32Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.32Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.32Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
26.32Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
26.32Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
26.32Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
26.32Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
26.32Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
26.32Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
26.32Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
26.32Single8IWESpermidine8IWE-TA9-Spermidine
26.32Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
26.32Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
26.32Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.32Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
26.32Single8Y0HVUF114188Y0H-CXCR3-VUF11418
26.32Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
26.32Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
26.32Consensusalpha2_offOrthosteric Ligandalpha2c_off
26.32Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
26.32Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
26.32Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
26.32Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
26.32Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.32Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.09Single4LDEBI1671074LDE-β2-BI167107
26.09Single5X33BIIL2605X33-BLT1-BIIL260
26.09Single6A93Risperidone6A93-5-HT2A-Risperidone
26.09Single6CM4Risperidone6CM4-D2-Risperidone
26.09Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
26.09Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
26.09Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
26.09Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
26.09Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
26.09Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
26.09Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
26.09Single8JJ8Formoterol8JJ8-β2-Formoterol
26.09Single8XYIVUF106618XYI-CXCR3-VUF10661
26.09Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
26.09Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
26.09Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
26.09Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
26.09Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
26.09Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
26.09Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
26.09Consensuslpl_offOrthosteric Ligands1p_off lpa_off
26.09Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
25.93Single5WF5UK-4320975WF5-A2A-UK-432097
25.93Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
25.81Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
25.81Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
25.81Consensusbradykinin_onOrthosteric Ligandbk2_on
25.81Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
25.81Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
25.00Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
25.00Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
25.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
25.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
25.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
25.00Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
25.00Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
25.00Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
25.00Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
25.00Single6FFIMMPEP6FFI-mGlu5-MMPEP
25.00Single6IBLArformoterol6IBL-β1-Arformoterol
25.00Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
25.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
25.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
25.00Single6PS4ICI118-5516PS4-β2-ICI118-551
25.00Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
25.00Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
25.00Single6TPGEMPA6TPG-OX2-EMPA
25.00Single7AROLUF58337ARO-A2A-LUF5833-Na
25.00Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
25.00Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
25.00Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
25.00Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
25.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
25.00Single7EZCUKA7EZC-A2A-UKA
25.00Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
25.00Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
25.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
25.00Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
25.00Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
25.00Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
25.00Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
25.00Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
25.00Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
25.00Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
25.00Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
25.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
25.00Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
25.00Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
25.00Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
25.00Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
25.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
25.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
25.00Single8IHKAcifran8IHK-HCA3-Acifran
25.00Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
25.00Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
25.00Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
25.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
25.00Single8K2WAMG4878K2W-CXCR3-AMG487
25.00Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
25.00Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
25.00Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
25.00Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
25.00Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Single8XVJMacitentan8XVJ-ETA-Macitentan
25.00Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
25.00Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
25.00Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
25.00Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
25.00Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
25.00Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
25.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
25.00Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
25.00Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
25.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
25.00Consensusalpha1_onOrthosteric Ligandalpha1a_on
25.00Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
25.00Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
25.00Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
25.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
25.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
25.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
25.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
25.00Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
25.00Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
25.00Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
25.00Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
25.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
25.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
25.00Consensushca_onOrthosteric Ligandhca2_on
24.14Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
24.14Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
24.14Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
24.14Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
24.14Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
24.00Single3NY9ICI118-5513NY9-β2-ICI118-551
24.00Single4UG2CGS216804UG2-A2A-CGS21680
24.00Single5WF6UK-4320975WF6-A2A-UK-432097
24.00Single5ZTYAM102575ZTY-CB2-AM10257
24.00Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
24.00Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
24.00Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
24.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
24.00Single8X5YAstemizole8X5Y-H1-Astemizole
24.00Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
24.00Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
24.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
23.81Single2Y04Salbutamol2Y04-β1-Salbutamol
23.81Single3NY8ICI118-5513NY8-β2-ICI118-551
23.81Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
23.81Single4EJ4Naltrindole4EJ4-δ-Naltrindole
23.81Single4GBRS-Carazolol4GBR-β2-S-Carazolol
23.81Single4QKX35V4QKX-β2-35V
23.81Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
23.81Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
23.81Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
23.81Single5UENDU1725UEN-A1-DU172
23.81Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
23.81Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
23.81Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
23.81Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
23.81Single6FFHFenobam6FFH-mGlu5-Fenobam
23.81Single6H7MSalbutamol6H7M-β1-Salbutamol
23.81Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
23.81Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
23.81Single6PS1Timolol6PS1-β2-Timolol
23.81Single6TOTLemborexant6TOT-OX1-Lemborexant
23.81Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
23.81Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
23.81Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
23.81Single7BU7BI1671077BU7-β1-BI167107
23.81Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
23.81Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
23.81Single7UL4Alvimopan7UL4-μ-Alvimopan
23.81Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
23.81Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
23.81Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
23.81Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
23.81Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
23.81Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
23.81Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
23.81Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
23.81Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
23.81Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
23.81Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
23.81Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
23.81Single8JJOAlprenolol8JJO-β2-Alprenolol
23.81Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
23.81Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
23.81Single8JXRLSD8JXR-D1-LSD
23.81Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
23.81Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
23.81Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
23.81Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
23.81Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
23.81Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
23.81Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
23.81Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
23.81Single9CHXS-Carazolol9CHX-β2-S-Carazolol
23.81Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
23.81Consensusa3_onOrthosteric Liganda3a_on
23.81Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
23.81Consensusalpha2_onOrthosteric Ligandalpha2b_on
23.81Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
23.81Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
23.81Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
23.81Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
23.81Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
23.81Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
23.81Consensusdopamine_offOrthosteric Ligandd2_off d3_off
23.81Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
23.81Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
23.81Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
23.81Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
23.81Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
23.81Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
23.81Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
23.81Consensushca_on_gpOrthosteric Ligandhca2_on_gp
23.81Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
23.81Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
23.53Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
23.53Single9CHUNoradrenaline9CHU-β2-Noradrenaline
23.33Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
23.33Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
23.08Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
23.08Single4IARErgotamine4IAR-5-HT1B-Ergotamine
23.08Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
23.08Single7QA8Peptide7QA8-STE2-Peptide
23.08Single7QA8Peptide7QA8-STE2-Peptide
23.08Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
23.08Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
23.08Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
23.08Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
23.08Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
23.08Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
23.08Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.73Single2RH1S-Carazolol2RH1-β2-S-Carazolol
22.73Single2Y03Isoprenaline2Y03-β1-Isoprenaline
22.73Single2YCWS-Carazolol2YCW-β1-S-Carazolol
22.73Single4JKVTaladegib4JKV-SMO-Taladegib
22.73Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
22.73Single5C1MBU725C1M-μ-BU72
22.73Single5D6LS-Carazolol5D6L-β2-S-Carazolol
22.73Single5JQHS-Carazolol5JQH-β2-S-Carazolol
22.73Single5N2RPSB-365N2R-A2A-PSB-36-Na
22.73Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
22.73Single5WQCEMPA5WQC-OX2-EMPA
22.73Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
22.73Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
22.73Single6D26Fevipiprant6D26-DP2-Fevipiprant
22.73Single6E67BI1671076E67-β2-BI167107-Gs (fused)
22.73Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
22.73Single6GPXMK08126GPX-CCR2-MK0812
22.73Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
22.73Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
22.73Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
22.73Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
22.73Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
22.73Single6PS6Timolol6PS6-β2-Timolol
22.73Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
22.73Single6TP6Filorexant6TP6-OX1-Filorexant
22.73Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
22.73Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
22.73Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
22.73Single7WC6LSD7WC6-5-HT2A-LSD
22.73Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
22.73Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
22.73Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
22.73Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
22.73Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
22.73Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
22.73Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
22.73Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
22.73Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
22.73Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
22.73Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
22.73Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
22.73Single8S4DCMF-0198S4D-Apelin-CMF-019
22.73Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
22.73Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
22.73Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
22.73Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
22.73Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
22.73Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
22.73Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
22.73Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
22.73Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
22.73Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
22.73Consensusa3_on_gpOrthosteric Liganda3a_on_gp
22.73Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
22.73Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
22.73Consensusadenosine_offOrthosteric Liganda1_off a2_off
22.73Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
22.73Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
22.73Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
22.73Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
22.73Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
22.73Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
22.73Consensusamine_offonOrthosteric Ligandamine_off amine_on
22.73Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
22.73Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
22.73Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
22.73Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
22.73Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
22.73Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
22.73Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
22.73Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
22.73Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.73Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
22.73Consensusdp_offOrthosteric Liganddp2_off
22.73Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
22.73Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
22.73Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
22.73Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
22.73Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
22.73Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
22.73Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.58Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
22.22Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
22.22Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
22.22Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
22.22Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
22.22Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
22.22Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
22.22Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
22.22Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
22.22Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
22.22Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
22.22Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
22.22Consensus5ht2_onOrthosteric Ligand5ht2b_on
22.22Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
21.74Single3P0GBI1671073P0G-β2-BI167107
21.74Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
21.74Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
21.74Single4U15Tiotropium4U15-M3-Tiotropium
21.74Single5D5AS-Carazolol5D5A-β2-S-Carazolol
21.74Single5D5BS-Carazolol5D5B-β2-S-Carazolol
21.74Single5V56TC1145V56-SMO-TC114
21.74Single5V57TC1145V57-SMO-TC114
21.74Single5XR8AM8415XR8-CB1-AM841
21.74Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
21.74Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
21.74Single6H7JIsoprenaline6H7J-β1-Isoprenaline
21.74Single6J21Aprepitant6J21-NK1-Aprepitant
21.74Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
21.74Single6OL9Tiotropium6OL9-M5-Tiotropium
21.74Single6TQ7SB-3348676TQ7-OX1-SB-334867
21.74Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
21.74Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
21.74Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
21.74Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
21.74Single7P2L4YI7P2L-mGlu5-4YI
21.74Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
21.74Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
21.74Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
21.74Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
21.74Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
21.74Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
21.74Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
21.74Single8E0GBU728E0G-μ-BU72
21.74Single8EA0Iperoxo8EA0-M3-Iperoxo
21.74Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
21.74Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
21.74Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
21.74Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.74Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
21.74Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
21.74Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
21.74Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
21.74Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
21.74Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
21.74Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
21.74Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
21.74Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
21.74Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
21.74Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
21.74Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
21.74Consensusa2_onOrthosteric Liganda2b_on
21.74Consensusa2_on_gpOrthosteric Liganda2b_on_gp
21.74Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
21.74Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
21.74Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
21.74Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
21.74Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
21.74Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
21.74Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
21.74Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.74Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
21.74Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
21.74Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
21.74Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
21.74Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
21.74Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
21.74Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
21.74Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
21.74Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
21.74Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
21.43Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
21.43Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
21.43Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.43Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
21.43Consensusangiotensin_onOrthosteric Ligandat1_on
21.43Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
21.43Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
21.43Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
21.43Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
21.05Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
21.05Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
21.05Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
21.05Single7SRQLSD7SRQ-5-HT2B-LSD
21.05Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
21.05Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
21.05Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
21.05Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
21.05Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.05Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
21.05Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
21.05Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
21.05Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
21.05Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
21.05Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.05Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
21.05Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
21.05Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
21.05Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
21.05Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
21.05Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
21.05Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.83Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
20.83Single3D4STimolol3D4S-β2-Timolol
20.83Single4AMIBucindolol4AMI-β1-Bucindolol
20.83Single4RWADIPP-NH24RWA-δ-DIPP-NH2
20.83Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
20.83Single5CXVTiotropium5CXV-M1-Tiotropium
20.83Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
20.83Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
20.83Single6MXTSalmeterol6MXT-β2-Salmeterol
20.83Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
20.83Single6ZG4HTL00099366ZG4-M1-HTL0009936
20.83Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
20.83Single7DFPSpiperone7DFP-D2-Spiperone
20.83Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
20.83Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.83Single7K15MKD0467K15-BLT1-MKD046-Na
20.83Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
20.83Single7YITNalfurafine7YIT-κ-Nalfurafine
20.83Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
20.83Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
20.83Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
20.83Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
20.83Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
20.83Single8JJLOlodaterol8JJL-β2-Olodaterol
20.83Single8JWY2-1188JWY-A2A-2-118
20.83Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
20.83Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
20.83Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.83Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.83Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.83Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.83Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.83Consensusalpha1_offOrthosteric Ligandalpha1a_off
20.83Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
20.83Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.83Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
20.83Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
20.83Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
20.83Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
20.83Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
20.83Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
20.83Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
20.83Consensuslpa_offOrthosteric Ligandlpa1_off
20.83Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
20.83Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
20.83Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
20.83Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
20.83Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
20.69Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
20.69Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
20.69Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
20.69Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
20.69Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
20.69Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
20.69Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
20.69Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
20.00Single3PWHZM-2413853PWH-A2A-ZM-241385
20.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
20.00Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
20.00Single4S0VSuvorexant4S0V-OX2-Suvorexant
20.00Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
20.00Single5WS3EMPA5WS3-OX2-EMPA
20.00Single5X93K-87945X93-ETB-K-8794
20.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
20.00Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
20.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
20.00Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
20.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.00Single6TPJSuvorexant6TPJ-OX2-Suvorexant
20.00Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
20.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
20.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
20.00Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
20.00Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
20.00Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
20.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
20.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
20.00Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
20.00Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
20.00Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
20.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
20.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
20.00Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
20.00Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
20.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
20.00Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
20.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
20.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
20.00Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
20.00Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
20.00Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
20.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
20.00Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
20.00Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
20.00Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
20.00Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
20.00Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
20.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
20.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Consensusangiotensin_offOrthosteric Ligandat1_off
20.00Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
20.00Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
20.00Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
20.00Consensusendothelin_offOrthosteric Ligandetb_off
20.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
20.00Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
20.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
20.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
20.00Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.00Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.00Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
20.00Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
20.00Consensusorexin_offOrthosteric Ligandox2_off ox1_off
20.00Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
20.00Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
20.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
20.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
20.00Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.35Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
19.35Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
19.35Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
19.35Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
19.35Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
19.23Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
19.23Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
19.23Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
19.23Single7XN9L-054,5227XN9-SST2-L-054,522
19.23Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
19.23Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
19.23Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
19.23Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
19.23Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
19.23Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
19.23Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
19.05Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
19.05Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
19.05Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
19.05Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
19.05Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
19.05Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
19.05Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
19.05Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
19.05Single5IUBQ274563445IUB-A2A-Q27456344-Na
19.05Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
19.05Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
19.05Single6AQFZM-2413856AQF-A2A-ZM-241385
19.05Single6KUXRS-799486KUX-α2a-RS-79948
19.05Single6PS5S-Propranolol6PS5-β2-S-Propranolol
19.05Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
19.05Single6TP3Nemorexant6TP3-OX1-Nemorexant
19.05Single6V9SGTPL114036V9S-OX1-GTPL11403
19.05Single6VI4JDTic6VI4-κ-JDTic
19.05Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
19.05Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
19.05Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
19.05Single6ZG9GSK10347026ZG9-M1-GSK1034702
19.05Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
19.05Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
19.05Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
19.05Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
19.05Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
19.05Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.05Single7T32ZM-2413857T32-A2A-ZM-241385
19.05Single7UL3Famotidine7UL3-H2-Famotidine
19.05Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
19.05Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.05Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
19.05Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
19.05Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
19.05Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
19.05Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
19.05Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
19.05Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
19.05Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
19.05Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
19.05Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
19.05Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
19.05Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
19.05Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
19.05Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
19.05Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
19.05Consensusopsins_offOrthosteric Ligandrhodopsin_off
19.05Consensussensory_offOrthosteric Ligandopsins_off
18.75Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
18.75Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
18.75Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
18.75Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
18.75Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
18.75Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
18.75Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
18.75Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
18.75Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
18.75Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
18.75Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
18.75Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
18.52Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
18.52Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
18.52Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
18.52Single7F8XNN90567F8X-CCKA-NN9056
18.52Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
18.52Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
18.52Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
18.52Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
18.52Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
18.52Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
18.52Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
18.52Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
18.52Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
18.52Consensuslpl_onOrthosteric Ligands1p_on lpa_on
18.52Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
18.52Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
18.42Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
18.42Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
18.18Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
18.18Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
18.18Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
18.18Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
18.18Single4DAJTiotropium4DAJ-M3-Tiotropium
18.18Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
18.18Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
18.18Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
18.18Single4MQSIperoxo4MQS-M2-Iperoxo
18.18Single4QIMANTA XV4QIM-SMO-ANTA XV
18.18Single4U14Tiotropium4U14-M3-Tiotropium
18.18Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
18.18Single4YAYZD-71554YAY-AT1-ZD-7155
18.18Single5DHHSB-6121115DHH-NOP-SB-612111
18.18Single5DSGTiotropium5DSG-M4-Tiotropium
18.18Single5IU8Q274563475IU8-A2A-Q27456347-Na
18.18Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
18.18Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
18.18Single6D27CAY104716D27-DP2-CAY10471
18.18Single6DRXLisuride6DRX-5-HT2B-Lisuride
18.18Single6GPSMK08126GPS-CCR2-MK0812
18.18Single6IGLIRL16206IGL-ETB-IRL1620
18.18Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
18.18Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
18.18Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
18.18Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
18.18Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
18.18Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
18.18Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
18.18Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
18.18Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.18Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
18.18Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
18.18Single7PYRPSB-21157PYR-A2A-PSB-2115
18.18Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
18.18Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
18.18Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
18.18Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
18.18Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
18.18Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
18.18Single7V3ZCP559407V3Z-CB1-CP55940
18.18Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
18.18Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
18.18Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
18.18Single7WC7Lisuride7WC7-5-HT2A-Lisuride
18.18Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
18.18Single8CU6LJ-45178CU6-A2A-LJ-4517
18.18Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
18.18Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
18.18Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
18.18Single8K5DGSK2560738K5D-HCA2-GSK256073
18.18Single8RLNLUF58348RLN-A2A-LUF5834
18.18Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
18.18Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
18.18Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
18.18Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
18.18Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
18.18Single8X63Mepyramine8X63-H1-Mepyramine
18.18Single8X64Desloratadine8X64-H1-Desloratadine
18.18Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
18.18Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
18.18Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
18.18Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.18Consensus5ht5_onOrthosteric Ligand5ht5a_on
18.18Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
18.18Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
18.18Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
18.18Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
18.18Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
18.18Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
18.18Consensusblt_onOrthosteric Ligandblt1_on
18.18Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
18.18Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
18.18Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
18.18Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
18.18Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
18.18Consensushistamine_offOrthosteric Ligandh1_off
18.18Consensusleukotriene_onOrthosteric Ligandblt_on
18.18Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
18.18Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
18.18Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
18.18Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
17.86Single6HLOAprepitant6HLO-NK1-Aprepitant
17.86Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
17.86Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
17.86Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
17.86Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
17.86Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
17.86Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
17.86Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
17.86Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
17.86Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
17.86Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
17.86Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
17.86Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
17.65Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
17.65Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
17.65Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
17.65Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
17.65Single8PWNTheophylline8PWN-A2A-Theophylline
17.65Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.65Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.65Consensusbombesin_onOrthosteric Ligandbb2_on
17.65Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
17.65Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.50Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
17.39Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
17.39Single5IUAQ274563485IUA-A2A-Q27456348-Na
17.39Single5N2SPSB365N2S-A1-PSB36
17.39Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
17.39Single5TVNLSD5TVN-5-HT2B-LSD
17.39Single5WIUNemonapride5WIU-D4-Nemonapride
17.39Single5WIVNemonapride5WIV-D4-Nemonapride-Na
17.39Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
17.39Single6LUQHaloperidol6LUQ-D2-Haloperidol
17.39Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
17.39Single6S0QZM-2413856S0Q-A2A-ZM-241385
17.39Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
17.39Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
17.39Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
17.39Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
17.39Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
17.39Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
17.39Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
17.39Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
17.39Single7SINNPS-21437SIN-CaS-NPS-2143
17.39Single7SINNPS-21437SIN-CaS-NPS-2143
17.39Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
17.39Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
17.39Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
17.39Single7W41PD1762527W41-BB2-PD176252
17.39Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
17.39Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
17.39Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
17.39Single8JXSPF-61428JXS-D1-PF-6142
17.39Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
17.39Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
17.39Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
17.39Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
17.39Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
17.39Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
17.39Single8ZMFA1L108ZMF-5-HT2C-A1L10
17.39Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
17.39Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
17.39Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
17.39Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
17.39Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
17.39Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
17.39Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
17.39Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
17.39Consensusblt_offOrthosteric Ligandblt1_off
17.39Consensusbombesin_offOrthosteric Ligandbb2_off
17.39Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
17.39Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
17.24Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
17.24Single6PT2KGCHM076PT2-δ-KGCHM07
17.24Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
17.24Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
17.24Single6W25SHU91196W25-MC4-SHU9119-Ca
17.24Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
17.24Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
17.24Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
17.24Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
17.24Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.24Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
17.24Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
17.24Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
17.24Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
17.24Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
17.24Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
17.24Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
17.14Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
17.14Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
17.14Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
17.14Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
17.14Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
16.67Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
16.67Single4DJHJDTic4DJH-κ-JDTic
16.67Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
16.67Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
16.67Single5V54Methiothepin5V54-5-HT1B-Methiothepin
16.67Single5XRAAM115425XRA-CB1-AM11542
16.67Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
16.67Single6JODAngiotensin II6JOD-AT2-Angiotensin II
16.67Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
16.67Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
16.67Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
16.67Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
16.67Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
16.67Single6WGTLSD6WGT-5-HT2A-LSD
16.67Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
16.67Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
16.67Single7B6WCyclazosin7B6W-α1b-Cyclazosin
16.67Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
16.67Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
16.67Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
16.67Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
16.67Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
16.67Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
16.67Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
16.67Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
16.67Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
16.67Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
16.67Single7PX4PSB-21137PX4-A2A-PSB-2113
16.67Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
16.67Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
16.67Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
16.67Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
16.67Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
16.67Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
16.67Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
16.67Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
16.67Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
16.67Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
16.67Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
16.67Single8A2OTheophylline8A2O-A2A-Theophylline-Na
16.67Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
16.67Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
16.67Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
16.67Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
16.67Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
16.67Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
16.67Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
16.67Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
16.67Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
16.67Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Single8XVLZibotentan8XVL-ETA-Zibotentan
16.67Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
16.67Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
16.67Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
16.67Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
16.67Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Consensus5ht1_offOrthosteric Ligand5ht1b_off
16.67Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
16.67Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
16.67Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
16.67Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
16.67Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
16.67Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
16.67Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
16.67Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
16.67Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
16.67Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
16.67Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
16.67Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
16.67Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
16.67Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
16.67Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
16.67Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
16.67Consensussensory_onOrthosteric Ligandopsins_on
16.67Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
16.67Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
16.67Consensusvasop-oxy_onOrthosteric Ligandv2_on
16.67Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
16.22Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
16.22Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
16.22Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
16.22Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
16.22Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.13Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
16.13Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
16.13Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
16.13Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
16.13Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
16.13Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
16.13Single8ZRTET-18ZRT-ETB-ET-1
16.13Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
16.13Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
16.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
16.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
16.00Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
16.00Single6KQICP559406KQI-CB1-CP55940-Org27569
16.00Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
16.00Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
16.00Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
16.00Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
16.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
16.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
16.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
16.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
16.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
16.00Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.00Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
16.00Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
16.00Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
16.00Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
16.00Single8JWZAB9288JWZ-A2A-AB928-Na
16.00Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
16.00Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
16.00Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
16.00Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
16.00Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
16.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.00Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
16.00Consensusorexin_onOrthosteric Ligandox2_on
16.00Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.00Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.91Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.79Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
15.79Single3OE6IT1t3OE6-CXCR4-IT1t
15.79Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
15.79Single3UZAGTPL92363UZA-A2A-GTPL9236
15.79Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
15.79Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
15.79Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
15.79Single7WC5Psilocin7WC5-5-HT2A-Psilocin
15.79Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
15.79Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.79Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
15.79Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
15.79Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.79Consensusgi_sensoryOrthosteric Ligandgi_opsins
15.79Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
15.79Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.79Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.79Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
15.79Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
15.79Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
15.62Single4XT3Fractalkine4XT3-US28-Fractalkine
15.62Single6FJ3PTH6FJ3-PTH1-PTH
15.62Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
15.62Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
15.62Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
15.62Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
15.62Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.62Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
15.62Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
15.62Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
15.62Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
15.62Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
15.62Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
15.62Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
15.62Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
15.38Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
15.38Single6K1QIRL25006K1Q-ETB-IRL2500
15.38Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
15.38Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
15.38Single7UM4AS26747237UM4-5-HT5A-AS2674723
15.38Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
15.38Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
15.38Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
15.38Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
15.38Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
15.38Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
15.38Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
15.38Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
15.38Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
15.38Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
15.38Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
15.38Consensuscck_onOrthosteric Ligandccka_on cckb_on
15.38Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
15.38Consensuschemerin_onOrthosteric Ligandcml1_on
15.38Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
15.38Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
15.38Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
15.15Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
15.15Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
15.15Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
15.15Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
15.15Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
15.15Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
15.15Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
15.15Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
15.15Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
15.15Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
15.15Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
15.15Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
15.00Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
15.00Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
15.00Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
15.00Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
15.00Single3OE9IT1t3OE9-CXCR4-IT1t
15.00Single3PBLEticlopride3PBL-D3-Eticlopride
15.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
15.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
15.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
15.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
15.00Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
15.00Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
15.00Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
15.00Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
15.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
15.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
15.00Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
15.00Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
15.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
15.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
15.00Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
15.00Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
15.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
15.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
15.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
14.81Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
14.81Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
14.81Single8QJ2pN1628QJ2-MC4-pN162-Gs
14.81Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
14.81Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
14.81Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
14.81Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
14.71Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
14.71Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
14.71Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
14.71Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
14.71Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
14.71Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
14.71Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
14.71Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
14.71Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusendothelin_onOrthosteric Ligandetb_on eta_on
14.29Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
14.29Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
14.29Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
14.29Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
14.29Single3ODUIT1t3ODU-CXCR4-IT1t
14.29Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
14.29Single4XT1Fractalkine4XT1-US28-Fractalkine
14.29Single5GLHEndothelin-15GLH-ETB-Endothelin-1
14.29Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
14.29Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
14.29Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
14.29Single6B73MP11046B73-κ-MP1104
14.29Single6IGKEndothelin-36IGK-ETB-Endothelin-3
14.29Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
14.29Single6ME2Ramelteon6ME2-MT1-Ramelteon
14.29Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
14.29Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
14.29Single7F8ULintitript7F8U-CCKA-Lintitript
14.29Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
14.29Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
14.29Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
14.29Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
14.29Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
14.29Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
14.29Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
14.29Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
14.29Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
14.29Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
14.29Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
14.29Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
14.29Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
14.29Single7XRRLemborexant7XRR-OX2-Lemborexant
14.29Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
14.29Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
14.29Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
14.29Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
14.29Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
14.29Single8IEBA1LYA8IEB-GPR156-A1LYA
14.29Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
14.29Single8KIGSHU91198KIG-MC3-SHU9119-Ca
14.29Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
14.29Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
14.29Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
14.29Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
14.29Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
14.29Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
14.29Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
14.29Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
14.29Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
14.29Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
14.29Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
14.29Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
14.29Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
14.29Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
14.29Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
14.29Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
14.29Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
14.29Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
14.29Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
14.29Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
14.29Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
13.89Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
13.89Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
13.89Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
13.89Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
13.89Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
13.79Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
13.79Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
13.79Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
13.79Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
13.79Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
13.79Single7XNACYN1548067XNA-SST2-CYN154806
13.79Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
13.79Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
13.79Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
13.79Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
13.79Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
13.79Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
13.79Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
13.79Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
13.79Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
13.79Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
13.79Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
13.64Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
13.64Single3REYXAC3REY-A2A-XAC
13.64Single3RZECidoxepin3RZE-H1-Cidoxepin
13.64Single5IU7Q274563465IU7-A2A-Q27456346-Na
13.64Single5JTBZM-2413855JTB-A2A-ZM-241385
13.64Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
13.64Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
13.64Single6A94Zotepine6A94-5-HT2A-Zotepine
13.64Single6IQLL7458706IQL-D4-L745870
13.64Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
13.64Single6MH8ZM-2413856MH8-A2A-ZM-241385
13.64Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
13.64Single6TPKRetosiban6TPK-OT-Retosiban
13.64Single6TPNHTL66416TPN-OX2-HTL6641
13.64Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
13.64Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
13.64Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
13.64Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
13.64Single7VODCariprazine7VOD-5-HT2A-Cariprazine
13.64Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
13.64Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
13.64Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
13.64Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
13.64Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
13.64Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
13.64Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
13.64Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
13.64Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
13.64Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
13.64Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
13.64Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
13.64Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
13.64Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single9BJKNaloxone9BJK-μ-Naloxone-NAM
13.64Consensusa2_offOrthosteric Liganda2a_off
13.64Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
13.64Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
13.64Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
13.64Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
13.64Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
13.64Consensusvasop-oxy_offOrthosteric Ligandot_off
13.51Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
13.33Single3OE0CVX153OE0-CXCR4-CVX15
13.33Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
13.33Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
13.33Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
13.33Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
13.33Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
13.33Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
13.33Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
13.33Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
13.16Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.04Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
13.04Single2Y02Carmoterol2Y02-β1-Carmoterol
13.04Single3EMLZM-2413853EML-A2A-ZM-241385
13.04Single5DHGC-355DHG-NOP-C-35
13.04Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
13.04Single5UIGCmpd-15UIG-A2A-Cmpd-1
13.04Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
13.04Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
13.04Single6S0LZM-2413856S0L-A2A-ZM-241385
13.04Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
13.04Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
13.04Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
13.04Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
13.04Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
13.04Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
13.04Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
13.04Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
13.04Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
13.04Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
13.04Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
13.04Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
13.04Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
13.04Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
13.04Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
13.04Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
13.04Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
13.04Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
13.04Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
12.90Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
12.90Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
12.90Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
12.90Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
12.90Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
12.90Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
12.90Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
12.82Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
12.50Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
12.50Single5XPRBosentan5XPR-ETB-Bosentan
12.50Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
12.50Single6HLPNetupitant6HLP-NK1-Netupitant
12.50Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
12.50Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
12.50Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
12.50Single7C4SS1P7C4S-S1P3-S1P
12.50Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
12.50Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
12.50Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
12.50Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
12.50Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
12.50Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
12.50Single8GNEKW-63568GNE-A2A-KW-6356-Na
12.50Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
12.50Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
12.50Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
12.50Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
12.50Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
12.50Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
12.50Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
12.50Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
12.50Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
12.50Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
12.20Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
12.12Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
12.12Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
12.12Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
12.12Single7SK3CXCL127SK3-ACKR3-CXCL12
12.12Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
12.12Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
12.12Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
12.12Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
12.12Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
12.12Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
12.00Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
12.00Single6E59L-7607356E59-NK1-L-760735
12.00Single6J20Aprepitant6J20-NK1-Aprepitant
12.00Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
12.00Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
12.00Single7FEECP559407FEE-CB1-CP55940-ZCZ011
12.00Single7R0CAVP7R0C-V2-AVP-Arrestin2
12.00Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
12.00Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
12.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
12.00Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
12.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
12.00Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
12.00Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
12.00Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
12.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
12.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
12.00Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
12.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
12.00Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
12.00Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
12.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
12.00Consensuslpa_onOrthosteric Ligandlpa1_on
12.00Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
12.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
12.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
12.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
12.00Consensustachykinin_offOrthosteric Ligandnk1_off
11.76Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
11.76Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
11.76Single5MZPCaffeine5MZP-A2A-Caffeine-Na
11.76Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
11.76Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
11.76Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
11.76Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
11.76Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
11.76Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
11.76Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
11.76Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
11.76Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
11.63Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
11.54Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
11.54Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
11.54Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
11.54Single6OS2TRV0266OS2-AT1-TRV026
11.54Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
11.54Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
11.54Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
11.54Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
11.54Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
11.54Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
11.54Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
11.54Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
11.54Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
11.54Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
11.43Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
11.43Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
11.43Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
11.43Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
11.43Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
11.43Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
11.43Single8IY6Endothelin-18IY6-ETB-Endothelin-1
11.43Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
11.11Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
11.11Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
11.11Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
11.11Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
11.11Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
11.11Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
11.11Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single7WC4Serotonin7WC4-5-HT2A-Serotonin
11.11Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
11.11Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
11.11Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.11Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
11.11Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
11.11Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
11.11Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
11.11Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
11.11Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
11.11Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
11.11Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
10.81Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
10.81Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
10.81Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
10.71Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
10.71Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
10.71Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
10.71Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
10.71Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
10.71Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
10.71Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
10.71Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
10.71Single8IEIA1LYA8IEI-GPR156-A1LYA
10.71Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
10.71Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
10.71Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
10.71Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
10.71Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
10.71Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.71Consensuskisspeptin_onOrthosteric Ligandkiss1_on
10.71Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
10.53Single3OE8IT1t3OE8-CXCR4-IT1t
10.53Single3RFMCaffeine3RFM-A2A-Caffeine
10.53Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.53Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
10.34Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
10.34Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
10.34Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
10.34Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
10.34Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
10.34Single8IEIA1LYA8IEI-GPR156-A1LYA
10.34Single8IEPA1LYA8IEP-GPR156-A1LYA
10.34Single8IEPA1LYA8IEP-GPR156-A1LYA
10.34Single8WKYPG-9348WKY-MC4-PG-934
10.34Single8XWNCXCL88XWN-CXCR2-CXCL8
10.34Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.34Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.34Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.34Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
10.34Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
10.34Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
10.34Consensussomatostatin_offOrthosteric Ligandsst2_off
10.26Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
10.00Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
10.00Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
10.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
10.00Single6ME5Agomelatine6ME5-MT1-Agomelatine
10.00Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
10.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
10.00Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
10.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
10.00Single7F61Cholesterol7F61-H3-PF-03654746-Cholesterol
10.00Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
10.00Single7SK5CXCL127SK5-ACKR3-CXCL12
10.00Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8IEBA1LYA8IEB-GPR156-A1LYA
10.00Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.00Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
10.00Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
10.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
10.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
10.00Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
10.00Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
10.00Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
9.68Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
9.68Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
9.68Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
9.68Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
9.68Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
9.52Single4O9RCyclopamine4O9R-SMO-Cyclopamine
9.52Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
9.52Single6HLLCP999946HLL-NK1-CP99994
9.52Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
9.52Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
9.52Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
9.52Single6TP4ACT-4622066TP4-OX1-ACT-462206
9.52Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
9.52Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
9.52Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
9.52Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
9.52Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
9.52Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
9.38Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
9.38Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
9.38Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
9.38Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
9.38Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
9.09Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
9.09Single4QINSAG1.54QIN-SMO-SAG1.5
9.09Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
9.09Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
9.09Single6ME9Ramelteon6ME9-MT2-Ramelteon
9.09Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
9.09Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
9.09Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
9.09Single7BR3Elagolix7BR3-GnRH1-Elagolix
9.09Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
9.09Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
9.09Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
9.09Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
9.09Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
9.09Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
9.09Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
9.09Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
9.09Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
9.09Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
9.09Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
9.09Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
9.09Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
9.09Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
9.09Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
9.09Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
9.09Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
9.09Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
9.09Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
8.82Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
8.82Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
8.70Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
8.70Single5UVIZM-2413855UVI-A2A-ZM-241385
8.70Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
8.70Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
8.70Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
8.70Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
8.70Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
8.70Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
8.70Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
8.70Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
8.70Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
8.70Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
8.70Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
8.70Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
8.70Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
8.70Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.70Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
8.70Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
8.70Consensusgrh_offOrthosteric Ligandgnrh1_off
8.70Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
8.57Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
8.33Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
8.33Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
8.33Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
8.33Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
8.33Single7F83PF-051904577F83-Ghrelin-PF-05190457
8.33Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
8.33Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
8.33Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
8.33Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
8.33Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
8.33Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
8.33Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
8.33Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
8.33Consensuscck_offOrthosteric Ligandccka_off
8.33Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
8.11Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
8.00Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
8.00Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
8.00Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
8.00Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
8.00Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
8.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
8.00Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
8.00Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
8.00Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
8.00Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.00Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
8.00Single8QOTNanobody-E8QOT-μ-Nanobody-E
8.00Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
8.00Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
8.00Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
8.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
8.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
8.00Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
8.00Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
7.69Single5TZRMK86665TZR-FFA1-MK8666
7.69Single6OS1TRV0266OS1-AT1-TRV026
7.69Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
7.69Single7F1TMIP-1a7F1T-CCR5-MIP-1a
7.69Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
7.69Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
7.69Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
7.69Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
7.69Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
7.69Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
7.69Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
7.69Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
7.69Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
7.69Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
7.69Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
7.50Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
7.41Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
7.41Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
7.41Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
7.41Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
7.41Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
7.41Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
7.41Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
7.41Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
7.41Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
7.14Single8XVUCXCL28XVU-CXCR2-CXCL2
7.14Single8XWFCXCL38XWF-CXCR2-CXCL3
7.14Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
7.14Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
7.14Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
6.90Single6KNMJN241-96KNM-Apelin-JN241-9
6.90Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
6.90Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
6.90Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single8XQJJN2418XQJ-Apelin-JN241
6.90Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
6.90Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
6.90Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
6.67Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
6.67Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
6.67Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
6.67Single8W8SAA-148W8S-GPR101-AA-14
6.67Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
6.67Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
6.67Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
6.67Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
6.45Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
6.45Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
6.45Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
6.45Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
6.25Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
6.25Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
6.25Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
6.25Single8W8RAA-148W8R-GPR101-AA-14-chim(NtGi1-Gs)/β1/γ2
6.25Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
6.25Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
6.06Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
5.88Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
5.88Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
5.88Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
5.88Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
5.56Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
5.26Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
5.26Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
5.26Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
5.26Single8HS2Fab0468HS2-GPR20-Fab046
5.26Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
5.26Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.26Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
5.26Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
5.00Single6TQ9SB-4081246TQ9-OX1-SB-408124
5.00Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
5.00Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
5.00Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
5.00Consensusp2y_offOrthosteric Ligandp2y1_off
4.76Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
4.76Single4XNWMRS25004XNW-P2Y1-MRS2500
4.76Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
4.76Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
4.76Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
4.76Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.76Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
4.76Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
4.76Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
4.76Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.76Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
4.76Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
4.76Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
4.76Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
4.55Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
4.55Single7FEEZCZ0117FEE-CB1-CP55940-ZCZ011
4.55Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
4.55Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
4.55Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
4.55Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.55Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
4.55Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.55Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
4.55Consensusgq_nucleotideOrthosteric Ligandgq_p2y
4.55Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
4.35Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
4.35Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
4.35Single4BWBNeurotensin4BWB-NTS1-Neurotensin
4.35Single4XNVBPTU4XNV-P2Y1-BPTU
4.35Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
4.35Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
4.35Single7F8YDevazepide7F8Y-CCKA-Devazepide
4.35Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.35Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
4.35Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
4.35Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
4.35Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
4.35Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
4.35Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
4.35Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
4.35Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
4.35Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
4.17Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7VV6C48/807VV6-MRGPRX2-C48/80
4.17Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
4.17Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
4.17Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
4.00Single5T04Neurotensin5T04-NTS1-Neurotensin
4.00Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
4.00Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
4.00Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.00Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
4.00Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
4.00Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
4.00Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
4.00Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
4.00Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
4.00Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.00Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
4.00Single9IYAONO-97105319IYA-GPR55-ONO-9710531
4.00Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
4.00Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
4.00Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
3.85Single4NTJAZD12834NTJ-P2Y12-AZD1283
3.85Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
3.85Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
3.85Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
3.70Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
3.70Single4BV0Neurotensin4BV0-NTS1-Neurotensin
3.70Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
3.70Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
3.70Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
3.70Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
3.70Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
3.70Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
3.70Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
3.70Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
3.70Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
3.70Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
3.70Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
3.70Consensusneurotensin_onOrthosteric Ligandnts1_on
3.70Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
3.57Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
3.57Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
3.57Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
3.57Single4PY02MeSATP4PY0-P2Y12-2MeSATP
3.57Single4XEENeurotensin4XEE-NTS1-Neurotensin
3.57Single4XESNeurotensin4XES-NTS1-Neurotensin
3.57Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
3.57Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
3.57Single6YVRNTS8-136YVR-NTS1-NTS8-13
3.57Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
3.57Single7SHEPI; PE7SHE-GPR158-PI; PE
3.57Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.57Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.57Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
3.57Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
3.57Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
3.57Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
3.57Single8XQJJN2418XQJ-Apelin-JN241
3.57Single8XWACXCL18XWA-CXCR2-CXCL1
3.57Single8XWMCXCL68XWM-CXCR2-CXCL6
3.57Single8XWSCXCL58XWS-CXCR2-CXCL5
3.57Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
3.57Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
3.57Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
3.57Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
3.57Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
3.45Single4BUONeurotensin4BUO-NTS1-Neurotensin
3.45Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
3.45Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
3.45Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.45Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
3.45Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
3.45Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
3.45Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
3.45Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
3.45Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.45Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.33Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
3.33Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
3.33Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
3.33Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
3.23Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
3.23Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.23Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
3.12Single7SHEPI; PE7SHE-GPR158-PI; PE
3.12Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7

Consensus Members
Id Members
8IUK 8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
8IUL 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
8IUM 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
Net Summary
Imin 2.78
Number of Linked Nodes 893
Number of Links 1026
Number of Hubs 144
Number of Links mediated by Hubs 540
Number of Communities 28
Number of Nodes involved in Communities 210
Number of Links involved in Communities 295
Path Summary
Number Of Nodes in MetaPath 118
Number Of Links MetaPath 117
Number of Shortest Paths 802553
Length Of Smallest Path 3
Average Path Length 35.2058
Length of Longest Path 95
Minimum Path Strength 0.466667
Average Path Strength 6.40657
Maximum Path Strength 19.6367
Minimum Path Correlation 0.706667
Average Path Correlation 0.975895
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.51515
Average % Of Corr. Nodes 43.0823
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 44.1614
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
prostanoid_on_gptp_on_gp
fp-alpha_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download fp-alpha_on_gp.zip



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