Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 1.4492602
2G.HN.37 1.93207403
3G.hns1.03 1.58948504
4G.S1.02 5.28782475
5G.S1.06 4.41324178
6G.H1.01 3.716424179
7G.S2.03 4.96203419
8G.S2.05 3.95237513
9G.S2.06 6.53932409
10G.S2.08 7.61254475
11G.S3.01 4.34569474
12G.S3.03 7.22844577
13G.S3.04 8.09203416
14G.S3.06 7.59284515
15G.S3.07 3.524624179
16G.s3h2.03 4.31696519
17G.H2.02 3.68371418
18G.H2.06 4.92768719
19G.H2.07 4.71158719
20G.H2.09 5.58032418
21G.h2s4.01 5.54087619
22G.s4h3.04 5.63633698
23G.s4h3.05 6.17005499
24G.H3.01 5.04348409
25G.H3.09 5.04426759
26G.H3.13 3.09135555
27G.H3.14 5.45778408
28G.H3.17 6.848615
29G.H3.18 6.056694189
30G.S5.04 4.06247559
31G.S5.05 3.577876139
32G.S5.06 5.43679408
33G.S5.07 3.95223409
34G.HG.04 5.31912599
35G.hgh4.02 6.153845197
36G.hgh4.05 8.73609407
37G.H4.03 6.33901404
38G.H4.08 0.0979624403
39G.H4.10 9.416284196
40G.H4.15 4.98761458
41G.h4s6.01 3.29748404
42G.h4s6.02 5.03115458
43G.h4s6.12 3.77335504
44G.S6.02 5.944625207
45G.H5.03 4.848014138
46G.H5.08 5.95046478
47G.H5.13 3.679925208
48G.H5.17 2.42193505
49G.H5.20 3.41831409
50G.H5.26 4.213605
51b.1x11 2.42564408
52b.lh12x2 4.10548408
53b.h2x1 3.73205405
54b.lhb1x3 2.03669602
55b.lhb1x11 3.22965404
56b.b1x4 3.13691567
57b.b1x6 7.48447409
58b.l1x3 8.28463639
59b.b2x1 7.74731518
60b.b2x5 6.12067637
61b.b3x3 3.52726408
62b.l3x2 5.01876539
63b.b4x2 5.0586408
64b.b4x3 4.795744147
65b.b4x4 8.57853438
66b.b4x5 3.9507487
67b.b4x6 9.36139639
68b.l4x2 10.4443464
69b.b5x2 5.40208407
70b.b5x3 6.63122639
71b.b5x5 5.06575485
72b.b5x7 5.73897407
73b.l5x1 4.101095148
74b.l5x2 2.39636406
75b.l5x5 7.03052719
76b.b6x5 3.78702786
77b.l6x5 5.975184154
78b.b7x1 5.390335154
79b.l7x2 4.04384419
80b.l7x4 3.61031409
81b.b8x4 5.73898406
82b.l8x3 3.11769403
83b.b9x2 0.594815405
84b.b9x3 3.65134406
85b.l9x3 6.73597619
86b.l9x6 4.9366918
87b.b10x3 3.4063408
88b.b10x5 4.36873609
89b.b11x2 4.35511407
90b.b11x4 5.55735419
91b.l11x2 7.87414419
92b.b12x6 7.82031718
93b.b12x7 5.289224229
94b.b13x7 7.63138547
95b.l13x3 7.6339649
96b.l13x6 4.59397519
97b.l13x7 4.47334449
98b.b14x3 4.33789445
99b.b15x1 6.37215549
100b.b15x2 6.39063416
101b.b15x3 4.47881449
102b.l15x1 5.12234417
103b.l15x2 5.32813549
104b.b16x4 10.5523446
105b.b16x5 4.14019505
106b.b16x6 7.29967748
107b.b17x5 5.69078517
108b.b17x7 8.49322418
109b.l17x3 8.67695619
110b.l17x6 6.9433419
111b.b18x3 4.86819418
112b.b18x5 5.13718405
113b.l18x1 5.318398116
114b.l18x2 5.669354117
115b.l18x3 6.240364115
116b.b19x2 7.37702516
117b.b19x4 6.03165418
118b.l19x2 6.13883519
119b.b20x4 10.22518
120b.b20x6 7.86537516
121b.b20x7 3.67392409
122b.l20x2 4.81944509
123b.b21x1 6.09596617
124b.b21x2 2.84204406
125b.b21x4 3.194405
126b.b21x5 4.87068404
127b.b21x7 5.94554605
128b.l21x2 4.45878404
129b.b22x5 5.437885117
130b.l22x5 5.991066129
131b.b23x6 6.928546167
132b.l23x1 7.67247406
133b.b24x4 7.495944166
134b.b24x6 6.879674168
135b.l24x2 4.213614126
136b.l24x3 4.58201405
137b.l25x3 8.354295109
138b.b26x3 3.62998406
139b.l27x1 10.1295719
140b.l27x2 7.719094109
141b.b28x3 4.1601407
142b.b28x4 7.576514106
143b.b28x6 8.409125109
144g.h1x1 1.19499702
145g.l1x4 4.40192408
146g.h2x11 8.497954116
147g.ctx3 5.29366609
148g.ctx6 3.32802406
149g.ctx14 4.994469
150g.ctx15 6.13967469
151g.ctx16 4.38687868
152NT 4.603981023
1531x39 4.13001407
1541x60 1.84278606
1552x40 2.768844239
1562x42 4.10788508
1572x44 1.83388506
1582x46 4.08841429
1592x50 5.68909529
160E1x50 4.85944528
161E1x52 4.19955406
1623x22 2.62259424
1633x49 4.00887409
1643x50 5.68099529
1654x56 3.60435406
166E2 8.479312023
1675x47 5.5909408
1685x50 3.11114409
1695x58 4.91498629
170I3 1.3617405
1716x32 1.42578408
1726x44 4.655429
1736x48 6.15833528
1746x49 2.92566406
1756x51 4.23888527
1766x59 2.40992406
177E3 2.46013823
1787x32 0.98148523
1797x34 3.43778425
1807x42 3.63498627
1817x49 5.19276429
1827x52 2.65099429
1837x53 4.66573629
1848x48 2.31089406
1858x50 3.84795239
1868x54 1.8994407
187Lig 6.524332220
188H.HA.26 0.0328489400
189H.hahb.08 0.0237225400
190H.hbhc.04 0.0266809400
191H.hbhc.13 0.0270078400
192H.HC.11 0.0680201600
193H.hchd.01 0.0367394400
194H.hdhe.01 0.0432141500
195H.hdhe.03 0.0269533400
196H.hehf.04 0.0729282400
197H.hehf.06 0.038378500
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b3x2 b.b4x6 12.93434.99694NoYes359
2b.b2x3 b.b3x2 12.97762.89107NoNo365
3b.b26x2 b.b2x3 31.12525.27508NoNo076
4b.b26x1 b.b26x2 31.40712.90612NoNo097
5b.b26x1 b.l27x1 31.69265.52462NoYes099
6b.b2x1 b.l27x1 69.91447.43088YesYes189
7b.b2x1 b.l3x1 73.372915.0701YesNo189
8b.l3x1 b.l5x5 76.27816.44245NoYes199
9G.h2s4.01 b.l5x5 34.69449.67656YesYes199
10G.H2.07 G.h2s4.01 37.77333.90144YesYes199
11G.H2.04 G.H2.07 99.98834.20567NoYes099
12G.H2.04 G.H3.08 99.98214.26253NoNo099
13G.H3.08 G.S4.04 1005.37889NoNo099
14G.S4.04 G.S5.04 91.93192.98223NoYes599
15G.S5.04 G.S5.06 89.63763.71869YesYes098
16G.S5.06 G.s4h3.01 89.64167.35746YesNo087
17G.HG.04 G.s4h3.01 89.61098.53586YesNo097
18G.HG.04 G.s4h3.04 89.11866.07219YesYes998
19G.HG.07 G.s4h3.04 93.71635.03949NoYes998
20G.HG.07 G.s4h3.02 94.13742.92988NoNo099
21G.s4h3.02 G.s5hg.01 94.08344.67706NoNo099
22G.S5.07 G.s5hg.01 93.62712.15564YesNo099
23G.S5.07 G.s6h5.01 93.47657.3804YesNo099
24G.S5.05 G.s6h5.01 93.03264.68662YesNo1399
25b.l5x5 b.l7x2 43.88765.38522YesYes199
26G.H2.07 b.l7x2 34.81843.53585YesYes199
27b.b10x1 b.l9x6 21.70512.87705NoYes098
28b.b10x1 b.b11x5 21.5553.2907NoNo096
29b.b11x5 b.b14x3 15.46195.49681NoYes065
30b.b10x2 b.b14x3 12.63514.65259NoYes065
31b.b10x2 b.b10x4 12.50024.11452NoNo066
32b.b10x4 b.b2x4 11.979112.315NoNo066
33b.b2x4 b.b6x5 11.88832.85655NoYes066
34G.H2.06 b.l9x6 40.92893.57536YesYes198
35G.H2.06 b.l17x6 39.91697.94556YesYes199
36G.H3.06 G.hgh4.02 10.51645.03124NoYes067
37b.l25x6 b.l27x1 37.091919.45NoYes189
38G.S5.03 G.S5.05 91.48613.57227NoYes089
39G.H5.10 G.S5.03 91.40843.48319NoNo068
40G.H5.10 G.S6.02 91.36945.26151NoYes067
41G.S6.02 G.h4s6.12 46.297410.1487YesYes074
42G.H5.13 G.S6.02 44.83826.53689YesYes2087
43G.H5.17 G.h4s6.12 45.0883.12453YesYes054
44G.H5.13 G.H5.17 44.65534.57479YesYes085
45G.H5.17 G.H5.26 89.26573.1938YesYes055
463x50 G.H5.25 73.24926.9395YesNo097
47G.H5.20 G.H5.25 73.63843.73377YesNo097
48G.H5.20 G.H5.26 78.49853.56817YesYes095
49b.l17x5 b.l17x6 42.2883.79409NoYes169
50b.l17x5 b.l19x2 42.13983.33987NoYes169
51b.l17x3 b.l19x2 29.18014.39373YesYes199
52b.b19x4 b.l17x3 16.40488.18317YesYes189
53b.b19x4 b.b20x6 11.42897.59447YesYes186
54b.b17x7 b.b20x6 32.480410.696YesYes186
55b.b17x7 b.b21x1 30.2875.64422YesYes187
56b.1x19 b.b21x1 26.94437.3364NoYes067
57b.1x15 b.1x19 24.0993.11439NoNo076
58b.1x12 b.1x15 22.29892.88005NoNo067
59b.1x12 g.h1x11 21.69852.68728NoNo069
60b.1x11 g.h1x11 18.54954.26422YesNo089
61b.1x11 g.h1x12 12.52872.29884YesNo086
62g.h1x12 g.h1x9 11.32281.99412NoNo066
63g.h1x5 g.h1x9 10.11621.39534NoNo066
64b.b20x4 b.l17x3 12.014117.2911YesYes189
65b.b20x4 b.b20x6 22.84234.28835YesYes186
66b.b20x2 b.l19x2 12.39768.5973NoYes069
67b.b20x2 b.b20x4 12.01385.8999NoYes068
68b.l26x5 g.ctx4 13.1746.20724NoNo057
69g.ctx3 g.ctx4 12.54564.09969YesNo097
70g.ctx3 g.ctx6 10.23116.44221YesYes096
71b.b2x5 b.l26x1 11.399211.6434YesNo377
72b.l11x1 b.l9x6 29.6496.75878NoYes198
73b.b11x6 b.l11x1 32.20823.25986NoNo199
74b.b11x6 b.l9x3 30.984514.6267NoYes199
75b.b12x6 b.l9x3 29.21575.5945YesYes189
76b.b11x2 b.b12x6 28.0723.04788YesYes078
77b.l26x1 b.l26x3 10.82895.71145NoNo377
78b.l26x3 b.l26x5 10.58745.52364NoNo075
79b.b7x1 b.b8x3 10.6253.18813YesNo046
80b.b11x2 b.l12x1 21.05853.41964YesNo076
81b.l23x1 b.l25x6 36.974519.6776YesNo068
82b.l21x7 b.l23x1 25.45674.49467NoYes056
83b.l21x7 b.l23x2 24.8496.53571NoNo058
84b.b23x6 b.l23x2 23.62883.90719YesNo078
85b.b23x6 b.b24x6 19.94436.9039YesYes1678
86b.b21x7 b.b24x6 19.422510.5328YesYes058
87b.b21x7 b.b23x2 12.39015.51742YesNo056
88b.b22x5 b.b23x2 11.45388.95377YesNo076
89b.b22x1 b.l23x1 11.29263.2892NoYes086
90b.b22x1 b.b22x2 10.98783.00706NoNo088
91b.b22x2 b.b26x3 10.6945.40817NoYes086
921x39 7x42 10.20963.4372YesYes077
933x36 Lig 32.94.56177NoYes270
943x36 6x48 33.083.96141NoYes278
956x44 6x48 32.68056.42417YesYes298
965x54 6x44 37.633.67481NoYes289
975x54 5x58 37.53562.98991NoYes289
983x50 5x58 42.96746.23034YesYes299
992x53 7x46 10.73423.81463NoNo089
1002x50 7x46 14.79486.76035YesNo099
1012x46 3x43 11.86813.57237YesNo298
1023x43 7x53 22.96875.96388NoYes289
1033x50 7x53 24.73616.00345YesYes299
1043x43 7x49 10.89063.59262NoYes289
1056x32 G.H5.26 10.12022.4046YesYes085
106b.b9x2 b.l12x1 15.50372.25039YesNo056
107H.HA.14 b.b9x2 10.86440.0331319NoYes005
108H.HA.14 H.HE.05 10.35350.0620659NoNo000
109H.HA.11 H.HE.05 10.01280.0588022NoNo000
110G.H2.07 b.l9x6 65.07323.93206YesYes198
111b.b2x3 b.b2x5 17.874.19932NoYes367
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
1x397x423.43720YesYes7721
2x563x324.249150NoNo7721
2x577x425.073650NoYes7721
2x60Lig3.946242NoYes7010
3x22E25.973852YesYes4321
3x294x653.700992NoNo6612
3x29Lig3.153932NoYes6010
3x32Lig5.631452NoYes7010
3x334x574.095772NoNo6812
3x33Lig7.578522NoYes6010
3x366x483.961412NoYes7812
3x36Lig4.561772NoYes7010
4x605x396.835382NoNo8822
4x64E26.4012NoYes5321
E2E244.55892YesYes3311
E2E2x517.077052YesNo3411
E2Lig8.826072YesYes3010
E2x51Lig4.011092NoYes4010
E2E2x525.573652YesNo3511
E2x52Lig6.267912NoYes5010
5x39E25.667922NoYes8321
5x395x434.603242NoNo8721
6x516x523.0822YesNo7712
6x516x555.025472YesNo7711
6x517x373.350552YesNo7612
6x517x383.110692YesNo7611
6x51Lig6.62572YesYes7010
6x547x343.141950NoYes5521
6x547x374.357980NoNo5622
6x55Lig3.622152NoYes7010
6x58Lig3.091382NoYes4010
E3E33.861582YesYes3322
7x34Lig4.168212YesYes5010
7x387x422.842862NoYes6711
7x38Lig6.884392NoYes6010
5x43Lig3.702822NoYes7010
7x42Lig4.271952YesYes7010
3x25E23.303792NoYes9321
4x60E23.717152NoYes8321
5x36E28.268570NoYes5321
LigNT3.951462YesYes0301
NTNT10.94332YesYes3311
2x537x423.222730NoYes8721
2x603x283.393092NoNo7612
3x327x422.961472NoYes7711
3x375x434.492290NoNo7721
5x406x553.6512NoNo6721
6x587x343.496362NoYes4511
E2NT12.8592YesYes3311
5x40E22.910082NoYes6321
E1x49NT3.175172NoYes4321
7x34E22.944592YesYes5311
5x35E22.615652NoYes4321
5x38E22.500620NoYes4321
2x64Lig2.365490NoYes6010
6x58E32.131682NoYes4312
1x32NT1.864992NoYes4321
E1Lig1.682692NoYes0010
5x32E21.621572NoYes5321
6x62Lig1.379692NoYes0010
7x32NT1.036852YesYes3321
3x20E10.9885710NoNo0021
5x336x620.8979780NoNo2021
7x24NT0.5286810NoYes0321
E1x501NT0.5054550NoYes0321
3x19E10.290NoNo0021
E1x48NT0.2315712NoYes0321
1x25Lig0.0979670NoYes0010
4x69E20.08684760NoYes0321
5x28E20.07117742NoYes0321
5x27E20.04978022NoYes0321

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
85.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
82.61Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
75.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
72.00Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
72.00Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
72.00Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
68.18Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
66.67Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
62.50Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
60.87Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
60.71Single5GLHEndothelin-15GLH-ETB-Endothelin-1
60.00Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
58.33Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
58.33Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
58.33Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
57.69Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
57.69Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
57.69Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
57.69Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
57.14Single8E0GBU728E0G-μ-BU72
57.14Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
57.14Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
57.14Consensusbradykinin_onOrthosteric Ligandbk2_on
57.14Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
57.14Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
57.14Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
56.67Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
56.52Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
56.00Consensusangiotensin_onOrthosteric Ligandat1_on
56.00Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
56.00Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
55.56Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
55.56Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
55.56Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
55.56Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
55.17Single6IGKEndothelin-36IGK-ETB-Endothelin-3
55.00Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
55.00Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
55.00Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
55.00Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
55.00Consensushca_on_gpOrthosteric Ligandhca2_on_gp
54.55Single4RWADIPP-NH24RWA-δ-DIPP-NH2
54.55Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
54.55Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
54.55Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
54.17Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
54.17Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
54.17Consensuslpl_onOrthosteric Ligands1p_on lpa_on
54.17Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
54.17Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
53.85Single6JODAngiotensin II6JOD-AT2-Angiotensin II
53.85Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
53.85Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
53.85Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
53.85Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
53.57Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
53.57Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
52.38Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
52.38Single5C1MBU725C1M-μ-BU72
52.38Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
52.38Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
52.38Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
52.38Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
52.38Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
52.17Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
52.17Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
52.00Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
52.00Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
52.00Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
52.00Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
52.00Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
51.85Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
51.85Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
51.85Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
51.85Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
51.72Single6IGLIRL16206IGL-ETB-IRL1620
51.72Consensusendothelin_onOrthosteric Ligandetb_on eta_on
50.00Single4UG2CGS216804UG2-A2A-CGS21680
50.00Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
50.00Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
50.00Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
50.00Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
50.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
50.00Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
50.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
50.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
50.00Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
50.00Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
50.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
50.00Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
50.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
50.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
50.00Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
50.00Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
50.00Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
50.00Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
50.00Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
50.00Consensushca_onOrthosteric Ligandhca2_on
50.00Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
50.00Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
50.00Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
48.39Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
48.28Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
48.15Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
48.15Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
48.15Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
48.15Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
48.15Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
48.15Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
48.15Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
48.00Single4IARErgotamine4IAR-5-HT1B-Ergotamine
48.00Single4XT1Fractalkine4XT1-US28-Fractalkine
48.00Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
48.00Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
48.00Single8WDTphotoNECA8WDT-A2A-photoNECA
48.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
48.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
48.00Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
48.00Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
48.00Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
48.00Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
48.00Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
47.83Single6MXTSalmeterol6MXT-β2-Salmeterol
47.83Single7YITNalfurafine7YIT-κ-Nalfurafine
47.83Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
47.83Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
47.83Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
47.83Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
47.83Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
47.83Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
47.83Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
47.83Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
47.83Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
47.83Consensuslpa_offOrthosteric Ligandlpa1_off
47.83Consensuslpl_offOrthosteric Ligands1p_off lpa_off
47.83Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
47.83Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
47.83Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
47.83Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
47.83Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
47.62Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
47.62Single7UL4Alvimopan7UL4-μ-Alvimopan
47.62Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
47.62Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
47.62Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
47.62Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
47.62Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
47.62Single8K5DGSK2560738K5D-HCA2-GSK256073
47.62Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.62Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.62Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.62Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
47.62Consensusa3_onOrthosteric Liganda3a_on
47.62Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
47.62Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
47.62Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
47.62Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
47.62Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
47.62Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
46.88Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
46.67Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
46.67Single8IY6Endothelin-18IY6-ETB-Endothelin-1
46.67Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
46.43Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
46.43Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
46.43Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
46.43Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
46.43Single8ZRTET-18ZRT-ETB-ET-1
46.43Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
46.43Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
46.15Single3QAKUK-4320973QAK-A2A-UK-432097
46.15Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
46.15Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
46.15Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
46.15Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
46.15Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
46.15Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
46.15Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
45.83Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
45.83Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
45.83Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
45.83Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
45.83Single7EZCUKA7EZC-A2A-UKA
45.83Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
45.83Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
45.83Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
45.83Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
45.83Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
45.83Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
45.83Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
45.83Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
45.83Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
45.83Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
45.45Single7C61Ergotamine7C61-5-HT1B-Ergotamine
45.45Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
45.45Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
45.45Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
45.45Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
45.45Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
45.45Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
45.45Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
45.45Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
45.45Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
45.45Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
45.45Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
45.45Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
45.45Single8S4DCMF-0198S4D-Apelin-CMF-019
45.45Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
45.45Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
45.45Consensusa3_on_gpOrthosteric Liganda3a_on_gp
45.45Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
45.45Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
45.45Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
45.45Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
45.45Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
45.45Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
45.45Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
45.45Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
45.16Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
45.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
45.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
45.00Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
45.00Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
45.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
45.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
44.83Single4XT3Fractalkine4XT3-US28-Fractalkine
44.83Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
44.83Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
44.83Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
44.44Single5WF5UK-4320975WF5-A2A-UK-432097
44.44Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
44.44Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
44.44Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
44.44Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
44.44Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
44.44Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
44.44Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
44.44Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
44.44Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
44.44Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
44.00Single3NY9ICI118-5513NY9-β2-ICI118-551
44.00Single5WF6UK-4320975WF6-A2A-UK-432097
44.00Single5ZTYAM102575ZTY-CB2-AM10257
44.00Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
44.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
44.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
44.00Single7XN9L-054,5227XN9-SST2-L-054,522
44.00Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
44.00Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
44.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
44.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
44.00Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
44.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
44.00Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
44.00Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
44.00Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
44.00Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
44.00Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
44.00Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
43.75Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
43.75Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
43.48Single2YDVNECA2YDV-A2A-NECA
43.48Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
43.48Single4UHRCGS216804UHR-A2A-CGS21680
43.48Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
43.48Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
43.48Single5G53NECA5G53-A2A-NECA-Gs
43.48Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
43.48Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
43.48Single6H7JIsoprenaline6H7J-β1-Isoprenaline
43.48Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
43.48Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
43.48Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
43.48Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
43.48Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
43.48Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
43.48Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
43.48Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
43.48Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
43.48Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
43.48Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
43.48Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
43.48Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
43.48Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
43.48Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
43.48Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
43.48Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Consensusa2_onOrthosteric Liganda2b_on
43.48Consensusa2_on_gpOrthosteric Liganda2b_on_gp
43.48Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
43.48Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
43.48Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
43.48Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
43.48Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
43.48Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
43.48Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
43.48Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
43.33Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
43.33Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
43.33Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
43.33Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
43.33Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
43.33Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
43.33Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
42.86Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
42.86Single4ZJCSB-6740424ZJC-OX1-SB-674042
42.86Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
42.86Single6PS0S-Carazolol6PS0-β2-S-Carazolol
42.86Single6PS4ICI118-5516PS4-β2-ICI118-551
42.86Single6TPGEMPA6TPG-OX2-EMPA
42.86Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
42.86Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
42.86Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
42.86Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
42.86Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
42.86Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
42.86Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
42.86Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
42.86Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
42.86Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
42.86Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
42.86Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
42.86Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
42.86Single8K5CAcipimox8K5C-HCA2-Acipimox
42.86Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.86Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
42.86Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
42.86Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
42.86Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
42.86Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
42.86Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
42.86Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
42.86Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
42.31Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
42.31Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
42.31Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
42.31Single7F8XNN90567F8X-CCKA-NN9056
42.31Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
42.31Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
42.31Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
42.31Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
42.31Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
42.31Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
42.31Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
42.31Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.94Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
41.67Single4AMIBucindolol4AMI-β1-Bucindolol
41.67Single4LDEBI1671074LDE-β2-BI167107
41.67Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
41.67Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
41.67Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
41.67Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
41.67Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
41.67Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
41.67Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
41.67Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
41.67Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
41.67Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
41.67Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
41.67Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
41.67Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
41.67Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
41.67Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
41.67Single8JJ8Formoterol8JJ8-β2-Formoterol
41.67Single8JJLOlodaterol8JJL-β2-Olodaterol
41.67Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
41.67Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
41.67Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
41.67Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
41.67Single8XYIVUF106618XYI-CXCR3-VUF10661
41.67Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
41.67Consensusalpha1_offOrthosteric Ligandalpha1a_off
41.67Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
41.67Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
41.67Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
41.67Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
41.67Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
41.67Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
41.67Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
41.67Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
41.67Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
41.67Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
41.38Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
41.38Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
41.38Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
41.38Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
41.38Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
41.38Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
41.38Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
41.38Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
40.91Single2Y04Salbutamol2Y04-β1-Salbutamol
40.91Single3NY8ICI118-5513NY8-β2-ICI118-551
40.91Single4EJ4Naltrindole4EJ4-δ-Naltrindole
40.91Single4GBRS-Carazolol4GBR-β2-S-Carazolol
40.91Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
40.91Single6PS1Timolol6PS1-β2-Timolol
40.91Single6TOTLemborexant6TOT-OX1-Lemborexant
40.91Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
40.91Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
40.91Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
40.91Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
40.91Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
40.91Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
40.91Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
40.91Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
40.91Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
40.91Single7V3ZCP559407V3Z-CB1-CP55940
40.91Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
40.91Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
40.91Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
40.91Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
40.91Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
40.91Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
40.91Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
40.91Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
40.91Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
40.91Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
40.91Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
40.91Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
40.91Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
40.91Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
40.91Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
40.91Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.91Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
40.91Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
40.91Single9CHXS-Carazolol9CHX-β2-S-Carazolol
40.91Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
40.91Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
40.91Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
40.91Consensusdopamine_offOrthosteric Ligandd2_off d3_off
40.91Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
40.91Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
40.74Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
40.74Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
40.74Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
40.74Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
40.74Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
40.74Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
40.74Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
40.74Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
40.74Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
40.74Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
40.74Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
40.74Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
40.62Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
40.62Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
40.62Consensusbombesin_onOrthosteric Ligandbb2_on
40.62Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
40.62Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
40.62Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
40.62Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
40.62Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
40.62Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
40.00Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
40.00Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
40.00Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
40.00Single5X93K-87945X93-ETB-K-8794
40.00Single6IBLArformoterol6IBL-β1-Arformoterol
40.00Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
40.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
40.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
40.00Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
40.00Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
40.00Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
40.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
40.00Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
40.00Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
40.00Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
40.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
40.00Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
40.00Single8K5BNiacin8K5B-HCA2-Niacin
40.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
40.00Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
40.00Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
40.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
40.00Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
40.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
40.00Consensuscck_onOrthosteric Ligandccka_on cckb_on
40.00Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
40.00Consensuschemerin_onOrthosteric Ligandcml1_on
40.00Consensusendothelin_offOrthosteric Ligandetb_off
40.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
40.00Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
40.00Consensusprostanoid_offOrthosteric Ligandep_off dp_off
39.39Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
39.39Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
39.29Single3OE0CVX153OE0-CXCR4-CVX15
39.29Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
39.29Single6PT2KGCHM076PT2-δ-KGCHM07
39.29Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
39.29Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
39.29Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
39.29Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
39.29Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
39.29Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
39.29Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
39.13Single2RH1S-Carazolol2RH1-β2-S-Carazolol
39.13Single2Y03Isoprenaline2Y03-β1-Isoprenaline
39.13Single2YCWS-Carazolol2YCW-β1-S-Carazolol
39.13Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
39.13Single5D6LS-Carazolol5D6L-β2-S-Carazolol
39.13Single5JQHS-Carazolol5JQH-β2-S-Carazolol
39.13Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
39.13Single5WQCEMPA5WQC-OX2-EMPA
39.13Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
39.13Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
39.13Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
39.13Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
39.13Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
39.13Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
39.13Single6TP6Filorexant6TP6-OX1-Filorexant
39.13Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
39.13Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
39.13Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
39.13Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
39.13Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
39.13Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
39.13Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
39.13Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
39.13Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
39.13Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
39.13Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
39.13Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
39.13Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
39.13Single8JXSPF-61428JXS-D1-PF-6142
39.13Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
39.13Single8TF5Oleic acid8TF5-GPR6-Oleic acid
39.13Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
39.13Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
39.13Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
39.13Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
39.13Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
39.13Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
39.13Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
39.13Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
39.13Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
39.13Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
39.13Consensusamine_offonOrthosteric Ligandamine_off amine_on
39.13Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
39.13Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
39.13Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
39.13Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
39.13Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
39.13Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
39.13Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
39.13Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
39.13Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
39.13Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
39.13Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
39.13Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
39.13Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
39.13Consensustrace-amine_onOrthosteric Ligandta1_on
38.71Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
38.71Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
38.71Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
38.71Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
38.46Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
38.46Single6PT3DPI-2876PT3-δ-DPI-287
38.46Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
38.46Single7SK9CCX6627SK9-ACKR3-CCX662
38.46Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
38.46Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
38.46Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
38.46Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
38.46Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
38.46Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
38.46Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
38.46Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
38.46Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
38.46Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
38.46Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
38.10Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
38.10Single5WS3EMPA5WS3-OX2-EMPA
38.10Single6AKXA4R6AKX-CCR5-A4R
38.10Single6B73MP11046B73-κ-MP1104
38.10Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
38.10Single6TODEMPA6TOD-OX1-EMPA-Na
38.10Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
38.10Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
38.10Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
38.10Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
38.10Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
38.10Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
38.10Single8GNGIstradefylline8GNG-A2A-Istradefylline
38.10Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
38.10Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
38.10Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
38.10Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
38.10Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.10Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
38.10Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
38.10Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
38.10Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
38.10Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
38.10Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
38.10Consensusalpha2_offOrthosteric Ligandalpha2c_off
38.10Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
38.10Consensusorexin_offOrthosteric Ligandox2_off ox1_off
38.10Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
38.10Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
38.10Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
38.10Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
37.93Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
37.93Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
37.93Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
37.93Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
37.93Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
37.93Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
37.93Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
37.93Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
37.93Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
37.93Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
37.93Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
37.93Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
37.93Consensusvasop-oxy_onOrthosteric Ligandv2_on
37.93Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
37.84Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
37.50Single3P0GBI1671073P0G-β2-BI167107
37.50Single4DJHJDTic4DJH-κ-JDTic
37.50Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
37.50Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
37.50Single5D5AS-Carazolol5D5A-β2-S-Carazolol
37.50Single5D5BS-Carazolol5D5B-β2-S-Carazolol
37.50Single5XR8AM8415XR8-CB1-AM841
37.50Single5XRAAM115425XRA-CB1-AM11542
37.50Single6J21Aprepitant6J21-NK1-Aprepitant
37.50Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
37.50Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
37.50Single6TQ7SB-3348676TQ7-OX1-SB-334867
37.50Single6WGTLSD6WGT-5-HT2A-LSD
37.50Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
37.50Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
37.50Single7FEECP559407FEE-CB1-CP55940-ZCZ011
37.50Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
37.50Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
37.50Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
37.50Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
37.50Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
37.50Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
37.50Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
37.50Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
37.50Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
37.50Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
37.50Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
37.50Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
37.50Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
37.50Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
37.50Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
37.50Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
37.50Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
37.50Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
37.50Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
37.50Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
37.50Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
37.50Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
37.50Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
37.50Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
37.50Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
37.50Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
37.50Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
37.50Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
37.50Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
37.50Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
37.50Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
37.50Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
37.50Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
37.50Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
37.50Consensuslpa_onOrthosteric Ligandlpa1_on
37.50Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
37.50Consensusrelaxin_onOrthosteric Ligandrxfp4_on
37.50Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
37.50Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.50Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
37.04Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
37.04Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
37.04Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
37.04Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
37.04Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
37.04Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
37.04Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
37.04Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
37.04Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
37.04Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
37.04Single8WKYPG-9348WKY-MC4-PG-934
37.04Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.04Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
37.04Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
37.04Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
37.04Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
37.04Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
37.04Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
36.67Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
36.67Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
36.67Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.67Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
36.67Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
36.67Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
36.67Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
36.67Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
36.67Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
36.36Single2YDOAdenosine2YDO-A2A-Adenosine
36.36Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
36.36Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
36.36Single4MBSMaraviroc4MBS-CCR5-Maraviroc
36.36Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
36.36Single6KUXRS-799486KUX-α2a-RS-79948
36.36Single6PS5S-Propranolol6PS5-β2-S-Propranolol
36.36Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
36.36Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
36.36Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
36.36Single6V9SGTPL114036V9S-OX1-GTPL11403
36.36Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
36.36Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
36.36Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
36.36Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
36.36Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
36.36Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
36.36Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
36.36Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.36Single7UL3Famotidine7UL3-H2-Famotidine
36.36Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
36.36Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
36.36Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
36.36Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
36.36Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
36.36Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
36.36Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
36.36Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
36.36Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
36.36Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
36.36Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
36.36Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
36.36Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
36.36Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
36.36Single8IHKAcifran8IHK-HCA3-Acifran
36.36Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
36.36Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
36.36Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
36.36Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.36Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
36.36Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
36.36Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
36.36Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
36.36Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
36.36Consensusalpha1_onOrthosteric Ligandalpha1a_on
36.36Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
36.36Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
36.36Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
36.36Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
36.36Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
36.36Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
36.00Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
36.00Single3D4STimolol3D4S-β2-Timolol
36.00Single4XEENeurotensin4XEE-NTS1-Neurotensin
36.00Single4XESNeurotensin4XES-NTS1-Neurotensin
36.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
36.00Single6A93Risperidone6A93-5-HT2A-Risperidone
36.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
36.00Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
36.00Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
36.00Single6KQICP559406KQI-CB1-CP55940-Org27569
36.00Single6OS2TRV0266OS2-AT1-TRV026
36.00Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
36.00Single7DFPSpiperone7DFP-D2-Spiperone
36.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
36.00Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
36.00Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
36.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
36.00Single7K15MKD0467K15-BLT1-MKD046-Na
36.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
36.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
36.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
36.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
36.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
36.00Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
36.00Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
36.00Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
36.00Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
36.00Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
36.00Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
36.00Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
36.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
36.00Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
36.00Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
36.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
36.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
36.00Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
36.00Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
36.00Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
36.00Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
36.00Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
36.00Consensusorexin_onOrthosteric Ligandox2_on
36.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
35.71Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
35.71Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
35.71Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
35.71Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
35.71Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
35.48Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
35.48Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
35.48Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
35.48Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
35.29Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
35.14Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
35.14Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
35.00Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
35.00Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
35.00Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
34.78Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
34.78Single2Y02Carmoterol2Y02-β1-Carmoterol
34.78Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
34.78Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
34.78Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
34.78Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
34.78Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
34.78Single4QKX35V4QKX-β2-35V
34.78Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
34.78Single4YAYZD-71554YAY-AT1-ZD-7155
34.78Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
34.78Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
34.78Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
34.78Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
34.78Single6H7MSalbutamol6H7M-β1-Salbutamol
34.78Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
34.78Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
34.78Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
34.78Single7BU7BI1671077BU7-β1-BI167107
34.78Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
34.78Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
34.78Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
34.78Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
34.78Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
34.78Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
34.78Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
34.78Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
34.78Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
34.78Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
34.78Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
34.78Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
34.78Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
34.78Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
34.78Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
34.78Single8JJOAlprenolol8JJO-β2-Alprenolol
34.78Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
34.78Single8JXRLSD8JXR-D1-LSD
34.78Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
34.78Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
34.78Single8T1WCVN4248T1W-GPR6-CVN424
34.78Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
34.78Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
34.78Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
34.78Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
34.78Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
34.78Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
34.78Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
34.78Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
34.78Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
34.78Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
34.78Consensus5ht5_onOrthosteric Ligand5ht5a_on
34.78Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
34.78Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
34.78Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
34.78Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
34.62Single4BUONeurotensin4BUO-NTS1-Neurotensin
34.62Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
34.62Single6H7LDobutamine6H7L-β1-Dobutamine
34.62Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
34.62Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
34.62Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
34.62Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
34.62Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
34.62Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
34.62Single7UM4AS26747237UM4-5-HT5A-AS2674723
34.62Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
34.62Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
34.62Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
34.62Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
34.62Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
34.62Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
34.62Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
34.62Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
34.62Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
34.62Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
34.62Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
34.62Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
34.62Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
34.62Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
34.62Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
34.48Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
34.48Single6W25SHU91196W25-MC4-SHU9119-Ca
34.48Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
34.48Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
33.33Single3OE9IT1t3OE9-CXCR4-IT1t
33.33Single3PBLEticlopride3PBL-D3-Eticlopride
33.33Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
33.33Single5N2RPSB-365N2R-A2A-PSB-36-Na
33.33Single5N2SPSB365N2S-A1-PSB36
33.33Single5TVNLSD5TVN-5-HT2B-LSD
33.33Single5WIUNemonapride5WIU-D4-Nemonapride
33.33Single5WIVNemonapride5WIV-D4-Nemonapride-Na
33.33Single6D26Fevipiprant6D26-DP2-Fevipiprant
33.33Single6E67BI1671076E67-β2-BI167107-Gs (fused)
33.33Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
33.33Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
33.33Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
33.33Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
33.33Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
33.33Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
33.33Single6PS6Timolol6PS6-β2-Timolol
33.33Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
33.33Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
33.33Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
33.33Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
33.33Single7C4SS1P7C4S-S1P3-S1P
33.33Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
33.33Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
33.33Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
33.33Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
33.33Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
33.33Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
33.33Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
33.33Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
33.33Single7WC6LSD7WC6-5-HT2A-LSD
33.33Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
33.33Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
33.33Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
33.33Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
33.33Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
33.33Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
33.33Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
33.33Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
33.33Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
33.33Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
33.33Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
33.33Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
33.33Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
33.33Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
33.33Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single8X5YAstemizole8X5Y-H1-Astemizole
33.33Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
33.33Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
33.33Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
33.33Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
33.33Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
33.33Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
33.33Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
33.33Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
33.33Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
33.33Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
33.33Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
33.33Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
33.33Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
33.33Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
33.33Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
33.33Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
33.33Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
33.33Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
33.33Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
33.33Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
33.33Consensusdp_offOrthosteric Liganddp2_off
33.33Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
33.33Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
32.35Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
32.35Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
32.26Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
32.26Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
32.26Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
32.26Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
32.26Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
32.26Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
32.26Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
32.14Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
32.14Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
32.14Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
32.00Single4BV0Neurotensin4BV0-NTS1-Neurotensin
32.00Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
32.00Single6OS1TRV0266OS1-AT1-TRV026
32.00Single7B6WCyclazosin7B6W-α1b-Cyclazosin
32.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
32.00Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
32.00Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
32.00Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
32.00Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
32.00Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
32.00Single7TUYGSK682753A7TUY-GPR183-GSK682753A
32.00Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.00Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
32.00Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
32.00Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
32.00Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
32.00Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
32.00Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
32.00Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
32.00Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
32.00Single8XVLZibotentan8XVL-ETA-Zibotentan
32.00Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
32.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
32.00Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
32.00Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
32.00Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
32.00Consensusneurotensin_onOrthosteric Ligandnts1_on
32.00Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
32.00Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
31.82Single3PWHZM-2413853PWH-A2A-ZM-241385
31.82Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
31.82Single4S0VSuvorexant4S0V-OX2-Suvorexant
31.82Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
31.82Single6AKYMaraviroc6AKY-CCR5-Maraviroc
31.82Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
31.82Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
31.82Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
31.82Single6TPJSuvorexant6TPJ-OX2-Suvorexant
31.82Single7BR3Elagolix7BR3-GnRH1-Elagolix
31.82Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
31.82Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
31.82Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
31.82Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
31.82Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
31.82Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
31.82Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
31.82Single7XRRLemborexant7XRR-OX2-Lemborexant
31.82Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
31.82Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
31.82Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
31.82Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
31.82Single8IWESpermidine8IWE-TA9-Spermidine
31.82Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
31.82Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
31.82Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
31.82Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
31.82Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
31.82Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.82Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.82Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
31.82Single8Y0HVUF114188Y0H-CXCR3-VUF11418
31.82Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
31.82Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
31.82Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
31.82Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
31.82Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
31.82Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
31.82Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
31.82Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
31.43Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
31.25Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
31.25Single6FJ3PTH6FJ3-PTH1-PTH
31.25Single7SK3CXCL127SK3-ACKR3-CXCL12
31.25Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
31.25Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
31.25Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
31.25Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
31.25Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
31.03Single6HLOAprepitant6HLO-NK1-Aprepitant
31.03Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
31.03Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
31.03Single7SK5CXCL127SK5-ACKR3-CXCL12
31.03Single7XNACYN1548067XNA-SST2-CYN154806
31.03Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
31.03Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
31.03Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
31.03Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
30.77Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
30.77Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
30.77Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
30.77Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
30.77Single6YVRNTS8-136YVR-NTS1-NTS8-13
30.77Single6ZG4HTL00099366ZG4-M1-HTL0009936
30.77Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
30.77Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
30.77Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.77Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
30.77Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
30.77Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
30.77Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
30.77Single8JWY2-1188JWY-A2A-2-118
30.77Single8JWZAB9288JWZ-A2A-AB928-Na
30.77Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
30.77Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
30.77Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
30.77Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
30.77Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
30.77Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
30.77Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
30.56Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
30.43Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
30.43Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
30.43Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
30.43Single6IQLL7458706IQL-D4-L745870
30.43Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
30.43Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
30.43Single6MH8ZM-2413856MH8-A2A-ZM-241385
30.43Single6TP3Nemorexant6TP3-OX1-Nemorexant
30.43Single6TPNHTL66416TPN-OX2-HTL6641
30.43Single6VI4JDTic6VI4-κ-JDTic
30.43Single7AROLUF58337ARO-A2A-LUF5833-Na
30.43Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
30.43Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
30.43Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
30.43Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
30.43Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
30.43Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
30.43Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
30.43Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
30.43Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
30.43Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
30.43Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
30.43Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
30.43Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
30.43Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
30.43Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
30.43Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.43Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
30.43Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
30.43Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
30.43Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
30.43Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
30.43Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
30.43Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
30.43Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
30.43Single9BJKNaloxone9BJK-μ-Naloxone-NAM
30.43Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
30.43Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
30.43Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
30.43Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
30.43Consensusgrh_offOrthosteric Ligandgnrh1_off
30.43Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
30.30Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
30.30Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
30.30Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
30.30Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
30.30Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
30.30Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
30.23Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
30.00Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
30.00Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
30.00Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
30.00Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
30.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
30.00Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
30.00Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
30.00Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
30.00Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
30.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
30.00Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
30.00Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
29.73Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.63Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
29.63Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
29.63Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
29.63Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.63Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
29.63Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
29.63Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
29.63Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.63Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
29.63Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
29.63Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
29.63Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.63Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
29.63Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
29.63Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.63Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.41Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
29.41Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
29.41Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
29.41Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
29.17Single2Y01Dobutamine2Y01-β1-Dobutamine
29.17Single4QIMANTA XV4QIM-SMO-ANTA XV
29.17Single5DHGC-355DHG-NOP-C-35
29.17Single5DHHSB-6121115DHH-NOP-SB-612111
29.17Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
29.17Single5TGZAM65385TGZ-CB1-AM6538
29.17Single5UENDU1725UEN-A1-DU172
29.17Single5UIGCmpd-15UIG-A2A-Cmpd-1
29.17Single6D27CAY104716D27-DP2-CAY10471
29.17Single6DRXLisuride6DRX-5-HT2B-Lisuride
29.17Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
29.17Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
29.17Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
29.17Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
29.17Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
29.17Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
29.17Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
29.17Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
29.17Single7WC7Lisuride7WC7-5-HT2A-Lisuride
29.17Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
29.17Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
29.17Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
29.17Single8CU6LJ-45178CU6-A2A-LJ-4517
29.17Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
29.17Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
29.17Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
29.17Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
29.17Single8RLNLUF58348RLN-A2A-LUF5834
29.17Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
29.17Single8X64Desloratadine8X64-H1-Desloratadine
29.17Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
29.17Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
29.17Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
29.17Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
29.17Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
29.17Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
29.17Consensusalpha2_onOrthosteric Ligandalpha2b_on
29.17Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
29.17Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
29.17Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
29.17Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
29.17Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
29.17Consensusblt_onOrthosteric Ligandblt1_on
29.17Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
29.17Consensuscck_offOrthosteric Ligandccka_off
29.17Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
29.17Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
29.17Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
29.17Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
29.17Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
29.17Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
29.17Consensusleukotriene_onOrthosteric Ligandblt_on
29.17Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
29.03Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
29.03Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
29.03Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
29.03Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
29.03Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
28.57Single3OE6IT1t3OE6-CXCR4-IT1t
28.57Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
28.57Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
28.57Single6KNMJN241-96KNM-Apelin-JN241-9
28.57Single6ME5Agomelatine6ME5-MT1-Agomelatine
28.57Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
28.57Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
28.57Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
28.57Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
28.57Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
28.57Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
28.57Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
28.57Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
28.57Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
28.57Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
28.57Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
28.57Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8XQJJN2418XQJ-Apelin-JN241
28.57Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
28.57Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
28.57Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
28.57Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
28.57Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
28.57Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
28.57Consensus5ht2_onOrthosteric Ligand5ht2b_on
28.57Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
28.57Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
28.57Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
28.12Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
28.12Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
28.12Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
28.00Single2Y00Dobutamine2Y00-β1-Dobutamine
28.00Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
28.00Single5XPRBosentan5XPR-ETB-Bosentan
28.00Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
28.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
28.00Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
28.00Single7SINNPS-21437SIN-CaS-NPS-2143
28.00Single7SINNPS-21437SIN-CaS-NPS-2143
28.00Single7W41PD1762527W41-BB2-PD176252
28.00Single8GNEKW-63568GNE-A2A-KW-6356-Na
28.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
28.00Single8QOTNanobody-E8QOT-μ-Nanobody-E
28.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
28.00Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
28.00Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
28.00Single8ZMFA1L108ZMF-5-HT2C-A1L10
28.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
28.00Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
28.00Consensusadenosine_offOrthosteric Liganda1_off a2_off
28.00Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
28.00Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
28.00Consensusblt_offOrthosteric Ligandblt1_off
28.00Consensusbombesin_offOrthosteric Ligandbb2_off
28.00Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
28.00Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
28.00Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
27.78Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
27.59Single7QA8Peptide7QA8-STE2-Peptide
27.59Single7QA8Peptide7QA8-STE2-Peptide
27.59Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
27.59Single8IEBA1LYA8IEB-GPR156-A1LYA
27.59Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
27.59Single8XWNCXCL88XWN-CXCR2-CXCL8
27.59Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
27.59Consensussomatostatin_offOrthosteric Ligandsst2_off
27.27Single6HLLCP999946HLL-NK1-CP99994
27.27Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
27.27Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
27.27Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
27.27Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
27.27Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
27.27Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
27.27Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
27.27Single7SRQLSD7SRQ-5-HT2B-LSD
27.27Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
27.27Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
27.27Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
27.27Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
27.27Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
27.27Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
27.27Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
27.27Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
27.27Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
27.27Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
27.27Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
27.27Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
27.27Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
27.27Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
27.27Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
27.27Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
27.27Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
27.27Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
27.27Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
27.27Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
27.27Consensusgq_nucleotideOrthosteric Ligandgq_p2y
27.27Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
27.03Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
26.92Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
26.92Single4U15Tiotropium4U15-M3-Tiotropium
26.92Single5V54Methiothepin5V54-5-HT1B-Methiothepin
26.92Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
26.92Single6J20Aprepitant6J20-NK1-Aprepitant
26.92Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
26.92Single6OL9Tiotropium6OL9-M5-Tiotropium
26.92Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
26.92Single7PX4PSB-21137PX4-A2A-PSB-2113
26.92Single7R0CAVP7R0C-V2-AVP-Arrestin2
26.92Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
26.92Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
26.92Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
26.92Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
26.92Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
26.92Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
26.92Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
26.92Consensus5ht1_offOrthosteric Ligand5ht1b_off
26.92Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
26.92Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
26.92Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
26.92Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
26.92Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
26.92Consensustachykinin_offOrthosteric Ligandnk1_off
26.67Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
26.67Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
26.67Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
26.67Single8IEBA1LYA8IEB-GPR156-A1LYA
26.67Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
26.67Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
26.47Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
26.47Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
26.47Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
26.47Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
26.32Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
26.32Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
26.09Single3ODUIT1t3ODU-CXCR4-IT1t
26.09Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
26.09Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
26.09Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
26.09Single5ZKQABT-4915ZKQ-PAF-ABT-491
26.09Single6DS0Ly2660976DS0-5-HT2B-Ly266097
26.09Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
26.09Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
26.09Single6ME2Ramelteon6ME2-MT1-Ramelteon
26.09Single6ME9Ramelteon6ME9-MT2-Ramelteon
26.09Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
26.09Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
26.09Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
26.09Single7F8ULintitript7F8U-CCKA-Lintitript
26.09Single7F8YDevazepide7F8Y-CCKA-Devazepide
26.09Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
26.09Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
26.09Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
26.09Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.09Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.09Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
26.09Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
26.09Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
26.09Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
26.09Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
26.09Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
26.09Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
26.09Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
26.09Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
26.09Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
26.09Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
26.09Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
26.09Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
26.09Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
26.09Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Consensusangiotensin_offOrthosteric Ligandat1_off
26.09Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
26.09Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
26.09Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
26.09Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
26.09Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.09Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.09Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
26.09Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
26.09Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
26.09Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
25.93Single4N4WSANT-14N4W-SMO-SANT-1
25.93Single4PY02MeSATP4PY0-P2Y12-2MeSATP
25.93Single5CXVTiotropium5CXV-M1-Tiotropium
25.93Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
25.93Single6CM4Risperidone6CM4-D2-Risperidone
25.93Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
25.93Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
25.93Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
25.93Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
25.93Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
25.93Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
25.93Single8XQJJN2418XQJ-Apelin-JN241
25.93Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
25.93Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
25.93Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
25.81Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
25.81Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
25.81Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
25.81Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
25.81Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
25.81Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
25.71Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
25.71Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
25.71Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
25.64Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
25.00Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
25.00Single3REYXAC3REY-A2A-XAC
25.00Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
25.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
25.00Single5IUBQ274563445IUB-A2A-Q27456344-Na
25.00Single5JTBZM-2413855JTB-A2A-ZM-241385
25.00Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
25.00Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
25.00Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
25.00Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
25.00Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
25.00Single6A94Zotepine6A94-5-HT2A-Zotepine
25.00Single6AQFZM-2413856AQF-A2A-ZM-241385
25.00Single6K1QIRL25006K1Q-ETB-IRL2500
25.00Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
25.00Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
25.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
25.00Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
25.00Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
25.00Single6ZG9GSK10347026ZG9-M1-GSK1034702
25.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
25.00Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
25.00Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
25.00Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
25.00Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
25.00Single7T32ZM-2413857T32-A2A-ZM-241385
25.00Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
25.00Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
25.00Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
25.00Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
25.00Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
25.00Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
25.00Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
25.00Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
25.00Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
25.00Single8PWNTheophylline8PWN-A2A-Theophylline
25.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
25.00Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
25.00Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
25.00Single8XVJMacitentan8XVJ-ETA-Macitentan
25.00Single8XVUCXCL28XVU-CXCR2-CXCL2
25.00Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
25.00Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
25.00Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
25.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
25.00Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
25.00Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
25.00Consensusa2_offOrthosteric Liganda2a_off
25.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
25.00Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
25.00Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
25.00Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
25.00Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
24.32Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
24.32Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
24.32Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
24.24Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
24.24Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
24.14Single5EE7MK08935EE7-Glucagon-MK0893
24.14Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.14Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
24.14Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
24.14Consensuskisspeptin_onOrthosteric Ligandkiss1_on
24.00Single3EMLZM-2413853EML-A2A-ZM-241385
24.00Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
24.00Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
24.00Single5IU8Q274563475IU8-A2A-Q27456347-Na
24.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
24.00Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
24.00Single5T04Neurotensin5T04-NTS1-Neurotensin
24.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
24.00Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
24.00Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
24.00Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
24.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
24.00Single6GPSMK08126GPS-CCR2-MK0812
24.00Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
24.00Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
24.00Single6S0LZM-2413856S0L-A2A-ZM-241385
24.00Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
24.00Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
24.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
24.00Single7PYRPSB-21157PYR-A2A-PSB-2115
24.00Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
24.00Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
24.00Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
24.00Single7YXAONO-54306087YXA-S1P5-ONO-5430608
24.00Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
24.00Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
24.00Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
24.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
24.00Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
24.00Single8X63Mepyramine8X63-H1-Mepyramine
24.00Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
24.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
24.00Single9IYAONO-97105319IYA-GPR55-ONO-9710531
24.00Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
24.00Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
24.00Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
24.00Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
24.00Consensushistamine_offOrthosteric Ligandh1_off
24.00Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
24.00Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
24.00Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
23.81Single3RFMCaffeine3RFM-A2A-Caffeine
23.81Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
23.81Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
23.81Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
23.81Single9CHUNoradrenaline9CHU-β2-Noradrenaline
23.81Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
23.81Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
23.81Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
23.81Consensusp2y_offOrthosteric Ligandp2y1_off
23.81Consensussensory_onOrthosteric Ligandopsins_on
23.68Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
23.68Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
23.68Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
23.68Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.53Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
23.53Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
23.53Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
23.53Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
23.33Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
23.33Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
23.33Single8IEIA1LYA8IEI-GPR156-A1LYA
23.33Single8IEPA1LYA8IEP-GPR156-A1LYA
23.33Single8IEPA1LYA8IEP-GPR156-A1LYA
23.33Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
23.33Single8KIGSHU91198KIG-MC3-SHU9119-Ca
23.33Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
23.33Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
23.33Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
23.33Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
23.33Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
23.08Single4NTJAZD12834NTJ-P2Y12-AZD1283
23.08Single5IUAQ274563485IUA-A2A-Q27456348-Na
23.08Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
23.08Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
23.08Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
23.08Single6GPXMK08126GPX-CCR2-MK0812
23.08Single6HLPNetupitant6HLP-NK1-Netupitant
23.08Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
23.08Single6LUQHaloperidol6LUQ-D2-Haloperidol
23.08Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
23.08Single6S0QZM-2413856S0Q-A2A-ZM-241385
23.08Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
23.08Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
23.08Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
23.08Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
23.08Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
23.08Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
23.08Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
23.08Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
23.08Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
23.08Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
23.08Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
23.08Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
23.08Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
23.08Consensusep_offOrthosteric Ligandep4_off
23.08Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
23.08Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
23.08Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
23.08Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.86Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
22.86Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
22.73Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
22.73Single3UZAGTPL92363UZA-A2A-GTPL9236
22.73Single4XNWMRS25004XNW-P2Y1-MRS2500
22.73Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
22.73Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
22.73Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
22.73Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
22.73Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
22.73Single7V6A-7V6A-M4-PubChem 9864275-Gi1/β1/γ2
22.73Single7WC5Psilocin7WC5-5-HT2A-Psilocin
22.73Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
22.73Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
22.73Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
22.73Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
22.73Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
22.73Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
22.73Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
22.73Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
22.73Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
22.73Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
22.73Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
22.73Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
22.58Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
22.58Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
22.58Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
22.58Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
22.22Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
22.22Single5TZRMK86665TZR-FFA1-MK8666
22.22Single5V56TC1145V56-SMO-TC114
22.22Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
22.22Single6E59L-7607356E59-NK1-L-760735
22.22Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
22.22Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
22.22Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
22.22Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
22.22Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
22.22Single7F1TMIP-1a7F1T-CCR5-MIP-1a
22.22Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
22.22Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
22.22Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
22.22Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
22.22Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8EA0Iperoxo8EA0-M3-Iperoxo
22.22Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
22.22Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
22.22Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
22.22Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
22.22Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
22.22Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
22.22Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
22.22Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
22.22Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
22.22Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
21.74Single4O9RCyclopamine4O9R-SMO-Cyclopamine
21.74Single5L7IVismodegib5L7I-SMO-Vismodegib
21.74Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
21.74Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
21.74Single6TP4ACT-4622066TP4-OX1-ACT-462206
21.74Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
21.74Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
21.74Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
21.74Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
21.74Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
21.74Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
21.74Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
21.74Single9B9Y7DY9B9Y-CB1-7DY
21.74Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
21.74Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
21.62Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
21.43Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
21.43Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
21.43Single5X33BIIL2605X33-BLT1-BIIL260
21.43Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
21.43Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
21.43Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
21.43Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
21.43Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
21.43Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
21.43Single8XWACXCL18XWA-CXCR2-CXCL1
21.43Single8XWMCXCL68XWM-CXCR2-CXCL6
21.43Single8XWSCXCL58XWS-CXCR2-CXCL5
21.43Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
21.43Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
21.43Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
21.43Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
21.21Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
21.21Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
21.21Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
20.93Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
20.83Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
20.83Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
20.83Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
20.83Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
20.83Single4BWBNeurotensin4BWB-NTS1-Neurotensin
20.83Single4QINSAG1.54QIN-SMO-SAG1.5
20.83Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
20.83Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
20.83Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
20.83Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
20.83Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
20.83Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
20.83Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
20.83Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
20.83Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
20.83Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
20.83Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
20.83Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
20.83Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
20.83Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
20.83Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
20.69Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
20.69Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
20.69Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single8XWFCXCL38XWF-CXCR2-CXCL3
20.69Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
20.69Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
20.45Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
20.00Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
20.00Single3RZECidoxepin3RZE-H1-Cidoxepin
20.00Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
20.00Single5MZPCaffeine5MZP-A2A-Caffeine-Na
20.00Single5UVIZM-2413855UVI-A2A-ZM-241385
20.00Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
20.00Single6TPKRetosiban6TPK-OT-Retosiban
20.00Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
20.00Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
20.00Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
20.00Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
20.00Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
20.00Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
20.00Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
20.00Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
20.00Single8IEIA1LYA8IEI-GPR156-A1LYA
20.00Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
20.00Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
20.00Single8K2WAMG4878K2W-CXCR3-AMG487
20.00Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
20.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
20.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
20.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
20.00Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
20.00Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
20.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
20.00Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
20.00Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
20.00Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
20.00Consensusopsins_offOrthosteric Ligandrhodopsin_off
20.00Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
20.00Consensussensory_offOrthosteric Ligandopsins_off
20.00Consensusvasop-oxy_offOrthosteric Ligandot_off
19.44Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
19.44Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
19.44Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
19.44Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
19.35Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
19.35Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.35Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
19.35Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
19.23Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
19.23Single4DAJTiotropium4DAJ-M3-Tiotropium
19.23Single4MQSIperoxo4MQS-M2-Iperoxo
19.23Single4U14Tiotropium4U14-M3-Tiotropium
19.23Single5DSGTiotropium5DSG-M4-Tiotropium
19.23Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
19.23Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
19.23Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
19.23Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
19.23Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
19.23Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
19.23Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.23Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
19.23Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
19.05Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
19.05Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
19.05Single7WC4Serotonin7WC4-5-HT2A-Serotonin
18.92Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
18.92Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
18.92Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
18.75Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
18.52Single4JKVTaladegib4JKV-SMO-Taladegib
18.52Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
18.52Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
18.52Single5CGCHTL142425CGC-mGlu5-HTL14242
18.52Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
18.52Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
18.52Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
18.52Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
18.52Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.52Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
18.52Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
18.52Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
18.52Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
18.52Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
18.52Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
18.52Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
18.18Single3OE8IT1t3OE8-CXCR4-IT1t
18.18Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
18.18Single6TQ9SB-4081246TQ9-OX1-SB-408124
18.18Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
18.18Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
17.95Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
17.95Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.86Single5V57TC1145V57-SMO-TC114
17.86Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
17.86Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
17.86Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
17.86Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
17.86Single9BJKNAM9BJK-μ-Naloxone-NAM
17.86Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
17.65Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
17.39Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
17.39Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
17.39Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
17.39Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.39Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
17.39Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
17.39Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
17.39Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
17.39Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
17.39Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
17.39Consensusgi_sensoryOrthosteric Ligandgi_opsins
17.39Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
17.39Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
17.24Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
17.24Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
17.24Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
17.14Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
17.14Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
16.67Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
16.67Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
16.67Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
16.67Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
16.67Single5CGDHTL142425CGD-mGlu5-HTL14242
16.67Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
16.67Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
16.67Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
16.67Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
16.67Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
16.67Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
16.67Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
16.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
16.67Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
16.67Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
16.67Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
16.13Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
16.13Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
16.13Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
16.00Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
16.00Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
16.00Single5U09Taranabant5U09-CB1-Taranabant
16.00Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
16.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
16.00Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
16.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
16.00Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
16.00Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
16.00Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
16.00Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
16.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
16.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
16.00Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
16.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
16.00Single9BA0A1AKN9BA0-CB1-A1AKN
16.00Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
15.62Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
15.62Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
15.62Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
15.38Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
15.38Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
15.38Single6ZINSR486926ZIN-NTS1-SR48692
15.38Single7VODCariprazine7VOD-5-HT2A-Cariprazine
15.00Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
14.81Single6IIVDaltroban6IIV-TP-Daltroban
14.81Single7F83PF-051904577F83-Ghrelin-PF-05190457
14.81Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
14.81Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
14.81Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
14.81Single9B9ZA1AKO9B9Z-CB1-A1AKO
14.81Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
14.29Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
14.29Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
14.29Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
14.29Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
14.29Single6Z4SSR486926Z4S-NTS1-SR48692
14.29Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
14.29Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
14.29Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
14.29Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
14.29Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.79Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
13.79Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
13.79Single7P2L4YI7P2L-mGlu5-4YI
13.79Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
13.64Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
13.64Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
13.64Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
13.64Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
13.33Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
13.33Single6IIURamatroban6IIU-TP-Ramatroban
13.33Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
13.33Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
13.04Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
13.04Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
12.90Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
12.90Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
12.90Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
12.50Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
12.50Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
12.50Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
12.50Single8JPSCCL78JPS-ACKR1-CCL7
12.50Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
12.00Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
12.00Single6LI0C176LI0-GPR52-C17
12.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
12.00Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
12.00Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
12.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
12.00Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
11.54Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
11.54Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
11.54Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
11.54Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
11.54Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
11.11Single6FFIMMPEP6FFI-mGlu5-MMPEP
11.11Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
11.11Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
11.11Single7VV6C48/807VV6-MRGPRX2-C48/80
11.11Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
10.71Single6FFHFenobam6FFH-mGlu5-Fenobam
10.71Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
10.71Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
10.34Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
10.34Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
10.34Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
10.34Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
10.34Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
10.00Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
10.00Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
9.68Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
9.38Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
9.09Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
8.82Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
8.70Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.70Single8HS2Fab0468HS2-GPR20-Fab046
8.70Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
8.70Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.33Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
8.00Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
8.00Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
8.00Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
7.69Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
7.69Single7UL2SR486927UL2-NTS1-SR48692-Na
7.69Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
7.69Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.69Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
7.69Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.69Consensusneurotensin_offOrthosteric Ligandnts1_off
7.69Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
7.14Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
6.67Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.67Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.45Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
5.56Single7SHEPI; PE7SHE-GPR158-PI; PE
5.00Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.00Single6D35Cholesterol6D35-SMO-Cholesterol
5.00Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.00Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.00Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
5.00Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
5.00Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
5.00Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
5.00Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
5.00Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
5.00Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
5.00Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
5.00Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.00Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.00Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
5.00Single7DTTCa7DTT-CaS-Ca-Ca
5.00Single7DTTCa7DTT-CaS-Ca-Ca
5.00Single7DTUTryptophan7DTU-CaS-Tryptophan
5.00Single7DTUTryptophan7DTU-CaS-Tryptophan
5.00Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.00Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.00Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.00Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.00Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.00Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.00Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.00Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.00Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
5.00Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.00Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.00Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.00Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.00Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.00Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.00Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
5.00Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
5.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.00Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.00Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.00Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.00Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.00Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.00Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.00Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.00Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.00Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
5.00Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.00Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.00Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.00Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.00Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.00Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.00Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
5.00Single7XW7K1-707XW7-TSH-K1-70
5.00Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.00Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.00Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.00Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.00Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.00Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.00Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.00Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.00Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.00Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.00Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.00Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.00Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
5.00Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.00Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.00Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.00Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.00Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
5.00Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
5.00Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.00Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.00Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
5.00Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
5.00Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
5.00Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
5.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
5.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
5.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
5.00Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.00Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.00Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.00Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.00Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.00Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.00Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.00Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.00Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.00Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.00Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.00Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.00Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.00Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.00Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.00Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.00Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.00Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.00Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
5.00Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
5.00Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
5.00Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
5.00Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
5.00Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
5.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.00Single8WVXNorrin8WVX-LGR4-Norrin
5.00Single8WVYNorrin8WVY-LGR4-Norrin
5.00Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.00Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.00Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.00Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.00Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.00Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.00Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
5.00Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.00Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.00Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.00Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.00Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.00Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.00Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.00Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.00Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.00Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.00Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.00Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.76Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.76Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.76Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.76Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.76Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.55Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.55Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.35Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.35Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.35Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
4.35Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.35Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.35Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
4.17Single5L7DCholesterol5L7D-SMO-Cholesterol
4.17Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.17Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.00Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
3.85Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
3.57Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
3.45Single8IYXYL-3658IYX-GPR34-YL-365
3.03Single7SHEPI; PE7SHE-GPR158-PI; PE
2.94Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
2.78Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.78Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.70Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
2.63Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.63Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.56Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.38Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
gi_peptide gi_cck
gi_apelin
gi_compl-pept
gi_endothelin
gi_formylpeptide
gi_galanin
gi_ghrelin
gi_npy
gi_neurotensin
gi_opioid
gi_orexin
gi_relaxin
gi_somatostatin
gi_sensory gi_opsins
gi_alicarboxylic gi_hca
gi_succinate
gi_amine gi_5ht
gi_muscarinic
gi_adrenergic
gi_dopamine
gi_histamine
gi_lipid gi_cannabinoid
gi_ffa
gi_leukotriene
gi_lpa
gi_s1p
gi_nucleotide gi_adenosine
gi_p2y
gi_protein gi_chemokine
gi_chemerin
Net Summary
Imin 2.81442
Number of Linked Nodes 1159
Number of Links 1343
Number of Hubs 197
Number of Links mediated by Hubs 785
Number of Communities 24
Number of Nodes involved in Communities 230
Number of Links involved in Communities 328
Path Summary
Number Of Nodes in MetaPath 112
Number Of Links MetaPath 111
Number of Shortest Paths 2272762
Length Of Smallest Path 3
Average Path Length 32.4831
Length of Longest Path 67
Minimum Path Strength 0.0976534
Average Path Strength 5.17232
Maximum Path Strength 20.6486
Minimum Path Correlation 0.700443
Average Path Correlation 0.964094
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.6129
Average % Of Corr. Nodes 31.3358
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 52.0857
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .




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