Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg Int. Strength Num Of Links Community ConSurf
1A:A:N50 8.0125109
2A:A:V214 5.665455
3A:A:F219 6.675658
4A:A:M221 4.476508
5A:A:F222 5.742506
6A:A:K233 5.862519
7A:A:W234 4.7375409
8A:A:C237 5.7175418
9A:A:F246 5.08754149
10A:A:D249 9.984108
11A:A:D252 9.34754108
12A:A:Y253 8.5675409
13A:A:R265 10.7185109
14A:A:L270 6.16406
15A:A:F273 4.5085149
16A:A:W277 8.5285146
17A:A:W281 7.80333615
18A:A:I288 6.324119
19A:A:F290 5.2245119
20A:A:L291 4.4054129
21A:A:Q294 6.4054126
22A:A:I308 6.79254177
23A:A:F312 4.474178
24A:A:F315 11.01254176
25A:A:E330 7.5545123
26A:A:V334 4.535404
27A:A:K338 10.24254125
28A:A:Y339 6.70667603
29A:A:F340 10.74754176
30A:A:R342 5.562505
31A:A:F345 7.2775408
32A:A:Y360 7.395408
33A:A:T364 6.18754119
34A:A:N371 7.17754119
35A:A:R374 6.00254114
36A:A:F376 8.8525459
37A:A:I383 6.73458
38A:A:R385 7.815256
39A:A:Y391 6.6425404
40B:B:D27 5.0725408
41B:B:L51 6.47409
42B:B:H54 6.57286799
43B:B:K57 13.5575419
44B:B:W63 6.64167607
45B:B:Q75 8.8475419
46B:B:D76 6.166599
47B:B:I80 6.15333698
48B:B:I81 4.80254187
49B:B:W82 10.234599
50B:B:Y85 10.74754154
51B:B:K89 9.815499
52B:B:L95 4.2375408
53B:B:W99 10.122509
54B:B:M101 6.415419
55B:B:Y105 4.875717186
56B:B:N110 6.88754194
57B:B:Y111 6.155194
58B:B:D118 4.4675409
59B:B:Y124 7.0675406
60B:B:T128 4.355403
61B:B:H142 7.2775419
62B:B:Y145 5.81167618
63B:B:F151 5.26609
64B:B:L152 3.96403
65B:B:T159 4.6125419
66B:B:S161 6.8325419
67B:B:D163 6.7125419
68B:B:W169 9.266518
69B:B:F180 5.67567
70B:B:H183 7.47667669
71B:B:D186 7.274519
72B:B:F199 7.9075469
73B:B:V200 5.875436
74B:B:C204 5.61417
75B:B:D205 6.44469
76B:B:K209 10.64466
77B:B:W211 7.48833668
78B:B:F222 7.745438
79B:B:H225 9.38167639
80B:B:D228 6.124519
81B:B:F234 4.47405
82B:B:F235 8.9845206
83B:B:N237 9.334205
84B:B:F241 7.254536
85B:B:D247 8.125439
86B:B:T249 7.6825436
87B:B:R251 7.53333638
88B:B:F253 6.36833636
89B:B:D254 8.1875409
90B:B:R256 11.7175409
91B:B:D258 11.0925437
92B:B:Q259 4.09406
93B:B:M262 5.68404
94B:B:Y264 6.656505
95B:B:H266 4.07474
96B:B:I269 3.2475474
97B:B:F278 5.565407
98B:B:R283 8.47409
99B:B:Y289 6.20286777
100B:B:N295 8.385476
101B:B:W297 7.72478
102B:B:R304 6.446575
103B:B:V307 5.2875473
104B:B:L308 4.745407
105B:B:H311 6.4965309
106B:B:R314 10.6267618
107B:B:W332 14.3067619
108B:B:D333 6.01254309
109B:B:W339 7.435409
110G:G:L19 3.946509
111G:G:R27 8.4325438
112G:G:Y40 8.47254206
113G:G:D48 6.9665299
114G:G:P49 3.9425407
115G:G:L51 4.62506
116G:G:P60 8.434159
117G:G:F61 5.458336158
118L:L:Q6 7.5325400
119L:L:H14 8.0954320
120L:L:R20 8.14254210
121L:L:W23 5.7465160
122L:L:L24 8.8275400
123L:L:R25 3.4525400
124R:R:V31 6.064216
125R:R:K34 3.9854164
126R:R:Q37 6.5025407
127R:R:C108 4.95754229
128R:R:P132 5.55667689
129R:R:Y134 5.1785
130R:R:I135 5.78487
131R:R:F138 6.60571784
132R:R:Y145 5.18254134
133R:R:R146 6.165408
134R:R:R147 4.474133
135R:R:W154 5.27254229
136R:R:E155 8.60254134
137R:R:W164 5.45754135
138R:R:E169 3485
139R:R:Y191 5.054507
140R:R:Y195 6.25429727
141R:R:F212 5.12507
142R:R:T218 4.21407
143R:R:R219 7.358509
144R:R:F230 8.584528
145R:R:R233 9.13428
146R:R:F288 6.736507
147R:R:L289 4.438547
148R:R:Y290 5.62254349
149R:R:N295 11.4775428
150R:R:Y296 8.5125427
151R:R:Y297 8.3175406
152R:R:W298 11.58509
153R:R:L300 6.7725408
154R:R:E302 8.17409
155R:R:Y305 9.38408
156R:R:I310 4.944268
157R:R:F311 5.314266
158R:R:F314 16.22457
159R:R:F315 9.52429756
160R:R:E317 6.62406
161R:R:F335 6.176505
162R:R:W339 6.484548
163R:R:V342 3.44405
164R:R:R343 6.2025448
165R:R:W352 11.242548
166R:R:K359 4.4125443
167R:R:W361 6.2975448
168R:R:Q364 8.095447
169R:R:F378 9.3054359
170R:R:K405 3.635408
171R:R:F417 8.408336359
172R:R:H420 10.798528
173R:R:Y421 13.798528
174R:R:F424 9.05527
175R:R:M425 3.37406
176R:R:Y429 9.736546
177R:R:W437 7.296676315
178R:R:M441 7.9525406
179R:R:Y443 8.665424
180R:R:E444 7.88427
181R:R:M445 5.622506
182R:R:Q451 8.8025429
183R:R:Y459 7.3275408
184R:R:N463 5.19409
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Int. Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.

Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1B:B:M61 B:B:W63 70.81535.82NoYes067
2B:B:C317 B:B:M61 70.69994.86NoNo076
3B:B:C317 B:B:S316 70.58443.44NoNo079
4B:B:S316 B:B:W332 70.46884.94NoYes099
5B:B:K57 B:B:W332 46.464926.69YesYes199
6B:B:K57 B:B:Q75 46.261612.2YesYes199
7R:R:K388 R:R:V384 15.94744.55NoNo098
8R:R:I310 R:R:V384 16.06034.61YesNo2688
9R:R:I310 R:R:I381 24.12664.42YesNo089
10R:R:I381 R:R:L306 24.28877.14NoNo099
11A:A:Y391 R:R:L306 19.69938.21YesNo049
12A:A:Y391 R:R:R219 21.763411.32YesYes049
13R:R:N220 R:R:R219 96.35486.03NoYes099
14R:R:L215 R:R:N220 96.41355.49NoNo099
15R:R:F212 R:R:L215 99.49974.87YesNo079
16R:R:E469 R:R:F212 99.716510.49NoYes097
17R:R:E469 R:R:R214 99.770410.47NoNo097
18B:B:D312 R:R:R214 99.877713.1NoNo057
19B:B:D312 B:B:D333 99.93113.99NoYes059
20B:B:D333 B:B:H311 99.97463.78YesYes3099
21B:B:H311 B:B:T329 49.97336.85YesNo098
22B:B:T329 B:B:W339 49.95647.28NoYes089
23B:B:L308 B:B:W339 1005.69YesYes079
24B:B:L308 B:B:V296 99.71994.47YesNo075
25B:B:L286 B:B:V296 99.64954.47NoNo075
26B:B:L286 B:B:V327 99.5794.47NoNo076
27B:B:V327 G:G:L50 99.36654.47NoNo069
28G:G:D48 G:G:L50 99.16754.07YesNo2999
29G:G:D48 G:G:P49 78.2244.83YesYes097
30B:B:M325 G:G:P49 77.58613.35NoYes057
31B:B:H311 B:B:K337 50.22576.55YesNo096
32B:B:K337 B:B:W339 50.18574.64NoYes069
33A:A:D378 A:A:Y360 10.44076.9NoYes078
34A:A:I244 A:A:I285 21.9914.42NoNo087
35A:A:I285 A:A:L282 22.2094.28NoNo079
36A:A:L282 A:A:N279 22.36813.73NoNo098
37A:A:N279 A:A:W281 22.52954.52NoYes085
38A:A:W281 B:B:W332 23.11845.62YesYes159
39A:A:L291 A:A:Q294 12.69335.32YesYes1296
40A:A:L289 A:A:L291 17.99554.15NoYes099
41A:A:F345 A:A:L289 18.15928.53YesNo089
42A:A:F273 A:A:F345 18.8154.29YesYes098
43A:A:F273 A:A:V287 20.07293.93YesNo1495
44A:A:I244 A:A:V287 22.0757.68NoNo085
45B:B:G162 B:B:S161 24.26653.71NoYes199
46B:B:G162 B:B:Y145 24.52824.35NoYes198
47B:B:M101 B:B:Y145 30.27467.18YesYes198
48A:A:C237 B:B:M101 21.91234.86YesYes189
49A:A:C237 B:B:Q75 21.99067.63YesYes189
50B:B:M101 B:B:Y59 21.68878.38YesNo198
51B:B:Q75 B:B:Y59 21.84077.89YesNo198
52G:G:D48 G:G:L51 39.31686.79YesYes096
53B:B:R283 G:G:L51 37.92514.86YesYes096
54B:B:L300 B:B:R283 36.2849.72NoYes069
55B:B:L300 B:B:T34 35.97754.42NoNo065
56B:B:L30 B:B:T34 35.8244.42NoNo055
57B:B:L30 B:B:M262 35.36285.65NoYes054
58B:B:M262 B:B:Y264 34.745710.78YesYes045
59B:B:L285 B:B:Y264 23.05245.86NoYes065
60B:B:F278 B:B:L285 22.72298.53YesNo076
61B:B:F235 B:B:F278 22.23155.36YesYes067
62B:B:F235 B:B:N237 20.544614.5YesYes2065
63B:B:G238 B:B:N237 20.43023.39NoYes075
64B:B:F234 B:B:G238 20.09454.52YesNo057
65B:B:F234 B:B:V200 18.91525.24YesYes056
66B:B:G116 B:B:M101 13.41355.24NoYes099
67B:B:D118 B:B:G116 13.0881.68YesNo099
68B:B:D118 B:B:G115 11.1381.68YesNo099
69B:B:G115 B:B:L146 10.81293.42NoNo097
70B:B:L146 B:B:T159 10.50864.42NoYes079
71B:B:C149 B:B:T159 21.06475.07NoYes089
72B:B:C149 B:B:T102 20.42873.38NoNo088
73B:B:H142 B:B:S161 21.336912.55YesYes199
74B:B:H142 B:B:T159 11.19014.11YesYes199
75B:B:C148 B:B:T102 19.15633.38NoNo068
76B:B:C148 B:B:R150 17.88335.57NoNo066
77B:B:H62 B:B:R150 17.246611.28NoNo066
78B:B:H62 B:B:Y105 16.60974.36NoYes066
79B:B:T321 B:B:W63 73.65969.7NoYes077
80B:B:D323 B:B:M325 73.986711.09NoNo075
81R:R:H223 R:R:R219 75.525611.28NoYes099
82R:R:E302 R:R:H223 74.95718.62YesNo099
83R:R:E302 R:R:L226 82.91329.28YesNo099
84R:R:L226 R:R:S229 39.77724.5NoNo099
85R:R:N295 R:R:S229 37.06037.45YesNo089
86R:R:N295 R:R:R233 73.69513.26YesYes288
87L:L:E4 R:R:R233 59.45284.65NoYes208
88L:L:E4 R:R:M445 59.68148.12NoYes006
89L:L:L7 R:R:M445 54.73455.65NoYes006
90R:R:F230 R:R:L226 43.14027.31YesNo089
91R:R:F230 R:R:N295 36.836218.12YesYes288
92R:R:R233 R:R:Y195 14.186711.32YesYes287
93R:R:I237 R:R:Y195 11.01767.25NoYes077
94R:R:F288 R:R:I237 10.75823.77YesNo077
95L:L:L7 R:R:F184 50.90133.65NoNo006
96L:L:L11 R:R:F184 48.22028.53NoNo006
97L:L:L11 L:L:L15 48.44674.15NoNo000
98L:L:H14 L:L:L15 47.33773.86YesNo3200
99L:L:H14 L:L:M18 47.731113.13YesNo000
100L:L:M18 L:L:S17 46.64921.53NoNo000
101L:L:R20 L:L:S17 37.8923.95YesNo2100
102L:L:R20 R:R:D137 31.128613.1YesNo005
103L:L:L24 R:R:D137 30.855714.93YesNo005
104R:R:M32 R:R:Y136 12.49475.99NoNo064
105R:R:M32 R:R:Q37 10.87724.08NoYes067
106L:L:L24 R:R:F138 27.252212.18YesYes004
107R:R:F138 R:R:P132 19.658.67YesYes849
108R:R:L116 R:R:P132 16.6566.57NoYes859
109R:R:L116 R:R:W118 16.55999.11NoNo059
110R:R:D113 R:R:W118 15.70015.58NoNo099
111R:R:A44 R:R:Y134 10.24645.34NoYes075
112R:R:D113 R:R:E111 13.40115.59NoNo097
113R:R:E111 R:R:R146 10.20745.82NoYes078
114B:B:D323 B:B:T321 73.72917.23NoNo2877
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1 Node2 LinkStrength Comm IsNode1Hub? IsNode2Hub? Node1Cons Node2Cons Node1Shell Node2Shell
L:L:V2 R:R:Q364 7.16 4 No Yes 0 7 0 1
L:L:V2 R:R:I367 4.61 4 No No 0 7 0 1
L:L:S3 R:R:E444 11.5 0 No Yes 0 7 0 1
L:L:E4 R:R:Y195 6.73 2 No Yes 0 7 0 1
L:L:E4 R:R:R233 4.65 2 No Yes 0 8 0 1
L:L:E4 R:R:M445 8.12 2 No Yes 0 6 0 1
L:L:I5 R:R:L289 4.28 4 No Yes 0 7 0 1
L:L:I5 R:R:Q364 4.12 4 No Yes 0 7 0 1
L:L:Q6 R:R:Y429 12.4 0 Yes Yes 0 6 0 1
L:L:Q6 R:R:M441 6.8 0 Yes Yes 0 6 0 1
L:L:L7 R:R:F184 3.65 0 No No 0 6 0 1
L:L:L7 R:R:M441 5.65 0 No Yes 0 6 0 1
L:L:L7 R:R:M445 5.65 0 No Yes 0 6 0 1
L:L:M8 R:R:F288 3.73 0 No Yes 0 7 0 1
L:L:M8 R:R:D353 4.16 0 No No 0 5 0 1
L:L:H9 R:R:S355 8.37 4 No No 0 7 0 1
L:L:H9 R:R:K360 3.93 4 No No 0 7 0 1
L:L:H9 R:R:Y429 4.36 4 No Yes 0 6 0 1
L:L:N10 R:R:V432 4.43 31 No No 0 5 0 1
L:L:N10 R:R:W437 7.91 31 No Yes 0 5 0 1
L:L:L11 R:R:F184 8.53 0 No No 0 6 0 1
L:L:L11 R:R:Y245 14.07 0 No No 0 4 0 1
L:L:K13 R:R:V31 9.11 0 No Yes 0 6 0 1
L:L:H14 R:R:E180 8.62 32 Yes No 0 3 0 1
L:L:H14 R:R:R181 6.77 32 Yes No 0 3 0 1
L:L:L15 R:R:R181 3.64 32 No No 0 3 0 1
L:L:N16 R:R:T33 7.31 16 No No 0 7 0 1
L:L:N16 R:R:E35 5.26 16 No No 0 5 0 1
L:L:S17 R:R:V31 4.85 21 No Yes 0 6 0 1
L:L:M18 R:R:E177 5.41 0 No No 0 1 0 1
L:L:E19 R:R:K34 4.05 0 No Yes 0 4 0 1
L:L:R20 R:R:V31 5.23 21 Yes Yes 0 6 0 1
L:L:R20 R:R:Y136 10.29 21 Yes No 0 4 0 1
L:L:R20 R:R:D137 13.1 21 Yes No 0 5 0 1
L:L:W23 R:R:K34 3.48 16 Yes Yes 0 4 0 1
L:L:W23 R:R:Q37 4.38 16 Yes Yes 0 7 0 1
L:L:W23 R:R:I38 5.87 16 Yes No 0 7 0 1
L:L:L24 R:R:D137 14.93 0 Yes No 0 5 0 1
L:L:L24 R:R:F138 12.18 0 Yes Yes 0 4 0 1
L:L:R25 R:R:V171 3.92 0 Yes No 0 3 0 1
L:L:L28 R:R:F138 7.31 0 No Yes 0 4 0 1
L:L:D30 R:R:H114 6.3 33 No No 0 4 0 1
L:L:V31 R:R:D113 4.38 0 No No 0 9 0 1
L:L:V31 R:R:H114 4.15 0 No No 0 4 0 1
L:L:F34 R:R:H114 5.66 33 No No 0 4 0 1
R:R:V31 R:R:Y136 5.05 21 Yes No 6 4 1 1
R:R:E36 R:R:M32 10.83 0 No No 6 6 2 2
R:R:M32 R:R:Q37 4.08 0 No Yes 6 7 2 1
R:R:M32 R:R:Y136 5.99 0 No No 6 4 2 1
R:R:E35 R:R:T33 12.7 16 No No 5 7 1 1
R:R:E36 R:R:T33 15.52 0 No No 6 7 2 1
R:R:E35 R:R:K34 4.05 16 No Yes 5 4 1 1
R:R:I38 R:R:K34 4.36 16 No Yes 7 4 1 1
R:R:L40 R:R:Q37 9.32 0 No Yes 5 7 2 1
R:R:I135 R:R:Q37 8.23 8 Yes Yes 7 7 2 1
R:R:D113 R:R:E111 15.59 0 No No 9 7 1 2
R:R:D113 R:R:W118 5.58 0 No No 9 9 1 2
R:R:I135 R:R:P132 5.08 8 Yes Yes 7 9 2 2
R:R:F138 R:R:P132 8.67 8 Yes Yes 4 9 1 2
R:R:F138 R:R:I135 3.77 8 Yes Yes 4 7 1 2
R:R:F138 R:R:Y167 6.19 8 Yes No 4 5 1 2
R:R:C170 R:R:F138 4.19 8 No Yes 9 4 2 1
R:R:F138 R:R:V171 3.93 8 Yes No 4 3 1 1
R:R:E180 R:R:V432 5.7 0 No No 3 5 1 1
R:R:D185 R:R:R181 9.53 0 No No 2 3 2 1
R:R:F184 R:R:W437 4.01 0 No Yes 6 5 1 1
R:R:L187 R:R:M441 4.24 0 No Yes 5 6 2 1
R:R:L187 R:R:M445 4.24 0 No Yes 5 6 2 1
R:R:Y191 R:R:Y195 4.96 0 Yes Yes 7 7 2 1
R:R:M445 R:R:Y191 7.18 0 Yes Yes 6 7 1 2
R:R:R233 R:R:Y195 11.32 2 Yes Yes 8 7 1 1
R:R:A234 R:R:Y195 5.34 0 No Yes 8 7 2 1
R:R:I237 R:R:Y195 7.25 0 No Yes 7 7 2 1
R:R:S449 R:R:Y195 5.09 0 No Yes 9 7 2 1
R:R:L292 R:R:R233 7.29 0 No Yes 6 8 2 1
R:R:N295 R:R:R233 13.26 2 Yes Yes 8 8 2 1
R:R:F288 R:R:S236 3.96 0 Yes No 7 7 1 2
R:R:F288 R:R:I237 3.77 0 Yes No 7 7 1 2
R:R:K240 R:R:L244 4.23 0 No No 7 5 2 2
R:R:F288 R:R:K240 16.13 0 Yes No 7 7 1 2
R:R:L244 R:R:Y245 9.38 0 No No 5 4 2 1
R:R:F288 R:R:L289 6.09 0 Yes Yes 7 7 1 1
R:R:L289 R:R:W339 4.56 4 Yes Yes 7 8 1 2
R:R:I363 R:R:L289 4.28 4 No Yes 7 7 2 1
R:R:L292 R:R:Y296 5.86 0 No Yes 6 7 2 2
R:R:I367 R:R:Y296 8.46 0 No Yes 7 7 1 2
R:R:I363 R:R:W339 10.57 4 No Yes 7 8 2 2
R:R:C351 R:R:D353 4.67 0 No No 9 5 2 1
R:R:D353 R:R:L354 6.79 0 No No 5 5 1 1
R:R:K360 R:R:W361 8.12 4 No Yes 7 8 1 2
R:R:K360 R:R:Y429 17.91 4 No Yes 7 6 1 1
R:R:Q364 R:R:W361 10.95 4 Yes Yes 7 8 1 2
R:R:W361 R:R:Y429 3.86 4 Yes Yes 8 6 2 1
R:R:Q364 R:R:Y429 10.15 4 Yes Yes 7 6 1 1
R:R:F424 R:R:Y443 7.22 2 Yes Yes 7 4 2 2
R:R:E444 R:R:F424 3.5 2 Yes Yes 7 7 1 2
R:R:T430 R:R:W437 3.64 0 No Yes 5 5 2 1
R:R:V432 R:R:W437 9.81 31 No Yes 5 5 1 1
R:R:M441 R:R:W437 15.12 0 Yes Yes 6 5 1 1
R:R:E444 R:R:Y443 3.37 2 Yes Yes 7 4 1 2
R:R:E444 R:R:N448 13.15 2 Yes No 7 6 1 2
R:R:Q438 R:R:W437 3.29 0 No Yes 4 5 2 1
R:R:S168 R:R:V171 3.23 0 No No 6 3 2 1
R:R:F238 R:R:Y195 3.09 0 No Yes 7 7 2 1
R:R:L244 R:R:V285 2.98 0 No No 5 6 2 2
R:R:L289 R:R:V285 2.98 4 Yes No 7 6 1 2
R:R:I190 R:R:M445 2.92 0 No Yes 6 6 2 1
L:L:G12 R:R:L354 1.71 0 No No 0 5 0 1
R:R:E177 R:R:T178 1.41 0 No No 1 3 1 2

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
70.37Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
69.23Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
69.23Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
69.23Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
68.97Consensuspth_onOrthosteric Ligandpth1_on pth2_on
67.86Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
65.52Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
65.38Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
64.29Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
62.50Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
62.07Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
61.54Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
60.61Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
60.00Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
60.00Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
59.26Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
58.33Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
57.69Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
57.69Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
57.14Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
57.14Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
57.14Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
57.14Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
57.14Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
57.14Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
57.14Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
57.14Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
56.00Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
55.56Single6FJ3PTH6FJ3-PTH1-PTH
55.56Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
55.56Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
55.56Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
55.56Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
55.17Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
55.17Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
54.84Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
54.55Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
53.85Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
53.57Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
53.57Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
53.33Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
52.78Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
51.85Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
51.85Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
51.85Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
51.85Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
51.61Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
50.00Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
50.00Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
50.00Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
50.00Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
50.00Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
50.00Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
50.00Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
50.00Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
50.00Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
48.48Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
48.48Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
48.28Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
48.28Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
48.28Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
48.28Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
48.28Consensusglp_onOrthosteric Ligandglp1_on glp2_on
48.28Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
48.15Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
48.15Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
48.15Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
48.15Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
48.00Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
48.00Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
46.67Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
46.67Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
46.43Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
46.43Consensuspac_onOrthosteric Ligandpac1_on
46.15Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
44.83Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
44.83Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
44.44Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
44.44Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
43.33Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
42.86Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
42.86Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
42.42Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
41.38Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
41.38Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
41.18Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
41.18Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
40.62Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
40.00Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
40.00Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
40.00Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
39.39Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
39.29Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
38.71Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
38.71Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
38.24Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
38.24Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
37.93Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
37.93Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
37.50Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
37.50Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
37.14Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
37.14Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
36.67Consensuscalcitonin_onOrthosteric Ligandctlike_on
35.48Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
35.48Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
35.48Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
35.29Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
34.62Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
34.62Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
34.48Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
34.38Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
34.38Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
34.38Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
34.29Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
33.33Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
33.33Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
33.33Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
33.33Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
33.33Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
32.35Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
32.35Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
32.14Single4XT1Fractalkine4XT1-US28-Fractalkine
32.14Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
31.43Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
31.25Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
31.03Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
30.30Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
30.30Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
29.41Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
29.41Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
29.41Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
29.41Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
29.03Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
29.03Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
29.03Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
28.57Single6IGKEndothelin-36IGK-ETB-Endothelin-3
28.57Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
28.57Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
28.12Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
28.12Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
28.00Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
28.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
27.78Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
27.59Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
27.59Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
27.59Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
27.27Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
27.27Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
27.27Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
27.27Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
26.92Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
26.83Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
26.67Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
26.67Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
26.67Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
26.67Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
26.47Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
26.47Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.47Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
26.47Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.47Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.47Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
26.47Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
26.19Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
26.09Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
25.93Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
25.93Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
25.93Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
25.81Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
25.81Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
25.81Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
25.81Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
25.81Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
25.81Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
25.71Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
25.71Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
25.71Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
25.00Single5GLHEndothelin-15GLH-ETB-Endothelin-1
25.00Single7T32ZM-2413857T32-A2A-ZM-241385
25.00Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
25.00Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
25.00Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
25.00Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
25.00Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
25.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
25.00Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
25.00Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
25.00Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
24.39Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
24.24Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
24.24Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
24.24Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
24.24Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
24.24Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
24.24Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
24.24Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
24.24Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
24.24Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.14Single3NY9ICI118-5513NY9-β2-ICI118-551
24.14Single4UG2CGS216804UG2-A2A-CGS21680
24.14Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
24.14Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
24.14Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8QJ2pN1628QJ2-MC4-pN162-Gs
24.14Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
24.14Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
24.14Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
24.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
24.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
24.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
23.68Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
23.68Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
23.53Single4XT3Fractalkine4XT3-US28-Fractalkine
23.53Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
23.53Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
23.53Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
23.53Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
23.53Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
23.53Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
23.53Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
23.53Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
23.53Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
23.33Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
23.33Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
23.33Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
23.33Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
23.33Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
23.33Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
23.33Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
23.33Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single5N2RPSB-365N2R-A2A-PSB-36-Na
23.08Single5N2SPSB365N2S-A1-PSB36
23.08Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
23.08Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
23.08Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
23.08Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
23.08Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
23.08Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
23.08Single8QOTNanobody-E8QOT-μ-Nanobody-E
23.08Single8S4DCMF-0198S4D-Apelin-CMF-019
23.08Single8TF5Oleic acid8TF5-GPR6-Oleic acid
23.08Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
23.08Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single9EHSLUF76029EHS-A3A-LUF7602
23.08Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
23.08Consensusadenosine_offOrthosteric Liganda1_off a2_off
23.08Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
22.86Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
22.86Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
22.86Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
22.73Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.58Single3QAKUK-4320973QAK-A2A-UK-432097
22.58Single6HLOAprepitant6HLO-NK1-Aprepitant
22.58Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
22.58Single7XNACYN1548067XNA-SST2-CYN154806
22.58Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
22.58Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
22.58Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
22.58Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
22.58Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
22.22Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
22.22Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
22.22Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
22.22Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
22.22Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
22.22Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
22.22Single7F1TMIP-1a7F1T-CCR5-MIP-1a
22.22Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
22.22Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
22.22Single7PX4PSB-21137PX4-A2A-PSB-2113
22.22Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
22.22Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
22.22Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
22.22Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
22.22Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
22.22Single8IY6Endothelin-18IY6-ETB-Endothelin-1
22.22Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
22.22Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
22.22Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
22.22Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
22.22Consensusendothelin_onOrthosteric Ligandetb_on eta_on
22.22Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
22.22Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
21.95Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
21.88Single3OE0CVX153OE0-CXCR4-CVX15
21.88Single5WF5UK-4320975WF5-A2A-UK-432097
21.88Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
21.88Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
21.88Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
21.88Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
21.88Consensusangiotensin_onOrthosteric Ligandat1_on
21.88Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
21.88Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
21.88Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
21.88Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
21.88Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
21.62Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
21.62Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
21.62Consensusbombesin_onOrthosteric Ligandbb2_on
21.62Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
21.62Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.62Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
21.62Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
21.62Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
21.43Single4XEENeurotensin4XEE-NTS1-Neurotensin
21.43Single4XESNeurotensin4XES-NTS1-Neurotensin
21.43Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
21.43Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
21.43Single6OS2TRV0266OS2-AT1-TRV026
21.43Single6YVRNTS8-136YVR-NTS1-NTS8-13
21.43Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
21.43Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
21.43Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
21.43Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
21.43Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
21.43Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
21.43Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
21.43Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.43Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
21.43Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
21.43Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
21.43Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
21.43Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
21.43Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
21.43Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
21.43Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
21.43Consensuslpa_offOrthosteric Ligandlpa1_off
21.43Consensuslpl_offOrthosteric Ligands1p_off lpa_off
21.43Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
21.43Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
21.21Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
21.21Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
21.21Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
21.21Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.21Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
21.21Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
21.21Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
21.21Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
21.21Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
21.21Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
21.21Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
21.21Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
21.21Consensusvasop-oxy_onOrthosteric Ligandv2_on
21.21Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
21.05Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
21.05Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.83Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
20.83Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
20.83Single4BWBNeurotensin4BWB-NTS1-Neurotensin
20.83Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
20.83Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
20.83Single5U09Taranabant5U09-CB1-Taranabant
20.83Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
20.83Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
20.83Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
20.83Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
20.83Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
20.83Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
20.83Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GNGIstradefylline8GNG-A2A-Istradefylline
20.83Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
20.83Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
20.83Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
20.83Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
20.83Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
20.69Single4BUONeurotensin4BUO-NTS1-Neurotensin
20.69Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
20.69Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
20.69Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
20.69Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
20.69Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
20.69Single7EZCUKA7EZC-A2A-UKA
20.69Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
20.69Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
20.69Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
20.69Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
20.69Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
20.69Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
20.69Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
20.69Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
20.69Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
20.69Single8XVUCXCL28XVU-CXCR2-CXCL2
20.69Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
20.69Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
20.69Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
20.69Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
20.69Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.69Consensuscck_onOrthosteric Ligandccka_on cckb_on
20.69Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
20.69Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
20.69Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
20.59Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
20.59Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
20.59Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
20.59Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
20.59Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
20.59Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Single8ZRTET-18ZRT-ETB-ET-1
20.59Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
20.59Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
20.59Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
20.59Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
20.51Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.00Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
20.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
20.00Single5IUBQ274563445IUB-A2A-Q27456344-Na
20.00Single5JTBZM-2413855JTB-A2A-ZM-241385
20.00Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
20.00Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
20.00Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
20.00Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
20.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
20.00Single7AROLUF58337ARO-A2A-LUF5833-Na
20.00Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
20.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
20.00Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
20.00Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
20.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
20.00Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
20.00Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
20.00Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
20.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
20.00Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
20.00Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
20.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
20.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
20.00Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
20.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
20.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
20.00Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
20.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
20.00Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
20.00Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
20.00Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
20.00Consensusa2_offOrthosteric Liganda2a_off
20.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
20.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
20.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
20.00Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
20.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
20.00Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
20.00Consensusgrh_offOrthosteric Ligandgnrh1_off
20.00Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
20.00Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
20.00Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
20.00Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
19.51Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
19.44Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
19.44Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
19.44Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
19.44Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
19.44Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
19.44Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
19.35Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
19.35Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
19.35Single7F8XNN90567F8X-CCKA-NN9056
19.35Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
19.35Single7QA8Peptide7QA8-STE2-Peptide
19.35Single7QA8Peptide7QA8-STE2-Peptide
19.35Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
19.35Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
19.35Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
19.35Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
19.35Single8WDTphotoNECA8WDT-A2A-photoNECA
19.35Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
19.35Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.35Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
19.35Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
19.35Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
19.35Consensussomatostatin_offOrthosteric Ligandsst2_off
19.35Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.23Single3EMLZM-2413853EML-A2A-ZM-241385
19.23Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
19.23Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
19.23Single5IU8Q274563475IU8-A2A-Q27456347-Na
19.23Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
19.23Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
19.23Single5UENDU1725UEN-A1-DU172
19.23Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
19.23Single6D27CAY104716D27-DP2-CAY10471
19.23Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
19.23Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
19.23Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
19.23Single6PS1Timolol6PS1-β2-Timolol
19.23Single6S0LZM-2413856S0L-A2A-ZM-241385
19.23Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
19.23Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
19.23Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
19.23Single7PYRPSB-21157PYR-A2A-PSB-2115
19.23Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
19.23Single7V3ZCP559407V3Z-CB1-CP55940
19.23Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
19.23Single8CU6LJ-45178CU6-A2A-LJ-4517
19.23Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
19.23Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
19.23Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
19.23Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
19.23Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
19.23Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
19.23Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
19.23Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
19.23Single9AS1DMT9AS1-5-HT2A-DMT
19.23Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
19.23Single9CHXS-Carazolol9CHX-β2-S-Carazolol
19.23Consensusa3_onOrthosteric Liganda3a_on
19.23Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
19.23Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
19.23Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
19.23Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
19.05Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
18.92Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
18.92Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
18.75Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
18.75Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
18.75Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
18.75Single7SK5CXCL127SK5-ACKR3-CXCL12
18.75Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
18.75Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
18.75Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
18.75Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
18.75Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
18.75Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.75Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
18.75Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.75Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
18.75Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
18.75Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
18.52Single5C1MBU725C1M-μ-BU72
18.52Single5IUAQ274563485IUA-A2A-Q27456348-Na
18.52Single5JQHS-Carazolol5JQH-β2-S-Carazolol
18.52Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
18.52Single5TVNLSD5TVN-5-HT2B-LSD
18.52Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
18.52Single6D26Fevipiprant6D26-DP2-Fevipiprant
18.52Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
18.52Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
18.52Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
18.52Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
18.52Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
18.52Single6PS6Timolol6PS6-β2-Timolol
18.52Single6S0QZM-2413856S0Q-A2A-ZM-241385
18.52Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
18.52Single7C61Ergotamine7C61-5-HT1B-Ergotamine
18.52Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
18.52Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
18.52Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
18.52Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
18.52Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
18.52Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
18.52Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
18.52Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8GNEKW-63568GNE-A2A-KW-6356-Na
18.52Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
18.52Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
18.52Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
18.52Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
18.52Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
18.52Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
18.52Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
18.52Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
18.52Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
18.52Single9B9ZA1AKO9B9Z-CB1-A1AKO
18.52Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
18.52Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
18.52Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
18.52Consensusa3_on_gpOrthosteric Liganda3a_on_gp
18.52Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
18.52Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
18.52Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
18.52Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
18.52Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
18.52Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
18.52Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
18.52Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
18.52Consensusdp_offOrthosteric Liganddp2_off
18.52Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
18.52Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
18.52Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
18.52Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.52Consensustrace-amine_onOrthosteric Ligandta1_on
18.42Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
18.42Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
18.42Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
18.42Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
18.18Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
18.18Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
18.18Single8A2OTheophylline8A2O-A2A-Theophylline-Na
18.18Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
18.18Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.18Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.18Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
18.18Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
18.18Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.18Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
18.18Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
17.95Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
17.95Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
17.95Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
17.86Single2YDVNECA2YDV-A2A-NECA
17.86Single3P0GBI1671073P0G-β2-BI167107
17.86Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
17.86Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
17.86Single4BV0Neurotensin4BV0-NTS1-Neurotensin
17.86Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
17.86Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
17.86Single4UHRCGS216804UHR-A2A-CGS21680
17.86Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
17.86Single5G53NECA5G53-A2A-NECA-Gs
17.86Single5XR8AM8415XR8-CB1-AM841
17.86Single5XRAAM115425XRA-CB1-AM11542
17.86Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
17.86Single6WGTLSD6WGT-5-HT2A-LSD
17.86Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
17.86Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
17.86Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
17.86Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
17.86Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
17.86Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
17.86Single7TUYGSK682753A7TUY-GPR183-GSK682753A
17.86Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
17.86Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
17.86Single8E0GBU728E0G-μ-BU72
17.86Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
17.86Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
17.86Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
17.86Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
17.86Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
17.86Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
17.86Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
17.86Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
17.86Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.86Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
17.86Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
17.86Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
17.86Single8ZWFJR14a8ZWF-C3aB-JR14a
17.86Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
17.86Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
17.86Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
17.86Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
17.86Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
17.86Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
17.86Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
17.86Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
17.86Consensuslpa_onOrthosteric Ligandlpa1_on
17.86Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
17.86Consensusneurotensin_onOrthosteric Ligandnts1_on
17.86Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.86Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
17.65Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
17.65Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
17.65Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
17.65Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
17.65Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
17.65Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
17.65Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
17.65Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
17.65Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
17.65Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
17.65Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
17.65Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
17.65Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
17.65Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
17.50Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
17.39Single4XNWMRS25004XNW-P2Y1-MRS2500
17.39Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
17.39Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
17.39Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
17.39Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
17.39Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
17.39Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
17.39Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
17.24Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
17.24Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
17.24Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
17.24Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
17.24Single6CM4Risperidone6CM4-D2-Risperidone
17.24Single6IIURamatroban6IIU-TXA2-Ramatroban
17.24Single6KQICP559406KQI-CB1-CP55940-Org27569
17.24Single6MXTSalmeterol6MXT-β2-Salmeterol
17.24Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
17.24Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
17.24Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
17.24Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
17.24Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
17.24Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
17.24Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
17.24Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
17.24Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
17.24Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
17.24Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
17.24Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
17.24Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
17.24Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
17.24Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
17.24Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
17.24Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
17.24Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
17.24Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
17.24Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
17.24Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
17.24Single8JJ8Formoterol8JJ8-β2-Formoterol
17.24Single8JJLOlodaterol8JJL-β2-Olodaterol
17.24Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
17.24Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
17.24Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
17.24Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8XWMCXCL68XWM-CXCR2-CXCL6
17.24Single8XWSCXCL58XWS-CXCR2-CXCL5
17.24Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
17.24Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
17.24Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
17.24Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
17.24Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
17.24Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
17.24Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
17.24Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
17.24Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
17.24Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
17.24Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
17.24Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
17.24Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
17.24Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
17.24Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.24Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
17.24Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
17.24Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
17.24Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
17.24Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.24Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
17.14Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
17.14Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
17.14Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
17.14Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
17.14Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
17.14Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
17.14Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
17.14Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
16.67Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
16.67Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
16.67Single3OE9IT1t3OE9-CXCR4-IT1t
16.67Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
16.67Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
16.67Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
16.67Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
16.67Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
16.67Single6LI0C176LI0-GPR52-C17
16.67Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
16.67Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
16.67Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.67Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
16.67Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
16.67Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
16.67Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
16.67Single7SK3CXCL127SK3-ACKR3-CXCL12
16.67Single7UM4AS26747237UM4-5-HT5A-AS2674723
16.67Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
16.67Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
16.67Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
16.67Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
16.67Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
16.67Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
16.67Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
16.67Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
16.67Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
16.67Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
16.67Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
16.67Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
16.67Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
16.67Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
16.67Single8K5BNiacin8K5B-HCA2-Niacin
16.67Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
16.67Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
16.67Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
16.67Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
16.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
16.67Single8XWFCXCL38XWF-CXCR2-CXCL3
16.67Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
16.67Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
16.67Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
16.67Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
16.67Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9B9Y7DY9B9Y-CB1-7DY
16.67Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
16.67Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
16.67Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
16.67Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
16.67Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.67Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.67Consensuschemerin_onOrthosteric Ligandcml1_on
16.67Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
16.67Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
16.67Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
16.67Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
16.67Consensusprostanoid_offOrthosteric Ligandep_off dp_off
16.67Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
16.67Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
16.67Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
16.67Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
16.28Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
16.22Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
16.22Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
16.22Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
16.22Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
16.22Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
16.13Single5WF6UK-4320975WF6-A2A-UK-432097
16.13Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
16.13Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
16.13Single6PT3DPI-2876PT3-δ-DPI-287
16.13Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
16.13Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
16.13Single7XN9L-054,5227XN9-SST2-L-054,522
16.13Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
16.13Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
16.13Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
16.13Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
16.13Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
16.13Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
16.13Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
16.13Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
16.13Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
16.13Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
16.13Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
16.13Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
16.13Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
16.13Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
16.00Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
16.00Single3PWHZM-2413853PWH-A2A-ZM-241385
16.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
16.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
16.00Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
16.00Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
16.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
16.00Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
16.00Single7BR3Elagolix7BR3-GnRH1-Elagolix
16.00Single7F8ULintitript7F8U-CCKA-Lintitript
16.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
16.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
16.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
16.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
16.00Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
16.00Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
16.00Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
16.00Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
16.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
16.00Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
16.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
16.00Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.00Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
16.00Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
16.00Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
16.00Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
16.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
16.00Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
16.00Single8IWESpermidine8IWE-TA9-Spermidine
16.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
16.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
16.00Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
16.00Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
16.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
16.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
16.00Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
16.00Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
16.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
16.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
16.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
16.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
16.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
16.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
16.00Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
16.00Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
16.00Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
16.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
16.00Consensusangiotensin_offOrthosteric Ligandat1_off
16.00Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
16.00Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
16.00Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
16.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
16.00Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
16.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
16.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
16.00Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
16.00Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
16.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
16.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.79Single6IGLIRL16206IGL-ETB-IRL1620
15.79Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
15.79Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
15.79Consensusbradykinin_onOrthosteric Ligandbk2_on
15.79Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
15.79Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
15.79Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
15.79Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
15.62Single4IARErgotamine4IAR-5-HT1B-Ergotamine
15.62Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
15.62Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
15.62Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
15.62Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
15.62Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
15.62Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
15.62Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
15.62Single8IEBA1LYA8IEB-GPR156-A1LYA
15.62Single8IEIA1LYA8IEI-GPR156-A1LYA
15.62Single8IEPA1LYA8IEP-GPR156-A1LYA
15.62Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
15.62Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
15.62Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.62Single8XWNCXCL88XWN-CXCR2-CXCL8
15.62Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
15.62Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
15.62Consensuslpl_onOrthosteric Ligands1p_on lpa_on
15.62Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
15.38Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
15.38Single2YDOAdenosine2YDO-A2A-Adenosine
15.38Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
15.38Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
15.38Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
15.38Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
15.38Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
15.38Single5UVIZM-2413855UVI-A2A-ZM-241385
15.38Single6AQFZM-2413856AQF-A2A-ZM-241385
15.38Single6KUXRS-799486KUX-α2a-RS-79948
15.38Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
15.38Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
15.38Single6MH8ZM-2413856MH8-A2A-ZM-241385
15.38Single6PS0S-Carazolol6PS0-β2-S-Carazolol
15.38Single6PS4ICI118-5516PS4-β2-ICI118-551
15.38Single6PS5S-Propranolol6PS5-β2-S-Propranolol
15.38Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
15.38Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
15.38Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
15.38Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
15.38Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
15.38Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
15.38Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
15.38Single7F61PF-036547467F61-H3-PF-03654746
15.38Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
15.38Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
15.38Single7UL3Famotidine7UL3-H2-Famotidine
15.38Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
15.38Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
15.38Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.38Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
15.38Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
15.38Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
15.38Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
15.38Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
15.38Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
15.38Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
15.38Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
15.38Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
15.38Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
15.38Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
15.38Single8K5CAcipimox8K5C-HCA2-Acipimox
15.38Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
15.38Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
15.38Single8RLNLUF58348RLN-A2A-LUF5834
15.38Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
15.38Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
15.38Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
15.38Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
15.38Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
15.38Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
15.38Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
15.38Single9AS5Mescaline9AS5-5-HT2A-Mescaline
15.38Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
15.38Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9BA0A1AKN9BA0-CB1-A1AKN
15.38Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
15.38Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
15.38Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
15.38Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
15.38Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
15.38Consensushca_onOrthosteric Ligandhca2_on
15.38Consensusopsins_offOrthosteric Ligandrhodopsin_off
15.38Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.38Consensussensory_offOrthosteric Ligandopsins_off
15.15Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
15.15Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
15.15Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
15.15Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
15.15Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
15.15Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
15.15Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
15.15Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
15.15Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
15.15Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
15.15Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
15.15Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
15.00Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
15.00Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
14.81Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
14.81Single2Y01Dobutamine2Y01-β1-Dobutamine
14.81Single2Y02Carmoterol2Y02-β1-Carmoterol
14.81Single2Y04Salbutamol2Y04-β1-Salbutamol
14.81Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
14.81Single3NY8ICI118-5513NY8-β2-ICI118-551
14.81Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
14.81Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
14.81Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
14.81Single4DAJTiotropium4DAJ-M3-Tiotropium
14.81Single4GBRS-Carazolol4GBR-β2-S-Carazolol
14.81Single4QKX35V4QKX-β2-35V
14.81Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
14.81Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
14.81Single4YAYZD-71554YAY-AT1-ZD-7155
14.81Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
14.81Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
14.81Single5T04Neurotensin5T04-NTS1-Neurotensin
14.81Single5TGZAM65385TGZ-CB1-AM6538
14.81Single5UIGCmpd-15UIG-A2A-Cmpd-1
14.81Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
14.81Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
14.81Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
14.81Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
14.81Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
14.81Single6H7MSalbutamol6H7M-β1-Salbutamol
14.81Single6IIVDaltroban6IIV-TXA2-Daltroban
14.81Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
14.81Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
14.81Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
14.81Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
14.81Single7BU7BI1671077BU7-β1-BI167107
14.81Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
14.81Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
14.81Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
14.81Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
14.81Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
14.81Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
14.81Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
14.81Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
14.81Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
14.81Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
14.81Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
14.81Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
14.81Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
14.81Single7WC7Lisuride7WC7-5-HT2A-Lisuride
14.81Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
14.81Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
14.81Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
14.81Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
14.81Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
14.81Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
14.81Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
14.81Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
14.81Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
14.81Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
14.81Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
14.81Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
14.81Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
14.81Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
14.81Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
14.81Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
14.81Single8JJOAlprenolol8JJO-β2-Alprenolol
14.81Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
14.81Single8JXRLSD8JXR-D1-LSD
14.81Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
14.81Single8T1WCVN4248T1W-GPR6-CVN424
14.81Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
14.81Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
14.81Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
14.81Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
14.81Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
14.81Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
14.81Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
14.81Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
14.81Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
14.81Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
14.81Single9H37A1IR09H37-A2A-A1IR0-Na
14.81Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
14.81Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
14.81Consensus5ht5_onOrthosteric Ligand5ht5a_on
14.81Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
14.81Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
14.81Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
14.81Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
14.81Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
14.81Consensusdopamine_offOrthosteric Ligandd2_off d3_off
14.81Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
14.81Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
14.81Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
14.81Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
14.81Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
14.81Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
14.81Consensushca_on_gpOrthosteric Ligandhca2_on_gp
14.71Single6PT2KGCHM076PT2-δ-KGCHM07
14.71Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
14.71Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.71Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
14.71Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
14.71Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
14.71Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
14.71Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
14.71Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
14.71Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.63Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
14.29Single2RH1S-Carazolol2RH1-β2-S-Carazolol
14.29Single2Y00Dobutamine2Y00-β1-Dobutamine
14.29Single2Y03Isoprenaline2Y03-β1-Isoprenaline
14.29Single2YCWS-Carazolol2YCW-β1-S-Carazolol
14.29Single4JKVTaladegib4JKV-SMO-Taladegib
14.29Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
14.29Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
14.29Single5CGCHTL142425CGC-mGlu5-HTL14242
14.29Single5D6LS-Carazolol5D6L-β2-S-Carazolol
14.29Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
14.29Single5XPRBosentan5XPR-ETB-Bosentan
14.29Single6E67BI1671076E67-β2-BI167107-Gs(CT)
14.29Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
14.29Single6JODAngiotensin II6JOD-AT2-Angiotensin II
14.29Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
14.29Single6LUQHaloperidol6LUQ-D2-Haloperidol
14.29Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
14.29Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
14.29Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
14.29Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
14.29Single7C4SS1P7C4S-S1P3-S1P
14.29Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
14.29Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
14.29Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
14.29Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
14.29Single7SINNPS-21437SIN-CaS-NPS-2143
14.29Single7SINNPS-21437SIN-CaS-NPS-2143
14.29Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
14.29Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
14.29Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
14.29Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
14.29Single7W41PD1762527W41-BB2-PD176252
14.29Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
14.29Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
14.29Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
14.29Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
14.29Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
14.29Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
14.29Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
14.29Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
14.29Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
14.29Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
14.29Single8JXSPF-61428JXS-D1-PF-6142
14.29Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
14.29Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
14.29Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
14.29Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
14.29Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
14.29Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
14.29Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
14.29Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
14.29Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
14.29Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
14.29Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
14.29Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
14.29Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
14.29Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
14.29Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
14.29Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
14.29Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
14.29Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
14.29Consensusamine_offonOrthosteric Ligandamine_off amine_on
14.29Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
14.29Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
14.29Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
14.29Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
14.29Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
14.29Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
14.29Consensusblt_offOrthosteric Ligandblt1_off
14.29Consensusbombesin_offOrthosteric Ligandbb2_off
14.29Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
14.29Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
14.29Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
14.29Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
14.29Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
14.29Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
14.29Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
14.29Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
14.29Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
14.29Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
13.89Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
13.89Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
13.89Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.89Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.89Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
13.79Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
13.79Single5D5AS-Carazolol5D5A-β2-S-Carazolol
13.79Single5D5BS-Carazolol5D5B-β2-S-Carazolol
13.79Single5V54Methiothepin5V54-5-HT1B-Methiothepin
13.79Single5V56TC1145V56-SMO-TC114
13.79Single5V57TC1145V57-SMO-TC114
13.79Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
13.79Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
13.79Single6H7JIsoprenaline6H7J-β1-Isoprenaline
13.79Single6J21Aprepitant6J21-NK1-Aprepitant
13.79Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
13.79Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
13.79Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.79Single6OS1TRV0266OS1-AT1-TRV026
13.79Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
13.79Single7B6WCyclazosin7B6W-α1b-Cyclazosin
13.79Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
13.79Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
13.79Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
13.79Single7FEECP559407FEE-CB1-CP55940-ZCZ011
13.79Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
13.79Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
13.79Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
13.79Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
13.79Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
13.79Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
13.79Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
13.79Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
13.79Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
13.79Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
13.79Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
13.79Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
13.79Single8EA0Iperoxo8EA0-M3-Iperoxo
13.79Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
13.79Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
13.79Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
13.79Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
13.79Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
13.79Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
13.79Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.79Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
13.79Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
13.79Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
13.79Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
13.79Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.79Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
13.79Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
13.79Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
13.79Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.79Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
13.79Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
13.79Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
13.79Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
13.79Single9AS9RS130-1809AS9-5-HT2A-RS130-180
13.79Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
13.79Single9BJKNaloxone9BJK-μ-Naloxone-NAM
13.79Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
13.79Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
13.79Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
13.79Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Consensus5ht1_offOrthosteric Ligand5ht1b_off
13.79Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
13.79Consensusa2_onOrthosteric Liganda2b_on
13.79Consensusa2_on_gpOrthosteric Liganda2b_on_gp
13.79Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
13.79Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
13.79Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
13.79Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
13.79Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
13.79Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
13.79Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
13.79Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.79Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.79Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
13.79Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
13.79Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
13.79Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
13.79Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
13.79Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.79Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.79Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
13.79Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
13.79Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
13.79Consensusrelaxin_onOrthosteric Ligandrxfp4_on
13.79Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
13.64Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
13.64Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
13.64Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.64Single8HS2Fab0468HS2-GPR20-Fab046
13.64Single8PWNTheophylline8PWN-A2A-Theophylline
13.51Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
13.51Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
13.51Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.51Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.33Single3D4STimolol3D4S-β2-Timolol
13.33Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
13.33Single4AMIBucindolol4AMI-β1-Bucindolol
13.33Single4LDEBI1671074LDE-β2-BI167107
13.33Single4RWADIPP-NH24RWA-δ-DIPP-NH2
13.33Single5CXVTiotropium5CXV-M1-Tiotropium
13.33Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
13.33Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
13.33Single6A93Risperidone6A93-5-HT2A-Risperidone
13.33Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
13.33Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
13.33Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
13.33Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
13.33Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
13.33Single7DFPSpiperone7DFP-D2-Spiperone
13.33Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.33Single7K15MKD0467K15-BLT1-MKD046-Na
13.33Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
13.33Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.33Single7YITNalfurafine7YIT-κ-Nalfurafine
13.33Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
13.33Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
13.33Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
13.33Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
13.33Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
13.33Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
13.33Single8JWY2-1188JWY-A2A-2-118
13.33Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8XWACXCL18XWA-CXCR2-CXCL1
13.33Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
13.33Single9DGIZ85267113509DGI-CB1-Z8526711350
13.33Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
13.33Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
13.33Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
13.33Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
13.33Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.33Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.33Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
13.33Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
13.33Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.33Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
13.33Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
13.33Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
13.33Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
13.33Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
13.33Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
13.33Consensusorexin_onOrthosteric Ligandox2_on
13.33Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.33Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.16Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
13.16Single9KDFRES-701-39KDF-ETB-RES-701-3
13.04Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
13.04Single3RFMCaffeine3RFM-A2A-Caffeine
13.04Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
13.04Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
13.04Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
13.04Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
13.04Single9CHUNoradrenaline9CHU-β2-Noradrenaline
13.04Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
13.04Consensusp2y_offOrthosteric Ligandp2y1_off
12.90Single5CGDHTL142425CGD-mGlu5-HTL14242
12.90Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
12.90Single5X93K-87945X93-ETB-K-8794
12.90Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
12.90Single6H7LDobutamine6H7L-β1-Dobutamine
12.90Single6IBLArformoterol6IBL-β1-Arformoterol
12.90Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
12.90Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.90Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
12.90Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
12.90Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
12.90Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
12.90Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
12.90Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
12.90Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
12.90Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
12.90Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.90Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8XVJMacitentan8XVJ-ETA-Macitentan
12.90Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
12.90Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
12.90Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
12.90Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
12.90Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
12.90Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
12.90Consensusendothelin_offOrthosteric Ligandetb_off
12.90Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
12.90Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
12.90Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
12.50Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
12.50Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
12.50Single3OE6IT1t3OE6-CXCR4-IT1t
12.50Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
12.50Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
12.50Single5ZTYAM102575ZTY-CB2-AM10257
12.50Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
12.50Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
12.50Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
12.50Single6ME5Agomelatine6ME5-MT1-Agomelatine
12.50Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
12.50Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
12.50Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
12.50Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
12.50Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
12.50Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
12.50Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
12.50Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
12.50Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
12.50Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
12.50Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
12.50Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
12.50Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
12.50Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
12.50Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
12.50Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
12.50Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
12.50Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
12.50Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
12.50Single8XQJJN2418XQJ-Apelin-JN241
12.50Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
12.50Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
12.50Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
12.50Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
12.50Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
12.50Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
12.50Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
12.50Single9IPYJR14a9IPY-C3aB-JR14a
12.50Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.50Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
12.50Single9LRCHistamine9LRC-H4-Histamine
12.50Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
12.50Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
12.50Consensus5ht2_onOrthosteric Ligand5ht2b_on
12.50Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
12.50Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Consensusgi_sensoryOrthosteric Ligandgi_opsins
12.50Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.50Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.50Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.50Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.12Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
12.12Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
12.12Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
12.12Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
12.12Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
12.12Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
12.12Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
12.12Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
12.12Single8IEIA1LYA8IEI-GPR156-A1LYA
12.12Single8IEPA1LYA8IEP-GPR156-A1LYA
12.12Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
12.12Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
12.12Single8WKYPG-9348WKY-MC4-PG-934
12.12Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
12.12Single9M4TSilodosin9M4T-Alpha1A-Silodosin
12.12Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
12.12Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
12.12Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
12.12Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
12.12Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
12.00Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
12.00Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
12.00Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
12.00Single3PBLEticlopride3PBL-D3-Eticlopride
12.00Single4O9RCyclopamine4O9R-SMO-Cyclopamine
12.00Single5L7IVismodegib5L7I-SMO-Vismodegib
12.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
12.00Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
12.00Single6HLLCP999946HLL-NK1-CP99994
12.00Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
12.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
12.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
12.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.00Single7SRQLSD7SRQ-5-HT2B-LSD
12.00Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
12.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
12.00Single7UL2SR486927UL2-NTS1-SR48692-Na
12.00Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
12.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
12.00Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.00Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
12.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
12.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
12.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
12.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
12.00Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
12.00Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
12.00Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
12.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
12.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
12.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
12.00Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
12.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
12.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
12.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
12.00Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
12.00Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
12.00Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
12.00Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single9AS7Psilocin9AS7-5-HT2A-Psilocin
12.00Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
12.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
12.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
12.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
12.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
12.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
12.00Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
12.00Consensusneurotensin_offOrthosteric Ligandnts1_off
12.00Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
11.76Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
11.76Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
11.76Single8IEBA1LYA8IEB-GPR156-A1LYA
11.76Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
11.76Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
11.76Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
11.76Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
11.76Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
11.76Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
11.76Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
11.54Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
11.54Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
11.54Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
11.54Single3ODUIT1t3ODU-CXCR4-IT1t
11.54Single4QINSAG1.54QIN-SMO-SAG1.5
11.54Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
11.54Single5ZKQABT-4915ZKQ-PAF-ABT-491
11.54Single6AKXA4R6AKX-CCR5-A4R
11.54Single6AKYMaraviroc6AKY-CCR5-Maraviroc
11.54Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
11.54Single6DS0Ly2660976DS0-5-HT2B-Ly266097
11.54Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
11.54Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
11.54Single6ME2Ramelteon6ME2-MT1-Ramelteon
11.54Single6ME9Ramelteon6ME9-MT2-Ramelteon
11.54Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
11.54Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
11.54Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
11.54Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
11.54Single7F8YDevazepide7F8Y-CCKA-Devazepide
11.54Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
11.54Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
11.54Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
11.54Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.54Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.54Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
11.54Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
11.54Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
11.54Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
11.54Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
11.54Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
11.54Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
11.54Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
11.54Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
11.54Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
11.54Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
11.54Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
11.54Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
11.54Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
11.54Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
11.54Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
11.54Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
11.54Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
11.54Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
11.54Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
11.54Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
11.54Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
11.54Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
11.54Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
11.54Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
11.54Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
11.54Single9H2XA1IR19H2X-A2A-A1IR1-Na
11.54Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
11.54Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
11.54Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
11.54Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
11.54Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
11.54Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
11.54Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.54Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
11.54Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.54Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
11.54Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
11.54Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.54Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.54Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
11.54Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
11.54Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
11.43Single6W25SHU91196W25-MC4-SHU9119-Ca
11.43Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
11.43Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
11.43Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
11.43Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
11.43Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
11.43Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
11.43Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.43Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.43Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
11.43Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
11.11Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
11.11Single3REYXAC3REY-A2A-XAC
11.11Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
11.11Single4MBSMaraviroc4MBS-CCR5-Maraviroc
11.11Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
11.11Single6A94Zotepine6A94-5-HT2A-Zotepine
11.11Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
11.11Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
11.11Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
11.11Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
11.11Single6V9SGTPL114036V9S-OX1-GTPL11403
11.11Single6VI4JDTic6VI4-κ-JDTic
11.11Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
11.11Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
11.11Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
11.11Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
11.11Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
11.11Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
11.11Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
11.11Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
11.11Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
11.11Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
11.11Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
11.11Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
11.11Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
11.11Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
11.11Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
11.11Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
11.11Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
11.11Single7VV6C48/807VV6-MRGPRX2-C48/80
11.11Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
11.11Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
11.11Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
11.11Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
11.11Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
11.11Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
11.11Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
11.11Single8IHKAcifran8IHK-HCA3-Acifran
11.11Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
11.11Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
11.11Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
11.11Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
11.11Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
11.11Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
11.11Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8ZPMAMD0708ZPM-CXCR4-AMD070
11.11Single8ZPNAMD31008ZPN-CXCR4-AMD3100
11.11Single9ARXSerotonin9ARX-5-HT2A-Serotonin
11.11Single9AS3LSD9AS3-5-HT2A-LSD
11.11Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
11.11Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
11.11Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
11.11Consensusalpha1_onOrthosteric Ligandalpha1a_on
11.11Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
11.11Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
11.11Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
11.11Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
11.11Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
11.11Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
11.11Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
10.71Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
10.71Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
10.71Single4EJ4Naltrindole4EJ4-δ-Naltrindole
10.71Single4MQSIperoxo4MQS-M2-Iperoxo
10.71Single4QIMANTA XV4QIM-SMO-ANTA XV
10.71Single4U14Tiotropium4U14-M3-Tiotropium
10.71Single5DHHSB-6121115DHH-NOP-SB-612111
10.71Single5DSGTiotropium5DSG-M4-Tiotropium
10.71Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
10.71Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
10.71Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
10.71Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
10.71Single6DRXLisuride6DRX-5-HT2B-Lisuride
10.71Single6GPSMK08126GPS-CCR2-MK0812
10.71Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.71Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
10.71Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
10.71Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
10.71Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.71Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
10.71Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
10.71Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
10.71Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
10.71Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
10.71Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
10.71Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
10.71Single7UL4Alvimopan7UL4-μ-Alvimopan
10.71Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
10.71Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
10.71Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
10.71Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
10.71Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
10.71Single7YXAONO-54306087YXA-S1P5-ONO-5430608
10.71Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
10.71Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
10.71Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
10.71Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
10.71Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
10.71Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
10.71Single8K5DGSK2560738K5D-HCA2-GSK256073
10.71Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
10.71Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
10.71Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
10.71Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
10.71Single8X63Mepyramine8X63-H1-Mepyramine
10.71Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
10.71Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
10.71Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
10.71Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
10.71Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
10.71Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
10.71Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
10.71Single9IYAONO-97105319IYA-GPR55-ONO-9710531
10.71Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
10.71Single9JEAAtropine9JEA-M1-Atropine
10.71Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
10.71Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
10.71Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
10.71Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
10.71Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.71Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.71Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
10.71Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
10.71Consensusalpha2_onOrthosteric Ligandalpha2b_on
10.71Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
10.71Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.71Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.71Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
10.71Consensuscck_offOrthosteric Ligandccka_off
10.71Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
10.71Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
10.71Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
10.71Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
10.71Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
10.71Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
10.71Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
10.71Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
10.71Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
10.71Consensushistamine_offOrthosteric Ligandh1_off
10.71Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
10.71Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
10.71Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
10.34Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
10.34Single5WIUNemonapride5WIU-D4-Nemonapride
10.34Single5WIVNemonapride5WIV-D4-Nemonapride-Na
10.34Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
10.34Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
10.34Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
10.34Single6GPXMK08126GPX-CCR2-MK0812
10.34Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
10.34Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
10.34Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
10.34Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
10.34Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
10.34Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
10.34Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
10.34Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
10.34Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
10.34Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
10.34Single7WC6LSD7WC6-5-HT2A-LSD
10.34Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
10.34Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
10.34Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
10.34Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
10.34Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
10.34Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
10.34Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
10.34Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
10.34Single8ZMFA1L108ZMF-5-HT2C-A1L10
10.34Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
10.34Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
10.34Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
10.34Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
10.34Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
10.34Single9HAPTolvaptan9HAP-V2-Tolvaptan
10.34Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
10.34Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
10.34Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
10.34Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
10.34Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
10.34Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
10.34Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
10.34Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
10.34Consensusep_offOrthosteric Ligandep4_off
10.34Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
10.34Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
10.34Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
10.34Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
10.34Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
10.26Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
10.26Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
10.00Single4DJHJDTic4DJH-κ-JDTic
10.00Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
10.00Single4U15Tiotropium4U15-M3-Tiotropium
10.00Single5TZRMK86665TZR-FFA1-MK8666
10.00Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
10.00Single6J20Aprepitant6J20-NK1-Aprepitant
10.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
10.00Single6OL9Tiotropium6OL9-M5-Tiotropium
10.00Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
10.00Single6TQ7SB-3348676TQ7-OX1-SB-334867
10.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
10.00Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
10.00Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
10.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
10.00Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
10.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
10.00Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
10.00Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
10.00Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
10.00Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
10.00Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
10.00Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
10.00Single8XVLZibotentan8XVL-ETA-Zibotentan
10.00Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
10.00Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
10.00Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
10.00Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
10.00Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
10.00Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
10.00Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
10.00Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
10.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
10.00Consensustachykinin_offOrthosteric Ligandnk1_off
9.68Single4N4WSANT-14N4W-SMO-SANT-1
9.68Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
9.68Single4PY02MeSATP4PY0-P2Y12-2MeSATP
9.68Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
9.68Single5X33BIIL2605X33-BLT1-BIIL260
9.68Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
9.68Single6ZG4HTL00099366ZG4-M1-HTL0009936
9.68Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
9.68Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
9.68Single8JWZAB9288JWZ-A2A-AB928-Na
9.68Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
9.68Single8XQJJN2418XQJ-Apelin-JN241
9.68Single8XYIVUF106618XYI-CXCR3-VUF10661
9.68Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
9.68Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
9.68Consensusalpha1_offOrthosteric Ligandalpha1a_off
9.68Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
9.68Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
9.68Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
9.38Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
9.38Single6K1QIRL25006K1Q-ETB-IRL2500
9.38Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
9.38Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
9.38Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
9.38Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
9.38Single8ZPLHF511168ZPL-CXCR4-HF51116
9.38Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single5MZPCaffeine5MZP-A2A-Caffeine-Na
9.09Single6KNMJN241-96KNM-Apelin-JN241-9
9.09Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
9.09Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
9.09Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
9.09Single7SK9CCX6627SK9-ACKR3-CCX662
9.09Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
9.09Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8X5YAstemizole8X5Y-H1-Astemizole
9.09Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9JF4PD1683689JF4-BB1-PD168368
9.09Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
9.09Consensuskisspeptin_onOrthosteric Ligandkiss1_on
8.82Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
8.82Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.82Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
8.82Single8KIGSHU91198KIG-MC3-SHU9119-Ca
8.82Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
8.82Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.82Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
8.82Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.82Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.82Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
8.82Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
8.82Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
8.70Single7WC4Serotonin7WC4-5-HT2A-Serotonin
8.70Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
8.70Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
8.70Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.70Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.57Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
8.57Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.57Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
8.57Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
8.57Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
8.33Single3OE8IT1t3OE8-CXCR4-IT1t
8.33Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
8.33Single6TQ9SB-4081246TQ9-OX1-SB-408124
8.33Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
8.33Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
8.33Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
8.33Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
8.33Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
8.33Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
8.33Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
8.33Consensussensory_onOrthosteric Ligandopsins_on
8.11Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
8.00Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
8.00Single3UZAGTPL92363UZA-A2A-GTPL9236
8.00Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
8.00Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
8.00Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
8.00Single7WC5Psilocin7WC5-5-HT2A-Psilocin
8.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.00Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
8.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
8.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
8.00Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
8.00Single8JPSCCL78JPS-ACKR1-CCL7
8.00Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
8.00Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
8.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
8.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
8.00Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
8.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
8.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
8.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
7.89Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
7.89Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
7.89Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
7.69Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
7.69Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
7.69Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.69Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
7.69Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
7.69Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
7.69Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.69Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
7.69Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.69Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
7.69Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
7.69Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
7.69Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
7.69Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
7.69Consensusgq_nucleotideOrthosteric Ligandgq_p2y
7.69Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
7.69Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.41Single4S0VSuvorexant4S0V-OX2-Suvorexant
7.41Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
7.41Single5WS3EMPA5WS3-OX2-EMPA
7.41Single6B73MP11046B73-κ-MP1104
7.41Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
7.41Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
7.41Single6TODEMPA6TOD-OX1-EMPA-Na
7.41Single6TPJSuvorexant6TPJ-OX2-Suvorexant
7.41Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
7.41Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
7.41Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
7.41Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
7.41Single7XRRLemborexant7XRR-OX2-Lemborexant
7.41Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
7.41Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
7.41Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
7.41Single8Y0HVUF114188Y0H-CXCR3-VUF11418
7.41Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
7.41Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
7.41Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
7.41Consensusorexin_offOrthosteric Ligandox2_off ox1_off
7.41Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
7.41Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
7.14Single3RZECidoxepin3RZE-H1-Cidoxepin
7.14Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
7.14Single4ZJCSB-6740424ZJC-OX1-SB-674042
7.14Single6IQLL7458706IQL-D4-L745870
7.14Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
7.14Single6TP3Nemorexant6TP3-OX1-Nemorexant
7.14Single6TPGEMPA6TPG-OX2-EMPA
7.14Single6TPNHTL66416TPN-OX2-HTL6641
7.14Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
7.14Single6ZG9GSK10347026ZG9-M1-GSK1034702
7.14Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
7.14Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
7.14Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
7.14Single7VODCariprazine7VOD-5-HT2A-Cariprazine
7.14Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
7.14Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
7.14Single8K2WAMG4878K2W-CXCR3-AMG487
7.14Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
7.14Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
7.14Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
7.14Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
7.14Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
7.14Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
7.14Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
7.14Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
7.14Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
7.14Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
7.14Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
7.14Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
6.90Single5DHGC-355DHG-NOP-C-35
6.90Single6TOTLemborexant6TOT-OX1-Lemborexant
6.90Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
6.90Single7F83PF-051904577F83-Ghrelin-PF-05190457
6.90Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
6.90Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
6.90Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
6.90Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
6.90Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
6.90Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.90Single8X64Desloratadine8X64-H1-Desloratadine
6.90Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
6.90Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
6.90Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
6.90Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
6.90Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
6.90Consensusblt_onOrthosteric Ligandblt1_on
6.90Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
6.90Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
6.90Consensusleukotriene_onOrthosteric Ligandblt_on
6.90Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
6.90Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
6.67Single4NTJAZD12834NTJ-P2Y12-AZD1283
6.67Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
6.67Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
6.67Single5WQCEMPA5WQC-OX2-EMPA
6.67Single6HLPNetupitant6HLP-NK1-Netupitant
6.67Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
6.67Single6TP6Filorexant6TP6-OX1-Filorexant
6.67Single6Z4SSR486926Z4S-NTS1-SR48692
6.67Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.67Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
6.67Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
6.67Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
6.67Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
6.67Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
6.67Single9HC04YI9HC0-mGlu5-4YI
6.67Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
6.67Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
6.45Single6E59L-7607356E59-NK1-L-760735
6.45Single7P2L4YI7P2L-mGlu5-4YI
6.45Single7R0CAVP7R0C-V2-AVP-Arrestin2
6.45Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
6.45Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
6.45Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
6.45Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.45Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.45Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
6.45Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
6.45Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
6.25Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
6.25Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
6.25Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
6.25Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
6.25Single9BJKNAM9BJK-μ-Naloxone-NAM
6.25Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.25Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
6.25Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
6.06Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
6.06Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
6.06Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
6.06Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
6.06Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
5.88Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
5.88Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
5.71Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
5.71Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.00Single6D35Cholesterol6D35-SMO-Cholesterol
5.00Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.00Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.00Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
5.00Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
5.00Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
5.00Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
5.00Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
5.00Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
5.00Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
5.00Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
5.00Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.00Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.00Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
5.00Single7DTTCa7DTT-CaS-Ca-Ca
5.00Single7DTTCa7DTT-CaS-Ca-Ca
5.00Single7DTUTryptophan7DTU-CaS-Tryptophan
5.00Single7DTUTryptophan7DTU-CaS-Tryptophan
5.00Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.00Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.00Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.00Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.00Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.00Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.00Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.00Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.00Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
5.00Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.00Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.00Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.00Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.00Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.00Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.00Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
5.00Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
5.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.00Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.00Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.00Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.00Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.00Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.00Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.00Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.00Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.00Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
5.00Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.00Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.00Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.00Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.00Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.00Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.00Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
5.00Single7XW7K1-707XW7-TSH-K1-70
5.00Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.00Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.00Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.00Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.00Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.00Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.00Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.00Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.00Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.00Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.00Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.00Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.00Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
5.00Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.00Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.00Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.00Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.00Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.00Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.00Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.00Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.00Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.00Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.00Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.00Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
5.00Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.00Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.00Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.00Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.00Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.00Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.00Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.00Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.00Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.00Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.00Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.00Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.00Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.00Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.00Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.00Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.00Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
5.00Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
5.00Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
5.00Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
5.00Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
5.00Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
5.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.00Single8WVXNorrin8WVX-LGR4-Norrin
5.00Single8WVYNorrin8WVY-LGR4-Norrin
5.00Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.00Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.00Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.00Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.00Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.00Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.00Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
5.00Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.00Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.00Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.00Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.00Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.00Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.00Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.00Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.00Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.00Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.00Single9KHHNorrin9KHH-LGR4-Norrin
5.00Single9S37NB219S37-LGR4-NB21
5.00Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.76Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.76Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.76Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.76Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.76Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.76Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.76Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.76Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.76Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.55Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.55Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.55Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.55Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.35Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.35Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.35Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.35Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.35Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.17Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
4.17Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
4.17Single5L7DCholesterol5L7D-SMO-Cholesterol
4.17Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
4.17Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.17Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.00Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
4.00Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
3.85Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
3.70Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
3.70Single6TP4ACT-4622066TP4-OX1-ACT-462206
3.70Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
3.70Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
3.70Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
3.70Single8HNNSCH5467388HNN-CXCR3-SCH546738
3.70Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
3.70Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
3.57Single4XNVBPTU4XNV-P2Y1-BPTU
3.57Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
3.57Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
3.57Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.57Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
3.45Single6TPKRetosiban6TPK-OT-Retosiban
3.45Single6ZINSR486926ZIN-NTS1-SR48692
3.45Single8IYXYL-3658IYX-GPR34-YL-365
3.45Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.45Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
3.45Consensusvasop-oxy_offOrthosteric Ligandot_off
3.33Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
3.23Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.23Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.12Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.12Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
2.94Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
2.78Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.78Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.63Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.63Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.56Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.38Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

PDB Summary
PDB 8HA0
Class B1
SubFamily Peptide
Type Parathyroid Hormone
SubType PTH1
Species Homo Sapiens
Ligand PTH
Other Ligand(s) -
Protein Partners chim(NtGi1-Gs)/Beta1/Gamma2
PDB Resolution 2.62
Date 2022-12-21
D.O.I. doi.org/10.1038/s41401-022-01032-z
Net Summary
Imin 3.35
Number of Linked Nodes 975
Number of Links 1151
Number of Hubs 184
Number of Links mediated by Hubs 675
Number of Communities 35
Number of Nodes involved in Communities 236
Number of Links involved in Communities 323
Path Summary
Number Of Nodes in MetaPath 115
Number Of Links MetaPath 114
Number of Shortest Paths 1893370
Length Of Smallest Path 3
Average Path Length 43.1608
Length of Longest Path 90
Minimum Path Strength 1.35
Average Path Strength 6.9068
Maximum Path Strength 26.34
Minimum Path Correlation 0.7
Average Path Correlation 0.990651
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.78571
Average % Of Corr. Nodes 48.0516
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 43.5859
Maximum Path Hubs % 100
AnnotationTypeLinks
Gene OntologyMolecular Function
Gene OntologyBiological Process
Gene OntologyCellular Component
SCOP2Domain Identifier• Transducin (heterotrimeric G protein), gamma chain   • G protein-coupled receptor-like
SCOP2Family Identifier• Transducin (heterotrimeric G protein), gamma chain   • G protein-coupled receptor-like
Membrane Protein Annotations-• Orientations of Proteins in Membranes database (OPM)   • Protein Data Bank of Transmembrane Proteins (PDBTM)   • MemProtMD


Details about the values in these tables can be found in the corresponding documentation page .
PDBsumOpen PDBsum Page
ChainA
ProteinG Protein α Sub unit
UniProtP04896
Sequence
>8HA0_Chain_A
LSAEDKAAV ERSKMIEKQ LQKDKQVYR ATHRLLLLG ADNSGKSTI 
VKQMRIYHV TSGIFETKF QVDKVNFHM FDVGAQRDE RRKWIQCFN 
DVTAIIFVV DSSDYNRLQ EALNDFKSI WNNRWLRTI SVILFLNKQ 
DLLAEKVLA GKSKIEDYF PEFARYTTP EDATPEPGE DPRVTRAKY 
FIRDEFLRI STASGDGRH YCYPHFTCS VDTENARRI FNDCRDIIQ 
RMHLRQYEL L


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainB
ProteinG Protein β Sub unit
UniProtP54311
Sequence
>8HA0_Chain_B
ELDQLRQEA EQLKNQIRD ARKACADAT LSQITNNID PVGRIQMRT 
RRTLRGHLA KIYAMHWGT DSRLLVSAS QDGKLIIWD SYTTNKVHA 
IPLRSSWVM TCAYAPSGN YVACGGLDN ICSIYNLKT REGNVRVSR 
ELAGHTGYL SCCRFLDDN QIVTSSGDT TCALWDIET GQQTTTFTG 
HTGDVMSLS LAPDTRLFV SGACDASAK LWDVREGMC RQTFTGHES 
DINAICFFP NGNAFATGS DDATCRLFD LRADQELMT YSHDNIICG 
ITSVSFSKS GRLLLAGYD DFNCNVWDA LKADRAGVL AGHDNRVSC 
LGVTDDGMA VATGSWDSF LKIWN


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainG
ProteinG Protein γ Sub unit
UniProtP63212
Sequence
>8HA0_Chain_G
TASIAQARK LVEQLKMEA NIDRIKVSK AAADLMAYC EAHAKEDPL 
LTPVPASEN PFR


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainR
ProteinReceptor
UniProtQ03431
Sequence
>8HA0_Chain_R
VMTKEEQIF LLHRAQAQC EKGRPCLPE WDHILCWPL GAPGEVVAV 
PCPDYIYDF NHKGHAYRR CDRNGSWEL VPGHNRTWA NYSECVKET 
REREVFDRL AMIYTVGYS VSLASLTVA VLILAYFRR LHCTRNYIH 
MHLFLSFML RAVSIFVKD AVLYSAGYA GCRVAVTFF LYFLATNYY 
WILVEGLYL HSLIFMAFF SEKKYLWGF TVFGWGLPA VFVAVWVSV 
RATLANTGC WDLSSGNKK WIIQVPILA SIVLNFILF INIVRVLAT 
KLRETNTRQ QYRKLLKST LVLMPLFGV HYIVFMATP YTEVSGTLW 
QVQMHYEML FNSFQGFFV AIIYCFCNG EVQAEIKKS WSRWTLAL


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  



This network is also present in following consensuses:
IdComponents
pth1_on6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
7Y36-PTH1-Teriparatide-Gs/β1/γ2
7Y35-PTH1-Abaloparatide-Gs/β1/γ2
pth1_on_gp6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
7Y36-PTH1-Teriparatide-Gs/β1/γ2
7Y35-PTH1-Abaloparatide-Gs/β1/γ2

This receptor, from the same or other species and bound to the same or other ligands, is also present in the following networks:
Show PDB Class SubFamily Type SubType Species Orthosteric Ligand Other Ligand(s) Protein Partners Resolution Date DOI
8GW8B1PeptideParathyroid HormonePTH1Homo sapiens-PCO371Gs/β1/γ22.92023-06-14doi.org/10.1038/s41586-023-06169-3
8GW8 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiens-PCO3712.92023-06-14doi.org/10.1038/s41586-023-06169-3
8JR9B1PeptideParathyroid HormonePTH1Homo sapiens-PCO371chim(NtGi1-Gs)/β1/γ22.572023-08-02doi.org/10.1038/s41586-023-06467-w
8JR9 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiens-PCO3712.572023-08-02doi.org/10.1038/s41586-023-06467-w
7VVJB1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-Gs/β1/γ23.22022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVJ (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-3.22022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVKB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ23.32022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVK (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.32022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVLB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ22.82022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVL (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVMB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ23.22022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVM (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.22022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVNB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ23.82022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVN (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.82022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVOB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ24.12022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVO (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-4.12022-08-03doi.org/10.1016/j.molcel.2022.07.003
8FLQB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ22.552023-04-26doi.org/10.1016/j.str.2023.04.002
8FLQ (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.552023-04-26doi.org/10.1016/j.str.2023.04.002
8FLRB1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-Gs/β1/γ22.942023-04-26doi.org/10.1016/j.str.2023.04.002
8FLR (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-2.942023-04-26doi.org/10.1016/j.str.2023.04.002
8FLSB1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-Gs/β1/γ23.092023-04-26doi.org/10.1016/j.str.2023.04.002
8FLS (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-3.092023-04-26doi.org/10.1016/j.str.2023.04.002
8FLTB1PeptideParathyroid HormonePTH1Homo sapiensM-PTH(1-14)-Gs/β1/γ23.032023-04-26doi.org/10.1016/j.str.2023.04.002
8FLT (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensM-PTH(1-14)-3.032023-04-26doi.org/10.1016/j.str.2023.04.002
8FLUB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH-Gs/β1/γ22.762023-04-26doi.org/10.1016/j.str.2023.04.002
8FLU (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH-2.762023-04-26doi.org/10.1016/j.str.2023.04.002
8HA0B1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1-Gs)/β1/γ22.622022-12-21doi.org/10.1038/s41401-022-01032-z
8HA0 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.622022-12-21doi.org/10.1038/s41401-022-01032-z
8HAFB1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-chim(NtGi1-Gs)/β1/γ23.252022-12-21doi.org/10.1038/s41401-022-01032-z
8HAF (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-3.252022-12-21doi.org/10.1038/s41401-022-01032-z
8HAOB1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1-Gs)/β1/γ23.762022-12-21doi.org/10.1038/s41401-022-01032-z
8HAO (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.762022-12-21doi.org/10.1038/s41401-022-01032-z
6FJ3B1PeptideParathyroid HormonePTH1Homo sapiensPTH--2.52018-11-21doi.org/10.1038/s41594-018-0151-4
6NBFB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-Gs/β1/γ232019-04-17doi.org/10.1126/science.aav7942
6NBF (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-32019-04-17doi.org/10.1126/science.aav7942
6NBHB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-Gs/β1/γ23.52019-04-17doi.org/10.1126/science.aav7942
6NBH (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-3.52019-04-17doi.org/10.1126/science.aav7942
6NBIB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-Gs/β1/γ242019-04-17doi.org/10.1126/science.aav7942
6NBI (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-42019-04-17doi.org/10.1126/science.aav7942
9B5YB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH-chim(NtGi1-Gq)/β1/γ23.492025-03-19doi.org/10.1073/pnas.2426178122
9B5Y (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH-3.492025-03-19doi.org/10.1073/pnas.2426178122
7Y35B1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-Gs/β1/γ22.92023-07-05To be published
7Y35 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-2.92023-07-05To be published
7Y36B1PeptideParathyroid HormonePTH1Homo sapiensTeriparatide-Gs/β1/γ22.82023-07-05To be published
7Y36 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensTeriparatide-2.82023-07-05To be published
9JR2B1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1L-Gs-CtGq)/β1/γ22.82024-10-16To be published
9JR2 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82024-10-16To be published
9JR3B1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1L-Gs-CtGq)/β1/γ22.82024-10-16To be published
9JR3 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82024-10-16To be published




You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

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