Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg Int. Strength Num Of Links Community ConSurf
1A:A:L37 8.4325419
2A:A:K46 4.2145199
3A:A:I184 4.774519
4A:A:E186 6.5675419
5A:A:F191 8.51254125
6A:A:L194 4.514124
7A:A:F196 8.4865127
8A:A:K197 8.8825416
9A:A:M198 4.4475407
10A:A:F199 10.446515
11A:A:Q204 4.30833619
12A:A:R208 6.3725419
13A:A:K210 7.275619
14A:A:W211 7.135619
15A:A:H213 6.17754138
16A:A:F215 9.38519
17A:A:F223 8.6075419
18A:A:Y230 4.85408
19A:A:L232 7.9554208
20A:A:F250 8.292519
21A:A:S252 4.6525417
22A:A:I253 5.6525418
23A:A:C254 4.6525415
24A:A:W258 7.876505
25A:A:F259 7.5875419
26A:A:L266 6.2275419
27A:A:F267 7.13254169
28A:A:I278 6.0154146
29A:A:L283 5.05754147
30A:A:Y287 11.024147
31A:A:Y296 4.4775404
32A:A:F307 5.17418
33A:A:Y320 6.4545157
34A:A:N331 9.4654168
35A:A:F336 5.7045128
36A:A:V342 4.46254157
37A:A:L353 4.77407
38A:A:F354 5.712505
39B:B:L7 4.1275408
40B:B:D27 5.5054238
41B:B:V40 4.6375483
42B:B:L51 10.235439
43B:B:H54 8.92333639
44B:B:Y59 8.666138
45B:B:W63 7.648537
46B:B:L70 6.3425435
47B:B:V71 4.164508
48B:B:S72 6.6125439
49B:B:L79 5.4254177
50B:B:I80 8.53538
51B:B:I81 5.28254267
52B:B:W82 10.3914739
53B:B:D83 7.6954258
54B:B:S84 5.825435
55B:B:K89 6.04333639
56B:B:H91 7.38254265
57B:B:I93 6.2825407
58B:B:L95 5.7465178
59B:B:W99 8.88428719
60B:B:Y105 5.55833606
61B:B:Y111 6.38544
62B:B:C114 4.065178
63B:B:L117 4.258519
64B:B:C121 4.615448
65B:B:I123 4.98546
66B:B:Y124 6.918506
67B:B:L126 5.66405
68B:B:E130 3.71254273
69B:B:H142 8.1225449
70B:B:Y145 5.11333918
71B:B:F151 6.175649
72B:B:L152 4.2463
73B:B:I157 4.6875447
74B:B:V158 4.8425465
75B:B:T159 5.484549
76B:B:D163 8.1475449
77B:B:T165 5.8625447
78B:B:C166 4.235468
79B:B:W169 8.908548
80B:B:I171 4.515446
81B:B:F180 7.8025467
82B:B:H183 7.04857769
83B:B:D186 5.088519
84B:B:V187 4.426569
85B:B:L190 5.7975405
86B:B:L192 4.63465
87B:B:R197 8.365425
88B:B:F199 5.846569
89B:B:S201 4.565469
90B:B:K209 11.0867666
91B:B:L210 7.39425
92B:B:W211 9.74167668
93B:B:Q220 9.495427
94B:B:F222 10.39428
95B:B:H225 6.04529
96B:B:I232 6.382528
97B:B:F235 4.86333696
98B:B:P236 5.6275497
99B:B:F241 7.11833626
100B:B:D247 8.5225429
101B:B:R251 8.1275428
102B:B:F253 9.465426
103B:B:D254 4.2275409
104B:B:R256 7.59499
105B:B:D258 10.6575427
106B:B:Q259 4.9475406
107B:B:Y264 18.185105
108B:B:F278 5.726597
109B:B:R283 8.68167689
110B:B:L284 5.7775485
111B:B:Y289 7.282867107
112B:B:V296 5.47585
113B:B:W297 18.61254108
114B:B:D298 8.9225489
115B:B:L300 5.4875486
116B:B:H311 8.17254119
117B:B:V315 4.454117
118B:B:M325 5.5625405
119B:B:W332 14.37836139
120B:B:K337 7.8165116
121B:B:W339 11.7085119
122G:G:Q18 4.064569
123G:G:D36 5.558595
124G:G:M38 4.0225484
125G:G:D48 8.66409
126G:G:P49 5.5175407
127G:G:N59 4.1325439
128G:G:F61 6.1475838
129R:R:N44 5.335409
130R:R:M55 3.755405
131R:R:I62 5.0075407
132R:R:Y64 6.17578
133R:R:D71 7.3145299
134R:R:F74 9.6557
135R:R:L78 8.7475408
136R:R:F80 10.33254316
137R:R:W91 11.2025319
138R:R:W95 9.0454324
139R:R:C98 9.1975409
140R:R:K99 9.23254327
141R:R:I107 3.7405
142R:R:I119 5.2479
143R:R:R123 8.38167679
144R:R:C126 5.3854228
145R:R:N135 3.475404
146R:R:R137 10.624227
147R:R:I169 5.5245181
148R:R:Y175 10.67754183
149R:R:F180 5.7565336
150R:R:R201 5.274555
151R:R:R205 6.702555
152R:R:F206 5.695456
153R:R:F210 7.032559
154R:R:P213 5.0975409
155R:R:I216 3.825406
156R:R:Y221 7.15857778
157R:R:K231 4.93254155
158R:R:M233 4.67754153
159R:R:L243 6.3175478
160R:R:F250 6.46409
161R:R:W254 5.816559
162R:R:F255 7.855456
163R:R:F257 5.07167657
164R:R:Q258 7.3175458
165R:R:F273 5.8925405
166R:R:F292 7.035457
167R:R:F293 5.24475
168R:R:N298 8.254299
169R:R:L301 4.708578
170R:R:Y302 6.6779
171R:R:F304 4.64254287
172R:R:F309 7.1775408
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Int. Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.

Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1B:B:D83 B:B:R68 16.137614.29YesNo085
2B:B:R68 B:B:Y85 15.705316.46NoNo054
3B:B:Y85 G:G:F61 13.6510.32NoYes048
4A:A:K345 R:R:M233 10.23534.32NoYes053
5A:A:F354 A:A:K345 24.52443.72YesNo055
6A:A:F354 R:R:K235 92.70938.69YesNo055
7A:A:D315 R:R:K235 93.12014.15NoNo035
8A:A:D315 A:A:T316 93.32615.78NoNo033
9A:A:K317 A:A:T316 94.1493NoNo073
10A:A:C254 A:A:K317 47.21854.85YesNo157
11A:A:C254 A:A:F250 47.56014.19YesYes159
12A:A:F223 A:A:F250 99.927617.15YesYes199
13A:A:F223 A:A:L249 49.98216.09YesNo199
14A:A:L249 A:A:R208 49.92793.64NoYes199
15A:A:R208 A:A:W211 1009YesYes199
16A:A:Q204 A:A:W211 43.85163.29YesYes199
17A:A:Q204 A:A:S206 21.45324.33YesNo198
18A:A:S206 B:B:D186 21.3875.89NoYes189
19B:B:D186 B:B:G185 64.29291.68YesNo095
20B:B:D205 B:B:G185 64.08351.68NoNo095
21B:B:D205 B:B:S207 63.66777.36NoNo095
22B:B:H183 B:B:S207 63.25474.18YesNo095
23B:B:H183 B:B:W211 50.68123.17YesYes698
24B:B:F199 B:B:W211 50.97989.02YesYes698
25B:B:F199 B:B:L192 49.44353.65YesYes695
26B:B:L192 B:B:R150 47.89324.86YesNo056
27B:B:H62 B:B:R150 47.74418.05NoNo066
28B:B:H62 B:B:Y105 47.31523.27NoYes066
29B:B:L69 B:B:Y105 17.8987.03NoYes056
30B:B:D83 B:B:L69 17.67464.07YesNo085
31A:A:I264 A:A:K317 47.13597.27NoNo167
32A:A:F250 A:A:I264 47.23035.02YesNo196
33A:A:F223 A:A:I253 49.9827.54YesYes198
34A:A:I253 A:A:R208 49.98196.26YesYes189
35A:A:Q204 B:B:Y145 22.24475.64YesYes198
36B:B:D186 B:B:Y145 43.24568.05YesYes198
37A:A:W211 B:B:L117 38.70823.42YesYes199
38B:B:L117 B:B:Y145 22.73293.52YesYes198
39R:R:R123 R:R:Y64 10.91427.2YesYes798
40A:A:L353 R:R:R123 65.27513.64YesYes079
41A:A:L348 A:A:L353 68.61265.54NoYes097
42A:A:F354 A:A:L348 68.82756.09YesNo059
43B:B:L117 B:B:W99 16.68743.42YesYes199
44A:A:N346 A:A:V342 13.83134.43NoYes047
45A:A:K345 A:A:N346 14.06455.6NoNo054
46A:A:F215 A:A:W211 17.08114.01YesYes199
47A:A:F215 B:B:W99 16.31812.03YesYes199
48B:B:Q75 B:B:Y59 32.384913.53NoYes098
49B:B:Q75 B:B:W99 32.52917.67NoYes099
50B:B:D290 B:B:R314 29.53421.44NoNo068
51B:B:C271 B:B:D290 29.26564.67NoNo056
52B:B:C271 B:B:D291 13.80679.34NoNo058
53B:B:D291 B:B:N293 13.664310.77NoNo085
54B:B:N293 B:B:V307 13.38774.43NoNo053
55B:B:G306 B:B:V307 14.27441.84NoNo043
56B:B:G306 B:B:V296 14.13061.84NoYes045
57B:B:R314 B:B:W332 29.58829.99NoYes089
58B:B:V71 B:B:Y105 26.81695.05YesYes086
59B:B:L79 B:B:V71 22.54284.47YesYes078
60B:B:C114 B:B:L79 21.12853.17YesYes1787
61B:B:C114 B:B:G115 20.49473.92YesNo089
62B:B:G115 B:B:L146 20.25693.42NoNo097
63B:B:L146 B:B:T159 18.0924.42NoYes079
64R:R:R123 R:R:Y302 52.35778.23YesYes799
65R:R:I116 R:R:Y302 49.482810.88NoYes089
66R:R:F250 R:R:I116 36.02788.79YesNo098
67R:R:F250 R:R:W254 28.51414.01YesYes099
68R:R:F257 R:R:W254 19.02784.01YesYes579
69R:R:F257 R:R:R205 17.23813.21YesYes575
70R:R:R201 R:R:R205 13.10117.46YesYes555
71R:R:I204 R:R:R201 10.17892.51NoYes045
72R:R:I116 R:R:N298 13.30968.5NoYes089
73R:R:F74 R:R:V105 13.01515.24YesNo076
74R:R:T77 R:R:V105 12.54797.93NoNo076
75R:R:I101 R:R:T77 10.31569.12NoNo057
76B:B:W332 B:B:Y59 30.399211.58YesYes1398
77B:B:C271 B:B:Y289 15.35544.03NoYes057
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1 Node2 LinkStrength Comm IsNode1Hub? IsNode2Hub? Node1Cons Node2Cons Node1Shell Node2Shell
L:L:?1 R:R:Y175 5.3 0 No Yes 0 3 0 1
L:L:?1 R:R:T177 6.66 0 No No 0 3 0 1
L:L:?1 R:R:R205 10.3 0 No Yes 0 5 0 1
R:R:D173 R:R:K90 15.21 18 No No 3 4 2 2
R:R:K90 R:R:Y175 11.94 18 No Yes 4 3 2 1
R:R:T177 R:R:V167 3.17 0 No No 3 1 1 2
R:R:D173 R:R:I169 9.8 18 No Yes 3 1 2 2
R:R:I169 R:R:Y175 3.63 18 Yes Yes 1 3 2 1
R:R:D173 R:R:Y175 21.84 18 No Yes 3 3 2 1
R:R:R201 R:R:R205 7.46 5 Yes Yes 5 5 2 1
R:R:F257 R:R:R205 3.21 5 Yes Yes 7 5 2 1
R:R:Q258 R:R:R205 7.01 5 Yes Yes 8 5 2 1
R:R:A261 R:R:R205 5.53 0 No Yes 5 5 2 1
R:R:F257 R:R:Q258 5.86 5 Yes Yes 7 8 2 2

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
42.86Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
42.86Single6ME5Agomelatine6ME5-MT1-Agomelatine
42.86Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
37.50Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
33.33Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
33.33Single6ME9Ramelteon6ME9-MT2-Ramelteon
33.33Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
33.33Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
30.00Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
30.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
30.00Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
30.00Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
30.00Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
28.57Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
28.57Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
27.27Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
27.27Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
27.27Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
27.27Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
25.00Single3OE6IT1t3OE6-CXCR4-IT1t
25.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
25.00Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
25.00Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
25.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
25.00Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
25.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
25.00Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
25.00Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
25.00Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.00Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
23.08Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
23.08Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
23.08Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
23.08Consensusrelaxin_onOrthosteric Ligandrxfp4_on
23.08Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
22.22Single3OE9IT1t3OE9-CXCR4-IT1t
22.22Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
22.22Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
22.22Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
22.22Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
22.22Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
22.22Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
22.22Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
22.22Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
22.22Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
22.22Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
22.22Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
22.22Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
22.22Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
22.22Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
22.22Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
22.22Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
22.22Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
22.22Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
22.22Consensusgq_nucleotideOrthosteric Ligandgq_p2y
22.22Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
21.43Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
21.43Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
21.43Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
21.43Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
21.43Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
21.43Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
21.43Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
21.43Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
21.43Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
21.43Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
20.00Single3ODUIT1t3ODU-CXCR4-IT1t
20.00Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
20.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
20.00Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
20.00Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
20.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
20.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
20.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
20.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
20.00Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
20.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
20.00Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
20.00Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
20.00Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
20.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
20.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
20.00Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
20.00Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
20.00Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
20.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
20.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
20.00Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
20.00Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
20.00Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
20.00Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
20.00Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
20.00Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
20.00Consensuschemerin_onOrthosteric Ligandcml1_on
20.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
20.00Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
20.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
20.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
20.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
18.75Single5WF6UK-4320975WF6-A2A-UK-432097
18.75Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
18.75Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
18.75Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
18.75Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
18.75Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
18.75Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
18.18Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
18.18Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
18.18Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
18.18Single6KUXRS-799486KUX-α2a-RS-79948
18.18Single6MH8ZM-2413856MH8-A2A-ZM-241385
18.18Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
18.18Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
18.18Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
18.18Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
18.18Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
18.18Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
18.18Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
18.18Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
18.18Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
18.18Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
18.18Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
18.18Single7UL3Famotidine7UL3-H2-Famotidine
18.18Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
18.18Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
18.18Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
18.18Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
18.18Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
18.18Single8IHKAcifran8IHK-HCA3-Acifran
18.18Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
18.18Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
18.18Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
18.18Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
18.18Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
18.18Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
18.18Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
18.18Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
18.18Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
18.18Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
18.18Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
18.18Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
18.18Consensushca_onOrthosteric Ligandhca2_on
18.18Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
17.65Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
17.65Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
17.65Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
17.65Single8IEIA1LYA8IEI-GPR156-A1LYA
17.65Single8IEPA1LYA8IEP-GPR156-A1LYA
17.65Single8IEPA1LYA8IEP-GPR156-A1LYA
17.65Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
17.65Single8WDTphotoNECA8WDT-A2A-photoNECA
17.65Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
17.65Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.65Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
17.65Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
17.65Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
17.65Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
17.65Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
17.65Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
16.67Single2Y02Carmoterol2Y02-β1-Carmoterol
16.67Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
16.67Single4QIMANTA XV4QIM-SMO-ANTA XV
16.67Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
16.67Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
16.67Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
16.67Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
16.67Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
16.67Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
16.67Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
16.67Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
16.67Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
16.67Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
16.67Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
16.67Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
16.67Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
16.67Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
16.67Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
16.67Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
16.67Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
16.67Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
16.67Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
16.67Single7V3ZCP559407V3Z-CB1-CP55940
16.67Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
16.67Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
16.67Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
16.67Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
16.67Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
16.67Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
16.67Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
16.67Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
16.67Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
16.67Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
16.67Single8IEBA1LYA8IEB-GPR156-A1LYA
16.67Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
16.67Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
16.67Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
16.67Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
16.67Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
16.67Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
16.67Single8T1WCVN4248T1W-GPR6-CVN424
16.67Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
16.67Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
16.67Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
16.67Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
16.67Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
16.67Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
16.67Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
16.67Single9CHXS-Carazolol9CHX-β2-S-Carazolol
16.67Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
16.67Single9IYAONO-97105319IYA-GPR55-ONO-9710531
16.67Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
16.67Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
16.67Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
16.67Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
16.67Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
16.67Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
16.67Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
16.67Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
16.67Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
16.67Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
16.67Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
16.67Consensushca_on_gpOrthosteric Ligandhca2_on_gp
16.67Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
16.67Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
16.67Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
15.79Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
15.79Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
15.79Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
15.79Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
15.79Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.79Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
15.79Consensusangiotensin_onOrthosteric Ligandat1_on
15.79Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
15.79Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
15.79Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
15.79Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
15.79Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
15.79Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
15.79Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
15.38Single4JKVTaladegib4JKV-SMO-Taladegib
15.38Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
15.38Single6D26Fevipiprant6D26-DP2-Fevipiprant
15.38Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
15.38Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
15.38Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
15.38Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
15.38Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
15.38Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
15.38Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
15.38Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
15.38Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
15.38Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
15.38Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
15.38Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
15.38Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
15.38Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
15.38Single8JXSPF-61428JXS-D1-PF-6142
15.38Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
15.38Single8TF5Oleic acid8TF5-GPR6-Oleic acid
15.38Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
15.38Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
15.38Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
15.38Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
15.38Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
15.38Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
15.38Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
15.38Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
15.38Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
15.38Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
15.38Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
15.38Consensusdp_offOrthosteric Liganddp2_off
15.38Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
15.38Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
15.38Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
15.38Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
15.38Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
15.38Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Consensustrace-amine_onOrthosteric Ligandta1_on
15.00Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
15.00Single6JODAngiotensin II6JOD-AT2-Angiotensin II
15.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
15.00Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
15.00Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
15.00Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
15.00Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
15.00Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
15.00Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.00Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
15.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
15.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
15.00Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
15.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
15.00Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
15.00Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
15.00Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
15.00Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
14.29Single2YDVNECA2YDV-A2A-NECA
14.29Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
14.29Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
14.29Single4UHRCGS216804UHR-A2A-CGS21680
14.29Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
14.29Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
14.29Single5G53NECA5G53-A2A-NECA-Gs
14.29Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
14.29Single5TZRMK86665TZR-FFA1-MK8666
14.29Single5V56TC1145V56-SMO-TC114
14.29Single5V57TC1145V57-SMO-TC114
14.29Single5XR8AM8415XR8-CB1-AM841
14.29Single5XRAAM115425XRA-CB1-AM11542
14.29Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
14.29Single6J21Aprepitant6J21-NK1-Aprepitant
14.29Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
14.29Single6OS1TRV0266OS1-AT1-TRV026
14.29Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
14.29Single6WGTLSD6WGT-5-HT2A-LSD
14.29Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
14.29Single7F1TMIP-1a7F1T-CCR5-MIP-1a
14.29Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
14.29Single7FEECP559407FEE-CB1-CP55940-ZCZ011
14.29Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
14.29Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
14.29Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
14.29Single7PX4PSB-21137PX4-A2A-PSB-2113
14.29Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
14.29Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
14.29Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
14.29Single7WC4Serotonin7WC4-5-HT2A-Serotonin
14.29Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
14.29Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
14.29Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
14.29Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
14.29Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
14.29Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
14.29Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
14.29Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
14.29Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
14.29Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
14.29Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
14.29Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
14.29Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
14.29Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
14.29Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
14.29Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
14.29Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
14.29Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
14.29Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
14.29Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
14.29Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
14.29Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
14.29Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
14.29Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
14.29Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
14.29Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
14.29Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
14.29Single8PWNTheophylline8PWN-A2A-Theophylline
14.29Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
14.29Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
14.29Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
14.29Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
14.29Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
14.29Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
14.29Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
14.29Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
14.29Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
14.29Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusa2_onOrthosteric Liganda2b_on
14.29Consensusa2_on_gpOrthosteric Liganda2b_on_gp
14.29Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.29Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.29Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
14.29Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
14.29Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
14.29Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
14.29Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
14.29Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
14.29Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
14.29Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
14.29Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
14.29Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
14.29Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
14.29Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
14.29Consensuslpa_onOrthosteric Ligandlpa1_on
14.29Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
14.29Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
13.64Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
13.64Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
13.64Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
13.64Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
13.64Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
13.64Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
13.64Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
13.64Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.64Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.64Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
13.33Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
13.33Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
13.33Single4AMIBucindolol4AMI-β1-Bucindolol
13.33Single4N4WSANT-14N4W-SMO-SANT-1
13.33Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
13.33Single4PY02MeSATP4PY0-P2Y12-2MeSATP
13.33Single4RWADIPP-NH24RWA-δ-DIPP-NH2
13.33Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
13.33Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
13.33Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
13.33Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
13.33Single6KQICP559406KQI-CB1-CP55940-Org27569
13.33Single6MXTSalmeterol6MXT-β2-Salmeterol
13.33Single6OS2TRV0266OS2-AT1-TRV026
13.33Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
13.33Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
13.33Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
13.33Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.33Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
13.33Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
13.33Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
13.33Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
13.33Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
13.33Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
13.33Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
13.33Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
13.33Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
13.33Single8JJLOlodaterol8JJL-β2-Olodaterol
13.33Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
13.33Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
13.33Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
13.33Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
13.33Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.33Single8XQJJN2418XQJ-Apelin-JN241
13.33Single8XWACXCL18XWA-CXCR2-CXCL1
13.33Single8XWMCXCL68XWM-CXCR2-CXCL6
13.33Single8XWSCXCL58XWS-CXCR2-CXCL5
13.33Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
13.33Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
13.33Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
13.33Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
13.33Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.33Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.33Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
13.33Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
13.33Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
13.33Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
13.33Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
13.33Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
13.33Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
13.33Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
13.33Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
13.33Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
13.33Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.33Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
13.33Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
13.33Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
13.33Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.33Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
13.33Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
13.33Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
13.33Consensuslpa_offOrthosteric Ligandlpa1_off
13.33Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
13.33Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.33Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
13.04Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
13.04Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
13.04Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
13.04Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
13.04Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
13.04Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
13.04Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
13.04Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
13.04Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
12.50Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
12.50Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
12.50Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
12.50Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
12.50Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
12.50Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
12.50Single6IBLArformoterol6IBL-β1-Arformoterol
12.50Single6IGLIRL16206IGL-ETB-IRL1620
12.50Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.50Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
12.50Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
12.50Single6TQ9SB-4081246TQ9-OX1-SB-408124
12.50Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
12.50Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
12.50Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
12.50Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
12.50Single7EZCUKA7EZC-A2A-UKA
12.50Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
12.50Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
12.50Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
12.50Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
12.50Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
12.50Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
12.50Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
12.50Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
12.50Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
12.50Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
12.50Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
12.50Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
12.50Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
12.50Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
12.50Single8A2OTheophylline8A2O-A2A-Theophylline-Na
12.50Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
12.50Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
12.50Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
12.50Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
12.50Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
12.50Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
12.50Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
12.50Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
12.50Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
12.50Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
12.50Single8IY6Endothelin-18IY6-ETB-Endothelin-1
12.50Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
12.50Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
12.50Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
12.50Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
12.50Single8XVUCXCL28XVU-CXCR2-CXCL2
12.50Single8XWFCXCL38XWF-CXCR2-CXCL3
12.50Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
12.50Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
12.50Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
12.50Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
12.50Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
12.50Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
12.50Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
12.50Consensusbradykinin_onOrthosteric Ligandbk2_on
12.50Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
12.50Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
12.50Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
12.50Consensuscck_onOrthosteric Ligandccka_on cckb_on
12.50Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
12.50Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
12.50Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
12.50Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
12.50Consensusendothelin_onOrthosteric Ligandetb_on eta_on
12.50Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
12.50Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
12.50Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
12.50Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
12.50Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
12.50Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
12.50Consensusp2y_offOrthosteric Ligandp2y1_off
12.50Consensusprostanoid_offOrthosteric Ligandep_off dp_off
12.50Consensussensory_onOrthosteric Ligandopsins_on
12.00Single5GLHEndothelin-15GLH-ETB-Endothelin-1
12.00Single6IGKEndothelin-36IGK-ETB-Endothelin-3
12.00Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
12.00Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
12.00Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
12.00Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
12.00Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
11.76Single3NY9ICI118-5513NY9-β2-ICI118-551
11.76Single4UG2CGS216804UG2-A2A-CGS21680
11.76Single5ZTYAM102575ZTY-CB2-AM10257
11.76Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
11.76Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
11.76Single6KNMJN241-96KNM-Apelin-JN241-9
11.76Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
11.76Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
11.76Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
11.76Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
11.76Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
11.76Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
11.76Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
11.76Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
11.76Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
11.76Single7XN9L-054,5227XN9-SST2-L-054,522
11.76Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
11.76Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
11.76Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
11.76Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
11.76Single8IEIA1LYA8IEI-GPR156-A1LYA
11.76Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
11.76Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
11.76Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
11.76Single8XQJJN2418XQJ-Apelin-JN241
11.76Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
11.76Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
11.76Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
11.76Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
11.76Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
11.76Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
11.76Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
11.76Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
11.76Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
11.76Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
11.76Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
11.76Consensuskisspeptin_onOrthosteric Ligandkiss1_on
11.76Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
11.76Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
11.76Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
11.76Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
11.54Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
11.54Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
11.54Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
11.54Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
11.11Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
11.11Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
11.11Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
11.11Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
11.11Single4IARErgotamine4IAR-5-HT1B-Ergotamine
11.11Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
11.11Single4XNWMRS25004XNW-P2Y1-MRS2500
11.11Single4XT1Fractalkine4XT1-US28-Fractalkine
11.11Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
11.11Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
11.11Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
11.11Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
11.11Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
11.11Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
11.11Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
11.11Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
11.11Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
11.11Single7F8XNN90567F8X-CCKA-NN9056
11.11Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
11.11Single7QA8Peptide7QA8-STE2-Peptide
11.11Single7QA8Peptide7QA8-STE2-Peptide
11.11Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
11.11Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
11.11Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
11.11Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
11.11Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single7WC5Psilocin7WC5-5-HT2A-Psilocin
11.11Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
11.11Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.11Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
11.11Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
11.11Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
11.11Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
11.11Single8IEBA1LYA8IEB-GPR156-A1LYA
11.11Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
11.11Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
11.11Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
11.11Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
11.11Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
11.11Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
11.11Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
11.11Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
11.11Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
11.11Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
11.11Single8XWNCXCL88XWN-CXCR2-CXCL8
11.11Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
11.11Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
11.11Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
11.11Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
11.11Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
11.11Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
11.11Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
11.11Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
11.11Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
11.11Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
11.11Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
11.11Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
11.11Consensuslpl_onOrthosteric Ligands1p_on lpa_on
11.11Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
11.11Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
11.11Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
11.11Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
11.11Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
11.11Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
11.11Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
11.11Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
10.71Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
10.53Single3QAKUK-4320973QAK-A2A-UK-432097
10.53Single6HLOAprepitant6HLO-NK1-Aprepitant
10.53Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
10.53Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
10.53Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
10.53Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
10.53Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
10.53Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
10.53Single7XNACYN1548067XNA-SST2-CYN154806
10.53Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
10.53Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
10.53Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
10.53Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
10.53Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
10.53Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
10.53Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
10.53Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
10.53Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
10.53Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
10.53Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
10.53Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
10.53Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
10.53Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
10.53Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
10.00Single3OE0CVX153OE0-CXCR4-CVX15
10.00Single3PBLEticlopride3PBL-D3-Eticlopride
10.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
10.00Single4O9RCyclopamine4O9R-SMO-Cyclopamine
10.00Single5L7IVismodegib5L7I-SMO-Vismodegib
10.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
10.00Single5WF5UK-4320975WF5-A2A-UK-432097
10.00Single6HLLCP999946HLL-NK1-CP99994
10.00Single6LI0C176LI0-GPR52-C17
10.00Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
10.00Single6TP4ACT-4622066TP4-OX1-ACT-462206
10.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
10.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
10.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
10.00Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
10.00Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
10.00Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
10.00Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
10.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
10.00Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
10.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
10.00Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
10.00Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.00Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
10.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
10.00Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
10.00Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
10.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
10.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
10.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
10.00Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
10.00Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
10.00Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
10.00Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
10.00Single8K5BNiacin8K5B-HCA2-Niacin
10.00Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
10.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
10.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
10.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
10.00Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
10.00Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
10.00Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
10.00Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
10.00Single9B9Y7DY9B9Y-CB1-7DY
10.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
10.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
10.00Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
10.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
10.00Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
10.00Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
10.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
10.00Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
10.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
10.00Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
10.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
10.00Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
9.52Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
9.52Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
9.52Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
9.52Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
9.52Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
9.52Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
9.52Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
9.52Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
9.52Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
9.52Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
9.52Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
9.52Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
9.52Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
9.52Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
9.52Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
9.52Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
9.52Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
9.52Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
9.52Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
9.52Consensusvasop-oxy_onOrthosteric Ligandv2_on
9.52Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
9.09Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
9.09Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
9.09Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
9.09Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
9.09Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
9.09Single3PWHZM-2413853PWH-A2A-ZM-241385
9.09Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
9.09Single4BWBNeurotensin4BWB-NTS1-Neurotensin
9.09Single4QINSAG1.54QIN-SMO-SAG1.5
9.09Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
9.09Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
9.09Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
9.09Single5U09Taranabant5U09-CB1-Taranabant
9.09Single5WS3EMPA5WS3-OX2-EMPA
9.09Single6AKXA4R6AKX-CCR5-A4R
9.09Single6AKYMaraviroc6AKY-CCR5-Maraviroc
9.09Single6B73MP11046B73-κ-MP1104
9.09Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
9.09Single6DS0Ly2660976DS0-5-HT2B-Ly266097
9.09Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
9.09Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
9.09Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
9.09Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
9.09Single6TODEMPA6TOD-OX1-EMPA-Na
9.09Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
9.09Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
9.09Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
9.09Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
9.09Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
9.09Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
9.09Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
9.09Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
9.09Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
9.09Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
9.09Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
9.09Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
9.09Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
9.09Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
9.09Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
9.09Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
9.09Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
9.09Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
9.09Single7XRRLemborexant7XRR-OX2-Lemborexant
9.09Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
9.09Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
9.09Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
9.09Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
9.09Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
9.09Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
9.09Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
9.09Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
9.09Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
9.09Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
9.09Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
9.09Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
9.09Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
9.09Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
9.09Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
9.09Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
9.09Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
9.09Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
9.09Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
9.09Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
9.09Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
9.09Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
9.09Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
9.09Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
9.09Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
9.09Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
9.09Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
9.09Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
9.09Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
9.09Single8ZRTET-18ZRT-ETB-ET-1
9.09Single9BA0A1AKN9BA0-CB1-A1AKN
9.09Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
9.09Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
9.09Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
9.09Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
9.09Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
9.09Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
9.09Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
9.09Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
9.09Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
9.09Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
9.09Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
9.09Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
9.09Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
9.09Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
9.09Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
9.09Consensusorexin_offOrthosteric Ligandox2_off ox1_off
9.09Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
9.09Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
9.09Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
9.09Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
9.09Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
8.70Single4XT3Fractalkine4XT3-US28-Fractalkine
8.70Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
8.70Single6FJ3PTH6FJ3-PTH1-PTH
8.70Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
8.70Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
8.70Single7SK3CXCL127SK3-ACKR3-CXCL12
8.70Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
8.70Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
8.70Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
8.70Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
8.70Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
8.70Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
8.33Single2YDOAdenosine2YDO-A2A-Adenosine
8.33Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
8.33Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
8.33Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
8.33Single4MBSMaraviroc4MBS-CCR5-Maraviroc
8.33Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
8.33Single4ZJCSB-6740424ZJC-OX1-SB-674042
8.33Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
8.33Single5IU7Q274563465IU7-A2A-Q27456346-Na
8.33Single5IUBQ274563445IUB-A2A-Q27456344-Na
8.33Single5JTBZM-2413855JTB-A2A-ZM-241385
8.33Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
8.33Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
8.33Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
8.33Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
8.33Single5UVIZM-2413855UVI-A2A-ZM-241385
8.33Single6A94Zotepine6A94-5-HT2A-Zotepine
8.33Single6AQFZM-2413856AQF-A2A-ZM-241385
8.33Single6PS0S-Carazolol6PS0-β2-S-Carazolol
8.33Single6PS4ICI118-5516PS4-β2-ICI118-551
8.33Single6PS5S-Propranolol6PS5-β2-S-Propranolol
8.33Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
8.33Single6TPGEMPA6TPG-OX2-EMPA
8.33Single6TPNHTL66416TPN-OX2-HTL6641
8.33Single6VI4JDTic6VI4-κ-JDTic
8.33Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
8.33Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
8.33Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
8.33Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
8.33Single7AROLUF58337ARO-A2A-LUF5833-Na
8.33Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
8.33Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
8.33Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
8.33Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
8.33Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
8.33Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
8.33Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
8.33Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
8.33Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
8.33Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
8.33Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.33Single7T32ZM-2413857T32-A2A-ZM-241385
8.33Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
8.33Single7VODCariprazine7VOD-5-HT2A-Cariprazine
8.33Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
8.33Single7VV6C48/807VV6-MRGPRX2-C48/80
8.33Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
8.33Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
8.33Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
8.33Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
8.33Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
8.33Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
8.33Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
8.33Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
8.33Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
8.33Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
8.33Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
8.33Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
8.33Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
8.33Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
8.33Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
8.33Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
8.33Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
8.33Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
8.33Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
8.33Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
8.33Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
8.33Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.33Single8K5CAcipimox8K5C-HCA2-Acipimox
8.33Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
8.33Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
8.33Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
8.33Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
8.33Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
8.33Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
8.33Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
8.33Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
8.33Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
8.33Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
8.33Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
8.33Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
8.33Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
8.33Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
8.33Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
8.33Single9BJKNaloxone9BJK-μ-Naloxone-NAM
8.33Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
8.33Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
8.33Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
8.33Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
8.33Consensusa2_offOrthosteric Liganda2a_off
8.33Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
8.33Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
8.33Consensusalpha1_onOrthosteric Ligandalpha1a_on
8.33Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
8.33Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
8.33Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
8.33Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
8.33Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
8.33Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
8.33Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
8.33Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
8.33Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
8.33Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
8.33Consensusopsins_offOrthosteric Ligandrhodopsin_off
8.33Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
8.33Consensussensory_offOrthosteric Ligandopsins_off
8.00Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
8.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
8.00Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
8.00Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
8.00Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
8.00Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
8.00Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
7.69Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
7.69Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
7.69Single2Y01Dobutamine2Y01-β1-Dobutamine
7.69Single2Y04Salbutamol2Y04-β1-Salbutamol
7.69Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
7.69Single3EMLZM-2413853EML-A2A-ZM-241385
7.69Single3NY8ICI118-5513NY8-β2-ICI118-551
7.69Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
7.69Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
7.69Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
7.69Single4EJ4Naltrindole4EJ4-δ-Naltrindole
7.69Single4GBRS-Carazolol4GBR-β2-S-Carazolol
7.69Single4QKX35V4QKX-β2-35V
7.69Single5IU8Q274563475IU8-A2A-Q27456347-Na
7.69Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
7.69Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
7.69Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
7.69Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
7.69Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
7.69Single5T04Neurotensin5T04-NTS1-Neurotensin
7.69Single5TGZAM65385TGZ-CB1-AM6538
7.69Single5UENDU1725UEN-A1-DU172
7.69Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
7.69Single6D27CAY104716D27-DP2-CAY10471
7.69Single6DRXLisuride6DRX-5-HT2B-Lisuride
7.69Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
7.69Single6H7MSalbutamol6H7M-β1-Salbutamol
7.69Single6IIVDaltroban6IIV-TP-Daltroban
7.69Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
7.69Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
7.69Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
7.69Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
7.69Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
7.69Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
7.69Single6S0LZM-2413856S0L-A2A-ZM-241385
7.69Single6TOTLemborexant6TOT-OX1-Lemborexant
7.69Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
7.69Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
7.69Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
7.69Single7BU7BI1671077BU7-β1-BI167107
7.69Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
7.69Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
7.69Single7PYRPSB-21157PYR-A2A-PSB-2115
7.69Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
7.69Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
7.69Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
7.69Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
7.69Single7UL4Alvimopan7UL4-μ-Alvimopan
7.69Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
7.69Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
7.69Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
7.69Single7WC7Lisuride7WC7-5-HT2A-Lisuride
7.69Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
7.69Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
7.69Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
7.69Single8CU6LJ-45178CU6-A2A-LJ-4517
7.69Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
7.69Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
7.69Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
7.69Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
7.69Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
7.69Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
7.69Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
7.69Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
7.69Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
7.69Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
7.69Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
7.69Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
7.69Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
7.69Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
7.69Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
7.69Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
7.69Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
7.69Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
7.69Single8JXRLSD8JXR-D1-LSD
7.69Single8K5DGSK2560738K5D-HCA2-GSK256073
7.69Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
7.69Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
7.69Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
7.69Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
7.69Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
7.69Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
7.69Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
7.69Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
7.69Single8X64Desloratadine8X64-H1-Desloratadine
7.69Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
7.69Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
7.69Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
7.69Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
7.69Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
7.69Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
7.69Single9B9ZA1AKO9B9Z-CB1-A1AKO
7.69Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
7.69Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
7.69Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
7.69Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
7.69Consensus5ht5_onOrthosteric Ligand5ht5a_on
7.69Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
7.69Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
7.69Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
7.69Consensusa3_onOrthosteric Liganda3a_on
7.69Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
7.69Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
7.69Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
7.69Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
7.69Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
7.69Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
7.69Consensusblt_onOrthosteric Ligandblt1_on
7.69Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
7.69Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
7.69Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
7.69Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
7.69Consensusdopamine_offOrthosteric Ligandd2_off d3_off
7.69Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
7.69Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
7.69Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
7.69Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
7.69Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
7.69Consensusleukotriene_onOrthosteric Ligandblt_on
7.69Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
7.69Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
7.69Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
7.41Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
7.41Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
7.41Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
7.14Single2RH1S-Carazolol2RH1-β2-S-Carazolol
7.14Single2Y00Dobutamine2Y00-β1-Dobutamine
7.14Single2Y03Isoprenaline2Y03-β1-Isoprenaline
7.14Single2YCWS-Carazolol2YCW-β1-S-Carazolol
7.14Single4NTJAZD12834NTJ-P2Y12-AZD1283
7.14Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
7.14Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
7.14Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
7.14Single5C1MBU725C1M-μ-BU72
7.14Single5D6LS-Carazolol5D6L-β2-S-Carazolol
7.14Single5IUAQ274563485IUA-A2A-Q27456348-Na
7.14Single5JQHS-Carazolol5JQH-β2-S-Carazolol
7.14Single5N2RPSB-365N2R-A2A-PSB-36-Na
7.14Single5N2SPSB365N2S-A1-PSB36
7.14Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
7.14Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
7.14Single5TVNLSD5TVN-5-HT2B-LSD
7.14Single5WIUNemonapride5WIU-D4-Nemonapride
7.14Single5WIVNemonapride5WIV-D4-Nemonapride-Na
7.14Single5WQCEMPA5WQC-OX2-EMPA
7.14Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
7.14Single5XPRBosentan5XPR-ETB-Bosentan
7.14Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
7.14Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
7.14Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
7.14Single6E67BI1671076E67-β2-BI167107-Gs (fused)
7.14Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
7.14Single6HLPNetupitant6HLP-NK1-Netupitant
7.14Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
7.14Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
7.14Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
7.14Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
7.14Single6S0QZM-2413856S0Q-A2A-ZM-241385
7.14Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
7.14Single6TP6Filorexant6TP6-OX1-Filorexant
7.14Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
7.14Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
7.14Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
7.14Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
7.14Single7C61Ergotamine7C61-5-HT1B-Ergotamine
7.14Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
7.14Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
7.14Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
7.14Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
7.14Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
7.14Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
7.14Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
7.14Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
7.14Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
7.14Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
7.14Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
7.14Single7W41PD1762527W41-BB2-PD176252
7.14Single7WC6LSD7WC6-5-HT2A-LSD
7.14Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
7.14Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
7.14Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
7.14Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
7.14Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
7.14Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
7.14Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
7.14Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
7.14Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
7.14Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.14Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.14Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.14Single8GNEKW-63568GNE-A2A-KW-6356-Na
7.14Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
7.14Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
7.14Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
7.14Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
7.14Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
7.14Single8QOTNanobody-E8QOT-μ-Nanobody-E
7.14Single8S4DCMF-0198S4D-Apelin-CMF-019
7.14Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
7.14Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
7.14Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
7.14Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.14Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.14Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
7.14Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
7.14Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
7.14Single8ZMFA1L108ZMF-5-HT2C-A1L10
7.14Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.14Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.14Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
7.14Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
7.14Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
7.14Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
7.14Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
7.14Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
7.14Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
7.14Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
7.14Consensusa3_on_gpOrthosteric Liganda3a_on_gp
7.14Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
7.14Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
7.14Consensusadenosine_offOrthosteric Liganda1_off a2_off
7.14Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
7.14Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
7.14Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
7.14Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
7.14Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
7.14Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
7.14Consensusamine_offonOrthosteric Ligandamine_off amine_on
7.14Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
7.14Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
7.14Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
7.14Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
7.14Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
7.14Consensusbombesin_offOrthosteric Ligandbb2_off
7.14Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
7.14Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
7.14Consensusep_offOrthosteric Ligandep4_off
7.14Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
7.14Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
7.14Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
7.14Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
7.14Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
7.14Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
7.14Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
6.67Single3P0GBI1671073P0G-β2-BI167107
6.67Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
6.67Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
6.67Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
6.67Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
6.67Single4BV0Neurotensin4BV0-NTS1-Neurotensin
6.67Single4DJHJDTic4DJH-κ-JDTic
6.67Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
6.67Single4U15Tiotropium4U15-M3-Tiotropium
6.67Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
6.67Single5D5AS-Carazolol5D5A-β2-S-Carazolol
6.67Single5D5BS-Carazolol5D5B-β2-S-Carazolol
6.67Single5V54Methiothepin5V54-5-HT1B-Methiothepin
6.67Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
6.67Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
6.67Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
6.67Single6H7JIsoprenaline6H7J-β1-Isoprenaline
6.67Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
6.67Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
6.67Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
6.67Single6OL9Tiotropium6OL9-M5-Tiotropium
6.67Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
6.67Single7B6WCyclazosin7B6W-α1b-Cyclazosin
6.67Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
6.67Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
6.67Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
6.67Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
6.67Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
6.67Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
6.67Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
6.67Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
6.67Single7R0CAVP7R0C-V2-AVP-Arrestin2
6.67Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
6.67Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
6.67Single7TUYGSK682753A7TUY-GPR183-GSK682753A
6.67Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
6.67Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
6.67Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
6.67Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
6.67Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
6.67Single8E0GBU728E0G-μ-BU72
6.67Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
6.67Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
6.67Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
6.67Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
6.67Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
6.67Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
6.67Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
6.67Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
6.67Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
6.67Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
6.67Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
6.67Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
6.67Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
6.67Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
6.67Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
6.67Single8XVLZibotentan8XVL-ETA-Zibotentan
6.67Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
6.67Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
6.67Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
6.67Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
6.67Consensus5ht1_offOrthosteric Ligand5ht1b_off
6.67Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
6.67Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
6.67Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
6.67Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
6.67Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
6.67Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
6.67Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
6.67Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
6.67Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
6.67Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
6.67Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
6.67Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
6.67Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
6.67Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
6.67Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
6.67Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
6.67Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
6.67Consensusneurotensin_onOrthosteric Ligandnts1_on
6.67Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
6.67Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
6.67Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
6.67Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
6.67Consensustachykinin_offOrthosteric Ligandnk1_off
6.45Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
6.45Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
6.25Single3D4STimolol3D4S-β2-Timolol
6.25Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
6.25Single4LDEBI1671074LDE-β2-BI167107
6.25Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
6.25Single4XEENeurotensin4XEE-NTS1-Neurotensin
6.25Single4XESNeurotensin4XES-NTS1-Neurotensin
6.25Single5CXVTiotropium5CXV-M1-Tiotropium
6.25Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
6.25Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
6.25Single6A93Risperidone6A93-5-HT2A-Risperidone
6.25Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
6.25Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
6.25Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
6.25Single6IIURamatroban6IIU-TP-Ramatroban
6.25Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
6.25Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
6.25Single6YVRNTS8-136YVR-NTS1-NTS8-13
6.25Single7DFPSpiperone7DFP-D2-Spiperone
6.25Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
6.25Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
6.25Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
6.25Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
6.25Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
6.25Single7K15MKD0467K15-BLT1-MKD046-Na
6.25Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
6.25Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
6.25Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
6.25Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
6.25Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
6.25Single7YITNalfurafine7YIT-κ-Nalfurafine
6.25Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
6.25Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
6.25Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
6.25Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
6.25Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
6.25Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
6.25Single8JJ8Formoterol8JJ8-β2-Formoterol
6.25Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
6.25Single8JWY2-1188JWY-A2A-2-118
6.25Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
6.25Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
6.25Single8XYIVUF106618XYI-CXCR3-VUF10661
6.25Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
6.25Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
6.25Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
6.25Consensusalpha1_offOrthosteric Ligandalpha1a_off
6.25Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
6.25Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
6.25Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
6.25Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
6.25Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
6.25Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
6.25Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
6.25Consensuslpl_offOrthosteric Ligands1p_off lpa_off
6.25Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
6.25Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
6.25Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
6.25Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
6.25Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
6.25Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
6.25Consensusorexin_onOrthosteric Ligandox2_on
6.25Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
6.25Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
5.88Single4BUONeurotensin4BUO-NTS1-Neurotensin
5.88Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
5.88Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
5.88Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
5.88Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
5.88Single5X93K-87945X93-ETB-K-8794
5.88Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
5.88Single6H7LDobutamine6H7L-β1-Dobutamine
5.88Single6K1QIRL25006K1Q-ETB-IRL2500
5.88Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
5.88Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
5.88Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
5.88Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
5.88Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.88Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
5.88Single7UM4AS26747237UM4-5-HT5A-AS2674723
5.88Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
5.88Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
5.88Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
5.88Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
5.88Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8XVJMacitentan8XVJ-ETA-Macitentan
5.88Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
5.88Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
5.88Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
5.88Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
5.88Consensusendothelin_offOrthosteric Ligandetb_off
5.88Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
5.88Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
5.88Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
5.88Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
5.88Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
5.88Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
5.88Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single5EE7MK08935EE7-Glucagon-MK0893
5.56Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
5.56Single6PT3DPI-2876PT3-δ-DPI-287
5.56Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
5.56Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
5.56Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single7SK9CCX6627SK9-ACKR3-CCX662
5.56Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
5.56Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
5.56Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
5.56Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
5.56Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single8QJ2pN1628QJ2-MC4-pN162-Gs
5.56Single8X5YAstemizole8X5Y-H1-Astemizole
5.56Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
5.56Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
5.56Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
5.41Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
5.26Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
5.26Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
5.26Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
5.26Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
5.26Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
5.26Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
5.26Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
5.26Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
5.26Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.26Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
5.26Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
5.26Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
5.26Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
5.26Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
5.26Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
5.26Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
5.26Consensussomatostatin_offOrthosteric Ligandsst2_off
5.00Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
5.00Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
5.00Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
5.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
5.00Single7SK5CXCL127SK5-ACKR3-CXCL12
5.00Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
5.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
5.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
5.00Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
5.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
5.00Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
5.00Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
4.76Single6PT2KGCHM076PT2-δ-KGCHM07
4.76Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
4.76Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
4.76Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
4.76Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
4.76Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
4.76Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
4.76Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
4.76Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
4.55Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
4.55Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
4.55Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
4.55Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
4.55Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
4.55Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
4.55Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
4.55Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
4.55Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
4.55Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
4.55Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
4.55Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
4.55Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.55Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
4.55Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
4.55Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
4.55Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
4.35Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
4.35Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
4.35Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
4.35Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
4.35Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
4.35Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
4.35Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
4.35Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
4.35Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
4.35Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
4.35Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
4.35Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
4.35Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
4.35Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
4.17Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
4.17Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
4.17Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
4.17Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
4.17Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
4.17Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
4.17Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
4.17Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
4.17Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
4.17Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
4.17Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
4.17Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
4.00Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
4.00Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
4.00Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
4.00Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
4.00Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
4.00Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
4.00Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
4.00Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
4.00Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
4.00Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
4.00Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
4.00Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
4.00Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
4.00Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
4.00Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
3.85Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
3.85Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
3.85Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
3.85Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
3.85Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
3.85Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
3.85Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
3.85Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
3.85Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
3.85Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
3.85Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
3.85Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
3.85Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
3.85Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
3.70Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
3.70Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
3.70Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
3.70Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
3.70Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
3.70Consensusbombesin_onOrthosteric Ligandbb2_on
3.70Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
3.70Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
3.57Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
3.57Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
3.57Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
3.57Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
3.57Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
3.57Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
3.45Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
3.45Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
3.45Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
3.45Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
3.45Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
3.45Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.33Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
3.33Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
3.33Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
3.33Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
3.33Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
3.33Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
3.33Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.23Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
2.94Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
2.86Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3

PDB Summary
PDB 8Y63
Class A
SubFamily Peptide
Type Formylpeptide
SubType FPR2-ALX
Species Homo Sapiens
Ligand C20:0 Ceramide
Other Ligand(s) -
Protein Partners Gi1/Beta1/Gamma2
PDB Resolution 3.2
Date 2025-02-05
D.O.I. To be published
Net Summary
Imin 3
Number of Linked Nodes 843
Number of Links 1038
Number of Hubs 172
Number of Links mediated by Hubs 618
Number of Communities 34
Number of Nodes involved in Communities 264
Number of Links involved in Communities 373
Path Summary
Number Of Nodes in MetaPath 78
Number Of Links MetaPath 77
Number of Shortest Paths 2924450
Length Of Smallest Path 3
Average Path Length 35.0644
Length of Longest Path 66
Minimum Path Strength 1.315
Average Path Strength 6.7726
Maximum Path Strength 34.25
Minimum Path Correlation 0.7
Average Path Correlation 0.988112
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.94118
Average % Of Corr. Nodes 36.7582
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 51.8853
Maximum Path Hubs % 100
AnnotationTypeLinks
Gene OntologyMolecular Function• molecular transducer activity   • signaling receptor activity   • amide binding   • amyloid-beta binding   • binding   • peptide binding   • G protein-coupled receptor activity   • transmembrane signaling receptor activity   • complement receptor activity   • immune receptor activity   • cargo receptor activity   • protein binding   • signaling receptor binding   • scavenger receptor binding   • peptide receptor activity   • N-formyl peptide receptor activity   • G protein-coupled peptide receptor activity   • positive regulation of cytosolic calcium ion concentration   • biological regulation   • regulation of biological quality   • regulation of biological process   • regulation of cellular process   • reactive oxygen species metabolic process   • positive regulation of biological process   • regulation of superoxide metabolic process   • positive regulation of reactive oxygen species metabolic process   • superoxide metabolic process   • positive regulation of metabolic process   • superoxide anion generation   • metabolic process   • cellular process
Gene OntologyBiological Process• positive regulation of cytosolic calcium ion concentration   • biological regulation   • regulation of biological quality   • regulation of biological process   • regulation of cellular process   • reactive oxygen species metabolic process   • positive regulation of biological process   • regulation of superoxide metabolic process   • positive regulation of reactive oxygen species metabolic process   • superoxide metabolic process   • positive regulation of metabolic process   • superoxide anion generation   • metabolic process   • cellular process   • positive regulation of superoxide anion generation   • regulation of superoxide anion generation   • regulation of metabolic process   • regulation of reactive oxygen species metabolic process   • positive regulation of cellular process   • cellular response to stimulus   • positive regulation of cell communication   • positive regulation of signal transduction   • response to stimulus   • signaling   • regulation of signal transduction   • intracellular signal transduction   • cell communication   • positive regulation of response to stimulus   • positive regulation of ERK1 and ERK2 cascade   • regulation of intracellular signal transduction   • intracellular signaling cassette   • signal transduction   • regulation of signaling   • positive regulation of MAPK cascade   • positive regulation of intracellular signal transduction   • regulation of MAPK cascade   • regulation of response to stimulus   • MAPK cascade   • regulation of cell communication   • ERK1 and ERK2 cascade   • regulation of ERK1 and ERK2 cascade   • positive regulation of signaling   • immune response-regulating cell surface receptor signaling pathway   • complement receptor mediated signaling pathway   • immune response-activating signaling pathway   • immune response-regulating signaling pathway   • positive regulation of immune response   • regulation of immune system process   • positive regulation of immune system process   • cell surface receptor signaling pathway   • immune response-activating cell surface receptor signaling pathway   • immune response   • immune system process   • regulation of immune response   • activation of immune response   • regulation of defense response   • regulation of response to external stimulus   • negative regulation of inflammatory response   • defense response   • negative regulation of response to stimulus   • negative regulation of biological process   • response to external stimulus   • regulation of inflammatory response   • response to stress   • negative regulation of response to external stimulus   • regulation of response to stress   • negative regulation of defense response   • inflammatory response   • positive chemotaxis   • chemotaxis   • taxis   • response to chemical   • locomotion   • regulation of localization   • import into cell   • positive regulation of cellular component organization   • regulation of cellular component organization   • transport   • vesicle-mediated transport   • cellular component organization   • localization   • positive regulation of endocytosis   • phagocytosis   • cellular component organization or biogenesis   • regulation of endocytosis   • regulation of transport   • regulation of phagocytosis   • regulation of vesicle-mediated transport   • establishment of localization   • positive regulation of phagocytosis   • positive regulation of transport   • endocytosis   • regulation of phosphatidylinositol 3-kinase/protein kinase B signal transduction   • positive regulation of phosphatidylinositol 3-kinase/protein kinase B signal transduction   • phosphatidylinositol 3-kinase/protein kinase B signal transduction   • calcium-mediated signaling   • biological process involved in interspecies interaction between organisms   • response to other organism   • response to biotic stimulus   • defense response to bacterium   • defense response to other organism   • response to bacterium   • response to external biotic stimulus   • multicellular organismal process   • cellular developmental process   • astrocyte differentiation   • cell development   • astrocyte activation   • glial cell development   • multicellular organism development   • neurogenesis   • astrocyte development   • gliogenesis   • cell differentiation   • anatomical structure development   • system development   • developmental process   • cell activation   • nervous system development   • central nervous system development   • glial cell differentiation   • glial cell activation   • neuroinflammatory response   • positive regulation of monocyte chemotaxis   • positive regulation of locomotion   • regulation of cell motility   • positive regulation of chemotaxis   • positive regulation of cell migration   • regulation of monocyte chemotaxis   • positive regulation of response to external stimulus   • positive regulation of cell motility   • regulation of cell migration   • myeloid leukocyte migration   • positive regulation of mononuclear cell migration   • cell migration   • cell motility   • regulation of mononuclear cell migration   • cell chemotaxis   • regulation of leukocyte chemotaxis   • regulation of leukocyte migration   • positive regulation of leukocyte migration   • positive regulation of leukocyte chemotaxis   • regulation of chemotaxis   • monocyte chemotaxis   • leukocyte migration   • cellular response to chemical stimulus   • regulation of locomotion   • mononuclear cell migration   • leukocyte chemotaxis   • phospholipase C-activating G protein-coupled receptor signaling pathway   • G protein-coupled receptor signaling pathway   • cell adhesion   • adenylate cyclase-inhibiting G protein-coupled receptor signaling pathway   • adenylate cyclase-modulating G protein-coupled receptor signaling pathway   • positive regulation of response to biotic stimulus   • regulation of response to biotic stimulus   • innate immune response   • positive regulation of innate immune response   • regulation of innate immune response   • defense response to symbiont   • positive regulation of defense response   • cellular response to nitrogen compound   • response to oxygen-containing compound   • response to nitrogen compound   • cellular response to amyloid-beta   • cellular response to oxygen-containing compound   • response to amyloid-beta   • myeloid leukocyte activation   • leukocyte activation   • macrophage activation   • leukocyte activation involved in inflammatory response   • microglial cell activation   • receptor-mediated endocytosis   • membrane-bounded organelle   • intracellular anatomical structure   • tertiary granule membrane   • membrane   • intracellular vesicle   • intracellular membrane-bounded organelle   • endomembrane system   • tertiary granule   • intracellular organelle   • cytoplasmic vesicle membrane   • cellular anatomical structure   • bounding membrane of organelle   • vesicle membrane   • cytoplasmic vesicle
Gene OntologyCellular Component• membrane-bounded organelle   • intracellular anatomical structure   • tertiary granule membrane   • membrane   • intracellular vesicle   • intracellular membrane-bounded organelle   • endomembrane system   • tertiary granule   • intracellular organelle   • cytoplasmic vesicle membrane   • cellular anatomical structure   • bounding membrane of organelle   • vesicle membrane   • cytoplasmic vesicle   • organelle   • secretory granule   • secretory vesicle   • cytoplasm   • vesicle   • organelle membrane   • secretory granule membrane   • specific granule membrane   • specific granule   • cell periphery   • plasma membrane   • ficolin-1-rich granule membrane   • ficolin-1-rich granule   • D2 dopamine receptor binding   • protein binding   • binding   • signaling receptor binding   • G protein-coupled receptor binding   • dopamine receptor binding   • phosphorus-oxygen lyase activity   • enzyme regulator activity   • cyclase regulator activity   • molecular function regulator activity   • cyclase activity   • adenylate cyclase regulator activity   • lyase activity   • catalytic activity   • adenylate cyclase activity   • guanyl nucleotide binding   • GTP binding   • nucleotide binding   • guanyl ribonucleotide binding   • purine ribonucleotide binding   • purine ribonucleoside triphosphate binding   • nucleoside phosphate binding   • ion binding   • purine nucleotide binding   • anion binding   • heterocyclic compound binding   • carbohydrate derivative binding   • ribonucleotide binding   • small molecule binding   • cation binding   • magnesium ion binding   • metal ion binding   • GDP binding   • G protein-coupled serotonin receptor binding   • protein-containing complex binding   • G-protein beta/gamma-subunit complex binding   • pyrophosphatase activity   • GTPase activity   • G protein activity   • ribonucleoside triphosphate phosphatase activity   • hydrolase activity, acting on acid anhydrides, in phosphorus-containing anhydrides   • hydrolase activity   • hydrolase activity, acting on acid anhydrides   • cellular response to stimulus   • regulation of biological process   • regulation of cellular process   • response to stimulus   • signaling   • biological regulation   • adenylate cyclase-inhibiting serotonin receptor signaling pathway   • G protein-coupled serotonin receptor signaling pathway   • cell communication   • adenylate cyclase-inhibiting G protein-coupled receptor signaling pathway   • adenylate cyclase-modulating G protein-coupled receptor signaling pathway   • G protein-coupled receptor signaling pathway   • cellular process   • signal transduction   • response to hormone   • response to chemical   • response to endogenous stimulus   • response to peptide hormone   • response to oxygen-containing compound   • response to nitrogen compound   • cell division   • leukocyte migration   • immune system process   • mononuclear cell migration   • lymphocyte migration   • cell migration   • T cell migration   • cell motility   • regulation of steroid biosynthetic process   • regulation of cholesterol biosynthetic process   • regulation of cholesterol metabolic process   • steroid metabolic process   • regulation of lipid metabolic process   • sterol metabolic process   • positive regulation of biological process   • cholesterol metabolic process   • lipid biosynthetic process   • alcohol metabolic process   • regulation of primary metabolic process   • positive regulation of metabolic process   • regulation of small molecule metabolic process   • positive regulation of biosynthetic process   • positive regulation of lipid metabolic process   • small molecule metabolic process   • steroid biosynthetic process   • positive regulation of cellular process   • regulation of biosynthetic process   • secondary alcohol biosynthetic process   • regulation of alcohol biosynthetic process   • small molecule biosynthetic process   • regulation of steroid metabolic process   • cholesterol biosynthetic process   • positive regulation of cholesterol biosynthetic process   • primary metabolic process   • secondary alcohol metabolic process   • positive regulation of steroid biosynthetic process   • biosynthetic process   • sterol biosynthetic process   • positive regulation of lipid biosynthetic process   • regulation of sterol biosynthetic process   • alcohol biosynthetic process   • positive regulation of cholesterol metabolic process   • positive regulation of steroid metabolic process   • metabolic process   • regulation of lipid biosynthetic process   • positive regulation of small molecule metabolic process   • regulation of metabolic process   • positive regulation of alcohol biosynthetic process   • positive regulation of sterol biosynthetic process   • lipid metabolic process   • regulation of cytoskeleton organization   • regulation of cellular component organization   • microtubule cytoskeleton organization   • regulation of mitotic spindle organization   • mitotic cell cycle   • cellular component organization   • cell cycle   • cellular component organization or biogenesis   • regulation of cell cycle   • microtubule cytoskeleton organization involved in mitosis   • spindle organization   • cell cycle process   • regulation of cell cycle process   • regulation of microtubule-based process   • regulation of spindle organization   • regulation of organelle organization   • mitotic spindle organization   • organelle organization   • mitotic cell cycle process   • microtubule-based process   • cytoskeleton organization   • regulation of microtubule cytoskeleton organization   • protein localization   • positive regulation of protein localization to cell periphery   • regulation of localization   • protein localization to cell periphery   • cellular localization   • regulation of protein localization   • positive regulation of protein localization to cell cortex   • regulation of protein localization to cell periphery   • localization   • regulation of cellular localization   • regulation of protein localization to cell cortex   • cellular macromolecule localization   • macromolecule localization   • positive regulation of protein localization   • protein localization to cell cortex   • response to ketone   • response to prostaglandin   • response to lipid   • response to alcohol   • response to prostaglandin E   • cellular response to forskolin   • cellular response to oxygen-containing compound   • cellular response to chemical stimulus   • cellular response to alcohol   • response to forskolin   • cellular response to lipid   • cellular response to ketone   • midbody   • nucleus   • membrane-enclosed lumen   • intracellular membraneless organelle   • nucleolus   • intracellular organelle lumen   • organelle lumen   • membraneless organelle   • nuclear lumen   • cell cortex   • protein-containing complex   • extrinsic component of plasma membrane   • catalytic complex   • plasma membrane protein complex   • cytoplasmic side of membrane   • membrane protein complex   • heterotrimeric G-protein complex   • side of membrane   • cytoplasmic side of plasma membrane   • GTPase complex   • extrinsic component of membrane   • extrinsic component of cytoplasmic side of plasma membrane   • extracellular exosome   • extracellular vesicle   • extracellular organelle   • extracellular region   • extracellular space   • extracellular membrane-bounded organelle   • centrosome   • microtubule organizing center   • cytoskeleton   • microtubule cytoskeleton   • cytosol   • nucleoplasm   • vacuolar membrane   • lytic vacuole   • vacuole   • lytic vacuole membrane   • lysosomal membrane   • lysosome   • enzyme binding   • GTPase binding   • signaling receptor complex adaptor activity   • protein-macromolecule adaptor activity   • molecular adaptor activity   • signaling adaptor activity   • multicellular organismal process   • system process   • sensory perception of chemical stimulus   • sensory perception   • nervous system process   • sensory perception of taste   • developmental process   • sensory organ development   • eye development   • animal organ development   • retina development in camera-type eye   • visual system development   • multicellular organism development   • camera-type eye development   • anatomical structure development   • sensory system development   • system development   • cell population proliferation   • cellular response to prostaglandin stimulus   • cellular response to endogenous stimulus   • cellular response to prostaglandin E stimulus   • cellular response to hormone stimulus   • small GTPase-mediated signal transduction   • Ras protein signal transduction   • intracellular signal transduction   • intracellular signaling cassette   • phospholipase C-activating G protein-coupled receptor signaling pathway   • cellular response to nitrogen compound   • response to dopamine   • cellular response to dopamine   • response to monoamine   • response to catecholamine   • adenylate cyclase-activating dopamine receptor signaling pathway   • cellular response to catecholamine stimulus   • G protein-coupled dopamine receptor signaling pathway   • adenylate cyclase-activating G protein-coupled receptor signaling pathway   • cellular response to monoamine stimulus   • synaptic signaling   • cellular response to acetylcholine   • cell-cell signaling   • acetylcholine receptor signaling pathway   • postsynaptic signal transduction   • G protein-coupled acetylcholine receptor signaling pathway   • response to acetylcholine   • non-motile cilium   • 9+0 non-motile cilium   • cilium   • neuron projection   • photoreceptor disc membrane   • photoreceptor outer segment   • plasma membrane bounded cell projection   • cell projection   • photoreceptor cell cilium   • synapse   • cell junction   • G-protein beta-subunit binding   • fibroblast proliferation
SCOP2Domain Identifier
SCOP2Family Identifier
Membrane Protein Annotations-• Orientations of Proteins in Membranes database (OPM)   • Protein Data Bank of Transmembrane Proteins (PDBTM)   • MemProtMD


Details about the values in these tables can be found in the corresponding documentation page .
CodeA1L
PDB ResiduesL:L:?1
Environment DetailsOpen EMBL-EBI Page
CodeA1L
Name[2-[[(2S)-1-[bis(phenylmethyl)amino]-5-[[N-(methylcarbamoyl)carbamimidoyl]amino]-1-oxidanylidene-pentan-2-yl]amino]-2-oxidanylidene-ethyl]-diazonio-azanide
Synonyms
Identifier
FormulaC24 H31 N9 O3
Molecular Weight493.561
SMILES
PubChem44129754
Formal Charge0
Total Atoms67
Total Chiral Atoms1
Total Bonds68
Total Aromatic Bonds12



PDBsumOpen PDBsum Page
This receptor, from the same or other species and bound to the same or other ligands, is also present in the following networks:
Show PDB Class SubFamily Type SubType Species Orthosteric Ligand Other Ligand(s) Protein Partners Resolution Date DOI
8Y63APeptideFormylpeptideFPR2-ALXHomo sapiensC20:0 Ceramide-Gi1/β1/γ23.22025-02-05To be published
8Y62APeptideFormylpeptideFPR2-ALXHomo sapiensC16:0 Ceramide-Gi1/β1/γ23.22025-02-05To be published
7WVYAPeptideFormylpeptideFPR2-ALXHomo sapiensAmyloid-β42-Gi2/β1/γ232022-04-1310.1038/s41467-022-29361-x
7WVXAPeptideFormylpeptideFPR2-ALXHomo sapiensHumanin-Gi2/β1/γ22.82022-04-1310.1038/s41467-022-29361-x
7WVWAPeptideFormylpeptideFPR2-ALXHomo sapiensfMYFINILTL-Gi2/β1/γ23.12022-04-1310.1038/s41467-022-29361-x
7WVVAPeptideFormylpeptideFPR2-ALXHomo sapiensfMLFII-Gi2/β1/γ22.92022-04-1310.1038/s41467-022-29361-x
7T6VAPeptideFormylpeptideFPR2-ALXHomo sapiensfMLFII-Gi1/β1/γ23.12022-03-3010.1038/s41467-022-28586-0
7T6UAPeptideFormylpeptideFPR2-ALXHomo sapiensCGEN-855A-Gi1/β1/γ22.92022-03-3010.1038/s41467-022-28586-0
7T6SAPeptideFormylpeptideFPR2-ALXHomo sapiensPubChem 24776341-Gi1/β1/γ232022-03-3010.1038/s41467-022-28586-0
6LW5APeptideFormylpeptideFPR2-ALXHomo sapiensWKYMVm--2.82020-03-2510.1038/s41467-020-15009-1
6OMMAPeptideFormylpeptideFPR2-ALXHomo sapiensWKYMVX-Gi1/β1/γ23.172020-02-2610.1038/s41467-020-14728-9




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