Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
11x27 2.99405
21x39 7.8925437
31x50 6.4425409
41x53 2.0375409
51x57 3.8375407
62x37 5.10254147
72x38 8.195426
82x42 5.64167627
92x44 3.5575406
102x46 2.968529
112x49 3.5975428
122x53 5.074506
132x56 3.718537
142x60 8.4575436
15E1x50 4.88857738
163x28 5.714536
173x29 7.8625436
183x32 7.4775436
193x33 3.055405
203x36 6.872527
213x37 3.87667627
223x42 6.475827
233x44 4.245428
243x45 5.47426
253x47 3.6725429
263x49 6.65428
27I2x57 6.404527
284x50 4.63857729
294x65 5.445435
30E2.Y193 6.03254154
31E2.F194 6.59534
325x43 6.685425
335x50 5.6125428
345x53 3.3125426
355x58 4.83833628
365x61 4.065408
376x44 6.57629
386x47 5.72428
396x48 9.16529
406x49 7.325405
416x51 8.1925406
426x61 4.5625434
436x64 3.4225161
447x38 7.4725435
457x42 5.4275407
467x45 9.088529
477x53 4.765629
48Lig 33.4452630
49G.HN.11 2.916502
50G.HN.43 2.8354119
51G.HN.47 2.8354116
52G.S1.02 5.034545
53G.S1.04 4.075447
54G.S1.06 4.2448
55G.S1.07 4.506519
56G.s1h1.01 2.45419
57G.s1h1.02 2.475407
58G.H1.01 4.355449
59G.H1.07 4.975409
60G.H1.08 5.8725408
61G.S2.01 3.5075419
62G.S2.08 7.38667645
63G.S3.02 6.9025414
64G.S3.03 6.23429747
65G.S3.04 7.16416
66G.S3.06 6.59333615
67G.s3h2.03 6.54419
68G.H2.03 4.514519
69G.H2.06 4.705819
70G.H2.07 5.50571719
71G.H2.09 6.0725418
72G.H2.10 3.4975417
73G.h2s4.01 6.33714719
74G.S4.02 5.3675418
75G.S4.03 3.145447
76G.S4.04 5.01143719
77G.s4h3.01 5.5497
78G.s4h3.04 8.454598
79G.H3.06 3.5725406
80G.H3.08 3.6275419
81G.H3.09 4.988509
82G.H3.13 4.40254135
83G.H3.17 6.82615
84G.H3.18 7.8825419
85G.S5.03 2.978548
86G.S5.04 3.9275409
87G.S5.05 4.12429749
88G.HG.04 5.04571799
89G.HG.08 4.262596
90G.HG.15 3.64333697
91G.hgh4.01 4.2075496
92G.hgh4.02 6.45857797
93G.H4.03 3.35404
94G.H4.11 3.156597
95G.H4.15 3.61508
96G.h4s6.10 2.86403
97G.h4s6.11 4.48254137
98G.S6.02 3.44857747
99G.S6.05 4.02494
100G.H5.03 5.23448
101G.H5.08 6.62548
102G.H5.15 3.3575407
103G.H5.20 4.758509
104G.H5.26 8.006505
105b.h2x5 3.735455
106b.lhb1x3 4.95452
107b.lhb1x6 5.3575453
108b.b1x3 4.4175487
109b.l1x3 7.703336119
110b.b2x1 6.992518
111b.b2x5 7.555687
112b.l2x5 10.785485
113b.b3x3 4.0875418
114b.b3x4 5.37254119
115b.b4x3 4.6275417
116b.b4x4 7.79254118
117b.b4x6 8.192867119
118b.l4x1 4.17485
119b.l4x2 12.155484
120b.b5x2 5.9225407
121b.b5x3 6.037119
122b.b5x5 5.64405
123b.b5x7 6.115417
124b.l5x1 4.8775418
125b.l5x5 7.69625819
126b.b6x5 4.12833616
127b.l6x1 2.075416
128b.l6x3 4.9625416
129b.b7x1 6.225414
130b.b7x4 3.154518
131b.b7x5 1.9419
132b.l7x2 4.50857719
133b.b8x2 4.18418
134b.b8x3 3.388516
135b.b8x4 5.32286716
136b.l8x8 5.4725414
137b.l8x10 4.72414
138b.b9x3 5.0725416
139b.b9x4 6.6409
140b.l9x3 7.23143719
141b.l9x5 1.8725408
142b.l9x6 3.4681018
143b.l9x7 2.8775417
144b.b10x2 5406
145b.b10x5 3.9925419
146b.l10x1 4.52403
147b.b11x2 3.762517
148b.b11x4 4.584519
149b.l11x1 2.975419
150b.l11x2 9.6975419
151b.b12x3 3.738578
152b.b12x6 8.545618
153b.b13x5 4.315474
154b.b13x7 9.078577
155b.l13x3 7.80667679
156b.l13x6 5.2375419
157b.l13x7 4.344579
158b.b14x3 5.372575
159b.b15x1 7.50167679
160b.b15x3 4.205679
161b.l15x1 5.9125417
162b.l15x2 4.962579
163b.b16x4 10.5025476
164b.b16x6 9.29667678
165b.b17x5 8.4925467
166b.b17x7 9.5975468
167b.l17x3 7.2669
168b.l17x6 6.102519
169b.b18x3 5.095468
170b.b18x5 5.6405
171b.l18x1 5.99286756
172b.l18x3 7.2525455
173b.b19x2 6.615666
174b.b19x4 4.27167668
175b.b19x5 2.7025405
176b.l19x1 6.195419
177b.l19x2 5.6175409
178b.b20x4 10.814568
179b.b20x6 6.65833666
180b.l20x2 9.1775409
181b.b21x7 4.68286705
182b.l21x5 5.682514
183b.l21x7 3.495415
184b.b22x3 2.59406
185b.b22x5 6.5425457
186b.l22x1 4.645459
187b.l22x4 2.19459
188b.l22x5 6.4559
189b.b23x1 4.695405
190b.b23x5 2.78254107
191b.b23x6 6.80429717
192b.l23x1 6.2075416
193b.b24x3 4.2954105
194b.b24x4 5.696516
195b.b24x5 4.2875405
196b.b24x6 6.215418
197b.b25x3 6.224515
198b.b25x6 3.525413
199b.l25x3 10.1665109
200b.b26x3 4.885106
201b.l26x1 6.3225487
202b.b27x1 3.7975406
203b.b27x3 4.8754108
204b.l27x1 11.5914719
205b.l27x2 9.60754109
206b.b28x3 4.5154117
207b.b28x4 6.584106
208b.b28x6 8.4265109
209b.b28x7 9.29489
210g.h1x11 2.125409
211g.h2x11 6.6325456
212g.ctx3 6.642559
213g.ctx4 3.1407
214g.ctx6 4.7725456
215g.ctx14 5.22589
216g.ctx16 5.20556988
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
16x48 7x45 24.434417.98YesYes299
26x48 6x51 18.27261.93YesYes096
36x51 7x38 16.431411.22YesYes065
47x38 Lig 16.05386.29YesYes350
52x50 7x46 19.36227.78NoNo098
62x53 7x46 19.16284.19YesNo068
72x53 3x32 15.998912.38YesYes066
83x32 Lig 16.24599.74YesYes360
93x34 4x50 13.84722.35NoYes069
103x34 4x57 13.03594.64NoNo067
112x38 2x42 13.9348.21YesYes267
122x42 3x42 25.29874.13YesYes277
132x46 2x50 22.62144.07YesNo099
143x42 4x50 22.444510.02YesYes279
152x42 3x49 13.9342.3YesYes278
162x38 I2x57 14.286613.36YesYes267
173x49 I2x57 14.286611.91YesYes287
182x46 7x53 23.36622.34YesYes299
197x49 7x53 32.66074.65NoYes299
207x45 7x49 32.619710.2YesNo299
213x50 7x53 59.68847.2NoYes099
223x50 G.H5.23 67.04764.18NoNo094
233x53 G.H5.23 67.22761.81NoNo084
243x53 G.H5.19 96.60673.13NoNo088
25G.H5.15 G.H5.19 96.77772.83YesNo078
26G.S1.04 G.S4.03 97.88714.28YesYes477
27G.S1.02 G.S1.04 48.40432.98YesYes457
28G.H5.11 G.S1.02 48.36496.41NoYes485
29G.H5.11 G.H5.15 97.28943.07NoYes087
30G.S1.04 G.S3.03 49.25656.09YesYes477
31G.H5.11 G.S3.03 49.09466.55NoYes487
32b.b26x1 b.b26x2 14.20363.44NoNo097
33b.b26x1 b.l27x1 14.37088.65NoYes099
34G.H3.17 b.l27x1 12.31052.81YesYes159
35G.H3.15 G.H3.17 36.79075.65NoYes185
36G.H3.15 G.H3.18 37.03024.83NoYes189
37G.H3.18 G.S4.02 36.931111.3YesYes198
38G.S1.07 G.S4.02 37.20434.28YesYes198
39G.S1.07 G.s1h1.01 88.74461.71YesYes199
40G.s1h1.01 G.s1h1.05 91.00531.86YesNo099
41G.s1h1.02 G.s1h1.05 90.99721.71YesNo079
42G.s1h1.02 G.s1h1.03 1001.95YesNo078
43G.H1.01 G.s1h1.03 99.98941.74YesNo098
44G.H1.01 G.S1.06 99.75795.64YesYes498
45G.S1.06 G.S4.03 98.39532.85YesYes487
46G.S1.05 G.h2s4.01 72.365812.18NoYes199
47G.S1.05 G.S1.07 72.25475.54NoYes199
48G.H2.07 b.l9x6 15.11424.82YesYes198
49G.H2.07 G.h2s4.01 30.39224.01YesYes199
50b.l7x2 b.l9x6 16.58992.34YesYes198
51G.h2s4.01 b.l7x2 34.01842.44YesYes199
52G.H2.03 G.H2.07 15.62262.18YesYes199
53G.H2.03 G.H2.06 10.18884.05YesYes199
54G.H2.06 b.l9x6 22.50583.58YesYes198
55G.H3.09 G.S4.04 10.202310.72YesYes099
56G.H4.15 G.S4.06 11.23672.62YesNo087
57G.H4.11 G.H4.15 13.50842.51YesYes078
58b.b6x1 b.l7x2 20.3252.83NoYes199
59b.b6x1 b.l7x1 20.94781.75NoNo199
60b.b7x5 b.l7x1 13.94782.11YesNo199
61b.b6x2 b.b7x5 14.73641.82NoYes089
62b.b10x2 b.b6x2 15.41963.38YesNo068
63b.b10x2 b.b14x3 15.66527.94YesYes065
64b.l17x5 b.l17x6 20.70135.89NoYes169
65b.l17x5 b.l19x2 35.28045.89NoYes069
66b.b19x6 b.l19x2 17.56375.89NoYes099
67b.b19x6 b.l17x3 14.95236.97NoYes099
68b.b20x6 b.l17x3 12.15534.53YesYes669
69b.b17x7 b.b20x6 23.93087.5YesYes686
70G.H2.06 b.l17x6 15.77958.3YesYes199
71G.H2.06 b.l19x1 15.77992.77YesYes199
72b.l17x5 b.l19x1 15.4575.89NoYes169
73b.b20x2 b.l19x2 16.15982.89NoYes069
74b.b20x2 b.b20x4 14.4096.47NoYes068
75b.b20x4 b.b20x6 11.9216.41YesYes686
76G.H3.17 b.l25x6 24.67136YesNo158
77b.l23x1 b.l25x6 27.082515.48YesNo168
78b.l21x7 b.l23x1 11.45853.11YesYes156
79b.b23x6 b.l21x7 10.06422.69YesYes175
80b.b17x5 b.b17x7 16.015812.88YesYes678
81b.b16x5 b.b17x5 12.07967.99NoYes657
82b.b16x5 b.l14x6 10.24114.15NoNo653
833x53 I2x57 29.31752.77NoYes087
84G.S1.07 G.S4.04 20.48082.44YesYes199
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
LigNT.G291.743YesNo0101
NT.A30NT.P311.873NoNo4411
LigNT.A301.813YesNo0401
NT.K34NT.P315.020NoNo5421
LigNT.P31113YesNo0401
E3.C277NT.C327.280NoNo6921
LigNT.C325.383YesNo0901
7x31NT.H335.043NoNo4311
LigNT.H334.023YesNo0301
1x277x312.920YesNo5421
1x282x6611.193NoNo5412
1x317x354.930NoNo3421
1x351x3916.410NoYes6721
1x357x357.990NoNo6421
1x392x612.673YesNo7712
1x397x428.383YesYes7712
1x39Lig4.113YesYes7010
2x533x3212.380YesYes6621
2x537x423.730YesYes6722
2x562x607.283YesYes7621
2x563x283.893YesYes7622
2x602x632.473YesNo6412
2x603x2823YesYes6612
2x60Lig22.083YesYes6010
2x63E1x504.940NoYes4822
3x25E1x503.923NoYes9822
3x28E1x503.013YesYes6822
E1x50E2x509.143YesNo8921
3x25E2x507.283NoNo9921
3x264x6530NoYes7521
3x293x301.823YesNo6612
3x293x332.743YesYes6512
3x294x6514.133YesYes6511
3x29Lig12.763YesYes6010
3x323x332.183YesYes6512
3x327x385.613YesYes6511
3x32Lig9.743YesYes6010
4x614x651.820NoYes4521
4x61E2.F1943.010NoYes4421
4x64E2.F1947.50NoYes4421
4x65Lig2.833YesYes5010
E2.D185Lig8.610NoYes3010
E2x50Lig6.13NoYes9010
E2x51E2x524.063NoNo4411
E2x51Lig6.633NoYes4010
E2x52Lig14.563NoYes4010
5x36E2.F1946.043NoYes3411
5x39E2.F19412.440NoYes5421
E2.F194Lig3.963YesYes4010
5x36Lig7.453NoYes3010
6x517x3811.220YesYes6521
6x547x343.170NoNo5421
6x586x613.960NoYes4421
6x61E3.S2752.893YesNo4311
6x617x272.833YesNo4211
6x61Lig8.573YesYes4010
E3.S275Lig8.93NoYes3010
7x27Lig12.483NoYes2010
7x31Lig4.633NoYes4010
7x34Lig4.343NoYes4010
7x35Lig3.033NoYes4010
7x387x426.773YesYes5712
7x38Lig6.293YesYes5010
1x28Lig1.613NoYes5010

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
100.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
66.67Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
66.67Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
65.22Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
64.00Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
64.00Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
60.00Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
58.33Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
57.69Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
57.69Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
56.52Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
54.55Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
54.17Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
54.17Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
53.85Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
51.85Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
51.72Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
50.00Single4XT1Fractalkine4XT1-US28-Fractalkine
50.00Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
50.00Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
50.00Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
48.28Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
48.28Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
48.28Consensusbradykinin_onOrthosteric Ligandbk2_on
48.28Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
48.28Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
48.15Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
48.15Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
48.15Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
48.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
48.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
47.83Single8ZPLHF511168ZPL-CXCR4-HF51116
47.83Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
46.67Single5GLHEndothelin-15GLH-ETB-Endothelin-1
46.43Single4XT3Fractalkine4XT3-US28-Fractalkine
46.43Single7SK3CXCL127SK3-ACKR3-CXCL12
46.43Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
46.43Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
46.15Single3OE0CVX153OE0-CXCR4-CVX15
46.15Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
45.83Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
45.83Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
45.83Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
45.83Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
45.83Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
45.45Single7F1TMIP-1a7F1T-CCR5-MIP-1a
45.00Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
44.83Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
44.83Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
44.44Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
44.44Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
44.44Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
44.44Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
44.44Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
44.44Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
44.44Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
44.00Single8XWNCXCL88XWN-CXCR2-CXCL8
44.00Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
43.48Single6OS2TRV0266OS2-AT1-TRV026
43.48Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
43.48Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
43.48Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
42.86Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
42.86Single6D27CAY104716D27-DP2-CAY10471
42.86Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
42.86Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
42.86Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
42.31Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
42.31Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
42.31Single7XNACYN1548067XNA-SST2-CYN154806
42.31Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
42.31Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
41.94Single6IGKEndothelin-36IGK-ETB-Endothelin-3
41.94Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
41.67Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
41.67Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
41.67Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.91Single6D26Fevipiprant6D26-DP2-Fevipiprant
40.91Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
40.91Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
40.91Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
40.91Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
40.91Consensusdp_offOrthosteric Liganddp2_off
40.74Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
40.74Consensusangiotensin_onOrthosteric Ligandat1_on
40.74Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
40.74Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
40.62Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
40.00Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
40.00Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
40.00Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
40.00Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
40.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
40.00Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
40.00Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
39.39Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
39.29Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
39.29Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
39.13Single6OS1TRV0266OS1-AT1-TRV026
39.13Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
39.13Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
39.13Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
39.13Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
39.13Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
39.13Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
39.13Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
39.13Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
38.71Consensusendothelin_onOrthosteric Ligandetb_on eta_on
38.46Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
38.46Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
38.46Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
38.46Consensussomatostatin_offOrthosteric Ligandsst2_off
38.10Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
38.10Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
38.10Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
38.10Single8ZPMAMD0708ZPM-CXCR4-AMD070
37.93Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
37.93Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
37.93Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
37.93Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
37.93Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
37.93Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
37.50Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
37.50Single6YVRNTS8-136YVR-NTS1-NTS8-13
37.50Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
37.50Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
37.50Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
37.50Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
37.50Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
37.50Single8XWACXCL18XWA-CXCR2-CXCL1
37.50Single8XWMCXCL68XWM-CXCR2-CXCL6
37.50Single8XWSCXCL58XWS-CXCR2-CXCL5
37.50Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
37.50Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
37.50Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
37.50Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
37.50Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
37.50Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
37.50Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
37.50Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
37.04Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
37.04Single7SK5CXCL127SK5-ACKR3-CXCL12
37.04Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
37.04Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.04Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
37.04Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
36.67Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
36.67Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
36.36Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
36.36Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
36.36Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
36.36Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
36.36Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
36.00Single4BUONeurotensin4BUO-NTS1-Neurotensin
36.00Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
36.00Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
36.00Single8XVUCXCL28XVU-CXCR2-CXCL2
36.00Single8XWFCXCL38XWF-CXCR2-CXCL3
36.00Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
36.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
36.00Consensusprostanoid_offOrthosteric Ligandep_off dp_off
35.71Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
35.71Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
35.71Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
35.71Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
35.71Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
35.71Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
35.48Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
35.48Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
35.29Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
35.00Single3OE9IT1t3OE9-CXCR4-IT1t
34.78Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
34.78Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
34.78Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
34.78Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
34.78Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
34.62Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
34.62Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
34.62Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
34.62Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
34.62Single9IPYJR14a9IPY-C3aB-JR14a
34.48Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
34.48Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
34.48Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
34.48Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
34.48Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.48Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
34.48Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
34.48Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
34.48Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
34.48Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
34.48Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
34.48Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
34.48Consensusvasop-oxy_onOrthosteric Ligandv2_on
34.48Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
34.38Single6IGLIRL16206IGL-ETB-IRL1620
34.38Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
34.38Single8IY6Endothelin-18IY6-ETB-Endothelin-1
34.29Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
33.33Single3ODUIT1t3ODU-CXCR4-IT1t
33.33Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
33.33Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single7PX4PSB-21137PX4-A2A-PSB-2113
33.33Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
33.33Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
33.33Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
33.33Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
33.33Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
33.33Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
33.33Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
33.33Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
33.33Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
33.33Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
33.33Single8GNGIstradefylline8GNG-A2A-Istradefylline
33.33Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
33.33Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
33.33Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
33.33Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
33.33Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
33.33Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
33.33Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
33.33Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
33.33Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
33.33Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
33.33Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
33.33Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
33.33Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8ZRTET-18ZRT-ETB-ET-1
33.33Single8ZWFJR14a8ZWF-C3aB-JR14a
33.33Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
33.33Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
33.33Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
33.33Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
33.33Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
33.33Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
33.33Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
33.33Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
33.33Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
33.33Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
33.33Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
33.33Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
33.33Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusneurotensin_onOrthosteric Ligandnts1_on
33.33Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
33.33Consensuspac_onOrthosteric Ligandpac1_on
32.26Single6FJ3PTH6FJ3-PTH1-PTH
32.26Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
32.26Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
32.26Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
32.26Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
32.26Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
32.26Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
32.26Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
32.26Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
32.26Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
32.14Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
32.14Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
32.14Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
32.14Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
32.14Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
32.14Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
32.14Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
32.14Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
32.14Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
32.14Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
32.14Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
32.14Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
32.14Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
32.14Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
32.00Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
32.00Single4XEENeurotensin4XEE-NTS1-Neurotensin
32.00Single4XESNeurotensin4XES-NTS1-Neurotensin
32.00Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
32.00Single7K15MKD0467K15-BLT1-MKD046-Na
32.00Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
32.00Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
32.00Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
32.00Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
32.00Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
32.00Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
32.00Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
32.00Consensuslpl_offOrthosteric Ligands1p_off lpa_off
32.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
31.82Single7AROLUF58337ARO-A2A-LUF5833-Na
31.82Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
31.82Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
31.82Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
31.82Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
31.82Single8K5CAcipimox8K5C-HCA2-Acipimox
31.82Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
31.82Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
31.82Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
31.82Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
31.82Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
31.82Consensushca_onOrthosteric Ligandhca2_on
31.82Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
31.25Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
31.25Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
31.25Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
31.25Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
31.25Single9KDFRES-701-39KDF-ETB-RES-701-3
31.25Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
31.25Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
31.03Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
31.03Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
31.03Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
31.03Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
31.03Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
31.03Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.03Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
31.03Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
31.03Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
31.03Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
30.77Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
30.77Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
30.77Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
30.77Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
30.77Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
30.77Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
30.77Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
30.77Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
30.77Consensuscck_onOrthosteric Ligandccka_on cckb_on
30.77Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
30.56Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
30.43Single4YAYZD-71554YAY-AT1-ZD-7155
30.43Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
30.43Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
30.43Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
30.43Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
30.43Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
30.43Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
30.43Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
30.43Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
30.43Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
30.43Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
30.43Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
30.43Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
30.43Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
30.43Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
30.43Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
30.43Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
30.43Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
30.43Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
30.43Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
30.43Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
30.43Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
30.43Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
30.43Consensushca_on_gpOrthosteric Ligandhca2_on_gp
30.43Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
30.30Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
30.30Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
30.30Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
30.00Single3OE6IT1t3OE6-CXCR4-IT1t
30.00Single6JODAngiotensin II6JOD-AT2-Angiotensin II
30.00Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
30.00Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
30.00Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
30.00Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
30.00Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
30.00Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
30.00Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
30.00Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
30.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
30.00Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
29.63Single6KNMJN241-96KNM-Apelin-JN241-9
29.63Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
29.63Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
29.63Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
29.63Single8QJ2pN1628QJ2-MC4-pN162-Gs
29.63Single8XQJJN2418XQJ-Apelin-JN241
29.63Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
29.63Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
29.63Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
29.63Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
29.41Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
29.41Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
29.41Consensusbombesin_onOrthosteric Ligandbb2_on
29.41Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
29.41Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
29.41Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
29.41Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
29.17Single5IUAQ274563485IUA-A2A-Q27456348-Na
29.17Single5N2RPSB-365N2R-A2A-PSB-36-Na
29.17Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
29.17Single6S0QZM-2413856S0Q-A2A-ZM-241385
29.17Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
29.17Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
29.17Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
29.17Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
29.17Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
29.17Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
29.17Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
29.17Consensusadenosine_offOrthosteric Liganda1_off a2_off
29.17Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
29.17Consensusblt_offOrthosteric Ligandblt1_off
29.17Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
29.17Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
29.03Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
29.03Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.03Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
29.03Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
29.03Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
29.03Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
29.03Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.95Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
28.95Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
28.57Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
28.57Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
28.57Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
28.57Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
28.57Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
28.57Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
28.57Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
28.57Single8WDTphotoNECA8WDT-A2A-photoNECA
28.57Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
28.57Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
28.57Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
28.57Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
28.57Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
28.57Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
28.57Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
28.57Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
28.57Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
28.57Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
28.57Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
28.57Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
28.57Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.12Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
28.12Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
28.12Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
28.12Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
28.12Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
28.00Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
28.00Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
28.00Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
28.00Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
28.00Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
28.00Single7TUYGSK682753A7TUY-GPR183-GSK682753A
28.00Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
28.00Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
28.00Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
28.00Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
28.00Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
28.00Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
28.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
28.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
28.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
27.59Single3QAKUK-4320973QAK-A2A-UK-432097
27.59Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
27.59Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
27.59Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
27.59Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
27.59Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
27.59Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
27.59Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
27.59Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
27.59Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
27.27Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
27.27Single4BWBNeurotensin4BWB-NTS1-Neurotensin
27.27Single5ZKQABT-4915ZKQ-PAF-ABT-491
27.27Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
27.27Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
27.27Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
27.27Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
27.27Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
27.27Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
27.27Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
27.27Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
27.27Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
27.27Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
27.27Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
27.27Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
27.27Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
27.27Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
27.27Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
27.27Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
27.27Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
27.27Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
27.27Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
27.27Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
27.27Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
27.27Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
27.27Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
27.27Consensusangiotensin_offOrthosteric Ligandat1_off
27.27Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
27.27Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
27.27Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
27.27Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
27.27Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
27.27Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
27.03Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
27.03Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
26.92Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
26.92Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
26.92Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
26.92Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
26.92Single8XQJJN2418XQJ-Apelin-JN241
26.92Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
26.92Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
26.92Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
26.92Consensuslpa_offOrthosteric Ligandlpa1_off
26.92Consensusorexin_onOrthosteric Ligandox2_on
26.67Single5WF5UK-4320975WF5-A2A-UK-432097
26.67Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
26.67Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
26.67Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
26.67Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
26.67Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
26.67Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
26.47Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
26.47Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
26.47Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
26.47Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
26.47Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
26.47Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
26.47Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
26.47Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
26.47Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
26.32Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
26.32Consensuspth_onOrthosteric Ligandpth1_on pth2_on
26.09Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
26.09Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
26.09Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
26.09Single5IUBQ274563445IUB-A2A-Q27456344-Na
26.09Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
26.09Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
26.09Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
26.09Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
26.09Single6MH8ZM-2413856MH8-A2A-ZM-241385
26.09Single6ZINSR486926ZIN-NTS1-SR48692
26.09Single7F61PF-036547467F61-H3-PF-03654746
26.09Single7T32ZM-2413857T32-A2A-ZM-241385
26.09Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
26.09Single8IHKAcifran8IHK-HCA3-Acifran
26.09Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
26.09Single8K2WAMG4878K2W-CXCR3-AMG487
26.09Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
26.09Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
26.09Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
26.09Single8ZPNAMD31008ZPN-CXCR4-AMD3100
26.09Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
26.09Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
26.09Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
26.09Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
26.09Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
25.93Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
25.93Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
25.93Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
25.93Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
25.93Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
25.93Single7EZCUKA7EZC-A2A-UKA
25.93Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
25.93Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
25.93Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
25.93Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
25.93Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
25.93Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
25.93Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.93Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
25.93Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
25.93Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
25.93Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
25.93Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
25.93Consensuschemerin_onOrthosteric Ligandcml1_on
25.93Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
25.93Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
25.81Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
25.81Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
25.81Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
25.81Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
25.81Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
25.81Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
25.81Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.81Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
25.71Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
25.71Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
25.00Single3EMLZM-2413853EML-A2A-ZM-241385
25.00Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
25.00Single5IU8Q274563475IU8-A2A-Q27456347-Na
25.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
25.00Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
25.00Single5T04Neurotensin5T04-NTS1-Neurotensin
25.00Single5UENDU1725UEN-A1-DU172
25.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
25.00Single5WF6UK-4320975WF6-A2A-UK-432097
25.00Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
25.00Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
25.00Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
25.00Single6S0LZM-2413856S0L-A2A-ZM-241385
25.00Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
25.00Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
25.00Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
25.00Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
25.00Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
25.00Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
25.00Single7PYRPSB-21157PYR-A2A-PSB-2115
25.00Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
25.00Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
25.00Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
25.00Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
25.00Single7V3ZCP559407V3Z-CB1-CP55940
25.00Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
25.00Single7XN9L-054,5227XN9-SST2-L-054,522
25.00Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
25.00Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
25.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
25.00Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
25.00Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
25.00Single7YXAONO-54306087YXA-S1P5-ONO-5430608
25.00Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
25.00Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
25.00Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
25.00Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
25.00Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
25.00Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8K5DGSK2560738K5D-HCA2-GSK256073
25.00Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
25.00Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
25.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
25.00Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
25.00Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
25.00Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
25.00Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
25.00Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
25.00Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
25.00Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
25.00Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
25.00Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
25.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
25.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
25.00Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
25.00Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
24.32Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
24.32Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
24.24Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
24.24Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
24.24Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
24.24Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
24.24Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
24.24Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
24.14Single4IARErgotamine4IAR-5-HT1B-Ergotamine
24.14Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
24.14Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
24.14Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
24.14Single7F8XNN90567F8X-CCKA-NN9056
24.14Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
24.14Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
24.14Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
24.14Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.14Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.14Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
24.14Consensuslpl_onOrthosteric Ligands1p_on lpa_on
24.14Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
24.14Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
24.14Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
24.00Single4JKVTaladegib4JKV-SMO-Taladegib
24.00Single5N2SPSB365N2S-A1-PSB36
24.00Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
24.00Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
24.00Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
24.00Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
24.00Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
24.00Single6Z4SSR486926Z4S-NTS1-SR48692
24.00Single7C61Ergotamine7C61-5-HT1B-Ergotamine
24.00Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
24.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
24.00Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
24.00Single7W41PD1762527W41-BB2-PD176252
24.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
24.00Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
24.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
24.00Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
24.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
24.00Single8QOTNanobody-E8QOT-μ-Nanobody-E
24.00Single8S4DCMF-0198S4D-Apelin-CMF-019
24.00Single8TF5Oleic acid8TF5-GPR6-Oleic acid
24.00Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
24.00Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
24.00Single9B9ZA1AKO9B9Z-CB1-A1AKO
24.00Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
24.00Single9EHSLUF76029EHS-A3A-LUF7602
24.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
24.00Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
24.00Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
24.00Consensusbombesin_offOrthosteric Ligandbb2_off
24.00Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
24.00Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
24.00Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
24.00Consensusep_offOrthosteric Ligandep4_off
24.00Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
24.00Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
24.00Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
24.00Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
23.81Single4XNWMRS25004XNW-P2Y1-MRS2500
23.81Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
23.81Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
23.81Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
23.81Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
23.81Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
23.53Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
23.53Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
23.53Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
23.53Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
23.53Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
23.53Consensusglp_onOrthosteric Ligandglp1_on glp2_on
23.53Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
23.33Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
23.33Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
23.33Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
23.33Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
23.33Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
23.33Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
23.33Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
23.33Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
23.08Single4BV0Neurotensin4BV0-NTS1-Neurotensin
23.08Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
23.08Single5V56TC1145V56-SMO-TC114
23.08Single5V57TC1145V57-SMO-TC114
23.08Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
23.08Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
23.08Single7B6WCyclazosin7B6W-α1b-Cyclazosin
23.08Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
23.08Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
23.08Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
23.08Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
23.08Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
23.08Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
23.08Single8E0GBU728E0G-μ-BU72
23.08Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
23.08Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
23.08Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
23.08Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
23.08Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.08Consensuslpa_onOrthosteric Ligandlpa1_on
23.08Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
23.08Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
23.08Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
22.86Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
22.86Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
22.86Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
22.86Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
22.86Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
22.86Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
22.73Single6LI0C176LI0-GPR52-C17
22.73Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
22.73Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
22.73Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
22.73Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
22.73Single8K5BNiacin8K5B-HCA2-Niacin
22.73Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
22.73Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
22.73Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.73Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
22.73Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
22.73Consensusgq_nucleotideOrthosteric Ligandgq_p2y
22.73Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
22.58Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
22.58Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
22.58Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.58Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
22.58Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
22.58Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
22.58Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
22.58Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
22.58Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.58Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
22.58Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
22.58Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
22.22Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
22.22Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
22.22Single6A93Risperidone6A93-5-HT2A-Risperidone
22.22Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
22.22Single6MXTSalmeterol6MXT-β2-Salmeterol
22.22Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
22.22Single7DFPSpiperone7DFP-D2-Spiperone
22.22Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
22.22Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
22.22Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
22.22Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
22.22Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
22.22Single8JJLOlodaterol8JJL-β2-Olodaterol
22.22Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
22.22Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
22.22Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
22.22Single8XYIVUF106618XYI-CXCR3-VUF10661
22.22Single9BJKNAM9BJK-μ-Naloxone-NAM
22.22Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
22.22Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
22.22Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
22.22Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
22.22Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
22.22Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
22.22Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
22.22Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
22.22Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
22.22Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
22.22Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
22.22Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
21.95Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
21.88Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
21.88Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
21.88Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
21.88Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
21.88Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
21.74Single3PWHZM-2413853PWH-A2A-ZM-241385
21.74Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
21.74Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
21.74Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
21.74Single5U09Taranabant5U09-CB1-Taranabant
21.74Single6AKYMaraviroc6AKY-CCR5-Maraviroc
21.74Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
21.74Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
21.74Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
21.74Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
21.74Single7F8YDevazepide7F8Y-CCKA-Devazepide
21.74Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
21.74Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
21.74Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
21.74Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
21.74Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
21.74Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
21.74Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
21.74Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
21.62Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
21.62Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
21.43Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
21.43Single6IBLArformoterol6IBL-β1-Arformoterol
21.43Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
21.43Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
21.43Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
21.43Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
21.43Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
21.43Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
21.43Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
21.43Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
21.43Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
21.43Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
21.43Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
21.43Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
21.43Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
21.05Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
21.05Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
21.05Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.05Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
21.05Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
20.83Single3REYXAC3REY-A2A-XAC
20.83Single4MBSMaraviroc4MBS-CCR5-Maraviroc
20.83Single5IU7Q274563465IU7-A2A-Q27456346-Na
20.83Single5JTBZM-2413855JTB-A2A-ZM-241385
20.83Single5UVIZM-2413855UVI-A2A-ZM-241385
20.83Single6AQFZM-2413856AQF-A2A-ZM-241385
20.83Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
20.83Single6V9SGTPL114036V9S-OX1-GTPL11403
20.83Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
20.83Single6ZG9GSK10347026ZG9-M1-GSK1034702
20.83Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
20.83Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
20.83Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
20.83Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
20.83Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
20.83Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
20.83Single9BA0A1AKN9BA0-CB1-A1AKN
20.83Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
20.83Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
20.83Consensusa2_offOrthosteric Liganda2a_off
20.83Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
20.83Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
20.83Consensusgrh_offOrthosteric Ligandgnrh1_off
20.69Single4UG2CGS216804UG2-A2A-CGS21680
20.69Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
20.69Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.69Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
20.69Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
20.69Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
20.69Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
20.69Single9JF4PD1683689JF4-BB1-PD168368
20.69Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
20.69Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
20.59Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
20.59Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
20.59Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
20.59Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
20.59Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
20.59Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
20.59Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
20.59Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
20.59Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
20.59Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
20.51Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
20.51Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.51Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
20.00Single4QIMANTA XV4QIM-SMO-ANTA XV
20.00Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
20.00Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
20.00Single5TGZAM65385TGZ-CB1-AM6538
20.00Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
20.00Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
20.00Single6GPSMK08126GPS-CCR2-MK0812
20.00Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
20.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
20.00Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
20.00Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.00Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
20.00Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
20.00Single7QA8Peptide7QA8-STE2-Peptide
20.00Single7QA8Peptide7QA8-STE2-Peptide
20.00Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
20.00Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
20.00Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
20.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
20.00Single7UL4Alvimopan7UL4-μ-Alvimopan
20.00Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
20.00Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
20.00Single8CU6LJ-45178CU6-A2A-LJ-4517
20.00Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
20.00Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
20.00Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
20.00Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
20.00Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
20.00Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
20.00Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
20.00Single8KIGSHU91198KIG-MC3-SHU9119-Ca
20.00Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
20.00Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
20.00Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
20.00Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
20.00Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
20.00Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
20.00Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
20.00Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
20.00Single9H37A1IR09H37-A2A-A1IR0-Na
20.00Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
20.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
20.00Consensuscck_offOrthosteric Ligandccka_off
20.00Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
20.00Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
20.00Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
20.00Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
20.00Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
19.44Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
19.44Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
19.44Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
19.44Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
19.44Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
19.44Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
19.44Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
19.44Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
19.35Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
19.35Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
19.35Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
19.35Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
19.35Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
19.35Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
19.35Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
19.35Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
19.23Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
19.23Single5C1MBU725C1M-μ-BU72
19.23Single5WQCEMPA5WQC-OX2-EMPA
19.23Single6GPXMK08126GPX-CCR2-MK0812
19.23Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
19.23Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
19.23Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
19.23Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
19.23Single7C4SS1P7C4S-S1P3-S1P
19.23Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
19.23Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
19.23Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
19.23Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
19.23Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
19.23Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
19.23Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
19.23Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
19.23Single8GNEKW-63568GNE-A2A-KW-6356-Na
19.23Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
19.23Single8JXSPF-61428JXS-D1-PF-6142
19.23Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
19.23Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
19.23Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
19.23Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
19.23Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
19.23Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
19.23Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
19.23Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
19.23Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
19.23Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
19.05Single3OE8IT1t3OE8-CXCR4-IT1t
19.05Single8A2OTheophylline8A2O-A2A-Theophylline-Na
19.05Consensusp2y_offOrthosteric Ligandp2y1_off
18.92Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
18.92Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
18.92Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
18.92Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
18.75Single6PT2KGCHM076PT2-δ-KGCHM07
18.75Single6W25SHU91196W25-MC4-SHU9119-Ca
18.75Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
18.75Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
18.75Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
18.52Single3P0GBI1671073P0G-β2-BI167107
18.52Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
18.52Single4DJHJDTic4DJH-κ-JDTic
18.52Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
18.52Single5XR8AM8415XR8-CB1-AM841
18.52Single5XRAAM115425XRA-CB1-AM11542
18.52Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
18.52Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
18.52Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
18.52Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
18.52Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
18.52Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
18.52Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
18.52Single7FEECP559407FEE-CB1-CP55940-ZCZ011
18.52Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
18.52Single7R0CAVP7R0C-V2-AVP-Arrestin2
18.52Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
18.52Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
18.52Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
18.52Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
18.52Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
18.52Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
18.52Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
18.52Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
18.52Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
18.52Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
18.52Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
18.52Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
18.52Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
18.52Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
18.52Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
18.52Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
18.52Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
18.52Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
18.52Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
18.52Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
18.52Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
18.52Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
18.42Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
18.42Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
18.18Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
18.18Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
18.18Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
18.18Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
18.18Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
18.18Single8JPSCCL78JPS-ACKR1-CCL7
18.18Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
18.18Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
18.18Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
17.95Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
17.86Single4LDEBI1671074LDE-β2-BI167107
17.86Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
17.86Single4PY02MeSATP4PY0-P2Y12-2MeSATP
17.86Single4RWADIPP-NH24RWA-δ-DIPP-NH2
17.86Single5X33BIIL2605X33-BLT1-BIIL260
17.86Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
17.86Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
17.86Single6KQICP559406KQI-CB1-CP55940-Org27569
17.86Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
17.86Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
17.86Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
17.86Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
17.86Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
17.86Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
17.86Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
17.86Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
17.86Single7YITNalfurafine7YIT-κ-Nalfurafine
17.86Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
17.86Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
17.86Single8JJ8Formoterol8JJ8-β2-Formoterol
17.86Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
17.86Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
17.86Single9DGIZ85267113509DGI-CB1-Z8526711350
17.86Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
17.86Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
17.86Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
17.86Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
17.86Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
17.86Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
17.86Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
17.86Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
17.86Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
17.86Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
17.86Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
17.86Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
17.86Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
17.65Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
17.65Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
17.65Consensuscalcitonin_onOrthosteric Ligandctlike_on
17.65Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
17.65Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
17.50Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
17.50Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
17.39Single4O9RCyclopamine4O9R-SMO-Cyclopamine
17.39Single5L7IVismodegib5L7I-SMO-Vismodegib
17.39Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
17.39Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
17.39Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
17.39Single9B9Y7DY9B9Y-CB1-7DY
17.24Single5X93K-87945X93-ETB-K-8794
17.24Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
17.24Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
17.24Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
17.24Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
17.24Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.24Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
17.24Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
17.24Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
17.24Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
17.24Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
17.24Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
17.24Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
17.24Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
17.24Consensusendothelin_offOrthosteric Ligandetb_off
17.24Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
17.24Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
17.24Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
17.14Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
17.14Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
17.14Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
17.14Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
17.07Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
16.67Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
16.67Single3NY9ICI118-5513NY9-β2-ICI118-551
16.67Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
16.67Single4QINSAG1.54QIN-SMO-SAG1.5
16.67Single4S0VSuvorexant4S0V-OX2-Suvorexant
16.67Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
16.67Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
16.67Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
16.67Single5WS3EMPA5WS3-OX2-EMPA
16.67Single5ZTYAM102575ZTY-CB2-AM10257
16.67Single6AKXA4R6AKX-CCR5-A4R
16.67Single6DS0Ly2660976DS0-5-HT2B-Ly266097
16.67Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
16.67Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
16.67Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
16.67Single6TPJSuvorexant6TPJ-OX2-Suvorexant
16.67Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
16.67Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
16.67Single7BR3Elagolix7BR3-GnRH1-Elagolix
16.67Single7F8ULintitript7F8U-CCKA-Lintitript
16.67Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
16.67Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
16.67Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single7SK9CCX6627SK9-ACKR3-CCX662
16.67Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
16.67Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
16.67Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
16.67Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
16.67Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
16.67Single7XRRLemborexant7XRR-OX2-Lemborexant
16.67Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
16.67Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
16.67Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
16.67Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
16.67Single8Y0HVUF114188Y0H-CXCR3-VUF11418
16.67Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
16.67Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
16.67Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
16.67Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
16.67Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
16.67Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
16.67Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
16.67Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
16.67Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
16.67Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
16.67Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
16.67Consensuskisspeptin_onOrthosteric Ligandkiss1_on
16.67Consensusorexin_offOrthosteric Ligandox2_off ox1_off
16.67Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
16.67Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
16.67Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
16.22Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
16.22Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
16.22Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
16.13Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
16.13Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
16.13Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
16.13Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
16.13Single8IEBA1LYA8IEB-GPR156-A1LYA
16.13Single8IEIA1LYA8IEI-GPR156-A1LYA
16.13Single8IEIA1LYA8IEI-GPR156-A1LYA
16.13Single8IEPA1LYA8IEP-GPR156-A1LYA
16.13Single8IEPA1LYA8IEP-GPR156-A1LYA
16.13Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
16.13Single8WKYPG-9348WKY-MC4-PG-934
16.13Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
16.13Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
16.13Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
16.13Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
16.13Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
16.13Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
16.13Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
16.00Single2YDOAdenosine2YDO-A2A-Adenosine
16.00Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
16.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
16.00Single6KUXRS-799486KUX-α2a-RS-79948
16.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
16.00Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
16.00Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
16.00Single6TP3Nemorexant6TP3-OX1-Nemorexant
16.00Single6TPGEMPA6TPG-OX2-EMPA
16.00Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
16.00Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
16.00Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
16.00Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.00Single7UL3Famotidine7UL3-H2-Famotidine
16.00Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
16.00Single7VV6C48/807VV6-MRGPRX2-C48/80
16.00Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
16.00Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
16.00Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
16.00Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.00Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
16.00Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
16.00Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
16.00Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
16.00Single8RLNLUF58348RLN-A2A-LUF5834
16.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.00Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
16.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
16.00Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
16.00Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
16.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
16.00Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
16.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
15.91Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
15.79Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
15.62Single6HLOAprepitant6HLO-NK1-Aprepitant
15.62Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
15.62Single8IEBA1LYA8IEB-GPR156-A1LYA
15.62Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.38Single2Y01Dobutamine2Y01-β1-Dobutamine
15.38Single2Y02Carmoterol2Y02-β1-Carmoterol
15.38Single2Y04Salbutamol2Y04-β1-Salbutamol
15.38Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
15.38Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
15.38Single5DHHSB-6121115DHH-NOP-SB-612111
15.38Single5UIGCmpd-15UIG-A2A-Cmpd-1
15.38Single6DRXLisuride6DRX-5-HT2B-Lisuride
15.38Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
15.38Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
15.38Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
15.38Single6PS1Timolol6PS1-β2-Timolol
15.38Single6TOTLemborexant6TOT-OX1-Lemborexant
15.38Single7BU7BI1671077BU7-β1-BI167107
15.38Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
15.38Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
15.38Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
15.38Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
15.38Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
15.38Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
15.38Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
15.38Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
15.38Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
15.38Single8T1WCVN4248T1W-GPR6-CVN424
15.38Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
15.38Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
15.38Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
15.38Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
15.38Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
15.38Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
15.38Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
15.38Single9CHXS-Carazolol9CHX-β2-S-Carazolol
15.38Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
15.38Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
15.38Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
15.38Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
15.38Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
15.38Consensusa3_onOrthosteric Liganda3a_on
15.38Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
15.15Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
15.15Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.15Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.00Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
15.00Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single2Y00Dobutamine2Y00-β1-Dobutamine
14.81Single2Y03Isoprenaline2Y03-β1-Isoprenaline
14.81Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
14.81Single6E67BI1671076E67-β2-BI167107-Gs(CT)
14.81Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
14.81Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
14.81Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
14.81Single6TP6Filorexant6TP6-OX1-Filorexant
14.81Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
14.81Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
14.81Single7SINNPS-21437SIN-CaS-NPS-2143
14.81Single7SINNPS-21437SIN-CaS-NPS-2143
14.81Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
14.81Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
14.81Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
14.81Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
14.81Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
14.81Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
14.81Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
14.81Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
14.81Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
14.81Single9HAPTolvaptan9HAP-V2-Tolvaptan
14.81Consensusa3_on_gpOrthosteric Liganda3a_on_gp
14.81Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.81Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.81Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
14.81Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
14.81Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.81Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
14.81Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
14.81Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.81Consensustrace-amine_onOrthosteric Ligandta1_on
14.71Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
14.71Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
14.71Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
14.63Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
14.29Single2YDVNECA2YDV-A2A-NECA
14.29Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
14.29Single4UHRCGS216804UHR-A2A-CGS21680
14.29Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
14.29Single5G53NECA5G53-A2A-NECA-Gs
14.29Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
14.29Single5TZRMK86665TZR-FFA1-MK8666
14.29Single6H7JIsoprenaline6H7J-β1-Isoprenaline
14.29Single6J20Aprepitant6J20-NK1-Aprepitant
14.29Single6J21Aprepitant6J21-NK1-Aprepitant
14.29Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
14.29Single6TQ7SB-3348676TQ7-OX1-SB-334867
14.29Single6WGTLSD6WGT-5-HT2A-LSD
14.29Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
14.29Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
14.29Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
14.29Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
14.29Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
14.29Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
14.29Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
14.29Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
14.29Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
14.29Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
14.29Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
14.29Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
14.29Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
14.29Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
14.29Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
14.29Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
14.29Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
14.29Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
14.29Single8PWNTheophylline8PWN-A2A-Theophylline
14.29Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
14.29Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
14.29Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.29Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
14.29Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single8XVLZibotentan8XVL-ETA-Zibotentan
14.29Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
14.29Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
14.29Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
14.29Consensusa2_onOrthosteric Liganda2b_on
14.29Consensusa2_on_gpOrthosteric Liganda2b_on_gp
14.29Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.29Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.29Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
14.29Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
14.29Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
14.29Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
14.29Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
14.29Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
13.89Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
13.79Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
13.79Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
13.79Single4AMIBucindolol4AMI-β1-Bucindolol
13.79Single4N4WSANT-14N4W-SMO-SANT-1
13.79Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
13.79Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
13.79Single6CM4Risperidone6CM4-D2-Risperidone
13.79Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
13.79Single6IIURamatroban6IIU-TXA2-Ramatroban
13.79Single6ZG4HTL00099366ZG4-M1-HTL0009936
13.79Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
13.79Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
13.79Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
13.79Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.79Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
13.79Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
13.79Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
13.79Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
13.79Single8JWY2-1188JWY-A2A-2-118
13.79Single8JWZAB9288JWZ-A2A-AB928-Na
13.79Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
13.79Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
13.79Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
13.79Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
13.79Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
13.79Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
13.79Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.79Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
13.79Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
13.79Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.79Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.64Single3RFMCaffeine3RFM-A2A-Caffeine
13.64Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
13.64Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
13.64Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
13.64Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
13.64Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
13.64Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
13.51Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
13.51Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
13.33Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
13.33Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
13.33Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
13.33Single6H7LDobutamine6H7L-β1-Dobutamine
13.33Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
13.33Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
13.33Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
13.33Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
13.33Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
13.33Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
13.33Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
13.33Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
13.33Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
13.33Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
13.33Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
13.33Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
13.33Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.33Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.33Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
13.33Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
13.33Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
13.16Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
13.04Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
13.04Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
13.04Single6ME5Agomelatine6ME5-MT1-Agomelatine
13.04Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
13.04Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
13.04Single7WC5Psilocin7WC5-5-HT2A-Psilocin
13.04Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.04Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
13.04Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
13.04Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.90Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
12.90Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
12.90Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
12.90Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
12.90Single8X5YAstemizole8X5Y-H1-Astemizole
12.90Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.90Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
12.50Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
12.50Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
12.50Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
12.50Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
12.50Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
12.50Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
12.50Single7UL2SR486927UL2-NTS1-SR48692-Na
12.50Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
12.50Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
12.50Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
12.50Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
12.50Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
12.50Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
12.50Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
12.50Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
12.50Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
12.50Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
12.50Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
12.50Consensusneurotensin_offOrthosteric Ligandnts1_off
12.50Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
12.00Single6B73MP11046B73-κ-MP1104
12.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
12.00Single6ME9Ramelteon6ME9-MT2-Ramelteon
12.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
12.00Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
12.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.00Single6TODEMPA6TOD-OX1-EMPA-Na
12.00Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
12.00Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
12.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
12.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
12.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
12.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
12.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
12.00Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
12.00Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.00Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
12.00Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
12.00Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
12.00Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
12.00Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
12.00Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
12.00Single8IWESpermidine8IWE-TA9-Spermidine
12.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
12.00Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.00Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.00Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.00Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
12.00Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
12.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
12.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
12.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
12.00Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
12.00Single9H2XA1IR19H2X-A2A-A1IR1-Na
12.00Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
12.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
12.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
11.90Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
11.54Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
11.54Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
11.54Single6IQLL7458706IQL-D4-L745870
11.54Single6PS0S-Carazolol6PS0-β2-S-Carazolol
11.54Single6PS4ICI118-5516PS4-β2-ICI118-551
11.54Single6PS5S-Propranolol6PS5-β2-S-Propranolol
11.54Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
11.54Single6TPKRetosiban6TPK-OT-Retosiban
11.54Single6VI4JDTic6VI4-κ-JDTic
11.54Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
11.54Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
11.54Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
11.54Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
11.54Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
11.54Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
11.54Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
11.54Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
11.54Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
11.54Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
11.54Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.54Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
11.54Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
11.54Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
11.54Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
11.54Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
11.54Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
11.54Single9AS5Mescaline9AS5-5-HT2A-Mescaline
11.54Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
11.54Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
11.54Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
11.54Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
11.54Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
11.54Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
11.54Consensusvasop-oxy_offOrthosteric Ligandot_off
11.43Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
11.43Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
11.43Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
11.43Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
11.43Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
11.11Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
11.11Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
11.11Single3NY8ICI118-5513NY8-β2-ICI118-551
11.11Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
11.11Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
11.11Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
11.11Single4GBRS-Carazolol4GBR-β2-S-Carazolol
11.11Single4QKX35V4QKX-β2-35V
11.11Single5DHGC-355DHG-NOP-C-35
11.11Single6H7MSalbutamol6H7M-β1-Salbutamol
11.11Single6IIVDaltroban6IIV-TXA2-Daltroban
11.11Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
11.11Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
11.11Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
11.11Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
11.11Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
11.11Single7F83PF-051904577F83-Ghrelin-PF-05190457
11.11Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
11.11Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
11.11Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
11.11Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
11.11Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
11.11Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
11.11Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
11.11Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
11.11Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
11.11Single7WC7Lisuride7WC7-5-HT2A-Lisuride
11.11Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
11.11Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
11.11Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
11.11Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
11.11Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
11.11Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
11.11Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
11.11Single8JJOAlprenolol8JJO-β2-Alprenolol
11.11Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
11.11Single8JXRLSD8JXR-D1-LSD
11.11Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
11.11Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
11.11Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
11.11Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
11.11Single9AS1DMT9AS1-5-HT2A-DMT
11.11Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
11.11Single9IYAONO-97105319IYA-GPR55-ONO-9710531
11.11Consensus5ht5_onOrthosteric Ligand5ht5a_on
11.11Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
11.11Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
11.11Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
11.11Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
11.11Consensusblt_onOrthosteric Ligandblt1_on
11.11Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
11.11Consensusdopamine_offOrthosteric Ligandd2_off d3_off
11.11Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
11.11Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
11.11Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
11.11Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
11.11Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
11.11Consensusleukotriene_onOrthosteric Ligandblt_on
11.11Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
10.81Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
10.81Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
10.71Single2RH1S-Carazolol2RH1-β2-S-Carazolol
10.71Single2YCWS-Carazolol2YCW-β1-S-Carazolol
10.71Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
10.71Single5D6LS-Carazolol5D6L-β2-S-Carazolol
10.71Single5JQHS-Carazolol5JQH-β2-S-Carazolol
10.71Single5TVNLSD5TVN-5-HT2B-LSD
10.71Single5WIUNemonapride5WIU-D4-Nemonapride
10.71Single5WIVNemonapride5WIV-D4-Nemonapride-Na
10.71Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
10.71Single5XPRBosentan5XPR-ETB-Bosentan
10.71Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
10.71Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
10.71Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
10.71Single6LUQHaloperidol6LUQ-D2-Haloperidol
10.71Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
10.71Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
10.71Single6PS6Timolol6PS6-β2-Timolol
10.71Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
10.71Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
10.71Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
10.71Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
10.71Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
10.71Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
10.71Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
10.71Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
10.71Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
10.71Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.71Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
10.71Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
10.71Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
10.71Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
10.71Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
10.71Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
10.71Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
10.71Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
10.71Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
10.71Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
10.71Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
10.71Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
10.71Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
10.71Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
10.71Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
10.71Consensusamine_offonOrthosteric Ligandamine_off amine_on
10.71Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
10.71Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
10.71Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
10.71Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
10.71Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
10.71Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
10.34Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
10.34Single5D5AS-Carazolol5D5A-β2-S-Carazolol
10.34Single5D5BS-Carazolol5D5B-β2-S-Carazolol
10.34Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
10.34Single6E59L-7607356E59-NK1-L-760735
10.34Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
10.34Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
10.34Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
10.34Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
10.34Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
10.34Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
10.34Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
10.34Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
10.34Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
10.34Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
10.34Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
10.34Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
10.34Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
10.34Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
10.34Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
10.34Single9BJKNaloxone9BJK-μ-Naloxone-NAM
10.34Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
10.34Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
10.34Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
10.34Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
10.34Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
10.34Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
10.34Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
10.34Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
10.34Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
10.34Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
10.34Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
10.34Consensustachykinin_offOrthosteric Ligandnk1_off
10.26Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
10.00Single3D4STimolol3D4S-β2-Timolol
10.00Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
10.00Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
10.00Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
10.00Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
10.00Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
10.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
10.00Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
10.00Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
10.00Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.00Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
10.00Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
10.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
10.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
10.00Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
9.68Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
9.68Single6K1QIRL25006K1Q-ETB-IRL2500
9.68Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
9.68Single7UM4AS26747237UM4-5-HT5A-AS2674723
9.68Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
9.68Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
9.68Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
9.52Single5MZPCaffeine5MZP-A2A-Caffeine-Na
9.52Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
9.38Single6PT3DPI-2876PT3-δ-DPI-287
9.38Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
9.38Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
9.38Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
9.38Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single7WC4Serotonin7WC4-5-HT2A-Serotonin
9.09Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
9.09Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
9.09Single9M4TSilodosin9M4T-Alpha1A-Silodosin
8.70Single6TQ9SB-4081246TQ9-OX1-SB-408124
8.70Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
8.70Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
8.70Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
8.70Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
8.70Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.70Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
8.70Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single9CHUNoradrenaline9CHU-β2-Noradrenaline
8.70Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
8.70Consensussensory_onOrthosteric Ligandopsins_on
8.33Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
8.33Single3UZAGTPL92363UZA-A2A-GTPL9236
8.33Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
8.33Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
8.33Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
8.33Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
8.33Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
8.33Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
8.33Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
8.33Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
8.33Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.33Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
8.33Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
8.33Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
8.33Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
8.33Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
8.33Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
8.33Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
8.33Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
8.33Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
8.33Single9LRCHistamine9LRC-H4-Histamine
8.33Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
8.33Consensus5ht2_onOrthosteric Ligand5ht2b_on
8.33Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.33Consensusgi_sensoryOrthosteric Ligandgi_opsins
8.33Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
8.33Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
8.33Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.33Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.33Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
8.33Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
8.33Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
8.00Single3PBLEticlopride3PBL-D3-Eticlopride
8.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
8.00Single6HLLCP999946HLL-NK1-CP99994
8.00Single6TP4ACT-4622066TP4-OX1-ACT-462206
8.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
8.00Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
8.00Single7SRQLSD7SRQ-5-HT2B-LSD
8.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
8.00Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
8.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
8.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
8.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
8.00Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
8.00Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
8.00Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
8.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
8.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
8.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
8.00Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
8.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
8.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
8.00Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
8.00Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
8.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
8.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
8.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
8.00Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
7.69Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
7.69Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
7.69Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
7.69Single6ME2Ramelteon6ME2-MT1-Ramelteon
7.69Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
7.69Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
7.69Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
7.69Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.69Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
7.69Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
7.69Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
7.69Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
7.69Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
7.69Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
7.69Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
7.69Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
7.69Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
7.69Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
7.69Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
7.69Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
7.69Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.69Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
7.69Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
7.69Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
7.69Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
7.69Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.69Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
7.69Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.69Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
7.69Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
7.69Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
7.69Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
7.69Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
7.69Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
7.41Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
7.41Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
7.41Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
7.41Single6A94Zotepine6A94-5-HT2A-Zotepine
7.41Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
7.41Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
7.41Single6TPNHTL66416TPN-OX2-HTL6641
7.41Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
7.41Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
7.41Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
7.41Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
7.41Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
7.41Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
7.41Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
7.41Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
7.41Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
7.41Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
7.41Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
7.41Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
7.41Single7VODCariprazine7VOD-5-HT2A-Cariprazine
7.41Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
7.41Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.41Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
7.41Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
7.41Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
7.41Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
7.41Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
7.41Single9AS3LSD9AS3-5-HT2A-LSD
7.41Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
7.41Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
7.41Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
7.41Consensusalpha1_onOrthosteric Ligandalpha1a_on
7.41Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
7.41Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
7.41Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
7.41Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
7.41Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
7.41Consensusopsins_offOrthosteric Ligandrhodopsin_off
7.41Consensussensory_offOrthosteric Ligandopsins_off
7.32Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
7.14Single4DAJTiotropium4DAJ-M3-Tiotropium
7.14Single4EJ4Naltrindole4EJ4-δ-Naltrindole
7.14Single4MQSIperoxo4MQS-M2-Iperoxo
7.14Single4U14Tiotropium4U14-M3-Tiotropium
7.14Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
7.14Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
7.14Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
7.14Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
7.14Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
7.14Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
7.14Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
7.14Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
7.14Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
7.14Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
7.14Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
7.14Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
7.14Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
7.14Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
7.14Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
7.14Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
7.14Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
7.14Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
7.14Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
7.14Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
7.14Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
7.14Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
7.14Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
7.14Single8X63Mepyramine8X63-H1-Mepyramine
7.14Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
7.14Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
7.14Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
7.14Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
7.14Single9JEAAtropine9JEA-M1-Atropine
7.14Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
7.14Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
7.14Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
7.14Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
7.14Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
7.14Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
7.14Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
7.14Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
7.14Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
7.14Consensusalpha2_onOrthosteric Ligandalpha2b_on
7.14Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
7.14Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
7.14Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
7.14Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
7.14Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
7.14Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
7.14Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
7.14Consensushistamine_offOrthosteric Ligandh1_off
7.14Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
7.14Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
6.98Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
6.90Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
6.90Single5CGCHTL142425CGC-mGlu5-HTL14242
6.90Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
6.90Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
6.90Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
6.90Single7WC6LSD7WC6-5-HT2A-LSD
6.90Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
6.90Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
6.90Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
6.90Single8ZMFA1L108ZMF-5-HT2C-A1L10
6.90Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
6.90Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
6.90Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
6.90Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
6.90Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
6.90Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
6.90Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
6.90Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
6.90Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
6.90Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
6.90Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
6.90Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single4U15Tiotropium4U15-M3-Tiotropium
6.67Single5V54Methiothepin5V54-5-HT1B-Methiothepin
6.67Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
6.67Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
6.67Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
6.67Single6OL9Tiotropium6OL9-M5-Tiotropium
6.67Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
6.67Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
6.67Single8EA0Iperoxo8EA0-M3-Iperoxo
6.67Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
6.67Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
6.67Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.67Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
6.67Consensus5ht1_offOrthosteric Ligand5ht1b_off
6.67Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
6.67Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
6.67Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
6.67Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
6.67Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
6.67Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
6.45Single5CXVTiotropium5CXV-M1-Tiotropium
6.45Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
6.45Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.45Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
6.45Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
6.25Single5CGDHTL142425CGD-mGlu5-HTL14242
6.25Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single8XVJMacitentan8XVJ-ETA-Macitentan
6.25Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
6.25Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.26Single6D35Cholesterol6D35-SMO-Cholesterol
5.26Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.26Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.26Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
5.26Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
5.26Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
5.26Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
5.26Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
5.26Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
5.26Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
5.26Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
5.26Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
5.26Single7DTTCa7DTT-CaS-Ca-Ca
5.26Single7DTTCa7DTT-CaS-Ca-Ca
5.26Single7DTUTryptophan7DTU-CaS-Tryptophan
5.26Single7DTUTryptophan7DTU-CaS-Tryptophan
5.26Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.26Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.26Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.26Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.26Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.26Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.26Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.26Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.26Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
5.26Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.26Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.26Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.26Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.26Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.26Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.26Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
5.26Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
5.26Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.26Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.26Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.26Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.26Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.26Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.26Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.26Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.26Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.26Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.26Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.26Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.26Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.26Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
5.26Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.26Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.26Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.26Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.26Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.26Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.26Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
5.26Single7XW7K1-707XW7-TSH-K1-70
5.26Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.26Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.26Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.26Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.26Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.26Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.26Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.26Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.26Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.26Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.26Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.26Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.26Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
5.26Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.26Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.26Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.26Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.26Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.26Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.26Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.26Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.26Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.26Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.26Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.26Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.26Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.26Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.26Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
5.26Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.26Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.26Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.26Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.26Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.26Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.26Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.26Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.26Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.26Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.26Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.26Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.26Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.26Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.26Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.26Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.26Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
5.26Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
5.26Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
5.26Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
5.26Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
5.26Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
5.26Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.26Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.26Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.26Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.26Single8WVXNorrin8WVX-LGR4-Norrin
5.26Single8WVYNorrin8WVY-LGR4-Norrin
5.26Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.26Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.26Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.26Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.26Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.26Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.26Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
5.26Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.26Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.26Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.26Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.26Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.26Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.26Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.26Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.26Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.26Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.26Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.26Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.26Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.26Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.26Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.26Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.26Single9KHHNorrin9KHH-LGR4-Norrin
5.26Single9S37NB219S37-LGR4-NB21
5.26Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
5.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.00Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.00Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.00Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
5.00Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.76Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.76Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.76Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.76Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.55Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.55Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.55Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.55Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.55Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.35Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
4.35Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
4.35Single5L7DCholesterol5L7D-SMO-Cholesterol
4.35Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.35Single8HS2Fab0468HS2-GPR20-Fab046
4.35Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.17Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
4.17Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
4.17Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
4.17Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
4.17Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
4.00Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
4.00Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
4.00Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
4.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
4.00Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.00Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
4.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
4.00Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
4.00Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
4.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
4.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
4.00Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
3.85Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
3.85Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
3.85Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
3.85Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
3.85Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
3.85Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
3.85Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
3.85Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
3.85Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
3.85Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
3.85Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
3.85Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
3.85Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
3.85Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
3.85Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.85Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
3.85Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.85Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
3.85Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.85Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.85Single9AS7Psilocin9AS7-5-HT2A-Psilocin
3.85Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
3.85Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
3.85Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
3.70Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
3.70Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
3.70Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
3.70Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
3.70Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
3.70Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
3.70Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
3.70Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
3.70Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
3.70Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
3.70Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
3.70Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
3.70Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
3.70Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
3.70Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
3.70Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
3.70Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
3.57Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
3.57Single3RZECidoxepin3RZE-H1-Cidoxepin
3.57Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
3.57Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
3.57Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
3.57Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
3.57Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
3.57Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
3.57Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.57Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
3.57Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
3.57Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.57Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
3.57Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
3.57Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
3.57Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
3.57Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
3.57Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
3.57Single9ARXSerotonin9ARX-5-HT2A-Serotonin
3.57Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
3.45Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
3.45Single5DSGTiotropium5DSG-M4-Tiotropium
3.45Single8X64Desloratadine8X64-H1-Desloratadine
3.45Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
3.45Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
3.33Single4NTJAZD12834NTJ-P2Y12-AZD1283
3.33Single6HLPNetupitant6HLP-NK1-Netupitant
3.33Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
3.33Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single9HC04YI9HC0-mGlu5-4YI
3.23Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
3.23Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
3.23Single7P2L4YI7P2L-mGlu5-4YI
3.23Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.23Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.23Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.23Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.23Single9AS9RS130-1809AS9-5-HT2A-RS130-180
3.23Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
3.12Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
2.86Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.86Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.70Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.70Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.63Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.44Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
7XA3 7XA3-CCR2-CCL2-Gi1/β1/γ2
Net Summary
Imin 1.71
Number of Linked Nodes 856
Number of Links 1145
Number of Hubs 216
Number of Links mediated by Hubs 777
Number of Communities 19
Number of Nodes involved in Communities 320
Number of Links involved in Communities 513
Path Summary
Number Of Nodes in MetaPath 85
Number Of Links MetaPath 84
Number of Shortest Paths 1718976
Length Of Smallest Path 3
Average Path Length 26.6613
Length of Longest Path 55
Minimum Path Strength 1.265
Average Path Strength 4.9428
Maximum Path Strength 21.92
Minimum Path Correlation 0.7
Average Path Correlation 0.985184
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.7027
Average % Of Corr. Nodes 48.7887
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 59.4197
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following differences:
Id1st Network2nd Network
ccr2_off_on_gpccr2_on_gpccr2_off
This network is also present in following consensuses:
IdComponents
ccr_on_gpccr6_on_gp
ccr8_on_gp
ccr2_on_gp
ccr1_on_gp
ccr5_on_gp



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Download ccr2_on_gp.zip



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