Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg Int. Strength Num Of Links Community ConSurf
1A:A:Q19 7.95754194
2A:A:Y37 9.064204
3A:A:L43 4.72254117
4A:A:L46 4.0375408
5A:A:S51 4.3445259
6A:A:K53 7.40254259
7A:A:F219 6.53667608
8A:A:H220 11.195427
9A:A:M221 5.7675408
10A:A:F222 7.89667627
11A:A:Q227 5.88333629
12A:A:E230 5.9525429
13A:A:K233 6.54833629
14A:A:W234 6.25729
15A:A:F238 9.015629
16A:A:F246 5.335409
17A:A:Y253 7.422508
18A:A:R265 10.08254269
19A:A:F273 5.458336159
20A:A:W277 8.788577156
21A:A:W281 13.205625
22A:A:I288 5.3275409
23A:A:F290 5.708336119
24A:A:E314 3.88406
25A:A:F315 13.38406
26A:A:P321 3.89575
27A:A:E330 6.98473
28A:A:K338 9.2375475
29A:A:Y339 6.20167673
30A:A:F340 11.3325407
31A:A:R342 6.848574
32A:A:E344 6.025405
33A:A:F345 7.8125408
34A:A:Y358 9.5125404
35A:A:Y360 7.754568
36A:A:F363 10.26575
37A:A:T364 7.454119
38A:A:D368 5.7954119
39A:A:N371 8.43754119
40A:A:R373 7.09254145
41A:A:R374 6.60754114
42A:A:F376 6.475717148
43A:A:R380 4.10754147
44A:A:R385 9565
45A:A:L388 5.22468
46A:A:L393 5.275468
47A:A:L394 5.7375468
48B:B:R22 7.68406
49B:B:I37 4.8075492
50B:B:V40 4.63593
51B:B:I43 4.9025493
52B:B:H54 11.2125409
53B:B:K57 10.088529
54B:B:Y59 8.528528
55B:B:M61 4.2425486
56B:B:W63 6.46687
57B:B:D76 6.4085209
58B:B:K78 5.3525408
59B:B:W82 10.7085249
60B:B:D83 9.57754198
61B:B:K89 6.143336249
62B:B:I93 7.0525407
63B:B:L95 5.4285228
64B:B:W99 11.354529
65B:B:M101 7.015429
66B:B:Y105 5.081437166
67B:B:N110 6.5075424
68B:B:Y111 4.9575424
69B:B:C114 5.014228
70B:B:D118 4.8175409
71B:B:C121 4.5325428
72B:B:I123 5.03526
73B:B:Y124 7.0575406
74B:B:L139 7.64409
75B:B:H142 7.864529
76B:B:Y145 7.14125828
77B:B:C149 3.772528
78B:B:F151 5.70167629
79B:B:L152 3.7975433
80B:B:I157 5.6275427
81B:B:V158 4.245435
82B:B:T159 6.702529
83B:B:S160 5.2436
84B:B:D163 9.47429
85B:B:C166 4.235438
86B:B:W169 8.635628
87B:B:D170 6.435439
88B:B:Q176 7.1425424
89B:B:F180 8.632537
90B:B:H183 8.898539
91B:B:D186 6.29529
92B:B:V187 5.4925439
93B:B:L190 5.73435
94B:B:F199 9.425439
95B:B:S201 4.416539
96B:B:C204 6.3427
97B:B:D205 6.072539
98B:B:K209 9.628536
99B:B:W211 9.054538
100B:B:R219 5.4125445
101B:B:Q220 6.284547
102B:B:F222 9.145448
103B:B:H225 9.43714749
104B:B:D228 8.434529
105B:B:I232 5.8625448
106B:B:F235 7.2156236
107B:B:P236 6.714237
108B:B:F241 8.848546
109B:B:T243 7448
110B:B:D246 6.545429
111B:B:D247 8.215449
112B:B:T249 7.2025446
113B:B:R251 12.228548
114B:B:F253 7.67646
115B:B:D258 6.488547
116B:B:Q259 5.06506
117B:B:Y264 5.96714705
118B:B:I269 4.4654124
119B:B:F278 5.8345237
120B:B:R283 8.256599
121B:B:L284 5.244595
122B:B:L285 4.8375406
123B:B:Y289 7.825717127
124B:B:D290 7.635426
125B:B:C294 4.69254105
126B:B:N295 8.6654126
127B:B:V296 4.124595
128B:B:W297 8.4254128
129B:B:R304 7.72754125
130B:B:H311 8.0665109
131B:B:R314 15.408528
132B:B:V315 4.42754107
133B:B:M325 8.445485
134B:B:T329 5.0945108
135B:B:W332 11.3243729
136B:B:D333 8.734109
137B:B:F335 7.2775404
138B:B:L336 4.602587
139B:B:K337 9.3254106
140B:B:W339 7.6085109
141G:G:R27 5.8825448
142G:G:D48 6.438599
143G:G:P49 4.7825407
144G:G:V54 4.29754286
145G:G:N59 7.5825409
146G:G:P60 8.545489
147G:G:F61 5.41143788
148L:L:V2 7.295410
149L:L:E4 6.79410
150L:L:I5 5.345410
151L:L:Q6 10.978510
152L:L:H9 6.97410
153L:L:H14 7.366510
154L:L:R20 12.7325400
155L:L:W23 10.75170
156L:L:K27 9.44254170
157R:R:C108 4.66459
158R:R:L116 7.2475455
159R:R:W118 10.9383659
160R:R:V129 6.6925455
161R:R:C131 5.385459
162R:R:Y134 8.835455
163R:R:F138 7.54143754
164R:R:R146 12.352558
165R:R:W154 11.304559
166R:R:V157 8.624294
167R:R:R162 8.68754293
168R:R:Y167 6.705405
169R:R:E180 5.625413
170R:R:F184 5.308516
171R:R:Y191 5.944517
172R:R:Y195 6.96717
173R:R:F212 9.7885137
174R:R:R214 8.16407
175R:R:L215 5.295139
176R:R:T218 5.86754217
177R:R:R219 7.426676139
178R:R:N220 6.6485139
179R:R:H223 5.614139
180R:R:H225 13.61418
181R:R:F227 4.59254309
182R:R:F230 9.17618
183R:R:R233 6.93286718
184R:R:K240 7.322517
185R:R:L244 5.17615
186R:R:Y245 7.502514
187R:R:F288 7.125417
188R:R:L289 5.35417
189R:R:Y290 6.2525409
190R:R:N295 10.82418
191R:R:Y296 8.89833617
192R:R:Y297 6.5885316
193R:R:W298 12.4067619
194R:R:I299 5.42419
195R:R:L300 5.188508
196R:R:E302 9.51409
197R:R:Y305 6.908336218
198R:R:H307 11.54254188
199R:R:F311 8.2285186
200R:R:F315 8.0375406
201R:R:E317 6.00254216
202R:R:W329 9.114519
203R:R:W339 6.23667618
204R:R:R343 8.5925418
205R:R:W352 10.226518
206R:R:K360 8.4575417
207R:R:Q364 7.42517
208R:R:F378 8.066569
209R:R:K388 8.04469
210R:R:M414 3.9575468
211R:R:F417 6.744569
212R:R:H420 8.664518
213R:R:Y421 11.6083618
214R:R:F424 8.242517
215R:R:M425 3.802506
216R:R:T427 5.0775415
217R:R:Y429 12.096516
218R:R:V432 8.64415
219R:R:W437 9.956515
220R:R:Q440 7.984516
221R:R:M441 8.785416
222R:R:Y443 7.402514
223R:R:E444 8.24417
224R:R:M445 5.6475406
225R:R:N448 8.712516
226R:R:Q451 7.172519
227R:R:F453 5.965406
228R:R:C460 3.95754309
229R:R:E469 9.2054139
230R:R:R476 3.2925407
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Int. Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.

Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1B:B:W332 B:B:Y59 20.22635.79YesYes298
2B:B:R314 B:B:W332 22.275118.99YesYes289
3B:B:R314 B:B:T274 22.74346.47YesNo288
4B:B:S275 B:B:T274 23.31973.2NoNo088
5B:B:L318 B:B:S275 23.3667.51NoNo068
6B:B:L318 B:B:T329 23.51164.42NoYes068
7B:B:H311 B:B:T329 53.69246.85YesYes1098
8B:B:D333 B:B:H311 84.38586.3YesYes1099
9B:B:D312 B:B:D333 42.20976.65NoYes059
10B:B:D312 R:R:R214 42.208610.72NoYes057
11R:R:E469 R:R:R214 1006.98YesYes097
12R:R:E469 R:R:L215 99.61919.28YesYes1399
13R:R:L215 R:R:N220 93.8964.12YesYes1399
14A:A:Y391 R:R:R219 10.797413.38NoYes049
15B:B:D333 B:B:F335 42.2613.14YesYes094
16B:B:F335 R:R:R214 50.03114.28YesYes047
17R:R:H223 R:R:N220 87.19915.1YesYes1399
18R:R:E302 R:R:H223 80.97457.39YesYes099
19R:R:F417 R:R:L416 10.6464.87YesNo099
20R:R:F417 R:R:L413 10.94193.65YesNo699
21A:A:L393 R:R:L413 10.93938.3YesNo689
22B:B:L284 B:B:V40 38.12384.47YesYes953
23B:B:R283 B:B:V40 68.65617.85YesYes993
24B:B:L300 B:B:R283 66.58218.5NoYes969
25B:B:L300 B:B:T34 66.07284.42NoNo065
26B:B:L30 B:B:T34 65.03652.95NoNo055
27B:B:L30 B:B:M262 59.85329.9NoNo054
28B:B:M262 B:B:Y264 58.81617.18NoYes045
29B:B:L252 B:B:Y264 38.02917.03NoYes075
30B:B:L252 B:B:L261 33.36415.54NoNo075
31B:B:L261 G:G:V30 31.28292.98NoNo058
32B:B:Q259 G:G:V30 30.76267.16YesNo068
33B:B:Q259 B:B:R22 28.68079.35YesYes066
34B:B:D258 B:B:R22 25.55573.57YesYes076
35B:B:L284 B:B:V296 39.98745.96YesYes955
36B:B:L286 B:B:V296 74.48252.98NoYes075
37B:B:L286 B:B:V327 74.73242.98NoNo076
38B:B:V327 G:G:L50 74.98384.47NoNo069
39B:B:M45 G:G:L50 75.23878.48NoNo049
40B:B:L308 B:B:M45 75.49795.65NoNo074
41B:B:L308 B:B:W339 45.440313.67NoYes079
42B:B:K337 B:B:W339 30.81825.8YesYes1069
43B:B:T329 B:B:W339 15.61976.06YesYes1089
44B:B:H311 B:B:K337 15.533610.48YesYes1096
45B:B:K337 B:B:T50 15.550612.01YesNo063
46B:B:R52 B:B:T50 15.58489.06NoNo073
47B:B:D258 B:B:F222 16.69465.97YesYes478
48B:B:C294 B:B:L308 30.31916.35YesNo057
49B:B:C294 B:B:T329 15.28233.38YesYes1058
50R:R:E302 R:R:L226 74.244417.23YesNo099
51R:R:F230 R:R:L226 74.18237.31YesNo089
52R:R:F230 R:R:Q451 24.66410.54YesYes189
53R:R:F230 R:R:N295 49.456718.12YesYes188
54R:R:N295 R:R:R233 51.55412.05YesYes188
55R:R:R233 R:R:Y296 22.24112.35YesYes187
56L:L:V2 R:R:Y296 44.02723.79YesYes107
57R:R:Q451 R:R:Y421 23.24327.89YesYes198
58R:R:Y296 R:R:Y421 22.237216.88YesYes178
59L:L:I5 L:L:V2 42.90677.68YesYes100
60R:R:R233 R:R:Y195 27.19459.26YesYes187
61R:R:I237 R:R:Y195 22.4018.46NoYes177
62R:R:F288 R:R:I237 22.37113.77YesNo177
63R:R:F288 R:R:L289 21.48694.87YesYes177
64L:L:I5 R:R:L289 42.6244.28YesYes107
65R:R:L289 R:R:W339 63.59477.97YesYes178
66R:R:V340 R:R:W339 30.84743.68NoYes158
67R:R:V340 R:R:W352 30.60694.9NoYes158
68R:R:R282 R:R:W352 59.760824.99NoYes188
69R:R:R282 R:R:Y278 59.2755.14NoNo084
70R:R:E35 R:R:Y278 58.29924.49NoNo054
71R:R:E35 R:R:T33 57.81288.47NoNo057
72L:L:N16 R:R:T33 55.86072.92NoNo007
73L:L:N16 L:L:S17 55.37262.98NoNo000
74L:L:R20 L:L:S17 54.88447.91YesNo000
75R:R:R343 R:R:W339 32.56158YesYes188
76R:R:R343 R:R:W352 30.619613YesYes188
77L:L:R20 R:R:Q37 50.98115.19YesNo007
78L:L:W23 R:R:Q37 50.492518.62YesNo007
79L:L:K27 L:L:W23 45.10629.28YesYes1700
80L:L:K27 R:R:I115 43.65055.82YesNo005
81R:R:F138 R:R:I115 37.29113.77YesNo045
82R:R:C170 R:R:F138 19.630411.17NoYes594
83R:R:C170 R:R:Y167 19.14128.06NoYes095
84R:R:W118 R:R:Y167 17.67076.75YesYes095
85R:R:L116 R:R:V129 11.77967.45YesYes555
86R:R:P130 R:R:V129 16.20153.53NoYes055
87R:R:H143 R:R:P130 14.72889.15NoNo035
88R:R:H143 R:R:Y145 11.78334.36NoNo034
89B:B:H311 B:B:V315 15.24524.15YesYes1097
90B:B:C294 B:B:V315 15.14335.12YesYes1057
91B:B:I43 B:B:V296 33.37084.61YesYes935
92B:B:I43 B:B:V40 33.12814.61YesYes933
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1 Node2 LinkStrength Comm IsNode1Hub? IsNode2Hub? Node1Cons Node2Cons Node1Shell Node2Shell
L:L:S1 R:R:Y429 5.09 1 No Yes 0 6 0 1
L:L:V2 R:R:Y296 3.79 1 Yes Yes 0 7 0 1
L:L:V2 R:R:Q364 10.03 1 Yes Yes 0 7 0 1
L:L:V2 R:R:I367 7.68 1 Yes No 0 7 0 1
L:L:S3 R:R:Q440 4.33 0 No Yes 0 6 0 1
L:L:S3 R:R:E444 12.94 0 No Yes 0 7 0 1
L:L:E4 R:R:Y195 8.98 1 Yes Yes 0 7 0 1
L:L:E4 R:R:R233 3.49 1 Yes Yes 0 8 0 1
L:L:E4 R:R:M445 8.12 1 Yes Yes 0 6 0 1
L:L:E4 R:R:N448 6.57 1 Yes Yes 0 6 0 1
L:L:I5 R:R:L289 4.28 1 Yes Yes 0 7 0 1
L:L:I5 R:R:Q364 4.12 1 Yes Yes 0 7 0 1
L:L:Q6 R:R:Y429 22.55 1 Yes Yes 0 6 0 1
L:L:Q6 R:R:Q440 8.96 1 Yes Yes 0 6 0 1
L:L:Q6 R:R:M441 6.8 1 Yes Yes 0 6 0 1
L:L:L7 R:R:M445 4.24 0 No Yes 0 6 0 1
L:L:M8 R:R:K240 5.76 1 No Yes 0 7 0 1
L:L:M8 R:R:F288 3.73 1 No Yes 0 7 0 1
L:L:H9 R:R:S355 5.58 1 Yes No 0 7 0 1
L:L:H9 R:R:K360 3.93 1 Yes Yes 0 7 0 1
L:L:H9 R:R:Y429 13.07 1 Yes Yes 0 6 0 1
L:L:N10 R:R:V432 4.43 1 No Yes 0 5 0 1
L:L:N10 R:R:W437 9.04 1 No Yes 0 5 0 1
L:L:L11 R:R:F184 4.87 1 No Yes 0 6 0 1
L:L:L11 R:R:Y245 16.41 1 No Yes 0 4 0 1
L:L:H14 R:R:E180 6.15 1 Yes Yes 0 3 0 1
L:L:H14 R:R:R181 4.51 1 Yes No 0 3 0 1
L:L:H14 R:R:F184 7.92 1 Yes Yes 0 6 0 1
L:L:L15 R:R:Y245 3.52 1 No Yes 0 4 0 1
L:L:E19 R:R:K34 10.8 0 No No 0 4 0 1
L:L:R20 R:R:Q37 15.19 0 Yes No 0 7 0 1
L:L:R20 R:R:Y136 12.35 0 Yes No 0 4 0 1
L:L:R20 R:R:D137 15.48 0 Yes No 0 5 0 1
L:L:V21 R:R:D137 8.76 0 No No 0 5 0 1
L:L:W23 R:R:K34 4.64 17 Yes No 0 4 0 1
L:L:W23 R:R:Q37 18.62 17 Yes No 0 7 0 1
L:L:W23 R:R:I38 15.27 17 Yes No 0 7 0 1
L:L:W23 R:R:L41 5.69 17 Yes No 0 8 0 1
L:L:L24 R:R:I135 5.71 5 No No 0 7 0 1
L:L:L24 R:R:F138 10.96 5 No Yes 0 4 0 1
L:L:K27 R:R:L41 5.64 17 Yes No 0 8 0 1
L:L:K27 R:R:H114 17.03 17 Yes No 0 4 0 1
L:L:K27 R:R:I115 5.82 17 Yes No 0 5 0 1
L:L:D30 R:R:H114 18.91 0 No No 0 4 0 1
L:L:V31 R:R:D113 11.69 0 No No 0 9 0 1
L:L:H32 R:R:R162 6.77 0 No Yes 0 3 0 1
L:L:F34 R:R:R162 3.21 0 No Yes 0 3 0 1
R:R:E35 R:R:T33 8.47 0 No No 5 7 2 1
R:R:I38 R:R:K34 5.82 17 No No 7 4 1 1
R:R:L41 R:R:W112 4.56 17 No No 8 7 1 2
R:R:D113 R:R:I115 4.2 0 No No 9 5 1 1
R:R:F138 R:R:I115 3.77 5 Yes No 4 5 1 1
R:R:C131 R:R:F138 4.19 5 Yes Yes 9 4 2 1
R:R:C131 R:R:C170 7.28 5 Yes No 9 9 2 2
R:R:I135 R:R:Y134 4.84 5 No Yes 7 5 1 2
R:R:F138 R:R:I135 16.33 5 Yes No 4 7 1 1
R:R:C170 R:R:F138 11.17 5 No Yes 9 4 2 1
R:R:F138 R:R:V171 3.93 5 Yes No 4 3 1 2
R:R:R162 R:R:V157 11.77 29 Yes Yes 3 4 1 2
R:R:V157 R:R:W164 12.26 29 Yes No 4 5 2 2
R:R:R162 R:R:W164 13 29 Yes No 3 5 1 2
R:R:R181 R:R:T178 3.88 0 No No 3 3 1 2
R:R:E180 R:R:F184 3.5 1 Yes Yes 3 6 1 1
R:R:E180 R:R:V432 11.41 1 Yes Yes 3 5 1 1
R:R:D185 R:R:R181 13.1 0 No No 2 3 2 1
R:R:F184 R:R:V432 5.24 1 Yes Yes 6 5 1 1
R:R:F184 R:R:W437 5.01 1 Yes Yes 6 5 1 1
R:R:L187 R:R:M441 5.65 0 No Yes 5 6 2 1
R:R:L187 R:R:M445 4.24 0 No Yes 5 6 2 1
R:R:Y191 R:R:Y195 5.96 1 Yes Yes 7 7 2 1
R:R:I237 R:R:Y191 3.63 1 No Yes 7 7 2 2
R:R:D241 R:R:Y191 6.9 1 No Yes 8 7 2 2
R:R:M445 R:R:Y191 5.99 0 Yes Yes 6 7 1 2
R:R:R233 R:R:Y195 9.26 1 Yes Yes 8 7 1 1
R:R:A234 R:R:Y195 5.34 0 No Yes 8 7 2 1
R:R:I237 R:R:Y195 8.46 1 No Yes 7 7 2 1
R:R:S449 R:R:Y195 7.63 0 No Yes 9 7 2 1
R:R:L292 R:R:R233 3.64 1 No Yes 6 8 2 1
R:R:N295 R:R:R233 12.05 1 Yes Yes 8 8 2 1
R:R:R233 R:R:Y296 12.35 1 Yes Yes 8 7 1 1
R:R:R233 R:R:Y421 4.12 1 Yes Yes 8 8 1 2
R:R:N448 R:R:R233 3.62 1 Yes Yes 6 8 1 1
R:R:F288 R:R:I237 3.77 1 Yes No 7 7 1 2
R:R:D241 R:R:K240 6.91 1 No Yes 8 7 2 1
R:R:K240 R:R:L244 4.23 1 Yes Yes 7 5 1 2
R:R:K240 R:R:Y245 3.58 1 Yes Yes 7 4 1 1
R:R:F288 R:R:K240 16.13 1 Yes Yes 7 7 1 1
R:R:D241 R:R:Y245 3.45 1 No Yes 8 4 2 1
R:R:L244 R:R:Y245 10.55 1 Yes Yes 5 4 2 1
R:R:D353 R:R:L244 5.43 0 No Yes 5 5 2 2
R:R:F288 R:R:L289 4.87 1 Yes Yes 7 7 1 1
R:R:L289 R:R:W339 7.97 1 Yes Yes 7 8 1 2
R:R:I363 R:R:L289 4.28 1 No Yes 7 7 2 1
R:R:L292 R:R:Y296 5.86 1 No Yes 6 7 2 1
R:R:A293 R:R:I367 3.25 0 No No 6 7 2 1
R:R:I367 R:R:Y296 9.67 1 No Yes 7 7 1 1
R:R:I371 R:R:Y296 4.84 1 No Yes 7 7 2 1
R:R:Y296 R:R:Y421 16.88 1 Yes Yes 7 8 1 2
R:R:I363 R:R:W339 9.4 1 No Yes 7 8 2 2
R:R:D353 R:R:L354 4.07 0 No No 5 5 2 1
R:R:K360 R:R:W361 15.08 1 Yes No 7 8 1 2
R:R:K360 R:R:Q364 4.07 1 Yes Yes 7 7 1 1
R:R:K360 R:R:Y429 10.75 1 Yes Yes 7 6 1 1
R:R:Q364 R:R:W361 9.86 1 Yes No 7 8 1 2
R:R:Q364 R:R:Y429 9.02 1 Yes Yes 7 6 1 1
R:R:I371 R:R:Y421 6.04 1 No Yes 7 8 2 2
R:R:H420 R:R:Y421 19.6 1 Yes Yes 8 8 2 2
R:R:H420 R:R:Y443 5.44 1 Yes Yes 8 4 2 2
R:R:H420 R:R:N448 5.1 1 Yes Yes 8 6 2 1
R:R:N448 R:R:Y421 15.12 1 Yes Yes 6 8 1 2
R:R:F424 R:R:T427 3.89 1 Yes Yes 7 5 2 2
R:R:F424 R:R:Q440 14.05 1 Yes Yes 7 6 2 1
R:R:F424 R:R:Y443 9.28 1 Yes Yes 7 4 2 2
R:R:E444 R:R:F424 3.5 1 Yes Yes 7 7 1 2
R:R:Q440 R:R:T427 8.5 1 Yes Yes 6 5 1 2
R:R:T430 R:R:W437 3.64 0 No Yes 5 5 2 1
R:R:V432 R:R:W437 13.48 1 Yes Yes 5 5 1 1
R:R:M441 R:R:W437 18.61 1 Yes Yes 6 5 1 1
R:R:M441 R:R:Q440 4.08 1 Yes Yes 6 6 1 1
R:R:E444 R:R:Y443 3.37 1 Yes Yes 7 4 1 2
R:R:E444 R:R:N448 13.15 1 Yes Yes 7 6 1 1
R:R:F238 R:R:Y195 3.09 0 No Yes 7 7 2 1
L:L:N16 R:R:T33 2.92 0 No No 0 7 0 1
R:R:E36 R:R:T33 2.82 0 No No 6 7 2 1
L:L:L28 R:R:F138 2.44 0 No Yes 0 4 0 1
L:L:R25 R:R:N176 2.41 0 No No 0 3 0 1
L:L:F34 R:R:D113 2.39 0 No No 0 9 0 1
L:L:G12 R:R:L354 1.71 0 No No 0 5 0 1
L:L:V21 R:R:L174 1.49 0 No No 0 3 0 1
R:R:E180 R:R:S433 1.44 1 Yes No 3 3 1 2
R:R:L174 R:R:N176 1.37 0 No No 3 3 1 1

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
82.14Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
79.31Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
78.57Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
75.86Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
74.07Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
73.33Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
73.33Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
71.43Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
69.23Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
66.67Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
64.29Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
60.71Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
60.00Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
60.00Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
58.62Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
56.67Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
56.25Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
54.84Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
54.84Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
54.84Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
53.33Single6FJ3PTH6FJ3-PTH1-PTH
53.33Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
53.33Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
53.12Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
51.61Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
51.61Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
51.61Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
50.00Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
48.65Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
48.39Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
48.39Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
48.39Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
46.88Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
46.88Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
45.71Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
45.16Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
45.16Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
45.16Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
44.44Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
44.44Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
43.75Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
43.75Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
43.75Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
43.75Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
43.33Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
42.86Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
42.42Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
41.94Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
41.94Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
41.94Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
41.18Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
41.18Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
41.18Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
40.62Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
40.62Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
40.00Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
40.00Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
40.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
39.47Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
39.39Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
38.24Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
38.24Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
37.50Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
37.50Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
37.50Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
37.14Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
37.14Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
37.14Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
37.14Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
36.84Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
36.67Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
36.11Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
35.29Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
35.14Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
35.14Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
34.38Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
34.29Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
34.29Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
34.29Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
34.21Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
34.21Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
33.33Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
33.33Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
33.33Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
33.33Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
33.33Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
33.33Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
33.33Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
32.43Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
32.35Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
32.26Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
31.58Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
31.25Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
31.03Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
30.77Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
30.56Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
30.56Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
30.30Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
30.23Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
30.00Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
29.55Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
29.41Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
29.03Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
29.03Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
28.95Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
28.57Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
28.12Single4XT1Fractalkine4XT1-US28-Fractalkine
28.12Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
27.59Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
27.59Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
27.59Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
27.59Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
27.27Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
27.27Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
26.67Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
26.67Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
26.67Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
26.67Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
26.47Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
25.81Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
25.71Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
25.71Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
25.00Single5EE7MK08935EE7-Glucagon-MK0893
25.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
25.00Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
25.00Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
25.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
25.00Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
25.00Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
25.00Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
24.32Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
24.32Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
24.32Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
24.32Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
24.32Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
24.32Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
24.24Single7QA8Peptide7QA8-STE2-Peptide
24.24Single7QA8Peptide7QA8-STE2-Peptide
24.24Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
24.14Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
24.14Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
24.14Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
24.14Single8S4DCMF-0198S4D-Apelin-CMF-019
24.14Single8TF5Oleic acid8TF5-GPR6-Oleic acid
24.14Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
23.68Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
23.68Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
23.68Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
23.68Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
23.53Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
23.53Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
23.53Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
23.53Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
23.33Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
23.33Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
23.33Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
23.33Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
22.86Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
22.86Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
22.86Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
22.86Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
22.86Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
22.86Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
22.58Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
22.58Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
22.58Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
22.58Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
22.58Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
22.58Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.58Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
22.58Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
22.58Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
22.58Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
22.58Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
22.58Consensuslpl_offOrthosteric Ligands1p_off lpa_off
22.58Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
22.58Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
22.50Single6IGKEndothelin-36IGK-ETB-Endothelin-3
22.22Single5U09Taranabant5U09-CB1-Taranabant
22.22Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
22.22Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
22.22Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.22Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
22.22Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
21.95Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
21.88Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
21.88Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
21.88Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
21.88Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
21.88Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
21.88Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
21.88Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
21.88Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
21.88Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
21.88Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
21.88Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
21.88Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
21.62Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.62Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
21.62Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
21.62Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
21.62Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
21.62Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
21.62Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
21.62Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
21.62Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.43Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
21.43Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
21.43Consensusgrh_offOrthosteric Ligandgnrh1_off
21.21Single4UG2CGS216804UG2-A2A-CGS21680
21.21Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
21.21Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
21.21Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
21.21Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
21.21Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
21.05Single4XT3Fractalkine4XT3-US28-Fractalkine
21.05Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
21.05Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
21.05Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
21.05Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
20.69Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
20.69Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
20.69Single7V3ZCP559407V3Z-CB1-CP55940
20.69Single9B9ZA1AKO9B9Z-CB1-A1AKO
20.69Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
20.59Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
20.59Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
20.59Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
20.59Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
20.59Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
20.59Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
20.59Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
20.59Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
20.59Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
20.59Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.51Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.51Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
20.51Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
20.51Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
20.51Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
20.51Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
20.51Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
20.00Single3QAKUK-4320973QAK-A2A-UK-432097
20.00Single5C1MBU725C1M-μ-BU72
20.00Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
20.00Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
20.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
20.00Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
20.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
20.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
20.00Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
20.00Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
20.00Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
20.00Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8IY6Endothelin-18IY6-ETB-Endothelin-1
20.00Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
20.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
20.00Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
20.00Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
20.00Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
20.00Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
20.00Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
20.00Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
20.00Consensusendothelin_onOrthosteric Ligandetb_on eta_on
20.00Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
20.00Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
20.00Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.00Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
19.51Single5GLHEndothelin-15GLH-ETB-Endothelin-1
19.51Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
19.51Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
19.51Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
19.51Consensusbombesin_onOrthosteric Ligandbb2_on
19.51Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
19.51Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
19.51Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
19.51Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
19.51Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
19.44Single5WF5UK-4320975WF5-A2A-UK-432097
19.44Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
19.44Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.44Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
19.44Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
19.44Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
19.44Consensusangiotensin_onOrthosteric Ligandat1_on
19.44Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
19.44Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
19.44Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
19.44Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
19.44Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
19.44Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
19.44Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
19.44Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
19.35Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
19.35Single5XRAAM115425XRA-CB1-AM11542
19.35Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
19.35Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
19.35Single7F1TMIP-1a7F1T-CCR5-MIP-1a
19.35Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
19.35Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
19.35Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
19.35Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
19.35Single8E0GBU728E0G-μ-BU72
19.35Single8EA0Iperoxo8EA0-M3-Iperoxo
19.35Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
19.35Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
19.35Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
19.35Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
19.35Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
19.35Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
19.35Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
19.35Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
19.35Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
19.35Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
19.05Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
19.05Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
18.92Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
18.92Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
18.92Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
18.92Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
18.92Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
18.92Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
18.92Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
18.92Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
18.92Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
18.92Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
18.92Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
18.92Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
18.92Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
18.92Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
18.92Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
18.92Consensusvasop-oxy_onOrthosteric Ligandv2_on
18.92Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
18.75Single6A93Risperidone6A93-5-HT2A-Risperidone
18.75Single6KQICP559406KQI-CB1-CP55940-Org27569
18.75Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
18.75Single6OS2TRV0266OS2-AT1-TRV026
18.75Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
18.75Single7DFPSpiperone7DFP-D2-Spiperone
18.75Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
18.75Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
18.75Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
18.75Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
18.75Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
18.75Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
18.75Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
18.75Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
18.75Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
18.75Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
18.75Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
18.75Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
18.75Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
18.75Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
18.75Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
18.75Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
18.75Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
18.75Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
18.75Consensuslpa_offOrthosteric Ligandlpa1_off
18.75Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
18.75Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
18.75Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
18.60Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
18.52Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
18.42Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
18.42Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
18.42Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
18.42Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
18.42Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
18.42Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
18.42Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
18.42Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
18.42Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
18.42Single8ZRTET-18ZRT-ETB-ET-1
18.42Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
18.42Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
18.42Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.42Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
18.42Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
18.42Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
18.18Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
18.18Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
18.18Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
18.18Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
18.18Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
18.18Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
18.18Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
18.18Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
18.18Single8XVUCXCL28XVU-CXCR2-CXCL2
18.18Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
18.18Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
18.18Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
18.18Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
18.18Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
17.95Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
17.95Single7SK3CXCL127SK3-ACKR3-CXCL12
17.86Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
17.86Single4BWBNeurotensin4BWB-NTS1-Neurotensin
17.86Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
17.86Single7BR3Elagolix7BR3-GnRH1-Elagolix
17.86Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
17.86Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
17.86Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
17.86Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
17.86Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
17.86Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
17.86Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
17.86Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
17.65Single3NY9ICI118-5513NY9-β2-ICI118-551
17.65Single5ZTYAM102575ZTY-CB2-AM10257
17.65Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
17.65Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
17.65Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
17.65Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
17.65Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
17.65Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
17.65Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.50Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
17.50Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
17.50Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
17.50Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
17.50Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
17.39Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
17.39Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
17.24Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
17.24Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
17.24Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
17.24Single7T32ZM-2413857T32-A2A-ZM-241385
17.24Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
17.24Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
17.24Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
17.24Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
17.24Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
17.24Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
17.24Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
17.24Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
17.24Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
17.24Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
17.24Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
17.14Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
17.14Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
17.14Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
17.14Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
17.14Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
17.14Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
17.14Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
17.14Single8WDTphotoNECA8WDT-A2A-photoNECA
17.14Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
17.14Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
17.14Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
17.14Consensuslpl_onOrthosteric Ligands1p_on lpa_on
17.14Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
17.14Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
17.07Single6IGLIRL16206IGL-ETB-IRL1620
17.07Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
17.07Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
16.67Single4DAJTiotropium4DAJ-M3-Tiotropium
16.67Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
16.67Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
16.67Single5TGZAM65385TGZ-CB1-AM6538
16.67Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
16.67Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
16.67Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
16.67Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
16.67Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
16.67Single6HLOAprepitant6HLO-NK1-Aprepitant
16.67Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
16.67Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
16.67Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
16.67Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
16.67Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
16.67Single7SK5CXCL127SK5-ACKR3-CXCL12
16.67Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
16.67Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
16.67Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
16.67Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
16.67Single7XNACYN1548067XNA-SST2-CYN154806
16.67Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
16.67Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
16.67Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
16.67Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
16.67Single8T1WCVN4248T1W-GPR6-CVN424
16.67Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
16.67Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
16.67Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
16.67Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
16.67Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
16.67Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
16.67Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
16.67Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
16.67Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
16.67Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
16.67Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
16.67Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
16.67Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
16.67Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
16.67Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
16.67Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
16.67Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
16.28Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
16.28Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
16.22Single3OE0CVX153OE0-CXCR4-CVX15
16.22Single6PT2KGCHM076PT2-δ-KGCHM07
16.22Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
16.22Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.22Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.22Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
16.22Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
16.22Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
16.22Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single5N2RPSB-365N2R-A2A-PSB-36-Na
16.13Single5N2SPSB365N2S-A1-PSB36
16.13Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
16.13Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
16.13Single6D26Fevipiprant6D26-DP2-Fevipiprant
16.13Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
16.13Single7C4SS1P7C4S-S1P3-S1P
16.13Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
16.13Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
16.13Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
16.13Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
16.13Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
16.13Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
16.13Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
16.13Single8JXSPF-61428JXS-D1-PF-6142
16.13Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
16.13Single8QOTNanobody-E8QOT-μ-Nanobody-E
16.13Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
16.13Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
16.13Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
16.13Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
16.13Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
16.13Consensusadenosine_offOrthosteric Liganda1_off a2_off
16.13Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
16.13Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
16.13Consensusdp_offOrthosteric Liganddp2_off
16.13Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
16.13Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
16.13Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
16.13Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
16.00Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
15.91Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
15.79Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
15.79Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
15.79Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
15.79Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
15.79Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
15.79Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
15.79Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.79Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
15.79Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
15.79Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
15.79Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
15.79Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
15.79Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
15.79Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
15.62Single2YDVNECA2YDV-A2A-NECA
15.62Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
15.62Single4BV0Neurotensin4BV0-NTS1-Neurotensin
15.62Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
15.62Single4UHRCGS216804UHR-A2A-CGS21680
15.62Single5G53NECA5G53-A2A-NECA-Gs
15.62Single5XR8AM8415XR8-CB1-AM841
15.62Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
15.62Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
15.62Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
15.62Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
15.62Single6OS1TRV0266OS1-AT1-TRV026
15.62Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
15.62Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
15.62Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
15.62Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
15.62Single7FEECP559407FEE-CB1-CP55940-ZCZ011
15.62Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
15.62Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
15.62Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
15.62Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
15.62Single7PX4PSB-21137PX4-A2A-PSB-2113
15.62Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
15.62Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
15.62Single7TUYGSK682753A7TUY-GPR183-GSK682753A
15.62Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
15.62Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
15.62Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
15.62Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
15.62Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
15.62Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
15.62Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
15.62Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.62Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
15.62Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
15.62Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
15.62Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
15.62Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
15.62Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
15.62Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
15.62Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
15.62Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
15.62Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
15.62Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
15.62Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
15.62Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
15.62Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
15.62Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.62Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
15.62Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
15.62Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
15.62Consensuslpa_onOrthosteric Ligandlpa1_on
15.62Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
15.62Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
15.62Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
15.62Consensusneurotensin_onOrthosteric Ligandnts1_on
15.62Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
15.38Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
15.38Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
15.38Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.38Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
15.38Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
15.38Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
15.15Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
15.15Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
15.15Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
15.15Single4XEENeurotensin4XEE-NTS1-Neurotensin
15.15Single4XESNeurotensin4XES-NTS1-Neurotensin
15.15Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
15.15Single5CXVTiotropium5CXV-M1-Tiotropium
15.15Single6CM4Risperidone6CM4-D2-Risperidone
15.15Single6IIURamatroban6IIU-TP-Ramatroban
15.15Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
15.15Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
15.15Single6YVRNTS8-136YVR-NTS1-NTS8-13
15.15Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
15.15Single7K15MKD0467K15-BLT1-MKD046-Na
15.15Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
15.15Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
15.15Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
15.15Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
15.15Single7YITNalfurafine7YIT-κ-Nalfurafine
15.15Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
15.15Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
15.15Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
15.15Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
15.15Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
15.15Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
15.15Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
15.15Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8XWMCXCL68XWM-CXCR2-CXCL6
15.15Single8XWSCXCL58XWS-CXCR2-CXCL5
15.15Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
15.15Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
15.15Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
15.15Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
15.15Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
15.15Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
15.15Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
15.15Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
15.15Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
15.15Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
15.15Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
15.15Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
15.15Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
15.15Consensusorexin_onOrthosteric Ligandox2_on
15.00Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.00Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
15.00Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
15.00Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
15.00Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
15.00Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
14.81Single3OE6IT1t3OE6-CXCR4-IT1t
14.81Single4XNWMRS25004XNW-P2Y1-MRS2500
14.81Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
14.81Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
14.81Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
14.81Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
14.81Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
14.81Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
14.81Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
14.81Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
14.81Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
14.81Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
14.81Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
14.71Single4BUONeurotensin4BUO-NTS1-Neurotensin
14.71Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
14.71Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
14.71Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
14.71Single5CGDHTL142425CGD-mGlu5-HTL14242
14.71Single5X93K-87945X93-ETB-K-8794
14.71Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
14.71Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
14.71Single7EZCUKA7EZC-A2A-UKA
14.71Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
14.71Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.71Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
14.71Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
14.71Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
14.71Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
14.71Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
14.71Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
14.71Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
14.71Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
14.71Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
14.71Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
14.71Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
14.71Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single8XWFCXCL38XWF-CXCR2-CXCL3
14.71Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
14.71Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
14.71Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
14.71Consensuscck_onOrthosteric Ligandccka_on cckb_on
14.71Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
14.71Consensusendothelin_offOrthosteric Ligandetb_off
14.71Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
14.71Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.71Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.71Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
14.71Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
14.71Consensusprostanoid_offOrthosteric Ligandep_off dp_off
14.71Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
14.71Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
14.71Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
14.63Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
14.63Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
14.29Single3OE9IT1t3OE9-CXCR4-IT1t
14.29Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
14.29Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
14.29Single5WF6UK-4320975WF6-A2A-UK-432097
14.29Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
14.29Single6LI0C176LI0-GPR52-C17
14.29Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
14.29Single6PT3DPI-2876PT3-δ-DPI-287
14.29Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
14.29Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
14.29Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
14.29Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
14.29Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7SK9CCX6627SK9-ACKR3-CCX662
14.29Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
14.29Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
14.29Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
14.29Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
14.29Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
14.29Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
14.29Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
14.29Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
14.29Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
14.29Single8K5BNiacin8K5B-HCA2-Niacin
14.29Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
14.29Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
14.29Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8X5YAstemizole8X5Y-H1-Astemizole
14.29Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
14.29Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
14.29Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
14.29Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
14.29Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
14.29Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
14.29Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
14.29Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
14.29Single9B9Y7DY9B9Y-CB1-7DY
14.29Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
14.29Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
14.29Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
14.29Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
14.29Consensusbradykinin_onOrthosteric Ligandbk2_on
14.29Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
14.29Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
14.29Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
14.29Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
14.29Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
14.29Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
14.29Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
14.29Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.95Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
13.89Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
13.89Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
13.89Single7F8XNN90567F8X-CCKA-NN9056
13.89Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
13.89Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
13.89Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
13.89Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
13.89Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
13.89Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
13.89Single8IEBA1LYA8IEB-GPR156-A1LYA
13.89Single8IEIA1LYA8IEI-GPR156-A1LYA
13.89Single8IEPA1LYA8IEP-GPR156-A1LYA
13.89Single8WKYPG-9348WKY-MC4-PG-934
13.89Single8XWNCXCL88XWN-CXCR2-CXCL8
13.89Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.89Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
13.89Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
13.89Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
13.89Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
13.89Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Consensussomatostatin_offOrthosteric Ligandsst2_off
13.79Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
13.79Single3ODUIT1t3ODU-CXCR4-IT1t
13.79Single4S0VSuvorexant4S0V-OX2-Suvorexant
13.79Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
13.79Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
13.79Single5ZKQABT-4915ZKQ-PAF-ABT-491
13.79Single6AKXA4R6AKX-CCR5-A4R
13.79Single6AKYMaraviroc6AKY-CCR5-Maraviroc
13.79Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
13.79Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
13.79Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
13.79Single6TPJSuvorexant6TPJ-OX2-Suvorexant
13.79Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
13.79Single7F8ULintitript7F8U-CCKA-Lintitript
13.79Single7F8YDevazepide7F8Y-CCKA-Devazepide
13.79Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
13.79Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
13.79Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
13.79Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
13.79Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
13.79Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
13.79Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
13.79Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
13.79Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
13.79Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
13.79Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
13.79Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
13.79Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GNGIstradefylline8GNG-A2A-Istradefylline
13.79Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
13.79Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
13.79Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
13.79Single8IWESpermidine8IWE-TA9-Spermidine
13.79Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
13.79Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
13.79Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
13.79Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
13.79Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
13.79Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
13.79Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
13.79Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
13.79Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
13.79Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
13.79Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
13.79Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
13.79Single8Y0HVUF114188Y0H-CXCR3-VUF11418
13.79Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
13.79Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
13.79Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
13.79Single9BA0A1AKN9BA0-CB1-A1AKN
13.79Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
13.79Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
13.79Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
13.79Consensusangiotensin_offOrthosteric Ligandat1_off
13.79Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
13.79Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
13.79Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
13.79Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
13.79Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
13.79Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
13.79Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
13.79Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
13.79Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
13.79Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
13.79Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
13.64Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
13.51Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
13.51Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
13.51Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
13.51Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
13.51Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
13.51Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
13.51Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
13.51Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
13.51Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
13.51Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
13.51Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
13.51Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
13.51Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
13.33Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
13.33Single2YDOAdenosine2YDO-A2A-Adenosine
13.33Single4MBSMaraviroc4MBS-CCR5-Maraviroc
13.33Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
13.33Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
13.33Single5IU7Q274563465IU7-A2A-Q27456346-Na
13.33Single5IUBQ274563445IUB-A2A-Q27456344-Na
13.33Single5JTBZM-2413855JTB-A2A-ZM-241385
13.33Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
13.33Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
13.33Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
13.33Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
13.33Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
13.33Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
13.33Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
13.33Single6TP3Nemorexant6TP3-OX1-Nemorexant
13.33Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
13.33Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
13.33Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
13.33Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
13.33Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
13.33Single7AROLUF58337ARO-A2A-LUF5833-Na
13.33Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
13.33Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
13.33Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.33Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
13.33Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
13.33Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
13.33Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
13.33Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
13.33Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
13.33Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
13.33Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
13.33Single8IHKAcifran8IHK-HCA3-Acifran
13.33Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
13.33Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
13.33Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
13.33Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
13.33Single8K5CAcipimox8K5C-HCA2-Acipimox
13.33Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
13.33Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
13.33Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.33Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
13.33Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
13.33Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
13.33Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
13.33Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
13.33Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
13.33Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
13.33Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
13.33Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
13.33Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
13.33Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
13.33Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
13.33Consensusa2_offOrthosteric Liganda2a_off
13.33Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
13.33Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
13.33Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
13.33Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
13.33Consensushca_onOrthosteric Ligandhca2_on
13.33Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
13.33Consensusopsins_offOrthosteric Ligandrhodopsin_off
13.33Consensussensory_offOrthosteric Ligandopsins_off
13.16Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
13.16Single6W25SHU91196W25-MC4-SHU9119-Ca
13.16Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
13.16Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
13.16Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
13.16Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
13.16Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.16Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
13.16Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
13.16Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
13.16Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
13.16Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.16Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
12.90Single3EMLZM-2413853EML-A2A-ZM-241385
12.90Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
12.90Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
12.90Single4MQSIperoxo4MQS-M2-Iperoxo
12.90Single4U14Tiotropium4U14-M3-Tiotropium
12.90Single4YAYZD-71554YAY-AT1-ZD-7155
12.90Single5DHHSB-6121115DHH-NOP-SB-612111
12.90Single5DSGTiotropium5DSG-M4-Tiotropium
12.90Single5IU8Q274563475IU8-A2A-Q27456347-Na
12.90Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
12.90Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
12.90Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
12.90Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
12.90Single5T04Neurotensin5T04-NTS1-Neurotensin
12.90Single5UENDU1725UEN-A1-DU172
12.90Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
12.90Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
12.90Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
12.90Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
12.90Single6D27CAY104716D27-DP2-CAY10471
12.90Single6GPSMK08126GPS-CCR2-MK0812
12.90Single6IIVDaltroban6IIV-TP-Daltroban
12.90Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
12.90Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
12.90Single6PS1Timolol6PS1-β2-Timolol
12.90Single6S0LZM-2413856S0L-A2A-ZM-241385
12.90Single6TOTLemborexant6TOT-OX1-Lemborexant
12.90Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
12.90Single7F83PF-051904577F83-Ghrelin-PF-05190457
12.90Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
12.90Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
12.90Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
12.90Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
12.90Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
12.90Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
12.90Single7PYRPSB-21157PYR-A2A-PSB-2115
12.90Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
12.90Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
12.90Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
12.90Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
12.90Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
12.90Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
12.90Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
12.90Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.90Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
12.90Single7YXAONO-54306087YXA-S1P5-ONO-5430608
12.90Single8CU6LJ-45178CU6-A2A-LJ-4517
12.90Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
12.90Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
12.90Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
12.90Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
12.90Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
12.90Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
12.90Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
12.90Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
12.90Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
12.90Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
12.90Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
12.90Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
12.90Single8JXRLSD8JXR-D1-LSD
12.90Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
12.90Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
12.90Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
12.90Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
12.90Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
12.90Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.90Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.90Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.90Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
12.90Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
12.90Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
12.90Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
12.90Single8X63Mepyramine8X63-H1-Mepyramine
12.90Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
12.90Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
12.90Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
12.90Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
12.90Single9CHXS-Carazolol9CHX-β2-S-Carazolol
12.90Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
12.90Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
12.90Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
12.90Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
12.90Consensusa3_onOrthosteric Liganda3a_on
12.90Consensuscck_offOrthosteric Ligandccka_off
12.90Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
12.90Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
12.90Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
12.90Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
12.90Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
12.90Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
12.90Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
12.90Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
12.90Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
12.90Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
12.90Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
12.90Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
12.90Consensushca_on_gpOrthosteric Ligandhca2_on_gp
12.90Consensushistamine_offOrthosteric Ligandh1_off
12.90Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
12.90Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
12.90Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
12.82Single6JODAngiotensin II6JOD-AT2-Angiotensin II
12.82Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
12.82Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
12.82Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
12.82Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
12.82Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
12.82Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
12.50Single4JKVTaladegib4JKV-SMO-Taladegib
12.50Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
12.50Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
12.50Single5CGCHTL142425CGC-mGlu5-HTL14242
12.50Single5IUAQ274563485IUA-A2A-Q27456348-Na
12.50Single5JQHS-Carazolol5JQH-β2-S-Carazolol
12.50Single5TVNLSD5TVN-5-HT2B-LSD
12.50Single5XPRBosentan5XPR-ETB-Bosentan
12.50Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
12.50Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
12.50Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
12.50Single6GPXMK08126GPX-CCR2-MK0812
12.50Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
12.50Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
12.50Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
12.50Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
12.50Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
12.50Single6PS6Timolol6PS6-β2-Timolol
12.50Single6S0QZM-2413856S0Q-A2A-ZM-241385
12.50Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
12.50Single6TP6Filorexant6TP6-OX1-Filorexant
12.50Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
12.50Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
12.50Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
12.50Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
12.50Single7C61Ergotamine7C61-5-HT1B-Ergotamine
12.50Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
12.50Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
12.50Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
12.50Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
12.50Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
12.50Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
12.50Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
12.50Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
12.50Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
12.50Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
12.50Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
12.50Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
12.50Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
12.50Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
12.50Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
12.50Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
12.50Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
12.50Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
12.50Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.50Single8GNEKW-63568GNE-A2A-KW-6356-Na
12.50Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
12.50Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
12.50Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.50Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.50Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
12.50Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
12.50Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
12.50Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
12.50Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
12.50Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
12.50Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
12.50Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
12.50Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
12.50Consensusa3_on_gpOrthosteric Liganda3a_on_gp
12.50Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
12.50Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
12.50Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
12.50Consensusblt_offOrthosteric Ligandblt1_off
12.50Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
12.50Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
12.50Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.50Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
12.50Consensusep_offOrthosteric Ligandep4_off
12.50Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
12.50Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
12.50Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
12.50Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
12.50Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
12.50Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Consensustrace-amine_onOrthosteric Ligandta1_on
12.20Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
12.12Single3P0GBI1671073P0G-β2-BI167107
12.12Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
12.12Single4DJHJDTic4DJH-κ-JDTic
12.12Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
12.12Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
12.12Single4U15Tiotropium4U15-M3-Tiotropium
12.12Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
12.12Single5V54Methiothepin5V54-5-HT1B-Methiothepin
12.12Single5V56TC1145V56-SMO-TC114
12.12Single5V57TC1145V57-SMO-TC114
12.12Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
12.12Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
12.12Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
12.12Single6OL9Tiotropium6OL9-M5-Tiotropium
12.12Single6TQ7SB-3348676TQ7-OX1-SB-334867
12.12Single6WGTLSD6WGT-5-HT2A-LSD
12.12Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
12.12Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
12.12Single7P2L4YI7P2L-mGlu5-4YI
12.12Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
12.12Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
12.12Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
12.12Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
12.12Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
12.12Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
12.12Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
12.12Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
12.12Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
12.12Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
12.12Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
12.12Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
12.12Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
12.12Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
12.12Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
12.12Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
12.12Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
12.12Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.12Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
12.12Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
12.12Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
12.12Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
12.12Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
12.12Consensus5ht1_offOrthosteric Ligand5ht1b_off
12.12Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
12.12Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
12.12Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
12.12Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
12.12Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
12.12Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
12.12Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
12.12Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
12.12Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
12.12Consensusrelaxin_onOrthosteric Ligandrxfp4_on
12.12Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
12.12Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.12Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
12.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
11.90Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
11.76Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
11.76Single4N4WSANT-14N4W-SMO-SANT-1
11.76Single4RWADIPP-NH24RWA-δ-DIPP-NH2
11.76Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
11.76Single5X33BIIL2605X33-BLT1-BIIL260
11.76Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
11.76Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
11.76Single6MXTSalmeterol6MXT-β2-Salmeterol
11.76Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
11.76Single6ZG4HTL00099366ZG4-M1-HTL0009936
11.76Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
11.76Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
11.76Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
11.76Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
11.76Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
11.76Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
11.76Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
11.76Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
11.76Single8JJ8Formoterol8JJ8-β2-Formoterol
11.76Single8JJLOlodaterol8JJL-β2-Olodaterol
11.76Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
11.76Single8XWACXCL18XWA-CXCR2-CXCL1
11.76Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
11.76Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
11.76Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
11.76Consensusalpha1_offOrthosteric Ligandalpha1a_off
11.76Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
11.76Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
11.76Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
11.76Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
11.76Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
11.63Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
11.54Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
11.54Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.54Single8HS2Fab0468HS2-GPR20-Fab046
11.54Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
11.54Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.43Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
11.43Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
11.43Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
11.43Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
11.43Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
11.43Single6K1QIRL25006K1Q-ETB-IRL2500
11.43Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
11.43Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
11.43Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
11.43Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.43Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
11.43Single7UM4AS26747237UM4-5-HT5A-AS2674723
11.43Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
11.43Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
11.43Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.43Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
11.43Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
11.43Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
11.43Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Single8XVJMacitentan8XVJ-ETA-Macitentan
11.43Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
11.43Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
11.43Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
11.43Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
11.43Consensuschemerin_onOrthosteric Ligandcml1_on
11.43Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
11.11Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
11.11Single3OE8IT1t3OE8-CXCR4-IT1t
11.11Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
11.11Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
11.11Single6TQ9SB-4081246TQ9-OX1-SB-408124
11.11Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
11.11Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
11.11Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
11.11Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
11.11Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
11.11Single7XN9L-054,5227XN9-SST2-L-054,522
11.11Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
11.11Single8A2OTheophylline8A2O-A2A-Theophylline-Na
11.11Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
11.11Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
11.11Single8IEIA1LYA8IEI-GPR156-A1LYA
11.11Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
11.11Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
11.11Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
11.11Single8XQJJN2418XQJ-Apelin-JN241
11.11Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
11.11Single9CHUNoradrenaline9CHU-β2-Noradrenaline
11.11Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
11.11Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
11.11Consensusp2y_offOrthosteric Ligandp2y1_off
11.11Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
11.11Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
10.81Single4IARErgotamine4IAR-5-HT1B-Ergotamine
10.81Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
10.81Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
10.81Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
10.81Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
10.81Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.81Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
10.81Single8IEPA1LYA8IEP-GPR156-A1LYA
10.81Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.81Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
10.81Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
10.81Single8KIGSHU91198KIG-MC3-SHU9119-Ca
10.81Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
10.81Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.81Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
10.81Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
10.81Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
10.81Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
10.71Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
10.71Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
10.71Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
10.71Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
10.71Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
10.71Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
10.71Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
10.71Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
10.71Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
10.71Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
10.71Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
10.71Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
10.71Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
10.71Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
10.71Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
10.71Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
10.71Consensus5ht2_onOrthosteric Ligand5ht2b_on
10.71Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
10.53Single8IEBA1LYA8IEB-GPR156-A1LYA
10.53Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
10.53Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
10.34Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
10.34Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
10.34Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
10.34Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
10.34Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
10.34Single4O9RCyclopamine4O9R-SMO-Cyclopamine
10.34Single5L7IVismodegib5L7I-SMO-Vismodegib
10.34Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
10.34Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
10.34Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
10.34Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
10.34Single7SRQLSD7SRQ-5-HT2B-LSD
10.34Single7UL2SR486927UL2-NTS1-SR48692-Na
10.34Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
10.34Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.34Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
10.34Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
10.34Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
10.34Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
10.34Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
10.34Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
10.34Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
10.34Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
10.34Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
10.34Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
10.34Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
10.34Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
10.34Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
10.34Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
10.34Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
10.34Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
10.34Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
10.34Consensusneurotensin_offOrthosteric Ligandnts1_off
10.34Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
10.26Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.26Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.00Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
10.00Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
10.00Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
10.00Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
10.00Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
10.00Single3PWHZM-2413853PWH-A2A-ZM-241385
10.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
10.00Single4QINSAG1.54QIN-SMO-SAG1.5
10.00Single5WS3EMPA5WS3-OX2-EMPA
10.00Single6B73MP11046B73-κ-MP1104
10.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
10.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
10.00Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
10.00Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
10.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
10.00Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
10.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.00Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
10.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
10.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
10.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
10.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
10.00Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
10.00Single7XRRLemborexant7XRR-OX2-Lemborexant
10.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
10.00Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
10.00Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
10.00Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
10.00Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
10.00Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
10.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
10.00Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
10.00Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.00Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
10.00Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
10.00Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
10.00Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
10.00Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
10.00Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
10.00Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
10.00Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
10.00Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
10.00Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
10.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
10.00Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
10.00Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
10.00Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
10.00Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
10.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
10.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
10.00Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.00Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.00Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
10.00Consensusorexin_offOrthosteric Ligandox2_off ox1_off
10.00Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
10.00Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
10.00Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
10.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.00Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
10.00Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
9.76Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
9.76Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
9.76Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
9.68Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
9.68Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
9.68Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
9.68Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
9.68Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
9.68Single4ZJCSB-6740424ZJC-OX1-SB-674042
9.68Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
9.68Single5UVIZM-2413855UVI-A2A-ZM-241385
9.68Single6AQFZM-2413856AQF-A2A-ZM-241385
9.68Single6IQLL7458706IQL-D4-L745870
9.68Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
9.68Single6KUXRS-799486KUX-α2a-RS-79948
9.68Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
9.68Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
9.68Single6MH8ZM-2413856MH8-A2A-ZM-241385
9.68Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
9.68Single6PS0S-Carazolol6PS0-β2-S-Carazolol
9.68Single6PS4ICI118-5516PS4-β2-ICI118-551
9.68Single6PS5S-Propranolol6PS5-β2-S-Propranolol
9.68Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
9.68Single6TPGEMPA6TPG-OX2-EMPA
9.68Single6V9SGTPL114036V9S-OX1-GTPL11403
9.68Single6VI4JDTic6VI4-κ-JDTic
9.68Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
9.68Single6ZG9GSK10347026ZG9-M1-GSK1034702
9.68Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
9.68Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
9.68Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
9.68Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
9.68Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
9.68Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
9.68Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
9.68Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
9.68Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
9.68Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
9.68Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single7UL3Famotidine7UL3-H2-Famotidine
9.68Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
9.68Single7VV6C48/807VV6-MRGPRX2-C48/80
9.68Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.68Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
9.68Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
9.68Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
9.68Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
9.68Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
9.68Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
9.68Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
9.68Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
9.68Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
9.68Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
9.68Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
9.68Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.68Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.68Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
9.68Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
9.68Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
9.68Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
9.68Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
9.68Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
9.68Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
9.68Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
9.68Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
9.68Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
9.68Single8K2WAMG4878K2W-CXCR3-AMG487
9.68Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.68Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
9.68Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
9.68Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.68Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.68Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
9.68Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
9.68Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
9.68Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
9.68Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
9.68Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
9.68Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
9.68Consensusalpha1_onOrthosteric Ligandalpha1a_on
9.68Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
9.68Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
9.68Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
9.68Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
9.68Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
9.68Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
9.68Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
9.68Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.38Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
9.38Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
9.38Single2Y01Dobutamine2Y01-β1-Dobutamine
9.38Single2Y02Carmoterol2Y02-β1-Carmoterol
9.38Single2Y04Salbutamol2Y04-β1-Salbutamol
9.38Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
9.38Single3NY8ICI118-5513NY8-β2-ICI118-551
9.38Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
9.38Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
9.38Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
9.38Single4EJ4Naltrindole4EJ4-δ-Naltrindole
9.38Single4GBRS-Carazolol4GBR-β2-S-Carazolol
9.38Single4QIMANTA XV4QIM-SMO-ANTA XV
9.38Single4QKX35V4QKX-β2-35V
9.38Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
9.38Single5DHGC-355DHG-NOP-C-35
9.38Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
9.38Single5UIGCmpd-15UIG-A2A-Cmpd-1
9.38Single6DRXLisuride6DRX-5-HT2B-Lisuride
9.38Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
9.38Single6H7MSalbutamol6H7M-β1-Salbutamol
9.38Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
9.38Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
9.38Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
9.38Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
9.38Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
9.38Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
9.38Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
9.38Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
9.38Single7BU7BI1671077BU7-β1-BI167107
9.38Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
9.38Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
9.38Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
9.38Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
9.38Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
9.38Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
9.38Single7UL4Alvimopan7UL4-μ-Alvimopan
9.38Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
9.38Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
9.38Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
9.38Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
9.38Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
9.38Single7WC7Lisuride7WC7-5-HT2A-Lisuride
9.38Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
9.38Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
9.38Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
9.38Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
9.38Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
9.38Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
9.38Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
9.38Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
9.38Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
9.38Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
9.38Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
9.38Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
9.38Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
9.38Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
9.38Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
9.38Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
9.38Single8JJOAlprenolol8JJO-β2-Alprenolol
9.38Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
9.38Single8K5DGSK2560738K5D-HCA2-GSK256073
9.38Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
9.38Single8RLNLUF58348RLN-A2A-LUF5834
9.38Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
9.38Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.38Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
9.38Single8X64Desloratadine8X64-H1-Desloratadine
9.38Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
9.38Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
9.38Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
9.38Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
9.38Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
9.38Consensus5ht5_onOrthosteric Ligand5ht5a_on
9.38Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
9.38Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
9.38Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
9.38Consensusalpha2_onOrthosteric Ligandalpha2b_on
9.38Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
9.38Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
9.38Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
9.38Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
9.38Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
9.38Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
9.38Consensusblt_onOrthosteric Ligandblt1_on
9.38Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
9.38Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
9.38Consensusdopamine_offOrthosteric Ligandd2_off d3_off
9.38Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
9.38Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
9.38Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
9.38Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
9.38Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
9.38Consensusleukotriene_onOrthosteric Ligandblt_on
9.38Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
9.38Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
9.09Single2RH1S-Carazolol2RH1-β2-S-Carazolol
9.09Single2Y00Dobutamine2Y00-β1-Dobutamine
9.09Single2Y03Isoprenaline2Y03-β1-Isoprenaline
9.09Single2YCWS-Carazolol2YCW-β1-S-Carazolol
9.09Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
9.09Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
9.09Single5D6LS-Carazolol5D6L-β2-S-Carazolol
9.09Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
9.09Single5WIUNemonapride5WIU-D4-Nemonapride
9.09Single5WIVNemonapride5WIV-D4-Nemonapride-Na
9.09Single5WQCEMPA5WQC-OX2-EMPA
9.09Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
9.09Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
9.09Single6E67BI1671076E67-β2-BI167107-Gs (fused)
9.09Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
9.09Single6LUQHaloperidol6LUQ-D2-Haloperidol
9.09Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
9.09Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
9.09Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
9.09Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
9.09Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
9.09Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
9.09Single7SINNPS-21437SIN-CaS-NPS-2143
9.09Single7SINNPS-21437SIN-CaS-NPS-2143
9.09Single7W41PD1762527W41-BB2-PD176252
9.09Single7WC6LSD7WC6-5-HT2A-LSD
9.09Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
9.09Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
9.09Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
9.09Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
9.09Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
9.09Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
9.09Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
9.09Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
9.09Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
9.09Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
9.09Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
9.09Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
9.09Single8ZMFA1L108ZMF-5-HT2C-A1L10
9.09Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
9.09Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
9.09Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
9.09Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
9.09Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
9.09Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
9.09Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
9.09Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
9.09Consensusamine_offonOrthosteric Ligandamine_off amine_on
9.09Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
9.09Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
9.09Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
9.09Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
9.09Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
9.09Consensusbombesin_offOrthosteric Ligandbb2_off
9.09Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
9.09Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
9.09Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
9.09Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
8.82Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
8.82Single5D5AS-Carazolol5D5A-β2-S-Carazolol
8.82Single5D5BS-Carazolol5D5B-β2-S-Carazolol
8.82Single5TZRMK86665TZR-FFA1-MK8666
8.82Single6H7JIsoprenaline6H7J-β1-Isoprenaline
8.82Single6J21Aprepitant6J21-NK1-Aprepitant
8.82Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
8.82Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
8.82Single7B6WCyclazosin7B6W-α1b-Cyclazosin
8.82Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
8.82Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
8.82Single7R0CAVP7R0C-V2-AVP-Arrestin2
8.82Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
8.82Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
8.82Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
8.82Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
8.82Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
8.82Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
8.82Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
8.82Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
8.82Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
8.82Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
8.82Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
8.82Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
8.82Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
8.82Single8XVLZibotentan8XVL-ETA-Zibotentan
8.82Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
8.82Single9BJKNAM9BJK-μ-Naloxone-NAM
8.82Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
8.82Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
8.82Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
8.82Consensusa2_onOrthosteric Liganda2b_on
8.82Consensusa2_on_gpOrthosteric Liganda2b_on_gp
8.82Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
8.82Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
8.82Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
8.82Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
8.82Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
8.82Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
8.82Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
8.82Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
8.82Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
8.82Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
8.82Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
8.82Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
8.82Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
8.82Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
8.82Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
8.57Single3D4STimolol3D4S-β2-Timolol
8.57Single4AMIBucindolol4AMI-β1-Bucindolol
8.57Single4LDEBI1671074LDE-β2-BI167107
8.57Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
8.57Single4PY02MeSATP4PY0-P2Y12-2MeSATP
8.57Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
8.57Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
8.57Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
8.57Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
8.57Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
8.57Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
8.57Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
8.57Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
8.57Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.57Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
8.57Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
8.57Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
8.57Single8JWY2-1188JWY-A2A-2-118
8.57Single8JWZAB9288JWZ-A2A-AB928-Na
8.57Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.57Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
8.57Single8XQJJN2418XQJ-Apelin-JN241
8.57Single8XYIVUF106618XYI-CXCR3-VUF10661
8.57Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
8.57Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
8.57Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
8.57Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
8.57Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
8.57Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
8.57Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
8.57Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.57Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.33Single6H7LDobutamine6H7L-β1-Dobutamine
8.33Single6IBLArformoterol6IBL-β1-Arformoterol
8.33Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
8.33Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
8.33Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
8.33Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
8.33Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
8.33Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
8.33Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
8.33Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
8.11Single6KNMJN241-96KNM-Apelin-JN241-9
8.11Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
8.11Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
8.11Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
8.11Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
8.11Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
8.11Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
8.11Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.11Consensuskisspeptin_onOrthosteric Ligandkiss1_on
7.89Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
7.89Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
7.89Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
7.89Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
7.89Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
7.89Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
7.89Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
7.69Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
7.69Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
7.69Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
7.41Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
7.41Single7WC4Serotonin7WC4-5-HT2A-Serotonin
7.41Single8PWNTheophylline8PWN-A2A-Theophylline
7.41Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
7.14Single3RFMCaffeine3RFM-A2A-Caffeine
7.14Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
7.14Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
7.14Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
7.14Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
7.14Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
7.14Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
7.14Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
7.14Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
6.90Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
6.90Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
6.90Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
6.90Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
6.90Single6ME5Agomelatine6ME5-MT1-Agomelatine
6.90Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
6.90Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
6.90Single7V6A-7V6A-M4-PubChem 9864275-Gi1/β1/γ2
6.90Single7WC5Psilocin7WC5-5-HT2A-Psilocin
6.90Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.90Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
6.90Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
6.90Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
6.90Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
6.90Single8JPSCCL78JPS-ACKR1-CCL7
6.90Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
6.90Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
6.90Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
6.90Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
6.90Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
6.90Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
6.90Consensusgi_sensoryOrthosteric Ligandgi_opsins
6.90Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
6.90Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
6.90Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
6.67Single3PBLEticlopride3PBL-D3-Eticlopride
6.67Single6HLLCP999946HLL-NK1-CP99994
6.67Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
6.67Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
6.67Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
6.67Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
6.67Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
6.67Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
6.67Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
6.67Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
6.67Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
6.67Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
6.67Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
6.67Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.67Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.67Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
6.67Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
6.67Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
6.45Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
6.45Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
6.45Single6ME2Ramelteon6ME2-MT1-Ramelteon
6.45Single6ME9Ramelteon6ME9-MT2-Ramelteon
6.45Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
6.45Single6TODEMPA6TOD-OX1-EMPA-Na
6.45Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
6.45Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
6.45Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
6.45Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
6.45Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
6.45Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
6.45Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.45Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
6.45Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
6.45Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
6.45Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.45Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.45Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
6.45Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
6.45Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
6.45Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
6.45Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
6.45Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
6.45Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
6.45Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
6.45Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
6.45Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
6.25Single3REYXAC3REY-A2A-XAC
6.25Single3RZECidoxepin3RZE-H1-Cidoxepin
6.25Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
6.25Single6A94Zotepine6A94-5-HT2A-Zotepine
6.25Single6FFIMMPEP6FFI-mGlu5-MMPEP
6.25Single6TPNHTL66416TPN-OX2-HTL6641
6.25Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
6.25Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
6.25Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
6.25Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
6.25Single7VODCariprazine7VOD-5-HT2A-Cariprazine
6.25Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
6.25Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
6.25Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
6.25Single8JD6N-(3-chlorophenyl)pyridine-2-carboxamide8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
6.25Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
6.25Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
6.25Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
6.25Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
6.25Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
6.25Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
6.25Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
6.25Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
6.25Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
6.25Single9BJKNaloxone9BJK-μ-Naloxone-NAM
6.25Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
6.25Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
6.06Single6FFHFenobam6FFH-mGlu5-Fenobam
6.06Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
6.06Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
6.06Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.06Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
6.06Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
6.06Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
6.06Single9IYAONO-97105319IYA-GPR55-ONO-9710531
6.06Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
6.06Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
6.06Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
6.06Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
5.88Single4NTJAZD12834NTJ-P2Y12-AZD1283
5.88Single6HLPNetupitant6HLP-NK1-Netupitant
5.88Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
5.88Single6Z4SSR486926Z4S-NTS1-SR48692
5.88Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
5.88Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.88Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
5.88Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
5.88Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
5.88Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
5.88Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
5.88Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
5.88Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
5.88Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
5.71Single6E59L-7607356E59-NK1-L-760735
5.71Single6J20Aprepitant6J20-NK1-Aprepitant
5.71Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
5.71Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
5.71Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
5.71Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.71Consensustachykinin_offOrthosteric Ligandnk1_off
5.56Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
5.56Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
5.56Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.56Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.56Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
5.56Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.41Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
5.41Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
5.13Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
5.00Single7SHEPI; PE7SHE-GPR158-PI; PE
4.17Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.17Single6D35Cholesterol6D35-SMO-Cholesterol
4.17Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.17Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.17Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.17Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.17Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
4.17Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
4.17Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
4.17Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
4.17Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.17Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
4.17Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.17Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.17Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.17Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.17Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.17Single7DTTCa7DTT-CaS-Ca-Ca
4.17Single7DTTCa7DTT-CaS-Ca-Ca
4.17Single7DTUTryptophan7DTU-CaS-Tryptophan
4.17Single7DTUTryptophan7DTU-CaS-Tryptophan
4.17Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.17Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.17Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.17Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.17Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.17Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.17Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.17Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.17Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.17Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.17Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.17Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.17Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.17Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.17Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.17Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.17Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.17Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.17Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.17Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.17Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.17Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.17Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.17Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.17Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.17Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.17Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.17Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.17Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.17Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.17Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
4.17Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.17Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.17Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.17Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.17Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.17Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.17Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.17Single7XW7K1-707XW7-TSH-K1-70
4.17Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.17Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.17Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.17Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.17Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.17Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.17Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.17Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.17Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.17Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.17Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.17Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.17Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.17Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.17Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.17Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.17Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.17Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
4.17Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
4.17Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.17Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.17Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
4.17Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
4.17Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.17Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.17Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.17Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.17Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.17Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
4.17Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
4.17Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
4.17Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
4.17Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
4.17Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
4.17Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.17Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.17Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.17Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.17Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.17Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.17Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.17Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.17Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.17Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.17Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.17Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.17Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.17Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.17Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.17Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.17Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.17Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
4.17Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
4.17Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.17Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
4.17Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
4.17Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.17Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.17Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.17Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.17Single8WVXNorrin8WVX-LGR4-Norrin
4.17Single8WVYNorrin8WVY-LGR4-Norrin
4.17Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.17Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.17Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.17Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.17Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.17Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.17Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.17Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.17Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.17Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.17Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.17Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.17Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.17Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.17Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.17Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.17Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.17Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.17Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.17Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.17Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.17Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.17Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.17Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.17Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.17Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.17Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.00Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.00Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.85Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
3.85Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
3.85Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
3.85Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
3.70Single5MZPCaffeine5MZP-A2A-Caffeine-Na
3.70Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
3.70Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
3.70Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
3.70Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
3.70Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.70Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
3.57Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
3.57Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
3.57Single5L7DCholesterol5L7D-SMO-Cholesterol
3.57Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
3.57Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.57Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
3.57Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
3.57Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.45Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
3.45Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
3.45Consensussensory_onOrthosteric Ligandopsins_on
3.33Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
3.33Single3UZAGTPL92363UZA-A2A-GTPL9236
3.33Single8ZPLCholesterol8ZPL-CXCR4-HF51116-Cholesterol
3.33Single8ZPMCholesterol8ZPM-CXCR4-AMD070-Cholesterol
3.33Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
3.33Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
3.33Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
3.23Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
3.23Single6TP4ACT-4622066TP4-OX1-ACT-462206
3.23Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
3.23Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
3.23Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.23Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
3.23Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
3.23Single8HNNSCH5467388HNN-CXCR3-SCH546738
3.23Consensusgq_nucleotideOrthosteric Ligandgq_p2y
3.23Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
3.12Single4K5YCP-3763954K5Y-CRF1-CP-376395
3.12Single4XNVBPTU4XNV-P2Y1-BPTU
3.12Single6C1QNDT95137276C1Q-C5a1-PMX53-NDT9513727
3.12Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
3.12Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
3.03Single6TPKRetosiban6TPK-OT-Retosiban
3.03Single6ZINSR486926ZIN-NTS1-SR48692
3.03Single8IYXYL-3658IYX-GPR34-YL-365
3.03Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
3.03Consensusvasop-oxy_offOrthosteric Ligandot_off
2.94Single4Z9GCP-3763954Z9G-CRF1-CP-376395
2.94Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
2.94Single8GTIBMK-C2058GTI-CRF1-BMK-C205
2.94Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
2.86Single8GTGBMK-I1528GTG-CRF1-BMK-I152
2.86Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
2.70Single8GTMBMK-C2038GTM-CRF1-BMK-C203
2.50Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.50Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.44Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
2.38Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.38Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.33Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.17Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

PDB Summary
PDB 7VVL
Class B1
SubFamily Peptide
Type Parathyroid Hormone
SubType PTH1
Species Homo Sapiens
Ligand PTH
Other Ligand(s) -
Protein Partners Gs/Beta1/Gamma2
PDB Resolution 2.8
Date 2022-08-03
D.O.I. 10.1016/j.molcel.2022.07.003
Net Summary
Imin 3.2
Number of Linked Nodes 944
Number of Links 1214
Number of Hubs 230
Number of Links mediated by Hubs 816
Number of Communities 32
Number of Nodes involved in Communities 344
Number of Links involved in Communities 516
Path Summary
Number Of Nodes in MetaPath 93
Number Of Links MetaPath 92
Number of Shortest Paths 6982621
Length Of Smallest Path 3
Average Path Length 41.9822
Length of Longest Path 73
Minimum Path Strength 1.395
Average Path Strength 7.64966
Maximum Path Strength 25.49
Minimum Path Correlation 0.7
Average Path Correlation 0.99688
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.32558
Average % Of Corr. Nodes 47.5143
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 59.234
Maximum Path Hubs % 100
AnnotationTypeLinks
Gene OntologyMolecular Function• binding   • guanyl nucleotide binding   • GTP binding   • nucleotide binding   • guanyl ribonucleotide binding   • purine ribonucleotide binding   • purine ribonucleoside triphosphate binding   • nucleoside phosphate binding   • ion binding   • purine nucleotide binding   • anion binding   • heterocyclic compound binding   • carbohydrate derivative binding   • ribonucleotide binding   • small molecule binding   • D1 dopamine receptor binding   • protein binding   • signaling receptor binding   • G protein-coupled receptor binding   • dopamine receptor binding   • protein-containing complex binding   • G-protein beta/gamma-subunit complex binding   • pyrophosphatase activity   • GTPase activity   • G protein activity   • ribonucleoside triphosphate phosphatase activity   • molecular function regulator activity   • hydrolase activity, acting on acid anhydrides, in phosphorus-containing anhydrides   • hydrolase activity   • hydrolase activity, acting on acid anhydrides   • catalytic activity   • enzyme regulator activity   • molecular function activator activity   • phosphorus-oxygen lyase activity   • cyclase regulator activity   • enzyme activator activity   • cyclase activator activity   • cyclase activity   • adenylate cyclase regulator activity   • lyase activity   • adenylate cyclase activator activity   • adenylate cyclase activity   • cation binding   • metal ion binding   • developmental process   • multicellular organismal process   • epithelium development   • ectodermal placode morphogenesis   • epidermis development   • molting cycle process   • hair cycle   • animal organ development   • hair follicle placode formation   • tissue development   • ectodermal placode formation   • anatomical structure morphogenesis   • skin development   • skin epidermis development   • hair follicle development
Gene OntologyBiological Process• developmental process   • multicellular organismal process   • epithelium development   • ectodermal placode morphogenesis   • epidermis development   • molting cycle process   • hair cycle   • animal organ development   • hair follicle placode formation   • tissue development   • ectodermal placode formation   • anatomical structure morphogenesis   • skin development   • skin epidermis development   • hair follicle development   • molting cycle   • anatomical structure development   • anatomical structure formation involved in morphogenesis   • ectodermal placode development   • hair cycle process   • system process   • sensory perception of chemical stimulus   • sensory perception   • nervous system process   • sensory perception of smell   • cellular response to stimulus   • cellular response to nitrogen compound   • response to stimulus   • response to endogenous stimulus   • response to peptide hormone   • cellular response to peptide hormone stimulus   • response to oxygen-containing compound   • response to nitrogen compound   • response to glucagon   • cellular response to oxygen-containing compound   • cellular response to glucagon stimulus   • cellular response to endogenous stimulus   • cellular response to chemical stimulus   • response to hormone   • response to chemical   • cellular process   • cellular response to hormone stimulus   • multicellular organism development   • skeletal system development   • bone development   • system development   • regulation of body fluid levels   • wound healing   • homotypic cell-cell adhesion   • cell activation   • hemostasis   • biological regulation   • platelet aggregation   • blood coagulation   • cell adhesion   • cell-cell adhesion   • response to stress   • coagulation   • regulation of biological quality   • response to wounding   • platelet activation   • response to fluid shear stress   • vascular endothelial cell response to laminar fluid shear stress   • response to laminar fluid shear stress   • cellular response to stress   • cellular response to laminar fluid shear stress   • vascular endothelial cell response to fluid shear stress   • cellular response to fluid shear stress   • cognition   • developmental growth   • growth   • response to ketone   • response to prostaglandin   • response to lipid   • response to alcohol   • cellular response to prostaglandin stimulus   • cellular response to prostaglandin E stimulus   • cellular response to alcohol   • cellular response to lipid   • response to prostaglandin E   • cellular response to ketone   • regulation of biological process   • regulation of cellular process   • signaling   • adenylate cyclase-activating G protein-coupled receptor signaling pathway   • cell communication   • adenylate cyclase-modulating G protein-coupled receptor signaling pathway   • G protein-coupled receptor signaling pathway   • signal transduction   • homeostatic process   • positive regulation of biological process   • adaptive thermogenesis   • positive regulation of metabolic process   • multicellular organismal-level homeostasis   • regulation of cold-induced thermogenesis   • cold-induced thermogenesis   • temperature homeostasis   • positive regulation of cold-induced thermogenesis   • positive regulation of multicellular organismal process   • metabolic process   • regulation of multicellular organismal process   • regulation of metabolic process   • positive regulation of cellular process   • protein localization   • regulation of localization   • establishment of protein localization   • nitrogen compound transport   • localization   • cellular macromolecule localization   • regulation of peptide hormone secretion   • regulation of hormone levels   • establishment of protein localization to extracellular region   • protein secretion   • establishment of localization   • regulation of protein secretion   • regulation of secretion   • cellular localization   • regulation of hormone secretion   • regulation of protein localization   • regulation of peptide secretion   • transport   • hormone secretion   • protein localization to extracellular region   • peptide secretion   • regulation of secretion by cell   • secretion by cell   • amide transport   • signal release   • regulation of signaling   • regulation of transport   • secretion   • regulation of peptide transport   • regulation of establishment of protein localization   • export from cell   • cell-cell signaling   • regulation of protein transport   • peptide transport   • protein transport   • regulation of cellular localization   • regulation of insulin secretion   • peptide hormone secretion   • macromolecule localization   • hormone transport   • regulation of cell communication   • insulin secretion   • adenylate cyclase-activating adrenergic receptor signaling pathway   • adrenergic receptor signaling pathway   • establishment of localization in cell   • intracellular transport   • regulation of defense response   • regulation of response to external stimulus   • negative regulation of inflammatory response   • negative regulation of biological process   • inflammatory response to antigenic stimulus   • regulation of response to stress   • regulation of immune system process   • negative regulation of inflammatory response to antigenic stimulus   • defense response   • immune response   • negative regulation of response to stimulus   • negative regulation of immune response   • regulation of inflammatory response to antigenic stimulus   • response to external stimulus   • regulation of inflammatory response   • regulation of response to stimulus   • negative regulation of immune system process   • immune system process   • negative regulation of response to external stimulus   • negative regulation of defense response   • regulation of immune response   • inflammatory response   • positive regulation of adenylate cyclase activity   • positive regulation of molecular function   • regulation of molecular function   • positive regulation of cyclase activity   • activation of adenylate cyclase activity   • regulation of adenylate cyclase activity   • regulation of catalytic activity   • positive regulation of catalytic activity   • positive regulation of lyase activity   • response to dopamine   • cellular response to dopamine   • response to monoamine   • response to catecholamine   • adenylate cyclase-activating dopamine receptor signaling pathway   • cellular response to catecholamine stimulus   • G protein-coupled dopamine receptor signaling pathway   • cellular response to monoamine stimulus   • renal system process   • chemical homeostasis   • multicellular organismal-level water homeostasis   • multicellular organismal-level chemical homeostasis   • renal water homeostasis   • cellular anatomical structure   • membrane   • protein-containing complex   • extrinsic component of plasma membrane   • catalytic complex   • plasma membrane protein complex   • cytoplasmic side of membrane   • plasma membrane   • membrane protein complex   • heterotrimeric G-protein complex   • side of membrane   • cell periphery   • cytoplasmic side of plasma membrane   • GTPase complex
Gene OntologyCellular Component• cellular anatomical structure   • membrane   • protein-containing complex   • extrinsic component of plasma membrane   • catalytic complex   • plasma membrane protein complex   • cytoplasmic side of membrane   • plasma membrane   • membrane protein complex   • heterotrimeric G-protein complex   • side of membrane   • cell periphery   • cytoplasmic side of plasma membrane   • GTPase complex   • extrinsic component of membrane   • extrinsic component of cytoplasmic side of plasma membrane   • extracellular exosome   • membrane-bounded organelle   • extracellular vesicle   • extracellular organelle   • extracellular region   • organelle   • extracellular space   • vesicle   • extracellular membrane-bounded organelle   • intracellular anatomical structure   • cytoplasm   • cytosol   • Golgi apparatus subcompartment   • Golgi apparatus   • organelle subcompartment   • trans-Golgi network membrane   • intracellular membrane-bounded organelle   • endomembrane system   • intracellular organelle   • trans-Golgi network   • organelle membrane   • cytoskeletal protein binding   • spectrin binding   • protein-containing complex binding   • protein binding   • binding   • enzyme binding   • GTPase binding   • phosphoric ester hydrolase activity   • alkylglycerophosphoethanolamine phosphodiesterase activity   • hydrolase activity, acting on ester bonds   • phosphoric diester hydrolase activity   • hydrolase activity   • catalytic activity   • pyrophosphatase activity   • GTPase activity   • ribonucleoside triphosphate phosphatase activity   • hydrolase activity, acting on acid anhydrides, in phosphorus-containing anhydrides   • hydrolase activity, acting on acid anhydrides   • signaling receptor complex adaptor activity   • protein-macromolecule adaptor activity   • molecular adaptor activity   • signaling adaptor activity   • positive regulation of cytosolic calcium ion concentration   • biological regulation   • regulation of biological quality   • multicellular organismal process   • system process   • sensory perception of chemical stimulus   • sensory perception   • nervous system process   • sensory perception of taste   • developmental process   • sensory organ development   • eye development   • animal organ development   • retina development in camera-type eye   • visual system development   • multicellular organism development   • camera-type eye development   • anatomical structure development   • sensory system development   • system development   • response to decreased oxygen levels   • cellular response to stimulus   • response to stimulus   • cellular response to oxygen levels   • cellular response to hypoxia   • cellular response to decreased oxygen levels   • cellular response to chemical stimulus   • cellular response to stress   • response to hypoxia   • response to stress   • response to chemical   • response to oxygen levels   • response to abiotic stimulus   • cellular process   • cell population proliferation   • regulation of biological process   • regulation of cellular process   • signaling   • phospholipase C-activating G protein-coupled receptor signaling pathway   • cell communication   • G protein-coupled receptor signaling pathway   • signal transduction   • muscle cell apoptotic process   • striated muscle cell apoptotic process   • apoptotic process   • cell death   • programmed cell death   • cardiac muscle cell apoptotic process   • photoreceptor inner segment   • somatodendritic compartment   • cell projection   • dendrite   • dendritic tree   • neuron projection   • plasma membrane bounded cell projection   • non-motile cilium   • 9+0 non-motile cilium   • cilium   • photoreceptor outer segment   • photoreceptor cell cilium   • ciliary membrane   • photoreceptor outer segment membrane   • bounding membrane of organelle   • plasma membrane region   • cell projection membrane   • synapse   • cell junction   • cell body   • G-protein beta-subunit binding   • cellular response to nitrogen compound   • response to dopamine   • cellular response to dopamine   • response to monoamine   • response to catecholamine   • adenylate cyclase-activating dopamine receptor signaling pathway   • cellular response to catecholamine stimulus   • G protein-coupled dopamine receptor signaling pathway   • response to oxygen-containing compound   • response to nitrogen compound   • adenylate cyclase-activating G protein-coupled receptor signaling pathway   • cellular response to oxygen-containing compound   • cellular response to monoamine stimulus   • adenylate cyclase-modulating G protein-coupled receptor signaling pathway   • response to ketone   • response to prostaglandin   • response to lipid   • response to endogenous stimulus   • response to alcohol   • cellular response to prostaglandin stimulus   • cellular response to endogenous stimulus   • cellular response to prostaglandin E stimulus   • cellular response to alcohol   • response to hormone   • cellular response to lipid   • response to prostaglandin E   • cellular response to ketone   • cellular response to hormone stimulus   • parathyroid hormone receptor binding   • signaling receptor binding   • G protein-coupled receptor binding   • type 1 parathyroid hormone receptor binding   • molecular transducer activity   • molecular function activator activity   • signaling receptor activity   • molecular function regulator activity   • signaling receptor regulator activity   • receptor ligand activity   • signaling receptor activator activity   • peptide hormone receptor binding   • hormone receptor binding   • hormone activity   • response to xenobiotic stimulus   • response to parathyroid hormone   • magnesium ion homeostasis   • inorganic ion homeostasis   • chemical homeostasis   • homeostatic process   • monoatomic ion homeostasis   • monoatomic cation homeostasis   • ossification   • bone mineralization   • biomineral tissue development   • tissue development   • multicellular organismal-level homeostasis   • homeostasis of number of cells within a tissue   • anatomical structure homeostasis   • tissue homeostasis   • homeostasis of number of cells   • biosynthetic process   • metabolic process   • macromolecule metabolic process   • macromolecule biosynthetic process   • skeletal system development   • regulation of biosynthetic process   • positive regulation of biological process   • regulation of macromolecule metabolic process   • gene expression   • positive regulation of macromolecule biosynthetic process   • regulation of gene expression   • positive regulation of metabolic process   • positive regulation of gene expression   • positive regulation of biosynthetic process   • regulation of macromolecule biosynthetic process   • positive regulation of macromolecule metabolic process   • regulation of metabolic process   • positive regulation of cellular process   • RNA metabolic process   • primary metabolic process   • nucleobase-containing compound biosynthetic process   • nucleic acid metabolic process   • RNA biosynthetic process   • nucleobase-containing compound metabolic process   • DNA-templated transcription   • nucleic acid biosynthetic process   • transcription by RNA polymerase II   • negative regulation of apoptotic process in bone marrow cell   • negative regulation of programmed cell death   • apoptotic process in bone marrow cell   • regulation of apoptotic process in bone marrow cell   • regulation of apoptotic process   • negative regulation of biological process   • regulation of programmed cell death   • negative regulation of apoptotic process   • negative regulation of cellular process   • regulation of generation of precursor metabolites and energy   • regulation of primary metabolic process   • positive regulation of glycogen metabolic process   • regulation of small molecule metabolic process   • small molecule metabolic process   • carbohydrate biosynthetic process   • hexose metabolic process   • positive regulation of glucose metabolic process   • positive regulation of glycogen biosynthetic process   • energy reserve metabolic process   • positive regulation of carbohydrate metabolic process   • regulation of glycogen metabolic process   • monosaccharide metabolic process   • regulation of glycogen biosynthetic process   • glucan biosynthetic process   • energy derivation by oxidation of organic compounds   • regulation of glucan biosynthetic process   • regulation of polysaccharide metabolic process   • polysaccharide metabolic process   • glucan metabolic process   • regulation of carbohydrate metabolic process   • regulation of glucose metabolic process   • carbohydrate metabolic process   • polysaccharide biosynthetic process   • glycogen metabolic process   • generation of precursor metabolites and energy   • glycogen biosynthetic process   • regulation of polysaccharide biosynthetic process   • regulation of carbohydrate biosynthetic process   • positive regulation of small molecule metabolic process   • glucose metabolic process   • phosphate ion homeostasis   • cell-cell signaling   • intracellular calcium ion homeostasis   • calcium ion homeostasis   • cellular homeostasis   • intracellular monoatomic cation homeostasis   • intracellular chemical homeostasis   • intracellular monoatomic ion homeostasis   • regulation of developmental process   • regulation of biomineral tissue development   • regulation of bone mineralization   • positive regulation of ossification   • positive regulation of developmental process   • positive regulation of biomineral tissue development   • regulation of multicellular organismal process   • regulation of multicellular organismal development   • positive regulation of bone mineralization   • positive regulation of multicellular organismal process   • regulation of ossification   • response to ethanol   • response to metal ion   • response to lead ion   • positive regulation of cell population proliferation   • positive regulation of cell proliferation in bone marrow   • cell proliferation in bone marrow   • regulation of cell proliferation in bone marrow   • regulation of cell population proliferation   • response to nutrient levels   • response to vitamin D   • response to nutrient   • response to vitamin   • hormone-mediated signaling pathway   • apoptotic signaling pathway   • hormone-mediated apoptotic signaling pathway   • nucleoside phosphate metabolic process   • ribose phosphate metabolic process   • cAMP metabolic process   • cyclic purine nucleotide metabolic process   • carbohydrate derivative metabolic process   • nucleotide metabolic process   • cyclic nucleotide metabolic process   • purine-containing compound metabolic process   • purine nucleotide metabolic process   • ribonucleotide metabolic process   • organophosphate metabolic process   • nucleobase-containing small molecule metabolic process   • phosphate-containing compound metabolic process   • purine ribonucleotide metabolic process   • phosphorus metabolic process   • regulation of cartilage development   • regulation of chondrocyte differentiation   • connective tissue development   • cellular developmental process   • negative regulation of cartilage development   • negative regulation of chondrocyte differentiation   • regulation of cell differentiation   • cell differentiation   • negative regulation of cell differentiation   • negative regulation of developmental process   • chondrocyte differentiation   • negative regulation of multicellular organismal process   • cartilage development   • negative regulation of metabolic process   • negative regulation of gene expression   • negative regulation of biosynthetic process   • negative regulation of macromolecule biosynthetic process   • negative regulation of macromolecule metabolic process   • regulation of localization   • hexose transmembrane transport   • D-glucose import   • transport   • carbohydrate transport   • positive regulation of D-glucose transmembrane transport   • localization   • positive regulation of transmembrane transport   • regulation of D-glucose import   • positive regulation of D-glucose import   • regulation of transport   • establishment of localization   • transmembrane transport   • regulation of transmembrane transport   • positive regulation of transport   • D-glucose transmembrane transport   • regulation of D-glucose transmembrane transport   • monosaccharide transmembrane transport   • carbohydrate transmembrane transport   • positive regulation of cell communication   • regulation of signaling   • positive regulation of signal transduction   • regulation of signal transduction   • positive regulation of response to stimulus   • regulation of response to stimulus   • regulation of cell communication   • positive regulation of signaling   • response to cadmium ion   • small GTPase-mediated signal transduction   • Rho protein signal transduction   • intracellular signal transduction   • intracellular signaling cassette   • regulation of leukocyte proliferation   • osteoclast proliferation   • regulation of osteoclast proliferation   • positive regulation of osteoclast proliferation   • leukocyte proliferation   • positive regulation of leukocyte proliferation   • bone maturation   • regulation of bone mineralization involved in bone maturation   • negative regulation of biomineral tissue development   • negative regulation of bone mineralization   • ossification involved in bone maturation   • bone development   • bone mineralization involved in bone maturation   • developmental maturation   • negative regulation of bone mineralization involved in bone maturation   • negative regulation of ossification   • anatomical structure maturation   • animal organ maturation   • positive regulation of DNA-templated transcription   • regulation of RNA metabolic process   • regulation of nucleobase-containing compound metabolic process   • regulation of RNA biosynthetic process   • regulation of transcription by RNA polymerase II   • positive regulation of nucleobase-containing compound metabolic process   • positive regulation of transcription by RNA polymerase II   • positive regulation of RNA metabolic process   • positive regulation of RNA biosynthetic process   • regulation of DNA-templated transcription   • regulation of inositol phosphate biosynthetic process   • alcohol metabolic process   • positive regulation of phosphate metabolic process   • inositol phosphate metabolic process   • regulation of phosphate metabolic process   • polyol biosynthetic process   • polyol metabolic process   • positive regulation of phosphorus metabolic process   • regulation of alcohol biosynthetic process   • small molecule biosynthetic process   • positive regulation of inositol phosphate biosynthetic process   • organophosphate biosynthetic process   • inositol phosphate biosynthetic process   • alcohol biosynthetic process   • regulation of phosphorus metabolic process   • positive regulation of alcohol biosynthetic process   • tissue remodeling   • bone remodeling   • bone resorption   • response to fibroblast growth factor   • response to growth factor   • identical protein binding   • protein homodimerization activity   • protein dimerization activity   • amide binding   • peptide hormone binding   • hormone binding   • peptide receptor activity   • G protein-coupled receptor activity   • G protein-coupled peptide receptor activity   • transmembrane signaling receptor activity   • parathyroid hormone receptor activity   • osteoblast development   • cell development   • osteoblast differentiation   • embryo development ending in birth or egg hatching   • chordate embryonic development   • embryo development   • in utero embryonic development   • cell maturation   • cell surface receptor signaling pathway   • negative regulation of cell population proliferation   • G protein-coupled receptor signaling pathway, coupled to cyclic nucleotide second messenger   • nucleus   • membrane-enclosed lumen   • intracellular membraneless organelle   • nucleolus   • intracellular organelle lumen   • organelle lumen   • membraneless organelle   • nuclear lumen   • apical part of cell   • apical plasma membrane   • basal part of cell   • basal plasma membrane   • basolateral plasma membrane   • receptor complex
SCOP2Domain Identifier• Transducin (heterotrimeric G protein), gamma chain   • G protein-coupled receptor-like
SCOP2Family Identifier• Transducin (heterotrimeric G protein), gamma chain   • G protein-coupled receptor-like
Membrane Protein Annotations-• Orientations of Proteins in Membranes database (OPM)   • Protein Data Bank of Transmembrane Proteins (PDBTM)   • MemProtMD


Details about the values in these tables can be found in the corresponding documentation page .
PDBsumOpen PDBsum Page
ChainA
ProteinG Protein α Sub unit
UniProtP63092
Sequence
>7VVL_Chain_A
QRNEEKAQR EANKKIEKQ LQKDKQVYR ATHRLLLLG ADNSGKSTI 
VKQMRIGIF ETKFQVDKV NFHMFDVGG QRDERRKWI QCFNDVTAI 
IFVVDSSDY NRLQEALNL FKSIWNNRW LRTISVILF LNKQDLLAE 
KVLAGKSKI EDYFPEFAR YTTPEDATP EPGEDPRVT RAKYFIRDE 
FLRISTASG DGRHYCYPH FTCAVDTEN ARRIFNDCR DIIQRMHLR 
QYELL


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainB
ProteinG Protein β Sub unit
UniProtP54311
Sequence
>7VVL_Chain_B
QLRQEAEQL KNQIRDARK ACADATLSQ ITNNIDPVG RIQMRTRRT 
LRGHLAKIY AMHWGTDSR LLVSASQDG KLIIWDSYT TNKVHAIPL 
RSSWVMTCA YAPSGNYVA CGGLDNICS IYNLKTREG NVRVSRELA 
GHTGYLSCC RFLDDNQIV TSSGDTTCA LWDIETGQQ TTTFTGHTG 
DVMSLSLAP DTRLFVSGA CDASAKLWD VREGMCRQT FTGHESDIN 
AICFFPNGN AFATGSDDA TCRLFDLRA DQELMTYSH DNIICGITS 
VSFSKSGRL LLAGYDDFN CNVWDALKA DRAGVLAGH DNRVSCLGV 
TDDGMAVAT GSWDSFLKI WN


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainG
ProteinG Protein γ Sub unit
UniProtP63212
Sequence
>7VVL_Chain_G
AQARKLVEQ LKMEANIDR IKVSKAAAD LMAYCEAHA KEDPLLTPV 
PASENPFR


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainR
ProteinReceptor
UniProtQ03431
Sequence
>7VVL_Chain_R
VMTKEEQIF LLHRAQAQC ECLPEWDHI LCWPVAVPC PDYIYDFNH 
KGHAYRRCD RNGSWELVP GHNRTWANY SECVKFLTN ETREREVFD 
RLGMIYTVG YSVSLASLT VAVLILAYF RRLHCTRNY IHMHLFLSF 
MLRAVSIFV KDAVLYSYA GCRVAVTFF LYFLATNYY WILVEGLYL 
HSLIFMAFF SEKKYLWGF TVFGWGLPA VFVAVWVSV RATLANTGC 
WDLSSGNKK WIIQVPILA SIVLNFILF INIVRVLAT KLRETDTRQ 
QYRKLLKST LVLMPLFGV HYIVFMATP YTEVSGTLW QVQMHYEML 
FNSFQGFFV AIIYCFCNG EVQAEIKKS WSRW


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  




This receptor, from the same or other species and bound to the same or other ligands, is also present in the following networks:
Show PDB Class SubFamily Type SubType Species Orthosteric Ligand Other Ligand(s) Protein Partners Resolution Date DOI
9JR3B1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1L-Gs-CtGq)/β1/γ22.82024-10-16To be published
9JR3 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82024-10-16To be published
9JR2B1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1L-Gs-CtGq)/β1/γ22.82024-10-16To be published
9JR2 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82024-10-16To be published
8JR9B1PeptideParathyroid HormonePTH1Homo sapiens-PCO371chim(NtGi1-Gs)/β1/γ22.572023-08-0210.1038/s41586-023-06467-w
8JR9 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiens-PCO3712.572023-08-0210.1038/s41586-023-06467-w
7Y36B1PeptideParathyroid HormonePTH1Homo sapiensTeriparatide-Gs/β1/γ22.82023-07-05To be published
7Y36 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensTeriparatide-2.82023-07-05To be published
7Y35B1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-Gs/β1/γ22.92023-07-05To be published
7Y35 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-2.92023-07-05To be published
8GW8B1PeptideParathyroid HormonePTH1Homo sapiens-KHFGs/β1/γ22.92023-06-1410.1038/s41586-023-06169-3
8GW8 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiens-KHF2.92023-06-1410.1038/s41586-023-06169-3
8FLUB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH-Gs/β1/γ22.762023-04-2610.1016/j.str.2023.04.002
8FLU (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH-2.762023-04-2610.1016/j.str.2023.04.002
8FLTB1PeptideParathyroid HormonePTH1Homo sapiensM-PTH(1-14)-Gs/β1/γ23.032023-04-2610.1016/j.str.2023.04.002
8FLT (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensM-PTH(1-14)-3.032023-04-2610.1016/j.str.2023.04.002
8FLSB1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-Gs/β1/γ23.092023-04-2610.1016/j.str.2023.04.002
8FLS (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-3.092023-04-2610.1016/j.str.2023.04.002
8FLRB1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-Gs/β1/γ22.942023-04-2610.1016/j.str.2023.04.002
8FLR (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-2.942023-04-2610.1016/j.str.2023.04.002
8FLQB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ22.552023-04-2610.1016/j.str.2023.04.002
8FLQ (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.552023-04-2610.1016/j.str.2023.04.002
8HAOB1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1-Gs)/β1/γ23.762022-12-2110.1038/s41401-022-01032-z
8HAO (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.762022-12-2110.1038/s41401-022-01032-z
8HAFB1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-chim(NtGi1-Gs)/β1/γ23.252022-12-2110.1038/s41401-022-01032-z
8HAF (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-3.252022-12-2110.1038/s41401-022-01032-z
8HA0B1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1-Gs)/β1/γ22.622022-12-2110.1038/s41401-022-01032-z
8HA0 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.622022-12-2110.1038/s41401-022-01032-z
7VVOB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ24.12022-08-0310.1016/j.molcel.2022.07.003
7VVO (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-4.12022-08-0310.1016/j.molcel.2022.07.003
7VVNB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ23.82022-08-0310.1016/j.molcel.2022.07.003
7VVN (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.82022-08-0310.1016/j.molcel.2022.07.003
7VVMB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ23.22022-08-0310.1016/j.molcel.2022.07.003
7VVM (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.22022-08-0310.1016/j.molcel.2022.07.003
7VVLB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ22.82022-08-0310.1016/j.molcel.2022.07.003
7VVL (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82022-08-0310.1016/j.molcel.2022.07.003
7VVKB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ23.32022-08-0310.1016/j.molcel.2022.07.003
7VVK (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.32022-08-0310.1016/j.molcel.2022.07.003
7VVJB1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-Gs/β1/γ23.22022-08-0310.1016/j.molcel.2022.07.003
7VVJ (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-3.22022-08-0310.1016/j.molcel.2022.07.003
6NBIB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-Gs/β1/γ242019-04-1710.1126/science.aav7942
6NBI (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-42019-04-1710.1126/science.aav7942
6NBHB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-Gs/β1/γ23.52019-04-1710.1126/science.aav7942
6NBH (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-3.52019-04-1710.1126/science.aav7942
6NBFB1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-Gs/β1/γ232019-04-1710.1126/science.aav7942
6NBF (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLong-Acting PTH Analog-32019-04-1710.1126/science.aav7942
6FJ3B1PeptideParathyroid HormonePTH1Homo sapiensPTH--2.52018-11-2110.1038/s41594-018-0151-4




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