Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.43 3.2475409
2G.S1.06 6.295418
3G.S1.07 4.62418
4G.s1h1.05 3.31419
5G.H1.01 4.45167619
6G.H1.04 4.7775417
7G.H1.08 6.325409
8G.S2.01 3.974519
9G.S3.03 6.69333608
10G.S3.04 7.895417
11G.S3.06 8.86517
12G.s3h2.03 4.675619
13G.H2.06 6.55333619
14G.H2.07 6.065619
15G.H2.10 5.34518
16G.h2s4.01 8.38333619
17G.S4.02 4.374518
18G.S4.03 4.7175417
19G.S4.05 4.3625417
20G.s4h3.03 5.305418
21G.H3.09 6.1619
22G.H3.13 9.15333616
23G.H3.17 10.745615
24G.S5.03 4.556519
25G.S5.04 5.18419
26G.S5.05 5.78819
27G.S5.06 4.982518
28G.S5.07 5.4409
29G.s5hg.01 6.222509
30G.HG.01 8.834516
31G.HG.03 4.2025406
32G.HG.15 6.2525417
33G.hgh4.01 8.0175406
34G.hgh4.05 7.546516
35G.hgh4.11 3.5275415
36G.hgh4.21 7.9954174
37G.H4.03 3.46754174
38G.H4.07 9.95415
39G.H4.08 7.272513
40G.H4.10 9.386517
41G.H4.11 4.084518
42G.H4.12 7.26833614
43G.H4.15 8.6525418
44G.H4.16 4.9414
45G.h4s6.02 4.1725417
46G.h4s6.20 6.355494
47G.S6.02 7.31833698
48G.S6.05 9.644515
49G.s6h5.01 7.12419
50G.H5.03 6.39519
51G.H5.06 9.9475414
52G.H5.07 3.924519
53G.H5.08 5.7185158
54G.H5.13 11.8875498
55G.H5.15 5.605448
56G.H5.20 3.7125408
57G.H5.25 4.0025408
58b.1x4 4.824108
59b.1x15 4.115417
60b.1x19 5.6875416
61b.h2x1 5.4625405
62b.h2x4 3.46573
63b.lhb1x3 4.808572
64b.lhb1x6 4.86333673
65b.lhb1x11 4.075484
66b.l1x3 10.2975459
67b.l1x7 3.576559
68b.b2x3 4.8556
69b.b2x5 7.21667657
70b.b3x1 4.808535
71b.b3x3 5.054538
72b.l3x1 7.4925419
73b.l3x2 7.706559
74b.b4x3 4.516537
75b.b4x4 6.712558
76b.b4x5 4.78167637
77b.b4x6 9.745659
78b.b4x7 8.64438
79b.l4x2 13.8625434
80b.b5x2 7.3975407
81b.b5x3 8.01559
82b.b5x7 5.405437
83b.l5x1 5.025438
84b.l5x5 10.205619
85b.b6x3 3.4275438
86b.b6x5 5.42736
87b.l6x5 7.9475414
88b.b7x1 6.6975414
89b.b7x2 4.27438
90b.l7x2 4.71419
91b.l7x4 5.435419
92b.b8x3 3.64667616
93b.b8x4 4.674536
94b.l8x1 3.8125435
95b.l8x3 2.93403
96b.l8x8 6.06434
97b.b9x4 7.7475409
98b.l9x3 7.175619
99b.l9x6 6.09718
100b.l9x7 4.465417
101b.b10x5 6.844519
102b.l10x1 3.9575463
103b.b11x2 5.49417
104b.b11x3 4.575465
105b.b11x4 5.785419
106b.b11x5 4.8225466
107b.l11x2 9.7525419
108b.b12x3 4.302568
109b.b12x6 9.968518
110b.b13x3 5.75504
111b.b13x7 9.196567
112b.l13x3 6.35143769
113b.l13x6 6.53419
114b.l13x7 5.364569
115b.b14x3 4.746565
116b.b15x1 8.66167669
117b.b15x3 4.478569
118b.l15x1 5.9125417
119b.l15x2 6.8875409
120b.b16x4 11.94466
121b.b16x5 4.6625405
122b.b16x6 8.68714768
123b.b17x5 8.0825417
124b.b17x7 8.5225418
125b.l17x3 9.01833619
126b.l17x6 8.994519
127b.b18x3 4.692518
128b.l18x1 7.0445126
129b.l18x2 5.30754127
130b.b19x2 9.062516
131b.b19x4 5.9175418
132b.l19x1 6.14419
133b.l19x2 8.244519
134b.b20x2 7.0175416
135b.b20x4 9.348518
136b.b20x6 9.2425416
137b.b20x7 6.385409
138b.b21x1 9.8725417
139b.b21x7 6.96605
140b.b22x5 7.054127
141b.l22x5 7.46667679
142b.b23x2 6.6725406
143b.b23x6 7.6285137
144b.l23x1 6.6575416
145b.b24x3 5.09485
146b.b24x4 7.8065136
147b.b24x6 8.44254138
148b.l24x2 6.098576
149b.l24x3 5.73405
150b.b25x3 6.07754135
151b.l25x3 8.832589
152b.l25x6 12.206518
153b.b27x3 5.4175408
154b.l27x1 9.56286719
155b.l27x2 9.4325489
156b.b28x3 4.434557
157b.b28x4 6.502586
158b.b28x6 8.405689
159g.h1x8 4.6825107
160g.h1x12 6.224106
161g.h2x11 11.84126
162g.ctx3 5.816579
163g.ctx4 3.8725407
164g.ctx6 3.47676
165g.ctx15 7.81439
166g.ctx16 4.89838
167Lig 8.490771320
1681x43 4.1775407
1691x46 3.14333628
1701x50 7.652509
171I1x50 7.45448
1722x39 4.196548
1732x42 7.9525408
1742x46 5.398529
1752x50 9.0975409
1762x56 4.455408
1772x57 4.84528
1782x60 9.596528
179E1x50 7.664148
1803x24 4.24754144
1813x37 6.5575428
1823x41 5.235427
1833x42 6.6425429
1843x43 5.2275429
1853x46 5.335429
1863x50 6.3429
1873x51 5.33408
1883x54 3.115408
189I2x53 7.536548
1904x42 4.02448
1914x50 4.424529
192E2.R180 3.385403
1935x39 6.27286708
1945x47 9.21629
1955x50 4.055409
1965x54 6.0525428
1975x58 6.945629
1985x68 8.084597
1996x37 3.398508
2006x44 5.892529
2016x48 7.25829
2026x51 12.0775428
2036x52 10.974528
2046x55 10.76427
205E3.V377 3.14754115
2067x33 3.87754116
2077x42 9.338528
2087x49 8.865429
2097x53 5.20857729
2108x50 8.35833648
2118x54 4.575448
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b26x1 b.l27x1 25.88453.71NoYes099
2G.H3.17 b.l27x1 13.07443.75YesYes159
3G.H3.15 G.H3.17 19.88084.52NoYes085
4G.H3.15 G.H3.18 19.97028.24NoNo089
5G.H3.18 G.S4.02 21.78114.28NoYes098
6G.S1.07 G.S4.02 26.46592.85YesYes188
7G.S1.07 G.s1h1.01 1001.71YesNo189
8G.H1.01 G.s1h1.01 62.77633.49YesNo199
9G.H1.01 G.S1.06 25.38335.64YesYes198
10G.S1.06 G.S4.03 25.07532.85YesYes187
11b.b2x1 b.l27x1 14.06516.75NoYes189
12G.H2.10 b.b2x1 14.03376.72YesNo188
13G.H2.10 G.h2s4.01 12.84014.19YesYes189
14G.S1.05 G.h2s4.01 69.409719.49NoYes199
15G.S1.05 G.S1.07 67.466211.07NoYes198
16G.S4.05 G.S5.05 73.00965.24YesYes179
17G.H1.01 G.S4.05 37.21954.55YesYes197
18G.S4.05 G.s1h1.05 37.23943.23YesYes179
19G.s1h1.01 G.s1h1.05 37.25213.71NoYes199
20G.H2.07 G.h2s4.01 53.75114.01YesYes199
21G.H2.06 b.l17x6 21.45449.68YesYes199
22G.H2.06 b.l9x6 43.06723.58YesYes198
23G.H2.06 b.l19x1 21.35285.53YesYes199
24G.S5.03 G.S5.05 36.50633.77YesYes199
25G.S4.03 G.S5.03 18.06714.42YesYes179
26G.S4.02 G.S5.02 12.03724.61YesNo186
27G.H3.09 G.S5.04 12.80677.31YesYes199
28G.S5.04 G.S5.06 12.42214.15YesYes198
29G.H5.10 G.S5.03 54.45238.4NoYes079
30G.H5.10 G.S6.02 90.601614.94NoYes078
31G.S6.02 G.h4s6.20 84.96543.97YesYes984
32G.S5.05 G.S6.04 36.40816.79YesNo199
33G.H5.10 G.S6.04 36.38018.82NoNo079
34G.H5.26 G.h4s6.20 83.61385.16NoYes084
35G.H5.20 G.H5.26 83.38574.87YesNo088
36G.H5.20 G.H5.25 80.83784.15YesYes088
375x58 6x37 76.84387.03YesYes098
386x37 G.H5.25 78.23844.15YesYes088
39b.l17x5 b.l17x6 22.72924.42NoYes169
40b.l17x5 b.l19x2 43.79832.94NoYes169
41b.l17x3 b.l19x2 27.307911.35YesYes199
42b.b19x4 b.l17x3 15.0039.58YesYes189
43b.b19x4 b.b20x6 10.45276.49YesYes186
44b.l17x5 b.l19x1 21.272.94NoYes169
45b.l17x3 b.l17x7 11.97179.28YesNo197
46b.b15x4 b.l17x7 11.81265.29NoNo067
47b.b15x4 b.l13x3 11.59643.18NoYes069
48b.b4x7 b.l4x2 14.31583.45YesYes384
49b.l4x2 g.ctx16 13.71926.19YesYes348
50b.b26x2 b.b2x3 18.9964.86NoYes076
51b.l4x1 g.ctx16 15.01735.28NoYes058
52b.b3x1 b.b4x7 14.31974.07YesYes358
53b.b6x5 b.l6x4 13.44072.9YesNo065
54b.l6x3 b.l6x4 13.84383.71NoNo065
55b.b7x1 b.b8x3 16.32143.63YesYes146
56b.b12x6 b.l9x3 18.71564.23YesYes189
57b.l11x1 b.l9x6 19.77127.24NoYes198
58b.b11x6 b.l11x1 21.1153.71NoNo199
59b.b11x6 b.l9x3 20.2912.55NoYes199
60b.b19x6 b.l19x2 14.644110.31NoYes199
61b.b19x5 b.b19x6 15.38793.71NoNo059
62b.b20x3 b.b21x7 11.37194.03NoYes085
63b.b20x3 b.l21x9 11.54764.91NoNo086
64b.b19x5 b.l21x9 14.80435.29NoNo056
653x36 Lig 18.47335.16NoYes080
663x36 6x48 18.72153.92NoYes089
676x44 6x48 44.8214.01YesYes299
685x54 6x44 71.23428.71YesYes289
695x54 5x58 71.59923.59YesYes289
706x52 Lig 36.740810.29YesYes280
716x48 6x52 24.52735.01YesYes298
725x47 6x52 24.25221.43YesYes298
735x47 6x44 25.68917.5YesYes299
743x32 Lig 19.658819.41NoYes290
752x56 3x32 18.93855.84YesNo089
762x56 3x28 16.71164.47YesNo087
772x59 3x28 15.95286.92NoNo067
782x59 3x24 15.19394.15NoYes064
793x21 3x24 11.39823NoYes074
805x40 6x55 15.854912.45NoYes077
815x37 6x59 12.33591.38NoNo067
825x40 6x59 14.09793.39NoNo077
835x37 E3.P373 10.573812.97NoNo061
84b.b2x5 b.l4x1 15.17754.94YesNo075
85b.b26x1 b.b26x2 19.1625.16NoNo097
86G.H2.07 b.l9x6 55.55693.86YesYes198
87b.b2x3 b.b2x5 17.92934.65YesYes567
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
2x60Lig4.752YesYes8010
3x29Lig6.430NoYes7010
3x32Lig19.412NoYes9010
3x33Lig9.680NoYes9010
3x36Lig5.160NoYes8010
5x43Lig5.860NoYes9010
5x44Lig2.932NoYes8010
5x461Lig3.92NoYes8010
6x51Lig14.252YesYes8010
6x52Lig10.292YesYes8010
6x55Lig11.72YesYes7010
7x38Lig3.832NoYes6010
7x42Lig12.192YesYes8010
2x532x564.470NoYes8822
2x537x425.860NoYes8821
2x563x325.840YesNo8921
2x577x428.212YesYes8821
2x602x649.332YesNo8612
2x607x386.492YesNo8611
2x607x3915.032YesNo8812
2x607x4212.382YesYes8811
2x647x3914.172NoNo6822
3x29E2x525.650NoNo7712
3x327x428.052NoYes9811
3x334x573.390NoNo9912
3x335x393.790NoYes9812
3x366x483.920NoYes8912
3x374x566.352YesNo8822
3x375x4619.592YesNo8821
4x565x4614.852NoNo8821
5x39E2x525.860YesNo8722
5x40E2x522.980NoNo7722
5x395x4313.990YesNo8921
5x406x5512.450NoYes7721
5x446x525.282NoYes8811
5x446x554.182NoYes8711
5x476x483.012YesYes9922
5x476x5221.432YesYes9821
6x486x525.012YesYes9821
6x516x5212.862YesYes8811
6x516x5514.712YesYes8711
6x517x386.492YesNo8611

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
92.31Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
78.57Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
76.92Single6TPGEMPA6TPG-OX2-EMPA
76.92Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
76.92Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
76.92Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
76.92Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
73.33Single6H7JIsoprenaline6H7J-β1-Isoprenaline
73.33Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
73.33Single6TQ7SB-3348676TQ7-OX1-SB-334867
73.33Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
73.33Single8E0GBU728E0G-μ-BU72
73.33Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
73.33Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
73.33Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
73.33Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
73.33Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
71.43Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
71.43Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
71.43Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
71.43Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
71.43Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
71.43Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
71.43Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
71.43Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
71.43Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
71.43Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
71.43Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
71.43Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
71.43Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
71.43Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
71.43Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
71.43Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
71.43Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
71.43Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
71.43Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
69.23Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
69.23Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
68.75Single4LDEBI1671074LDE-β2-BI167107
68.75Single7YITNalfurafine7YIT-κ-Nalfurafine
68.75Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
68.75Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
68.75Consensusalpha1_offOrthosteric Ligandalpha1a_off
68.75Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
68.75Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
68.75Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
68.75Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
66.67Single2RH1S-Carazolol2RH1-β2-S-Carazolol
66.67Single2Y03Isoprenaline2Y03-β1-Isoprenaline
66.67Single5C1MBU725C1M-μ-BU72
66.67Single5JQHS-Carazolol5JQH-β2-S-Carazolol
66.67Single5WQCEMPA5WQC-OX2-EMPA
66.67Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
66.67Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
66.67Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
66.67Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
66.67Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
66.67Single7WC6LSD7WC6-5-HT2A-LSD
66.67Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
66.67Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
66.67Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
66.67Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
66.67Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
66.67Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
66.67Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
66.67Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
66.67Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
66.67Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
66.67Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
66.67Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
66.67Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
66.67Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
66.67Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
66.67Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
66.67Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
66.67Consensusamine_offonOrthosteric Ligandamine_off amine_on
66.67Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
66.67Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
66.67Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
66.67Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
66.67Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
66.67Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
66.67Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
64.71Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
64.71Single5X93K-87945X93-ETB-K-8794
64.71Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
64.71Consensusendothelin_offOrthosteric Ligandetb_off
64.71Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
64.29Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
64.29Single4ZJCSB-6740424ZJC-OX1-SB-674042
64.29Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
64.29Single6PS0S-Carazolol6PS0-β2-S-Carazolol
64.29Single6PS4ICI118-5516PS4-β2-ICI118-551
64.29Single6PS5S-Propranolol6PS5-β2-S-Propranolol
64.29Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
64.29Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
64.29Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
64.29Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
64.29Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
64.29Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
64.29Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
64.29Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
64.29Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
64.29Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
64.29Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
64.29Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
64.29Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
64.29Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
64.29Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
64.29Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
64.29Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
64.29Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
64.29Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
64.29Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
64.29Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
64.29Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
64.29Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
64.29Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
64.29Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
64.29Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
64.29Consensusalpha1_onOrthosteric Ligandalpha1a_on
64.29Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
64.29Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
64.29Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
64.29Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
63.16Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
62.50Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
62.50Single5D5AS-Carazolol5D5A-β2-S-Carazolol
62.50Single5D5BS-Carazolol5D5B-β2-S-Carazolol
62.50Single6WGTLSD6WGT-5-HT2A-LSD
62.50Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
62.50Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
62.50Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
62.50Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
62.50Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
62.50Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
62.50Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
62.50Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
62.50Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
62.50Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
62.50Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
62.50Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
62.50Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
62.50Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
62.50Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
62.50Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
62.50Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
61.54Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
61.54Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
61.54Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
61.54Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
61.54Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
61.11Single3NY9ICI118-5513NY9-β2-ICI118-551
61.11Single8X5YAstemizole8X5Y-H1-Astemizole
60.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
60.00Single2Y04Salbutamol2Y04-β1-Salbutamol
60.00Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
60.00Single3NY8ICI118-5513NY8-β2-ICI118-551
60.00Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
60.00Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
60.00Single4GBRS-Carazolol4GBR-β2-S-Carazolol
60.00Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
60.00Single5DHGC-355DHG-NOP-C-35
60.00Single6H7MSalbutamol6H7M-β1-Salbutamol
60.00Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
60.00Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
60.00Single6PS1Timolol6PS1-β2-Timolol
60.00Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
60.00Single6TOTLemborexant6TOT-OX1-Lemborexant
60.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
60.00Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
60.00Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
60.00Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
60.00Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
60.00Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
60.00Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
60.00Single7UL4Alvimopan7UL4-μ-Alvimopan
60.00Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
60.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
60.00Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
60.00Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
60.00Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
60.00Single8JJOAlprenolol8JJO-β2-Alprenolol
60.00Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
60.00Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
60.00Single8T1WCVN4248T1W-GPR6-CVN424
60.00Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
60.00Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
60.00Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
60.00Single8X64Desloratadine8X64-H1-Desloratadine
60.00Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
60.00Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
60.00Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
60.00Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
60.00Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
60.00Consensusalpha2_onOrthosteric Ligandalpha2b_on
60.00Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
60.00Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
60.00Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
60.00Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
60.00Consensusdopamine_offOrthosteric Ligandd2_off d3_off
60.00Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
60.00Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
58.82Single3D4STimolol3D4S-β2-Timolol
58.82Single4AMIBucindolol4AMI-β1-Bucindolol
58.82Single4RWADIPP-NH24RWA-δ-DIPP-NH2
58.82Single5CXVTiotropium5CXV-M1-Tiotropium
58.82Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
58.82Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
58.82Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
58.82Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
58.82Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
58.82Single8JJ8Formoterol8JJ8-β2-Formoterol
58.82Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
58.82Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
58.82Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
58.82Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
58.82Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
58.82Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
57.89Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
57.89Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
57.89Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
57.14Single5WS3EMPA5WS3-OX2-EMPA
57.14Single6AKXA4R6AKX-CCR5-A4R
57.14Single6B73MP11046B73-κ-MP1104
57.14Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
57.14Single6TODEMPA6TOD-OX1-EMPA-Na
57.14Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
57.14Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
57.14Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
57.14Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
57.14Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
57.14Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
57.14Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
57.14Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
57.14Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
57.14Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
57.14Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
57.14Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
57.14Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
57.14Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
57.14Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
57.14Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
57.14Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
57.14Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
57.14Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
57.14Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
57.14Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
57.14Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
57.14Consensusalpha2_offOrthosteric Ligandalpha2c_off
57.14Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
57.14Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
57.14Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
57.14Consensusorexin_offOrthosteric Ligandox2_off ox1_off
57.14Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
57.14Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
56.25Single2YCWS-Carazolol2YCW-β1-S-Carazolol
56.25Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
56.25Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
56.25Single5D6LS-Carazolol5D6L-β2-S-Carazolol
56.25Single5TVNLSD5TVN-5-HT2B-LSD
56.25Single5WIUNemonapride5WIU-D4-Nemonapride
56.25Single5WIVNemonapride5WIV-D4-Nemonapride-Na
56.25Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
56.25Single6E67BI1671076E67-β2-BI167107-Gs (fused)
56.25Single6PS6Timolol6PS6-β2-Timolol
56.25Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
56.25Single6TP6Filorexant6TP6-OX1-Filorexant
56.25Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
56.25Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
56.25Single8JXSPF-61428JXS-D1-PF-6142
56.25Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
56.25Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
56.25Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
56.25Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
56.25Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
56.25Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
56.25Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
56.25Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
56.25Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
56.25Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
56.25Consensustrace-amine_onOrthosteric Ligandta1_on
55.56Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
55.56Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
55.56Single6H7LDobutamine6H7L-β1-Dobutamine
55.56Single6IBLArformoterol6IBL-β1-Arformoterol
55.56Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
55.56Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
55.56Single7UM4AS26747237UM4-5-HT5A-AS2674723
55.56Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
55.56Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
55.56Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
55.56Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
55.56Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
55.56Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
55.56Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
55.56Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
53.85Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
53.85Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
53.85Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
53.85Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
53.33Single4MBSMaraviroc4MBS-CCR5-Maraviroc
53.33Single6IQLL7458706IQL-D4-L745870
53.33Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
53.33Single6TPNHTL66416TPN-OX2-HTL6641
53.33Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
53.33Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
53.33Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
53.33Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
53.33Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
53.33Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
53.33Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.33Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
53.33Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
53.33Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
53.33Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
53.33Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
53.33Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.33Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
53.33Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
53.33Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
53.33Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
53.33Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
53.33Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
52.94Single2YDVNECA2YDV-A2A-NECA
52.94Single3P0GBI1671073P0G-β2-BI167107
52.94Single4DJHJDTic4DJH-κ-JDTic
52.94Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
52.94Single4U15Tiotropium4U15-M3-Tiotropium
52.94Single4UHRCGS216804UHR-A2A-CGS21680
52.94Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
52.94Single5G53NECA5G53-A2A-NECA-Gs
52.94Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
52.94Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
52.94Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
52.94Single6OL9Tiotropium6OL9-M5-Tiotropium
52.94Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
52.94Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
52.94Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
52.94Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
52.94Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
52.94Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
52.94Single8XVLZibotentan8XVL-ETA-Zibotentan
52.94Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
52.94Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
52.94Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
52.94Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
52.94Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
52.94Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
52.94Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
52.94Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
52.63Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
52.63Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
52.63Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Single2Y02Carmoterol2Y02-β1-Carmoterol
50.00Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
50.00Single3PBLEticlopride3PBL-D3-Eticlopride
50.00Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
50.00Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
50.00Single4DAJTiotropium4DAJ-M3-Tiotropium
50.00Single4EJ4Naltrindole4EJ4-δ-Naltrindole
50.00Single4IARErgotamine4IAR-5-HT1B-Ergotamine
50.00Single4QKX35V4QKX-β2-35V
50.00Single5DHHSB-6121115DHH-NOP-SB-612111
50.00Single5DSGTiotropium5DSG-M4-Tiotropium
50.00Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
50.00Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
50.00Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
50.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
50.00Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
50.00Single6MXTSalmeterol6MXT-β2-Salmeterol
50.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
50.00Single6ZG4HTL00099366ZG4-M1-HTL0009936
50.00Single7BU7BI1671077BU7-β1-BI167107
50.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
50.00Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
50.00Single7DFPSpiperone7DFP-D2-Spiperone
50.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
50.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
50.00Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
50.00Single7SRQLSD7SRQ-5-HT2B-LSD
50.00Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
50.00Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
50.00Single7WC7Lisuride7WC7-5-HT2A-Lisuride
50.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
50.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
50.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
50.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
50.00Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
50.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
50.00Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
50.00Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
50.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
50.00Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
50.00Single8JXRLSD8JXR-D1-LSD
50.00Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
50.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
50.00Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
50.00Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
50.00Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
50.00Single8X63Mepyramine8X63-H1-Mepyramine
50.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
50.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
50.00Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
50.00Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
50.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
50.00Single9CHXS-Carazolol9CHX-β2-S-Carazolol
50.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
50.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
50.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
50.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
50.00Consensus5ht5_onOrthosteric Ligand5ht5a_on
50.00Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
50.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
50.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
50.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
50.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
50.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
50.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
50.00Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
50.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
50.00Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
50.00Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
50.00Consensushistamine_offOrthosteric Ligandh1_off
50.00Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
50.00Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
50.00Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
50.00Consensusorexin_onOrthosteric Ligandox2_on
47.83Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
47.62Single6HLOAprepitant6HLO-NK1-Aprepitant
47.62Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
47.37Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
47.37Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
47.37Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
47.37Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
47.37Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
47.37Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
47.37Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
47.37Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
47.37Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
47.37Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
47.37Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
47.06Single5XPRBosentan5XPR-ETB-Bosentan
47.06Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
47.06Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
47.06Single7C61Ergotamine7C61-5-HT1B-Ergotamine
47.06Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
47.06Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
47.06Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
47.06Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
47.06Single8TF5Oleic acid8TF5-GPR6-Oleic acid
47.06Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
47.06Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
47.06Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
47.06Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
47.06Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
47.06Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
47.06Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
46.67Single4S0VSuvorexant4S0V-OX2-Suvorexant
46.67Single6AKYMaraviroc6AKY-CCR5-Maraviroc
46.67Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
46.67Single6TPJSuvorexant6TPJ-OX2-Suvorexant
46.67Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
46.67Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
46.67Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
46.67Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
46.67Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
46.67Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
46.67Single7XRRLemborexant7XRR-OX2-Lemborexant
46.67Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
46.67Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
46.67Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
46.67Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
46.67Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
46.67Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
46.67Single8Y0HVUF114188Y0H-CXCR3-VUF11418
46.67Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
46.67Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
46.67Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
46.67Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
46.67Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
46.67Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
46.15Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
46.15Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
46.15Single9CHUNoradrenaline9CHU-β2-Noradrenaline
46.15Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
46.15Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
45.83Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
45.45Single6PT2KGCHM076PT2-δ-KGCHM07
45.45Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
45.45Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
45.00Single4UG2CGS216804UG2-A2A-CGS21680
45.00Single5ZTYAM102575ZTY-CB2-AM10257
45.00Single6PT3DPI-2876PT3-δ-DPI-287
45.00Single7SK9CCX6627SK9-ACKR3-CCX662
45.00Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
45.00Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
45.00Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
44.44Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
44.44Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
44.44Single5V54Methiothepin5V54-5-HT1B-Methiothepin
44.44Single6E59L-7607356E59-NK1-L-760735
44.44Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
44.44Single6J20Aprepitant6J20-NK1-Aprepitant
44.44Single6J21Aprepitant6J21-NK1-Aprepitant
44.44Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
44.44Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
44.44Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
44.44Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
44.44Single8EA0Iperoxo8EA0-M3-Iperoxo
44.44Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
44.44Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
44.44Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
44.44Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
44.44Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
44.44Consensus5ht1_offOrthosteric Ligand5ht1b_off
44.44Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
44.44Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
44.44Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
44.44Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
44.44Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
44.44Consensustachykinin_offOrthosteric Ligandnk1_off
43.75Single3RZECidoxepin3RZE-H1-Cidoxepin
43.75Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
43.75Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
43.75Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
43.75Single6A94Zotepine6A94-5-HT2A-Zotepine
43.75Single6KUXRS-799486KUX-α2a-RS-79948
43.75Single6TP3Nemorexant6TP3-OX1-Nemorexant
43.75Single6V9SGTPL114036V9S-OX1-GTPL11403
43.75Single6VI4JDTic6VI4-κ-JDTic
43.75Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
43.75Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
43.75Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
43.75Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
43.75Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
43.75Single7UL3Famotidine7UL3-H2-Famotidine
43.75Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
43.75Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
43.75Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
43.75Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
43.75Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
43.75Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
43.75Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
43.75Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
43.75Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
43.75Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
43.75Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
43.75Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
43.75Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
43.75Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
43.75Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
43.75Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
43.75Single9BJKNaloxone9BJK-μ-Naloxone-NAM
43.75Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
43.48Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
42.86Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
42.86Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
42.86Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.86Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
42.86Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
42.86Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
42.86Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
42.86Single8WDTphotoNECA8WDT-A2A-photoNECA
42.86Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
42.86Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
42.86Consensus5ht2_onOrthosteric Ligand5ht2b_on
42.86Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.86Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
42.86Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
42.86Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
42.11Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
42.11Single6A93Risperidone6A93-5-HT2A-Risperidone
42.11Single6CM4Risperidone6CM4-D2-Risperidone
42.11Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
42.11Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
42.11Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
42.11Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
42.11Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
42.11Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
42.11Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
42.11Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
42.11Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
42.11Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
42.11Single8JJLOlodaterol8JJL-β2-Olodaterol
42.11Single8XYIVUF106618XYI-CXCR3-VUF10661
42.11Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
42.11Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
42.11Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
42.11Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
42.11Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
42.11Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
42.11Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
41.67Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
41.18Single2Y01Dobutamine2Y01-β1-Dobutamine
41.18Single4MQSIperoxo4MQS-M2-Iperoxo
41.18Single4U14Tiotropium4U14-M3-Tiotropium
41.18Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
41.18Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
41.18Single6DRXLisuride6DRX-5-HT2B-Lisuride
41.18Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
41.18Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
41.18Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
41.18Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
41.18Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
41.18Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
41.18Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
41.18Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
41.18Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
41.18Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
41.18Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
41.18Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
41.18Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
41.18Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
40.91Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
40.91Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
40.91Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
40.00Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
40.00Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
40.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
40.00Single6TP4ACT-4622066TP4-OX1-ACT-462206
40.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
40.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
40.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
40.00Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
40.00Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.00Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
40.00Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
40.00Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
40.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
40.00Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
40.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
40.00Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
40.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
40.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
40.00Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
40.00Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
40.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
40.00Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
40.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
40.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
40.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
40.00Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
39.13Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
39.13Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
39.13Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
39.13Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
39.13Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
38.89Single2Y00Dobutamine2Y00-β1-Dobutamine
38.89Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
38.89Single6HLPNetupitant6HLP-NK1-Netupitant
38.89Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
38.89Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
38.89Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
38.89Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
38.89Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
38.89Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
38.89Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
38.89Single7SINNPS-21437SIN-CaS-NPS-2143
38.89Single7SINNPS-21437SIN-CaS-NPS-2143
38.89Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
38.89Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
38.89Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
38.89Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
38.89Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
38.89Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
38.89Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
38.89Single8S4DCMF-0198S4D-Apelin-CMF-019
38.89Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
38.89Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
38.89Single8ZMFA1L108ZMF-5-HT2C-A1L10
38.89Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
38.89Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
38.89Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
38.46Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
38.46Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
38.46Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
38.10Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
38.10Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
38.10Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
38.10Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
38.10Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
38.10Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
38.10Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
37.50Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
37.50Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
37.50Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
37.50Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
37.50Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
37.50Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
37.50Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
37.50Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
37.50Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
37.50Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
37.50Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
37.50Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
37.50Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
37.50Single8IWESpermidine8IWE-TA9-Spermidine
37.50Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
37.50Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
37.50Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
37.50Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
37.50Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
37.50Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
37.50Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
37.50Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
37.50Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
37.50Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
37.50Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
37.50Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
37.50Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
37.50Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
37.50Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
37.50Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
36.84Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
36.84Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
36.84Single7B6WCyclazosin7B6W-α1b-Cyclazosin
36.84Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
36.84Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
36.84Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
36.84Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
36.84Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
36.84Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
36.84Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
36.84Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
36.84Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
36.84Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
36.84Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
36.84Consensusa2_onOrthosteric Liganda2b_on
36.84Consensusa2_on_gpOrthosteric Liganda2b_on_gp
36.84Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
36.84Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
36.84Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
36.84Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
36.84Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
36.84Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
36.36Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
36.36Single7QA8Peptide7QA8-STE2-Peptide
36.36Single7QA8Peptide7QA8-STE2-Peptide
36.36Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
36.36Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
36.36Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
36.36Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
36.36Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
36.36Consensuslpl_onOrthosteric Ligands1p_on lpa_on
36.36Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
36.36Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
36.36Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
36.00Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
35.71Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
35.71Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
35.71Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
35.71Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
35.71Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
35.71Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
35.71Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
35.71Consensusbombesin_onOrthosteric Ligandbb2_on
35.71Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
35.71Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
35.29Single2YDOAdenosine2YDO-A2A-Adenosine
35.29Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
35.29Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
35.29Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
35.29Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
35.29Single6ZG9GSK10347026ZG9-M1-GSK1034702
35.29Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
35.29Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
35.29Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
35.29Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
35.29Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
35.29Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
35.29Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
35.29Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
35.29Single8IHKAcifran8IHK-HCA3-Acifran
35.29Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
35.29Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
35.29Single8K5CAcipimox8K5C-HCA2-Acipimox
35.29Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
35.29Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
35.29Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
35.29Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
35.29Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
35.29Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
35.29Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
35.29Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
35.29Consensushca_onOrthosteric Ligandhca2_on
35.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
35.00Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
35.00Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
35.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
35.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
35.00Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
35.00Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
35.00Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
35.00Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
35.00Single8JWZAB9288JWZ-A2A-AB928-Na
35.00Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
35.00Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
35.00Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
35.00Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
35.00Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
35.00Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
35.00Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
35.00Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
35.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
35.00Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
35.00Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
35.00Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
35.00Consensuslpa_offOrthosteric Ligandlpa1_off
35.00Consensuslpl_offOrthosteric Ligands1p_off lpa_off
35.00Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
35.00Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.78Single3QAKUK-4320973QAK-A2A-UK-432097
34.78Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
34.78Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
34.78Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
34.78Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
34.78Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
34.78Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
34.62Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
34.62Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
34.62Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
33.33Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
33.33Single3UZAGTPL92363UZA-A2A-GTPL9236
33.33Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
33.33Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
33.33Single4YAYZD-71554YAY-AT1-ZD-7155
33.33Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
33.33Single5WF5UK-4320975WF5-A2A-UK-432097
33.33Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
33.33Single6GPSMK08126GPS-CCR2-MK0812
33.33Single6K1QIRL25006K1Q-ETB-IRL2500
33.33Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
33.33Single7EZCUKA7EZC-A2A-UKA
33.33Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
33.33Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
33.33Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
33.33Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
33.33Single7V3ZCP559407V3Z-CB1-CP55940
33.33Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
33.33Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
33.33Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
33.33Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
33.33Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
33.33Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
33.33Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
33.33Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
33.33Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
33.33Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
33.33Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
33.33Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
33.33Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
33.33Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
33.33Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
33.33Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
33.33Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
33.33Single8K5DGSK2560738K5D-HCA2-GSK256073
33.33Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
33.33Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
33.33Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
33.33Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8XVJMacitentan8XVJ-ETA-Macitentan
33.33Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
33.33Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
33.33Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
33.33Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
33.33Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
33.33Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
33.33Consensusa3_onOrthosteric Liganda3a_on
33.33Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusblt_onOrthosteric Ligandblt1_on
33.33Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
33.33Consensuscck_offOrthosteric Ligandccka_off
33.33Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
33.33Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
33.33Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
33.33Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
33.33Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
33.33Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
33.33Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
33.33Consensushca_on_gpOrthosteric Ligandhca2_on_gp
33.33Consensusleukotriene_onOrthosteric Ligandblt_on
33.33Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
33.33Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
33.33Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
33.33Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
33.33Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
33.33Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
33.33Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
32.14Single6IGLIRL16206IGL-ETB-IRL1620
32.14Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
32.00Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
32.00Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
32.00Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
32.00Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Consensusvasop-oxy_onOrthosteric Ligandv2_on
32.00Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
31.82Single5WF6UK-4320975WF6-A2A-UK-432097
31.82Single7XN9L-054,5227XN9-SST2-L-054,522
31.82Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
31.82Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
31.82Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
31.82Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
31.82Single8QJ2pN1628QJ2-MC4-pN162-Gs
31.82Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
31.82Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
31.82Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
31.58Single5CGCHTL142425CGC-mGlu5-HTL14242
31.58Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
31.58Single6GPXMK08126GPX-CCR2-MK0812
31.58Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
31.58Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
31.58Single7C4SS1P7C4S-S1P3-S1P
31.58Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
31.58Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
31.58Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
31.58Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
31.58Single7W41PD1762527W41-BB2-PD176252
31.58Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
31.58Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
31.58Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
31.58Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
31.58Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
31.58Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
31.58Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
31.58Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
31.58Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
31.58Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
31.58Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
31.58Consensusa3_on_gpOrthosteric Liganda3a_on_gp
31.58Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
31.58Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
31.58Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
31.58Consensusbombesin_offOrthosteric Ligandbb2_off
31.58Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
31.58Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
31.58Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
31.58Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
31.58Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
31.25Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
31.25Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
31.25Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
31.25Single6HLLCP999946HLL-NK1-CP99994
31.25Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
31.25Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
31.25Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
31.25Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
31.25Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
31.25Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
31.25Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
31.25Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
31.25Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
31.25Single8K5BNiacin8K5B-HCA2-Niacin
31.25Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
31.25Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
31.25Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
31.25Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
31.25Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
31.25Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
31.25Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
30.77Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
30.77Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
30.77Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single8ZRTET-18ZRT-ETB-ET-1
30.77Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
30.77Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
30.77Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.43Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
30.43Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
30.43Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
30.43Single8IEBA1LYA8IEB-GPR156-A1LYA
30.43Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
30.43Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
30.43Single8WKYPG-9348WKY-MC4-PG-934
30.43Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
30.43Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
30.00Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
30.00Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
30.00Single5XR8AM8415XR8-CB1-AM841
30.00Single5XRAAM115425XRA-CB1-AM11542
30.00Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
30.00Single7FEECP559407FEE-CB1-CP55940-ZCZ011
30.00Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
30.00Single7TUYGSK682753A7TUY-GPR183-GSK682753A
30.00Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
30.00Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
30.00Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
30.00Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
30.00Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
30.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
30.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
30.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
30.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
30.00Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
30.00Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
30.00Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.00Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
30.00Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
30.00Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
30.00Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
29.63Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
29.63Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.63Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
29.63Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
29.41Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
29.41Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
29.41Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
29.41Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
29.41Single6DS0Ly2660976DS0-5-HT2B-Ly266097
29.41Single6ME2Ramelteon6ME2-MT1-Ramelteon
29.41Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
29.41Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
29.41Single7BR3Elagolix7BR3-GnRH1-Elagolix
29.41Single7F8ULintitript7F8U-CCKA-Lintitript
29.41Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
29.41Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
29.41Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
29.41Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
29.41Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
29.41Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
29.41Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.41Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
29.41Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
29.41Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
29.41Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
29.41Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
29.41Consensusangiotensin_offOrthosteric Ligandat1_off
29.41Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
29.41Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
29.41Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
29.41Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
29.17Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
29.17Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
29.17Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
29.17Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
29.17Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
29.17Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
29.17Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
29.17Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
29.03Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
28.57Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
28.57Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
28.57Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
28.57Single6KQICP559406KQI-CB1-CP55940-Org27569
28.57Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
28.57Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
28.57Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
28.57Single7K15MKD0467K15-BLT1-MKD046-Na
28.57Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
28.57Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
28.57Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
28.57Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
28.57Single8JWY2-1188JWY-A2A-2-118
28.57Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
28.57Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
28.57Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
28.57Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
28.57Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
28.57Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
28.00Single6W25SHU91196W25-MC4-SHU9119-Ca
28.00Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
28.00Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
28.00Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
28.00Consensusangiotensin_onOrthosteric Ligandat1_on
28.00Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
28.00Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
28.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
27.78Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
27.78Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
27.78Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
27.78Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
27.78Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
27.78Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
27.78Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
27.78Single6TPKRetosiban6TPK-OT-Retosiban
27.78Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
27.78Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
27.78Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
27.78Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
27.78Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
27.78Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
27.78Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
27.78Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
27.78Consensusgrh_offOrthosteric Ligandgnrh1_off
27.78Consensusopsins_offOrthosteric Ligandrhodopsin_off
27.78Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
27.78Consensussensory_offOrthosteric Ligandopsins_off
27.78Consensusvasop-oxy_offOrthosteric Ligandot_off
27.59Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
27.59Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
27.59Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
27.59Consensusbradykinin_onOrthosteric Ligandbk2_on
27.59Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
27.59Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
27.27Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
27.27Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
27.27Single5CGDHTL142425CGD-mGlu5-HTL14242
27.27Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
27.27Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
27.27Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
27.27Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
27.27Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
27.27Consensusprostanoid_offOrthosteric Ligandep_off dp_off
26.92Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
26.92Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
26.92Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
26.92Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
26.92Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
26.92Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
26.92Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
26.92Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
26.92Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
26.92Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
26.67Single3OE8IT1t3OE8-CXCR4-IT1t
26.67Single5GLHEndothelin-15GLH-ETB-Endothelin-1
26.67Single6IGKEndothelin-36IGK-ETB-Endothelin-3
26.67Single6TQ9SB-4081246TQ9-OX1-SB-408124
26.67Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
26.67Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
26.67Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
26.67Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
26.67Consensussensory_onOrthosteric Ligandopsins_on
26.32Single5TGZAM65385TGZ-CB1-AM6538
26.32Single5UIGCmpd-15UIG-A2A-Cmpd-1
26.32Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
26.32Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
26.32Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
26.32Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
26.32Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
26.32Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
26.32Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
26.32Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
26.32Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
26.32Single7YXAONO-54306087YXA-S1P5-ONO-5430608
26.32Single8CU6LJ-45178CU6-A2A-LJ-4517
26.32Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
26.32Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
26.32Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
26.32Single8RLNLUF58348RLN-A2A-LUF5834
26.32Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
26.32Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
26.32Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
26.09Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
26.09Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
26.09Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
26.09Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
26.09Single8IEIA1LYA8IEI-GPR156-A1LYA
26.09Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
26.09Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
26.09Consensuskisspeptin_onOrthosteric Ligandkiss1_on
25.93Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
25.93Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
25.93Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.93Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
25.93Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
25.93Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
25.93Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
25.81Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
25.81Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
25.81Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
25.81Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
25.00Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
25.00Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
25.00Single3OE6IT1t3OE6-CXCR4-IT1t
25.00Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
25.00Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
25.00Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
25.00Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
25.00Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
25.00Single6D26Fevipiprant6D26-DP2-Fevipiprant
25.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
25.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
25.00Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
25.00Single6LUQHaloperidol6LUQ-D2-Haloperidol
25.00Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
25.00Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
25.00Single7F8XNN90567F8X-CCKA-NN9056
25.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
25.00Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Single7WC5Psilocin7WC5-5-HT2A-Psilocin
25.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single8IEIA1LYA8IEI-GPR156-A1LYA
25.00Single8IEPA1LYA8IEP-GPR156-A1LYA
25.00Single8IEPA1LYA8IEP-GPR156-A1LYA
25.00Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
25.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
25.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
25.00Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
25.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
25.00Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
25.00Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusadenosine_offOrthosteric Liganda1_off a2_off
25.00Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
25.00Consensusblt_offOrthosteric Ligandblt1_off
25.00Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
25.00Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
25.00Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
25.00Consensusdp_offOrthosteric Liganddp2_off
25.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
25.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
25.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
25.00Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.00Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
25.00Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
25.00Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
25.00Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
25.00Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
25.00Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
25.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
25.00Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
25.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
25.00Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.00Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.00Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
25.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
25.00Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.14Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
24.00Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
24.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
24.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
24.00Single8IEBA1LYA8IEB-GPR156-A1LYA
24.00Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
24.00Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
24.00Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
24.00Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
24.00Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
24.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
24.00Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
24.00Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
23.81Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
23.81Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
23.81Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
23.81Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
23.81Single7P2L4YI7P2L-mGlu5-4YI
23.81Single7R0CAVP7R0C-V2-AVP-Arrestin2
23.81Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
23.81Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
23.81Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
23.81Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
23.81Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
23.81Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
23.81Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.81Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
23.81Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
23.81Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
23.81Single9BJKNAM9BJK-μ-Naloxone-NAM
23.81Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
23.81Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
23.81Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.81Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
23.81Consensuslpa_onOrthosteric Ligandlpa1_on
23.81Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
23.81Consensusrelaxin_onOrthosteric Ligandrxfp4_on
23.81Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
23.53Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
23.53Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
23.53Single3OE9IT1t3OE9-CXCR4-IT1t
23.53Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
23.53Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
23.53Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
23.53Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
23.53Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
23.53Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
23.53Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
23.53Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
23.33Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
23.33Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
23.33Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
23.33Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
23.33Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
23.33Consensusendothelin_onOrthosteric Ligandetb_on eta_on
23.33Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
23.33Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
23.08Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
23.08Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
23.08Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
23.08Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
23.08Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
23.08Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
23.08Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
22.86Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
22.86Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
22.73Single4N4WSANT-14N4W-SMO-SANT-1
22.73Single5X33BIIL2605X33-BLT1-BIIL260
22.73Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
22.73Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
22.73Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
22.73Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
22.73Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
22.73Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
22.73Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.73Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
22.58Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
22.58Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
22.58Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
22.58Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
22.58Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
22.22Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
22.22Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
22.22Single3ODUIT1t3ODU-CXCR4-IT1t
22.22Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
22.22Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
22.22Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
22.22Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
22.22Single6JODAngiotensin II6JOD-AT2-Angiotensin II
22.22Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
22.22Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
22.22Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
22.22Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
22.22Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
22.22Single7F8YDevazepide7F8Y-CCKA-Devazepide
22.22Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
22.22Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
22.22Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
22.22Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
22.22Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
22.22Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
22.22Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
22.22Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
22.22Single8GNGIstradefylline8GNG-A2A-Istradefylline
22.22Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
22.22Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
22.22Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.22Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
22.22Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.22Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.22Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
22.22Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
22.22Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
21.88Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
21.88Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
21.88Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
21.74Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
21.74Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
21.74Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensuscck_onOrthosteric Ligandccka_on cckb_on
21.74Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
21.74Consensuschemerin_onOrthosteric Ligandcml1_on
21.74Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
21.43Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
21.43Single5MZPCaffeine5MZP-A2A-Caffeine-Na
21.43Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
21.43Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.43Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
21.43Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
21.43Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
21.43Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
21.43Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
21.43Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
21.43Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
21.05Single3REYXAC3REY-A2A-XAC
21.05Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
21.05Single5IU7Q274563465IU7-A2A-Q27456346-Na
21.05Single5IUBQ274563445IUB-A2A-Q27456344-Na
21.05Single5JTBZM-2413855JTB-A2A-ZM-241385
21.05Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
21.05Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
21.05Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
21.05Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
21.05Single6AQFZM-2413856AQF-A2A-ZM-241385
21.05Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
21.05Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
21.05Single7AROLUF58337ARO-A2A-LUF5833-Na
21.05Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
21.05Single7T32ZM-2413857T32-A2A-ZM-241385
21.05Single7VODCariprazine7VOD-5-HT2A-Cariprazine
21.05Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
21.05Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single8K2WAMG4878K2W-CXCR3-AMG487
21.05Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.05Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
21.05Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
21.05Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
21.05Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
21.05Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
21.05Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
21.05Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
21.05Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
21.05Consensusa2_offOrthosteric Liganda2a_off
21.05Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
21.05Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
20.83Single5EE7MK08935EE7-Glucagon-MK0893
20.83Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
20.83Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
20.83Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
20.83Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
20.83Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
20.83Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
20.69Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
20.69Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
20.59Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
20.59Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
20.59Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
20.59Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single3EMLZM-2413853EML-A2A-ZM-241385
20.00Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
20.00Single4XT1Fractalkine4XT1-US28-Fractalkine
20.00Single5IU8Q274563475IU8-A2A-Q27456347-Na
20.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
20.00Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
20.00Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
20.00Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
20.00Single5UENDU1725UEN-A1-DU172
20.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
20.00Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
20.00Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
20.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
20.00Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
20.00Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
20.00Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
20.00Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
20.00Single6S0LZM-2413856S0L-A2A-ZM-241385
20.00Single7F83PF-051904577F83-Ghrelin-PF-05190457
20.00Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
20.00Single7PYRPSB-21157PYR-A2A-PSB-2115
20.00Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
20.00Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7WC4Serotonin7WC4-5-HT2A-Serotonin
20.00Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
20.00Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
20.00Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.00Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
20.00Single8KIGSHU91198KIG-MC3-SHU9119-Ca
20.00Single8PWNTheophylline8PWN-A2A-Theophylline
20.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
20.00Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
20.00Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
20.00Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
20.00Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
20.00Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
20.00Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
20.00Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
20.00Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
20.00Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
20.00Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
20.00Single9IYAONO-97105319IYA-GPR55-ONO-9710531
20.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
20.00Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.00Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
20.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
20.00Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
20.00Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
19.51Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
19.35Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
19.35Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
19.35Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
19.35Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
19.35Single8IY6Endothelin-18IY6-ETB-Endothelin-1
19.23Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
19.23Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
19.23Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
19.23Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
19.23Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
19.23Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
19.05Single4NTJAZD12834NTJ-P2Y12-AZD1283
19.05Single5IUAQ274563485IUA-A2A-Q27456348-Na
19.05Single5N2RPSB-365N2R-A2A-PSB-36-Na
19.05Single5N2SPSB365N2S-A1-PSB36
19.05Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
19.05Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
19.05Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
19.05Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
19.05Single6S0QZM-2413856S0Q-A2A-ZM-241385
19.05Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
19.05Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
19.05Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
19.05Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
19.05Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
19.05Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
19.05Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
19.05Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
19.05Single8GNEKW-63568GNE-A2A-KW-6356-Na
19.05Single8QOTNanobody-E8QOT-μ-Nanobody-E
19.05Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
19.05Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
19.05Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
19.05Consensusep_offOrthosteric Ligandep4_off
18.75Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
18.75Single3RFMCaffeine3RFM-A2A-Caffeine
18.75Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
18.75Single8A2OTheophylline8A2O-A2A-Theophylline-Na
18.75Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
18.52Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
18.52Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
18.52Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
18.52Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
18.52Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
18.52Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.52Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.52Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
18.52Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
18.18Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
18.18Single7PX4PSB-21137PX4-A2A-PSB-2113
18.18Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
18.18Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
18.18Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
18.18Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
18.18Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
18.18Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
18.18Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
18.18Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
18.18Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
18.18Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
18.18Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
18.18Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
18.18Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
17.86Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
17.86Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
17.86Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
17.86Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
17.86Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
17.86Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
17.86Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
17.86Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
17.86Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
17.86Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
17.65Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
17.65Single6ME5Agomelatine6ME5-MT1-Agomelatine
17.65Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
17.65Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
17.65Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
17.65Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.65Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
17.65Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
17.65Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
17.65Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.65Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
17.65Consensusgi_sensoryOrthosteric Ligandgi_opsins
17.65Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
17.65Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
17.39Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
17.39Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
17.39Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
17.39Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
17.39Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
17.39Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
17.39Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
17.39Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
17.39Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
17.39Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
17.39Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
17.39Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
17.39Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
17.24Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
17.24Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
17.24Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
17.24Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
17.24Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
17.24Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
17.24Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
17.24Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
17.24Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.67Single4XT3Fractalkine4XT3-US28-Fractalkine
16.67Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
16.67Single6FJ3PTH6FJ3-PTH1-PTH
16.67Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
16.67Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
16.67Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
16.67Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
16.67Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.67Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
16.67Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
16.67Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
16.67Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
16.67Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
16.67Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
16.67Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
16.67Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
16.67Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
16.67Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
16.67Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
16.67Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
16.67Single9B9Y7DY9B9Y-CB1-7DY
16.67Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
16.67Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.67Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.67Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
16.67Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
16.67Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
16.67Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
16.67Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
16.13Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
16.13Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
16.13Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
16.13Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
16.00Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
16.00Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
16.00Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
16.00Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
16.00Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
16.00Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
16.00Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
16.00Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
16.00Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
16.00Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single3PWHZM-2413853PWH-A2A-ZM-241385
15.79Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
15.79Single5ZKQABT-4915ZKQ-PAF-ABT-491
15.79Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
15.79Single6ME9Ramelteon6ME9-MT2-Ramelteon
15.79Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
15.79Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
15.79Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
15.79Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
15.79Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
15.79Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
15.79Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
15.79Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
15.62Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
15.62Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
15.62Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
15.62Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
15.62Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
15.62Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
15.62Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
15.62Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
15.62Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
15.38Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
15.38Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
15.38Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
15.38Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.38Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
15.38Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
15.15Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
15.00Single5UVIZM-2413855UVI-A2A-ZM-241385
15.00Single6FFIMMPEP6FFI-mGlu5-MMPEP
15.00Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
15.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
15.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
15.00Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
15.00Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
15.00Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
15.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
15.00Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
14.81Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
14.81Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
14.81Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
14.81Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
14.81Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
14.71Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
14.71Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
14.71Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
14.29Single3OE0CVX153OE0-CXCR4-CVX15
14.29Single6D27CAY104716D27-DP2-CAY10471
14.29Single6FFHFenobam6FFH-mGlu5-Fenobam
14.29Single6IIVDaltroban6IIV-TP-Daltroban
14.29Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
14.29Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
14.29Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
14.29Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
14.29Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
14.29Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
14.29Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
14.29Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
14.29Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.29Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
13.89Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.79Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
13.79Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
13.79Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
13.79Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
13.79Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
13.79Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
13.64Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
13.64Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
13.64Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
13.64Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.64Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
13.64Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
13.64Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
13.64Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
13.51Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
13.33Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
13.33Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
13.33Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
13.33Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
13.33Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
13.04Single5TZRMK86665TZR-FFA1-MK8666
13.04Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
13.04Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
13.04Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
13.04Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
13.04Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
13.04Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
13.04Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.90Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
12.90Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
12.90Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
12.90Single7SK3CXCL127SK3-ACKR3-CXCL12
12.90Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
12.90Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
12.90Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
12.50Single4PY02MeSATP4PY0-P2Y12-2MeSATP
12.50Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
12.50Single6IIURamatroban6IIU-TP-Ramatroban
12.50Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
12.50Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
12.50Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
12.50Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
12.50Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
12.50Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
12.50Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.50Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
12.50Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.50Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
12.50Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
12.50Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.50Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.50Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.00Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
12.00Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
12.00Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
12.00Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
11.54Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
11.54Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
11.54Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
11.54Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
11.54Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
11.54Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
11.11Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
11.11Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
11.11Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
11.11Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
11.11Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
11.11Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
11.11Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.11Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
11.11Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
11.11Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
11.11Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
11.11Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
11.11Consensussomatostatin_offOrthosteric Ligandsst2_off
10.71Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
10.71Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
10.71Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
10.71Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
10.71Single7SK5CXCL127SK5-ACKR3-CXCL12
10.71Single7XNACYN1548067XNA-SST2-CYN154806
10.71Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.71Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
10.53Single5L7IVismodegib5L7I-SMO-Vismodegib
10.53Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
10.53Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
10.53Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
10.53Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
10.53Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
10.34Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
10.00Single5U09Taranabant5U09-CB1-Taranabant
10.00Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
10.00Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
10.00Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
10.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
10.00Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
10.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
10.00Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
10.00Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
10.00Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
10.00Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
10.00Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
10.00Single9BA0A1AKN9BA0-CB1-A1AKN
9.68Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
9.68Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
9.52Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
9.52Single6ZINSR486926ZIN-NTS1-SR48692
9.52Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
9.52Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
9.52Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.52Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
9.52Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.38Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
9.38Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
9.09Single4QIMANTA XV4QIM-SMO-ANTA XV
9.09Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
9.09Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
9.09Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
9.09Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
9.09Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
9.09Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
9.09Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
9.09Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
9.09Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
9.09Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
9.09Single9B9ZA1AKO9B9Z-CB1-A1AKO
9.09Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
9.09Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
9.09Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
8.82Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
8.70Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
8.70Single6Z4SSR486926Z4S-NTS1-SR48692
8.70Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
8.70Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
8.70Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
8.70Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
8.57Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
8.33Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
8.33Single4BV0Neurotensin4BV0-NTS1-Neurotensin
8.33Single5V56TC1145V56-SMO-TC114
8.33Single6OS1TRV0266OS1-AT1-TRV026
8.33Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
8.33Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
8.33Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
8.33Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
8.33Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
8.33Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
8.33Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
8.33Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
8.33Consensusneurotensin_onOrthosteric Ligandnts1_on
8.33Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
8.11Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
8.00Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
8.00Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
8.00Single4XEENeurotensin4XEE-NTS1-Neurotensin
8.00Single4XESNeurotensin4XES-NTS1-Neurotensin
8.00Single6OS2TRV0266OS2-AT1-TRV026
8.00Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
8.00Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
8.00Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
8.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
8.00Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
8.00Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
8.00Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
8.00Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
8.00Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
7.89Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
7.89Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
7.69Single4BUONeurotensin4BUO-NTS1-Neurotensin
7.69Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
7.69Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
7.69Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
7.69Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
7.69Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
7.41Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
7.41Single8XQJJN2418XQJ-Apelin-JN241
7.41Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
7.41Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
7.14Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
7.14Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
6.90Single7SHEPI; PE7SHE-GPR158-PI; PE
6.90Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
6.67Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
6.25Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
6.25Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
6.25Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
5.88Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
5.88Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
5.56Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
5.56Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
5.26Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
5.26Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
5.26Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
5.13Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
5.00Single6LI0C176LI0-GPR52-C17
5.00Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.00Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
5.00Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
5.00Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
5.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
5.00Consensusgq_nucleotideOrthosteric Ligandgq_p2y
5.00Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
4.76Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
4.76Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
4.76Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
4.76Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
4.55Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
4.55Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
4.55Single7VV6C48/807VV6-MRGPRX2-C48/80
4.55Single8IYXYL-3658IYX-GPR34-YL-365
4.55Single8JD6N-(3-chlorophenyl)pyridine-2-carboxamide8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.55Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
4.35Single5T04Neurotensin5T04-NTS1-Neurotensin
4.35Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.35Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
4.35Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
4.35Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
4.17Single4JKVTaladegib4JKV-SMO-Taladegib
4.17Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
4.00Single5V57TC1145V57-SMO-TC114
4.00Single7F1TMIP-1a7F1T-CCR5-MIP-1a
4.00Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.00Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
3.85Single6YVRNTS8-136YVR-NTS1-NTS8-13
3.85Single7SHEPI; PE7SHE-GPR158-PI; PE
3.85Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.85Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
3.85Single8XQJJN2418XQJ-Apelin-JN241
3.70Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
3.70Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
3.70Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
3.70Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
3.70Single8XVUCXCL28XVU-CXCR2-CXCL2
3.70Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
3.57Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
3.57Single6KNMJN241-96KNM-Apelin-JN241-9
3.57Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
3.57Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
3.45Single8XWNCXCL88XWN-CXCR2-CXCL8
3.33Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7

Consensus Members
Id Members
8IRU 8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
Net Summary
Imin 2.85
Number of Linked Nodes 823
Number of Links 1085
Number of Hubs 211
Number of Links mediated by Hubs 753
Number of Communities 17
Number of Nodes involved in Communities 307
Number of Links involved in Communities 479
Path Summary
Number Of Nodes in MetaPath 88
Number Of Links MetaPath 87
Number of Shortest Paths 3362484
Length Of Smallest Path 3
Average Path Length 30.8998
Length of Longest Path 55
Minimum Path Strength 1.245
Average Path Strength 6.24576
Maximum Path Strength 22.905
Minimum Path Correlation 0.7
Average Path Correlation 0.988555
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.7027
Average % Of Corr. Nodes 37.2701
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 64.7395
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
dopamine_on_gpd2_on_gp
d1_on_gp
d3_on_gp
d4_on_gp
d5_on_gp



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