Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1b.1x15 3.3625407
2b.lhb1x3 3.634512
3b.lhb1x6 5.826513
4b.lhb1x9 3.785403
5b.lhb1x11 3.87514
6b.b1x3 7.054127
7b.b1x4 4.80254127
8b.b1x6 5.335459
9b.l1x3 9.99167659
10b.l1x4 3.375406
11b.b2x1 8.05667618
12b.b2x3 4656
13b.b2x5 6.49667657
14b.l3x2 4.804559
15b.b4x3 3.8325477
16b.b4x5 3.49477
17b.b4x6 9.99659
18b.b5x2 5.8054137
19b.b5x3 5.78286759
20b.b5x5 4.28475
21b.b5x7 7.0225477
22b.l5x1 4.834578
23b.l5x5 9.562519
24b.b6x5 4.65375876
25b.b7x1 5.178594
26b.b7x4 3.42478
27b.l7x2 4.19429719
28b.b8x3 3.38496
29b.b8x4 5.49776
30b.l8x8 5.82474
31b.b9x4 7.355409
32b.l9x3 6.58286719
33b.l9x6 4.36222918
34b.b10x4 5.8625466
35b.b10x5 3.168509
36b.l10x1 3.462503
37b.b11x3 4.335465
38b.b11x4 4.4525419
39b.b11x5 4.3925406
40b.l11x1 3.2775419
41b.b12x5 3.7466
42b.b12x6 8.51618
43b.b13x3 6.6875414
44b.b13x7 6.814567
45b.l13x3 8.042569
46b.l13x6 4.6519
47b.b14x1 3.8875418
48b.b14x3 4.434565
49b.b15x1 6.19667669
50b.b15x2 6.224546
51b.l15x1 4.24333617
52b.b16x4 9.51466
53b.b16x5 3.0825445
54b.b16x6 8.36833668
55b.l16x3 9.4725443
56b.b17x3 5.635465
57b.b17x4 6.2825445
58b.b17x5 5.644547
59b.b17x7 7.374548
60b.l17x3 7.0975849
61b.l17x6 6.905619
62b.b18x3 5.2548
63b.b18x5 5.9775445
64b.l18x1 5.646516
65b.l18x2 4.44417
66b.l18x3 5.0825415
67b.b19x2 6.68429746
68b.b19x4 5.01548
69b.l19x2 6.0275449
70b.b20x2 3.78546
71b.b20x3 3.5875418
72b.b20x4 10.458548
73b.b20x6 6.69167646
74b.b20x7 4.158509
75b.l20x1 2.55546
76b.l20x2 7.565409
77b.b21x1 8.6447
78b.b21x5 4.075414
79b.b21x7 5.39167615
80b.l21x2 6.695414
81b.l21x5 4.2375414
82b.l21x7 3.83415
83b.b22x5 5.79143717
84b.l22x1 4.2375419
85b.l22x4 2.144519
86b.l22x5 6.49667619
87b.b23x6 6.015617
88b.l23x1 7.23416
89b.b24x2 3.93405
90b.b24x4 6.255416
91b.b24x6 4.4575418
92b.l24x2 4.4325416
93b.l24x3 5.825405
94b.b25x3 6.6415
95b.l25x3 8.268519
96b.l25x6 10.565418
97b.b26x3 5.2725406
98b.l26x1 8.0175457
99b.b27x1 3.825416
100b.b27x3 5.1525418
101b.l27x1 9.1875819
102b.l27x2 7.895419
103b.b28x3 3.27833657
104b.b28x4 6.005416
105b.b28x6 6.105619
106G.HN.43 2.835459
107G.S1.01 7.0675416
108G.S1.02 5.9375435
109G.S1.04 5.22437
110G.S1.06 4.2525438
111G.H1.01 8.63509
112G.S2.05 6.505419
113G.S2.06 9.105433
114G.S2.08 6.412534
115G.S3.03 6.455636
116G.S3.04 7.166517
117G.S3.05 4.012535
118G.S3.06 7.744519
119G.s3h2.03 5.198519
120G.H2.02 4.2925419
121G.H2.03 9.9325419
122G.H2.06 7.58167619
123G.H2.07 4.38143718
124G.H2.08 4.16418
125G.h2s4.01 6.85667617
126G.h2s4.02 5.3675415
127G.S4.02 5.1825417
128G.S4.03 4.21439
129G.S4.04 6.088517
130G.S4.06 3.47418
131G.s4h3.01 4.5875419
132G.s4h3.04 4.985619
133G.H3.09 6.41857715
134G.H3.13 4.2025418
135G.H3.17 6.68143719
136G.H3.18 6.574513
137G.S5.03 3.04539
138G.S5.04 4.182519
139G.S5.05 3.542538
140G.S5.06 4.864519
141G.HG.04 5.956515
142G.hgh4.01 4.605417
143G.hgh4.02 8.484515
144G.hgh4.05 6.616513
145G.H4.03 7.618514
146G.H4.05 4.8525417
147G.H4.10 9.8975417
148G.H4.11 3.71415
149G.H4.15 4.63613
150G.S6.01 5.315417
151G.S6.02 8.42143735
152G.S6.05 4.736519
153G.s6h5.01 5.945437
154G.s6h5.02 3.66409
155G.H5.03 7.7625437
156G.H5.08 5.50286734
157G.H5.25 5.03425
1581x35 2.5125425
1591x39 4.854528
1601x40 2.88406
1611x42 4.9075427
1621x43 6.0425407
1631x47 4.6825406
1641x50 4.635409
1651x57 7.46427
1662x39 3.43407
1672x43 6.6325428
1682x46 4.634529
1692x50 4.685629
1702x53 5.3275407
1712x54 3.9575406
1722x57 3.90333628
1732x60 7.93427
1743x30 3.614506
1753x32 6.47333627
1763x33 5.25375825
1773x36 3.52528
1783x37 5.822528
1793x38 4.82407
1803x40 5.6975428
1813x41 5.71525
1823x43 3.9975428
1833x50 5.946529
1844x50 4.075159
1854x56 7.3125424
186E2.Q148 14.16425
187E2.Y149 8.45485
188E2.E154 5.5075481
189E2.N160 7.526525
190E2.I162 5.365424
191E2.T163 4.372524
192E2x50 5.3725489
193E2x52 3.72525
194E2.F168 4.278524
1955x40 9.848525
1965x43 3.7525
1975x44 4.13426
1985x461 5.69167626
1995x47 6.264528
2005x48 2.8025424
2015x50 5.23429
2025x51 2.6825426
2035x58 7.40167628
2045x61 4.59528
2055x65 4.18428
206I3.H211 12.815433
207I3.V212 4.232503
2086x45 3.92833629
2096x48 6.13167629
2106x51 4.98125827
2116x52 7.9325428
2126x54 4.255425
2136x55 6.2875406
214E3.P252 4.148521
2157x33 4.265424
2167x34 6.00143725
2177x38 4.1225425
2187x45 7.342529
2197x49 7.0775429
220g.h1x11 2.0925409
221g.h1x14 6.0525469
222g.l1x4 4.756508
223g.ctx3 6.15519
224g.ctx6 2.804516
225g.ctx14 7.8025409
226Lig 6.432941720
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.1x15 g.h1x11 10.5251.43YesYes079
2b.b17x7 b.b21x1 14.49445.97YesYes487
3b.b17x7 b.b20x6 18.08028.57YesYes486
4b.b20x6 b.l17x3 22.39053.39YesYes469
5b.l17x3 b.l19x2 30.45395.04YesYes499
6b.l17x5 b.l19x2 32.50634.42NoYes069
7b.l17x5 b.l19x1 32.75992.94NoNo069
8b.l17x6 b.l19x1 33.012814.64YesNo199
9b.b14x1 b.l17x6 16.66374.16YesYes189
10b.b14x1 b.l9x6 17.17862.39YesYes188
11b.b6x1 b.l9x6 33.62142.39NoYes198
12b.b2x1 b.b6x1 34.82632.39YesNo189
13b.b2x1 b.l27x1 37.9439.65YesYes189
14b.b26x1 b.l27x1 86.02024.94NoYes099
15b.b26x1 b.b26x2 86.1333.44NoNo097
16b.b26x2 b.b2x3 43.21836.48NoYes076
17b.b28x3 b.b2x3 52.55022.83YesYes576
18G.H2.06 b.l17x6 16.66585.53YesYes199
19G.H2.06 b.l9x6 17.43755.97YesYes198
20b.b26x2 b.b27x4 43.03071.96NoNo075
21b.b27x4 b.b28x3 43.08413.42NoYes057
22b.b28x3 b.b4x6 32.05073.42YesYes579
23b.b28x3 b.l1x7 31.71212.85YesNo079
24b.l1x3 b.l1x7 31.71819.28YesNo099
25b.b28x3 b.b3x4 31.71043YesNo579
26b.b3x4 b.l1x3 31.71519.76NoYes599
27b.b4x6 b.l1x3 32.6828.46YesYes599
28b.l1x3 b.l3x2 96.47113.78YesYes599
29b.l1x4 b.l3x2 1004.07YesYes069
30G.H2.08 G.H3.17 20.47522.35YesYes189
31G.S6.02 I3.H211 12.537919.6YesYes353
32I3.H211 I3.P210 12.83533.05YesNo033
335x68 I3.P210 12.93364.74NoNo053
345x68 I3.V212 13.01774.3NoYes053
355x65 I3.V212 13.70373.04YesYes083
363x50 G.H5.25 13.37110.93YesYes295
373x46 3x50 14.43292.51NoYes099
382x43 3x46 14.60922.85YesNo089
391x57 2x43 15.583214.61YesYes278
401x57 2x47 99.56223.89YesNo078
411x54 2x47 99.62152.95NoNo078
421x54 1x58 99.76522.98NoNo074
431x58 1x59 99.79141.84NoNo044
441x59 1x63 99.84371.64NoNo045
451x63 I1.P39 99.86983.16NoNo053
46I1.P39 b.l1x4 99.89581.64NoYes036
47G.H3.12 G.S1.07 11.68237.14NoNo059
48G.S1.07 G.S4.04 13.51282.44NoYes097
49G.H2.08 G.H3.18 19.50956.28YesYes183
50G.H3.18 G.S4.02 26.0298.79YesYes137
51G.S4.02 G.S5.02 25.5427.36YesNo178
52G.H3.09 G.S5.02 23.56492.51YesNo158
53G.H3.09 G.H4.15 16.1136.43YesYes153
54G.H4.11 G.H4.15 12.52812.51YesYes153
552x46 2x50 16.78346.79YesYes299
562x46 7x53 75.04142.44YesNo299
571x57 7x53 74.74418.57YesNo279
583x30 Lig 13.69981.74YesYes060
593x33 Lig 20.66097.55YesYes250
603x33 3x36 24.95112.42YesYes258
613x36 6x48 45.80542.51YesYes289
626x45 6x48 17.20183.22YesYes299
633x43 6x45 24.92083.65YesYes289
642x46 3x43 41.54554.15YesYes298
656x51 Lig 37.31874.2YesYes270
663x36 6x51 20.26363.63YesYes287
676x51 7x41 20.26053.82YesNo278
686x48 7x41 20.44473.96YesNo298
696x48 7x45 49.271213.29YesYes299
703x43 7x45 16.65264.12YesYes289
712x50 7x45 16.68882.69YesYes299
727x45 7x49 16.631213.46YesYes299
732x46 7x49 16.67346.79YesYes299
74E1x52 E2x50 10.75633.17NoYes079
753x22 E2x50 15.36589.7NoYes829
763x22 E2.E161 18.43891.35NoNo823
77E2.E161 E2.Y149 19.974710.1NoYes835
78E2.T152 E2.Y149 29.19324.99NoYes035
79E2.I162 E2.T152 30.72954.56YesNo043
80E2.I162 E2.Q148 13.69389.61YesYes245
81E2.Q148 Lig 16.302122.87YesYes250
82E2.I162 E2.T163 18.57133.04YesYes244
83E2.T163 Lig 14.34576.33YesYes240
84G.H3.12 G.H3.18 10.90992.51NoYes053
85G.H3.15 G.H3.18 19.15883.62NoYes143
86G.H3.15 G.H3.17 19.27883.39NoYes149
87G.H3.17 b.l27x1 39.57753.75YesYes199
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
2x603x3213.652YesYes7722
2x603x334.782YesYes7521
3x303x314.520YesNo6512
3x304x546.430YesNo6312
3x304x572.790YesNo6712
3x304x582.590YesNo6412
3x323x333.092YesYes7521
3x327x382.622YesYes7522
3x333x362.422YesYes5812
3x33E2x523.372YesYes5511
3x336x519.932YesYes5711
3x337x342.062YesYes5511
3x337x388.832YesYes5512
3x33Lig7.552YesYes5010
3x366x513.632YesYes8721
3x367x416.192YesNo8822
3x375x435.862YesYes8521
3x375x4618.212YesYes8622
3x376x515.962YesYes8721
3x376x525.812YesYes8822
3x376x553.272YesYes8622
4x565x429.852YesNo4422
4x565x433.862YesYes4521
4x565x46110.292YesYes4622
4x60Lig11.730NoYes5010
4x61E2.N1608.50NoYes4512
4x61Lig4.090NoYes4010
E2.N151E2.V1472.960NoNo5421
E2.V147Lig5.330NoYes4010
E2.N160E2.Q14818.492YesYes5521
E2.I162E2.Q1489.612YesYes4521
E2.Q148E2.T1635.672YesYes5411
E2.Q148Lig22.872YesYes5010
E2.I162E2.N1604.252YesYes4522
E2.I162E2.T1633.042YesYes4421
E2.T163E2x524.232YesYes4511
E2.F168E2.T1632.592YesYes4411
E2.T163Lig6.332YesYes4010
E2.F168E2x522.332YesYes4511
7x34E2x525.822YesYes5511
E2x52Lig2.852YesYes5010
5x32E2.F16810.542NoYes1411
5x33E2.F1682.440NoYes1421
E2.F168Lig3.492YesYes4010
5x32Lig4.762NoYes1010
5x35Lig6.40NoYes3010
5x365x372.982NoNo4212
5x365x406.542NoYes4511
5x36Lig8.532NoYes4010
5x39Lig5.330NoYes4010
5x406x5514.672YesYes5612
5x40E3.S2515.272YesNo5412
5x407x3414.932YesYes5511
5x40Lig7.832YesYes5010
5x425x432.652NoYes4521
5x435x4614.152YesYes5612
5x43Lig1.982YesYes5010
6x516x524.652YesYes7812
6x517x345.142YesYes7511
6x517x382.522YesYes7512
6x517x413.822YesNo7812
6x51Lig4.22YesYes7010
6x546x552.792YesYes5622
6x54E3.P2525.342YesYes5122
6x547x343.952YesYes5521
E3.P252E3.S2513.562YesNo1422
7x34E3.P2525.762YesYes5112
7x34Lig4.352YesYes5010
3x30Lig1.740YesYes6010
4x62E2.V1471.540NoNo4421

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
92.86Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
87.50Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
66.67Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
58.82Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
58.82Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
58.82Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
58.82Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
57.89Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
55.56Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
55.56Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
47.37Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
47.37Single4PY02MeSATP4PY0-P2Y12-2MeSATP
44.44Single4NTJAZD12834NTJ-P2Y12-AZD1283
44.00Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
43.75Single6ME9Ramelteon6ME9-MT2-Ramelteon
43.48Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
42.86Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
42.11Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
42.11Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
41.67Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
41.67Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
40.91Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
40.00Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
40.00Single6ME5Agomelatine6ME5-MT1-Agomelatine
40.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
40.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
40.00Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
40.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
40.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
40.00Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
38.89Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
38.89Single9IYAONO-97105319IYA-GPR55-ONO-9710531
38.10Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
38.10Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
37.50Single6HLLCP999946HLL-NK1-CP99994
36.84Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
36.84Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
36.84Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
36.84Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.84Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
36.84Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
36.84Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
36.36Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
36.36Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
36.36Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
35.29Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
35.29Single6ME2Ramelteon6ME2-MT1-Ramelteon
35.29Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
35.29Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
35.29Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.00Single5TZRMK86665TZR-FFA1-MK8666
35.00Single6J21Aprepitant6J21-NK1-Aprepitant
35.00Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
35.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
35.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
35.00Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
35.00Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
35.00Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
35.00Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
35.00Consensustachykinin_offOrthosteric Ligandnk1_off
34.78Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
34.78Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
34.78Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
34.78Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
34.78Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
34.78Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
33.33Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
33.33Single6HLOAprepitant6HLO-NK1-Aprepitant
33.33Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
33.33Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
33.33Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
33.33Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
33.33Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
33.33Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
33.33Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
33.33Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
33.33Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
33.33Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
33.33Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
33.33Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
33.33Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
33.33Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
33.33Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
32.14Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
32.00Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
32.00Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
32.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
32.00Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
32.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
32.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
31.82Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
31.82Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.82Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
31.82Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
31.82Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
31.58Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
31.58Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
31.58Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
31.58Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.58Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
31.58Consensusa3_onOrthosteric Liganda3a_on
31.58Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
31.25Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
31.25Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
31.25Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
31.25Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
30.77Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
30.77Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
30.77Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.77Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
30.77Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
30.77Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
30.43Single3NY9ICI118-5513NY9-β2-ICI118-551
30.43Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
30.43Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
30.43Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
30.43Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
30.43Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
30.43Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
30.43Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
30.00Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
30.00Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
30.00Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
30.00Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
30.00Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
30.00Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
30.00Single7W41PD1762527W41-BB2-PD176252
30.00Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
30.00Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
30.00Single8QOTNanobody-E8QOT-μ-Nanobody-E
30.00Consensusa3_on_gpOrthosteric Liganda3a_on_gp
30.00Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
30.00Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
30.00Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
30.00Consensusbombesin_offOrthosteric Ligandbb2_off
30.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
30.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
29.63Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
29.63Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.41Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
29.41Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
29.41Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
29.41Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
29.17Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
29.17Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
29.17Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
29.17Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
29.17Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
29.17Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.17Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.17Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
28.57Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
28.57Single6J20Aprepitant6J20-NK1-Aprepitant
28.57Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
28.57Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
28.57Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
28.57Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
28.57Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.57Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
28.57Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
28.57Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
28.57Consensusa2_onOrthosteric Liganda2b_on
28.57Consensusa2_on_gpOrthosteric Liganda2b_on_gp
28.57Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
28.57Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
28.57Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
28.57Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
28.57Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
28.57Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
28.12Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
28.00Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
28.00Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
28.00Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
27.78Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
27.78Single3PWHZM-2413853PWH-A2A-ZM-241385
27.78Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
27.78Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
27.78Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
27.78Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
27.78Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
27.78Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
27.78Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.78Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
27.78Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
27.78Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
27.78Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.78Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
27.78Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
27.59Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
27.59Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
27.27Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
27.27Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
27.27Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
27.27Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
27.27Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
27.27Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
27.27Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
27.27Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
27.27Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
27.27Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
27.27Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
27.27Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.92Single3OE0CVX153OE0-CXCR4-CVX15
26.92Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
26.92Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
26.92Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
26.92Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
26.92Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
26.32Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
26.32Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
26.32Single5IU7Q274563465IU7-A2A-Q27456346-Na
26.32Single5IUBQ274563445IUB-A2A-Q27456344-Na
26.32Single5JTBZM-2413855JTB-A2A-ZM-241385
26.32Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
26.32Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
26.32Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
26.32Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
26.32Single5UVIZM-2413855UVI-A2A-ZM-241385
26.32Single6AQFZM-2413856AQF-A2A-ZM-241385
26.32Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
26.32Single6MH8ZM-2413856MH8-A2A-ZM-241385
26.32Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
26.32Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
26.32Single7AROLUF58337ARO-A2A-LUF5833-Na
26.32Single7T32ZM-2413857T32-A2A-ZM-241385
26.32Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
26.32Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
26.32Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
26.32Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
26.32Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
26.32Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.32Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
26.32Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
26.32Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Consensusa2_offOrthosteric Liganda2a_off
26.32Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
26.09Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
26.09Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
26.09Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
26.09Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
26.09Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
26.09Single7UM4AS26747237UM4-5-HT5A-AS2674723
26.09Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
26.09Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
26.09Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
26.09Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
26.09Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
26.09Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
26.09Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
26.09Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
26.09Consensuschemerin_onOrthosteric Ligandcml1_on
26.09Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
26.09Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
25.93Single6JODAngiotensin II6JOD-AT2-Angiotensin II
25.93Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
25.93Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
25.93Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
25.81Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
25.81Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
25.81Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
25.81Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
25.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
25.00Single3EMLZM-2413853EML-A2A-ZM-241385
25.00Single3RFMCaffeine3RFM-A2A-Caffeine
25.00Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
25.00Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
25.00Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
25.00Single4UG2CGS216804UG2-A2A-CGS21680
25.00Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
25.00Single5IU8Q274563475IU8-A2A-Q27456347-Na
25.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
25.00Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
25.00Single5UENDU1725UEN-A1-DU172
25.00Single5UIGCmpd-15UIG-A2A-Cmpd-1
25.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
25.00Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
25.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
25.00Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
25.00Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
25.00Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
25.00Single6S0LZM-2413856S0L-A2A-ZM-241385
25.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
25.00Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
25.00Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
25.00Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
25.00Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
25.00Single7PYRPSB-21157PYR-A2A-PSB-2115
25.00Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
25.00Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
25.00Single7XN9L-054,5227XN9-SST2-L-054,522
25.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
25.00Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
25.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
25.00Single8CU6LJ-45178CU6-A2A-LJ-4517
25.00Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
25.00Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
25.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
25.00Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
25.00Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
25.00Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
25.00Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
25.00Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
25.00Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
25.00Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
25.00Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
25.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
25.00Single9CHXS-Carazolol9CHX-β2-S-Carazolol
25.00Single9H37A1IR09H37-A2A-A1IR0-Na
25.00Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
25.00Single9JF4PD1683689JF4-BB1-PD168368
25.00Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
25.00Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
25.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
25.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
25.00Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
25.00Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
25.00Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
25.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
25.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
25.00Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.00Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
24.00Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
24.00Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
24.00Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.00Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
24.00Single8IEBA1LYA8IEB-GPR156-A1LYA
24.00Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
24.00Single8WDTphotoNECA8WDT-A2A-photoNECA
24.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.00Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
24.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
24.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
24.00Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
23.81Single2YCWS-Carazolol2YCW-β1-S-Carazolol
23.81Single5D6LS-Carazolol5D6L-β2-S-Carazolol
23.81Single5IUAQ274563485IUA-A2A-Q27456348-Na
23.81Single5N2SPSB365N2S-A1-PSB36
23.81Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
23.81Single5TVNLSD5TVN-5-HT2B-LSD
23.81Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
23.81Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
23.81Single6HLPNetupitant6HLP-NK1-Netupitant
23.81Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
23.81Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
23.81Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
23.81Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
23.81Single6S0QZM-2413856S0Q-A2A-ZM-241385
23.81Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
23.81Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
23.81Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
23.81Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
23.81Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.81Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
23.81Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
23.81Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8GNEKW-63568GNE-A2A-KW-6356-Na
23.81Single8JXSPF-61428JXS-D1-PF-6142
23.81Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
23.81Single8ZMFA1L108ZMF-5-HT2C-A1L10
23.81Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
23.81Single9EHSLUF76029EHS-A3A-LUF7602
23.81Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
23.81Single9HAPTolvaptan9HAP-V2-Tolvaptan
23.81Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
23.81Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
23.81Consensusadenosine_offOrthosteric Liganda1_off a2_off
23.81Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
23.81Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
23.81Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
23.81Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
23.81Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
23.81Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
23.81Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
23.81Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.81Consensustrace-amine_onOrthosteric Ligandta1_on
23.53Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
23.53Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
23.53Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
23.53Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.53Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
23.53Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
23.53Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
23.33Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
23.33Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
23.33Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
23.33Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
23.33Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
23.33Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
23.33Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
23.33Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
23.08Single3QAKUK-4320973QAK-A2A-UK-432097
23.08Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
23.08Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
23.08Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
23.08Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
23.08Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
23.08Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
23.08Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
23.08Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
23.08Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
23.08Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
23.08Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
23.08Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
23.08Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
23.08Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
22.73Single2YDVNECA2YDV-A2A-NECA
22.73Single3P0GBI1671073P0G-β2-BI167107
22.73Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
22.73Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
22.73Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
22.73Single4UHRCGS216804UHR-A2A-CGS21680
22.73Single5D5AS-Carazolol5D5A-β2-S-Carazolol
22.73Single5D5BS-Carazolol5D5B-β2-S-Carazolol
22.73Single5G53NECA5G53-A2A-NECA-Gs
22.73Single5V54Methiothepin5V54-5-HT1B-Methiothepin
22.73Single5XR8AM8415XR8-CB1-AM841
22.73Single6E59L-7607356E59-NK1-L-760735
22.73Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
22.73Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
22.73Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
22.73Single7F1TMIP-1a7F1T-CCR5-MIP-1a
22.73Single7PX4PSB-21137PX4-A2A-PSB-2113
22.73Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
22.73Single7TUYGSK682753A7TUY-GPR183-GSK682753A
22.73Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
22.73Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
22.73Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
22.73Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
22.73Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
22.73Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
22.73Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
22.73Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
22.73Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
22.73Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
22.73Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
22.73Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
22.73Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
22.73Single9BJKNaloxone9BJK-μ-Naloxone-NAM
22.73Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
22.73Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
22.73Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
22.73Consensus5ht1_offOrthosteric Ligand5ht1b_off
22.73Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
22.73Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
22.73Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
22.73Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
22.73Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
22.73Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
22.73Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
22.73Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
22.73Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
22.73Consensuslpa_onOrthosteric Ligandlpa1_on
22.73Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
22.73Consensusrelaxin_onOrthosteric Ligandrxfp4_on
22.73Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
22.73Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.73Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
22.58Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
22.58Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
22.58Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
22.58Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
22.58Consensusbradykinin_onOrthosteric Ligandbk2_on
22.58Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
22.58Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
22.22Single3PBLEticlopride3PBL-D3-Eticlopride
22.22Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
22.22Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
22.22Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
22.22Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
22.22Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
22.22Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
22.22Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
22.22Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
22.22Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
22.22Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
22.22Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
22.22Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
22.22Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
22.22Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.22Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
22.22Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
22.22Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
22.22Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
22.22Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
22.22Consensusangiotensin_onOrthosteric Ligandat1_on
22.22Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
22.22Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
22.22Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
21.74Single3D4STimolol3D4S-β2-Timolol
21.74Single4RWADIPP-NH24RWA-δ-DIPP-NH2
21.74Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
21.74Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
21.74Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
21.74Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
21.74Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
21.74Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
21.74Single6MXTSalmeterol6MXT-β2-Salmeterol
21.74Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
21.74Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
21.74Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
21.74Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
21.74Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
21.74Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
21.74Single7YITNalfurafine7YIT-κ-Nalfurafine
21.74Single8JJ8Formoterol8JJ8-β2-Formoterol
21.74Single8JJLOlodaterol8JJL-β2-Olodaterol
21.74Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
21.74Single8JWY2-1188JWY-A2A-2-118
21.74Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
21.74Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.74Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
21.74Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
21.74Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
21.74Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
21.74Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
21.74Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
21.74Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
21.74Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
21.74Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
21.74Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
21.74Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
21.74Consensuslpa_offOrthosteric Ligandlpa1_off
21.74Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
21.62Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
21.43Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
21.43Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
21.43Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
21.43Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
21.43Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
21.43Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
21.43Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
21.43Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
21.43Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
21.43Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
21.43Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.43Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
21.43Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
21.43Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
21.43Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
21.43Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
21.43Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
21.43Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
21.43Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
21.43Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
21.43Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
21.43Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
21.43Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
21.43Consensusvasop-oxy_onOrthosteric Ligandv2_on
21.43Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
21.21Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
21.21Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
21.05Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
21.05Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
21.05Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
21.05Single6AKYMaraviroc6AKY-CCR5-Maraviroc
21.05Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
21.05Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
21.05Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
21.05Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
21.05Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
21.05Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
21.05Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
21.05Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
21.05Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
21.05Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
21.05Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.05Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
21.05Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
21.05Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
21.05Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
21.05Single8GNGIstradefylline8GNG-A2A-Istradefylline
21.05Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
21.05Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
21.05Single8IWESpermidine8IWE-TA9-Spermidine
21.05Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
21.05Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
21.05Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
21.05Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
21.05Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
21.05Single9H2XA1IR19H2X-A2A-A1IR1-Na
21.05Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
21.05Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
21.05Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
21.05Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
21.05Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
21.05Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
21.05Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
21.05Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
21.05Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
20.83Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
20.83Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
20.83Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
20.83Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
20.83Single7EZCUKA7EZC-A2A-UKA
20.83Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
20.83Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
20.83Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.83Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
20.83Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
20.83Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
20.83Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
20.83Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
20.83Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.83Single8XVUCXCL28XVU-CXCR2-CXCL2
20.83Single8XWFCXCL38XWF-CXCR2-CXCL3
20.83Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
20.83Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
20.83Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
20.83Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
20.83Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
20.83Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
20.83Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.83Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
20.83Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
20.83Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
20.69Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.69Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
20.69Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
20.69Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
20.69Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
20.69Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
20.69Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
20.69Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
20.69Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
20.69Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
20.69Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
20.69Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.69Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.69Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
20.00Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
20.00Single3REYXAC3REY-A2A-XAC
20.00Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
20.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
20.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
20.00Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
20.00Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
20.00Single5WF6UK-4320975WF6-A2A-UK-432097
20.00Single5ZTYAM102575ZTY-CB2-AM10257
20.00Single6A94Zotepine6A94-5-HT2A-Zotepine
20.00Single6KNMJN241-96KNM-Apelin-JN241-9
20.00Single6KUXRS-799486KUX-α2a-RS-79948
20.00Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
20.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
20.00Single6PS4ICI118-5516PS4-β2-ICI118-551
20.00Single6PS5S-Propranolol6PS5-β2-S-Propranolol
20.00Single6PT3DPI-2876PT3-δ-DPI-287
20.00Single6TPNHTL66416TPN-OX2-HTL6641
20.00Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
20.00Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
20.00Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
20.00Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
20.00Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
20.00Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
20.00Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
20.00Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
20.00Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
20.00Single7UL3Famotidine7UL3-H2-Famotidine
20.00Single7VV6C48/807VV6-MRGPRX2-C48/80
20.00Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
20.00Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
20.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
20.00Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
20.00Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
20.00Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
20.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
20.00Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
20.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
20.00Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
20.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
20.00Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
20.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
20.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
20.00Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
20.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
20.00Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
20.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
20.00Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
20.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
20.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
20.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
20.00Single8XQJJN2418XQJ-Apelin-JN241
20.00Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
20.00Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
20.00Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
20.00Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
20.00Single9ARXSerotonin9ARX-5-HT2A-Serotonin
20.00Single9IPYJR14a9IPY-C3aB-JR14a
20.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
20.00Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
20.00Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
20.00Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
20.00Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
20.00Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
20.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
20.00Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
20.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
20.00Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.00Consensuskisspeptin_onOrthosteric Ligandkiss1_on
20.00Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
20.00Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
20.00Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
20.00Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
20.00Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
20.00Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
20.00Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
19.35Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
19.35Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
19.35Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
19.35Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
19.35Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
19.35Single9KDFRES-701-39KDF-ETB-RES-701-3
19.23Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
19.23Single4IARErgotamine4IAR-5-HT1B-Ergotamine
19.23Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
19.23Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
19.23Single7F8XNN90567F8X-CCKA-NN9056
19.23Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
19.23Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8IEIA1LYA8IEI-GPR156-A1LYA
19.23Single8IEPA1LYA8IEP-GPR156-A1LYA
19.23Single8IEPA1LYA8IEP-GPR156-A1LYA
19.23Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
19.23Single8KIGSHU91198KIG-MC3-SHU9119-Ca
19.23Single8WKYPG-9348WKY-MC4-PG-934
19.23Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.23Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
19.23Single8XWNCXCL88XWN-CXCR2-CXCL8
19.23Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
19.23Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
19.23Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
19.23Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single9M4TSilodosin9M4T-Alpha1A-Silodosin
19.23Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
19.23Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
19.23Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
19.23Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
19.23Consensuslpl_onOrthosteric Ligands1p_on lpa_on
19.23Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
19.23Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.05Single2Y01Dobutamine2Y01-β1-Dobutamine
19.05Single2Y02Carmoterol2Y02-β1-Carmoterol
19.05Single2Y04Salbutamol2Y04-β1-Salbutamol
19.05Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
19.05Single3NY8ICI118-5513NY8-β2-ICI118-551
19.05Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
19.05Single4EJ4Naltrindole4EJ4-δ-Naltrindole
19.05Single4GBRS-Carazolol4GBR-β2-S-Carazolol
19.05Single4QKX35V4QKX-β2-35V
19.05Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
19.05Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
19.05Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
19.05Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
19.05Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
19.05Single6H7MSalbutamol6H7M-β1-Salbutamol
19.05Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
19.05Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
19.05Single6PS1Timolol6PS1-β2-Timolol
19.05Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
19.05Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
19.05Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
19.05Single7BU7BI1671077BU7-β1-BI167107
19.05Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
19.05Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
19.05Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
19.05Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
19.05Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
19.05Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
19.05Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
19.05Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
19.05Single7V3ZCP559407V3Z-CB1-CP55940
19.05Single7WC7Lisuride7WC7-5-HT2A-Lisuride
19.05Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
19.05Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
19.05Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
19.05Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
19.05Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
19.05Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
19.05Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
19.05Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
19.05Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
19.05Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
19.05Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
19.05Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
19.05Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
19.05Single8JXRLSD8JXR-D1-LSD
19.05Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
19.05Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
19.05Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
19.05Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
19.05Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
19.05Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
19.05Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
19.05Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
19.05Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
19.05Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
19.05Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
19.05Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
19.05Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
19.05Consensus5ht5_onOrthosteric Ligand5ht5a_on
19.05Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
19.05Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
19.05Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
19.05Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
19.05Consensusdopamine_offOrthosteric Ligandd2_off d3_off
19.05Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
19.05Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
19.05Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
19.05Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
18.75Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
18.75Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
18.75Single8IY6Endothelin-18IY6-ETB-Endothelin-1
18.75Single8PWNTheophylline8PWN-A2A-Theophylline
18.75Consensusendothelin_onOrthosteric Ligandetb_on eta_on
18.75Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
18.52Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
18.52Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
18.52Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
18.52Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
18.52Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
18.52Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
18.52Single8IEBA1LYA8IEB-GPR156-A1LYA
18.52Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
18.52Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
18.52Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
18.52Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
18.52Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
18.52Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
18.52Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
18.52Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
18.52Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
18.52Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
18.52Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
18.52Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
18.52Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
18.52Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
18.18Single2RH1S-Carazolol2RH1-β2-S-Carazolol
18.18Single2Y00Dobutamine2Y00-β1-Dobutamine
18.18Single2Y03Isoprenaline2Y03-β1-Isoprenaline
18.18Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
18.18Single5C1MBU725C1M-μ-BU72
18.18Single5GLHEndothelin-15GLH-ETB-Endothelin-1
18.18Single5JQHS-Carazolol5JQH-β2-S-Carazolol
18.18Single5N2RPSB-365N2R-A2A-PSB-36-Na
18.18Single5WIUNemonapride5WIU-D4-Nemonapride
18.18Single5WIVNemonapride5WIV-D4-Nemonapride-Na
18.18Single5XPRBosentan5XPR-ETB-Bosentan
18.18Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
18.18Single6D26Fevipiprant6D26-DP2-Fevipiprant
18.18Single6E67BI1671076E67-β2-BI167107-Gs(CT)
18.18Single6IGKEndothelin-36IGK-ETB-Endothelin-3
18.18Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
18.18Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
18.18Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
18.18Single6PS6Timolol6PS6-β2-Timolol
18.18Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
18.18Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
18.18Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
18.18Single7C61Ergotamine7C61-5-HT1B-Ergotamine
18.18Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
18.18Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
18.18Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
18.18Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
18.18Single7WC6LSD7WC6-5-HT2A-LSD
18.18Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
18.18Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
18.18Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
18.18Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
18.18Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
18.18Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
18.18Single8S4DCMF-0198S4D-Apelin-CMF-019
18.18Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
18.18Single8TF5Oleic acid8TF5-GPR6-Oleic acid
18.18Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
18.18Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
18.18Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
18.18Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
18.18Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
18.18Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
18.18Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
18.18Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
18.18Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
18.18Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
18.18Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
18.18Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
18.18Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
18.18Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
18.18Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
18.18Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
18.18Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
18.18Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
18.18Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
18.18Consensusamine_offonOrthosteric Ligandamine_off amine_on
18.18Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
18.18Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
18.18Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
18.18Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
18.18Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
18.18Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
18.18Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
18.18Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
18.18Consensusdp_offOrthosteric Liganddp2_off
18.18Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
18.18Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
18.18Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Single5WF5UK-4320975WF5-A2A-UK-432097
17.86Single6PT2KGCHM076PT2-δ-KGCHM07
17.86Single6W25SHU91196W25-MC4-SHU9119-Ca
17.86Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
17.86Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
17.86Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
17.86Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
17.86Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
17.86Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
17.86Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
17.86Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
17.86Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
17.86Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.86Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.86Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
17.86Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
17.65Single6TQ9SB-4081246TQ9-OX1-SB-408124
17.65Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
17.65Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
17.65Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
17.65Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
17.65Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
17.65Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
17.65Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
17.65Consensussensory_onOrthosteric Ligandopsins_on
17.39Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
17.39Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
17.39Single5XRAAM115425XRA-CB1-AM11542
17.39Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
17.39Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
17.39Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
17.39Single6H7JIsoprenaline6H7J-β1-Isoprenaline
17.39Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
17.39Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
17.39Single6WGTLSD6WGT-5-HT2A-LSD
17.39Single7B6WCyclazosin7B6W-α1b-Cyclazosin
17.39Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
17.39Single7FEECP559407FEE-CB1-CP55940-ZCZ011
17.39Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
17.39Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
17.39Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
17.39Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
17.39Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
17.39Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
17.39Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
17.39Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
17.39Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
17.39Single8E0GBU728E0G-μ-BU72
17.39Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
17.39Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
17.39Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
17.39Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
17.39Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
17.39Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
17.39Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
17.39Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
17.39Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
17.39Single8ZWFJR14a8ZWF-C3aB-JR14a
17.39Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
17.39Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
17.39Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
17.39Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
17.39Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
17.39Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
17.39Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
17.39Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
17.39Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
17.39Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
17.39Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
17.39Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
17.39Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
17.39Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
17.24Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
17.24Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
17.24Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
17.24Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
17.14Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
17.14Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
16.67Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
16.67Single3UZAGTPL92363UZA-A2A-GTPL9236
16.67Single4AMIBucindolol4AMI-β1-Bucindolol
16.67Single4LDEBI1671074LDE-β2-BI167107
16.67Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
16.67Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
16.67Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
16.67Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
16.67Single6KQICP559406KQI-CB1-CP55940-Org27569
16.67Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
16.67Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
16.67Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
16.67Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
16.67Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
16.67Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
16.67Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
16.67Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
16.67Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
16.67Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
16.67Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
16.67Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
16.67Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
16.67Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
16.67Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
16.67Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
16.67Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
16.67Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
16.67Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
16.67Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
16.67Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
16.67Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
16.67Single8JWZAB9288JWZ-A2A-AB928-Na
16.67Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
16.67Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
16.67Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
16.67Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
16.67Single8XQJJN2418XQJ-Apelin-JN241
16.67Single8XWACXCL18XWA-CXCR2-CXCL1
16.67Single8XWMCXCL68XWM-CXCR2-CXCL6
16.67Single8XWSCXCL58XWS-CXCR2-CXCL5
16.67Single8XYIVUF106618XYI-CXCR3-VUF10661
16.67Single8ZRTET-18ZRT-ETB-ET-1
16.67Single9DGIZ85267113509DGI-CB1-Z8526711350
16.67Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
16.67Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.67Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.67Consensus5ht2_onOrthosteric Ligand5ht2b_on
16.67Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
16.67Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
16.67Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
16.67Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
16.67Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
16.67Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
16.67Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
16.67Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
16.67Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
16.67Consensusgi_sensoryOrthosteric Ligandgi_opsins
16.67Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
16.67Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
16.67Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
16.67Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
16.67Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
16.67Consensuslpl_offOrthosteric Ligands1p_off lpa_off
16.67Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
16.67Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
16.67Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
16.67Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
16.67Consensusorexin_onOrthosteric Ligandox2_on
16.67Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.67Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
16.67Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
16.13Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
16.13Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
16.13Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
16.13Single7SK3CXCL127SK3-ACKR3-CXCL12
16.13Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
16.13Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
16.13Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
16.00Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
16.00Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
16.00Single6H7LDobutamine6H7L-β1-Dobutamine
16.00Single6IBLArformoterol6IBL-β1-Arformoterol
16.00Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
16.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
16.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
16.00Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
16.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
16.00Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
16.00Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
16.00Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
16.00Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
16.00Single8ZPLHF511168ZPL-CXCR4-HF51116
16.00Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
16.00Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
16.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
16.00Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
16.00Consensuscck_onOrthosteric Ligandccka_on cckb_on
16.00Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
16.00Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
16.00Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
16.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
16.00Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
16.00Consensusprostanoid_offOrthosteric Ligandep_off dp_off
15.79Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
15.79Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
15.79Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
15.79Single6TP4ACT-4622066TP4-OX1-ACT-462206
15.79Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
15.79Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
15.79Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
15.79Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
15.79Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
15.79Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.79Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
15.79Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single9AS7Psilocin9AS7-5-HT2A-Psilocin
15.79Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
15.79Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
15.79Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.79Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.62Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
15.62Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
15.62Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
15.38Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
15.38Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
15.38Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
15.38Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
15.38Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
15.38Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
15.38Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
15.38Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
15.38Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
15.38Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
15.38Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
15.38Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
15.15Single6IGLIRL16206IGL-ETB-IRL1620
15.15Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
15.15Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
15.15Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
15.15Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
15.00Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
15.00Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
15.00Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
15.00Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
15.00Single5WS3EMPA5WS3-OX2-EMPA
15.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
15.00Single6AKXA4R6AKX-CCR5-A4R
15.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
15.00Single6TODEMPA6TOD-OX1-EMPA-Na
15.00Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
15.00Single7F8ULintitript7F8U-CCKA-Lintitript
15.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
15.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.00Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
15.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
15.00Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
15.00Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
15.00Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
15.00Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
15.00Single7XRRLemborexant7XRR-OX2-Lemborexant
15.00Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
15.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
15.00Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
15.00Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
15.00Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
15.00Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
15.00Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
15.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
15.00Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
15.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
15.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
15.00Consensusangiotensin_offOrthosteric Ligandat1_off
15.00Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
15.00Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
15.00Consensusorexin_offOrthosteric Ligandox2_off ox1_off
15.00Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
15.00Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
15.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
14.81Single4XT1Fractalkine4XT1-US28-Fractalkine
14.81Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
14.81Single7QA8Peptide7QA8-STE2-Peptide
14.81Single7QA8Peptide7QA8-STE2-Peptide
14.81Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
14.81Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
14.81Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
14.81Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
14.81Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
14.81Single8IEIA1LYA8IEI-GPR156-A1LYA
14.81Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.81Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
14.81Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
14.81Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
14.81Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
14.81Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
14.81Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
14.81Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
14.81Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
14.81Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
14.71Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
14.71Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
14.71Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
14.71Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
14.71Consensusbombesin_onOrthosteric Ligandbb2_on
14.71Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
14.71Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
14.71Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
14.71Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
14.71Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
14.29Single2YDOAdenosine2YDO-A2A-Adenosine
14.29Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
14.29Single4ZJCSB-6740424ZJC-OX1-SB-674042
14.29Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
14.29Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
14.29Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
14.29Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
14.29Single6TPKRetosiban6TPK-OT-Retosiban
14.29Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
14.29Single6V9SGTPL114036V9S-OX1-GTPL11403
14.29Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
14.29Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
14.29Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
14.29Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
14.29Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
14.29Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
14.29Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
14.29Single7F61PF-036547467F61-H3-PF-03654746
14.29Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
14.29Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
14.29Single7SK5CXCL127SK5-ACKR3-CXCL12
14.29Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
14.29Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
14.29Single7XNACYN1548067XNA-SST2-CYN154806
14.29Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
14.29Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
14.29Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
14.29Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
14.29Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
14.29Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.29Single8IYXYL-3658IYX-GPR34-YL-365
14.29Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
14.29Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
14.29Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
14.29Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
14.29Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
14.29Single8RLNLUF58348RLN-A2A-LUF5834
14.29Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
14.29Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
14.29Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
14.29Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
14.29Single9AS3LSD9AS3-5-HT2A-LSD
14.29Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9AS5Mescaline9AS5-5-HT2A-Mescaline
14.29Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
14.29Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
14.29Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
14.29Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
14.29Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
14.29Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
14.29Consensusalpha1_onOrthosteric Ligandalpha1a_on
14.29Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
14.29Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
14.29Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
14.29Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
14.29Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
14.29Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
14.29Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
14.29Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
14.29Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
14.29Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
14.29Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
14.29Consensusopsins_offOrthosteric Ligandrhodopsin_off
14.29Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
14.29Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
14.29Consensussensory_offOrthosteric Ligandopsins_off
14.29Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
14.29Consensusvasop-oxy_offOrthosteric Ligandot_off
13.89Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
13.89Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
13.79Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
13.79Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
13.79Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
13.79Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
13.79Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.79Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
13.79Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
13.79Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
13.79Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
13.79Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
13.64Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
13.64Single4YAYZD-71554YAY-AT1-ZD-7155
13.64Single6D27CAY104716D27-DP2-CAY10471
13.64Single6DRXLisuride6DRX-5-HT2B-Lisuride
13.64Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
13.64Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
13.64Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
13.64Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
13.64Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
13.64Single7UL4Alvimopan7UL4-μ-Alvimopan
13.64Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
13.64Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
13.64Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
13.64Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
13.64Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
13.64Single8JJOAlprenolol8JJO-β2-Alprenolol
13.64Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
13.64Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
13.64Single8T1WCVN4248T1W-GPR6-CVN424
13.64Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
13.64Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
13.64Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
13.64Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
13.64Single8X64Desloratadine8X64-H1-Desloratadine
13.64Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
13.64Single9AS1DMT9AS1-5-HT2A-DMT
13.64Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
13.64Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
13.64Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
13.64Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
13.64Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
13.64Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
13.64Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
13.64Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
13.64Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
13.64Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
13.64Consensusblt_onOrthosteric Ligandblt1_on
13.64Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
13.64Consensuscck_offOrthosteric Ligandccka_off
13.64Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
13.64Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
13.64Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
13.64Consensusleukotriene_onOrthosteric Ligandblt_on
13.64Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
13.33Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
13.33Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
13.33Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
13.33Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
13.33Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
13.33Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
13.33Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
13.16Consensuspth_onOrthosteric Ligandpth1_on pth2_on
13.04Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
13.04Single5WQCEMPA5WQC-OX2-EMPA
13.04Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
13.04Single6LUQHaloperidol6LUQ-D2-Haloperidol
13.04Single6TP6Filorexant6TP6-OX1-Filorexant
13.04Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
13.04Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
13.04Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
13.04Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
13.04Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
13.04Single7SINNPS-21437SIN-CaS-NPS-2143
13.04Single7SINNPS-21437SIN-CaS-NPS-2143
13.04Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
13.04Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
13.04Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
13.04Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
13.04Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
13.04Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
13.04Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
13.04Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
13.04Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
13.04Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
13.04Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
13.04Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
13.04Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
13.04Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
13.04Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
13.04Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
13.04Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
13.04Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.04Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.04Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
13.04Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.04Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
12.90Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
12.90Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
12.90Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
12.90Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
12.90Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
12.90Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
12.90Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
12.90Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
12.50Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
12.50Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
12.50Single4U15Tiotropium4U15-M3-Tiotropium
12.50Single4XT3Fractalkine4XT3-US28-Fractalkine
12.50Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
12.50Single5MZPCaffeine5MZP-A2A-Caffeine-Na
12.50Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
12.50Single6OL9Tiotropium6OL9-M5-Tiotropium
12.50Single6OS1TRV0266OS1-AT1-TRV026
12.50Single6TQ7SB-3348676TQ7-OX1-SB-334867
12.50Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
12.50Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
12.50Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
12.50Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
12.50Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
12.50Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
12.50Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
12.50Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
12.50Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
12.50Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
12.50Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
12.50Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
12.50Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
12.50Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
12.50Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
12.50Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
12.50Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
12.50Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
12.50Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
12.50Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.50Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
12.50Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
12.50Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
12.50Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.50Single8XVLZibotentan8XVL-ETA-Zibotentan
12.50Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
12.50Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
12.50Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
12.50Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
12.50Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.50Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
12.50Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
12.50Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
12.50Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
12.50Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
12.50Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
12.50Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
12.50Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
12.12Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
12.12Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
12.12Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
12.12Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
12.12Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
12.12Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
12.12Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
12.12Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
12.12Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
12.12Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
12.12Consensusglp_onOrthosteric Ligandglp1_on glp2_on
12.12Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
12.00Single4XEENeurotensin4XEE-NTS1-Neurotensin
12.00Single4XESNeurotensin4XES-NTS1-Neurotensin
12.00Single5CXVTiotropium5CXV-M1-Tiotropium
12.00Single6A93Risperidone6A93-5-HT2A-Risperidone
12.00Single6CM4Risperidone6CM4-D2-Risperidone
12.00Single6OS2TRV0266OS2-AT1-TRV026
12.00Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
12.00Single6YVRNTS8-136YVR-NTS1-NTS8-13
12.00Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
12.00Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
12.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
12.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
12.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
12.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
12.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
12.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
12.00Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
12.00Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
12.00Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
12.00Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
12.00Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
12.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
12.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
12.00Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
12.00Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
12.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
12.00Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
12.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
12.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
12.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
12.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
12.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
12.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
12.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
11.90Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
11.76Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
11.76Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
11.76Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
11.76Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
11.76Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
11.76Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
11.76Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
11.76Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
11.76Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
11.76Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
11.76Single7WC4Serotonin7WC4-5-HT2A-Serotonin
11.76Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.76Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
11.76Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
11.76Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
11.76Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
11.76Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
11.76Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.76Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
11.76Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
11.54Single4BUONeurotensin4BUO-NTS1-Neurotensin
11.54Single5X93K-87945X93-ETB-K-8794
11.54Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
11.54Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
11.54Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
11.54Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
11.54Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
11.54Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
11.54Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
11.54Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
11.54Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
11.54Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
11.54Single8XVJMacitentan8XVJ-ETA-Macitentan
11.54Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
11.54Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
11.54Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
11.54Consensusendothelin_offOrthosteric Ligandetb_off
11.54Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
11.43Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
11.11Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
11.11Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
11.11Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
11.11Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
11.11Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
11.11Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
11.11Single7SK9CCX6627SK9-ACKR3-CCX662
11.11Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
11.11Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
11.11Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
11.11Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
11.11Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
11.11Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8X5YAstemizole8X5Y-H1-Astemizole
11.11Single9CHUNoradrenaline9CHU-β2-Noradrenaline
11.11Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
11.11Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
11.11Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
11.11Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
11.11Consensusp2y_offOrthosteric Ligandp2y1_off
10.81Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
10.81Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
10.81Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
10.81Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
10.81Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
10.81Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
10.71Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
10.71Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
10.71Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
10.71Consensussomatostatin_offOrthosteric Ligandsst2_off
10.53Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
10.53Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
10.53Single4XNWMRS25004XNW-P2Y1-MRS2500
10.53Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
10.53Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
10.53Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
10.53Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
10.53Single7WC5Psilocin7WC5-5-HT2A-Psilocin
10.53Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
10.53Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
10.53Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
10.53Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
10.53Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
10.53Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
10.53Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
10.53Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
10.53Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
10.53Single9LRCHistamine9LRC-H4-Histamine
10.53Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
10.53Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
10.53Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
10.53Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
10.53Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
10.34Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
10.34Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
10.34Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
10.26Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
10.26Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
10.26Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
10.00Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
10.00Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
10.00Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
10.00Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
10.00Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
10.00Single3OE9IT1t3OE9-CXCR4-IT1t
10.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
10.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
10.00Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
10.00Single7SRQLSD7SRQ-5-HT2B-LSD
10.00Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
10.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
10.00Single7UL2SR486927UL2-NTS1-SR48692-Na
10.00Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
10.00Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
10.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
10.00Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
10.00Single8K5BNiacin8K5B-HCA2-Niacin
10.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
10.00Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
10.00Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
10.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
10.00Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
10.00Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
10.00Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
10.00Single9B9Y7DY9B9Y-CB1-7DY
10.00Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
10.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
10.00Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
10.00Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
10.00Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
10.00Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
10.00Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
10.00Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
10.00Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
10.00Consensusgq_nucleotideOrthosteric Ligandgq_p2y
10.00Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.00Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.00Consensusneurotensin_offOrthosteric Ligandnts1_off
10.00Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
9.76Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
9.68Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
9.68Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
9.68Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
9.68Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
9.68Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
9.68Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
9.68Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
9.52Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
9.52Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
9.52Single4BWBNeurotensin4BWB-NTS1-Neurotensin
9.52Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
9.52Single4S0VSuvorexant4S0V-OX2-Suvorexant
9.52Single6B73MP11046B73-κ-MP1104
9.52Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
9.52Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
9.52Single6TPJSuvorexant6TPJ-OX2-Suvorexant
9.52Single7BR3Elagolix7BR3-GnRH1-Elagolix
9.52Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
9.52Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
9.52Single7F8YDevazepide7F8Y-CCKA-Devazepide
9.52Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
9.52Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
9.52Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
9.52Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
9.52Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
9.52Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
9.52Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
9.52Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
9.52Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
9.52Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
9.52Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
9.52Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
9.52Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
9.52Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
9.52Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
9.52Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
9.52Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
9.52Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
9.52Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
9.52Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
9.52Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
9.52Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
9.52Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
9.52Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
9.52Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
9.52Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
9.52Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
9.52Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
9.52Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
9.52Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
9.52Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
9.52Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
9.52Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
9.52Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
9.52Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
9.52Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
9.52Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
9.52Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
9.52Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.52Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
9.52Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
9.52Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
9.38Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
9.38Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
9.38Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
9.38Consensuspac_onOrthosteric Ligandpac1_on
9.38Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
9.09Single3RZECidoxepin3RZE-H1-Cidoxepin
9.09Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
9.09Single6FJ3PTH6FJ3-PTH1-PTH
9.09Single6IQLL7458706IQL-D4-L745870
9.09Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
9.09Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
9.09Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
9.09Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
9.09Single6TP3Nemorexant6TP3-OX1-Nemorexant
9.09Single6TPGEMPA6TPG-OX2-EMPA
9.09Single6VI4JDTic6VI4-κ-JDTic
9.09Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
9.09Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
9.09Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
9.09Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
9.09Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
9.09Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
9.09Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
9.09Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
9.09Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
9.09Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
9.09Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
9.09Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
9.09Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.09Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
9.09Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
9.09Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
9.09Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
9.09Single8K5CAcipimox8K5C-HCA2-Acipimox
9.09Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
9.09Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
9.09Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
9.09Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8ZPNAMD31008ZPN-CXCR4-AMD3100
9.09Single9BA0A1AKN9BA0-CB1-A1AKN
9.09Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
9.09Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
9.09Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
9.09Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
9.09Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
9.09Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
9.09Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
9.09Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
9.09Consensusgrh_offOrthosteric Ligandgnrh1_off
9.09Consensushca_onOrthosteric Ligandhca2_on
9.09Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.09Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
9.09Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
9.09Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
9.09Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
8.89Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
8.82Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
8.82Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
8.82Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
8.82Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
8.82Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
8.82Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
8.82Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
8.70Single4DAJTiotropium4DAJ-M3-Tiotropium
8.70Single4MQSIperoxo4MQS-M2-Iperoxo
8.70Single4QIMANTA XV4QIM-SMO-ANTA XV
8.70Single4U14Tiotropium4U14-M3-Tiotropium
8.70Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
8.70Single5DSGTiotropium5DSG-M4-Tiotropium
8.70Single5TGZAM65385TGZ-CB1-AM6538
8.70Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
8.70Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
8.70Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
8.70Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
8.70Single6TOTLemborexant6TOT-OX1-Lemborexant
8.70Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.70Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
8.70Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
8.70Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
8.70Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
8.70Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
8.70Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
8.70Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
8.70Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
8.70Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
8.70Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
8.70Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
8.70Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
8.70Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
8.70Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
8.70Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
8.70Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
8.70Single8X63Mepyramine8X63-H1-Mepyramine
8.70Single8Y73MPAM-158Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
8.70Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
8.70Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
8.70Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
8.70Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
8.70Single9JEAAtropine9JEA-M1-Atropine
8.70Consensusalpha2_onOrthosteric Ligandalpha2b_on
8.70Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
8.70Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
8.70Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
8.70Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
8.70Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
8.70Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
8.70Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
8.70Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
8.70Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
8.70Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
8.70Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
8.70Consensushca_on_gpOrthosteric Ligandhca2_on_gp
8.70Consensushistamine_offOrthosteric Ligandh1_off
8.70Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
8.70Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
8.70Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
8.70Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
8.57Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
8.57Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
8.57Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
8.57Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
8.57Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
8.57Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
8.57Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
8.57Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
8.57Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
8.33Single4JKVTaladegib4JKV-SMO-Taladegib
8.33Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
8.33Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
8.33Single6Z4SSR486926Z4S-NTS1-SR48692
8.33Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
8.33Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
8.33Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
8.33Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
8.33Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
8.33Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
8.33Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
8.33Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
8.33Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
8.33Single9B9ZA1AKO9B9Z-CB1-A1AKO
8.33Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
8.33Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
8.33Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
8.33Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
8.33Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
8.33Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
8.33Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
8.00Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
8.00Single4BV0Neurotensin4BV0-NTS1-Neurotensin
8.00Single4DJHJDTic4DJH-κ-JDTic
8.00Single5V56TC1145V56-SMO-TC114
8.00Single5V57TC1145V57-SMO-TC114
8.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
8.00Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
8.00Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
8.00Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
8.00Single7R0CAVP7R0C-V2-AVP-Arrestin2
8.00Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
8.00Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
8.00Single8EA0Iperoxo8EA0-M3-Iperoxo
8.00Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
8.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
8.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
8.00Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
8.00Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
8.00Single9AS9RS130-1809AS9-5-HT2A-RS130-180
8.00Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
8.00Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
8.00Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Consensusneurotensin_onOrthosteric Ligandnts1_on
8.00Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
7.89Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
7.69Single4N4WSANT-14N4W-SMO-SANT-1
7.69Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
7.69Single6ZG4HTL00099366ZG4-M1-HTL0009936
7.69Single7DFPSpiperone7DFP-D2-Spiperone
7.69Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
7.69Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
7.69Single7K15MKD0467K15-BLT1-MKD046-Na
7.69Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
7.69Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
7.69Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
7.69Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
7.69Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
7.69Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
7.69Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
7.69Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
7.69Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
7.69Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
7.41Single6K1QIRL25006K1Q-ETB-IRL2500
7.41Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
7.41Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
7.41Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
7.41Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
7.41Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
7.41Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
7.14Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
6.90Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
6.90Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
6.90Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
6.90Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
6.67Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
6.67Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
6.67Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
6.45Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
6.25Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
6.25Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
6.25Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
6.25Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
6.25Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
6.25Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
6.25Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
6.06Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
6.06Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
6.06Consensuscalcitonin_onOrthosteric Ligandctlike_on
5.88Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
5.88Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
5.88Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
5.88Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
5.71Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
5.71Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
5.71Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
5.56Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
5.56Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
5.56Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
5.26Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
5.26Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
5.26Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
5.26Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
5.26Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
5.26Single8IKGQ2B8IKG-CB1-Q2B-Gi1/β1/γ1
5.26Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
5.26Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
5.26Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
5.26Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
5.00Single3OE6IT1t3OE6-CXCR4-IT1t
5.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
5.00Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
5.00Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
5.00Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
5.00Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
5.00Single8WG8Peptide8WG8-Glucagon-Peptide-chim(NtGi1-Gs)/β1/γ2
4.76Single4O9RCyclopamine4O9R-SMO-Cyclopamine
4.76Single5L7IVismodegib5L7I-SMO-Vismodegib
4.76Single6LI0C176LI0-GPR52-C17
4.76Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
4.76Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
4.76Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
4.76Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
4.76Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
4.76Single8IKHQ2L8IKH-CB1-Q2L-Gi1/β1/γ1
4.76Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.76Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
4.76Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.76Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.76Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
4.76Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
4.76Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
4.76Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
4.55Single3ODUIT1t3ODU-CXCR4-IT1t
4.55Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
4.55Single4QINSAG1.54QIN-SMO-SAG1.5
4.55Single5U09Taranabant5U09-CB1-Taranabant
4.55Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
4.55Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
4.55Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7WV9ZCZ0117WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
4.55Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
4.55Single8G94CD698G94-S1P1-CD69-Gi1/β1/γ2
4.55Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
4.55Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
4.55Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8Y0HVUF114188Y0H-CXCR3-VUF11418
4.55Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
4.55Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
4.55Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
4.55Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
4.44Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
4.35Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
4.35Single6FFIMMPEP6FFI-mGlu5-MMPEP
4.35Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
4.35Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
4.35Single6ZINSR486926ZIN-NTS1-SR48692
4.35Single7VODCariprazine7VOD-5-HT2A-Cariprazine
4.35Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
4.35Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
4.35Single8IHKAcifran8IHK-HCA3-Acifran
4.35Single8K2WAMG4878K2W-CXCR3-AMG487
4.35Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.35Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
4.35Single8ZPMAMD0708ZPM-CXCR4-AMD070
4.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
4.35Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
4.35Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
4.35Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
4.35Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
4.17Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
4.17Single5DHGC-355DHG-NOP-C-35
4.17Single5DHHSB-6121115DHH-NOP-SB-612111
4.17Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
4.17Single5T04Neurotensin5T04-NTS1-Neurotensin
4.17Single6FFHFenobam6FFH-mGlu5-Fenobam
4.17Single6GPSMK08126GPS-CCR2-MK0812
4.17Single6IIVDaltroban6IIV-TXA2-Daltroban
4.17Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
4.17Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
4.17Single7F83PF-051904577F83-Ghrelin-PF-05190457
4.17Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
4.17Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
4.17Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
4.17Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
4.17Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
4.17Single8K5DGSK2560738K5D-HCA2-GSK256073
4.17Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
4.17Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
4.17Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
4.17Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
4.00Single5CGCHTL142425CGC-mGlu5-HTL14242
4.00Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
4.00Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
4.00Single6GPXMK08126GPX-CCR2-MK0812
4.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
4.00Single7C4SS1P7C4S-S1P3-S1P
4.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
4.00Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
4.00Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
4.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
4.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.00Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.00Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.00Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
4.00Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
4.00Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
4.00Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
4.00Consensusblt_offOrthosteric Ligandblt1_off
4.00Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
4.00Consensusep_offOrthosteric Ligandep4_off
4.00Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
3.85Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
3.85Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
3.85Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.85Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.85Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.85Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
3.85Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
3.85Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
3.85Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
3.70Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
3.70Single6IIURamatroban6IIU-TXA2-Ramatroban
3.70Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
3.70Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
3.70Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
3.70Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
3.57Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
3.57Single5CGDHTL142425CGD-mGlu5-HTL14242
3.57Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
3.57Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
3.57Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.57Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
3.57Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
3.57Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
3.45Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
3.45Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
3.33Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
3.33Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
3.23Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
2.78Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
2.70Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2

Consensus Members
Id Members
8J22 8J22-FFA2-TUG-1375-Gi1/β1/γ2
Net Summary
Imin 1.86
Number of Linked Nodes 853
Number of Links 1159
Number of Hubs 226
Number of Links mediated by Hubs 786
Number of Communities 17
Number of Nodes involved in Communities 334
Number of Links involved in Communities 546
Path Summary
Number Of Nodes in MetaPath 88
Number Of Links MetaPath 87
Number of Shortest Paths 12355893
Length Of Smallest Path 3
Average Path Length 34.7266
Length of Longest Path 61
Minimum Path Strength 1.13
Average Path Strength 4.52903
Maximum Path Strength 20.68
Minimum Path Correlation 0.7
Average Path Correlation 0.997601
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.63158
Average % Of Corr. Nodes 33.8521
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 61.2207
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
ffa_on_gpffa2_on_gp
ffa3_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download ffa2_on_gp.zip



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