Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.36 6.83125444
2G.HN.40 5.4625447
3G.S2.03 4.6429
4G.S3.03 5.09167638
5G.S3.04 9.99125427
6G.S3.05 3.67875408
7G.S3.06 10.2225427
8G.H2.01 5.935409
9G.H2.05 5.35125428
10G.H2.06 4.79786729
11G.h2s4.01 9.8925409
12G.H3.01 4.98875409
13G.H3.09 5.065149
14G.H3.13 10.934146
15G.H3.17 9.68625
16G.S5.05 4.7554159
17G.s5hg.01 3.039509
18G.hgh4.01 9.45406
19G.hgh4.02 4.8975138
20G.hgh4.05 6.939506
21G.hgh4.08 8.24125406
22G.hgh4.11 5.3575405
23G.hgh4.20 5.7854163
24G.hgh4.21 4.09875404
25G.H4.03 4.27125404
26G.H4.05 7.73625405
27G.H4.07 8.538754165
28G.H4.10 8.3795137
29G.S6.02 7.90375438
30G.s6h5.01 6.733754159
31G.H5.08 5.50167638
32G.H5.17 9.12375435
33b.1x2 2.05375401
34b.1x3 2.70375408
35b.1x6 4.18625408
36b.lh12x2 5.72875408
37b.h2x5 4.3025405
38b.lhb1x6 4.583754103
39b.b1x4 4.34125407
40b.b1x6 8.525449
41b.l1x3 7.5725649
42b.l1x6 9.66529
43b.b2x1 6.80875428
44b.b2x5 7.66417607
45b.l3x2 6.53549
46b.b4x6 8.72749
47b.b4x7 8.24375448
48b.b5x3 6.79917649
49b.l5x5 10.145509
50b.b6x5 3.764506
51b.b8x5 4.4975404
52b.l8x5 4.03625403
53b.l9x3 7.8695209
54b.l9x6 6.3425128
55b.b10x5 5.535509
56b.l11x2 8.1555209
57b.b12x6 9.098508
58b.b13x7 7.843567
59b.l13x3 9.057569
60b.b15x2 5.88456
61b.l15x2 6.605469
62b.b16x4 9.648566
63b.b16x5 4.5225405
64b.b16x6 10.032568
65b.b17x5 7.8775457
66b.b17x7 8.3575458
67b.l17x3 9.8025659
68b.l17x6 7.59529
69b.b18x3 4.294558
70b.l18x1 7.408336216
71b.l18x3 8.115405
72b.b19x2 5.59656
73b.l19x2 8.87875409
74b.b20x2 8.15456
75b.b20x4 10.371558
76b.b20x6 5.815656
77b.b20x7 4.6645229
78b.l20x2 9.241254229
79b.b21x1 6.513557
80b.b21x7 5.17667605
81b.b22x5 6.25625407
82b.l22x5 8.863754109
83b.b23x6 5.74786727
84b.l23x1 6.532526
85b.b24x4 8.3075426
86b.b24x6 6.17875428
87b.b24x7 8.116254109
88b.l24x2 5.993754106
89b.l24x3 4.051505
90b.l25x3 8.25583679
91b.l25x6 12.452528
92b.l26x3 6.236254187
93b.l27x1 9.895729
94b.b28x3 4.60125447
95b.b28x6 9.113579
96b.b28x7 6.64489
97g.h1x8 4.15875407
98g.h1x10 3.41625409
99g.ctx3 6.386509
100g.ctx6 4.3165106
101g.ctx14 6.79375489
102g.ctx15 7.06375489
103g.ctx16 5.33143788
104Lig 27.14812410
105NT 292.373415
1061x31 6.035414
1071x32 9.77625414
1081x39 6.39083618
1091x43 6.223507
1101x60 3.479506
1112x39 6.422599
1122x43 6.32625499
1132x50 8.1725408
1142x53 7.49833618
1152x60 5.8625416
1162x64 5.02917617
117E1 21.1375613
1183x32 5.53083616
1193x33 4.92083617
1203x40 10.424517
1213x42 9.461676119
1223x46 8.7875409
1233x51 4.92125407
124I2 8.7751136
1254x46 5.9625407
1264x50 8.206254118
1274x53 3.4365239
128E2 11815
129E2x51 14.7212418
1305x41 8.78167615
1315x43 4.1675417
1325x52 2.14625404
1335x55 3.33406
1345x58 6.0735179
135I3 5.58111936
1366x32 4.47625408
1376x36 2.01875409
1386x44 6.1745179
1396x47 6.575509
1406x48 10.8588418
1416x51 7.61625416
142E3 6.4675815
1437x33 5.6025417
1447x37 7.59375418
1457x55 1.96625408
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1G.HN.40 b.b5x2 11.60728.85YesNo477
2G.HN.40 b.b5x3 13.25095.6YesYes479
3b.l1x3 b.l3x2 49.82493.78YesYes499
4b.b4x6 b.l1x3 39.9513.705YesYes499
5b.l1x4 b.l3x2 52.453910.855NoYes069
6G.hns1.01 b.l1x4 53.49614.69NoNo046
7G.S1.03 G.hns1.01 21.349423.665NoNo294
8G.h2s4.03 G.hns1.01 32.40693.45NoNo264
9G.S1.03 G.S3.06 22.01774.81NoYes297
10G.S3.06 b.l5x5 23.740519.54YesYes079
11b.l5x5 b.l7x2 23.64025.695YesNo099
12b.l7x2 b.l9x6 23.73863.515NoYes098
13G.s3h2.03 b.l9x6 98.60425.07NoYes098
14G.s3h2.03 b.l7x4 98.64393.96NoNo099
15G.hfs2.07 b.l7x4 99.58985.94NoNo089
16G.hfs2.06 G.hfs2.07 99.66163.71NoNo078
17G.S2.02 G.hfs2.06 99.69723.3NoNo057
18G.S2.02 G.S3.07 99.76813.58NoNo059
19G.S1.06 G.S3.07 99.80336.11NoNo089
20G.S1.06 G.S3.05 99.83844.95NoYes088
21G.S2.06 G.S3.05 99.96573.11NoYes098
22G.S2.06 G.S3.03 1009.11NoYes098
23G.S1.02 G.S3.03 33.25166.79NoYes368
24G.h2s4.03 b.l1x6 33.18866.915NoYes269
25b.b2x1 b.l1x6 21.42974.775YesYes289
26b.b2x1 b.b6x1 43.41744.19YesNo089
27b.b6x1 b.l9x6 43.53055.39NoYes098
28G.S1.02 I2 33.186.58NoYes366
29G.S3.01 G.S3.03 33.18033.93NoYes358
30G.S3.01 I2 33.14456.695NoYes356
31G.H5.08 G.S3.03 33.67273.755YesYes388
32G.H5.08 I2 33.38646.01YesYes386
33G.H5.16 I2 33.59086.38NoYes366
345x68 G.H5.16 33.37628.135NoNo396
355x68 G.H5.17 27.02666.805NoYes395
36G.H5.17 I3 25.15957.6YesYes356
37G.H4.16 I3 24.26444.75NoYes346
38G.H4.16 G.S6.03 24.03334.105NoNo045
39G.H4.12 G.S6.03 23.80215.04NoNo045
40G.H4.12 G.H4.13 22.13878.935NoNo043
41G.H4.13 G.hgh4.08 21.90699.195NoYes036
42G.H4.05 G.hgh4.08 12.51837.2YesYes056
43G.H4.02 G.H4.05 10.98529.065NoYes055
44G.H4.02 G.hgh4.21 10.02655.955NoYes054
45G.H2.01 b.l13x6 32.38765.36YesNo099
46b.l13x6 b.l9x6 32.49659.77NoYes1298
47G.H2.01 G.H2.03 32.070913.955YesNo099
48G.H2.03 G.H2.05 31.99973.49NoYes098
49G.H2.06 G.H2.09 15.55013.39YesNo298
50G.H3.17 b.l27x1 17.36244.685YesYes259
51b.l1x6 b.l27x1 13.085621.465YesYes299
52b.l25x6 b.l27x1 16.852720.49YesYes289
53G.H2.06 b.l17x6 15.21857.605YesYes299
54G.H3.17 b.l23x1 12.42287.26YesYes256
55b.l23x1 b.l25x6 12.392513.1YesYes268
562x43 3x46 16.582510.465YesYes099
572x42 3x46 66.93335.465NoYes099
582x42 3x42 67.31534.11NoYes099
593x42 3x45 69.34969.395YesNo098
603x45 4x46 69.75036.045NoYes087
614x42 4x46 70.35023.475NoYes047
624x42 I2 70.749414.32NoYes346
63b.l17x5 b.l17x6 46.32694.415NoYes069
64b.l17x5 b.l19x2 46.1855.89NoYes069
65b.b20x2 b.l19x2 42.643413.73YesYes069
66b.b20x2 b.b20x4 39.258210.995YesYes568
67b.b20x4 b.b20x6 38.86853.745YesYes586
68b.b17x7 b.b20x6 36.234410.72YesYes586
69b.b17x7 b.b21x1 34.60286.57YesYes587
70b.b21x1 g.h1x14 33.76614.545YesNo079
71g.h1x10 g.h1x14 18.13115.095YesNo099
72b.l21x7 b.l23x1 24.23515.445NoYes256
73b.b23x6 b.l21x7 22.74464.03YesNo275
74b.b23x6 b.b24x6 18.89153.375YesYes278
75b.b21x7 b.b24x6 17.42167.235YesYes058
76b.l26x5 g.ctx4 13.50763.35NoNo057
77g.ctx3 g.ctx4 12.95154.83YesNo097
78b.b1x6 b.b4x6 10.783319.93YesYes499
79b.b3x2 b.b4x6 20.47794.56NoYes059
80b.b2x5 b.b3x2 20.205510.25YesNo075
81b.b17x6 g.h1x14 15.48814.235NoNo079
82b.b16x4 b.b17x6 15.325910.51YesNo067
83b.b16x4 b.b16x6 12.54088.12YesYes668
84b.b13x7 b.b16x6 22.907614.535YesYes678
85b.b13x5 b.b13x7 22.01637.78NoYes047
86b.b12x5 b.b13x5 21.3486.63NoNo064
87b.b11x1 b.b12x5 19.67493.99NoNo056
88b.b11x1 b.l10x1 16.31763.99NoNo053
89b.b14x5 b.l10x1 15.64454.845NoNo053
90b.b10x4 b.b14x5 15.30763.645NoNo065
91b.b10x4 b.b2x4 14.970715.8NoNo066
92b.b17x3 g.h1x10 12.86673.815NoYes059
93b.b16x6 b.b17x3 12.67437.18YesNo685
94b.b2x4 b.b6x5 14.63363.815NoYes066
95b.l26x3 b.l26x5 13.61546.93YesNo075
96b.l26x1 b.l26x3 14.69315.785NoYes1877
97b.b2x5 b.l26x1 15.246417.59YesNo077
982x46 3x46 43.81189.28NoYes099
992x46 2x50 41.05053.655NoYes098
1002x50 3x39 38.089513.895YesNo089
1012x53 3x39 37.64810.245YesNo089
1022x53 Lig 28.93234.88YesYes180
103b.b2x1 b.l27x1 22.94095.305YesYes289
104G.H2.05 b.l17x6 31.294710.72YesYes289
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x32Lig4.8451YesYes6010
3x33Lig3.5851YesYes7010
3x36Lig11.291NoYes6010
3x40Lig10.391YesYes7010
5x41Lig9.8451YesYes5010
2x53Lig4.881YesYes8010
7x37Lig5.5151YesYes8010
7x38Lig8.921NoYes8010
E3Lig8.7251YesYes5010
7x30Lig4.5150NoYes5010
7x33Lig5.091YesYes7010
7x34Lig8.6850NoYes5010
1x32Lig28.651YesYes4010
1x35Lig4.2251NoYes6010
1x39Lig10.1651YesYes8010
2x60Lig6.0051YesYes6010
E1Lig36.581YesYes3010
E2x52Lig5.881NoYes6010
E2Lig27.0551YesYes5010
1x29Lig9.5851NoYes1010
LigNT96.3251YesYes0501
NTNT531.0151YesYes5511
E1NT11.1351YesYes3511
1x281x323.380NoYes1421
1x311x355.681YesNo4621
1x317x3111.831YesNo4421
1x361x397.1650NoYes5821
1x391x403.7451YesNo8712
1x391x434.4651YesYes8712
1x392x614.61YesNo8712
1x397x388.2051YesNo8811
1x432x536.170YesYes7821
1x432x576.940YesNo7722
2x533x369.8051YesNo8611
2x533x3910.2451YesNo8912
2x533x409.261YesYes8711
2x536x484.631YesYes8812
2x563x327.270NoYes6621
2x572x613.650NoNo7722
2x573x323.930NoYes7621
2x603x283.7951YesNo6612
2x603x328.6851YesYes6611
2x62E15.111NoYes4321
2x64E113.481YesYes7321
2x64E2x524.071YesNo7621
E1E130.261YesYes3311
3x26E24.841NoYes7521
3x26E2x5127.271NoYes7822
3x323x334.5251YesYes6711
3x323x363.931YesNo6611
3x334x606.8751YesNo7812
3x335x415.291YesYes7511
3x335x435.9651YesYes7712
3x405x4711.361YesNo7712
3x405x514.2351YesNo7712
3x406x4816.8751YesYes7812
E2E2x5112.841YesYes5812
E2E2x524.161YesNo5611
E2E28.7851YesYes5511
5x41E218.6451YesYes5511
5x415x434.111YesYes5712
5x415x4410.441YesNo5612
5x41E34.361YesYes5511
5x44E33.3751NoYes6521
6x487x375.051YesYes8821
6x517x338.0151YesYes6721
6x517x3713.9951YesYes6821
6x54E34.2850NoYes5521
E3E312.3151YesYes5511
7x33E33.491YesYes7511
7x337x375.8151YesYes7811
1x271x296.6550NoNo0121
1x311x323.4751YesYes4421
1x327x313.61YesNo4411
2x603x314.9651YesNo6412
2x612x643.3950NoYes7722
2x643x284.471YesNo7622
4x605x433.5251NoYes8722
7x31Lig5.261NoYes4010
3x293x333.2850NoYes6721
4x68E22.891NoYes5521
7x32E32.8750NoYes5521
1x341x352.4250NoNo4621
1x291x332.0351NoNo1212

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
95.45Consensuspac_onOrthosteric Ligandpac1_on
84.00Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
84.00Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
83.33Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
80.00Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
76.92Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
76.92Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
74.07Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
73.08Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
72.00Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
72.00Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
72.00Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
71.43Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
70.37Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
69.23Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
68.00Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
66.67Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
65.52Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
65.38Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
65.38Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
64.00Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
63.33Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
62.96Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
62.96Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
62.96Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
62.96Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
62.96Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
62.96Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
62.96Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
61.54Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
61.54Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
61.54Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
60.87Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
60.71Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
60.71Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
60.71Consensusglp_onOrthosteric Ligandglp1_on glp2_on
60.71Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
60.00Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
59.26Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
58.62Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
58.06Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
57.14Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
57.14Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
57.14Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
56.67Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
56.25Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
56.25Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
56.25Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
56.00Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
55.56Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
55.56Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
55.56Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
55.17Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
55.17Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
54.55Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
53.33Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
53.33Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
53.33Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
53.33Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
53.12Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
51.85Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
51.72Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
51.72Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
51.52Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
51.52Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
50.00Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
50.00Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
50.00Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
50.00Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
50.00Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
48.65Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
48.48Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
48.48Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
48.39Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
48.28Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
48.00Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
47.22Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
47.22Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
46.88Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
46.43Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
46.43Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
45.71Consensuspth_onOrthosteric Ligandpth1_on pth2_on
45.16Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
44.12Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
43.75Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
43.75Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
43.75Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
43.33Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
42.86Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
42.31Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
41.94Single6FJ3PTH6FJ3-PTH1-PTH
41.18Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
41.18Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
40.74Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
40.62Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
40.62Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
40.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
40.00Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
40.00Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
40.00Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
40.00Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
40.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
40.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
40.00Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
40.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
40.00Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
39.39Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
39.39Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
39.39Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
39.29Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
38.89Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
38.89Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
38.71Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
38.71Consensuscalcitonin_onOrthosteric Ligandctlike_on
38.71Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
38.46Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
38.46Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
37.93Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
37.93Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
37.93Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
37.84Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
37.50Single4XT3Fractalkine4XT3-US28-Fractalkine
37.50Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
37.50Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
37.50Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
37.50Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
37.50Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
37.50Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
37.50Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
37.50Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
37.50Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
37.50Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
37.04Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
36.67Consensusangiotensin_onOrthosteric Ligandat1_on
36.67Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
36.67Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
36.67Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
36.67Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
36.36Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
36.36Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
36.36Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
36.36Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
36.36Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
36.36Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
36.36Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
36.36Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
36.36Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
36.11Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
35.71Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
35.48Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
35.48Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
35.48Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
35.48Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
35.29Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
35.29Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
35.29Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
35.29Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
35.29Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
35.14Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
35.00Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
34.48Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
34.48Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
34.48Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
34.48Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
34.48Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
34.48Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
34.48Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.38Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
34.38Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
34.38Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
34.38Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
34.38Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
34.29Single6IGKEndothelin-36IGK-ETB-Endothelin-3
34.29Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
34.29Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.29Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.29Consensusbombesin_onOrthosteric Ligandbb2_on
34.29Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
34.29Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
33.33Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
33.33Single6OS2TRV0266OS2-AT1-TRV026
33.33Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
33.33Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
33.33Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
33.33Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
33.33Single7XNACYN1548067XNA-SST2-CYN154806
33.33Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
33.33Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
33.33Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
33.33Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
33.33Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
33.33Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
33.33Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
33.33Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
33.33Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
33.33Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
33.33Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
33.33Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
33.33Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
32.43Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
32.35Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
32.35Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
32.35Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
32.35Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
32.35Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
32.26Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
32.26Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
32.26Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
32.26Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
32.26Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
32.26Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
32.26Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
32.26Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
32.14Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
32.14Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
32.14Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
32.14Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
32.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
32.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
31.43Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
31.43Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
31.25Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
31.25Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.25Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
31.25Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
31.25Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
31.25Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
31.25Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
31.03Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
31.03Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
31.03Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
31.03Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
30.95Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
30.77Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
30.77Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
30.77Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
30.56Single5GLHEndothelin-15GLH-ETB-Endothelin-1
30.56Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
30.56Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
30.56Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
30.56Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
30.30Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
30.30Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
30.30Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
30.30Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
30.30Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
30.30Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
30.30Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
30.30Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
30.30Single8ZRTET-18ZRT-ETB-ET-1
30.30Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
30.30Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
30.30Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
30.30Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
30.30Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
30.00Single4XT1Fractalkine4XT1-US28-Fractalkine
30.00Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
30.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
30.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
30.00Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
30.00Consensussomatostatin_offOrthosteric Ligandsst2_off
29.73Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
29.73Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
29.63Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
29.63Single7TUYGSK682753A7TUY-GPR183-GSK682753A
29.63Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
29.63Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
29.63Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
29.41Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
29.41Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
29.41Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
29.27Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
29.17Single4BWBNeurotensin4BWB-NTS1-Neurotensin
29.17Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
29.17Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
29.03Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
29.03Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
29.03Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
29.03Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
29.03Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
29.03Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
29.03Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
28.95Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
28.57Single4XEENeurotensin4XEE-NTS1-Neurotensin
28.57Single4XESNeurotensin4XES-NTS1-Neurotensin
28.57Single6YVRNTS8-136YVR-NTS1-NTS8-13
28.57Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
28.57Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
28.57Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
28.57Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
28.57Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
28.57Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
28.57Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
28.57Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
28.57Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
28.57Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
28.57Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
28.57Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
28.57Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
28.57Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
28.57Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
28.57Consensuslpa_offOrthosteric Ligandlpa1_off
28.57Consensuslpl_offOrthosteric Ligands1p_off lpa_off
28.21Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
28.21Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
28.12Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
28.12Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.12Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.12Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
28.12Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
28.12Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
28.12Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
28.12Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
28.12Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
28.00Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
28.00Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
28.00Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
28.00Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
27.78Single6IGLIRL16206IGL-ETB-IRL1620
27.78Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
27.78Single8IY6Endothelin-18IY6-ETB-Endothelin-1
27.78Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
27.78Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
27.78Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
27.78Consensusbradykinin_onOrthosteric Ligandbk2_on
27.78Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
27.78Consensusendothelin_onOrthosteric Ligandetb_on eta_on
27.78Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
27.59Single4BUONeurotensin4BUO-NTS1-Neurotensin
27.59Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
27.59Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
27.59Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
27.59Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
27.59Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
27.59Consensuschemerin_onOrthosteric Ligandcml1_on
27.59Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.59Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single6JODAngiotensin II6JOD-AT2-Angiotensin II
27.27Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
27.27Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
27.27Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
27.27Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
27.27Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
27.27Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
27.27Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.27Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
27.27Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
27.27Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
27.27Consensusvasop-oxy_onOrthosteric Ligandv2_on
27.27Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
27.03Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
27.03Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
27.03Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
26.92Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
26.92Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
26.92Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
26.92Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
26.92Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
26.92Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
26.92Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
26.92Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
26.92Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
26.92Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
26.92Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
26.92Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
26.92Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
26.92Consensushca_on_gpOrthosteric Ligandhca2_on_gp
26.92Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
26.92Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
26.67Single4UG2CGS216804UG2-A2A-CGS21680
26.67Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
26.67Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
26.67Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
26.67Single8QJ2pN1628QJ2-MC4-pN162-Gs
26.67Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
26.67Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
26.67Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
26.67Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
26.67Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
26.47Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
26.47Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
26.47Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
26.47Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
26.47Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
26.47Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
26.47Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
26.47Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
26.47Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
26.47Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
26.32Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
26.09Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
25.93Single5C1MBU725C1M-μ-BU72
25.93Single6D26Fevipiprant6D26-DP2-Fevipiprant
25.93Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
25.93Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
25.93Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
25.93Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
25.93Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
25.93Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
25.93Single8S4DCMF-0198S4D-Apelin-CMF-019
25.93Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
25.93Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
25.93Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
25.93Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
25.93Single9B9ZA1AKO9B9Z-CB1-A1AKO
25.93Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
25.93Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
25.93Single9EHSLUF76029EHS-A3A-LUF7602
25.93Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
25.93Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
25.93Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
25.93Consensusdp_offOrthosteric Liganddp2_off
25.81Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
25.81Single7QA8Peptide7QA8-STE2-Peptide
25.81Single7QA8Peptide7QA8-STE2-Peptide
25.81Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
25.81Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
25.81Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
25.81Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
25.81Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
25.81Single8WDTphotoNECA8WDT-A2A-photoNECA
25.81Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
25.81Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
25.81Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
25.81Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
25.81Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
25.81Consensuslpl_onOrthosteric Ligands1p_on lpa_on
25.81Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
25.81Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
25.71Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
25.71Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.71Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
25.71Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
25.71Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
25.71Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
25.64Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
25.00Single3QAKUK-4320973QAK-A2A-UK-432097
25.00Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
25.00Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
25.00Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
25.00Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
25.00Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
25.00Single6OS1TRV0266OS1-AT1-TRV026
25.00Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
25.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
25.00Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
25.00Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
25.00Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
25.00Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
25.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
25.00Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
25.00Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
25.00Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single8E0GBU728E0G-μ-BU72
25.00Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
25.00Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
25.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
25.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
25.00Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
25.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
25.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
25.00Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
25.00Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
25.00Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
25.00Single8K5BNiacin8K5B-HCA2-Niacin
25.00Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
25.00Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
25.00Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
25.00Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
25.00Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
25.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
25.00Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
25.00Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
25.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
25.00Consensusneurotensin_onOrthosteric Ligandnts1_on
25.00Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
24.32Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
24.32Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
24.32Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
24.32Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
24.24Single3OE0CVX153OE0-CXCR4-CVX15
24.24Single5WF5UK-4320975WF5-A2A-UK-432097
24.24Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
24.24Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
24.24Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
24.24Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
24.24Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.24Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
24.24Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
24.24Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
24.24Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
24.14Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
24.14Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
24.14Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
24.14Single6A93Risperidone6A93-5-HT2A-Risperidone
24.14Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
24.14Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
24.14Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
24.14Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
24.14Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
24.14Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
24.14Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
24.14Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
24.14Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
24.14Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
24.14Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
24.14Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
24.14Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.14Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
24.14Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
24.14Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
24.14Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
24.14Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
24.14Single8XYIVUF106618XYI-CXCR3-VUF10661
24.14Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
24.14Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
24.14Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
24.14Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
24.14Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
24.14Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
24.14Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
24.14Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
24.14Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
24.14Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
24.14Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
24.14Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
24.14Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
24.14Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
24.14Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
24.14Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
24.14Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
24.14Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
24.14Consensusorexin_onOrthosteric Ligandox2_on
24.14Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
24.14Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
24.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
24.00Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
24.00Single5U09Taranabant5U09-CB1-Taranabant
24.00Single6AKXA4R6AKX-CCR5-A4R
24.00Single6AKYMaraviroc6AKY-CCR5-Maraviroc
24.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
24.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
24.00Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
24.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
24.00Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
24.00Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
24.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
24.00Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
24.00Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
24.00Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
24.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
24.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
24.00Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
24.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
24.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
24.00Consensusangiotensin_offOrthosteric Ligandat1_off
24.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
24.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
24.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
24.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
23.81Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
23.81Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
23.81Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
23.68Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
23.68Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
23.53Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
23.53Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
23.53Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
23.53Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
23.53Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
23.53Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
23.53Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
23.53Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
23.53Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
23.53Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
23.33Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
23.33Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
23.33Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
23.33Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
23.33Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
23.33Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
23.33Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
23.33Single7EZCUKA7EZC-A2A-UKA
23.33Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
23.33Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
23.33Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
23.33Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
23.33Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
23.33Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
23.33Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
23.33Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
23.33Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
23.33Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
23.33Single8XVUCXCL28XVU-CXCR2-CXCL2
23.33Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
23.33Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
23.33Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
23.33Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
23.33Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
23.33Consensuscck_onOrthosteric Ligandccka_on cckb_on
23.33Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
23.33Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
23.33Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
23.33Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
23.33Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
23.33Consensusprostanoid_offOrthosteric Ligandep_off dp_off
23.08Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
23.08Single4MBSMaraviroc4MBS-CCR5-Maraviroc
23.08Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
23.08Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
23.08Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
23.08Single7AROLUF58337ARO-A2A-LUF5833-Na
23.08Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
23.08Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
23.08Single7F61PF-036547467F61-H3-PF-03654746
23.08Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
23.08Single7T32ZM-2413857T32-A2A-ZM-241385
23.08Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
23.08Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
23.08Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
23.08Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
23.08Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
23.08Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
23.08Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
23.08Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
23.08Single8K5CAcipimox8K5C-HCA2-Acipimox
23.08Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
23.08Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
23.08Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
23.08Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
23.08Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
23.08Single8ZPMAMD0708ZPM-CXCR4-AMD070
23.08Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
23.08Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
23.08Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
23.08Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
23.08Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
23.08Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
23.08Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.08Consensushca_onOrthosteric Ligandhca2_on
23.08Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
23.08Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
23.08Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
22.86Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
22.86Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
22.86Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
22.86Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
22.86Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
22.86Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
22.73Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
22.73Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
22.58Single3NY9ICI118-5513NY9-β2-ICI118-551
22.58Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
22.58Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
22.58Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
22.58Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
22.58Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single7SK9CCX6627SK9-ACKR3-CCX662
22.58Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
22.58Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
22.58Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
22.58Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
22.58Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
22.58Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
22.58Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
22.58Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
22.58Single9IPYJR14a9IPY-C3aB-JR14a
22.58Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
22.58Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
22.58Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
22.58Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
22.58Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
22.58Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
22.22Single3EMLZM-2413853EML-A2A-ZM-241385
22.22Single4YAYZD-71554YAY-AT1-ZD-7155
22.22Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
22.22Single5UENDU1725UEN-A1-DU172
22.22Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
22.22Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
22.22Single6D27CAY104716D27-DP2-CAY10471
22.22Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
22.22Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
22.22Single6PS1Timolol6PS1-β2-Timolol
22.22Single6S0LZM-2413856S0L-A2A-ZM-241385
22.22Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
22.22Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
22.22Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
22.22Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
22.22Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
22.22Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
22.22Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
22.22Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
22.22Single7V3ZCP559407V3Z-CB1-CP55940
22.22Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
22.22Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
22.22Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
22.22Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
22.22Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
22.22Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
22.22Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
22.22Single8K5DGSK2560738K5D-HCA2-GSK256073
22.22Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
22.22Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
22.22Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
22.22Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
22.22Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
22.22Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
22.22Single9CHXS-Carazolol9CHX-β2-S-Carazolol
22.22Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
22.22Consensusa3_onOrthosteric Liganda3a_on
22.22Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
22.22Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
22.22Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
22.22Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
22.22Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
21.88Single4IARErgotamine4IAR-5-HT1B-Ergotamine
21.88Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
21.88Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
21.88Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
21.88Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
21.88Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
21.88Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
21.88Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
21.88Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
21.88Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
21.88Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.88Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
21.88Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
21.88Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.88Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single5IUAQ274563485IUA-A2A-Q27456348-Na
21.43Single5N2RPSB-365N2R-A2A-PSB-36-Na
21.43Single5N2SPSB365N2S-A1-PSB36
21.43Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
21.43Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
21.43Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
21.43Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
21.43Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
21.43Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
21.43Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
21.43Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
21.43Single6S0QZM-2413856S0Q-A2A-ZM-241385
21.43Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
21.43Single7C4SS1P7C4S-S1P3-S1P
21.43Single7C61Ergotamine7C61-5-HT1B-Ergotamine
21.43Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
21.43Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
21.43Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
21.43Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
21.43Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
21.43Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
21.43Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
21.43Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
21.43Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
21.43Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
21.43Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.43Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
21.43Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
21.43Single8JXSPF-61428JXS-D1-PF-6142
21.43Single8QOTNanobody-E8QOT-μ-Nanobody-E
21.43Single8TF5Oleic acid8TF5-GPR6-Oleic acid
21.43Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
21.43Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.43Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.43Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
21.43Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
21.43Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
21.43Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
21.43Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
21.43Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
21.43Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
21.43Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
21.43Consensusa3_on_gpOrthosteric Liganda3a_on_gp
21.43Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
21.43Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
21.43Consensusadenosine_offOrthosteric Liganda1_off a2_off
21.43Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
21.43Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
21.43Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
21.43Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
21.43Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
21.43Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
21.43Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
21.43Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
21.43Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
21.43Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.43Consensustrace-amine_onOrthosteric Ligandta1_on
21.21Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
21.21Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
21.21Single7SK5CXCL127SK5-ACKR3-CXCL12
21.21Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
21.21Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
21.21Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
21.21Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
21.21Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
21.21Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
21.21Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
21.21Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
21.21Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
21.21Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
21.05Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
21.05Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
20.83Single4XNWMRS25004XNW-P2Y1-MRS2500
20.83Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
20.83Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.83Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
20.83Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
20.69Single2YDVNECA2YDV-A2A-NECA
20.69Single3P0GBI1671073P0G-β2-BI167107
20.69Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
20.69Single4BV0Neurotensin4BV0-NTS1-Neurotensin
20.69Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
20.69Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
20.69Single4UHRCGS216804UHR-A2A-CGS21680
20.69Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
20.69Single5G53NECA5G53-A2A-NECA-Gs
20.69Single5XR8AM8415XR8-CB1-AM841
20.69Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
20.69Single7B6WCyclazosin7B6W-α1b-Cyclazosin
20.69Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
20.69Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
20.69Single7F1TMIP-1a7F1T-CCR5-MIP-1a
20.69Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
20.69Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
20.69Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
20.69Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
20.69Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
20.69Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
20.69Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.69Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
20.69Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
20.69Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
20.69Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
20.69Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
20.69Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
20.69Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.69Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
20.69Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
20.69Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
20.69Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
20.69Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
20.69Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
20.69Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
20.69Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
20.69Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
20.69Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
20.69Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
20.69Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
20.69Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.69Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
20.69Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
20.69Single8ZWFJR14a8ZWF-C3aB-JR14a
20.69Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
20.69Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
20.69Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
20.69Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
20.69Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
20.69Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
20.69Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
20.69Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
20.69Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
20.69Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
20.69Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
20.69Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
20.69Consensuslpa_onOrthosteric Ligandlpa1_on
20.69Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
20.69Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
20.69Consensusrelaxin_onOrthosteric Ligandrxfp4_on
20.69Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
20.69Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.69Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
20.59Single6PT2KGCHM076PT2-δ-KGCHM07
20.59Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
20.59Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
20.59Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
20.59Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
20.59Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
20.51Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
20.51Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
20.00Single3OE9IT1t3OE9-CXCR4-IT1t
20.00Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
20.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
20.00Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
20.00Single6LI0C176LI0-GPR52-C17
20.00Single6MXTSalmeterol6MXT-β2-Salmeterol
20.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
20.00Single7DFPSpiperone7DFP-D2-Spiperone
20.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
20.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
20.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
20.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
20.00Single7YITNalfurafine7YIT-κ-Nalfurafine
20.00Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
20.00Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
20.00Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
20.00Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
20.00Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
20.00Single8JJ8Formoterol8JJ8-β2-Formoterol
20.00Single8JJLOlodaterol8JJL-β2-Olodaterol
20.00Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
20.00Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
20.00Single8JWY2-1188JWY-A2A-2-118
20.00Single8JWZAB9288JWZ-A2A-AB928-Na
20.00Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
20.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
20.00Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
20.00Single8XWMCXCL68XWM-CXCR2-CXCL6
20.00Single8XWSCXCL58XWS-CXCR2-CXCL5
20.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
20.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
20.00Single9B9Y7DY9B9Y-CB1-7DY
20.00Single9DGIZ85267113509DGI-CB1-Z8526711350
20.00Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
20.00Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
20.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
20.00Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
20.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.00Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
20.00Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
20.00Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
20.00Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.00Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
20.00Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
20.00Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
20.00Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
20.00Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
20.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
20.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
20.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
20.00Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
20.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.00Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
19.51Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
19.44Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
19.44Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
19.44Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
19.35Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
19.35Single5X93K-87945X93-ETB-K-8794
19.35Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
19.35Single6IBLArformoterol6IBL-β1-Arformoterol
19.35Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
19.35Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
19.35Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
19.35Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
19.35Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
19.35Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.35Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
19.35Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
19.35Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
19.35Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
19.35Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
19.35Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
19.35Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
19.35Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
19.35Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
19.35Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
19.35Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
19.35Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.35Single8XWFCXCL38XWF-CXCR2-CXCL3
19.35Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
19.35Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
19.35Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
19.35Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
19.35Consensusendothelin_offOrthosteric Ligandetb_off
19.35Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
19.35Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
19.35Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
19.23Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
19.23Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
19.23Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
19.23Single5ZKQABT-4915ZKQ-PAF-ABT-491
19.23Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
19.23Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
19.23Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
19.23Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
19.23Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
19.23Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
19.23Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
19.23Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
19.23Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
19.23Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
19.23Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
19.23Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
19.23Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
19.23Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
19.23Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
19.23Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
19.23Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
19.23Single8IWESpermidine8IWE-TA9-Spermidine
19.23Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
19.23Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
19.23Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
19.23Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
19.23Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
19.23Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
19.23Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
19.23Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
19.23Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
19.23Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
19.23Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
19.23Consensusalpha2_offOrthosteric Ligandalpha2c_off
19.23Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
19.23Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
19.23Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
18.92Single7SK3CXCL127SK3-ACKR3-CXCL12
18.92Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
18.75Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
18.75Single5WF6UK-4320975WF6-A2A-UK-432097
18.75Single5ZTYAM102575ZTY-CB2-AM10257
18.75Single6PT3DPI-2876PT3-δ-DPI-287
18.75Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
18.75Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
18.75Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
18.75Single7XN9L-054,5227XN9-SST2-L-054,522
18.75Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
18.75Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
18.75Single8X5YAstemizole8X5Y-H1-Astemizole
18.75Single8XQJJN2418XQJ-Apelin-JN241
18.75Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
18.75Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
18.75Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
18.75Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
18.75Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
18.75Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
18.75Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
18.75Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single2YDOAdenosine2YDO-A2A-Adenosine
18.52Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
18.52Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
18.52Single5IU7Q274563465IU7-A2A-Q27456346-Na
18.52Single5IUBQ274563445IUB-A2A-Q27456344-Na
18.52Single5JTBZM-2413855JTB-A2A-ZM-241385
18.52Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
18.52Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
18.52Single5UVIZM-2413855UVI-A2A-ZM-241385
18.52Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
18.52Single6MH8ZM-2413856MH8-A2A-ZM-241385
18.52Single6PS0S-Carazolol6PS0-β2-S-Carazolol
18.52Single6PS4ICI118-5516PS4-β2-ICI118-551
18.52Single6PS5S-Propranolol6PS5-β2-S-Propranolol
18.52Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
18.52Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
18.52Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
18.52Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
18.52Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
18.52Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
18.52Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.52Single7UL3Famotidine7UL3-H2-Famotidine
18.52Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
18.52Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
18.52Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
18.52Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
18.52Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
18.52Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
18.52Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
18.52Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
18.52Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
18.52Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
18.52Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
18.52Single8IHKAcifran8IHK-HCA3-Acifran
18.52Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
18.52Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
18.52Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
18.52Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
18.52Single8K2WAMG4878K2W-CXCR3-AMG487
18.52Single8RLNLUF58348RLN-A2A-LUF5834
18.52Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
18.52Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
18.52Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
18.52Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
18.52Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
18.52Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
18.52Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
18.52Single8ZPNAMD31008ZPN-CXCR4-AMD3100
18.52Single9AS5Mescaline9AS5-5-HT2A-Mescaline
18.52Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single9BA0A1AKN9BA0-CB1-A1AKN
18.52Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
18.52Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
18.52Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
18.52Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
18.52Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
18.52Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
18.52Consensusa2_offOrthosteric Liganda2a_off
18.52Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
18.52Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
18.52Consensusgrh_offOrthosteric Ligandgnrh1_off
18.52Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
18.42Single9KDFRES-701-39KDF-ETB-RES-701-3
18.42Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
18.18Single7F8XNN90567F8X-CCKA-NN9056
18.18Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
18.18Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
18.18Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
18.18Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
18.18Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
18.18Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
18.18Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Single8XWNCXCL88XWN-CXCR2-CXCL8
18.18Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
18.18Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
18.18Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
18.18Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
18.18Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
18.18Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
17.95Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
17.86Single2Y04Salbutamol2Y04-β1-Salbutamol
17.86Single3NY8ICI118-5513NY8-β2-ICI118-551
17.86Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
17.86Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
17.86Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
17.86Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
17.86Single4GBRS-Carazolol4GBR-β2-S-Carazolol
17.86Single4QKX35V4QKX-β2-35V
17.86Single5DHHSB-6121115DHH-NOP-SB-612111
17.86Single5IU8Q274563475IU8-A2A-Q27456347-Na
17.86Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
17.86Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
17.86Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
17.86Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
17.86Single5T04Neurotensin5T04-NTS1-Neurotensin
17.86Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
17.86Single6GPSMK08126GPS-CCR2-MK0812
17.86Single6H7MSalbutamol6H7M-β1-Salbutamol
17.86Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
17.86Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
17.86Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
17.86Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
17.86Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
17.86Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
17.86Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
17.86Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
17.86Single7PYRPSB-21157PYR-A2A-PSB-2115
17.86Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
17.86Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
17.86Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
17.86Single7UL4Alvimopan7UL4-μ-Alvimopan
17.86Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
17.86Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
17.86Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
17.86Single7WC7Lisuride7WC7-5-HT2A-Lisuride
17.86Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
17.86Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
17.86Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
17.86Single8CU6LJ-45178CU6-A2A-LJ-4517
17.86Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
17.86Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
17.86Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
17.86Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
17.86Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
17.86Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
17.86Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
17.86Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
17.86Single8JJOAlprenolol8JJO-β2-Alprenolol
17.86Single8JXRLSD8JXR-D1-LSD
17.86Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
17.86Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
17.86Single8T1WCVN4248T1W-GPR6-CVN424
17.86Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
17.86Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
17.86Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
17.86Single8X63Mepyramine8X63-H1-Mepyramine
17.86Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
17.86Single9AS1DMT9AS1-5-HT2A-DMT
17.86Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
17.86Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
17.86Single9H37A1IR09H37-A2A-A1IR0-Na
17.86Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
17.86Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
17.86Consensus5ht5_onOrthosteric Ligand5ht5a_on
17.86Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
17.86Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
17.86Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
17.86Consensusdopamine_offOrthosteric Ligandd2_off d3_off
17.86Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
17.86Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
17.86Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
17.86Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
17.86Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
17.86Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
17.86Consensushistamine_offOrthosteric Ligandh1_off
17.65Single6HLOAprepitant6HLO-NK1-Aprepitant
17.65Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
17.65Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
17.65Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
17.65Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
17.65Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
17.65Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
17.65Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
17.65Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
17.39Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
17.39Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
17.39Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
17.24Single2RH1S-Carazolol2RH1-β2-S-Carazolol
17.24Single2Y03Isoprenaline2Y03-β1-Isoprenaline
17.24Single2YCWS-Carazolol2YCW-β1-S-Carazolol
17.24Single4JKVTaladegib4JKV-SMO-Taladegib
17.24Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
17.24Single5D6LS-Carazolol5D6L-β2-S-Carazolol
17.24Single5JQHS-Carazolol5JQH-β2-S-Carazolol
17.24Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
17.24Single5TVNLSD5TVN-5-HT2B-LSD
17.24Single5WIUNemonapride5WIU-D4-Nemonapride
17.24Single5WIVNemonapride5WIV-D4-Nemonapride-Na
17.24Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
17.24Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
17.24Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
17.24Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
17.24Single6E67BI1671076E67-β2-BI167107-Gs(CT)
17.24Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
17.24Single6GPXMK08126GPX-CCR2-MK0812
17.24Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
17.24Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
17.24Single6PS6Timolol6PS6-β2-Timolol
17.24Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
17.24Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
17.24Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
17.24Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
17.24Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
17.24Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
17.24Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
17.24Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
17.24Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
17.24Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
17.24Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
17.24Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GNEKW-63568GNE-A2A-KW-6356-Na
17.24Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
17.24Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
17.24Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
17.24Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
17.24Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
17.24Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
17.24Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
17.24Single8ZMFA1L108ZMF-5-HT2C-A1L10
17.24Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
17.24Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
17.24Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
17.24Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
17.24Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
17.24Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
17.24Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
17.24Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
17.24Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
17.24Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
17.24Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
17.24Consensusamine_offonOrthosteric Ligandamine_off amine_on
17.24Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
17.24Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
17.24Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
17.24Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
17.24Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
17.24Consensusblt_offOrthosteric Ligandblt1_off
17.24Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.24Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
17.24Consensusep_offOrthosteric Ligandep4_off
17.24Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
17.24Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.24Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
17.24Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.24Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.24Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.24Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
17.24Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
17.24Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
17.14Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
17.14Single6W25SHU91196W25-MC4-SHU9119-Ca
17.14Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
17.14Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
17.14Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
17.14Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
17.14Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
17.14Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
16.67Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
16.67Single4DJHJDTic4DJH-κ-JDTic
16.67Single5D5AS-Carazolol5D5A-β2-S-Carazolol
16.67Single5D5BS-Carazolol5D5B-β2-S-Carazolol
16.67Single5V54Methiothepin5V54-5-HT1B-Methiothepin
16.67Single5V56TC1145V56-SMO-TC114
16.67Single5V57TC1145V57-SMO-TC114
16.67Single5XRAAM115425XRA-CB1-AM11542
16.67Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
16.67Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
16.67Single6H7JIsoprenaline6H7J-β1-Isoprenaline
16.67Single6J21Aprepitant6J21-NK1-Aprepitant
16.67Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
16.67Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
16.67Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
16.67Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.67Single6TQ7SB-3348676TQ7-OX1-SB-334867
16.67Single6WGTLSD6WGT-5-HT2A-LSD
16.67Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
16.67Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
16.67Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
16.67Single7FEECP559407FEE-CB1-CP55940-ZCZ011
16.67Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
16.67Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
16.67Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
16.67Single7PX4PSB-21137PX4-A2A-PSB-2113
16.67Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
16.67Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
16.67Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
16.67Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
16.67Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
16.67Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
16.67Single8A2OTheophylline8A2O-A2A-Theophylline-Na
16.67Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
16.67Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8EA0Iperoxo8EA0-M3-Iperoxo
16.67Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
16.67Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
16.67Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
16.67Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
16.67Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
16.67Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
16.67Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
16.67Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
16.67Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
16.67Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
16.67Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
16.67Single9BJKNaloxone9BJK-μ-Naloxone-NAM
16.67Single9CHUNoradrenaline9CHU-β2-Noradrenaline
16.67Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
16.67Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
16.67Consensus5ht1_offOrthosteric Ligand5ht1b_off
16.67Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
16.67Consensusa2_onOrthosteric Liganda2b_on
16.67Consensusa2_on_gpOrthosteric Liganda2b_on_gp
16.67Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
16.67Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
16.67Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
16.67Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
16.67Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
16.67Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
16.67Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
16.67Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
16.67Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
16.67Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
16.67Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.67Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
16.67Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
16.67Consensusp2y_offOrthosteric Ligandp2y1_off
16.22Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.13Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
16.13Single3D4STimolol3D4S-β2-Timolol
16.13Single4AMIBucindolol4AMI-β1-Bucindolol
16.13Single4LDEBI1671074LDE-β2-BI167107
16.13Single4N4WSANT-14N4W-SMO-SANT-1
16.13Single4RWADIPP-NH24RWA-δ-DIPP-NH2
16.13Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
16.13Single6CM4Risperidone6CM4-D2-Risperidone
16.13Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
16.13Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
16.13Single6KQICP559406KQI-CB1-CP55940-Org27569
16.13Single6ZG4HTL00099366ZG4-M1-HTL0009936
16.13Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
16.13Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
16.13Single7K15MKD0467K15-BLT1-MKD046-Na
16.13Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
16.13Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
16.13Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
16.13Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
16.13Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.13Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
16.13Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
16.13Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
16.13Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
16.13Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
16.13Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
16.13Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8XQJJN2418XQJ-Apelin-JN241
16.13Single8XWACXCL18XWA-CXCR2-CXCL1
16.13Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
16.13Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
16.13Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
16.13Consensusalpha1_offOrthosteric Ligandalpha1a_off
16.13Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
16.13Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.13Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.00Single3OE6IT1t3OE6-CXCR4-IT1t
16.00Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
16.00Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
16.00Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
16.00Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
16.00Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
16.00Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
16.00Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
16.00Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
16.00Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
16.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
16.00Single9LRCHistamine9LRC-H4-Histamine
16.00Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
16.00Consensus5ht2_onOrthosteric Ligand5ht2b_on
16.00Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
16.00Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
15.62Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
15.62Single5CGDHTL142425CGD-mGlu5-HTL14242
15.62Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
15.62Single6H7LDobutamine6H7L-β1-Dobutamine
15.62Single6K1QIRL25006K1Q-ETB-IRL2500
15.62Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
15.62Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single7UM4AS26747237UM4-5-HT5A-AS2674723
15.62Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
15.62Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
15.62Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
15.62Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8XVJMacitentan8XVJ-ETA-Macitentan
15.62Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
15.62Single8ZPLHF511168ZPL-CXCR4-HF51116
15.62Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
15.62Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
15.62Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
15.62Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
15.62Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
15.62Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
15.62Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
15.62Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single4O9RCyclopamine4O9R-SMO-Cyclopamine
15.38Single7SRQLSD7SRQ-5-HT2B-LSD
15.38Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
15.38Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
15.38Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
15.38Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
15.38Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
15.38Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
15.38Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
15.38Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
15.38Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
15.38Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
15.38Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
15.38Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
15.38Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
15.38Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
15.38Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
15.38Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
15.38Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
15.38Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
15.38Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
15.38Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
15.38Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
15.38Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
15.38Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
15.38Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
15.38Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
15.38Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
15.38Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
15.15Single6KNMJN241-96KNM-Apelin-JN241-9
15.15Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
15.15Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
15.15Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
15.15Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
15.15Consensuskisspeptin_onOrthosteric Ligandkiss1_on
14.81Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
14.81Single3ODUIT1t3ODU-CXCR4-IT1t
14.81Single3PWHZM-2413853PWH-A2A-ZM-241385
14.81Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
14.81Single4QINSAG1.54QIN-SMO-SAG1.5
14.81Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
14.81Single6B73MP11046B73-κ-MP1104
14.81Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
14.81Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
14.81Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
14.81Single6ME2Ramelteon6ME2-MT1-Ramelteon
14.81Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
14.81Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
14.81Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
14.81Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
14.81Single7BR3Elagolix7BR3-GnRH1-Elagolix
14.81Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
14.81Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
14.81Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
14.81Single7F8ULintitript7F8U-CCKA-Lintitript
14.81Single7F8YDevazepide7F8Y-CCKA-Devazepide
14.81Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.81Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.81Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
14.81Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
14.81Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
14.81Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
14.81Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
14.81Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
14.81Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
14.81Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
14.81Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
14.81Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
14.81Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
14.81Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
14.81Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
14.81Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
14.81Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
14.81Single8Y0HVUF114188Y0H-CXCR3-VUF11418
14.81Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
14.81Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
14.81Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
14.81Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
14.81Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
14.81Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
14.81Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
14.81Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
14.81Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
14.81Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
14.81Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
14.81Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
14.81Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
14.81Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
14.81Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
14.81Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
14.81Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.81Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.81Consensusorexin_offOrthosteric Ligandox2_off ox1_off
14.81Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
14.81Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.81Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
14.71Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
14.71Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
14.71Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
14.71Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
14.71Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
14.71Single8KIGSHU91198KIG-MC3-SHU9119-Ca
14.71Single8WKYPG-9348WKY-MC4-PG-934
14.71Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
14.71Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
14.71Single9M4TSilodosin9M4T-Alpha1A-Silodosin
14.71Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
14.71Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
14.71Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
14.29Single3REYXAC3REY-A2A-XAC
14.29Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
14.29Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
14.29Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
14.29Single4ZJCSB-6740424ZJC-OX1-SB-674042
14.29Single6A94Zotepine6A94-5-HT2A-Zotepine
14.29Single6AQFZM-2413856AQF-A2A-ZM-241385
14.29Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
14.29Single6KUXRS-799486KUX-α2a-RS-79948
14.29Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
14.29Single6TPGEMPA6TPG-OX2-EMPA
14.29Single6V9SGTPL114036V9S-OX1-GTPL11403
14.29Single6VI4JDTic6VI4-κ-JDTic
14.29Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
14.29Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
14.29Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
14.29Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
14.29Single6ZG9GSK10347026ZG9-M1-GSK1034702
14.29Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
14.29Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
14.29Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
14.29Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
14.29Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
14.29Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
14.29Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
14.29Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
14.29Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
14.29Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
14.29Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
14.29Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
14.29Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
14.29Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
14.29Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
14.29Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
14.29Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
14.29Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
14.29Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9AS3LSD9AS3-5-HT2A-LSD
14.29Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
14.29Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
14.29Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
14.29Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
14.29Consensusalpha1_onOrthosteric Ligandalpha1a_on
14.29Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
14.29Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
14.29Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
14.29Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
14.29Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
14.29Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
14.29Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
13.89Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.89Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
13.89Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
13.89Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
13.79Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
13.79Single2Y01Dobutamine2Y01-β1-Dobutamine
13.79Single2Y02Carmoterol2Y02-β1-Carmoterol
13.79Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
13.79Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
13.79Single4DAJTiotropium4DAJ-M3-Tiotropium
13.79Single4EJ4Naltrindole4EJ4-δ-Naltrindole
13.79Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
13.79Single4MQSIperoxo4MQS-M2-Iperoxo
13.79Single4U14Tiotropium4U14-M3-Tiotropium
13.79Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
13.79Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
13.79Single5DHGC-355DHG-NOP-C-35
13.79Single5TGZAM65385TGZ-CB1-AM6538
13.79Single5UIGCmpd-15UIG-A2A-Cmpd-1
13.79Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
13.79Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
13.79Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
13.79Single6DRXLisuride6DRX-5-HT2B-Lisuride
13.79Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
13.79Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
13.79Single6TOTLemborexant6TOT-OX1-Lemborexant
13.79Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
13.79Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
13.79Single7BU7BI1671077BU7-β1-BI167107
13.79Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
13.79Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
13.79Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
13.79Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
13.79Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
13.79Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
13.79Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
13.79Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
13.79Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
13.79Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
13.79Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
13.79Single7YXAONO-54306087YXA-S1P5-ONO-5430608
13.79Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
13.79Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
13.79Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
13.79Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
13.79Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
13.79Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
13.79Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
13.79Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
13.79Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
13.79Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
13.79Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
13.79Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
13.79Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
13.79Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
13.79Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
13.79Single8X64Desloratadine8X64-H1-Desloratadine
13.79Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
13.79Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
13.79Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
13.79Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
13.79Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
13.79Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
13.79Single9JEAAtropine9JEA-M1-Atropine
13.79Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
13.79Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
13.79Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
13.79Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
13.79Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
13.79Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
13.79Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
13.79Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
13.79Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
13.79Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
13.79Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
13.79Consensusalpha2_onOrthosteric Ligandalpha2b_on
13.79Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
13.79Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
13.79Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
13.79Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
13.79Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
13.79Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
13.79Consensusblt_onOrthosteric Ligandblt1_on
13.79Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
13.79Consensuscck_offOrthosteric Ligandccka_off
13.79Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
13.79Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
13.79Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
13.79Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
13.79Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
13.79Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
13.79Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
13.79Consensusleukotriene_onOrthosteric Ligandblt_on
13.79Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
13.79Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
13.79Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
13.79Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
13.51Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
13.51Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
13.33Single2Y00Dobutamine2Y00-β1-Dobutamine
13.33Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
13.33Single5CGCHTL142425CGC-mGlu5-HTL14242
13.33Single5WQCEMPA5WQC-OX2-EMPA
13.33Single5XPRBosentan5XPR-ETB-Bosentan
13.33Single6LUQHaloperidol6LUQ-D2-Haloperidol
13.33Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
13.33Single6TP6Filorexant6TP6-OX1-Filorexant
13.33Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
13.33Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
13.33Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
13.33Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
13.33Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
13.33Single7W41PD1762527W41-BB2-PD176252
13.33Single7WC6LSD7WC6-5-HT2A-LSD
13.33Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
13.33Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
13.33Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
13.33Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
13.33Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
13.33Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
13.33Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
13.33Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
13.33Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
13.33Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
13.33Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
13.33Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
13.33Consensusbombesin_offOrthosteric Ligandbb2_off
13.33Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
13.33Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
13.33Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
13.33Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.16Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
13.04Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
12.90Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
12.90Single4U15Tiotropium4U15-M3-Tiotropium
12.90Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
12.90Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
12.90Single6J20Aprepitant6J20-NK1-Aprepitant
12.90Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
12.90Single6OL9Tiotropium6OL9-M5-Tiotropium
12.90Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
12.90Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
12.90Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
12.90Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
12.90Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
12.90Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
12.90Single9AS9RS130-1809AS9-5-HT2A-RS130-180
12.90Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
12.90Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
12.90Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.90Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
12.90Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
12.90Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
12.90Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
12.50Single5CXVTiotropium5CXV-M1-Tiotropium
12.50Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
12.50Single5X33BIIL2605X33-BLT1-BIIL260
12.50Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
12.50Single6IIURamatroban6IIU-TXA2-Ramatroban
12.50Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
12.50Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
12.50Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8HS2Fab0468HS2-GPR20-Fab046
12.50Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
12.50Single8PWNTheophylline8PWN-A2A-Theophylline
12.50Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.50Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
12.50Single9BJKNAM9BJK-μ-Naloxone-NAM
12.50Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.50Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.50Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
12.50Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
12.50Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
12.12Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
12.12Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
12.12Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single3OE8IT1t3OE8-CXCR4-IT1t
12.00Single3RFMCaffeine3RFM-A2A-Caffeine
12.00Single6TQ9SB-4081246TQ9-OX1-SB-408124
12.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
12.00Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
12.00Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
12.00Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
12.00Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
11.76Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
11.76Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
11.76Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
11.76Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
11.76Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
11.76Single9JF4PD1683689JF4-BB1-PD168368
11.76Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
11.54Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
11.54Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
11.54Single6ME5Agomelatine6ME5-MT1-Agomelatine
11.54Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
11.54Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.54Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
11.54Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.54Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
11.54Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
11.54Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
11.54Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
11.54Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
11.54Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
11.54Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
11.54Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
11.43Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.43Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.43Single8IEBA1LYA8IEB-GPR156-A1LYA
11.43Single8IEIA1LYA8IEI-GPR156-A1LYA
11.43Single8IEPA1LYA8IEP-GPR156-A1LYA
11.43Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.43Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
11.43Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.43Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Single3PBLEticlopride3PBL-D3-Eticlopride
11.11Single5L7IVismodegib5L7I-SMO-Vismodegib
11.11Single6HLLCP999946HLL-NK1-CP99994
11.11Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
11.11Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.11Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.11Single7UL2SR486927UL2-NTS1-SR48692-Na
11.11Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
11.11Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
11.11Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
11.11Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
11.11Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
11.11Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.11Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
11.11Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
11.11Single9AS7Psilocin9AS7-5-HT2A-Psilocin
11.11Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
11.11Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
11.11Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
11.11Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
11.11Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
11.11Consensusgq_nucleotideOrthosteric Ligandgq_p2y
11.11Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
11.11Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.11Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
11.11Consensusneurotensin_offOrthosteric Ligandnts1_off
11.11Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
10.71Single4S0VSuvorexant4S0V-OX2-Suvorexant
10.71Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
10.71Single5WS3EMPA5WS3-OX2-EMPA
10.71Single6DS0Ly2660976DS0-5-HT2B-Ly266097
10.71Single6ME9Ramelteon6ME9-MT2-Ramelteon
10.71Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
10.71Single6TODEMPA6TOD-OX1-EMPA-Na
10.71Single6TPJSuvorexant6TPJ-OX2-Suvorexant
10.71Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
10.71Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
10.71Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
10.71Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
10.71Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
10.71Single7XRRLemborexant7XRR-OX2-Lemborexant
10.71Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
10.71Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
10.71Single9H2XA1IR19H2X-A2A-A1IR1-Na
10.71Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
10.71Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
10.71Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
10.71Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
10.53Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
10.53Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
10.53Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
10.34Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
10.34Single3RZECidoxepin3RZE-H1-Cidoxepin
10.34Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
10.34Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
10.34Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
10.34Single6IQLL7458706IQL-D4-L745870
10.34Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
10.34Single6TP3Nemorexant6TP3-OX1-Nemorexant
10.34Single6TPNHTL66416TPN-OX2-HTL6641
10.34Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
10.34Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
10.34Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
10.34Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
10.34Single7VV6C48/807VV6-MRGPRX2-C48/80
10.34Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
10.34Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
10.34Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
10.34Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.34Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
10.34Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
10.34Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
10.34Single9ARXSerotonin9ARX-5-HT2A-Serotonin
10.34Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
10.34Consensusopsins_offOrthosteric Ligandrhodopsin_off
10.34Consensussensory_offOrthosteric Ligandopsins_off
10.00Single4QIMANTA XV4QIM-SMO-ANTA XV
10.00Single5DSGTiotropium5DSG-M4-Tiotropium
10.00Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
10.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
10.00Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
10.00Single6IIVDaltroban6IIV-TXA2-Daltroban
10.00Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
10.00Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7F83PF-051904577F83-Ghrelin-PF-05190457
10.00Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
10.00Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
10.00Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
10.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
10.00Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
10.00Single9IYAONO-97105319IYA-GPR55-ONO-9710531
10.00Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
9.68Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
9.68Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
9.68Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
9.68Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
9.68Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
9.68Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
9.68Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
9.68Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
9.68Single6Z4SSR486926Z4S-NTS1-SR48692
9.68Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
9.68Single7SINNPS-21437SIN-CaS-NPS-2143
9.68Single7SINNPS-21437SIN-CaS-NPS-2143
9.68Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
9.68Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
9.68Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
9.68Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
9.68Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
9.68Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
9.68Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
9.68Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
9.68Single9HAPTolvaptan9HAP-V2-Tolvaptan
9.68Single9HC04YI9HC0-mGlu5-4YI
9.68Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
9.68Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
9.68Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
9.38Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
9.38Single5TZRMK86665TZR-FFA1-MK8666
9.38Single6E59L-7607356E59-NK1-L-760735
9.38Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
9.38Single7P2L4YI7P2L-mGlu5-4YI
9.38Single7R0CAVP7R0C-V2-AVP-Arrestin2
9.38Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
9.38Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
9.38Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
9.38Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
9.38Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
9.38Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
9.38Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
9.38Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
9.38Single8XVLZibotentan8XVL-ETA-Zibotentan
9.38Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
9.38Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
9.38Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
9.38Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
9.38Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
9.38Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
9.38Consensustachykinin_offOrthosteric Ligandnk1_off
9.09Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
9.09Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
9.09Single4PY02MeSATP4PY0-P2Y12-2MeSATP
9.09Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
9.09Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
9.09Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
9.09Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
9.09Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
8.82Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
8.82Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
8.82Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
8.82Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
8.82Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
8.70Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
8.57Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single5MZPCaffeine5MZP-A2A-Caffeine-Na
8.33Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
8.33Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
8.33Single8IEIA1LYA8IEI-GPR156-A1LYA
8.33Single8IEPA1LYA8IEP-GPR156-A1LYA
8.33Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
8.11Single8IEBA1LYA8IEB-GPR156-A1LYA
8.00Single7WC4Serotonin7WC4-5-HT2A-Serotonin
7.69Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
7.69Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
7.69Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.69Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
7.69Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
7.69Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
7.69Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
7.69Consensussensory_onOrthosteric Ligandopsins_on
7.41Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
7.41Single3UZAGTPL92363UZA-A2A-GTPL9236
7.41Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
7.41Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
7.41Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
7.41Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
7.41Single7WC5Psilocin7WC5-5-HT2A-Psilocin
7.41Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.41Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.41Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
7.41Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
7.41Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
7.41Single8JPSCCL78JPS-ACKR1-CCL7
7.41Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
7.41Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
7.41Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.41Consensusgi_sensoryOrthosteric Ligandgi_opsins
7.41Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.41Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.41Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
7.41Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
7.41Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
7.14Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
7.14Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
7.14Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
7.14Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
7.14Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
7.14Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
7.14Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
7.14Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
7.14Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
7.14Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.14Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
7.14Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
7.14Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.14Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
7.14Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.14Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
7.14Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.90Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
6.90Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
6.90Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
6.90Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
6.90Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
6.90Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
6.90Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
6.90Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
6.90Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
6.90Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
6.90Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.90Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.90Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
6.90Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
6.90Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
6.90Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
6.90Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
6.90Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
6.90Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
6.90Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
6.90Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.90Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.90Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
6.90Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
6.67Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
6.67Single6FFIMMPEP6FFI-mGlu5-MMPEP
6.67Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
6.67Single6TPKRetosiban6TPK-OT-Retosiban
6.67Single6ZINSR486926ZIN-NTS1-SR48692
6.67Single7VODCariprazine7VOD-5-HT2A-Cariprazine
6.67Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
6.67Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
6.67Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
6.67Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
6.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.67Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
6.67Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
6.67Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
6.67Consensusvasop-oxy_offOrthosteric Ligandot_off
6.45Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
6.45Single6FFHFenobam6FFH-mGlu5-Fenobam
6.45Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
6.45Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.45Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
6.45Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
6.25Single4NTJAZD12834NTJ-P2Y12-AZD1283
6.25Single6HLPNetupitant6HLP-NK1-Netupitant
6.25Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
6.25Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.25Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
6.25Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
6.25Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.25Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.06Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.06Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.88Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.88Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.88Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.88Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.56Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
5.56Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
4.55Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.55Single6D35Cholesterol6D35-SMO-Cholesterol
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.55Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.55Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.55Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
4.55Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.55Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.55Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.55Single7XW7K1-707XW7-TSH-K1-70
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.55Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.55Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.55Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WVXNorrin8WVX-LGR4-Norrin
4.55Single8WVYNorrin8WVY-LGR4-Norrin
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.55Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9KHHNorrin9KHH-LGR4-Norrin
4.55Single9S37NB219S37-LGR4-NB21
4.55Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.35Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.17Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.17Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.17Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.00Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.00Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.00Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.00Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.85Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
3.85Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
3.85Single5L7DCholesterol5L7D-SMO-Cholesterol
3.85Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.85Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.70Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
3.70Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
3.57Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
3.57Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
3.57Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.45Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
3.45Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
3.45Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
3.45Single6TP4ACT-4622066TP4-OX1-ACT-462206
3.45Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.45Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
3.45Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.45Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
3.33Single4K5YCP-3763954K5Y-CRF1-CP-376395
3.33Single6C1QNDT95137276C1Q-C5a1-PMX53-NDT9513727
3.33Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
3.23Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
3.23Single8IYXYL-3658IYX-GPR34-YL-365
3.23Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.23Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
3.12Single4Z9GCP-3763954Z9G-CRF1-CP-376395
3.12Single8GTIBMK-C2058GTI-CRF1-BMK-C205
3.03Single8GTGBMK-I1528GTG-CRF1-BMK-I152
2.94Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
2.86Single8GTMBMK-C2038GTM-CRF1-BMK-C203
2.78Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
2.63Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.63Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.50Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.50Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.44Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.27Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
pac1_on_gp 8E3X-PAC1-PACAP27-Gs/β1/γ2
6M1H-PAC1-Maxadilan-Gs/β1/γ2
Net Summary
Imin 3.325
Number of Linked Nodes 856
Number of Links 1002
Number of Hubs 145
Number of Links mediated by Hubs 576
Number of Communities 24
Number of Nodes involved in Communities 184
Number of Links involved in Communities 263
Path Summary
Number Of Nodes in MetaPath 105
Number Of Links MetaPath 104
Number of Shortest Paths 1850876
Length Of Smallest Path 3
Average Path Length 36.5358
Length of Longest Path 75
Minimum Path Strength 0.755
Average Path Strength 6.66453
Maximum Path Strength 45.4067
Minimum Path Correlation 0.7
Average Path Correlation 0.991175
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.81818
Average % Of Corr. Nodes 45.4675
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 45.148
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
vip-pacap_on_gpvpac_on_gp
pac_on_gp



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