Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg Int. Strength Num Of Links Community ConSurf
1A:A:H41 6.43167686
2A:A:L44 8.145409
3A:A:V214 5.466586
4A:A:F219 7.5175488
5A:A:H220 9.2575417
6A:A:M221 5.1325408
7A:A:F222 9.406517
8A:A:Q227 5.87419
9A:A:R228 5.846519
10A:A:E230 8.3225419
11A:A:K233 7.616519
12A:A:W234 6.4375419
13A:A:I245 3.135407
14A:A:V248 2.9025407
15A:A:L270 6.545406
16A:A:F273 6.1525139
17A:A:W277 9.008336136
18A:A:W281 11.7025415
19A:A:L289 4.144139
20A:A:K300 3.875409
21A:A:Y311 10.61254226
22A:A:F312 5.742598
23A:A:F315 6.91596
24A:A:R333 3.845495
25A:A:R336 7.0675495
26A:A:K338 10.244145
27A:A:Y339 6.63254143
28A:A:F340 8.085497
29A:A:R342 5.784144
30A:A:E344 6.8175495
31A:A:F345 6.454138
32A:A:S349 3.9854137
33A:A:Y360 6.435408
34A:A:F363 6.855145
35A:A:R373 6.2975485
36A:A:F376 5.66167688
37A:A:H387 8.005408
38A:A:Y391 6.726104
39A:A:L393 4.43408
40B:B:L30 6.1375405
41B:B:I37 3.676502
42B:B:V40 4.2654153
43B:B:L51 7.4445119
44B:B:H54 9.9765119
45B:B:K57 10.775419
46B:B:Y59 5.9775418
47B:B:W63 6.944507
48B:B:L70 5.7754115
49B:B:V71 3.71754168
50B:B:Q75 6.7925419
51B:B:D76 7.77409
52B:B:L79 5.0185167
53B:B:W82 10.75176119
54B:B:D83 8.394208
55B:B:K89 6.326119
56B:B:I93 4.995407
57B:B:L95 4.0645168
58B:B:W99 7.86667619
59B:B:M101 5.545419
60B:B:N110 8.92754174
61B:B:Y111 6.1425174
62B:B:C114 4.51254168
63B:B:I123 3.85754176
64B:B:Y124 4.3025406
65B:B:H142 7.304559
66B:B:Y145 5.96286718
67B:B:C148 3.46406
68B:B:F151 3.9975409
69B:B:S161 8.09459
70B:B:D163 7.724559
71B:B:T165 4.405457
72B:B:C166 4.245448
73B:B:W169 9.7925458
74B:B:Q176 5.9525454
75B:B:F180 7.716547
76B:B:H183 8.93833649
77B:B:L190 4.494545
78B:B:F199 8.064549
79B:B:V200 9.1625436
80B:B:S201 4.24449
81B:B:C204 5.0125417
82B:B:D205 7.0625449
83B:B:K209 11.665446
84B:B:L210 4.448535
85B:B:W211 7.335648
86B:B:D212 5.69439
87B:B:C218 6.5575445
88B:B:Q220 7.15537
89B:B:F222 7.584538
90B:B:H225 8.945639
91B:B:D228 8.625419
92B:B:I232 4.705438
93B:B:F235 7.4725186
94B:B:F241 8.394536
95B:B:T243 5.6525438
96B:B:T249 4.8325436
97B:B:R251 9.332538
98B:B:F253 4.82667636
99B:B:R256 6.38254259
100B:B:D258 10.7125437
101B:B:Y264 6.3705
102B:B:I273 6.2475406
103B:B:R283 7.8385159
104B:B:L285 6.2125406
105B:B:Y289 10.006507
106B:B:C294 3.83465
107B:B:W297 8.32254268
108B:B:D298 7.10254159
109B:B:H311 9.422569
110B:B:R314 16.1425418
111B:B:L318 3.71466
112B:B:T329 6.235468
113B:B:W332 12.275619
114B:B:D333 8.78469
115B:B:L336 4.4285117
116B:B:K337 8.7675466
117B:B:W339 11.12469
118G:G:R27 7.17438
119G:G:Y40 9.7454186
120G:G:D48 7.034279
121G:G:N59 8.135409
122G:G:F61 5.268577238
123L:L:Y13 8.3725300
124L:L:F22 4.888570
125L:L:L26 7.0475470
126R:R:Q27 5.525405
127R:R:W36 7.62333676
128R:R:L50 8.2075423
129R:R:P53 4.4875403
130R:R:Y65 7.592576
131R:R:W68 14.098529
132R:R:T71 4.585427
133R:R:C81 6.715429
134R:R:Y84 6.84675
135R:R:L85 8.3975476
136R:R:P86 5.262573
137R:R:W87 6.11473
138R:R:R94 9.036525
139R:R:K98 13.106528
140R:R:C100 5.9025429
141R:R:W106 7.7225429
142R:R:R111 9.1454314
143R:R:Q113 7.24314
144R:R:R116 10.222526
145R:R:Q131 11.55403
146R:R:V134 4.76254302
147R:R:F141 5.535406
148R:R:Y145 7.1785287
149R:R:Y149 7.21667608
150R:R:R173 7.725109
151R:R:F181 3.9525338
152R:R:F184 9.1475408
153R:R:R201 7.844194
154R:R:M231 5.1025406
155R:R:Q232 5.6954127
156R:R:Y233 4.03509
157R:R:V236 4.19754126
158R:R:N238 7.64254369
159R:R:Y239 4.88254368
160R:R:W241 6.661676359
161R:R:E245 8.154109
162R:R:Y248 4.3645108
163R:R:Y267 3.516507
164R:R:P275 4.22409
165R:R:V279 2.8954126
166R:R:W282 5.5465129
167R:R:Q293 6.3325194
168R:R:W295 13.244379
169R:R:T296 3.51754295
170R:R:F303 5.648504
171R:R:W304 7.952506
172R:R:L307 5.4845127
173R:R:R308 6.8375406
174R:R:I321 3.2875408
175R:R:L357 4.4454109
176R:R:V360 3.25406
177R:R:L399 5.0854108
178R:R:Y400 8.024108
179R:R:C401 4.51254339
180R:R:E410 3.80254348
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Int. Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.

Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1B:B:L51 B:B:W82 25.09115.94YesYes1199
2B:B:I338 B:B:L51 24.9368.56NoYes059
3B:B:I338 G:G:F61 24.78443.77NoYes058
4B:B:D76 B:B:S74 31.89518.83YesNo099
5B:B:H54 B:B:S74 31.717111.16YesNo099
6B:B:H54 B:B:W82 29.18636.35YesYes1199
7B:B:D76 B:B:L55 32.104210.86YesNo096
8A:A:K34 B:B:L55 98.42555.64NoNo046
9A:A:K34 A:A:R38 98.47637.43NoNo044
10A:A:Y37 B:B:L55 77.63988.21NoNo046
11A:A:R42 A:A:Y37 83.183410.29NoNo094
12A:A:R38 R:R:L258 98.50167.29NoNo046
13A:A:H41 R:R:T257 98.55159.58YesNo067
14R:R:L258 R:R:T257 98.52662.95NoNo067
15A:A:F219 A:A:H41 11.69757.92YesYes886
16A:A:H41 A:A:I383 99.98613.98YesNo068
17A:A:R42 B:B:W99 81.78073NoYes199
18B:B:L117 B:B:W99 56.33825.69NoYes099
19A:A:Q227 B:B:L117 55.98587.99YesNo099
20A:A:Q227 A:A:W234 13.7574.38YesYes199
21A:A:Q227 B:B:Y145 42.02114.51YesYes198
22A:A:R231 A:A:W234 18.68217NoYes099
23A:A:L272 A:A:R231 18.36784.86NoNo089
24A:A:D240 B:B:W99 12.2956.7NoYes169
25B:B:K57 B:B:W332 11.897519.73YesYes199
26B:B:Q75 B:B:W99 13.08228.76YesYes199
27A:A:F246 A:A:L272 17.58056.09NoNo098
28A:A:F246 A:A:V248 17.42242.62NoYes097
29A:A:F345 A:A:V248 16.78852.62YesYes087
30A:A:H387 A:A:I383 1003.98YesNo088
31A:A:H387 A:A:Q390 50.88786.18YesNo084
32A:A:H387 R:R:L252 49.141218YesNo088
33A:A:Q390 R:R:R173 50.76077.01NoYes049
34A:A:Y391 R:R:R173 49.127313.38YesYes1049
35A:A:L393 A:A:Y391 90.41823.52YesYes084
36R:R:L252 R:R:Y248 48.96473.52NoYes088
37A:A:Y391 R:R:Y248 48.49613.97YesYes1048
38A:A:L393 R:R:I355 89.29645.71YesNo088
39B:B:N340 G:G:F61 20.16893.62NoYes098
40B:B:N340 B:B:R48 18.92168.44NoNo097
41B:B:R46 B:B:R48 18.67062.13NoNo057
42B:B:Q44 B:B:R46 18.53211.17NoNo045
43B:B:Q44 B:B:R42 18.39681.17NoNo042
44B:B:A305 B:B:R42 18.26482.77NoNo042
45B:B:A305 B:B:V40 18.14961.7NoYes043
46B:B:L30 B:B:T34 16.17762.95YesNo055
47B:B:L30 B:B:M262 13.795912.72YesNo054
48B:B:M262 B:B:Y264 13.26948.38NoYes045
49B:B:N313 B:B:W332 21.28244.52NoYes079
50B:B:F292 B:B:N313 20.75323.62NoNo047
51B:B:F292 R:R:R413 20.22392.14NoNo047
52B:B:D312 R:R:R413 19.16483.57NoNo057
53B:B:D312 B:B:D333 18.6357.98NoYes059
54B:B:D333 B:B:H311 13.85277.56YesYes699
55B:B:G162 B:B:Y145 47.14164.35NoYes098
56B:B:G162 B:B:S161 47.04673.71NoYes099
57B:B:H142 B:B:S161 20.689315.34YesYes599
58B:B:D163 B:B:S161 17.625710.31YesYes599
59B:B:H142 B:B:T165 17.65374.11YesYes597
60B:B:D163 B:B:T165 17.27217.23YesYes597
61B:B:T165 B:B:T181 34.77543.14YesNo072
62B:B:G182 B:B:T181 34.52293.64NoNo062
63B:B:G182 G:G:Q18 34.27164.93NoNo069
64B:B:Q220 B:B:R219 16.50533.5YesNo375
65B:B:D212 B:B:R219 25.57315.96YesNo395
66B:B:D212 B:B:E215 25.97697.8YesNo393
67B:B:E215 B:B:M217 26.99528.12NoNo033
68G:G:E17 G:G:Q18 27.73757.65NoNo069
69R:R:F322 R:R:I355 89.04585.02NoNo098
70R:R:F319 R:R:F322 88.54334.29NoNo079
71R:R:F319 R:R:V360 88.41855.24NoYes076
72R:R:I315 R:R:V360 86.53333.07NoYes076
73R:R:I315 R:R:Y239 86.40713.63NoYes078
74R:R:V311 R:R:Y239 86.18018.83NoYes088
75L:L:H1 R:R:V311 86.0499.69NoNo008
76L:L:H1 R:R:W304 85.25968.46NoYes006
77R:R:L307 R:R:W304 84.59764.56YesYes076
78R:R:L307 R:R:Q232 16.91556.65YesYes1277
79R:R:M231 R:R:Q232 16.63275.44YesYes067
80R:R:I194 R:R:M231 16.16355.83NoYes066
81R:R:I194 R:R:T296 16.0073.04NoYes065
82L:L:S11 R:R:T296 13.62256.4NoYes2905
83L:L:S11 R:R:S297 13.48144.89NoNo004
84R:R:Q27 R:R:S297 13.32438.66YesNo054
85L:L:D15 R:R:Q27 12.6796.53NoYes005
86L:L:D15 R:R:M29 12.71434.16NoNo005
87L:L:F22 R:R:M29 12.55657.46YesNo005
88L:L:F22 R:R:L32 23.8854.87YesNo004
89R:R:L32 R:R:P86 35.31386.57NoYes043
90R:R:P86 R:R:V28 28.99583.53YesNo033
91L:L:E16 R:R:V28 28.47252.85NoNo003
92L:L:E16 L:L:Y13 27.94925.61NoYes000
93L:L:Q17 L:L:Y13 16.366911.27NoYes000
94L:L:L14 L:L:Q17 15.84073.99NoNo000
95L:L:L14 L:L:Y10 15.31457.03NoNo000
96L:L:F6 L:L:Y10 14.78863.09NoNo000
97R:R:L307 R:R:W282 65.268510.25YesYes1279
98R:R:K286 R:R:W282 64.89674.64NoYes089
99R:R:K286 R:R:W295 63.585117.4NoYes089
100R:R:R225 R:R:W295 63.11925.99NoYes3789
101R:R:R225 R:R:V221 63.00166.54NoNo084
102R:R:D218 R:R:V221 62.85674.38NoNo044
103R:R:D218 R:R:W215 62.71235.58NoNo042
104R:R:F33 R:R:W215 62.56813.01NoNo042
105R:R:F33 R:R:W36 62.27964.01NoYes046
106L:L:F22 R:R:W36 12.29333.01YesYes706
107R:R:W36 R:R:Y84 31.452814.47YesYes765
108R:R:L32 R:R:Y84 11.98799.38NoYes045
109L:L:F6 R:R:Y145 11.11756.19NoYes007
110L:L:L26 R:R:W36 18.13915.69YesYes706
111L:L:L26 R:R:Y65 18.190910.55YesYes706
112R:R:Y65 R:R:Y84 18.04235.96YesYes765
113L:L:M27 R:R:Y65 31.84935.99NoYes006
114L:L:M27 R:R:R116 31.15584.96NoYes006
115R:R:P69 R:R:W68 12.116421.62NoYes269
116R:R:K98 R:R:R116 17.753814.85YesYes286
117B:B:M217 G:G:E17 27.48265.41NoNo036
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1 Node2 LinkStrength Comm IsNode1Hub? IsNode2Hub? Node1Cons Node2Cons Node1Shell Node2Shell
L:L:H1 R:R:W304 8.46 0 No Yes 0 6 0 1
L:L:H1 R:R:R308 15.8 0 No Yes 0 6 0 1
L:L:H1 R:R:V311 9.69 0 No No 0 8 0 1
L:L:S2 R:R:L377 3 0 No No 0 3 0 1
L:L:S2 R:R:D385 4.42 0 No No 0 7 0 1
L:L:S2 R:R:L386 4.5 0 No No 0 7 0 1
L:L:Q3 R:R:Y149 5.64 0 No Yes 0 8 0 1
L:L:F6 R:R:Y145 6.19 0 No Yes 0 7 0 1
L:L:F6 R:R:L386 7.31 0 No No 0 7 0 1
L:L:T7 R:R:M231 3.01 0 No Yes 0 6 0 1
L:L:S8 R:R:N298 2.98 0 No No 0 6 0 1
L:L:S11 R:R:L198 3 29 No No 0 6 0 1
L:L:S11 R:R:T296 6.4 29 No Yes 0 5 0 1
L:L:S11 R:R:S297 4.89 29 No No 0 4 0 1
L:L:Y13 R:R:V134 3.79 30 Yes Yes 0 2 0 1
L:L:Y13 R:R:Y138 19.86 30 Yes No 0 5 0 1
L:L:D15 R:R:Q27 6.53 0 No Yes 0 5 0 1
L:L:D15 R:R:M29 4.16 0 No No 0 5 0 1
L:L:D15 R:R:Q293 5.22 0 No Yes 0 4 0 1
L:L:K20 R:R:Q131 9.49 0 No Yes 0 3 0 1
L:L:F22 R:R:M29 7.46 7 Yes No 0 5 0 1
L:L:F22 R:R:L32 4.87 7 Yes No 0 4 0 1
L:L:F22 R:R:W36 3.01 7 Yes Yes 0 6 0 1
L:L:I23 R:R:Y65 7.25 7 No Yes 0 6 0 1
L:L:I23 R:R:L85 8.56 7 No Yes 0 6 0 1
L:L:L26 R:R:W36 5.69 7 Yes Yes 0 6 0 1
L:L:L26 R:R:Y65 10.55 7 Yes Yes 0 6 0 1
L:L:L26 R:R:Y84 5.86 7 Yes Yes 0 5 0 1
L:L:M27 R:R:Y65 5.99 0 No Yes 0 6 0 1
L:L:M27 R:R:R116 4.96 0 No Yes 0 6 0 1
R:R:Q27 R:R:V292 4.3 0 Yes No 5 4 1 2
R:R:Q27 R:R:S297 8.66 0 Yes No 5 4 1 1
R:R:P86 R:R:V28 3.53 7 Yes No 3 3 2 1
R:R:D30 R:R:V292 4.38 19 No No 5 4 2 2
R:R:D30 R:R:Q293 11.75 19 No Yes 5 4 2 1
R:R:L32 R:R:Y84 9.38 0 No Yes 4 5 1 1
R:R:L32 R:R:P86 6.57 0 No Yes 4 3 1 2
R:R:F33 R:R:W36 4.01 0 No Yes 4 6 2 1
R:R:K37 R:R:W36 4.64 0 No Yes 3 6 2 1
R:R:K64 R:R:W36 13.92 0 No Yes 4 6 2 1
R:R:W36 R:R:Y84 14.47 7 Yes Yes 6 5 1 1
R:R:Y39 R:R:Y84 2.98 0 No Yes 6 5 2 1
R:R:D63 R:R:R111 11.91 31 No Yes 9 4 2 2
R:R:D63 R:R:Q113 13.05 31 No Yes 9 4 2 1
R:R:Y65 R:R:Y84 5.96 7 Yes Yes 6 5 1 1
R:R:L85 R:R:Y65 8.21 7 Yes Yes 6 6 1 1
R:R:K98 R:R:S66 3.06 2 Yes No 8 5 2 2
R:R:R116 R:R:S66 11.86 2 Yes No 6 5 1 2
R:R:I79 R:R:K98 17.45 2 No Yes 4 8 2 2
R:R:I79 R:R:R116 12.53 2 No Yes 4 6 2 1
R:R:L85 R:R:P86 6.57 7 Yes Yes 6 3 1 2
R:R:L85 R:R:W87 10.25 7 Yes Yes 6 3 1 1
R:R:P86 R:R:W87 8.11 7 Yes Yes 3 3 2 1
R:R:M123 R:R:W87 3.49 0 No Yes 3 3 2 1
R:R:K98 R:R:R116 14.85 2 Yes Yes 8 6 2 1
R:R:Q113 R:R:R111 8.18 31 Yes Yes 4 4 1 2
R:R:P114 R:R:Q113 4.74 0 No Yes 5 4 2 1
R:R:A118 R:R:R116 6.91 2 No Yes 5 6 2 1
R:R:I128 R:R:Q131 8.23 0 No Yes 2 3 2 1
R:R:K132 R:R:Q131 25.76 0 No Yes 2 3 2 1
R:R:M137 R:R:V134 6.09 0 No Yes 4 2 2 1
R:R:V134 R:R:Y138 7.57 30 Yes No 2 5 1 1
R:R:Q142 R:R:Y145 4.51 28 No Yes 5 7 2 1
R:R:Q142 R:R:T146 4.25 28 No No 5 7 2 2
R:R:T146 R:R:Y145 8.74 28 No Yes 7 7 2 1
R:R:Y145 R:R:Y149 4.96 28 Yes Yes 7 8 1 1
R:R:D195 R:R:Y145 11.49 0 No Yes 7 7 2 1
R:R:L192 R:R:T146 2.95 0 No No 7 7 2 2
R:R:A188 R:R:Y149 4 0 No Yes 8 8 2 1
R:R:V191 R:R:Y149 6.31 0 No Yes 7 8 2 1
R:R:L192 R:R:Y149 5.86 0 No Yes 7 8 2 1
R:R:S390 R:R:Y149 16.53 0 No Yes 9 8 2 1
R:R:M231 R:R:S190 6.13 0 Yes No 6 5 1 2
R:R:D195 R:R:V191 5.84 0 No No 7 7 2 2
R:R:I194 R:R:M231 5.83 0 No Yes 6 6 2 1
R:R:I194 R:R:T296 3.04 0 No Yes 6 5 2 1
R:R:C294 R:R:L198 3.17 0 No No 9 6 2 1
R:R:L198 R:R:T296 2.95 29 No Yes 6 5 1 1
R:R:R201 R:R:Y202 11.32 19 Yes No 4 1 2 1
R:R:Q293 R:R:R201 7.01 19 Yes Yes 4 4 1 2
R:R:C294 R:R:R201 6.96 0 No Yes 9 4 2 2
R:R:Q293 R:R:Y202 3.38 19 Yes No 4 1 1 1
R:R:M231 R:R:Q232 5.44 0 Yes Yes 6 7 1 2
R:R:L307 R:R:Q232 6.65 12 Yes Yes 7 7 2 2
R:R:V311 R:R:Y239 8.83 0 No Yes 8 8 1 2
R:R:Q293 R:R:V292 4.3 19 Yes No 4 4 1 2
R:R:N298 R:R:W304 16.95 0 No Yes 6 6 1 1
R:R:M301 R:R:W304 6.98 0 No Yes 5 6 2 1
R:R:L307 R:R:W304 4.56 12 Yes Yes 7 6 2 1
R:R:R308 R:R:W305 3 0 Yes No 6 7 1 2
R:R:F312 R:R:R308 5.34 0 No Yes 5 6 2 1
R:R:F365 R:R:R308 3.21 0 No Yes 7 6 2 1
R:R:D385 R:R:V364 5.84 0 No No 7 6 1 2
R:R:L377 R:R:L382 8.3 0 No No 3 5 1 2
R:R:D385 R:R:S389 2.94 0 No No 7 6 1 2
L:L:E16 R:R:V28 2.85 0 No No 0 3 0 1
L:L:T29 R:R:Q113 2.83 0 No Yes 0 4 0 1
L:L:G4 R:R:W304 2.81 0 No Yes 0 6 0 1
R:R:M123 R:R:Q131 2.72 0 No Yes 3 3 2 1
L:L:A18 R:R:Y202 2.67 0 No No 0 1 0 1
R:R:D299 R:R:Q27 2.61 0 No Yes 4 5 2 1
L:L:A19 R:R:W87 2.59 0 No Yes 0 3 0 1
R:R:K35 R:R:Y84 2.39 0 No Yes 4 5 2 1
R:R:A228 R:R:T296 1.68 0 No Yes 5 5 2 1
R:R:V130 R:R:V134 1.6 0 No Yes 1 2 2 1
L:L:T5 R:R:L377 1.47 0 No No 0 3 0 1
L:L:M27 R:R:Q122 1.36 0 No No 0 3 0 1
L:L:Y13 R:R:A135 1.33 30 Yes No 0 3 0 1
L:L:D9 R:R:Y138 1.15 0 No No 0 5 0 1

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
66.67Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
58.33Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
58.33Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
57.69Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
55.56Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
55.56Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
55.17Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
52.00Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
52.00Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
51.85Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
51.85Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
50.00Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
50.00Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
50.00Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
50.00Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
48.48Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
48.28Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
48.15Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
48.00Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
46.15Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
46.15Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
44.83Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
44.83Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
44.83Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
44.44Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
44.44Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
44.44Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
44.44Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
42.86Single6FJ3PTH6FJ3-PTH1-PTH
42.86Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
42.86Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
42.86Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
42.86Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
42.86Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
42.86Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
42.31Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
41.94Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
41.94Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
41.38Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
41.38Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
40.74Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
40.74Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
40.74Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
40.62Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
40.62Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
40.62Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
40.00Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
40.00Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
40.00Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
39.39Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
39.39Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
39.39Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
39.29Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
38.46Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
38.24Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
37.93Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
37.93Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
37.93Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
37.93Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
37.50Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
37.50Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
37.04Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
36.67Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
36.67Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
36.67Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
36.67Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
36.67Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
35.48Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
35.48Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
35.29Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
35.29Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
35.29Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
34.62Single4XT1Fractalkine4XT1-US28-Fractalkine
34.62Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
34.38Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
33.33Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
33.33Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
32.35Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
32.26Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
32.26Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
32.26Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
32.00Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
31.43Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
31.25Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
31.03Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
31.03Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
30.00Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
29.63Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
29.41Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
29.41Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
29.41Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
29.17Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
29.03Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
28.57Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
28.57Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
28.57Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
28.57Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
28.12Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
28.00Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
27.27Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
26.92Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
26.67Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
26.47Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
26.47Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
26.09Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
26.09Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
25.93Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
25.81Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
25.00Single4XT3Fractalkine4XT3-US28-Fractalkine
25.00Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
25.00Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
25.00Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
24.39Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
24.00Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
23.81Single6LI0C176LI0-GPR52-C17
23.81Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
23.81Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
23.81Single8K5BNiacin8K5B-HCA2-Niacin
23.81Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
23.53Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
23.53Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
23.33Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
23.33Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
23.33Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
23.08Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
23.08Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
23.08Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
22.73Single5U09Taranabant5U09-CB1-Taranabant
22.73Single5ZKQABT-4915ZKQ-PAF-ABT-491
22.73Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
22.73Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
22.73Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
22.73Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.73Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.73Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
22.73Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.73Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.58Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
22.58Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
22.22Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
22.22Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
22.22Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
22.22Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
21.88Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
21.88Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
21.88Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
21.88Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
21.74Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
21.74Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
21.74Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
21.74Single8K5CAcipimox8K5C-HCA2-Acipimox
21.74Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
21.74Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
21.74Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
21.74Consensushca_onOrthosteric Ligandhca2_on
21.74Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
21.43Single5EE7MK08935EE7-Glucagon-MK0893
21.43Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
21.43Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
21.43Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
21.43Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
21.43Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
21.43Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
21.43Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
21.21Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
20.83Single4YAYZD-71554YAY-AT1-ZD-7155
20.83Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
20.83Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
20.83Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
20.83Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
20.83Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
20.83Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
20.83Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
20.83Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
20.83Single9B9ZA1AKO9B9Z-CB1-A1AKO
20.83Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
20.83Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
20.83Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
20.83Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
20.83Consensushca_on_gpOrthosteric Ligandhca2_on_gp
20.83Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
20.69Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
20.69Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
20.59Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
20.59Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
20.59Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
20.00Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
20.00Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
20.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
20.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
20.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
20.00Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
20.00Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
20.00Single8TF5Oleic acid8TF5-GPR6-Oleic acid
20.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
20.00Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
20.00Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
20.00Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
20.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
20.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
20.00Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
20.00Consensusep_offOrthosteric Ligandep4_off
20.00Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
19.44Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
19.35Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
19.35Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
19.35Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
19.23Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
19.23Single7TUYGSK682753A7TUY-GPR183-GSK682753A
19.23Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
19.23Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
19.23Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
19.23Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
19.23Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
19.23Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
19.05Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
19.05Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
19.05Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
18.75Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
18.75Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
18.75Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
18.75Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
18.75Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
18.75Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
18.75Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
18.75Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
18.75Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
18.52Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
18.52Single6IIURamatroban6IIU-TP-Ramatroban
18.52Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
18.52Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
18.52Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
18.52Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
18.52Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
18.52Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
18.52Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
18.52Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
18.52Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
18.52Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
18.52Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
18.52Single8XYIVUF106618XYI-CXCR3-VUF10661
18.52Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
18.52Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
18.52Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
18.52Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
18.18Single3OE9IT1t3OE9-CXCR4-IT1t
18.18Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
18.18Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
18.18Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
18.18Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
18.18Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
18.18Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
18.18Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
18.18Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
18.18Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
18.18Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
18.18Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single9B9Y7DY9B9Y-CB1-7DY
18.18Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
18.18Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
18.18Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
17.86Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
17.86Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
17.86Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
17.86Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
17.86Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
17.86Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
17.86Single7UM4AS26747237UM4-5-HT5A-AS2674723
17.86Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
17.86Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensuscck_onOrthosteric Ligandccka_on cckb_on
17.86Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
17.86Consensusprostanoid_offOrthosteric Ligandep_off dp_off
17.86Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
17.86Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
17.86Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
17.65Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
17.65Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
17.65Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
17.65Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
17.65Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
17.39Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
17.39Single3PWHZM-2413853PWH-A2A-ZM-241385
17.39Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
17.39Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
17.39Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
17.39Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
17.39Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
17.39Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
17.39Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
17.39Single8GNGIstradefylline8GNG-A2A-Istradefylline
17.39Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
17.39Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
17.39Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
17.39Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
17.39Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
17.39Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
17.39Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
17.39Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
17.39Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
17.39Single9BA0A1AKN9BA0-CB1-A1AKN
17.39Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
17.39Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
17.39Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
17.39Consensusangiotensin_offOrthosteric Ligandat1_off
17.39Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
17.24Single3NY9ICI118-5513NY9-β2-ICI118-551
17.24Single4UG2CGS216804UG2-A2A-CGS21680
17.24Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
17.24Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
17.24Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
17.24Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
17.24Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
17.24Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
17.24Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
17.24Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
17.14Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
17.14Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
17.14Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
17.14Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
17.14Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
16.67Single2YDOAdenosine2YDO-A2A-Adenosine
16.67Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
16.67Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
16.67Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
16.67Single7AROLUF58337ARO-A2A-LUF5833-Na
16.67Single7F8XNN90567F8X-CCKA-NN9056
16.67Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
16.67Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
16.67Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
16.67Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
16.67Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
16.67Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
16.67Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
16.67Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
16.67Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
16.67Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
16.67Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
16.67Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
16.67Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
16.67Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
16.67Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
16.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
16.67Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
16.67Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
16.67Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
16.67Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
16.67Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
16.67Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
16.67Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
16.67Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
16.22Single5GLHEndothelin-15GLH-ETB-Endothelin-1
16.22Single6IGKEndothelin-36IGK-ETB-Endothelin-3
16.22Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
16.22Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
16.22Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
16.13Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
16.13Single6HLOAprepitant6HLO-NK1-Aprepitant
16.13Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
16.13Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
16.13Single7XNACYN1548067XNA-SST2-CYN154806
16.13Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
16.13Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
16.13Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
16.13Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
16.13Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
16.13Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
16.13Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
16.13Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
16.13Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
16.13Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
16.13Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
16.00Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
16.00Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
16.00Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
16.00Single5TGZAM65385TGZ-CB1-AM6538
16.00Single5UENDU1725UEN-A1-DU172
16.00Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
16.00Single6D27CAY104716D27-DP2-CAY10471
16.00Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
16.00Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
16.00Single7V3ZCP559407V3Z-CB1-CP55940
16.00Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
16.00Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
16.00Single8CU6LJ-45178CU6-A2A-LJ-4517
16.00Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
16.00Single8K5DGSK2560738K5D-HCA2-GSK256073
16.00Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
16.00Single8RLNLUF58348RLN-A2A-LUF5834
16.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
16.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
16.00Single8T1WCVN4248T1W-GPR6-CVN424
16.00Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
16.00Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
16.00Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
16.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
16.00Single9CHXS-Carazolol9CHX-β2-S-Carazolol
16.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
16.00Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
16.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
16.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
16.00Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
15.79Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
15.79Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
15.79Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
15.62Single3OE0CVX153OE0-CXCR4-CVX15
15.62Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
15.62Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
15.62Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
15.62Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
15.62Consensusangiotensin_onOrthosteric Ligandat1_on
15.62Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
15.62Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
15.62Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.62Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
15.62Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
15.38Single5JQHS-Carazolol5JQH-β2-S-Carazolol
15.38Single5N2RPSB-365N2R-A2A-PSB-36-Na
15.38Single5N2SPSB365N2S-A1-PSB36
15.38Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
15.38Single5TVNLSD5TVN-5-HT2B-LSD
15.38Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
15.38Single6D26Fevipiprant6D26-DP2-Fevipiprant
15.38Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
15.38Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
15.38Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
15.38Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
15.38Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
15.38Single6PS6Timolol6PS6-β2-Timolol
15.38Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
15.38Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
15.38Single7C4SS1P7C4S-S1P3-S1P
15.38Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
15.38Single7SINNPS-21437SIN-CaS-NPS-2143
15.38Single7SINNPS-21437SIN-CaS-NPS-2143
15.38Single7W41PD1762527W41-BB2-PD176252
15.38Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
15.38Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
15.38Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
15.38Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
15.38Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
15.38Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
15.38Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
15.38Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
15.38Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
15.38Consensusadenosine_offOrthosteric Liganda1_off a2_off
15.38Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
15.38Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
15.38Consensusblt_offOrthosteric Ligandblt1_off
15.38Consensusbombesin_offOrthosteric Ligandbb2_off
15.38Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
15.38Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
15.38Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
15.38Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
15.38Consensusdp_offOrthosteric Liganddp2_off
15.38Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
15.38Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
15.38Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
15.38Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
15.38Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Consensustrace-amine_onOrthosteric Ligandta1_on
15.15Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
15.15Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
15.15Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
15.15Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
15.15Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
15.15Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.15Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.15Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
15.15Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
15.15Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
15.15Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
15.15Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
15.15Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
15.15Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
15.15Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
15.15Consensusvasop-oxy_onOrthosteric Ligandv2_on
15.15Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
15.00Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
15.00Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
15.00Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
15.00Single8HS2Fab0468HS2-GPR20-Fab046
15.00Single8PWNTheophylline8PWN-A2A-Theophylline
15.00Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
15.00Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
14.81Single2YDVNECA2YDV-A2A-NECA
14.81Single4UHRCGS216804UHR-A2A-CGS21680
14.81Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
14.81Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
14.81Single5G53NECA5G53-A2A-NECA-Gs
14.81Single5XR8AM8415XR8-CB1-AM841
14.81Single5XRAAM115425XRA-CB1-AM11542
14.81Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
14.81Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
14.81Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
14.81Single6WGTLSD6WGT-5-HT2A-LSD
14.81Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
14.81Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
14.81Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
14.81Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
14.81Single7F1TMIP-1a7F1T-CCR5-MIP-1a
14.81Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
14.81Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
14.81Single7PX4PSB-21137PX4-A2A-PSB-2113
14.81Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
14.81Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
14.81Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
14.81Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
14.81Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
14.81Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
14.81Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
14.81Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
14.81Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
14.81Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
14.81Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
14.81Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
14.81Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
14.81Consensusa2_onOrthosteric Liganda2b_on
14.81Consensusa2_on_gpOrthosteric Liganda2b_on_gp
14.81Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.81Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.81Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
14.81Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
14.81Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
14.81Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
14.81Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
14.81Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
14.81Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
14.81Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.81Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
14.71Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
14.71Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
14.71Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
14.71Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
14.71Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
14.71Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
14.29Single4XEENeurotensin4XEE-NTS1-Neurotensin
14.29Single4XESNeurotensin4XES-NTS1-Neurotensin
14.29Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
14.29Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
14.29Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
14.29Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
14.29Single6OS2TRV0266OS2-AT1-TRV026
14.29Single6YVRNTS8-136YVR-NTS1-NTS8-13
14.29Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
14.29Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
14.29Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
14.29Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
14.29Single7K15MKD0467K15-BLT1-MKD046-Na
14.29Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
14.29Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
14.29Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
14.29Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
14.29Single8A2OTheophylline8A2O-A2A-Theophylline-Na
14.29Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
14.29Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
14.29Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
14.29Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
14.29Single8JWY2-1188JWY-A2A-2-118
14.29Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
14.29Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
14.29Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
14.29Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
14.29Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
14.29Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
14.29Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
14.29Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
14.29Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
14.29Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
14.29Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
14.29Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
14.29Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
14.29Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
14.29Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
14.29Consensuslpa_offOrthosteric Ligandlpa1_off
14.29Consensuslpl_offOrthosteric Ligands1p_off lpa_off
14.29Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
14.29Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
13.89Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
13.89Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
13.89Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
13.89Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
13.89Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
13.89Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
13.89Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
13.79Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
13.79Single4BUONeurotensin4BUO-NTS1-Neurotensin
13.79Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
13.79Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
13.79Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
13.79Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
13.79Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
13.79Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
13.79Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
13.79Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
13.79Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
13.79Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
13.79Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
13.79Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
13.79Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
13.79Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
13.79Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
13.79Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
13.79Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
13.79Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
13.79Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8XVUCXCL28XVU-CXCR2-CXCL2
13.79Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
13.79Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
13.79Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
13.79Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
13.79Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
13.79Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
13.79Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
13.79Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
13.79Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
13.79Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
13.79Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
13.64Single3OE6IT1t3OE6-CXCR4-IT1t
13.64Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
13.64Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
13.64Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
13.64Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
13.64Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
13.64Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
13.64Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.64Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.64Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
13.64Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
13.64Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
13.64Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
13.64Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
13.64Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
13.64Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
13.64Consensusgi_sensoryOrthosteric Ligandgi_opsins
13.64Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
13.64Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
13.51Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
13.51Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
13.51Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
13.51Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
13.51Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
13.51Consensusbradykinin_onOrthosteric Ligandbk2_on
13.51Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
13.51Consensusendothelin_onOrthosteric Ligandetb_on eta_on
13.51Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
13.33Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
13.33Single5ZTYAM102575ZTY-CB2-AM10257
13.33Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
13.33Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
13.33Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
13.33Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
13.33Single7SK9CCX6627SK9-ACKR3-CCX662
13.33Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
13.33Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
13.33Single8IEIA1LYA8IEI-GPR156-A1LYA
13.33Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
13.33Single8QJ2pN1628QJ2-MC4-pN162-Gs
13.33Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
13.33Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
13.33Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
13.33Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
13.33Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
13.16Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
13.16Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
13.16Consensusbombesin_onOrthosteric Ligandbb2_on
13.16Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
13.16Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
13.04Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
13.04Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
13.04Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
13.04Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
13.04Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
13.04Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
13.04Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
13.04Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
13.04Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
13.04Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
13.04Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
13.04Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
13.04Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
13.04Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
13.04Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
13.04Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
13.04Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
13.04Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
13.04Consensusgq_nucleotideOrthosteric Ligandgq_p2y
13.04Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
12.90Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
12.90Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
12.90Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
12.90Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
12.90Single7QA8Peptide7QA8-STE2-Peptide
12.90Single7QA8Peptide7QA8-STE2-Peptide
12.90Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
12.90Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
12.90Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
12.90Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
12.90Single8IEBA1LYA8IEB-GPR156-A1LYA
12.90Single8IEIA1LYA8IEI-GPR156-A1LYA
12.90Single8IEPA1LYA8IEP-GPR156-A1LYA
12.90Single8IEPA1LYA8IEP-GPR156-A1LYA
12.90Single8KIGSHU91198KIG-MC3-SHU9119-Ca
12.90Single8WDTphotoNECA8WDT-A2A-photoNECA
12.90Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.90Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
12.90Single8XWNCXCL88XWN-CXCR2-CXCL8
12.90Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.90Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
12.90Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
12.90Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
12.90Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
12.90Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
12.90Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
12.90Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
12.90Consensuslpl_onOrthosteric Ligands1p_on lpa_on
12.90Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
12.90Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
12.90Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensussomatostatin_offOrthosteric Ligandsst2_off
12.90Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.82Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
12.50Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
12.50Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
12.50Single3ODUIT1t3ODU-CXCR4-IT1t
12.50Single3QAKUK-4320973QAK-A2A-UK-432097
12.50Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
12.50Single4BWBNeurotensin4BWB-NTS1-Neurotensin
12.50Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
12.50Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
12.50Single6AKXA4R6AKX-CCR5-A4R
12.50Single6AKYMaraviroc6AKY-CCR5-Maraviroc
12.50Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
12.50Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
12.50Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
12.50Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
12.50Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.50Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
12.50Single7BR3Elagolix7BR3-GnRH1-Elagolix
12.50Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
12.50Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
12.50Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
12.50Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
12.50Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
12.50Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
12.50Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
12.50Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
12.50Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
12.50Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
12.50Single7SK5CXCL127SK5-ACKR3-CXCL12
12.50Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
12.50Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
12.50Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
12.50Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
12.50Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
12.50Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
12.50Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.50Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.50Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
12.50Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
12.50Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
12.50Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
12.50Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
12.50Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
12.50Single8IEBA1LYA8IEB-GPR156-A1LYA
12.50Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
12.50Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
12.50Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
12.50Single8IWESpermidine8IWE-TA9-Spermidine
12.50Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
12.50Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
12.50Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
12.50Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
12.50Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
12.50Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
12.50Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.50Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.50Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.50Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
12.50Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
12.50Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
12.50Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
12.50Consensusalpha2_offOrthosteric Ligandalpha2c_off
12.50Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
12.50Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
12.50Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
12.50Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.50Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
12.50Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
12.50Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
12.50Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
12.20Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
12.12Single5WF5UK-4320975WF5-A2A-UK-432097
12.12Single6W25SHU91196W25-MC4-SHU9119-Ca
12.12Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
12.12Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
12.12Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.12Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.12Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
12.12Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
12.12Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.12Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
12.12Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
12.12Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
12.12Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
12.12Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
12.00Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
12.00Single3REYXAC3REY-A2A-XAC
12.00Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
12.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
12.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
12.00Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
12.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
12.00Single5IUBQ274563445IUB-A2A-Q27456344-Na
12.00Single5JTBZM-2413855JTB-A2A-ZM-241385
12.00Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
12.00Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
12.00Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
12.00Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
12.00Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
12.00Single6AQFZM-2413856AQF-A2A-ZM-241385
12.00Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
12.00Single6KUXRS-799486KUX-α2a-RS-79948
12.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
12.00Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
12.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
12.00Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
12.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
12.00Single6PS4ICI118-5516PS4-β2-ICI118-551
12.00Single6PS5S-Propranolol6PS5-β2-S-Propranolol
12.00Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
12.00Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
12.00Single6V9SGTPL114036V9S-OX1-GTPL11403
12.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
12.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
12.00Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
12.00Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
12.00Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
12.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
12.00Single7T32ZM-2413857T32-A2A-ZM-241385
12.00Single7UL3Famotidine7UL3-H2-Famotidine
12.00Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
12.00Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
12.00Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
12.00Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
12.00Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
12.00Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
12.00Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
12.00Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
12.00Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
12.00Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
12.00Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.00Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.00Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
12.00Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
12.00Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
12.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
12.00Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
12.00Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
12.00Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
12.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
12.00Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
12.00Single8IHKAcifran8IHK-HCA3-Acifran
12.00Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
12.00Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
12.00Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
12.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
12.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
12.00Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.00Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.00Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.00Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.00Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
12.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
12.00Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
12.00Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
12.00Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
12.00Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
12.00Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
12.00Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
12.00Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
12.00Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
12.00Consensusa2_offOrthosteric Liganda2a_off
12.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
12.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
12.00Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
12.00Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
12.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
12.00Consensusgrh_offOrthosteric Ligandgnrh1_off
12.00Consensusopsins_offOrthosteric Ligandrhodopsin_off
12.00Consensussensory_offOrthosteric Ligandopsins_off
11.76Single6JODAngiotensin II6JOD-AT2-Angiotensin II
11.76Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
11.76Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
11.76Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
11.76Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
11.76Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
11.76Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
11.76Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
11.76Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
11.76Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
11.54Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
11.54Single2Y01Dobutamine2Y01-β1-Dobutamine
11.54Single2Y02Carmoterol2Y02-β1-Carmoterol
11.54Single2Y04Salbutamol2Y04-β1-Salbutamol
11.54Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
11.54Single3EMLZM-2413853EML-A2A-ZM-241385
11.54Single3NY8ICI118-5513NY8-β2-ICI118-551
11.54Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
11.54Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
11.54Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
11.54Single4DAJTiotropium4DAJ-M3-Tiotropium
11.54Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
11.54Single4GBRS-Carazolol4GBR-β2-S-Carazolol
11.54Single4QIMANTA XV4QIM-SMO-ANTA XV
11.54Single4QKX35V4QKX-β2-35V
11.54Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
11.54Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
11.54Single5IU8Q274563475IU8-A2A-Q27456347-Na
11.54Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
11.54Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
11.54Single5T04Neurotensin5T04-NTS1-Neurotensin
11.54Single5UIGCmpd-15UIG-A2A-Cmpd-1
11.54Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
11.54Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
11.54Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
11.54Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
11.54Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
11.54Single6H7MSalbutamol6H7M-β1-Salbutamol
11.54Single6IIVDaltroban6IIV-TP-Daltroban
11.54Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
11.54Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
11.54Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
11.54Single6PS1Timolol6PS1-β2-Timolol
11.54Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
11.54Single6S0LZM-2413856S0L-A2A-ZM-241385
11.54Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
11.54Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
11.54Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
11.54Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
11.54Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
11.54Single7BU7BI1671077BU7-β1-BI167107
11.54Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
11.54Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
11.54Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
11.54Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
11.54Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
11.54Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
11.54Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
11.54Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
11.54Single7PYRPSB-21157PYR-A2A-PSB-2115
11.54Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
11.54Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
11.54Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
11.54Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
11.54Single7UL4Alvimopan7UL4-μ-Alvimopan
11.54Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
11.54Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
11.54Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
11.54Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
11.54Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
11.54Single7WC7Lisuride7WC7-5-HT2A-Lisuride
11.54Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
11.54Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
11.54Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
11.54Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
11.54Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
11.54Single7YXAONO-54306087YXA-S1P5-ONO-5430608
11.54Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
11.54Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
11.54Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
11.54Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
11.54Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
11.54Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
11.54Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.54Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
11.54Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
11.54Single8JJOAlprenolol8JJO-β2-Alprenolol
11.54Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
11.54Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
11.54Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
11.54Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
11.54Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
11.54Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
11.54Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
11.54Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
11.54Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
11.54Consensus5ht5_onOrthosteric Ligand5ht5a_on
11.54Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
11.54Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
11.54Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
11.54Consensusa3_onOrthosteric Liganda3a_on
11.54Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
11.54Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.54Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
11.54Consensusdopamine_offOrthosteric Ligandd2_off d3_off
11.54Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
11.54Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
11.54Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
11.43Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
11.43Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
11.43Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
11.43Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
11.43Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
11.43Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
11.43Single8ZRTET-18ZRT-ETB-ET-1
11.43Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
11.43Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
11.43Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
11.11Single2RH1S-Carazolol2RH1-β2-S-Carazolol
11.11Single2Y00Dobutamine2Y00-β1-Dobutamine
11.11Single2Y03Isoprenaline2Y03-β1-Isoprenaline
11.11Single2YCWS-Carazolol2YCW-β1-S-Carazolol
11.11Single4JKVTaladegib4JKV-SMO-Taladegib
11.11Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
11.11Single5C1MBU725C1M-μ-BU72
11.11Single5CGCHTL142425CGC-mGlu5-HTL14242
11.11Single5D6LS-Carazolol5D6L-β2-S-Carazolol
11.11Single5IUAQ274563485IUA-A2A-Q27456348-Na
11.11Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
11.11Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
11.11Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
11.11Single6E67BI1671076E67-β2-BI167107-Gs (fused)
11.11Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
11.11Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
11.11Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
11.11Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
11.11Single6LUQHaloperidol6LUQ-D2-Haloperidol
11.11Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
11.11Single6S0QZM-2413856S0Q-A2A-ZM-241385
11.11Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
11.11Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
11.11Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
11.11Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
11.11Single7C61Ergotamine7C61-5-HT1B-Ergotamine
11.11Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
11.11Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
11.11Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
11.11Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
11.11Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
11.11Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
11.11Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
11.11Single7SK3CXCL127SK3-ACKR3-CXCL12
11.11Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
11.11Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
11.11Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
11.11Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
11.11Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
11.11Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
11.11Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
11.11Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
11.11Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
11.11Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
11.11Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GNEKW-63568GNE-A2A-KW-6356-Na
11.11Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
11.11Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
11.11Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
11.11Single8QOTNanobody-E8QOT-μ-Nanobody-E
11.11Single8S4DCMF-0198S4D-Apelin-CMF-019
11.11Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
11.11Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
11.11Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
11.11Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
11.11Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
11.11Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
11.11Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
11.11Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
11.11Consensusa3_on_gpOrthosteric Liganda3a_on_gp
11.11Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
11.11Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
11.11Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
11.11Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
11.11Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
11.11Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
11.11Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
11.11Consensusamine_offonOrthosteric Ligandamine_off amine_on
11.11Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
11.11Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
11.11Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
11.11Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
11.11Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
11.11Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
11.11Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
11.11Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
11.11Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
11.11Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
11.11Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
11.11Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
11.11Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
11.11Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
11.11Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
11.11Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
11.11Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
11.11Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
10.81Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
10.81Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
10.71Single3P0GBI1671073P0G-β2-BI167107
10.71Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
10.71Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
10.71Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
10.71Single4BV0Neurotensin4BV0-NTS1-Neurotensin
10.71Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
10.71Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
10.71Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
10.71Single5D5AS-Carazolol5D5A-β2-S-Carazolol
10.71Single5D5BS-Carazolol5D5B-β2-S-Carazolol
10.71Single5V54Methiothepin5V54-5-HT1B-Methiothepin
10.71Single5V56TC1145V56-SMO-TC114
10.71Single5V57TC1145V57-SMO-TC114
10.71Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
10.71Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
10.71Single6H7JIsoprenaline6H7J-β1-Isoprenaline
10.71Single6J21Aprepitant6J21-NK1-Aprepitant
10.71Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
10.71Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
10.71Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
10.71Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.71Single7B6WCyclazosin7B6W-α1b-Cyclazosin
10.71Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
10.71Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
10.71Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
10.71Single7FEECP559407FEE-CB1-CP55940-ZCZ011
10.71Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
10.71Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
10.71Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
10.71Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
10.71Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
10.71Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
10.71Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
10.71Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
10.71Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
10.71Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
10.71Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
10.71Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
10.71Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
10.71Single8E0GBU728E0G-μ-BU72
10.71Single8EA0Iperoxo8EA0-M3-Iperoxo
10.71Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
10.71Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
10.71Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
10.71Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
10.71Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
10.71Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
10.71Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
10.71Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
10.71Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
10.71Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
10.71Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
10.71Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
10.71Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
10.71Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
10.71Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
10.71Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
10.71Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
10.71Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
10.71Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
10.71Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
10.71Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
10.71Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
10.71Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
10.71Single9BJKNAM9BJK-μ-Naloxone-NAM
10.71Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Consensus5ht1_offOrthosteric Ligand5ht1b_off
10.71Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
10.71Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
10.71Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
10.71Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
10.71Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
10.71Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
10.71Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
10.71Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
10.71Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
10.71Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
10.71Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
10.71Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
10.71Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
10.71Consensuslpa_onOrthosteric Ligandlpa1_on
10.71Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
10.71Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.71Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
10.71Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
10.71Consensusneurotensin_onOrthosteric Ligandnts1_on
10.71Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
10.71Consensusrelaxin_onOrthosteric Ligandrxfp4_on
10.71Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
10.53Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
10.53Single8IY6Endothelin-18IY6-ETB-Endothelin-1
10.53Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
10.34Single3D4STimolol3D4S-β2-Timolol
10.34Single4AMIBucindolol4AMI-β1-Bucindolol
10.34Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
10.34Single4LDEBI1671074LDE-β2-BI167107
10.34Single4N4WSANT-14N4W-SMO-SANT-1
10.34Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
10.34Single5CXVTiotropium5CXV-M1-Tiotropium
10.34Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
10.34Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
10.34Single5X33BIIL2605X33-BLT1-BIIL260
10.34Single6CM4Risperidone6CM4-D2-Risperidone
10.34Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
10.34Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
10.34Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
10.34Single6KQICP559406KQI-CB1-CP55940-Org27569
10.34Single6MXTSalmeterol6MXT-β2-Salmeterol
10.34Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
10.34Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
10.34Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
10.34Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
10.34Single7DFPSpiperone7DFP-D2-Spiperone
10.34Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
10.34Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
10.34Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
10.34Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
10.34Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
10.34Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
10.34Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
10.34Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
10.34Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
10.34Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
10.34Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
10.34Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
10.34Single8JJ8Formoterol8JJ8-β2-Formoterol
10.34Single8JJLOlodaterol8JJL-β2-Olodaterol
10.34Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
10.34Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
10.34Single8JWZAB9288JWZ-A2A-AB928-Na
10.34Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
10.34Single8XWMCXCL68XWM-CXCR2-CXCL6
10.34Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
10.34Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
10.34Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
10.34Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
10.34Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
10.34Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
10.34Consensusalpha1_offOrthosteric Ligandalpha1a_off
10.34Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
10.34Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
10.34Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
10.34Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
10.34Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
10.34Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
10.34Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
10.34Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
10.34Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
10.34Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
10.34Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
10.34Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
10.34Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
10.34Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
10.34Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
10.26Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
10.26Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
10.00Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
10.00Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
10.00Single5CGDHTL142425CGD-mGlu5-HTL14242
10.00Single5MZPCaffeine5MZP-A2A-Caffeine-Na
10.00Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
10.00Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
10.00Single6H7LDobutamine6H7L-β1-Dobutamine
10.00Single6IBLArformoterol6IBL-β1-Arformoterol
10.00Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
10.00Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
10.00Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
10.00Single7EZCUKA7EZC-A2A-UKA
10.00Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
10.00Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
10.00Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
10.00Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
10.00Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
10.00Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
10.00Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
10.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
10.00Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
10.00Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
10.00Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
10.00Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
10.00Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
10.00Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
10.00Single8XWFCXCL38XWF-CXCR2-CXCL3
10.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
10.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
10.00Consensuschemerin_onOrthosteric Ligandcml1_on
10.00Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
10.00Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single5WF6UK-4320975WF6-A2A-UK-432097
9.68Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
9.68Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
9.68Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
9.68Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
9.68Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
9.68Single7XN9L-054,5227XN9-SST2-L-054,522
9.68Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
9.68Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
9.68Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
9.68Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
9.68Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
9.68Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
9.52Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
9.38Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
9.38Single4IARErgotamine4IAR-5-HT1B-Ergotamine
9.38Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
9.38Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
9.38Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
9.38Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
9.38Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
9.38Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
9.38Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
9.38Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
9.38Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
9.38Single8WKYPG-9348WKY-MC4-PG-934
9.38Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
9.38Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
9.09Single3OE8IT1t3OE8-CXCR4-IT1t
9.09Single3RFMCaffeine3RFM-A2A-Caffeine
9.09Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
9.09Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
9.09Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
9.09Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
9.09Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
9.09Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
9.09Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
9.09Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
9.09Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
9.09Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
9.09Single9CHUNoradrenaline9CHU-β2-Noradrenaline
9.09Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
9.09Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
9.09Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
9.09Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
9.09Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
9.09Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
9.09Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
9.09Consensusp2y_offOrthosteric Ligandp2y1_off
9.09Consensussensory_onOrthosteric Ligandopsins_on
9.09Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
9.09Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
8.82Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
8.82Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
8.82Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
8.82Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
8.82Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
8.70Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
8.70Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
8.70Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
8.70Single3UZAGTPL92363UZA-A2A-GTPL9236
8.70Single4XNWMRS25004XNW-P2Y1-MRS2500
8.70Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
8.70Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
8.70Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
8.70Single6ME5Agomelatine6ME5-MT1-Agomelatine
8.70Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
8.70Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
8.70Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
8.70Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
8.70Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.70Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
8.70Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
8.70Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
8.70Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
8.70Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
8.70Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
8.70Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
8.70Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.70Consensus5ht2_onOrthosteric Ligand5ht2b_on
8.70Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.70Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
8.70Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
8.70Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
8.70Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
8.70Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
8.70Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
8.57Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
8.57Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
8.57Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
8.57Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
8.33Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
8.33Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
8.33Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
8.33Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
8.33Single3PBLEticlopride3PBL-D3-Eticlopride
8.33Single4O9RCyclopamine4O9R-SMO-Cyclopamine
8.33Single5L7IVismodegib5L7I-SMO-Vismodegib
8.33Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
8.33Single6HLLCP999946HLL-NK1-CP99994
8.33Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
8.33Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
8.33Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
8.33Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
8.33Single7SRQLSD7SRQ-5-HT2B-LSD
8.33Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
8.33Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
8.33Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
8.33Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
8.33Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
8.33Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
8.33Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
8.33Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
8.33Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
8.33Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
8.33Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
8.33Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
8.33Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
8.33Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
8.33Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
8.33Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
8.33Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
8.33Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
8.33Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
8.33Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
8.33Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
8.33Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
8.33Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
8.33Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
8.33Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
8.33Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
8.33Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
8.33Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
8.33Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
8.33Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
8.33Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
8.33Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
8.33Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
8.33Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
8.11Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
8.00Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
8.00Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
8.00Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
8.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
8.00Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
8.00Single4QINSAG1.54QIN-SMO-SAG1.5
8.00Single4S0VSuvorexant4S0V-OX2-Suvorexant
8.00Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
8.00Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
8.00Single5WS3EMPA5WS3-OX2-EMPA
8.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
8.00Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
8.00Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
8.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
8.00Single6ME9Ramelteon6ME9-MT2-Ramelteon
8.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
8.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
8.00Single6TODEMPA6TOD-OX1-EMPA-Na
8.00Single6TPJSuvorexant6TPJ-OX2-Suvorexant
8.00Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
8.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
8.00Single7F8ULintitript7F8U-CCKA-Lintitript
8.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
8.00Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
8.00Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
8.00Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
8.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
8.00Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
8.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
8.00Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
8.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
8.00Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
8.00Single7XRRLemborexant7XRR-OX2-Lemborexant
8.00Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
8.00Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
8.00Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
8.00Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
8.00Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
8.00Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
8.00Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
8.00Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
8.00Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
8.00Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
8.00Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
8.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
8.00Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
8.00Single8Y0HVUF114188Y0H-CXCR3-VUF11418
8.00Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
8.00Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
8.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
8.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
8.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
8.00Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.00Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.00Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
8.00Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
8.00Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
8.00Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
8.00Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
8.00Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
8.00Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
8.00Consensusorexin_offOrthosteric Ligandox2_off ox1_off
8.00Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
8.00Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
8.00Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
7.89Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
7.89Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
7.69Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
7.69Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
7.69Single4ZJCSB-6740424ZJC-OX1-SB-674042
7.69Single5UVIZM-2413855UVI-A2A-ZM-241385
7.69Single6A94Zotepine6A94-5-HT2A-Zotepine
7.69Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
7.69Single6IGLIRL16206IGL-ETB-IRL1620
7.69Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
7.69Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
7.69Single6TP3Nemorexant6TP3-OX1-Nemorexant
7.69Single6TPGEMPA6TPG-OX2-EMPA
7.69Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
7.69Single6VI4JDTic6VI4-κ-JDTic
7.69Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
7.69Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
7.69Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
7.69Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
7.69Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
7.69Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
7.69Single6ZG9GSK10347026ZG9-M1-GSK1034702
7.69Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
7.69Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
7.69Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
7.69Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
7.69Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
7.69Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
7.69Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
7.69Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
7.69Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
7.69Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
7.69Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
7.69Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
7.69Single7VODCariprazine7VOD-5-HT2A-Cariprazine
7.69Single7VV6C48/807VV6-MRGPRX2-C48/80
7.69Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
7.69Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
7.69Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
7.69Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
7.69Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
7.69Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
7.69Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
7.69Single8K2WAMG4878K2W-CXCR3-AMG487
7.69Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
7.69Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
7.69Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
7.69Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
7.69Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
7.69Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
7.69Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
7.69Consensusalpha1_onOrthosteric Ligandalpha1a_on
7.69Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
7.69Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
7.69Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
7.69Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
7.69Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
7.69Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
7.69Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
7.50Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
7.41Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
7.41Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
7.41Single4EJ4Naltrindole4EJ4-δ-Naltrindole
7.41Single4MQSIperoxo4MQS-M2-Iperoxo
7.41Single4U14Tiotropium4U14-M3-Tiotropium
7.41Single5DHHSB-6121115DHH-NOP-SB-612111
7.41Single5DSGTiotropium5DSG-M4-Tiotropium
7.41Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
7.41Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
7.41Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
7.41Single6DRXLisuride6DRX-5-HT2B-Lisuride
7.41Single6GPSMK08126GPS-CCR2-MK0812
7.41Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
7.41Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
7.41Single6TOTLemborexant6TOT-OX1-Lemborexant
7.41Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
7.41Single7F83PF-051904577F83-Ghrelin-PF-05190457
7.41Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
7.41Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
7.41Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
7.41Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
7.41Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
7.41Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
7.41Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
7.41Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
7.41Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.41Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
7.41Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
7.41Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
7.41Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
7.41Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
7.41Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
7.41Single8JXRLSD8JXR-D1-LSD
7.41Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
7.41Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
7.41Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
7.41Single8X63Mepyramine8X63-H1-Mepyramine
7.41Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
7.41Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
7.41Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
7.41Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
7.41Single9IYAONO-97105319IYA-GPR55-ONO-9710531
7.41Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
7.41Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
7.41Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
7.41Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
7.41Consensusalpha2_onOrthosteric Ligandalpha2b_on
7.41Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
7.41Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
7.41Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
7.41Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
7.41Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
7.41Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
7.41Consensusblt_onOrthosteric Ligandblt1_on
7.41Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
7.41Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
7.41Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
7.41Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.41Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.41Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.41Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
7.41Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
7.41Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
7.41Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
7.41Consensushistamine_offOrthosteric Ligandh1_off
7.41Consensusleukotriene_onOrthosteric Ligandblt_on
7.41Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
7.41Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
7.41Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
7.41Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
7.32Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
7.32Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
7.14Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
7.14Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
7.14Single5WIUNemonapride5WIU-D4-Nemonapride
7.14Single5WIVNemonapride5WIV-D4-Nemonapride-Na
7.14Single5WQCEMPA5WQC-OX2-EMPA
7.14Single5XPRBosentan5XPR-ETB-Bosentan
7.14Single6GPXMK08126GPX-CCR2-MK0812
7.14Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
7.14Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
7.14Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
7.14Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
7.14Single6TP6Filorexant6TP6-OX1-Filorexant
7.14Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.14Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
7.14Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
7.14Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
7.14Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
7.14Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
7.14Single7WC6LSD7WC6-5-HT2A-LSD
7.14Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
7.14Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
7.14Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
7.14Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
7.14Single8JXSPF-61428JXS-D1-PF-6142
7.14Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8ZMFA1L108ZMF-5-HT2C-A1L10
7.14Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
7.14Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
7.14Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
7.14Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
7.14Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
7.14Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
7.14Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
7.14Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
7.14Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
7.14Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
7.14Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
7.14Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single4DJHJDTic4DJH-κ-JDTic
6.90Single4U15Tiotropium4U15-M3-Tiotropium
6.90Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
6.90Single6J20Aprepitant6J20-NK1-Aprepitant
6.90Single6OL9Tiotropium6OL9-M5-Tiotropium
6.90Single6OS1TRV0266OS1-AT1-TRV026
6.90Single6TQ7SB-3348676TQ7-OX1-SB-334867
6.90Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
6.90Single7P2L4YI7P2L-mGlu5-4YI
6.90Single7R0CAVP7R0C-V2-AVP-Arrestin2
6.90Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
6.90Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
6.90Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
6.90Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
6.90Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
6.90Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
6.90Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
6.90Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
6.90Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
6.90Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
6.90Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
6.90Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.90Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
6.90Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.90Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
6.90Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
6.90Single8XVLZibotentan8XVL-ETA-Zibotentan
6.90Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
6.90Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
6.90Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
6.90Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
6.90Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
6.90Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
6.90Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
6.90Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
6.90Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
6.90Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
6.90Consensustachykinin_offOrthosteric Ligandnk1_off
6.67Single4RWADIPP-NH24RWA-δ-DIPP-NH2
6.67Single6A93Risperidone6A93-5-HT2A-Risperidone
6.67Single6ZG4HTL00099366ZG4-M1-HTL0009936
6.67Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
6.67Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
6.67Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
6.67Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
6.67Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.67Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
6.67Single7YITNalfurafine7YIT-κ-Nalfurafine
6.67Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
6.67Single8XQJJN2418XQJ-Apelin-JN241
6.67Single8XWACXCL18XWA-CXCR2-CXCL1
6.67Single8XWSCXCL58XWS-CXCR2-CXCL5
6.67Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
6.67Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
6.67Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
6.67Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
6.67Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
6.67Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
6.67Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
6.67Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
6.67Consensusorexin_onOrthosteric Ligandox2_on
6.67Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.67Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.45Single5X93K-87945X93-ETB-K-8794
6.45Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
6.45Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
6.45Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
6.45Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.45Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.45Single8XVJMacitentan8XVJ-ETA-Macitentan
6.45Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
6.45Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
6.45Consensusendothelin_offOrthosteric Ligandetb_off
6.45Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
6.45Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
6.45Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.45Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
6.45Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
6.25Single6KNMJN241-96KNM-Apelin-JN241-9
6.25Single6PT3DPI-2876PT3-δ-DPI-287
6.25Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
6.25Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
6.25Single8X5YAstemizole8X5Y-H1-Astemizole
6.25Single8XQJJN2418XQJ-Apelin-JN241
6.25Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
6.25Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
6.25Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
6.25Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
6.25Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
6.06Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
6.06Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
6.06Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.06Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
6.06Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
5.88Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
5.71Single6PT2KGCHM076PT2-δ-KGCHM07
5.71Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
5.71Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
5.71Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
5.71Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
5.71Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
5.71Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
5.56Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.56Single6D35Cholesterol6D35-SMO-Cholesterol
5.56Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.56Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.56Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
5.56Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
5.56Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
5.56Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
5.56Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
5.56Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
5.56Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
5.56Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
5.56Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
5.56Single7DTTCa7DTT-CaS-Ca-Ca
5.56Single7DTTCa7DTT-CaS-Ca-Ca
5.56Single7DTUTryptophan7DTU-CaS-Tryptophan
5.56Single7DTUTryptophan7DTU-CaS-Tryptophan
5.56Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.56Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.56Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.56Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.56Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.56Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.56Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.56Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.56Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
5.56Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.56Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.56Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.56Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.56Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.56Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.56Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
5.56Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
5.56Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.56Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.56Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.56Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.56Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.56Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.56Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.56Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.56Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.56Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.56Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.56Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.56Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.56Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.56Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
5.56Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.56Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.56Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.56Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.56Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.56Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.56Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
5.56Single7XW7K1-707XW7-TSH-K1-70
5.56Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.56Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.56Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.56Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.56Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.56Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.56Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.56Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.56Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.56Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.56Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.56Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.56Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
5.56Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.56Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.56Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.56Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.56Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
5.56Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
5.56Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.56Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.56Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
5.56Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
5.56Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
5.56Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
5.56Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.56Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.56Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.56Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
5.56Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
5.56Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
5.56Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
5.56Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.56Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.56Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.56Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.56Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.56Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.56Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.56Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.56Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.56Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.56Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.56Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.56Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.56Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.56Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.56Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.56Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.56Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.56Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
5.56Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
5.56Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
5.56Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
5.56Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
5.56Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
5.56Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.56Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.56Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single8WVXNorrin8WVX-LGR4-Norrin
5.56Single8WVYNorrin8WVY-LGR4-Norrin
5.56Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.56Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.56Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.56Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.56Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.56Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.56Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
5.56Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.56Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.56Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.56Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.56Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.56Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.56Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.56Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.56Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
5.26Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.26Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.26Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.26Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.26Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.26Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.26Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.26Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.26Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.00Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
5.00Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
5.00Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
5.00Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
4.76Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.76Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.76Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
4.76Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.76Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.76Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
4.55Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
4.55Single5L7DCholesterol5L7D-SMO-Cholesterol
4.55Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.55Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
4.55Single7WC4Serotonin7WC4-5-HT2A-Serotonin
4.55Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.55Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
4.35Single6TQ9SB-4081246TQ9-OX1-SB-408124
4.35Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
4.35Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
4.35Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
4.35Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
4.17Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
4.17Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
4.17Single7WC5Psilocin7WC5-5-HT2A-Psilocin
4.17Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
4.17Single8JPSCCL78JPS-ACKR1-CCL7
4.17Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
4.17Single8ZPLCholesterol8ZPL-CXCR4-HF51116-Cholesterol
4.17Single8ZPMCholesterol8ZPM-CXCR4-AMD070-Cholesterol
4.17Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
4.00Single6TP4ACT-4622066TP4-OX1-ACT-462206
4.00Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
4.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
4.00Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.00Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
4.00Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
4.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
4.00Single8HNNSCH5467388HNN-CXCR3-SCH546738
4.00Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
4.00Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.00Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.00Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
3.85Single4XNVBPTU4XNV-P2Y1-BPTU
3.85Single6B73MP11046B73-κ-MP1104
3.85Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
3.85Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
3.85Single7F8YDevazepide7F8Y-CCKA-Devazepide
3.85Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
3.85Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.85Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
3.85Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
3.85Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
3.85Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.85Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
3.85Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
3.85Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
3.70Single3RZECidoxepin3RZE-H1-Cidoxepin
3.70Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
3.70Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
3.70Single6IQLL7458706IQL-D4-L745870
3.70Single6TPKRetosiban6TPK-OT-Retosiban
3.70Single6TPNHTL66416TPN-OX2-HTL6641
3.70Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
3.70Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
3.70Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
3.70Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
3.70Single8JD6N-(3-chlorophenyl)pyridine-2-carboxamide8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
3.70Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
3.70Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
3.70Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
3.70Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
3.70Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
3.70Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
3.70Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
3.70Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
3.70Consensusvasop-oxy_offOrthosteric Ligandot_off
3.57Single5DHGC-355DHG-NOP-C-35
3.57Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
3.57Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
3.57Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
3.57Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.57Single8X64Desloratadine8X64-H1-Desloratadine
3.57Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
3.57Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
3.57Consensuscck_offOrthosteric Ligandccka_off
3.57Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
3.45Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
3.45Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
3.45Single6HLPNetupitant6HLP-NK1-Netupitant
3.45Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
3.45Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
3.45Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
3.45Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.45Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
3.45Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
3.45Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.45Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.45Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
3.45Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
3.45Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
3.45Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
3.45Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
3.33Single5TZRMK86665TZR-FFA1-MK8666
3.33Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
3.33Single6E59L-7607356E59-NK1-L-760735
3.33Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
3.33Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
3.33Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
3.33Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
3.33Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
3.33Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
3.33Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
3.33Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
3.33Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
3.23Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
3.23Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
3.23Single4PY02MeSATP4PY0-P2Y12-2MeSATP
3.23Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
3.23Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
3.23Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.23Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
3.23Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
3.12Single6K1QIRL25006K1Q-ETB-IRL2500
3.12Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
3.12Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.12Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
3.12Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
3.12Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
3.03Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
3.03Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
3.03Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
3.03Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
3.03Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
3.03Consensuskisspeptin_onOrthosteric Ligandkiss1_on
2.94Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
2.94Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
2.94Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
2.94Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.94Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.94Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
2.94Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
2.94Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
2.94Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
2.94Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
2.94Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
2.86Single7SHEPI; PE7SHE-GPR158-PI; PE
2.86Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
2.86Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
2.78Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.78Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.78Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
2.70Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.70Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
2.50Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

PDB Summary
PDB 6WHC
Class B1
SubFamily Peptide
Type Glucagon
SubType Glucagon
Species Homo Sapiens
Ligand Glu16 analog of GCG
Other Ligand(s) -
Protein Partners Gs/Beta1/Gamma2
PDB Resolution 3.4
Date 2020-05-27
D.O.I. 10.1074/jbc.RA120.013793
Net Summary
Imin 2.95
Number of Linked Nodes 945
Number of Links 1116
Number of Hubs 180
Number of Links mediated by Hubs 643
Number of Communities 37
Number of Nodes involved in Communities 252
Number of Links involved in Communities 346
Path Summary
Number Of Nodes in MetaPath 118
Number Of Links MetaPath 117
Number of Shortest Paths 1949245
Length Of Smallest Path 3
Average Path Length 40.9079
Length of Longest Path 76
Minimum Path Strength 1.17
Average Path Strength 6.58217
Maximum Path Strength 25.86
Minimum Path Correlation 0.71
Average Path Correlation 0.99056
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2
Average % Of Corr. Nodes 50.9397
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 42.7602
Maximum Path Hubs % 100
AnnotationTypeLinks
Gene OntologyMolecular Function• binding   • guanyl nucleotide binding   • GTP binding   • nucleotide binding   • guanyl ribonucleotide binding   • purine ribonucleotide binding   • purine ribonucleoside triphosphate binding   • nucleoside phosphate binding   • ion binding   • purine nucleotide binding   • anion binding   • heterocyclic compound binding   • carbohydrate derivative binding   • ribonucleotide binding   • small molecule binding   • D1 dopamine receptor binding   • protein binding   • signaling receptor binding   • G protein-coupled receptor binding   • dopamine receptor binding   • protein-containing complex binding   • G-protein beta/gamma-subunit complex binding   • pyrophosphatase activity   • GTPase activity   • G protein activity   • ribonucleoside triphosphate phosphatase activity   • molecular function regulator activity   • hydrolase activity, acting on acid anhydrides, in phosphorus-containing anhydrides   • hydrolase activity   • hydrolase activity, acting on acid anhydrides   • catalytic activity   • enzyme regulator activity   • molecular function activator activity   • phosphorus-oxygen lyase activity   • cyclase regulator activity   • enzyme activator activity   • cyclase activator activity   • cyclase activity   • adenylate cyclase regulator activity   • lyase activity   • adenylate cyclase activator activity   • adenylate cyclase activity   • cation binding   • metal ion binding   • developmental process   • multicellular organismal process   • epithelium development   • ectodermal placode morphogenesis   • epidermis development   • molting cycle process   • hair cycle   • animal organ development   • hair follicle placode formation   • tissue development   • ectodermal placode formation   • anatomical structure morphogenesis   • skin development   • skin epidermis development   • hair follicle development
Gene OntologyBiological Process• developmental process   • multicellular organismal process   • epithelium development   • ectodermal placode morphogenesis   • epidermis development   • molting cycle process   • hair cycle   • animal organ development   • hair follicle placode formation   • tissue development   • ectodermal placode formation   • anatomical structure morphogenesis   • skin development   • skin epidermis development   • hair follicle development   • molting cycle   • anatomical structure development   • anatomical structure formation involved in morphogenesis   • ectodermal placode development   • hair cycle process   • system process   • sensory perception of chemical stimulus   • sensory perception   • nervous system process   • sensory perception of smell   • cellular response to stimulus   • cellular response to nitrogen compound   • response to stimulus   • response to endogenous stimulus   • response to peptide hormone   • cellular response to peptide hormone stimulus   • response to oxygen-containing compound   • response to nitrogen compound   • response to glucagon   • cellular response to oxygen-containing compound   • cellular response to glucagon stimulus   • cellular response to endogenous stimulus   • cellular response to chemical stimulus   • response to hormone   • response to chemical   • cellular process   • cellular response to hormone stimulus   • multicellular organism development   • skeletal system development   • bone development   • system development   • regulation of body fluid levels   • wound healing   • homotypic cell-cell adhesion   • cell activation   • hemostasis   • biological regulation   • platelet aggregation   • blood coagulation   • cell adhesion   • cell-cell adhesion   • response to stress   • coagulation   • regulation of biological quality   • response to wounding   • platelet activation   • response to fluid shear stress   • vascular endothelial cell response to laminar fluid shear stress   • response to laminar fluid shear stress   • cellular response to stress   • cellular response to laminar fluid shear stress   • vascular endothelial cell response to fluid shear stress   • cellular response to fluid shear stress   • cognition   • developmental growth   • growth   • response to ketone   • response to prostaglandin   • response to lipid   • response to alcohol   • cellular response to prostaglandin stimulus   • cellular response to prostaglandin E stimulus   • cellular response to alcohol   • cellular response to lipid   • response to prostaglandin E   • cellular response to ketone   • regulation of biological process   • regulation of cellular process   • signaling   • adenylate cyclase-activating G protein-coupled receptor signaling pathway   • cell communication   • adenylate cyclase-modulating G protein-coupled receptor signaling pathway   • G protein-coupled receptor signaling pathway   • signal transduction   • homeostatic process   • positive regulation of biological process   • adaptive thermogenesis   • positive regulation of metabolic process   • multicellular organismal-level homeostasis   • regulation of cold-induced thermogenesis   • cold-induced thermogenesis   • temperature homeostasis   • positive regulation of cold-induced thermogenesis   • positive regulation of multicellular organismal process   • metabolic process   • regulation of multicellular organismal process   • regulation of metabolic process   • positive regulation of cellular process   • protein localization   • regulation of localization   • establishment of protein localization   • nitrogen compound transport   • localization   • cellular macromolecule localization   • regulation of peptide hormone secretion   • regulation of hormone levels   • establishment of protein localization to extracellular region   • protein secretion   • establishment of localization   • regulation of protein secretion   • regulation of secretion   • cellular localization   • regulation of hormone secretion   • regulation of protein localization   • regulation of peptide secretion   • transport   • hormone secretion   • protein localization to extracellular region   • peptide secretion   • regulation of secretion by cell   • secretion by cell   • amide transport   • signal release   • regulation of signaling   • regulation of transport   • secretion   • regulation of peptide transport   • regulation of establishment of protein localization   • export from cell   • cell-cell signaling   • regulation of protein transport   • peptide transport   • protein transport   • regulation of cellular localization   • regulation of insulin secretion   • peptide hormone secretion   • macromolecule localization   • hormone transport   • regulation of cell communication   • insulin secretion   • adenylate cyclase-activating adrenergic receptor signaling pathway   • adrenergic receptor signaling pathway   • establishment of localization in cell   • intracellular transport   • regulation of defense response   • regulation of response to external stimulus   • negative regulation of inflammatory response   • negative regulation of biological process   • inflammatory response to antigenic stimulus   • regulation of response to stress   • regulation of immune system process   • negative regulation of inflammatory response to antigenic stimulus   • defense response   • immune response   • negative regulation of response to stimulus   • negative regulation of immune response   • regulation of inflammatory response to antigenic stimulus   • response to external stimulus   • regulation of inflammatory response   • regulation of response to stimulus   • negative regulation of immune system process   • immune system process   • negative regulation of response to external stimulus   • negative regulation of defense response   • regulation of immune response   • inflammatory response   • positive regulation of adenylate cyclase activity   • positive regulation of molecular function   • regulation of molecular function   • positive regulation of cyclase activity   • activation of adenylate cyclase activity   • regulation of adenylate cyclase activity   • regulation of catalytic activity   • positive regulation of catalytic activity   • positive regulation of lyase activity   • response to dopamine   • cellular response to dopamine   • response to monoamine   • response to catecholamine   • adenylate cyclase-activating dopamine receptor signaling pathway   • cellular response to catecholamine stimulus   • G protein-coupled dopamine receptor signaling pathway   • cellular response to monoamine stimulus   • renal system process   • chemical homeostasis   • multicellular organismal-level water homeostasis   • multicellular organismal-level chemical homeostasis   • renal water homeostasis   • cellular anatomical structure   • membrane   • protein-containing complex   • extrinsic component of plasma membrane   • catalytic complex   • plasma membrane protein complex   • cytoplasmic side of membrane   • plasma membrane   • membrane protein complex   • heterotrimeric G-protein complex   • side of membrane   • cell periphery   • cytoplasmic side of plasma membrane   • GTPase complex
Gene OntologyCellular Component• cellular anatomical structure   • membrane   • protein-containing complex   • extrinsic component of plasma membrane   • catalytic complex   • plasma membrane protein complex   • cytoplasmic side of membrane   • plasma membrane   • membrane protein complex   • heterotrimeric G-protein complex   • side of membrane   • cell periphery   • cytoplasmic side of plasma membrane   • GTPase complex   • extrinsic component of membrane   • extrinsic component of cytoplasmic side of plasma membrane   • extracellular exosome   • membrane-bounded organelle   • extracellular vesicle   • extracellular organelle   • extracellular region   • organelle   • extracellular space   • vesicle   • extracellular membrane-bounded organelle   • intracellular anatomical structure   • cytoplasm   • cytosol   • Golgi apparatus subcompartment   • Golgi apparatus   • organelle subcompartment   • trans-Golgi network membrane   • intracellular membrane-bounded organelle   • endomembrane system   • intracellular organelle   • trans-Golgi network   • organelle membrane   • protein binding   • binding   • enzyme binding   • GTPase binding   • protein-containing complex binding   • pyrophosphatase activity   • GTPase activity   • ribonucleoside triphosphate phosphatase activity   • hydrolase activity, acting on acid anhydrides, in phosphorus-containing anhydrides   • hydrolase activity   • hydrolase activity, acting on acid anhydrides   • catalytic activity   • signaling receptor complex adaptor activity   • protein-macromolecule adaptor activity   • molecular adaptor activity   • signaling adaptor activity   • multicellular organismal process   • system process   • sensory perception of chemical stimulus   • sensory perception   • nervous system process   • sensory perception of taste   • developmental process   • sensory organ development   • eye development   • animal organ development   • retina development in camera-type eye   • visual system development   • multicellular organism development   • camera-type eye development   • anatomical structure development   • sensory system development   • system development   • cell population proliferation   • cellular process   • cellular response to stimulus   • regulation of biological process   • regulation of cellular process   • response to stimulus   • signaling   • biological regulation   • signal transduction   • cell communication   • response to ketone   • response to prostaglandin   • response to lipid   • response to endogenous stimulus   • response to alcohol   • cellular response to prostaglandin stimulus   • response to oxygen-containing compound   • cellular response to oxygen-containing compound   • cellular response to endogenous stimulus   • cellular response to prostaglandin E stimulus   • cellular response to chemical stimulus   • cellular response to alcohol   • response to hormone   • response to chemical   • cellular response to lipid   • response to prostaglandin E   • cellular response to ketone   • cellular response to hormone stimulus   • small GTPase-mediated signal transduction   • Ras protein signal transduction   • intracellular signal transduction   • intracellular signaling cassette   • phospholipase C-activating G protein-coupled receptor signaling pathway   • G protein-coupled receptor signaling pathway   • cellular response to nitrogen compound   • response to dopamine   • cellular response to dopamine   • response to monoamine   • response to catecholamine   • adenylate cyclase-activating dopamine receptor signaling pathway   • cellular response to catecholamine stimulus   • G protein-coupled dopamine receptor signaling pathway   • response to nitrogen compound   • adenylate cyclase-activating G protein-coupled receptor signaling pathway   • cellular response to monoamine stimulus   • adenylate cyclase-modulating G protein-coupled receptor signaling pathway   • synaptic signaling   • cellular response to acetylcholine   • cell-cell signaling   • acetylcholine receptor signaling pathway   • postsynaptic signal transduction   • G protein-coupled acetylcholine receptor signaling pathway   • response to acetylcholine   • non-motile cilium   • 9+0 non-motile cilium   • cilium   • neuron projection   • photoreceptor disc membrane   • photoreceptor outer segment   • plasma membrane bounded cell projection   • cell projection   • photoreceptor cell cilium   • vacuolar membrane   • lytic vacuole   • vacuole   • lytic vacuole membrane   • bounding membrane of organelle   • lysosomal membrane   • lysosome   • synapse   • cell junction   • G-protein beta-subunit binding   • fibroblast proliferation   • glucagon receptor activity   • peptide receptor activity   • molecular transducer activity   • G protein-coupled receptor activity   • G protein-coupled peptide receptor activity   • signaling receptor activity   • transmembrane signaling receptor activity   • amide binding   • peptide hormone binding   • hormone binding   • enzyme regulator activity   • guanyl nucleotide binding   • GTP binding   • nucleotide binding   • guanyl ribonucleotide binding   • GDP binding   • purine ribonucleotide binding   • ion binding   • anion binding   • molecular function regulator activity   • heterocyclic compound binding   • carbohydrate derivative binding   • ribonucleotide binding   • nucleoside-triphosphatase regulator activity   • GTPase regulator activity   • purine ribonucleoside triphosphate binding   • guanyl-nucleotide exchange factor activity   • nucleoside phosphate binding   • purine nucleotide binding   • small molecule binding   • circulatory system process   • regulation of blood pressure   • regulation of biological quality   • blood circulation   • regulation of biosynthetic process   • positive regulation of biological process   • regulation of macromolecule metabolic process   • gene expression   • macromolecule biosynthetic process   • positive regulation of macromolecule biosynthetic process   • regulation of gene expression   • positive regulation of metabolic process   • biosynthetic process   • positive regulation of gene expression   • positive regulation of biosynthetic process   • regulation of macromolecule biosynthetic process   • metabolic process   • positive regulation of macromolecule metabolic process   • macromolecule metabolic process   • regulation of metabolic process   • positive regulation of cellular process   • hormone-mediated signaling pathway   • response to peptide hormone   • cellular response to peptide hormone stimulus   • response to glucagon   • cellular response to glucagon stimulus   • carbohydrate metabolic process   • energy derivation by oxidation of organic compounds   • glycogen metabolic process   • primary metabolic process   • regulation of generation of precursor metabolites and energy   • generation of precursor metabolites and energy   • regulation of polysaccharide metabolic process   • regulation of primary metabolic process   • glucan metabolic process   • polysaccharide metabolic process   • energy reserve metabolic process   • regulation of glycogen metabolic process   • regulation of carbohydrate metabolic process   • cellular response to nutrient levels   • response to nutrient levels   • cellular response to stress   • response to stress   • response to starvation   • cellular response to starvation   • cell surface receptor signaling pathway   • response to nutrient   • localization   • secretion by cell   • exocytosis   • transport   • secretion   • export from cell   • establishment of localization   • vesicle-mediated transport   • chemical homeostasis   • homeostatic process   • glucose homeostasis   • carbohydrate homeostasis   • endosome   • intracellular vesicle   • cytoplasmic vesicle
SCOP2Domain Identifier• Transducin (heterotrimeric G protein), gamma chain   • G protein-coupled receptor-like   • FnI-like domain
SCOP2Family Identifier• Transducin (heterotrimeric G protein), gamma chain   • G protein-coupled receptor-like   • FnI-like domain
Membrane Protein Annotations-• Orientations of Proteins in Membranes database (OPM)   • Protein Data Bank of Transmembrane Proteins (PDBTM)   • MemProtMD


Details about the values in these tables can be found in the corresponding documentation page .
PDBsumOpen PDBsum Page
ChainA
ProteinG Protein α Sub unit
UniProtP63092
Sequence
>6WHC_Chain_A
TEDQRNEEK AQREANKKI EKQLQKDKQ VYRATHRLL LLGAGIFET 
KFQVDKVNF HMFDVGAQR DERRKWIQC FNDVTAIIF VVASSSTNR 
LQAALKLFD SIWNNKWLR DTSVILFLN KQDLLAEKV LAGKSKIED 
YFPEFARYT TPEDATPEP GEDPRVTRA KYFIRDEFL RISTASGDG 
RHYCYPHFT CAVDTENIR RVFNDCRDI IQRMHLRQY ELL


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainB
ProteinG Protein β Sub unit
UniProtP62873
Sequence
>6WHC_Chain_B
QEAEQLKNQ IRDARKACA DATLSQITN NIDPVGRIQ MRTRRTLRG 
HLAKIYAMH WGTDSRLLV SASQDGKLI IWDSYTTNK VHAIPLRSS 
WVMTCAYAP SGNYVACGG LDNICSIYN LKTREGNVR VSRELAGHT 
GYLSCCRFL DDNQIVTSS GDTTCALWD IETGQQTTT FTGHTGDVM 
SLSLAPDTR LFVSGACDA SAKLWDVRE GMCRQTFTG HESDINAIC 
FFPNGNAFA TGSDDATCR LFDLRADQE LMTYSHDNI ICGITSVSF 
SKSGRLLLA GYDDFNCNV WDALKADRA GVLAGHDNR VSCLGVTDD 
GMAVATGSW DSFLKIWN


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainG
ProteinG Protein γ Sub unit
UniProtP59768
Sequence
>6WHC_Chain_G
VEQLKMEAN IDRIKVSKA AADLMAYCE AHAKEDPLL TPVPASENP 
FR


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainR
ProteinReceptor
UniProtP47871
Sequence
>6WHC_Chain_R
QVMDFLFEK WKLYGDQCH HNLSLLPPP TELVCNRTF DKYSCWPDT 
PANTTANIS CPWYLPWHH KVQHRFVFK RCGPDGQWV RGPRGQPWR 
DASQCQMDG EEIEVQKEV AKMYSSFQV MYTVGYSLS LGALLLALA 
ILGGLSKLH CTRNAIHAN LFASFVLKA SSVLVIDGL LRTRYSTWL 
SDGAVAGCR VAAVFMQYG IVANYCWLL VEGLYLHNL LGLATLPER 
SFFSLYLGI GWGAPMLFV VPWAVVKCL FENVQCWTS NDNMGFWWI 
LRFPVFLAI LINFFIFVR IVQLLVAKL RARQMHYKF RLAKSTLTL 
IPLLGVHEV VFAFTLRSA KLFFDLFLS SFQGLLVAV LYCFLNKEV 
QSELRRRWH RW


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  




This receptor, from the same or other species and bound to the same or other ligands, is also present in the following networks:
Show PDB Class SubFamily Type SubType Species Orthosteric Ligand Other Ligand(s) Protein Partners Resolution Date DOI
9IVMB1PeptideGlucagonGLP-1Homo sapiensGLP-1 (Truncated)LSN3318839chim(NtGi1-Gs)/β2/γ23.222024-11-1310.1016/j.apsb.2024.09.002
9IVM (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensGLP-1 (Truncated)LSN33188393.222024-11-1310.1016/j.apsb.2024.09.002
8YW4B1PeptideGlucagonGIPHomo sapiensRetatrutide-chim(NtGi1-Gs)/β1/γ223.262024-09-18doi.org/10.1038/s41421-024-00700-0
8YW4 (No Gprot) B1PeptideGlucagonGIPHomo sapiensRetatrutide-3.262024-09-18doi.org/10.1038/s41421-024-00700-0
8YW3B1PeptideGlucagonGLP-1Homo sapiensRetatrutide-Gs/β1/γ22.682024-09-18doi.org/10.1038/s41421-024-00700-0
8YW3 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensRetatrutide-2.682024-09-18doi.org/10.1038/s41421-024-00700-0
8YW5B1PeptideGlucagonGlucagonHomo sapiensRetatrutide-Gs/β1/γ22.842024-09-18doi.org/10.1038/s41421-024-00700-0
8YW5 (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensRetatrutide-2.842024-09-18doi.org/10.1038/s41421-024-00700-0
8WG8B1PeptideGlucagonGlucagonHomo sapiens-Peptidechim(NtGi1-Gs)/β1/γ22.712024-03-0610.1038/s41421-024-00649-0
8WG8 (No Gprot) B1PeptideGlucagonGlucagonHomo sapiens-Peptide2.712024-03-0610.1038/s41421-024-00649-0
8WA3B1PeptideGlucagonGIPHomo sapiens--Gs/β1/γ22.862024-03-0610.1038/s41421-024-00649-0
8WA3 (No Gprot) B1PeptideGlucagonGIPHomo sapiens--2.862024-03-0610.1038/s41421-024-00649-0
8WG7B1PeptideGlucagonGLP-1Homo sapiens--Gs/β1/γ22.542024-03-0610.1038/s41421-024-00649-0
8WG7 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens--2.542024-03-0610.1038/s41421-024-00649-0
8JISB1PeptideGlucagonGLP-1Homo sapiensPeptide-15-chim(NtGi1-Gs)/β1/γ22.462023-11-0810.1073/pnas.2303696120
8JIS (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensPeptide-15-2.462023-11-0810.1073/pnas.2303696120
8ITMB1PeptideGlucagonGIPHomo sapiens--Gs/β1/γ23.132023-10-1810.1073/pnas.2306145120
8ITM (No Gprot) B1PeptideGlucagonGIPHomo sapiens--3.132023-10-1810.1073/pnas.2306145120
8ITLB1PeptideGlucagonGIPHomo sapiens--Gs/β1/γ23.232023-10-1810.1073/pnas.2306145120
8ITL (No Gprot) B1PeptideGlucagonGIPHomo sapiens--3.232023-10-1810.1073/pnas.2306145120
8JIRB1PeptideGlucagonGLP-1Homo sapiensSAR425899-chim(NtGi1-Gs)/β1/γ22.572023-09-0610.1073/pnas.2303696120
8JIR (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensSAR425899-2.572023-09-0610.1073/pnas.2303696120
8JIPB1PeptideGlucagonGLP-1Homo sapiensMEDI0382-chim(NtGi1-Gs)/β1/γ22.852023-09-0610.1073/pnas.2303696120
8JIP (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensMEDI0382-2.852023-09-0610.1073/pnas.2303696120
8JITB1PeptideGlucagonGlucagonHomo sapiensMEDI0382-Gs/β1/γ22.912023-09-0610.1073/pnas.2303696120
8JIT (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensMEDI0382-2.912023-09-0610.1073/pnas.2303696120
8JRVB1PeptideGlucagonGlucagonHomo sapiensGlucagon-Arrestin23.32023-08-1610.1038/s41586-023-06420-x
8JRUB1PeptideGlucagonGlucagonHomo sapiens--Arrestin23.52023-08-1610.1038/s41586-023-06420-x
8FU6B1PeptideGlucagonGlucagonHomo sapiensGlucagon derivative ZP3780-Gs/β1/γ22.92023-04-1210.1016/j.cell.2023.02.028
8FU6 (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensGlucagon derivative ZP3780-2.92023-04-1210.1016/j.cell.2023.02.028
9IVGB1PeptideGlucagonGLP-1Homo sapiensGLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ232024-11-2710.1016/j.apsb.2024.09.002
9IVG (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensGLP-1 (Truncated)-32024-11-2710.1016/j.apsb.2024.09.002
9J1PB1PeptideGlucagonGLP-1Homo sapiensg1:Ox-chim(NtGi1-Gs)/β1/γ22.992025-02-2610.1021/jacs.4c12808
9J1P (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensg1:Ox-2.992025-02-2610.1021/jacs.4c12808
8JIUB1PeptideGlucagonGlucagonHomo sapiensSAR425899-Gs/β1/γ22.762023-09-1310.1073/pnas.2303696120
8JIU (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensSAR425899-2.762023-09-1310.1073/pnas.2303696120
8JIQB1PeptideGlucagonGlucagonHomo sapiensPeptide-15-Gs/β1/γ23.42023-09-1310.1073/pnas.2303696120
8JIQ (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensPeptide-15-3.42023-09-1310.1073/pnas.2303696120
7X8SB1PeptideGlucagonGLP-1Homo sapiensWB4-24-Gs/β1/γ23.092022-06-2910.1073/pnas.2200155119
7X8S (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensWB4-24-3.092022-06-2910.1073/pnas.2200155119
7X8RB1PeptideGlucagonGLP-1Homo sapiensBOC5-Gs/β1/γ22.612022-06-2910.1073/pnas.2200155119
7X8R (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensBOC5-2.612022-06-2910.1073/pnas.2200155119
7S15B1PeptideGlucagonGLP-1Homo sapiensPubChem 134611223--3.82022-06-0810.1021/acs.jmedchem.1c01856
7RBTB1PeptideGlucagonGIPHomo sapiensTirzepatidePubChem 163183774chim(NtGi1-Gs)/β1/γ23.082022-04-1310.1073/pnas.2116506119
7RBT (No Gprot) B1PeptideGlucagonGIPHomo sapiensTirzepatidePubChem 1631837743.082022-04-1310.1073/pnas.2116506119
7RA3B1PeptideGlucagonGIPHomo sapiensGIP-chim(NtGi1-Gs)/β1/γ23.242022-04-1310.1073/pnas.2116506119
7RA3 (No Gprot) B1PeptideGlucagonGIPHomo sapiensGIP-3.242022-04-1310.1073/pnas.2116506119
7RGPB1PeptideGlucagonGLP-1Homo sapiensTirzepatide-chim(NtGi1-Gs)/β1/γ22.92022-04-1310.1073/pnas.2116506119
7RGP (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensTirzepatide-2.92022-04-1310.1073/pnas.2116506119
7RG9B1PeptideGlucagonGLP-1Homo sapiens--chim(NtGi1-Gs)/β1/γ23.22022-04-1310.1073/pnas.2116506119
7RG9 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens--3.22022-04-1310.1073/pnas.2116506119
7V9LB1PeptideGlucagonGHRH (SV1)Homo sapiens--chim(NtGi1-Gs)/β1/γ22.62022-04-0610.1073/pnas.2106606118
7V9L (No Gprot) B1PeptideGlucagonGHRH (SV1)Homo sapiens--2.62022-04-0610.1073/pnas.2106606118
7VBHB1PeptideGlucagonGLP-1Homo sapiensPeptide-20-Gs/β1/γ232022-04-0610.1038/s41467-022-28683-0
7VBH (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensPeptide-20-32022-04-0610.1038/s41467-022-28683-0
7VABB1PeptideGlucagonGIPHomo sapiensNon-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ23.22022-03-0210.1038/s41467-022-28683-0
7VAB (No Gprot) B1PeptideGlucagonGIPHomo sapiensNon-Acylated Tirzepatide-3.22022-03-0210.1038/s41467-022-28683-0
7FIYB1PeptideGlucagonGIPHomo sapiensTirzepatide-Gs/β1/γ23.42022-03-0210.1038/s41467-022-28683-0
7FIY (No Gprot) B1PeptideGlucagonGIPHomo sapiensTirzepatide-3.42022-03-0210.1038/s41467-022-28683-0
7VBIB1PeptideGlucagonGLP-1Homo sapiensNon-Acylated Tirzepatide-Gs/β1/γ232022-03-0210.1038/s41467-022-28683-0
7VBI (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensNon-Acylated Tirzepatide-32022-03-0210.1038/s41467-022-28683-0
7FIMB1PeptideGlucagonGLP-1Homo sapiensTirzepatide-Gs/β1/γ23.42022-03-0210.1038/s41467-022-28683-0
7FIM (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensTirzepatide-3.42022-03-0210.1038/s41467-022-28683-0
7V35B1PeptideGlucagonGlucagonHomo sapiensPeptide-20-Gs/β1/γ23.52022-03-0210.1038/s41467-022-28683-0
7V35 (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensPeptide-20-3.52022-03-0210.1038/s41467-022-28683-0
7FINB1PeptideGlucagonGIPHomo sapiensPeptide-20; GGL-Gs/β1/γ23.12022-02-2310.1038/s41467-022-28683-0
7FIN (No Gprot) B1PeptideGlucagonGIPHomo sapiensPeptide-20; GGL-3.12022-02-2310.1038/s41467-022-28683-0
7LLYB1PeptideGlucagonGLP-1Homo sapiensOxyntomodulin-Gs/β1/γ23.32022-01-1210.1038/s41467-021-27760-0
7LLY (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensOxyntomodulin-3.32022-01-1210.1038/s41467-021-27760-0
7LLLB1PeptideGlucagonGLP-1Homo sapiensExendin-4-Gs/β1/γ23.72022-01-1210.1038/s41467-021-27760-0
7LLL (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensExendin-4-3.72022-01-1210.1038/s41467-021-27760-0
7S3IB1PeptideGlucagonGLP-1Homo sapiens--Gs/β1/γ22.512022-01-0510.1038/s41589-021-00945-w
7S3I (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens--2.512022-01-0510.1038/s41589-021-00945-w
7S1MB1PeptideGlucagonGLP-1Homo sapiensEx4-D-Ala-Gs/β1/γ22.412022-01-0510.1038/s41589-021-00945-w
7S1M (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensEx4-D-Ala-2.412022-01-0510.1038/s41589-021-00945-w
7V9MB1PeptideGlucagonGHRH (SV1)Homo sapiensSomatoliberin-Gs/β1/γ23.292021-10-2010.1073/pnas.2106606118
7V9M (No Gprot) B1PeptideGlucagonGHRH (SV1)Homo sapiensSomatoliberin-3.292021-10-2010.1073/pnas.2106606118
7RTBB1PeptideGlucagonGLP-1Homo sapiensPeptide-19-Gs/β1/γ22.142021-10-0610.1016/j.bbrc.2021.09.016
7RTB (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensPeptide-19-2.142021-10-0610.1016/j.bbrc.2021.09.016
7EVMB1PeptideGlucagonGLP-1Homo sapiens-PubChem 156022738Gs/β1/γ22.52021-08-1110.1038/s41467-021-24058-z
7EVM (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens-PubChem 1560227382.52021-08-1110.1038/s41467-021-24058-z
7DURB1PeptideGlucagonGLP-1Homo sapiens-PubChem 156022738Gs/β1/γ23.32021-08-1110.1038/s41467-021-24058-z
7DUR (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens-PubChem 1560227383.32021-08-1110.1038/s41467-021-24058-z
7DTYB1PeptideGlucagonGIPHomo sapiensGIP-Gs/β1/γ22.982021-08-0410.7554/eLife.68719
7DTY (No Gprot) B1PeptideGlucagonGIPHomo sapiensGIP-2.982021-08-0410.7554/eLife.68719
7KI1B1PeptideGlucagonGLP-1Homo sapiensTaspoglutide-Gs/β1/γ22.52021-08-0410.1016/j.celrep.2021.109374
7KI1 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensTaspoglutide-2.52021-08-0410.1016/j.celrep.2021.109374
7KI0B1PeptideGlucagonGLP-1Homo sapiensSemaglutide-Gs/β1/γ22.52021-08-0410.1016/j.celrep.2021.109374
7KI0 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensSemaglutide-2.52021-08-0410.1016/j.celrep.2021.109374
7DUQB1PeptideGlucagonGLP-1Homo sapiensGLP-1PubChem 156022738Gs/β1/γ22.52021-07-1410.1038/s41467-021-24058-z
7DUQ (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensGLP-1PubChem 1560227382.52021-07-1410.1038/s41467-021-24058-z
7E14B1PeptideGlucagonGLP-1Homo sapiensOrforglipronPubChem 156022738Gs/β1/γ22.92021-07-0710.1038/s41467-021-24058-z
7E14 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensOrforglipronPubChem 1560227382.92021-07-0710.1038/s41467-021-24058-z
7LCKB1PeptideGlucagonGLP-1Homo sapiensDanuglipron--3.242021-01-2010.1016/j.str.2021.04.008
7LCJB1PeptideGlucagonGLP-1Homo sapiensDanuglipron--2.822021-01-2010.1016/j.str.2021.04.008
7LCIB1PeptideGlucagonGLP-1Homo sapiensDanuglipron-Gs/β1/γ22.92021-01-2010.1016/j.str.2021.04.008
7LCI (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensDanuglipron-2.92021-01-2010.1016/j.str.2021.04.008
7D68B1PeptideGlucagonGLP-2Homo sapiensGLP-2-Gs/β1/γ232020-12-1610.1038/s41422-020-00442-0
7D68 (No Gprot) B1PeptideGlucagonGLP-2Homo sapiensGLP-2-32020-12-1610.1038/s41422-020-00442-0
6XOXB1PeptideGlucagonGLP-1Homo sapiensOrforglipron-chim(NtGi1-Gs)/β1/γ23.12020-11-1810.1073/pnas.2014879117
6XOX (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensOrforglipron-3.12020-11-1810.1073/pnas.2014879117
7CZ5B1PeptideGlucagonGHRHHomo sapiensSomatoliberin-Gs/β1/γ22.62020-11-1810.1038/s41467-020-18945-0
7CZ5 (No Gprot) B1PeptideGlucagonGHRHHomo sapiensSomatoliberin-2.62020-11-1810.1038/s41467-020-18945-0
7D3SB1PeptideGlucagonSecretinHomo sapiensSecretin-Gs/β1/γ22.92020-11-0410.1016/j.bbrc.2020.08.042
7D3S (No Gprot) B1PeptideGlucagonSecretinHomo sapiensSecretin-2.92020-11-0410.1016/j.bbrc.2020.08.042
6X1AB1PeptideGlucagonGLP-1Homo sapiensDanuglipron-Gs/β1/γ22.52020-09-0910.1016/j.molcel.2020.09.020
6X1A (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensDanuglipron-2.52020-09-0910.1016/j.molcel.2020.09.020
6X19B1PeptideGlucagonGLP-1Homo sapiensCHU-128-Gs/β1/γ22.12020-09-0910.1016/j.molcel.2020.09.020
6X19 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensCHU-128-2.12020-09-0910.1016/j.molcel.2020.09.020
6X18B1PeptideGlucagonGLP-1Homo sapiensGLP-1-Gs/β1/γ22.12020-09-0910.1016/j.molcel.2020.09.020
6X18 (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensGLP-1-2.12020-09-0910.1016/j.molcel.2020.09.020
7C2EB1PeptideGlucagonGLP-1Homo sapiensPubChem 149050799-Gs/β1/γ24.22020-08-2610.1038/s41422-020-0384-8
7C2E (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensPubChem 149050799-4.22020-08-2610.1038/s41422-020-0384-8
6WPWB1PeptideGlucagonGlucagonHomo sapiensGlucagon derivative ZP3780-Gs/β1/γ23.12020-08-1210.1126/science.aba3373
6WPW (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensGlucagon derivative ZP3780-3.12020-08-1210.1126/science.aba3373
6WZGB1PeptideGlucagonSecretinHomo sapiensSecretin-Gs/β1/γ22.32020-08-1210.1038/s41467-020-17791-4
6WZG (No Gprot) B1PeptideGlucagonSecretinHomo sapiensSecretin-2.32020-08-1210.1038/s41467-020-17791-4
6WI9B1PeptideGlucagonSecretinHomo sapiensSecretin-Gs/β1/γ24.32020-08-1210.1038/s41467-020-17791-4
6WI9 (No Gprot) B1PeptideGlucagonSecretinHomo sapiensSecretin-4.32020-08-1210.1038/s41467-020-17791-4
6VCBB1PeptideGlucagonGLP-1Homo sapiensGLP-1LSN3160440Gs/β1/γ23.32020-07-2210.1038/s41589-020-0589-7
6VCB (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensGLP-1LSN31604403.32020-07-2210.1038/s41589-020-0589-7
6WHCB1PeptideGlucagonGlucagonHomo sapiensGlu16 analog of GCG-Gs/β1/γ23.42020-05-2710.1074/jbc.RA120.013793
6WHC (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensGlu16 analog of GCG-3.42020-05-2710.1074/jbc.RA120.013793
6LMLB1PeptideGlucagonGlucagonHomo sapiensGlucagon-Gi1/β1/γ13.92020-04-0110.1126/science.aaz5346
6LML (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensGlucagon-3.92020-04-0110.1126/science.aaz5346
6LMKB1PeptideGlucagonGlucagonHomo sapiensGlucagon-Gs/β1/γ23.72020-04-0110.1126/science.aaz5346
6LMK (No Gprot) B1PeptideGlucagonGlucagonHomo sapiensGlucagon-3.72020-04-0110.1126/science.aaz5346
6LN2B1PeptideGlucagonGLP-1Homo sapiens-PubChem 68178630-3.22020-03-1810.1038/s41467-020-14934-5
6ORVB1PeptideGlucagonGLP-1Homo sapiens-TT-OAD2Gs/β1/γ232020-01-0810.1038/s41586-019-1902-z
6ORV (No Gprot) B1PeptideGlucagonGLP-1Homo sapiens-TT-OAD232020-01-0810.1038/s41586-019-1902-z
6KK7B1PeptideGlucagonGLP-1Homo sapiens-PubChem 68178630-3.12019-11-1310.1107/S2052252519013496
6KK1B1PeptideGlucagonGLP-1Homo sapiens-PubChem 68178630-2.82019-11-1310.1107/S2052252519013496
6KJVB1PeptideGlucagonGLP-1Homo sapiens-PubChem 68178630-2.82019-11-1310.1107/S2052252519013496
6B3JB1PeptideGlucagonGLP-1Homo sapiensExendin-P5-Gs/β1/γ23.32018-02-2110.1038/nature25773
6B3J (No Gprot) B1PeptideGlucagonGLP-1Homo sapiensExendin-P5-3.32018-02-2110.1038/nature25773
5YQZB1PeptideGlucagonGlucagonHomo sapiensGlucagon analogue--32018-01-1710.1038/nature25153
5NX2B1PeptideGlucagonGLP-1Homo sapiensGLP-1 (Truncated)--3.72017-06-1410.1038/nature22800
5VEWB1PeptideGlucagonGLP-1Homo sapiens-PF-06372222-2.72017-05-2410.1038/nature22378
5XF1B1PeptideGlucagonGlucagonHomo sapiens-NNC0640-3.192017-05-2410.1038/nature22363
5XEZB1PeptideGlucagonGlucagonHomo sapiens-NNC0640-32017-05-2410.1038/nature22363
5VAIB1PeptideGlucagonGLP-1Oryctolagus cuniculusGLP-1-Gs/β1/γ24.12017-05-2410.1038/nature22394
5VAI (No Gprot) B1PeptideGlucagonGLP-1Oryctolagus cuniculusGLP-1-4.12017-05-2410.1038/nature22394
5VEXB1PeptideGlucagonGLP-1Homo sapiens-NNC0640-32017-05-1710.1038/nature22378
5EE7B1PeptideGlucagonGlucagonHomo sapiens-MK0893-2.52016-04-2010.1038/nature17414
4L6RB1PeptideGlucagonGlucagonHomo sapiens---3.32013-07-2410.1038/nature12393




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