Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.47 3.9025466
2G.S1.02 5.296595
3G.S1.05 5.932529
4G.s1h1.05 3.715179
5G.H1.01 4.26754179
6G.S2.08 6.57595
7G.S3.01 5.2825494
8G.S3.03 7.008597
9G.S3.04 7.5875426
10G.S3.06 9.866525
11G.S3.08 4.362529
12G.s3h2.03 4.605429
13G.H2.02 4.25428
14G.H2.03 6.085429
15G.H2.06 7.674529
16G.H2.07 4.722529
17G.h2s4.01 7.585629
18G.s4h3.04 7.10571738
19G.s4h3.05 7.045439
20G.H3.06 3.86436
21G.H3.09 7.30254209
22G.H3.15 5.795428
23G.H3.17 8.05625
24G.H3.18 6.282529
25G.S5.04 3.9125439
26G.S5.05 5.5275409
27G.S5.06 6.405438
28G.HG.01 5.03435
29G.HG.04 7.514539
30G.HG.07 7.3175439
31G.HG.13 3.8525437
32G.hgh4.01 3.9406
33G.hgh4.02 5.19833637
34G.hgh4.05 5.958537
35G.H4.03 6.58534
36G.H4.05 4.355434
37G.H4.10 8.1275436
38G.H4.15 6.655438
39G.h4s6.02 5.1625408
40G.S6.01 5.1854205
41G.S6.02 5.1956137
42G.S6.05 5.3075434
43G.H5.08 5.164598
44G.H5.25 3.99407
45b.1x11 3.07408
46b.1x19 7.015446
47b.h2x1 4.6675405
48b.lhb1x6 4.038503
49b.lhb1x11 4.7825484
50b.b1x6 9.1925409
51b.l1x3 8.188509
52b.b2x1 8.50167628
53b.b2x3 4.8875466
54b.b2x5 7.424567
55b.b4x4 8.57468
56b.b4x5 3.85577
57b.b4x6 11.562569
58b.l4x2 11.8825464
59b.b5x3 7.00571769
60b.b5x5 5.62475
61b.l5x1 5.982578
62b.l5x5 9.58529
63b.b6x5 4.565676
64b.l6x5 6.54254144
65b.b7x1 6.2254144
66b.b7x4 4.215478
67b.l7x2 5.4075429
68b.b8x4 6.636576
69b.l8x8 5.3825474
70b.l9x3 6.8485129
71b.l9x6 5.27667628
72b.l9x7 3.8254127
73b.b10x5 5.07333609
74b.l10x1 4.6975403
75b.l10x4 6.44403
76b.b11x3 3.9625405
77b.b11x4 6.47254129
78b.b12x3 4.235458
79b.b12x5 3.762556
80b.b12x6 8.798336128
81b.b13x3 6.6054124
82b.b13x7 6.072557
83b.l13x3 7.33286759
84b.l13x6 4.966529
85b.l13x7 4.3375459
86b.b14x1 6.745428
87b.b15x1 7.1975459
88b.b15x3 4.6075459
89b.l15x1 4.775627
90b.l15x2 7.6925459
91b.b16x4 10.495456
92b.b16x6 7.595658
93b.b17x7 7.75448
94b.l17x3 9.598549
95b.l17x6 7.2425429
96b.b18x3 5.09448
97b.l18x1 8.051676186
98b.l18x3 8.494185
99b.b19x2 7.365646
100b.b19x4 5.5575448
101b.l19x1 4.695429
102b.l19x2 4.9675409
103b.b20x4 11.2525448
104b.b20x6 8.956546
105b.b20x7 3.38409
106b.b21x1 10.406547
107b.b21x3 7.58446
108b.b21x5 7.04404
109b.b21x7 6.045105
110b.b22x5 5.0925407
111b.l22x5 7.8645229
112b.b23x1 3.2725405
113b.b23x2 4.2454106
114b.b23x6 6.561437107
115b.b24x2 6.70254105
116b.b24x4 6.3085106
117b.b24x5 2.7475405
118b.l24x2 3.99754226
119b.l24x3 4.905405
120b.b25x6 3.65754103
121b.l25x3 7.624589
122b.l25x6 13.3275428
123b.b26x3 4.15406
124b.b27x3 5.465488
125b.l27x1 13.6583629
126b.l27x2 5.32589
127b.b28x4 7.64486
128b.b28x6 7.85833689
129g.h1x11 2.7965219
130g.h2x11 6.67254186
131g.ctx3 6.426589
132g.ctx5 3.945489
133g.ctx6 3.18167606
134g.ctx15 7.6075469
135g.ctx16 5.14857768
1361x43 3.13416
1371x47 3.578517
1381x60 9.134116
139I1x49 5.584117
140I1x50 7.265118
1412x42 4.965618
1422x46 5.47167619
1432x50 7.262519
1442x53 5.075418
1452x54 3.5975407
1462x56 5.05417
1472x57 5.66617
148E1x50 7.076157
1493x24 7.43254156
1503x32 7.5125417
1513x34 5.56754166
1523x37 5.46406
1533x41 4.59405
1543x42 8.34167618
1553x44 4.2075418
1563x50 4.376519
1573x51 4.05408
1583x52 4.386514
159I2x52 4.7025404
160I2x53 7.085617
161I2x57 6.0625417
1624x58 7.4325164
1634x61 4.312515
164E2.N163 5.955415
165E2.I166 4.7575402
166E2x52 5.28414
167E2.M187 5.2325403
168E2.V188 4.12514
1695x36 5.4925404
1705x39 5.32714717
1715x47 8.7825418
1725x50 3.36408
1735x54 5.772518
1745x58 4.79619
1756x37 4.4425408
1766x44 5.75519
1776x48 7.2718
1786x52 9.3825407
1796x54 4.894514
1806x55 6.94415
1816x58 6.286513
182E3.V289 5.068514
1837x34 5.31614
1847x37 6.39406
1857x39 7.184516
1867x42 10.828517
1877x49 7.83419
1887x50 2.5325409
1897x53 4.9175419
1908x47 4.43408
1918x50 6.317118
1928x54 2.95754117
193Lig 9.31875810
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.l1x5 b.l3x1 10.14493.03NoNo079
2b.b2x1 b.l3x1 81.464710.15YesNo089
3b.b2x1 b.l27x1 81.112715.43YesYes289
4b.l25x5 b.l27x1 81.33776.78NoYes079
5b.l25x5 b.l27x2 81.33744.04NoYes079
6b.l25x4 b.l27x2 1009.31NoYes059
7I1x48 b.l25x4 99.96859.53NoNo065
8I1x48 I1x49 99.90585.84NoYes067
91x60 I1x49 99.15175.22YesYes1167
101x60 I1x50 99.380313.57YesYes1168
118x50 I1x50 98.900910.96YesYes1188
128x50 8x54 98.67133.22YesYes1187
131x53 8x54 98.65592.62NoYes097
141x53 7x50 98.58681.77NoYes099
151x50 7x50 98.48254.89NoYes099
161x50 2x50 90.96556.73NoYes099
172x46 2x50 24.10595.43YesYes199
182x46 3x46 15.53714.28YesNo099
192x42 3x46 13.30683.77YesNo089
202x42 3x49 14.15147.17YesNo188
213x49 I2x53 13.93810.34NoYes187
223x52 I2x53 12.97263.97YesYes147
23b.l3x1 b.l5x5 85.15445.48NoYes099
243x52 3x56 11.10744.03YesNo047
253x51 3x56 11.0015.38YesNo087
263x51 3x55 10.68134.03YesNo086
273x55 5x64 10.57456.76NoNo066
285x64 5x68 10.46772.74NoNo067
295x68 G.H5.12 10.24934.11NoNo976
30G.H5.08 G.H5.12 10.14652.59YesNo986
31G.h2s4.01 b.l5x5 42.255813.03YesYes299
32G.S4.04 G.S5.04 17.97073.65NoYes099
33G.H3.08 G.S4.04 22.15087.31NoNo099
34G.H2.04 G.H3.08 22.34833.64NoNo099
35G.H2.04 G.H2.07 22.74364NoYes099
36G.H2.07 G.h2s4.01 42.68064.01YesYes299
37G.H2.07 b.l7x2 42.14323.42YesYes299
38b.l5x5 b.l7x2 42.14416.83YesYes299
39G.H2.07 b.l9x6 75.184.82YesYes298
40b.l13x6 b.l9x6 17.47646.9YesYes298
41b.b14x1 b.l9x6 34.39693.59YesYes288
42b.l15x1 b.l17x6 17.068912.45YesYes279
43G.H2.06 b.b14x1 16.918211.52YesYes298
442x50 7x49 42.42349.42YesYes199
45b.l11x1 b.l9x6 22.57014.35NoYes298
46b.b11x6 b.l11x1 23.2123.71NoNo099
47b.b11x6 b.l9x3 23.052916.74NoYes099
48b.b11x4 b.l9x3 14.16455.48YesYes1299
49b.b10x2 b.b6x2 13.35643.38NoNo068
50b.b10x2 b.b14x3 11.379.52NoNo065
51g.h1x10 g.h1x11 13.30762.66NoYes099
52b.l17x5 b.l17x6 33.54642.94NoYes069
53b.l17x5 b.l19x2 49.01845.89NoYes069
54b.b20x2 b.l19x2 37.69022.89NoYes069
55b.b20x2 b.b20x4 36.07325.17NoYes068
56b.b20x4 b.b20x6 32.15023.21YesYes486
57b.b17x7 b.b20x6 20.478411.79YesYes486
58b.b17x7 b.b21x1 19.07894.78YesYes487
59b.1x19 b.b21x1 16.80815.48YesYes467
60b.1x19 g.h1x14 13.07463.49YesNo069
61g.h1x10 g.h1x14 11.01946.37NoNo099
62b.l17x5 b.l19x1 16.35385.89NoYes069
63b.b24x5 b.b25x5 10.21721.84YesNo054
64b.b25x5 b.b25x6 10.04981.84NoYes043
65b.b23x1 b.lhb1x9 10.65322.85YesNo053
66b.lhb1x11 b.lhb1x9 15.21952.92YesNo043
67b.b28x6 b.lhb1x11 25.13233.49YesYes894
68b.b28x4 b.b28x6 12.7745.8YesYes869
69b.b19x2 b.b20x6 10.995915YesYes466
70b.b27x3 b.b28x6 12.84686.06YesYes889
71b.l25x3 b.l27x2 26.84693.78YesYes899
72b.b27x3 b.l25x3 13.48538.21YesYes889
73b.b28x4 b.l25x3 13.00835.24YesYes869
742x53 7x46 22.96556.46YesNo089
752x50 7x46 25.336310.31YesNo099
762x53 2x56 20.70374.81YesYes187
772x56 3x32 18.98727.3YesYes177
783x32 Lig 19.25866.92YesYes170
793x36 Lig 19.54718.77NoYes170
803x36 6x48 19.70197.28NoYes178
816x48 7x45 40.52514.69YesNo189
827x45 7x49 40.69598.17NoYes199
836x52 Lig 20.29879.32YesYes070
846x48 6x52 19.99444.01YesYes087
85E2.Y183 E2x51 11.22815.05NoNo043
86E2.R173 E2.Y183 13.47348.23NoNo034
87E2.M187 E2.R173 24.69872.48YesNo033
885x36 E2.I166 23.57324.25YesYes042
895x36 5x39 26.92763.49YesYes047
905x39 E2.V188 19.58765.05YesYes174
91E2.V188 Lig 20.66063.8YesYes140
92E2.I170 E2.M187 13.47155.83NoYes043
935x39 E2.N162 10.09884.65YesNo175
945x39 5x43 20.12589.41YesNo075
955x43 Lig 20.10876.75NoYes050
966x51 7x34 14.16985.01NoYes064
977x38 7x42 10.110315.24NoYes057
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
2x563x327.31YesYes7721
2x567x425.051YesYes7722
3x323x364.341YesNo7711
3x327x4211.491YesYes7712
3x32Lig6.921YesYes7010
3x334x573.230NoNo5712
3x334x614.610NoYes5512
3x33Lig12.670NoYes5010
3x366x487.281NoYes7812
3x36Lig8.771NoYes7010
4x565x434.910NoNo5521
4x61E2x525.021YesYes5422
4x615x396.041YesYes5722
E2.V188E2x523.931YesYes4412
5x39E2x523.091YesYes7422
5x39E2.V1885.051YesYes7421
5x40E2.V1883.390NoYes5421
6x55E2.V1884.431YesYes5411
E2.V188Lig3.81YesYes4010
5x395x439.411YesNo7521
5x43Lig6.750NoYes5010
5x446x555.960NoYes6521
5x4616x522.770NoYes5721
5x476x5221.431YesYes8721
6x486x524.011YesYes8721
6x517x345.010NoYes6412
6x517x384.870NoNo6512
6x51Lig13.470NoYes6010
6x52Lig9.320YesYes7010
6x557x344.521YesYes5412
6x55Lig12.851YesYes5010
7x387x4215.240NoYes5722

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
100.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
88.89Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
80.00Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
80.00Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
80.00Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
77.78Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
77.78Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
77.78Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
77.78Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
77.78Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
75.00Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
75.00Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
72.73Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
72.73Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
72.73Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
72.73Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
72.73Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
72.73Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
72.73Single9CHXS-Carazolol9CHX-β2-S-Carazolol
72.73Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
72.73Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
70.00Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
70.00Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
70.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
70.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
70.00Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
70.00Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
70.00Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
70.00Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
70.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
70.00Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
70.00Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
66.67Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
66.67Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
66.67Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
66.67Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
66.67Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
66.67Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
63.64Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
63.64Single6PS0S-Carazolol6PS0-β2-S-Carazolol
63.64Single6PS4ICI118-5516PS4-β2-ICI118-551
63.64Single6PS5S-Propranolol6PS5-β2-S-Propranolol
63.64Single6TPNHTL66416TPN-OX2-HTL6641
63.64Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
63.64Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
63.64Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
63.64Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
63.64Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
63.64Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
63.64Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
63.64Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
63.64Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
63.64Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
63.64Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
63.64Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
63.64Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
63.64Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
63.64Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
63.64Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
63.64Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
63.64Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
63.64Consensusalpha1_onOrthosteric Ligandalpha1a_on
63.64Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
63.64Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
63.64Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
63.64Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
63.64Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
61.54Single2YDVNECA2YDV-A2A-NECA
61.54Single4UHRCGS216804UHR-A2A-CGS21680
61.54Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
61.54Single5G53NECA5G53-A2A-NECA-Gs
61.54Single6J21Aprepitant6J21-NK1-Aprepitant
61.54Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
61.54Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
61.54Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
61.54Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
61.54Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
60.00Single3PBLEticlopride3PBL-D3-Eticlopride
60.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
60.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
60.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
60.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
60.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
60.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
60.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
58.33Single3NY8ICI118-5513NY8-β2-ICI118-551
58.33Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
58.33Single4GBRS-Carazolol4GBR-β2-S-Carazolol
58.33Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
58.33Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
58.33Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
58.33Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
58.33Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
58.33Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
58.33Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
58.33Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
58.33Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
58.33Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
58.33Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
58.33Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
58.33Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
58.33Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
58.33Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
58.33Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
58.33Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
58.33Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
58.33Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
58.33Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.33Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
58.33Single8X64Desloratadine8X64-H1-Desloratadine
58.33Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
58.33Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
58.33Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
58.33Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
58.33Consensus5ht5_onOrthosteric Ligand5ht5a_on
58.33Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
58.33Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
58.33Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
58.33Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
58.33Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
58.33Consensusdopamine_offOrthosteric Ligandd2_off d3_off
58.33Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
58.33Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
58.33Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
57.14Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
57.14Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
57.14Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
57.14Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
55.56Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
55.56Single9CHUNoradrenaline9CHU-β2-Noradrenaline
54.55Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
54.55Single6AKXA4R6AKX-CCR5-A4R
54.55Single6ME2Ramelteon6ME2-MT1-Ramelteon
54.55Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
54.55Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
54.55Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
54.55Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
54.55Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
54.55Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
54.55Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
54.55Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
54.55Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
54.55Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
54.55Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
54.55Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
54.55Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
54.55Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
54.55Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
54.55Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
54.55Consensusalpha2_offOrthosteric Ligandalpha2c_off
53.85Single2RH1S-Carazolol2RH1-β2-S-Carazolol
53.85Single2YCWS-Carazolol2YCW-β1-S-Carazolol
53.85Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
53.85Single5C1MBU725C1M-μ-BU72
53.85Single5D6LS-Carazolol5D6L-β2-S-Carazolol
53.85Single5JQHS-Carazolol5JQH-β2-S-Carazolol
53.85Single5TVNLSD5TVN-5-HT2B-LSD
53.85Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
53.85Single6E67BI1671076E67-β2-BI167107-Gs (fused)
53.85Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
53.85Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
53.85Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
53.85Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
53.85Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
53.85Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
53.85Single7WC6LSD7WC6-5-HT2A-LSD
53.85Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
53.85Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
53.85Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
53.85Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
53.85Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
53.85Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
53.85Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.85Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.85Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.85Single8JXSPF-61428JXS-D1-PF-6142
53.85Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.85Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.85Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
53.85Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
53.85Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
53.85Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
53.85Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
53.85Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
53.85Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
53.85Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
53.85Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
53.85Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
53.85Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
53.85Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
53.85Consensusamine_offonOrthosteric Ligandamine_off amine_on
53.85Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
53.85Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
53.85Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
53.85Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
53.85Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
53.85Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
53.85Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
53.85Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
53.85Consensustrace-amine_onOrthosteric Ligandta1_on
53.33Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
53.33Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
53.33Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
53.33Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
53.33Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
50.00Single3NY9ICI118-5513NY9-β2-ICI118-551
50.00Single3P0GBI1671073P0G-β2-BI167107
50.00Single3RZECidoxepin3RZE-H1-Cidoxepin
50.00Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
50.00Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
50.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
50.00Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
50.00Single4UG2CGS216804UG2-A2A-CGS21680
50.00Single5D5AS-Carazolol5D5A-β2-S-Carazolol
50.00Single5D5BS-Carazolol5D5B-β2-S-Carazolol
50.00Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
50.00Single6A94Zotepine6A94-5-HT2A-Zotepine
50.00Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
50.00Single6H7JIsoprenaline6H7J-β1-Isoprenaline
50.00Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
50.00Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
50.00Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
50.00Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
50.00Single6TPGEMPA6TPG-OX2-EMPA
50.00Single6WGTLSD6WGT-5-HT2A-LSD
50.00Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
50.00Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
50.00Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
50.00Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
50.00Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
50.00Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
50.00Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
50.00Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
50.00Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
50.00Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
50.00Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
50.00Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
50.00Single8E0GBU728E0G-μ-BU72
50.00Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
50.00Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
50.00Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
50.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
50.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
50.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
50.00Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
50.00Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
50.00Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
50.00Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
50.00Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
50.00Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
50.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
50.00Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
50.00Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
50.00Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
50.00Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
50.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
50.00Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
50.00Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
50.00Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
50.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
50.00Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
50.00Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
50.00Single9BJKNaloxone9BJK-μ-Naloxone-NAM
50.00Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
50.00Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
50.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
50.00Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
50.00Consensus5ht2_onOrthosteric Ligand5ht2b_on
50.00Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
50.00Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
50.00Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
50.00Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
50.00Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
50.00Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
50.00Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
50.00Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
50.00Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
50.00Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
47.06Single8WDTphotoNECA8WDT-A2A-photoNECA
47.06Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
47.06Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
46.67Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
46.67Single3D4STimolol3D4S-β2-Timolol
46.67Single4AMIBucindolol4AMI-β1-Bucindolol
46.67Single4LDEBI1671074LDE-β2-BI167107
46.67Single4RWADIPP-NH24RWA-δ-DIPP-NH2
46.67Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
46.67Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
46.67Single6MXTSalmeterol6MXT-β2-Salmeterol
46.67Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
46.67Single7YITNalfurafine7YIT-κ-Nalfurafine
46.67Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
46.67Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
46.67Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
46.67Single8JJ8Formoterol8JJ8-β2-Formoterol
46.67Single8JJLOlodaterol8JJL-β2-Olodaterol
46.67Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
46.67Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
46.67Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
46.67Consensusalpha1_offOrthosteric Ligandalpha1a_off
46.67Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
46.67Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
46.67Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
46.67Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
46.67Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
46.67Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
46.67Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
46.67Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
46.67Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
46.67Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
46.15Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
46.15Single2Y02Carmoterol2Y02-β1-Carmoterol
46.15Single2Y04Salbutamol2Y04-β1-Salbutamol
46.15Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
46.15Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
46.15Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
46.15Single4EJ4Naltrindole4EJ4-δ-Naltrindole
46.15Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
46.15Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
46.15Single6H7MSalbutamol6H7M-β1-Salbutamol
46.15Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
46.15Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
46.15Single6PS1Timolol6PS1-β2-Timolol
46.15Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
46.15Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
46.15Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
46.15Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
46.15Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
46.15Single7WC7Lisuride7WC7-5-HT2A-Lisuride
46.15Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
46.15Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
46.15Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
46.15Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
46.15Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
46.15Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
46.15Single8JJOAlprenolol8JJO-β2-Alprenolol
46.15Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
46.15Single8JXRLSD8JXR-D1-LSD
46.15Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
46.15Single8T1WCVN4248T1W-GPR6-CVN424
46.15Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
46.15Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
46.15Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
46.15Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
46.15Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
46.15Single8X63Mepyramine8X63-H1-Mepyramine
46.15Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
46.15Consensusalpha2_onOrthosteric Ligandalpha2b_on
46.15Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
46.15Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
46.15Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
46.15Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
46.15Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
46.15Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
46.15Consensushistamine_offOrthosteric Ligandh1_off
45.45Single6HLLCP999946HLL-NK1-CP99994
45.45Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
45.45Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
45.45Single6TP4ACT-4622066TP4-OX1-ACT-462206
45.45Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
45.45Single7SRQLSD7SRQ-5-HT2B-LSD
45.45Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
45.45Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
45.45Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
45.45Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
45.45Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
45.45Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
45.45Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
44.44Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
44.44Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
43.75Single5X93K-87945X93-ETB-K-8794
43.75Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
43.75Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
43.75Single6H7LDobutamine6H7L-β1-Dobutamine
43.75Single6IBLArformoterol6IBL-β1-Arformoterol
43.75Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
43.75Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
43.75Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
43.75Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
43.75Single7UM4AS26747237UM4-5-HT5A-AS2674723
43.75Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
43.75Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
43.75Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
43.75Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
43.75Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
43.75Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
43.75Consensusendothelin_offOrthosteric Ligandetb_off
43.75Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
43.75Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
42.86Single2Y03Isoprenaline2Y03-β1-Isoprenaline
42.86Single5WIUNemonapride5WIU-D4-Nemonapride
42.86Single5WIVNemonapride5WIV-D4-Nemonapride-Na
42.86Single5WQCEMPA5WQC-OX2-EMPA
42.86Single5XPRBosentan5XPR-ETB-Bosentan
42.86Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
42.86Single6HLPNetupitant6HLP-NK1-Netupitant
42.86Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
42.86Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
42.86Single6PS6Timolol6PS6-β2-Timolol
42.86Single7C61Ergotamine7C61-5-HT1B-Ergotamine
42.86Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
42.86Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
42.86Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
42.86Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
42.86Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
42.86Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
42.86Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
42.86Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
42.86Single8TF5Oleic acid8TF5-GPR6-Oleic acid
42.86Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
42.86Single8ZMFA1L108ZMF-5-HT2C-A1L10
42.86Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
42.86Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
42.11Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
42.11Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
41.67Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
41.67Single6AKYMaraviroc6AKY-CCR5-Maraviroc
41.67Single6B73MP11046B73-κ-MP1104
41.67Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
41.67Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
41.67Single6TODEMPA6TOD-OX1-EMPA-Na
41.67Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
41.67Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
41.67Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
41.67Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
41.67Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
41.67Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
41.67Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
41.67Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
41.67Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
41.67Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
41.67Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
41.67Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
41.67Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
41.67Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
41.67Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
41.67Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
41.67Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
41.67Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
41.67Consensusorexin_offOrthosteric Ligandox2_off ox1_off
41.67Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
41.18Single5ZTYAM102575ZTY-CB2-AM10257
41.18Single6PT3DPI-2876PT3-δ-DPI-287
41.18Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
41.18Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
41.18Single8X5YAstemizole8X5Y-H1-Astemizole
41.18Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
41.18Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
41.18Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
41.18Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
41.18Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
40.00Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
40.00Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
40.00Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
40.00Single4U15Tiotropium4U15-M3-Tiotropium
40.00Single5V54Methiothepin5V54-5-HT1B-Methiothepin
40.00Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
40.00Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
40.00Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
40.00Single6E59L-7607356E59-NK1-L-760735
40.00Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
40.00Single6J20Aprepitant6J20-NK1-Aprepitant
40.00Single6OL9Tiotropium6OL9-M5-Tiotropium
40.00Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
40.00Single6TQ7SB-3348676TQ7-OX1-SB-334867
40.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
40.00Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
40.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
40.00Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
40.00Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
40.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
40.00Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
40.00Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.00Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
40.00Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
40.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
40.00Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
40.00Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
40.00Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
40.00Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
40.00Single8XVLZibotentan8XVL-ETA-Zibotentan
40.00Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
40.00Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
40.00Consensus5ht1_offOrthosteric Ligand5ht1b_off
40.00Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
40.00Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
40.00Consensusa2_onOrthosteric Liganda2b_on
40.00Consensusa2_on_gpOrthosteric Liganda2b_on_gp
40.00Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
40.00Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
40.00Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
40.00Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
40.00Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
40.00Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
40.00Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
40.00Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
40.00Consensustachykinin_offOrthosteric Ligandnk1_off
38.89Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
38.89Single4IARErgotamine4IAR-5-HT1B-Ergotamine
38.89Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
38.89Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
38.89Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
38.89Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
38.89Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
38.89Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
38.89Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
38.89Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
38.89Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
38.89Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
38.46Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
38.46Single2YDOAdenosine2YDO-A2A-Adenosine
38.46Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
38.46Single4ZJCSB-6740424ZJC-OX1-SB-674042
38.46Single6IQLL7458706IQL-D4-L745870
38.46Single6KUXRS-799486KUX-α2a-RS-79948
38.46Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
38.46Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
38.46Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
38.46Single6VI4JDTic6VI4-κ-JDTic
38.46Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
38.46Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
38.46Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
38.46Single7UL3Famotidine7UL3-H2-Famotidine
38.46Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
38.46Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
38.46Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.46Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
38.46Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
38.46Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.46Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
38.46Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
38.46Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
38.46Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
38.46Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
38.46Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
38.46Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
38.46Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
38.46Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
38.46Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
38.46Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
38.46Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
38.46Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
38.46Consensusopsins_offOrthosteric Ligandrhodopsin_off
38.46Consensussensory_offOrthosteric Ligandopsins_off
38.10Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
37.50Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
37.50Single5CXVTiotropium5CXV-M1-Tiotropium
37.50Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
37.50Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
37.50Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
37.50Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
37.50Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
37.50Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
37.50Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
37.50Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
37.50Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
37.50Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
37.50Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.50Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
37.50Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
37.50Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
37.50Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
37.50Single8JWY2-1188JWY-A2A-2-118
37.50Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.50Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
37.50Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
37.50Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
37.50Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
37.50Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
37.50Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
37.50Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
37.50Consensuslpa_offOrthosteric Ligandlpa1_off
37.50Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
37.50Consensusorexin_onOrthosteric Ligandox2_on
37.50Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
37.50Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
36.84Single3QAKUK-4320973QAK-A2A-UK-432097
36.84Single6HLOAprepitant6HLO-NK1-Aprepitant
36.36Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
36.36Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
36.36Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
36.36Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
36.36Single6ME5Agomelatine6ME5-MT1-Agomelatine
36.36Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
36.36Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
36.36Single7WC5Psilocin7WC5-5-HT2A-Psilocin
36.36Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.36Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
36.36Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
36.36Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
36.36Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
36.36Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
36.36Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
36.36Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
36.36Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
36.36Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
36.36Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
35.71Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
35.71Single2Y01Dobutamine2Y01-β1-Dobutamine
35.71Single4DAJTiotropium4DAJ-M3-Tiotropium
35.71Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
35.71Single4MQSIperoxo4MQS-M2-Iperoxo
35.71Single4QKX35V4QKX-β2-35V
35.71Single4U14Tiotropium4U14-M3-Tiotropium
35.71Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
35.71Single5DHGC-355DHG-NOP-C-35
35.71Single5DHHSB-6121115DHH-NOP-SB-612111
35.71Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
35.71Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
35.71Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
35.71Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
35.71Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
35.71Single6DRXLisuride6DRX-5-HT2B-Lisuride
35.71Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
35.71Single6TOTLemborexant6TOT-OX1-Lemborexant
35.71Single7BU7BI1671077BU7-β1-BI167107
35.71Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
35.71Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
35.71Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
35.71Single7UL4Alvimopan7UL4-μ-Alvimopan
35.71Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
35.71Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
35.71Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
35.71Single8CU6LJ-45178CU6-A2A-LJ-4517
35.71Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
35.71Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
35.71Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
35.71Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
35.71Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
35.71Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
35.71Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
35.71Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
35.71Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
35.71Consensusa3_onOrthosteric Liganda3a_on
35.71Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
35.29Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
35.29Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
35.29Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
35.29Single7EZCUKA7EZC-A2A-UKA
35.29Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
35.29Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
35.29Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
35.29Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
35.29Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
35.29Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
35.29Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.29Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
35.29Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
35.29Consensuschemerin_onOrthosteric Ligandcml1_on
35.29Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
35.29Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
35.29Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
35.00Single5WF5UK-4320975WF5-A2A-UK-432097
35.00Single6PT2KGCHM076PT2-δ-KGCHM07
35.00Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
35.00Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
34.78Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
33.33Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
33.33Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
33.33Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
33.33Single2Y00Dobutamine2Y00-β1-Dobutamine
33.33Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
33.33Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
33.33Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
33.33Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
33.33Single5WF6UK-4320975WF6-A2A-UK-432097
33.33Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
33.33Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
33.33Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
33.33Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
33.33Single6TP6Filorexant6TP6-OX1-Filorexant
33.33Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
33.33Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
33.33Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
33.33Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
33.33Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
33.33Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Single7SK9CCX6627SK9-ACKR3-CCX662
33.33Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
33.33Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
33.33Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
33.33Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
33.33Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
33.33Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
33.33Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
33.33Single7W41PD1762527W41-BB2-PD176252
33.33Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
33.33Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
33.33Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
33.33Single8QOTNanobody-E8QOT-μ-Nanobody-E
33.33Single8S4DCMF-0198S4D-Apelin-CMF-019
33.33Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
33.33Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
33.33Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
33.33Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
33.33Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
33.33Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
33.33Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
33.33Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
33.33Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
33.33Consensusa3_on_gpOrthosteric Liganda3a_on_gp
33.33Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
33.33Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
33.33Consensusadenosine_offOrthosteric Liganda1_off a2_off
33.33Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
33.33Consensusbombesin_offOrthosteric Ligandbb2_off
33.33Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
33.33Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
33.33Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
33.33Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
33.33Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
33.33Consensuskisspeptin_onOrthosteric Ligandkiss1_on
33.33Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
33.33Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
33.33Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
31.82Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
31.82Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
31.58Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
31.58Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
31.58Single8IEBA1LYA8IEB-GPR156-A1LYA
31.58Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
31.58Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.58Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
31.58Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
31.58Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
31.58Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
31.58Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
31.58Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
31.58Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
31.58Consensuslpl_onOrthosteric Ligands1p_on lpa_on
31.58Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
31.25Single4DJHJDTic4DJH-κ-JDTic
31.25Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
31.25Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
31.25Single5XR8AM8415XR8-CB1-AM841
31.25Single5XRAAM115425XRA-CB1-AM11542
31.25Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
31.25Single7B6WCyclazosin7B6W-α1b-Cyclazosin
31.25Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
31.25Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
31.25Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
31.25Single7TUYGSK682753A7TUY-GPR183-GSK682753A
31.25Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
31.25Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
31.25Single8EA0Iperoxo8EA0-M3-Iperoxo
31.25Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
31.25Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
31.25Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
31.25Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
31.25Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
31.25Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
31.25Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
31.25Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
31.25Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
31.25Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
31.25Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
31.25Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
31.25Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
31.25Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
31.25Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
31.25Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
30.77Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
30.77Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
30.77Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
30.77Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
30.77Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
30.77Single5WS3EMPA5WS3-OX2-EMPA
30.77Single6DS0Ly2660976DS0-5-HT2B-Ly266097
30.77Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
30.77Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
30.77Single6ME9Ramelteon6ME9-MT2-Ramelteon
30.77Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
30.77Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
30.77Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
30.77Single7F8ULintitript7F8U-CCKA-Lintitript
30.77Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
30.77Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
30.77Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
30.77Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
30.77Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
30.77Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
30.77Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
30.77Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
30.77Single7XRRLemborexant7XRR-OX2-Lemborexant
30.77Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
30.77Single8GNGIstradefylline8GNG-A2A-Istradefylline
30.77Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
30.77Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
30.77Single8IWESpermidine8IWE-TA9-Spermidine
30.77Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
30.77Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
30.77Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.77Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
30.77Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
30.77Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
30.77Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
30.77Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
30.77Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
30.77Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
30.77Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
30.77Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
30.77Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
30.43Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
30.43Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
30.00Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
30.00Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
30.00Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
30.00Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
30.00Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
30.00Single7WC4Serotonin7WC4-5-HT2A-Serotonin
30.00Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
30.00Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
30.00Single8PWNTheophylline8PWN-A2A-Theophylline
30.00Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
30.00Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
30.00Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
30.00Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
30.00Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
29.41Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
29.41Single6A93Risperidone6A93-5-HT2A-Risperidone
29.41Single6CM4Risperidone6CM4-D2-Risperidone
29.41Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
29.41Single7DFPSpiperone7DFP-D2-Spiperone
29.41Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
29.41Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.41Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
29.41Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
29.41Single8JWZAB9288JWZ-A2A-AB928-Na
29.41Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
29.41Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
29.41Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
29.41Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
29.41Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
29.41Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
29.41Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
29.41Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
29.41Consensuslpl_offOrthosteric Ligands1p_off lpa_off
29.41Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
29.41Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.41Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.17Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
29.17Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
29.17Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
29.17Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
29.17Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
29.17Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
28.57Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
28.57Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
28.57Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
28.57Single5IU7Q274563465IU7-A2A-Q27456346-Na
28.57Single5IUBQ274563445IUB-A2A-Q27456344-Na
28.57Single5JTBZM-2413855JTB-A2A-ZM-241385
28.57Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
28.57Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
28.57Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
28.57Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
28.57Single5UVIZM-2413855UVI-A2A-ZM-241385
28.57Single6AQFZM-2413856AQF-A2A-ZM-241385
28.57Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
28.57Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
28.57Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
28.57Single6TPKRetosiban6TPK-OT-Retosiban
28.57Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
28.57Single7AROLUF58337ARO-A2A-LUF5833-Na
28.57Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
28.57Single7T32ZM-2413857T32-A2A-ZM-241385
28.57Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
28.57Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
28.57Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
28.57Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
28.57Single7VODCariprazine7VOD-5-HT2A-Cariprazine
28.57Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
28.57Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
28.57Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
28.57Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
28.57Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
28.57Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
28.57Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
28.57Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
28.57Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
28.57Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
28.57Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
28.57Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
28.57Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
28.57Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
28.57Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.57Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.57Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
28.57Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
28.57Consensusa2_offOrthosteric Liganda2a_off
28.57Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
28.57Consensusangiotensin_onOrthosteric Ligandat1_on
28.57Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
28.57Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
28.57Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
28.57Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
28.57Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
28.57Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
28.57Consensusvasop-oxy_offOrthosteric Ligandot_off
28.00Single6IGLIRL16206IGL-ETB-IRL1620
28.00Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
28.00Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
27.78Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
27.78Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
27.78Single6K1QIRL25006K1Q-ETB-IRL2500
27.78Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
27.78Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
27.78Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
27.78Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
27.78Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
27.78Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
27.78Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
27.78Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
27.78Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
27.78Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
27.78Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
27.78Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
27.78Single8XVJMacitentan8XVJ-ETA-Macitentan
27.78Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
27.78Consensuscck_onOrthosteric Ligandccka_on cckb_on
27.78Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
27.78Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
27.78Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
27.78Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
27.78Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
27.78Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
27.27Single6TQ9SB-4081246TQ9-OX1-SB-408124
27.27Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
27.27Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
27.27Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
27.27Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
27.27Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
27.27Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
27.27Single8A2OTheophylline8A2O-A2A-Theophylline-Na
27.27Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
27.27Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
27.27Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
27.27Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
27.27Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
27.27Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
27.27Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
27.27Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
27.27Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
27.27Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
27.27Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
27.27Consensussensory_onOrthosteric Ligandopsins_on
27.27Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
27.27Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
27.27Consensusvasop-oxy_onOrthosteric Ligandv2_on
27.27Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
26.92Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
26.92Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
26.92Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
26.92Consensusbombesin_onOrthosteric Ligandbb2_on
26.92Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
26.92Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
26.92Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
26.67Single3EMLZM-2413853EML-A2A-ZM-241385
26.67Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
26.67Single5DSGTiotropium5DSG-M4-Tiotropium
26.67Single5IU8Q274563475IU8-A2A-Q27456347-Na
26.67Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
26.67Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
26.67Single5UENDU1725UEN-A1-DU172
26.67Single5UIGCmpd-15UIG-A2A-Cmpd-1
26.67Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
26.67Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
26.67Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
26.67Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
26.67Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
26.67Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
26.67Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
26.67Single6S0LZM-2413856S0L-A2A-ZM-241385
26.67Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.67Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
26.67Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
26.67Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
26.67Single7PYRPSB-21157PYR-A2A-PSB-2115
26.67Single7V3ZCP559407V3Z-CB1-CP55940
26.67Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
26.67Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
26.67Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
26.67Single8RLNLUF58348RLN-A2A-LUF5834
26.67Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
26.67Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
26.67Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
26.67Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
26.67Single9IYAONO-97105319IYA-GPR55-ONO-9710531
26.67Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
26.67Consensuscck_offOrthosteric Ligandccka_off
26.67Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
26.67Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
26.67Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
26.67Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
26.67Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
26.67Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
26.67Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
26.67Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
26.67Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
26.32Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
26.32Single7XN9L-054,5227XN9-SST2-L-054,522
26.32Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
26.32Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
26.32Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
26.32Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
26.32Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
26.32Single8IEIA1LYA8IEI-GPR156-A1LYA
26.32Single8QJ2pN1628QJ2-MC4-pN162-Gs
26.32Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
26.32Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
26.32Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
26.32Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
26.09Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
26.09Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
26.09Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Single8ZRTET-18ZRT-ETB-ET-1
26.09Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
26.09Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
26.09Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
26.09Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.93Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
25.93Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
25.00Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
25.00Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
25.00Single3UZAGTPL92363UZA-A2A-GTPL9236
25.00Single4NTJAZD12834NTJ-P2Y12-AZD1283
25.00Single5IUAQ274563485IUA-A2A-Q27456348-Na
25.00Single5N2RPSB-365N2R-A2A-PSB-36-Na
25.00Single5N2SPSB365N2S-A1-PSB36
25.00Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
25.00Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
25.00Single6D26Fevipiprant6D26-DP2-Fevipiprant
25.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
25.00Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
25.00Single6LUQHaloperidol6LUQ-D2-Haloperidol
25.00Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
25.00Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
25.00Single6S0QZM-2413856S0Q-A2A-ZM-241385
25.00Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
25.00Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
25.00Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
25.00Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
25.00Single7F8XNN90567F8X-CCKA-NN9056
25.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
25.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7QA8Peptide7QA8-STE2-Peptide
25.00Single7QA8Peptide7QA8-STE2-Peptide
25.00Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
25.00Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
25.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
25.00Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
25.00Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
25.00Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
25.00Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
25.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
25.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
25.00Single8GNEKW-63568GNE-A2A-KW-6356-Na
25.00Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
25.00Single8IEIA1LYA8IEI-GPR156-A1LYA
25.00Single8IEPA1LYA8IEP-GPR156-A1LYA
25.00Single8IEPA1LYA8IEP-GPR156-A1LYA
25.00Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
25.00Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
25.00Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
25.00Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
25.00Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
25.00Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
25.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
25.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
25.00Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
25.00Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
25.00Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
25.00Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
25.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
25.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
25.00Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
25.00Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
25.00Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
25.00Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
25.00Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
25.00Consensusdp_offOrthosteric Liganddp2_off
25.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
25.00Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
25.00Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
25.00Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
25.00Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
25.00Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
25.00Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
25.00Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
25.00Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
25.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
25.00Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
25.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
25.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
24.00Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
24.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
24.00Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
24.00Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
23.81Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
23.81Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
23.81Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
23.81Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
23.81Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
23.81Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
23.81Single8IEBA1LYA8IEB-GPR156-A1LYA
23.81Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
23.81Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
23.81Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
23.81Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
23.81Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
23.81Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
23.53Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
23.53Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
23.53Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
23.53Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
23.53Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
23.53Single7FEECP559407FEE-CB1-CP55940-ZCZ011
23.53Single7PX4PSB-21137PX4-A2A-PSB-2113
23.53Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
23.53Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
23.53Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
23.53Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
23.53Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
23.53Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
23.53Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
23.53Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
23.53Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
23.53Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
23.53Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
23.53Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
23.53Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.53Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
23.53Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
23.53Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
23.53Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
23.53Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.53Consensuslpa_onOrthosteric Ligandlpa1_on
23.53Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
23.53Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
23.53Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
23.53Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
23.08Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
23.08Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
23.08Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
23.08Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
23.08Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
23.08Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
23.08Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
23.08Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
23.08Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
23.08Single8IY6Endothelin-18IY6-ETB-Endothelin-1
23.08Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
23.08Single8K5BNiacin8K5B-HCA2-Niacin
23.08Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
23.08Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
23.08Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
23.08Single9B9Y7DY9B9Y-CB1-7DY
23.08Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
23.08Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
23.08Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
23.08Consensusbradykinin_onOrthosteric Ligandbk2_on
23.08Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
23.08Consensusendothelin_onOrthosteric Ligandetb_on eta_on
23.08Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
23.08Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
22.73Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
22.73Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
22.73Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
22.73Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
22.73Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
22.73Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
22.22Single4N4WSANT-14N4W-SMO-SANT-1
22.22Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
22.22Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
22.22Single5GLHEndothelin-15GLH-ETB-Endothelin-1
22.22Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
22.22Single6IGKEndothelin-36IGK-ETB-Endothelin-3
22.22Single6KQICP559406KQI-CB1-CP55940-Org27569
22.22Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
22.22Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
22.22Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
22.22Single6ZG4HTL00099366ZG4-M1-HTL0009936
22.22Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
22.22Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
22.22Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
22.22Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
22.22Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
22.22Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
22.22Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
22.22Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
22.22Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
22.22Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
22.22Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.22Single8XYIVUF106618XYI-CXCR3-VUF10661
22.22Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
22.22Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
22.22Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
22.22Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
22.22Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
22.22Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
22.22Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
21.74Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
21.74Single6JODAngiotensin II6JOD-AT2-Angiotensin II
21.74Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
21.74Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
21.74Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
21.74Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
21.74Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.74Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
21.74Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
21.74Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
21.43Single3PWHZM-2413853PWH-A2A-ZM-241385
21.43Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
21.43Single4S0VSuvorexant4S0V-OX2-Suvorexant
21.43Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
21.43Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
21.43Single6TPJSuvorexant6TPJ-OX2-Suvorexant
21.43Single7BR3Elagolix7BR3-GnRH1-Elagolix
21.43Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
21.43Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
21.43Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
21.43Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
21.43Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
21.43Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
21.43Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
21.43Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
21.43Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
21.43Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
21.43Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
21.43Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
21.43Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
21.43Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
21.43Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
21.43Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
21.43Single8Y0HVUF114188Y0H-CXCR3-VUF11418
21.43Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
21.43Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
21.43Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
21.43Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
21.43Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
21.43Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
21.43Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
21.43Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
21.05Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
21.05Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
21.05Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.05Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
21.05Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.05Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
21.05Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
21.05Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
21.05Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
21.05Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
21.05Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
21.05Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
21.05Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Consensusprostanoid_offOrthosteric Ligandep_off dp_off
20.83Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
20.83Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
20.83Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.83Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
20.83Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
20.83Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
20.83Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
20.83Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
20.83Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
20.83Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
20.83Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
20.00Single3REYXAC3REY-A2A-XAC
20.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
20.00Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
20.00Single5EE7MK08935EE7-Glucagon-MK0893
20.00Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
20.00Single5MZPCaffeine5MZP-A2A-Caffeine-Na
20.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
20.00Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
20.00Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
20.00Single6TP3Nemorexant6TP3-OX1-Nemorexant
20.00Single6V9SGTPL114036V9S-OX1-GTPL11403
20.00Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
20.00Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
20.00Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
20.00Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
20.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
20.00Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
20.00Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
20.00Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
20.00Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
20.00Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
20.00Single8IHKAcifran8IHK-HCA3-Acifran
20.00Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
20.00Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
20.00Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
20.00Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
20.00Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
20.00Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8K5CAcipimox8K5C-HCA2-Acipimox
20.00Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
20.00Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
20.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
20.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
20.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
20.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
20.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
20.00Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
20.00Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
20.00Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
20.00Consensusgrh_offOrthosteric Ligandgnrh1_off
20.00Consensushca_onOrthosteric Ligandhca2_on
20.00Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
19.23Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
19.23Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
19.23Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
19.23Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
19.23Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
19.23Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
19.23Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
19.23Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
19.05Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
19.05Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
19.05Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
19.05Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
19.05Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
19.05Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
19.05Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
19.05Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
19.05Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
19.05Single8WKYPG-9348WKY-MC4-PG-934
19.05Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
19.05Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
19.05Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
19.05Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
19.05Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.75Single5TGZAM65385TGZ-CB1-AM6538
18.75Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
18.75Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
18.75Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
18.75Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
18.75Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.75Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
18.75Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
18.75Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
18.75Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
18.75Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
18.75Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
18.75Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
18.75Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
18.75Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
18.75Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
18.75Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
18.75Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
18.75Consensusblt_onOrthosteric Ligandblt1_on
18.75Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
18.75Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
18.75Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
18.75Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
18.75Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
18.75Consensushca_on_gpOrthosteric Ligandhca2_on_gp
18.75Consensusleukotriene_onOrthosteric Ligandblt_on
18.75Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
18.75Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
18.75Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
18.52Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
18.52Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
18.52Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
18.52Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
18.18Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
18.18Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
18.18Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
18.18Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
18.18Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
18.18Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
18.18Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
18.18Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
18.18Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
18.18Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
18.18Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
17.86Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
17.86Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
17.86Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
17.86Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
17.86Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
17.86Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
17.65Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
17.65Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
17.65Single5CGCHTL142425CGC-mGlu5-HTL14242
17.65Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
17.65Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
17.65Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
17.65Single7C4SS1P7C4S-S1P3-S1P
17.65Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
17.65Single7SINNPS-21437SIN-CaS-NPS-2143
17.65Single7SINNPS-21437SIN-CaS-NPS-2143
17.65Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
17.65Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
17.65Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.65Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
17.65Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
17.65Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
17.65Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
17.65Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
17.65Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
17.65Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
17.65Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
17.65Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
17.65Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.65Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.65Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
17.39Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
17.39Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
17.39Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
17.39Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
17.39Single6W25SHU91196W25-MC4-SHU9119-Ca
17.39Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
17.39Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
17.39Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
17.39Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
17.39Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
17.39Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
17.39Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
17.39Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
17.39Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
17.24Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
16.67Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
16.67Single3RFMCaffeine3RFM-A2A-Caffeine
16.67Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
16.67Single5TZRMK86665TZR-FFA1-MK8666
16.67Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
16.67Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
16.67Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
16.67Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
16.67Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
16.67Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
16.67Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
16.67Single7R0CAVP7R0C-V2-AVP-Arrestin2
16.67Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
16.67Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
16.67Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
16.67Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
16.67Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
16.67Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
16.67Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
16.67Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
16.67Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
16.67Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
16.67Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
16.67Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
16.67Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
16.67Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
16.67Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
16.67Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
16.67Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
16.67Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
16.67Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
16.67Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
16.67Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
16.67Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
16.67Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
16.67Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
16.13Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
16.00Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
16.00Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
16.00Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
16.00Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
16.00Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
16.00Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
16.00Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
16.00Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
16.00Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
15.79Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
15.79Single4PY02MeSATP4PY0-P2Y12-2MeSATP
15.79Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
15.79Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
15.79Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
15.79Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
15.79Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.79Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
15.79Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
15.79Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
15.79Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
15.79Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
15.38Single3OE6IT1t3OE6-CXCR4-IT1t
15.38Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
15.38Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
15.38Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
15.38Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
15.38Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
15.38Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.38Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
15.38Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
15.38Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
15.38Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
15.38Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.38Consensusgi_sensoryOrthosteric Ligandgi_opsins
15.38Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.38Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.00Single5CGDHTL142425CGD-mGlu5-HTL14242
15.00Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
15.00Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
15.00Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
15.00Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
15.00Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
15.00Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
14.81Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
14.71Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
14.29Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
14.29Single3OE9IT1t3OE9-CXCR4-IT1t
14.29Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
14.29Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
14.29Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
14.29Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
14.29Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
14.29Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
14.29Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
14.29Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
14.29Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
14.29Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
14.29Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
14.29Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
14.29Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
14.29Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
14.29Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
14.29Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
14.29Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
14.29Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
14.29Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
14.29Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
14.29Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
14.29Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
14.29Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
14.29Single8XQJJN2418XQJ-Apelin-JN241
14.29Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
14.29Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
14.29Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
14.29Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
14.29Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
13.64Single4XT1Fractalkine4XT1-US28-Fractalkine
13.64Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
13.64Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
13.33Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
13.33Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
13.33Single3ODUIT1t3ODU-CXCR4-IT1t
13.33Single5U09Taranabant5U09-CB1-Taranabant
13.33Single5ZKQABT-4915ZKQ-PAF-ABT-491
13.33Single7F8YDevazepide7F8Y-CCKA-Devazepide
13.33Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
13.33Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
13.33Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
13.33Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
13.33Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
13.33Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
13.33Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
13.33Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
13.33Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
13.33Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
13.33Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
13.33Single9BA0A1AKN9BA0-CB1-A1AKN
13.33Consensusangiotensin_offOrthosteric Ligandat1_off
13.33Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
13.33Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
13.33Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
13.33Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
13.04Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
13.04Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
13.04Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
13.04Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
13.04Single7XNACYN1548067XNA-SST2-CYN154806
13.04Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
13.04Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
13.04Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
13.04Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
13.04Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
12.90Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
12.90Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
12.90Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single3OE0CVX153OE0-CXCR4-CVX15
12.50Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
12.50Single6FFIMMPEP6FFI-mGlu5-MMPEP
12.50Single6ZG9GSK10347026ZG9-M1-GSK1034702
12.50Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
12.50Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
12.50Single7VV6C48/807VV6-MRGPRX2-C48/80
12.50Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
12.50Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
12.50Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
12.50Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
12.50Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
12.50Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
12.50Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
12.50Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
12.12Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
12.00Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
12.00Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
12.00Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
12.00Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
12.00Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
12.00Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
12.00Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
12.00Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
12.00Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
11.76Single4QIMANTA XV4QIM-SMO-ANTA XV
11.76Single4YAYZD-71554YAY-AT1-ZD-7155
11.76Single6D27CAY104716D27-DP2-CAY10471
11.76Single6FFHFenobam6FFH-mGlu5-Fenobam
11.76Single6GPSMK08126GPS-CCR2-MK0812
11.76Single6IIVDaltroban6IIV-TP-Daltroban
11.76Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
11.76Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
11.76Single7F83PF-051904577F83-Ghrelin-PF-05190457
11.76Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
11.76Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
11.76Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
11.76Single8K5DGSK2560738K5D-HCA2-GSK256073
11.76Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
11.76Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
11.76Single9B9ZA1AKO9B9Z-CB1-A1AKO
11.76Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
11.54Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
11.54Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
11.54Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
11.54Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
11.11Single4XT3Fractalkine4XT3-US28-Fractalkine
11.11Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
11.11Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
11.11Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
11.11Single6FJ3PTH6FJ3-PTH1-PTH
11.11Single6GPXMK08126GPX-CCR2-MK0812
11.11Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
11.11Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
11.11Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
11.11Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
11.11Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
11.11Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
11.11Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
11.11Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
11.11Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
11.11Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
11.11Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
11.11Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
11.11Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
11.11Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
11.11Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
11.11Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
11.11Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
11.11Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
11.11Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
11.11Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
11.11Consensusep_offOrthosteric Ligandep4_off
11.11Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
11.11Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
11.11Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
10.71Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
10.71Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
10.71Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
10.71Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
10.71Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
10.71Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
10.71Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
10.71Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
10.53Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
10.53Single4BV0Neurotensin4BV0-NTS1-Neurotensin
10.53Single5V56TC1145V56-SMO-TC114
10.53Single6OS1TRV0266OS1-AT1-TRV026
10.53Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
10.53Single7F1TMIP-1a7F1T-CCR5-MIP-1a
10.53Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
10.53Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
10.53Single7P2L4YI7P2L-mGlu5-4YI
10.53Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
10.53Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
10.53Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
10.53Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
10.53Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Consensusneurotensin_onOrthosteric Ligandnts1_on
10.53Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
10.53Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
10.53Consensusrelaxin_onOrthosteric Ligandrxfp4_on
10.53Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
10.34Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
10.34Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
10.34Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
10.34Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
10.34Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
10.34Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
10.34Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
10.34Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
10.00Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
10.00Single4XEENeurotensin4XEE-NTS1-Neurotensin
10.00Single4XESNeurotensin4XES-NTS1-Neurotensin
10.00Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
10.00Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
10.00Single6IIURamatroban6IIU-TP-Ramatroban
10.00Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
10.00Single7K15MKD0467K15-BLT1-MKD046-Na
10.00Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
10.00Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
10.00Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
10.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
10.00Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
10.00Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
10.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
10.00Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
10.00Single8XQJJN2418XQJ-Apelin-JN241
10.00Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
10.00Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
10.00Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
10.00Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
10.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
10.00Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
10.00Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
9.68Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
9.68Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
9.68Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
9.68Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
9.52Single4BUONeurotensin4BUO-NTS1-Neurotensin
9.52Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
9.52Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
9.52Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
9.52Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
9.52Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
9.52Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
9.52Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
9.52Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
9.52Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
9.52Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
9.52Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
9.38Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
9.38Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
9.38Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
9.09Single6KNMJN241-96KNM-Apelin-JN241-9
9.09Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
9.09Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
9.09Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
9.09Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
9.09Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
9.09Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
9.09Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
9.09Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
8.70Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
8.70Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.70Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.70Single8KIGSHU91198KIG-MC3-SHU9119-Ca
8.70Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
8.70Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
8.70Consensussomatostatin_offOrthosteric Ligandsst2_off
8.33Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
8.33Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
8.33Single7SHEPI; PE7SHE-GPR158-PI; PE
8.33Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
8.33Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.33Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
8.33Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
8.33Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
8.33Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.33Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
8.33Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
8.11Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
8.00Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
8.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
8.00Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
8.00Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
8.00Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
7.89Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
7.69Single3OE8IT1t3OE8-CXCR4-IT1t
7.69Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
7.69Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
7.69Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
7.69Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
7.69Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
7.69Consensusp2y_offOrthosteric Ligandp2y1_off
7.41Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
7.41Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
7.41Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
7.41Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
7.41Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
7.41Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
7.41Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
7.41Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
7.41Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
7.14Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
7.14Single4XNWMRS25004XNW-P2Y1-MRS2500
7.14Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
7.14Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
7.14Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
7.14Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
7.14Single7SK3CXCL127SK3-ACKR3-CXCL12
7.14Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
7.14Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
7.14Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
7.14Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
7.14Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
6.90Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
6.90Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
6.90Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
6.90Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
6.67Single4O9RCyclopamine4O9R-SMO-Cyclopamine
6.67Single5L7IVismodegib5L7I-SMO-Vismodegib
6.67Single6LI0C176LI0-GPR52-C17
6.67Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
6.67Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
6.67Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
6.67Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
6.67Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
6.67Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
6.67Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
6.67Consensusgq_nucleotideOrthosteric Ligandgq_p2y
6.67Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
6.45Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
6.25Single4BWBNeurotensin4BWB-NTS1-Neurotensin
6.25Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
6.25Single4QINSAG1.54QIN-SMO-SAG1.5
6.25Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
6.25Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
6.25Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
6.25Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
6.25Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
6.25Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
6.25Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
6.25Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
6.25Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
6.25Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
6.25Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
6.25Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
6.25Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
6.25Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
6.25Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
6.25Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
6.25Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
6.25Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
5.88Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
5.88Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
5.88Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
5.88Single6ZINSR486926ZIN-NTS1-SR48692
5.88Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
5.88Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
5.88Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
5.88Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
5.88Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8IYXYL-3658IYX-GPR34-YL-365
5.88Single8JD6N-(3-chlorophenyl)pyridine-2-carboxamide8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
5.88Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
5.88Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
5.88Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
5.88Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
5.88Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
5.88Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
5.56Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
5.56Single5T04Neurotensin5T04-NTS1-Neurotensin
5.56Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
5.56Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
5.56Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
5.56Single7YXAONO-54306087YXA-S1P5-ONO-5430608
5.56Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
5.56Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
5.56Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
5.56Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
5.56Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
5.56Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
5.56Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
5.56Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
5.56Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
5.56Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
5.26Single4JKVTaladegib4JKV-SMO-Taladegib
5.26Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
5.26Single6Z4SSR486926Z4S-NTS1-SR48692
5.26Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
5.26Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
5.26Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
5.26Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
5.26Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
5.26Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
5.26Consensusblt_offOrthosteric Ligandblt1_off
5.00Single5V57TC1145V57-SMO-TC114
5.00Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
5.00Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.00Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.00Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
5.00Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
5.00Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
5.00Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
5.00Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
5.00Single9BJKNAM9BJK-μ-Naloxone-NAM
4.76Single5X33BIIL2605X33-BLT1-BIIL260
4.76Single6OS2TRV0266OS2-AT1-TRV026
4.76Single6YVRNTS8-136YVR-NTS1-NTS8-13
4.76Single7SHEPI; PE7SHE-GPR158-PI; PE
4.76Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
4.76Single8XWACXCL18XWA-CXCR2-CXCL1
4.76Single8XWMCXCL68XWM-CXCR2-CXCL6
4.76Single8XWSCXCL58XWS-CXCR2-CXCL5
4.76Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
4.76Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
4.76Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
4.76Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
4.55Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
4.55Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
4.55Single8XVUCXCL28XVU-CXCR2-CXCL2
4.55Single8XWFCXCL38XWF-CXCR2-CXCL3
4.55Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
4.55Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
4.55Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
4.35Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
4.35Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
4.35Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
4.17Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
4.17Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
4.17Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
4.17Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
4.17Single8XWNCXCL88XWN-CXCR2-CXCL8
4.17Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
4.17Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
4.00Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
4.00Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
4.00Single7SK5CXCL127SK5-ACKR3-CXCL12
3.85Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
3.70Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
3.57Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
2.86Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2

Consensus Members
Id Members
7XTA 7XTA-5-HT4-Serotonin-Gi1/β1/γ2
Net Summary
Imin 2.77
Number of Linked Nodes 832
Number of Links 1056
Number of Hubs 193
Number of Links mediated by Hubs 689
Number of Communities 22
Number of Nodes involved in Communities 278
Number of Links involved in Communities 413
Path Summary
Number Of Nodes in MetaPath 98
Number Of Links MetaPath 97
Number of Shortest Paths 2866021
Length Of Smallest Path 3
Average Path Length 33.7389
Length of Longest Path 61
Minimum Path Strength 1.265
Average Path Strength 6.42162
Maximum Path Strength 24.76
Minimum Path Correlation 0.7
Average Path Correlation 0.989064
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.63158
Average % Of Corr. Nodes 38.0775
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 60.5708
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
5ht_on_gp5ht1_on_gp
5ht2_on_gp
5ht4_on_gp
5ht5_on_gp
5ht6_on_gp
5ht7_on_gp



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