Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 2.4445402
2G.S1.02 5.79585
3G.S1.06 5.13254168
4G.H1.01 5.5124169
5G.H1.08 4.273408
6G.S2.03 5.699429
7G.S2.08 8.4205485
8G.S3.01 5.5095484
9G.S3.03 7.4312587
10G.S3.04 6.8595426
11G.S3.06 7.1512525
12G.S3.07 4.1034169
13G.s3h2.03 5.2315429
14G.H2.02 4.428428
15G.H2.06 5.17133629
16G.H2.07 5.44033629
17G.h2s4.01 7.167429
18G.S4.04 5.548439
19G.s4h3.04 5.67967638
20G.s4h3.14 1.0185406
21G.H3.01 7.6045409
22G.H3.06 5.3525436
23G.H3.09 5.51914739
24G.H3.13 4.438535
25G.H3.17 7.53533625
26G.H3.18 5.73354179
27G.S5.04 4.101439
28G.S5.05 4.49045139
29G.S5.07 4.938409
30G.HG.04 6.4565439
31G.HG.07 4.872439
32G.HG.15 4.729407
33G.hgh4.01 5.413436
34G.hgh4.02 6.87737
35G.hgh4.05 9.208407
36G.H4.03 5.7634
37G.H4.15 4.617638
38G.H4.16 3.4315433
39G.h4s6.02 4.9005438
40G.S6.02 7.7465407
41G.S6.04 8.7654139
42G.S6.05 5.186434
43G.s6h5.01 4.9125139
44G.s6h5.02 3.7515407
45G.H5.03 5.14725138
46G.H5.05 4.4575485
47G.H5.08 5.3595488
48G.H5.20 4.37354129
49b.1x2 2.98454191
50b.h2x1 4.2535405
51b.h2x5 4.0975405
52b.l1x3 9.3284549
53b.b2x1 8.3908528
54b.b2x3 4.0715446
55b.b2x5 6.579647
56b.b3x3 4.714478
57b.l3x2 4.194549
58b.b4x3 4.8325477
59b.b4x5 4.2475477
60b.b4x6 9.789649
61b.b5x2 5.842407
62b.b5x3 6.65667649
63b.b5x5 5.225475
64b.b5x7 5.6895477
65b.l5x1 4.444578
66b.l5x5 8.10314729
67b.b6x5 4.1285876
68b.b7x1 5.9265404
69b.b8x3 4.294406
70b.b8x4 5.368676
71b.l8x3 4.36254223
72b.l8x5 4.03554223
73b.b9x4 6.8225409
74b.l9x3 6.8088529
75b.l9x6 5.75886728
76b.l9x7 3.654427
77b.b10x5 4.48467609
78b.l10x1 3.721403
79b.b11x2 4.739407
80b.l11x2 7.4995429
81b.b12x5 3.712466
82b.b12x6 8.38533628
83b.b13x7 8.06567
84b.l13x3 7.245669
85b.l13x6 4.8295429
86b.l13x7 4.802469
87b.b15x1 7.646569
88b.b15x3 4.4585469
89b.l15x2 5.842469
90b.b16x4 10.265466
91b.b16x6 8.637668
92b.b17x5 6.639457
93b.b17x7 8.3885458
94b.l17x3 8.86867659
95b.l17x6 6.0848529
96b.b18x3 4.7475458
97b.b18x5 5.276405
98b.l18x1 6.882577116
99b.l18x2 5.80954117
100b.b19x2 6.452656
101b.b19x4 6.5945458
102b.l19x2 6.7945459
103b.b20x4 9.4088558
104b.b20x6 8.2048556
105b.b21x1 9.021457
106b.b21x3 5.96456
107b.b21x4 4.02405
108b.b21x5 5.941404
109b.b21x7 6.32933605
110b.l21x5 3.9084104
111b.b22x5 7.1314117
112b.l22x5 6.115676159
113b.b23x1 4.4275405
114b.b23x2 5.23954116
115b.b23x6 6.3447107
116b.b24x4 7.174106
117b.b24x6 7.1344108
118b.b25x3 6.79365105
119b.l25x3 7.6996599
120b.l25x6 12.219428
121b.b26x3 4.8355406
122b.l26x5 5.8045405
123b.l27x1 10.6949729
124b.l27x2 5.4284599
125b.b28x2 4.3988594
126b.b28x3 4.1545447
127b.b28x4 7.706496
128b.b28x6 8.8476599
129g.h1x1 2.1745402
130g.h1x12 2.6095406
131g.l1x4 6.7685408
132g.h2x11 8.6744116
133g.ctx3 6.5695409
134g.ctx6 3.8884506
135g.ctx16 5.46525208
136Lig 10.89632310
137NT 6.29861014
1381x35 5.562416
1391x39 4.92133617
1401x53 3.2375408
1411x57 2.9145406
1421x58 2.5485403
1432x42 3.7176507
1442x50 7.535409
1452x60 7.107616
1462x63 5.67415
147E1x50 6.44775818
148E1x52 6.8292516
1493x30 4.471405
1503x33 7.1548515
1513x37 6.486516
1523x50 5.2595409
1533x52 5.4735405
154I2x57 3.762607
1554x65 6.074515
156E2 16.121613
157E2x50 6.2765419
158E2x52 7.04415
1595x33 2.2335412
1605x47 7.491418
1615x50 3.6155409
1625x51 4.919416
1635x58 6.2844508
1645x65 4.9674128
1655x69 4.0285124
166I3 4.44554124
1676x36 6.4385407
1686x44 5.774518
1696x48 6.73833619
1706x51 8.4435416
1716x52 7.9564518
1726x55 4.617415
173E3 7.2784501
1747x26 6.458503
1757x34 5.1414
1767x42 6.431617
1777x49 6.20254249
1787x53 5.21067609
1797x55 3.4256506
1808x47 5.040336148
1818x49 5.34054147
1828x50 3.651409
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.l2x3 b.l2x5 40.1023.808NoNo085
2b.b3x1 b.l2x3 39.9527.328NoNo058
3b.b3x1 b.b6x5 39.80195.156NoYes056
4b.b26x2 b.b2x3 55.2744.536NoYes076
5b.b26x1 b.b26x2 55.40933.096NoNo097
6b.b26x1 b.l27x1 55.54524.448NoYes099
7b.b2x1 b.l27x1 68.07297.14YesYes289
8b.b2x1 b.l3x1 68.552717.36YesNo289
9b.l3x1 b.l5x5 68.79617.012NoYes299
10G.h2s4.01 b.l5x5 69.350410.424YesYes299
11G.S1.05 G.h2s4.01 66.87189.988NoYes099
12G.S1.05 G.S1.07 66.95136.92NoNo099
13G.S1.07 G.S4.04 67.11042.924NoYes099
14G.S4.04 G.S5.04 98.19233.65YesYes399
15G.S5.04 G.S6.03 98.56544.716YesNo395
16G.H4.16 G.S6.03 97.43374.232YesNo335
176x23 G.H4.16 99.89563.024NoYes023
186x23 G.h4s6.12 1004.42NoNo024
19G.H5.17 G.h4s6.12 85.23823.51NoNo054
205x69 G.H5.17 73.35865.208YesNo045
215x65 5x69 36.73145.024YesYes1284
225x65 G.H5.20 36.66463.71YesYes1289
23G.H5.20 G.H5.25 72.97983.322YesNo097
243x50 G.H5.25 72.87586.8YesNo097
253x50 7x53 44.24623.704YesYes099
265x69 6x33 36.66053.654YesNo1247
276x33 G.H5.20 36.62713.042NoYes1279
28G.S6.02 G.h4s6.12 18.725112.122YesNo074
29G.H3.15 G.H3.17 19.46355.424NoYes085
30G.H3.15 G.H3.18 19.57023.622NoYes089
31G.H2.08 G.H3.18 20.4284.518NoYes089
32G.H2.07 G.H2.08 20.53513.286YesNo098
33G.H2.07 G.s3h2.03 12.00856.794YesYes299
34G.H2.02 G.H2.07 20.7423.458YesYes289
35G.s3h2.03 b.l9x6 11.11844.734YesYes298
36G.H2.02 b.l9x6 11.10256.106YesYes288
37G.H2.04 G.H2.07 37.70466.4NoYes099
38G.H2.04 G.H3.08 37.81134.128NoNo099
39b.l25x6 b.l27x1 14.155923.39YesYes289
40G.H5.13 G.S6.02 17.9787.126NoYes087
41G.H5.13 G.H5.17 15.98376.358NoNo085
425x68 G.H5.13 29.92946.3NoNo058
43b.b2x4 b.b6x5 30.25073.052NoYes066
44b.b10x4 b.b2x4 30.092513.09NoNo066
45b.b10x4 b.b14x5 28.92963.156NoNo065
46b.b14x5 b.b15x1 26.77432.926NoYes059
47b.b15x1 b.b16x6 23.004913.63YesYes698
48b.b16x6 b.b17x3 21.50994.962YesNo685
49b.b17x3 g.h1x10 21.41434.88NoNo059
50g.h1x10 g.h1x13 21.09283.536NoNo091
51b.b17x2 g.h1x13 20.92734.044NoNo031
52b.b17x2 b.l16x3 20.76186.496NoNo033
53b.b16x7 b.l16x3 20.596110.914NoNo093
54b.b16x7 b.l14x6 20.26433.256NoNo093
55b.b16x5 b.l14x6 20.09823.876NoNo053
56b.b16x5 b.b17x5 12.47815.588NoYes057
57b.l2x5 b.l4x2 39.916325.928NoNo054
58b.l4x2 g.ctx16 39.77856.396NoYes048
59b.b2x5 b.l4x1 40.31285.436YesNo075
60b.l4x1 g.ctx16 40.16945.812NoYes058
61b.l11x1 b.l9x6 17.88577.534NoYes298
62b.b11x6 b.l11x1 26.26913.34NoNo299
63b.b11x6 b.l9x3 21.346113.948NoYes299
64b.b12x6 b.l9x3 17.53444.868YesYes289
65b.l23x1 b.l25x6 25.076918.58NoYes068
66b.l21x7 b.l23x1 24.51424.356NoNo056
67b.b23x6 b.l21x7 23.08544.032YesNo1075
68b.b23x6 b.b24x6 19.13614.628YesYes1078
69b.b21x7 b.b24x6 18.679713.118YesYes058
705x64 5x68 29.52613.012NoNo045
713x55 5x64 29.43884.762NoNo074
723x51 3x55 29.351612.62NoNo087
733x51 5x57 28.91674.572NoNo086
743x47 5x57 28.83054.474NoNo096
753x47 5x54 55.40267.358NoNo098
765x54 6x44 53.00673.734NoYes088
775x47 6x44 24.90935.146YesYes188
785x47 6x52 24.463614.028YesYes188
796x51 6x52 57.46389.146YesYes168
806x51 Lig 48.50310.884YesYes160
813x50 5x58 28.75458.026YesYes098
823x47 5x58 27.30968.648NoYes098
836x44 6x48 26.95627.818YesYes189
846x48 6x52 36.62924.44YesYes198
853x43 7x53 32.37066.332NoYes089
863x43 7x49 29.38013.844NoYes2489
877x45 7x49 14.00924.632NoYes099
886x48 7x45 13.47869.04YesNo099
892x50 7x49 15.58587.27YesYes099
902x50 7x46 14.26778.834YesNo098
912x53 7x46 14.12375.552NoNo068
922x53 7x42 12.70239.488NoYes067
937x42 Lig 10.31876.384YesYes170
94E2 Lig 16.764510.038YesYes130
952x60 Lig 10.219814.43YesYes160
96b.b2x3 b.b2x5 46.8023.724YesYes467
97G.H3.08 G.S4.04 37.86915.116NoYes099
98G.H3.17 b.l25x6 14.49543.8YesYes258
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
E2x51Lig4.1481NoYes4010
5x32Lig3.2581NoYes6010
5x36Lig11.7521NoYes4010
E2Lig10.0381YesYes3010
LigNT3.7921YesYes0401
6x58Lig12.321NoYes4010
7x34Lig9.8421YesYes4010
E2x52Lig7.5521YesYes5010
E1Lig13.7261NoYes4010
2x60Lig14.431YesYes6010
3x32Lig10.160NoYes6010
7x42Lig6.3841YesYes7010
3x33Lig8.4721YesYes5010
6x51Lig10.8841YesYes6010
7x38Lig4.821NoYes5010
4x61Lig4.0581NoYes4010
4x65Lig4.1341YesYes5010
4x60Lig3.4680NoYes8010
5x39Lig6.6621NoYes4010
7x24NT6.250NoYes8421
NTNT7.261YesYes4411
7x28NT3.730NoYes3421
7x27NT4.1381NoYes4421
7x31NT4.1461NoYes4421
E1NT3.2441NoYes4411
7x32NT15.4640NoYes2421
7x36NT7.7021NoYes5421
1x392x577.2681YesNo7722
1x397x383.4961YesNo7521
1x397x424.5681YesYes7721
1x427x424.0380NoYes7721
2x537x429.4880NoYes6721
2x577x429.6121NoYes7721
2x602x634.8241YesYes6512
2x60E1x506.9341YesYes6812
2x603x288.1541YesNo6512
2x604x653.61YesYes6511
2x60E2x504.71YesYes6912
2x63E16.951YesNo5421
2x63E1x507.5241YesYes5822
2x63E23.3821YesYes5321
E1x49E210.5861NoYes4321
3x25E1x507.3121NoYes9822
E1x50E23.4121YesYes8321
E1x50E2x507.8361YesYes8922
3x22E28.1640NoYes3321
3x25E23.0421NoYes9321
3x25E2x507.281NoYes9922
3x294x6512.3860NoYes5521
3x333x3710.3141YesYes5612
3x334x573.3281YesNo5712
3x334x619.9641YesNo5411
3x335x433.6961YesNo5412
3x375x435.0881YesNo6422
4x64E2x523.6741NoYes5521
4x64E211.6341NoYes5321
4x65E2x505.291YesYes5912
4x65E2x524.961YesYes5511
E2E2x5117.2221YesNo3411
E2E265.921YesYes3311
E2E2x5211.9741YesYes3511
5x32E210.9321NoYes6311
5x35E220.8321NoYes2321
5x36E25.441NoYes4311
5x31E27.4860NoYes4321
5x335x343.631YesNo2112
5x355x394.11NoNo2421
6x516x529.1461YesYes6812
6x516x5510.031YesYes6512
6x517x343.7141YesYes6411
6x526x553.4061YesYes8522
6x547x343.6680NoYes4421
6x587x274.141NoNo4412
6x587x317.4241NoNo4412
7x347x353.1761YesNo4412
7x387x424.4961NoYes5711
5x336x632.2781YesNo2112
2x67E21.9360NoYes6321
5x33Lig1.81YesYes2010
5x335x371.2261YesNo2312
5x42Lig0.5280NoYes4010

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
95.24Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
95.24Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
73.91Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
60.00Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
59.26Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
57.69Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
56.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
55.56Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
53.57Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
52.17Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
52.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
50.00Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
50.00Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
50.00Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
48.28Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
48.28Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
48.00Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
46.67Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
46.67Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
46.67Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
46.43Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
46.15Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
46.15Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
46.15Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
46.15Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
46.15Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
46.15Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
45.16Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
45.16Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
45.16Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
45.16Consensusbradykinin_onOrthosteric Ligandbk2_on
45.16Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
45.16Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
44.83Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
44.83Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
44.83Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
44.44Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
44.44Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
44.44Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
44.44Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
44.44Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
44.44Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
44.00Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
44.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
43.48Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
43.48Single8S4DCMF-0198S4D-Apelin-CMF-019
43.48Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
43.33Single7SK3CXCL127SK3-ACKR3-CXCL12
43.33Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
42.86Single3OE0CVX153OE0-CXCR4-CVX15
42.86Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
42.86Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
42.86Consensusangiotensin_onOrthosteric Ligandat1_on
42.86Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
42.86Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
42.42Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
42.31Single6KNMJN241-96KNM-Apelin-JN241-9
42.31Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
42.31Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
42.31Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
41.94Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
41.94Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
41.94Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
41.67Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
41.38Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
41.38Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
41.38Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
41.38Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
41.38Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
41.38Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
41.38Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
41.38Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
41.38Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
41.38Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
41.38Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
40.91Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
40.74Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
40.74Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
40.74Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
40.00Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
40.00Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
40.00Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
40.00Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
40.00Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
40.00Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
40.00Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
40.00Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
40.00Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
40.00Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
39.39Single5GLHEndothelin-15GLH-ETB-Endothelin-1
39.39Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
39.29Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
39.29Single7SK5CXCL127SK5-ACKR3-CXCL12
39.29Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
39.29Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
39.29Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
38.71Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
38.46Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
38.46Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
38.46Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
38.46Consensuschemerin_onOrthosteric Ligandcml1_on
38.46Consensusprostanoid_offOrthosteric Ligandep_off dp_off
37.93Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
37.93Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
37.93Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
37.93Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
37.93Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
37.93Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
37.50Single6D26Fevipiprant6D26-DP2-Fevipiprant
37.50Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
37.50Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
37.50Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
37.50Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
37.50Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
37.50Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
37.50Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
37.50Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
37.50Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
37.50Consensusdp_offOrthosteric Liganddp2_off
37.50Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
37.50Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
37.04Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
37.04Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
37.04Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
37.04Single7XN9L-054,5227XN9-SST2-L-054,522
37.04Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
37.04Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
37.04Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
37.04Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
37.04Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
36.67Single6JODAngiotensin II6JOD-AT2-Angiotensin II
36.67Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
36.67Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.67Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
36.67Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
36.67Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
36.36Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
36.36Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
36.36Consensusangiotensin_offOrthosteric Ligandat1_off
36.36Consensusendothelin_onOrthosteric Ligandetb_on eta_on
36.00Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
36.00Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
36.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
36.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
36.00Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
35.71Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
35.71Single7F8XNN90567F8X-CCKA-NN9056
35.71Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
35.71Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
35.71Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
35.71Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
35.71Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
35.48Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
35.48Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
35.48Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
35.48Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
35.48Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
35.48Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
35.48Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
35.48Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
35.48Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
35.48Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
35.48Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
35.29Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
35.29Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
35.29Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
34.78Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
34.78Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
34.62Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
34.62Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
34.62Single6OS2TRV0266OS2-AT1-TRV026
34.62Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
34.62Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
34.62Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
34.62Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
34.62Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.62Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
34.62Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
34.62Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
34.62Consensuslpl_offOrthosteric Ligands1p_off lpa_off
34.62Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.62Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.48Single3QAKUK-4320973QAK-A2A-UK-432097
34.48Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
34.48Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
34.48Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
34.48Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
34.48Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
34.48Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
34.48Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
34.38Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
34.38Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
34.29Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
33.33Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
33.33Single4YAYZD-71554YAY-AT1-ZD-7155
33.33Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
33.33Single5WF5UK-4320975WF5-A2A-UK-432097
33.33Single6D27CAY104716D27-DP2-CAY10471
33.33Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
33.33Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
33.33Single7EZCUKA7EZC-A2A-UKA
33.33Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
33.33Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
33.33Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
33.33Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
33.33Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
33.33Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
33.33Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
33.33Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
33.33Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
33.33Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
33.33Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
33.33Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
33.33Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
33.33Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
33.33Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
33.33Consensusa3_onOrthosteric Liganda3a_on
33.33Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
33.33Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
33.33Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
33.33Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
33.33Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
33.33Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
33.33Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
33.33Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
33.33Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
33.33Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
33.33Consensushca_on_gpOrthosteric Ligandhca2_on_gp
33.33Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
33.33Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
33.33Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
32.43Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
32.35Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
32.35Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
32.35Single8IY6Endothelin-18IY6-ETB-Endothelin-1
32.26Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
32.26Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
32.26Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
32.26Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
32.26Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
32.14Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
32.14Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
32.14Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
32.14Single8QJ2pN1628QJ2-MC4-pN162-Gs
32.14Single8XQJJN2418XQJ-Apelin-JN241
32.14Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
32.14Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
32.14Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
32.14Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
32.14Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
32.00Single5C1MBU725C1M-μ-BU72
32.00Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
32.00Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
32.00Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
32.00Single7C61Ergotamine7C61-5-HT1B-Ergotamine
32.00Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
32.00Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
32.00Single7W41PD1762527W41-BB2-PD176252
32.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.00Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
32.00Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
32.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
32.00Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
32.00Consensusa3_on_gpOrthosteric Liganda3a_on_gp
32.00Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
32.00Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
32.00Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
32.00Consensusbombesin_offOrthosteric Ligandbb2_off
32.00Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
32.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
32.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
32.00Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
32.00Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
31.43Single6IGKEndothelin-36IGK-ETB-Endothelin-3
31.43Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
31.43Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
31.43Consensusbombesin_onOrthosteric Ligandbb2_on
31.43Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
31.43Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
31.25Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
31.25Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
31.25Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
31.25Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
31.25Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
31.03Single4IARErgotamine4IAR-5-HT1B-Ergotamine
31.03Single4XT1Fractalkine4XT1-US28-Fractalkine
31.03Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
31.03Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
31.03Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
31.03Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
31.03Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
31.03Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
31.03Single8WDTphotoNECA8WDT-A2A-photoNECA
31.03Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.03Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
31.03Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
31.03Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
30.77Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
30.77Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
30.77Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
30.77Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
30.77Single6OS1TRV0266OS1-AT1-TRV026
30.77Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
30.77Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
30.77Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
30.77Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
30.77Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
30.77Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
30.77Single8E0GBU728E0G-μ-BU72
30.77Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
30.77Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
30.77Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
30.77Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
30.77Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
30.77Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
30.77Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
30.77Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
30.77Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
30.77Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
30.77Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
30.77Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
30.77Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
30.77Consensusrelaxin_onOrthosteric Ligandrxfp4_on
30.77Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
30.43Single6ME9Ramelteon6ME9-MT2-Ramelteon
30.43Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
30.43Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.43Single8GNGIstradefylline8GNG-A2A-Istradefylline
30.43Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
30.43Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
30.43Single8IWESpermidine8IWE-TA9-Spermidine
30.43Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
30.43Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
30.30Single4XT3Fractalkine4XT3-US28-Fractalkine
30.30Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
30.30Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
30.30Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
30.30Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
30.30Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
30.30Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
30.30Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
30.30Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
30.00Single6HLOAprepitant6HLO-NK1-Aprepitant
30.00Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
30.00Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
30.00Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
30.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
30.00Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
30.00Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
29.63Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
29.63Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
29.63Single4RWADIPP-NH24RWA-δ-DIPP-NH2
29.63Single6A93Risperidone6A93-5-HT2A-Risperidone
29.63Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
29.63Single6MXTSalmeterol6MXT-β2-Salmeterol
29.63Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
29.63Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
29.63Single7K15MKD0467K15-BLT1-MKD046-Na
29.63Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
29.63Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
29.63Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
29.63Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.63Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
29.63Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
29.63Single8XQJJN2418XQJ-Apelin-JN241
29.63Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
29.63Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
29.63Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
29.63Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
29.63Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
29.63Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
29.63Consensuslpa_offOrthosteric Ligandlpa1_off
29.17Single6KUXRS-799486KUX-α2a-RS-79948
29.17Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
29.17Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
29.17Single6V9SGTPL114036V9S-OX1-GTPL11403
29.17Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
29.17Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
29.17Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
29.17Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
29.17Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
29.17Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
29.17Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
29.17Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.17Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
29.17Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
29.17Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
29.17Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
29.17Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
29.17Consensushca_onOrthosteric Ligandhca2_on
29.17Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
29.03Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
29.03Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
29.03Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
29.03Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
29.03Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
29.03Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
29.03Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
29.03Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
28.57Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
28.57Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
28.57Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
28.57Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
28.57Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
28.57Single6IGLIRL16206IGL-ETB-IRL1620
28.57Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
28.57Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
28.57Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
28.57Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
28.57Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
28.57Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
28.57Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
28.57Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
28.57Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
28.57Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
28.57Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
28.57Single8XVUCXCL28XVU-CXCR2-CXCL2
28.57Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
28.57Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
28.57Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
28.57Consensuscck_onOrthosteric Ligandccka_on cckb_on
28.57Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
28.57Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
28.57Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
28.57Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
28.12Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.12Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
28.12Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
28.12Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
28.12Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
28.12Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
28.12Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.12Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
28.12Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.12Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.12Consensusvasop-oxy_onOrthosteric Ligandv2_on
28.12Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
28.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
28.00Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
28.00Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
28.00Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
28.00Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
28.00Single6PS1Timolol6PS1-β2-Timolol
28.00Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
28.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
28.00Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
28.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
28.00Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
28.00Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
28.00Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
28.00Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
28.00Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
28.00Single8K5DGSK2560738K5D-HCA2-GSK256073
28.00Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
28.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
28.00Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
28.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
28.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
28.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
28.00Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
28.00Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
28.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
28.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
27.78Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
27.78Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
27.59Single3NY9ICI118-5513NY9-β2-ICI118-551
27.59Single4UG2CGS216804UG2-A2A-CGS21680
27.59Single5WF6UK-4320975WF6-A2A-UK-432097
27.59Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.59Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
27.59Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
27.59Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
27.59Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
27.59Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
27.59Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
27.59Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
27.27Single6ME5Agomelatine6ME5-MT1-Agomelatine
27.27Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
27.27Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
27.27Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
27.27Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
27.27Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
27.27Single8ZRTET-18ZRT-ETB-ET-1
27.27Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
27.03Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
27.03Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
27.03Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
26.92Single2YCWS-Carazolol2YCW-β1-S-Carazolol
26.92Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
26.92Single5D6LS-Carazolol5D6L-β2-S-Carazolol
26.92Single5N2RPSB-365N2R-A2A-PSB-36-Na
26.92Single5N2SPSB365N2S-A1-PSB36
26.92Single5WQCEMPA5WQC-OX2-EMPA
26.92Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
26.92Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
26.92Single6PS6Timolol6PS6-β2-Timolol
26.92Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
26.92Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
26.92Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
26.92Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
26.92Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
26.92Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
26.92Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
26.92Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
26.92Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
26.92Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
26.92Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
26.92Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
26.92Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
26.92Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
26.92Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
26.92Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
26.92Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
26.92Single8QOTNanobody-E8QOT-μ-Nanobody-E
26.92Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
26.92Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
26.92Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
26.92Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
26.92Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
26.92Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
26.92Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.92Consensustrace-amine_onOrthosteric Ligandta1_on
26.67Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
26.67Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
26.67Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
26.67Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Single8WKYPG-9348WKY-MC4-PG-934
26.67Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.67Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
26.67Single8XWNCXCL88XWN-CXCR2-CXCL8
26.67Consensuslpl_onOrthosteric Ligands1p_on lpa_on
26.67Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
26.67Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
26.67Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
26.47Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
26.47Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
26.47Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
26.47Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
26.09Single3OE9IT1t3OE9-CXCR4-IT1t
26.09Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
26.09Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
26.09Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
26.09Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
26.09Single8K5BNiacin8K5B-HCA2-Niacin
26.09Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
26.09Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
26.09Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
26.09Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
26.09Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
25.93Single2YDVNECA2YDV-A2A-NECA
25.93Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
25.93Single4UHRCGS216804UHR-A2A-CGS21680
25.93Single5D5AS-Carazolol5D5A-β2-S-Carazolol
25.93Single5D5BS-Carazolol5D5B-β2-S-Carazolol
25.93Single5G53NECA5G53-A2A-NECA-Gs
25.93Single6J21Aprepitant6J21-NK1-Aprepitant
25.93Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
25.93Single6TQ7SB-3348676TQ7-OX1-SB-334867
25.93Single7B6WCyclazosin7B6W-α1b-Cyclazosin
25.93Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
25.93Single7F1TMIP-1a7F1T-CCR5-MIP-1a
25.93Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
25.93Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
25.93Single7R0CAVP7R0C-V2-AVP-Arrestin2
25.93Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
25.93Single7TUYGSK682753A7TUY-GPR183-GSK682753A
25.93Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
25.93Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
25.93Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
25.93Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
25.93Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
25.93Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
25.93Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
25.93Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
25.93Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
25.93Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
25.93Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
25.93Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.93Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
25.93Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
25.93Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
25.93Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
25.93Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
25.93Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
25.93Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
25.93Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
25.93Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
25.93Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
25.93Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
25.93Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.93Consensustachykinin_offOrthosteric Ligandnk1_off
25.93Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
25.81Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
25.81Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
25.81Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
25.81Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
25.71Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
25.71Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
25.71Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
25.71Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
25.71Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
25.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
25.00Single3D4STimolol3D4S-β2-Timolol
25.00Single4AMIBucindolol4AMI-β1-Bucindolol
25.00Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
25.00Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
25.00Single4PY02MeSATP4PY0-P2Y12-2MeSATP
25.00Single4S0VSuvorexant4S0V-OX2-Suvorexant
25.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
25.00Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
25.00Single5WS3EMPA5WS3-OX2-EMPA
25.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
25.00Single6AKYMaraviroc6AKY-CCR5-Maraviroc
25.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
25.00Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
25.00Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
25.00Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
25.00Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
25.00Single6PT2KGCHM076PT2-δ-KGCHM07
25.00Single6TPJSuvorexant6TPJ-OX2-Suvorexant
25.00Single6W25SHU91196W25-MC4-SHU9119-Ca
25.00Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
25.00Single6YVRNTS8-136YVR-NTS1-NTS8-13
25.00Single7BR3Elagolix7BR3-GnRH1-Elagolix
25.00Single7DFPSpiperone7DFP-D2-Spiperone
25.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
25.00Single7F8ULintitript7F8U-CCKA-Lintitript
25.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
25.00Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
25.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
25.00Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
25.00Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
25.00Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
25.00Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
25.00Single7YITNalfurafine7YIT-κ-Nalfurafine
25.00Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
25.00Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
25.00Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
25.00Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
25.00Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
25.00Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
25.00Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
25.00Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
25.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
25.00Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
25.00Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
25.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
25.00Single8JJ8Formoterol8JJ8-β2-Formoterol
25.00Single8JJLOlodaterol8JJL-β2-Olodaterol
25.00Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
25.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
25.00Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
25.00Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
25.00Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
25.00Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
25.00Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
25.00Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
25.00Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
25.00Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
25.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
25.00Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
25.00Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
25.00Single8XWACXCL18XWA-CXCR2-CXCL1
25.00Single8XWSCXCL58XWS-CXCR2-CXCL5
25.00Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
25.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
25.00Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
25.00Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
25.00Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
25.00Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
25.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
25.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
25.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
25.00Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
25.00Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
25.00Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
25.00Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
25.00Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
25.00Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
25.00Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
25.00Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
25.00Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
25.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
25.00Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
25.00Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
25.00Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
25.00Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
25.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
25.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
25.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
25.00Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
25.00Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
25.00Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
25.00Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
25.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
25.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
25.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
24.39Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
24.39Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
24.32Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
24.32Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
24.24Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
24.24Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
24.24Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
24.24Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
24.24Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
24.24Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
24.24Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
24.24Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
24.14Single4BUONeurotensin4BUO-NTS1-Neurotensin
24.14Single5X93K-87945X93-ETB-K-8794
24.14Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
24.14Single6IBLArformoterol6IBL-β1-Arformoterol
24.14Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
24.14Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
24.14Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
24.14Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.14Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
24.14Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
24.14Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
24.14Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
24.14Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
24.14Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.14Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
24.14Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
24.14Single8XWFCXCL38XWF-CXCR2-CXCL3
24.14Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
24.14Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
24.14Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
24.14Consensusendothelin_offOrthosteric Ligandetb_off
24.14Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
24.14Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
24.14Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single2YDOAdenosine2YDO-A2A-Adenosine
24.00Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
24.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
24.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
24.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
24.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
24.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
24.00Single6PS4ICI118-5516PS4-β2-ICI118-551
24.00Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
24.00Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
24.00Single6TP3Nemorexant6TP3-OX1-Nemorexant
24.00Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
24.00Single7AROLUF58337ARO-A2A-LUF5833-Na
24.00Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
24.00Single7T32ZM-2413857T32-A2A-ZM-241385
24.00Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
24.00Single7UL3Famotidine7UL3-H2-Famotidine
24.00Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
24.00Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
24.00Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
24.00Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
24.00Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
24.00Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
24.00Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
24.00Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
24.00Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
24.00Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
24.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
24.00Single8IHKAcifran8IHK-HCA3-Acifran
24.00Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
24.00Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
24.00Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
24.00Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
24.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
24.00Single8K5CAcipimox8K5C-HCA2-Acipimox
24.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
24.00Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
24.00Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
24.00Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
24.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
24.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
24.00Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
24.00Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
24.00Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
24.00Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
24.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
24.00Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
24.00Consensusgrh_offOrthosteric Ligandgnrh1_off
23.81Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
23.68Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
23.68Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
23.68Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
23.53Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
23.53Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.53Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
23.53Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
23.53Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
23.33Single5ZTYAM102575ZTY-CB2-AM10257
23.33Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
23.33Single6PT3DPI-2876PT3-δ-DPI-287
23.33Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
23.33Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
23.33Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
23.33Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
23.33Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
23.33Single7SK9CCX6627SK9-ACKR3-CCX662
23.33Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
23.33Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
23.33Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
23.33Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
23.33Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
23.33Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
23.33Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
23.08Single2Y01Dobutamine2Y01-β1-Dobutamine
23.08Single2Y02Carmoterol2Y02-β1-Carmoterol
23.08Single2Y04Salbutamol2Y04-β1-Salbutamol
23.08Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
23.08Single3NY8ICI118-5513NY8-β2-ICI118-551
23.08Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
23.08Single4EJ4Naltrindole4EJ4-δ-Naltrindole
23.08Single4GBRS-Carazolol4GBR-β2-S-Carazolol
23.08Single4QKX35V4QKX-β2-35V
23.08Single5T04Neurotensin5T04-NTS1-Neurotensin
23.08Single5TGZAM65385TGZ-CB1-AM6538
23.08Single5UENDU1725UEN-A1-DU172
23.08Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
23.08Single6DRXLisuride6DRX-5-HT2B-Lisuride
23.08Single6H7MSalbutamol6H7M-β1-Salbutamol
23.08Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
23.08Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
23.08Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
23.08Single7BU7BI1671077BU7-β1-BI167107
23.08Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
23.08Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
23.08Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
23.08Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
23.08Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
23.08Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
23.08Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
23.08Single7UL4Alvimopan7UL4-μ-Alvimopan
23.08Single7V3ZCP559407V3Z-CB1-CP55940
23.08Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
23.08Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
23.08Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
23.08Single8CU6LJ-45178CU6-A2A-LJ-4517
23.08Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
23.08Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
23.08Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
23.08Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
23.08Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
23.08Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
23.08Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
23.08Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
23.08Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
23.08Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
23.08Single8JJOAlprenolol8JJO-β2-Alprenolol
23.08Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
23.08Single8JXRLSD8JXR-D1-LSD
23.08Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
23.08Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
23.08Single8T1WCVN4248T1W-GPR6-CVN424
23.08Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
23.08Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
23.08Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
23.08Single9CHXS-Carazolol9CHX-β2-S-Carazolol
23.08Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
23.08Consensuscck_offOrthosteric Ligandccka_off
23.08Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
23.08Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
23.08Consensusdopamine_offOrthosteric Ligandd2_off d3_off
23.08Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
23.08Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
23.08Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
22.86Single6FJ3PTH6FJ3-PTH1-PTH
22.86Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
22.86Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
22.86Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
22.86Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
22.73Single8A2OTheophylline8A2O-A2A-Theophylline-Na
22.73Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
22.58Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
22.58Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
22.58Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
22.58Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
22.58Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
22.58Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
22.58Single8IEBA1LYA8IEB-GPR156-A1LYA
22.58Single8KIGSHU91198KIG-MC3-SHU9119-Ca
22.58Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
22.58Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
22.58Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
22.50Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
22.22Single2RH1S-Carazolol2RH1-β2-S-Carazolol
22.22Single2Y00Dobutamine2Y00-β1-Dobutamine
22.22Single2Y03Isoprenaline2Y03-β1-Isoprenaline
22.22Single4NTJAZD12834NTJ-P2Y12-AZD1283
22.22Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
22.22Single5JQHS-Carazolol5JQH-β2-S-Carazolol
22.22Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
22.22Single5TVNLSD5TVN-5-HT2B-LSD
22.22Single5WIUNemonapride5WIU-D4-Nemonapride
22.22Single5WIVNemonapride5WIV-D4-Nemonapride-Na
22.22Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
22.22Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
22.22Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
22.22Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
22.22Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
22.22Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
22.22Single6TP6Filorexant6TP6-OX1-Filorexant
22.22Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
22.22Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
22.22Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
22.22Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
22.22Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
22.22Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
22.22Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
22.22Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
22.22Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
22.22Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
22.22Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
22.22Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
22.22Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
22.22Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
22.22Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.22Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8GNEKW-63568GNE-A2A-KW-6356-Na
22.22Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
22.22Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
22.22Single8JXSPF-61428JXS-D1-PF-6142
22.22Single8TF5Oleic acid8TF5-GPR6-Oleic acid
22.22Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
22.22Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
22.22Single8ZMFA1L108ZMF-5-HT2C-A1L10
22.22Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
22.22Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
22.22Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
22.22Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
22.22Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
22.22Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
22.22Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
22.22Consensusadenosine_offOrthosteric Liganda1_off a2_off
22.22Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
22.22Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
22.22Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
22.22Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
22.22Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
22.22Consensusamine_offonOrthosteric Ligandamine_off amine_on
22.22Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
22.22Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
22.22Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
22.22Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
22.22Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
22.22Consensusblt_offOrthosteric Ligandblt1_off
22.22Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
22.22Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
22.22Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
22.22Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
22.22Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.22Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
22.22Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
21.95Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
21.88Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
21.88Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
21.88Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
21.88Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
21.88Single7XNACYN1548067XNA-SST2-CYN154806
21.88Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
21.88Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
21.88Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.88Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
21.88Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
21.88Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
21.88Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
21.88Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
21.88Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
21.88Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
21.74Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
21.74Single3OE6IT1t3OE6-CXCR4-IT1t
21.74Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
21.74Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
21.74Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
21.74Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
21.74Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
21.74Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
21.74Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
21.74Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
21.74Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
21.74Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
21.74Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
21.74Consensus5ht2_onOrthosteric Ligand5ht2b_on
21.74Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
21.74Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
21.62Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
21.62Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
21.62Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
21.62Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
21.62Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
21.43Single3P0GBI1671073P0G-β2-BI167107
21.43Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
21.43Single5TZRMK86665TZR-FFA1-MK8666
21.43Single5XR8AM8415XR8-CB1-AM841
21.43Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
21.43Single6H7JIsoprenaline6H7J-β1-Isoprenaline
21.43Single6J20Aprepitant6J20-NK1-Aprepitant
21.43Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
21.43Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
21.43Single6WGTLSD6WGT-5-HT2A-LSD
21.43Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
21.43Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
21.43Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
21.43Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
21.43Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
21.43Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
21.43Single7PX4PSB-21137PX4-A2A-PSB-2113
21.43Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
21.43Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
21.43Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
21.43Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
21.43Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
21.43Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
21.43Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
21.43Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
21.43Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
21.43Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
21.43Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
21.43Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
21.43Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.43Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
21.43Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
21.43Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
21.43Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
21.43Single8XVLZibotentan8XVL-ETA-Zibotentan
21.43Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
21.43Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
21.43Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
21.43Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
21.43Consensusa2_onOrthosteric Liganda2b_on
21.43Consensusa2_on_gpOrthosteric Liganda2b_on_gp
21.43Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
21.43Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
21.43Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
21.43Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
21.43Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
21.43Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.43Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
21.43Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
21.43Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
21.43Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
21.43Consensuslpa_onOrthosteric Ligandlpa1_on
21.43Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
21.43Consensusneurotensin_onOrthosteric Ligandnts1_on
21.43Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
21.43Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
21.28Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
21.21Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
21.21Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
21.21Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
21.21Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
21.21Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
21.21Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
21.21Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
21.21Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
21.05Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
21.05Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
20.83Single3PBLEticlopride3PBL-D3-Eticlopride
20.83Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
20.83Single6HLLCP999946HLL-NK1-CP99994
20.83Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
20.83Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
20.83Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
20.83Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
20.83Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
20.83Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
20.83Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
20.83Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
20.83Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
20.83Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
20.83Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
20.83Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
20.83Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
20.83Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
20.83Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
20.83Single9B9Y7DY9B9Y-CB1-7DY
20.83Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
20.83Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
20.83Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
20.69Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
20.69Single4LDEBI1671074LDE-β2-BI167107
20.69Single4XEENeurotensin4XEE-NTS1-Neurotensin
20.69Single4XESNeurotensin4XES-NTS1-Neurotensin
20.69Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
20.69Single6CM4Risperidone6CM4-D2-Risperidone
20.69Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
20.69Single6ZG4HTL00099366ZG4-M1-HTL0009936
20.69Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
20.69Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.69Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.69Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
20.69Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.69Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
20.69Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
20.69Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
20.69Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
20.69Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
20.69Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
20.69Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
20.69Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
20.69Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
20.69Single8XWMCXCL68XWM-CXCR2-CXCL6
20.69Single8XYIVUF106618XYI-CXCR3-VUF10661
20.69Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.69Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.69Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.69Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.69Consensusalpha1_offOrthosteric Ligandalpha1a_off
20.69Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
20.69Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
20.69Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
20.69Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
20.69Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.69Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
20.69Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
20.69Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
20.69Consensusorexin_onOrthosteric Ligandox2_on
20.69Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
20.59Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
20.59Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
20.59Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
20.59Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
20.59Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
20.51Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
20.51Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
20.51Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
20.51Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
20.45Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
20.00Single3ODUIT1t3ODU-CXCR4-IT1t
20.00Single3PWHZM-2413853PWH-A2A-ZM-241385
20.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
20.00Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
20.00Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
20.00Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
20.00Single6AKXA4R6AKX-CCR5-A4R
20.00Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
20.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
20.00Single6H7LDobutamine6H7L-β1-Dobutamine
20.00Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
20.00Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
20.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
20.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
20.00Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
20.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.00Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
20.00Single6TODEMPA6TOD-OX1-EMPA-Na
20.00Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
20.00Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
20.00Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
20.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
20.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
20.00Single7F8YDevazepide7F8Y-CCKA-Devazepide
20.00Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
20.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
20.00Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
20.00Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
20.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
20.00Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
20.00Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
20.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
20.00Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
20.00Single7UM4AS26747237UM4-5-HT5A-AS2674723
20.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
20.00Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
20.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
20.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
20.00Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
20.00Single7XRRLemborexant7XRR-OX2-Lemborexant
20.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
20.00Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
20.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
20.00Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
20.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
20.00Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
20.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
20.00Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
20.00Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
20.00Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
20.00Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
20.00Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
20.00Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
20.00Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
20.00Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
20.00Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
20.00Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
20.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
20.00Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
20.00Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
20.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
20.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
20.00Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
20.00Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
20.00Single8Y0HVUF114188Y0H-CXCR3-VUF11418
20.00Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
20.00Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
20.00Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
20.00Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
20.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
20.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
20.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
20.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.00Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
20.00Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
20.00Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
20.00Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
20.00Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
20.00Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
20.00Consensusorexin_offOrthosteric Ligandox2_off ox1_off
20.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
20.00Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
20.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
20.00Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
20.00Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
19.51Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
19.51Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
19.51Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
19.44Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
19.44Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
19.44Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
19.35Single5EE7MK08935EE7-Glucagon-MK0893
19.35Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
19.35Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
19.35Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
19.35Single8X5YAstemizole8X5Y-H1-Astemizole
19.23Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
19.23Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
19.23Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
19.23Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
19.23Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
19.23Single5IU7Q274563465IU7-A2A-Q27456346-Na
19.23Single5IUBQ274563445IUB-A2A-Q27456344-Na
19.23Single5JTBZM-2413855JTB-A2A-ZM-241385
19.23Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
19.23Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
19.23Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
19.23Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
19.23Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
19.23Single6AQFZM-2413856AQF-A2A-ZM-241385
19.23Single6IQLL7458706IQL-D4-L745870
19.23Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
19.23Single6PS5S-Propranolol6PS5-β2-S-Propranolol
19.23Single6TPGEMPA6TPG-OX2-EMPA
19.23Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
19.23Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
19.23Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
19.23Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
19.23Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
19.23Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
19.23Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
19.23Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
19.23Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
19.23Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
19.23Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
19.23Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
19.23Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.23Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
19.23Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
19.23Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
19.23Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
19.23Single7VV6C48/807VV6-MRGPRX2-C48/80
19.23Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
19.23Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
19.23Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
19.23Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
19.23Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
19.23Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
19.23Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
19.23Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
19.23Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
19.23Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
19.23Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
19.23Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
19.23Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
19.23Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
19.23Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
19.23Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
19.23Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
19.23Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
19.23Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
19.23Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
19.23Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
19.23Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
19.23Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
19.23Consensusa2_offOrthosteric Liganda2a_off
19.23Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
19.23Consensusalpha1_onOrthosteric Ligandalpha1a_on
19.23Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
19.23Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
19.23Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
19.23Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
19.23Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
19.23Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
19.23Consensusopsins_offOrthosteric Ligandrhodopsin_off
19.23Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
19.23Consensussensory_offOrthosteric Ligandopsins_off
19.05Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
18.92Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
18.92Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
18.75Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
18.75Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
18.75Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
18.75Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
18.75Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
18.75Consensussomatostatin_offOrthosteric Ligandsst2_off
18.52Single3EMLZM-2413853EML-A2A-ZM-241385
18.52Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
18.52Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
18.52Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
18.52Single4QIMANTA XV4QIM-SMO-ANTA XV
18.52Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
18.52Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
18.52Single5DHHSB-6121115DHH-NOP-SB-612111
18.52Single5IU8Q274563475IU8-A2A-Q27456347-Na
18.52Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
18.52Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
18.52Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
18.52Single5UIGCmpd-15UIG-A2A-Cmpd-1
18.52Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
18.52Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
18.52Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
18.52Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
18.52Single6GPSMK08126GPS-CCR2-MK0812
18.52Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
18.52Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
18.52Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
18.52Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
18.52Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
18.52Single6S0LZM-2413856S0L-A2A-ZM-241385
18.52Single6TOTLemborexant6TOT-OX1-Lemborexant
18.52Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
18.52Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
18.52Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.52Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
18.52Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
18.52Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
18.52Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
18.52Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
18.52Single7PYRPSB-21157PYR-A2A-PSB-2115
18.52Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
18.52Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
18.52Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
18.52Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
18.52Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
18.52Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
18.52Single7WC7Lisuride7WC7-5-HT2A-Lisuride
18.52Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
18.52Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
18.52Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
18.52Single7YXAONO-54306087YXA-S1P5-ONO-5430608
18.52Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
18.52Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
18.52Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
18.52Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
18.52Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
18.52Single8RLNLUF58348RLN-A2A-LUF5834
18.52Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
18.52Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
18.52Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
18.52Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
18.52Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
18.52Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
18.52Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
18.52Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
18.52Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
18.52Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
18.52Single9IYAONO-97105319IYA-GPR55-ONO-9710531
18.52Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.52Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.52Consensus5ht5_onOrthosteric Ligand5ht5a_on
18.52Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
18.52Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
18.52Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
18.52Consensusalpha2_onOrthosteric Ligandalpha2b_on
18.52Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
18.52Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
18.52Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
18.52Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
18.52Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
18.52Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
18.52Consensusblt_onOrthosteric Ligandblt1_on
18.52Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
18.52Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
18.52Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
18.52Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
18.52Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
18.52Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
18.52Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
18.52Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
18.52Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
18.52Consensusleukotriene_onOrthosteric Ligandblt_on
18.52Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
18.52Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
18.52Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
18.42Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
18.42Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
18.42Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
18.42Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
18.42Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
18.42Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
18.18Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
18.18Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
18.18Single7WC4Serotonin7WC4-5-HT2A-Serotonin
18.18Single8IEBA1LYA8IEB-GPR156-A1LYA
18.18Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
18.18Single8PWNTheophylline8PWN-A2A-Theophylline
18.18Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
17.95Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
17.86Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
17.86Single5IUAQ274563485IUA-A2A-Q27456348-Na
17.86Single5XPRBosentan5XPR-ETB-Bosentan
17.86Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
17.86Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
17.86Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
17.86Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
17.86Single6E67BI1671076E67-β2-BI167107-Gs (fused)
17.86Single6GPXMK08126GPX-CCR2-MK0812
17.86Single6HLPNetupitant6HLP-NK1-Netupitant
17.86Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
17.86Single6LUQHaloperidol6LUQ-D2-Haloperidol
17.86Single6S0QZM-2413856S0Q-A2A-ZM-241385
17.86Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
17.86Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
17.86Single7C4SS1P7C4S-S1P3-S1P
17.86Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
17.86Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
17.86Single7SINNPS-21437SIN-CaS-NPS-2143
17.86Single7SINNPS-21437SIN-CaS-NPS-2143
17.86Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
17.86Single7WC6LSD7WC6-5-HT2A-LSD
17.86Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
17.86Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
17.86Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
17.86Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
17.86Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
17.86Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
17.86Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
17.86Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
17.86Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
17.86Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
17.86Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
17.86Consensusep_offOrthosteric Ligandep4_off
17.86Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.86Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
17.86Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
17.86Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.86Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
17.86Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.65Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
17.65Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
17.50Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.39Single3RFMCaffeine3RFM-A2A-Caffeine
17.39Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
17.39Single6TQ9SB-4081246TQ9-OX1-SB-408124
17.39Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
17.39Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
17.39Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
17.39Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
17.39Single9CHUNoradrenaline9CHU-β2-Noradrenaline
17.39Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
17.39Consensusp2y_offOrthosteric Ligandp2y1_off
17.39Consensussensory_onOrthosteric Ligandopsins_on
17.24Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
17.24Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
17.24Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
17.24Single4BV0Neurotensin4BV0-NTS1-Neurotensin
17.24Single4DJHJDTic4DJH-κ-JDTic
17.24Single4U15Tiotropium4U15-M3-Tiotropium
17.24Single5V54Methiothepin5V54-5-HT1B-Methiothepin
17.24Single5XRAAM115425XRA-CB1-AM11542
17.24Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
17.24Single6E59L-7607356E59-NK1-L-760735
17.24Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
17.24Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.24Single6OL9Tiotropium6OL9-M5-Tiotropium
17.24Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
17.24Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
17.24Single7FEECP559407FEE-CB1-CP55940-ZCZ011
17.24Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
17.24Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
17.24Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
17.24Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
17.24Single8EA0Iperoxo8EA0-M3-Iperoxo
17.24Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
17.24Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
17.24Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
17.24Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
17.24Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
17.24Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
17.24Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
17.24Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
17.24Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
17.24Consensus5ht1_offOrthosteric Ligand5ht1b_off
17.24Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
17.24Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
17.24Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
17.24Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.24Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
17.24Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
17.24Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
17.14Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
17.14Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
17.14Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
17.07Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
17.07Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
16.67Single3UZAGTPL92363UZA-A2A-GTPL9236
16.67Single4N4WSANT-14N4W-SMO-SANT-1
16.67Single4XNWMRS25004XNW-P2Y1-MRS2500
16.67Single5CXVTiotropium5CXV-M1-Tiotropium
16.67Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
16.67Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
16.67Single6KQICP559406KQI-CB1-CP55940-Org27569
16.67Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
16.67Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
16.67Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
16.67Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
16.67Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
16.67Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
16.67Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
16.67Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
16.67Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
16.67Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
16.67Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
16.67Single7V6A-7V6A-M4-PubChem 9864275-Gi1/β1/γ2
16.67Single7WC5Psilocin7WC5-5-HT2A-Psilocin
16.67Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
16.67Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
16.67Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
16.67Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
16.67Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
16.67Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
16.67Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
16.67Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
16.67Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
16.67Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
16.67Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
16.67Single8JWY2-1188JWY-A2A-2-118
16.67Single8JWZAB9288JWZ-A2A-AB928-Na
16.67Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
16.67Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
16.67Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
16.67Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
16.67Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
16.67Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
16.67Consensusgi_sensoryOrthosteric Ligandgi_opsins
16.67Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
16.67Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
16.67Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
16.67Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
16.67Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
16.67Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
16.67Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
16.67Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
16.22Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
16.22Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
16.22Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
16.13Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
16.13Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8XVJMacitentan8XVJ-ETA-Macitentan
16.13Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
16.13Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
16.00Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
16.00Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
16.00Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
16.00Single4O9RCyclopamine4O9R-SMO-Cyclopamine
16.00Single5L7IVismodegib5L7I-SMO-Vismodegib
16.00Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
16.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
16.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
16.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
16.00Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
16.00Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
16.00Single7SRQLSD7SRQ-5-HT2B-LSD
16.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
16.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
16.00Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
16.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
16.00Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
16.00Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
16.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
16.00Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
16.00Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
16.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
16.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
16.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
16.00Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
16.00Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
15.79Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
15.79Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
15.79Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
15.62Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
15.62Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
15.62Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
15.62Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
15.62Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
15.62Consensuskisspeptin_onOrthosteric Ligandkiss1_on
15.38Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
15.38Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
15.38Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
15.38Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
15.38Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
15.38Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
15.38Single4BWBNeurotensin4BWB-NTS1-Neurotensin
15.38Single4QINSAG1.54QIN-SMO-SAG1.5
15.38Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
15.38Single5U09Taranabant5U09-CB1-Taranabant
15.38Single6B73MP11046B73-κ-MP1104
15.38Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
15.38Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
15.38Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
15.38Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
15.38Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
15.38Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
15.38Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
15.38Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
15.38Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
15.38Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
15.38Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
15.38Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
15.38Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
15.38Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
15.38Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
15.38Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
15.38Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
15.38Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
15.38Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
15.38Single9BA0A1AKN9BA0-CB1-A1AKN
15.38Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
15.38Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
15.38Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
15.38Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
15.38Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.38Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
15.15Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
15.15Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
15.15Single7QA8Peptide7QA8-STE2-Peptide
15.15Single7QA8Peptide7QA8-STE2-Peptide
15.15Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
15.15Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
15.15Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
15.15Single8IEIA1LYA8IEI-GPR156-A1LYA
15.15Single8IEPA1LYA8IEP-GPR156-A1LYA
15.15Single8IEPA1LYA8IEP-GPR156-A1LYA
15.15Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
15.15Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
15.15Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
15.15Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
15.15Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
14.81Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
14.81Single3REYXAC3REY-A2A-XAC
14.81Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
14.81Single5UVIZM-2413855UVI-A2A-ZM-241385
14.81Single6A94Zotepine6A94-5-HT2A-Zotepine
14.81Single6TPKRetosiban6TPK-OT-Retosiban
14.81Single6TPNHTL66416TPN-OX2-HTL6641
14.81Single6VI4JDTic6VI4-κ-JDTic
14.81Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
14.81Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
14.81Single6ZG9GSK10347026ZG9-M1-GSK1034702
14.81Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
14.81Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
14.81Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
14.81Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
14.81Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
14.81Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
14.81Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
14.81Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
14.81Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
14.81Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
14.81Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
14.81Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
14.81Single8K2WAMG4878K2W-CXCR3-AMG487
14.81Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
14.81Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
14.81Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
14.81Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
14.81Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single9BJKNaloxone9BJK-μ-Naloxone-NAM
14.81Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
14.81Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
14.81Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
14.81Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
14.81Consensusvasop-oxy_offOrthosteric Ligandot_off
14.71Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
14.71Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
14.29Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
14.29Single4DAJTiotropium4DAJ-M3-Tiotropium
14.29Single4MQSIperoxo4MQS-M2-Iperoxo
14.29Single4U14Tiotropium4U14-M3-Tiotropium
14.29Single5DHGC-355DHG-NOP-C-35
14.29Single5DSGTiotropium5DSG-M4-Tiotropium
14.29Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
14.29Single6IIVDaltroban6IIV-TP-Daltroban
14.29Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
14.29Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
14.29Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
14.29Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
14.29Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
14.29Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
14.29Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
14.29Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
14.29Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
14.29Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
14.29Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
14.29Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
14.29Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
14.29Single8X63Mepyramine8X63-H1-Mepyramine
14.29Single8X64Desloratadine8X64-H1-Desloratadine
14.29Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single9B9ZA1AKO9B9Z-CB1-A1AKO
14.29Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
14.29Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
14.29Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
14.29Consensushistamine_offOrthosteric Ligandh1_off
14.29Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
14.29Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
13.95Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
13.89Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
13.89Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
13.79Single4JKVTaladegib4JKV-SMO-Taladegib
13.79Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
13.79Single5CGCHTL142425CGC-mGlu5-HTL14242
13.79Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
13.79Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
13.79Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
13.79Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
13.79Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
13.79Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
13.79Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
13.79Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
13.79Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
13.79Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
13.79Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
13.79Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
13.79Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
13.79Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
13.79Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
13.64Single5MZPCaffeine5MZP-A2A-Caffeine-Na
13.64Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
13.64Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
13.51Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
13.51Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
13.33Single5V56TC1145V56-SMO-TC114
13.33Single5V57TC1145V57-SMO-TC114
13.33Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
13.33Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
13.33Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
13.33Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
13.33Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
13.33Single9BJKNAM9BJK-μ-Naloxone-NAM
13.33Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
13.33Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
13.33Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
13.16Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
13.04Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
13.04Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
13.04Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
13.04Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
13.04Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
13.04Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
13.04Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.90Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
12.90Single5X33BIIL2605X33-BLT1-BIIL260
12.90Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
12.90Single6IIURamatroban6IIU-TP-Ramatroban
12.90Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
12.90Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
12.90Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
12.90Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
12.90Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.82Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
12.82Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
12.50Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
12.50Single3OE8IT1t3OE8-CXCR4-IT1t
12.50Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
12.50Single5CGDHTL142425CGD-mGlu5-HTL14242
12.50Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
12.50Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
12.50Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
12.50Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.50Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
12.50Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
12.50Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
12.50Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
12.50Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
12.50Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
12.50Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
12.12Single8IEIA1LYA8IEI-GPR156-A1LYA
12.12Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
12.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
12.00Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
12.00Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
12.00Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
12.00Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
11.76Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
11.76Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.54Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
11.54Single6LI0C176LI0-GPR52-C17
11.54Single6TP4ACT-4622066TP4-OX1-ACT-462206
11.54Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
11.54Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.54Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
11.54Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
11.54Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
11.54Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
11.54Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
11.54Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.54Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
11.54Consensusgq_nucleotideOrthosteric Ligandgq_p2y
11.54Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
11.11Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
11.11Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
11.11Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
11.11Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
11.11Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
11.11Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
11.11Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
11.11Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
11.11Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
11.11Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
11.11Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
11.11Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
11.11Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
10.81Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
10.81Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
10.71Single3RZECidoxepin3RZE-H1-Cidoxepin
10.71Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
10.71Single6ZINSR486926ZIN-NTS1-SR48692
10.71Single7VODCariprazine7VOD-5-HT2A-Cariprazine
10.71Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.71Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
10.71Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
10.34Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
10.34Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
10.34Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
10.34Single7F83PF-051904577F83-Ghrelin-PF-05190457
10.34Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
10.34Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
10.34Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
10.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
10.00Single6Z4SSR486926Z4S-NTS1-SR48692
10.00Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
10.00Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
10.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
10.00Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
10.00Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
10.00Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
10.00Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
9.68Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
9.68Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
9.68Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
9.68Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
9.68Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
9.38Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
9.38Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
9.09Single6K1QIRL25006K1Q-ETB-IRL2500
9.09Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
9.09Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
8.82Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
8.70Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
8.70Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
8.57Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
8.33Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.33Single8HS2Fab0468HS2-GPR20-Fab046
8.33Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.33Single9GE2Cholesterol9GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
8.00Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
8.00Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
8.00Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
7.69Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
7.69Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
7.69Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
7.69Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
7.69Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
7.69Single8JPSCCL78JPS-ACKR1-CCL7
7.69Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.69Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.41Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
7.41Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
7.41Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
7.41Single7UL2SR486927UL2-NTS1-SR48692-Na
7.41Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
7.41Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
7.41Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
7.41Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.41Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
7.41Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.41Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Consensusneurotensin_offOrthosteric Ligandnts1_off
7.41Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
7.14Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
7.14Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.14Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.14Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.14Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
7.14Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
7.14Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.90Single6FFIMMPEP6FFI-mGlu5-MMPEP
6.90Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
6.90Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
6.90Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.90Single8IYXYL-3658IYX-GPR34-YL-365
6.90Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.90Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.67Single6FFHFenobam6FFH-mGlu5-Fenobam
6.45Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
6.45Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.45Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.45Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single7P2L4YI7P2L-mGlu5-4YI
6.25Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.25Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.06Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
4.76Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.76Single6D35Cholesterol6D35-SMO-Cholesterol
4.76Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.76Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.76Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.76Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.76Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
4.76Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
4.76Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
4.76Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
4.76Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.76Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
4.76Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.76Single7DTTCa7DTT-CaS-Ca-Ca
4.76Single7DTTCa7DTT-CaS-Ca-Ca
4.76Single7DTUTryptophan7DTU-CaS-Tryptophan
4.76Single7DTUTryptophan7DTU-CaS-Tryptophan
4.76Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.76Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.76Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.76Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.76Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.76Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.76Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.76Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.76Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.76Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.76Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.76Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.76Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.76Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.76Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.76Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.76Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.76Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.76Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.76Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.76Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.76Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.76Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.76Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.76Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.76Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.76Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.76Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.76Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.76Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.76Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
4.76Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.76Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.76Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.76Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.76Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.76Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.76Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.76Single7XW7K1-707XW7-TSH-K1-70
4.76Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.76Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.76Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.76Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.76Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.76Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.76Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.76Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.76Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.76Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.76Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.76Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.76Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.76Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.76Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.76Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.76Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.76Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
4.76Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
4.76Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.76Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.76Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
4.76Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
4.76Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.76Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.76Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
4.76Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
4.76Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
4.76Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
4.76Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
4.76Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
4.76Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.76Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.76Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.76Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.76Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.76Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.76Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.76Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.76Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.76Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.76Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.76Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.76Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.76Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.76Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.76Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.76Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.76Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
4.76Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
4.76Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.76Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
4.76Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
4.76Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.76Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.76Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8WVXNorrin8WVX-LGR4-Norrin
4.76Single8WVYNorrin8WVY-LGR4-Norrin
4.76Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.76Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.76Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.76Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.76Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.76Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.76Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.76Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.76Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.76Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.76Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.76Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.76Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.76Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.76Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.76Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.76Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.76Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.35Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.35Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.17Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.17Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.17Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
4.17Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.17Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.00Single5L7DCholesterol5L7D-SMO-Cholesterol
4.00Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.00Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.00Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
3.70Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
3.70Single8WG8Peptide8WG8-Glucagon-Peptide-chim(NtGi1-Gs)/β1/γ2
3.57Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
3.57Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
3.45Single8G94CD698G94-S1P1-CD69-Gi1/β1/γ2
3.23Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
3.12Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
3.12Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.12Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.03Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
3.03Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
2.70Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.70Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.63Single7SHEPI; PE7SHE-GPR158-PI; PE
2.56Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.56Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.50Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.33Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
8XZH 8XZH-Apelin-MM07-Gi1/β1/γ2
7W0M 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
8XZJ 8XZJ-Apelin-WN353-Gi1/β1/γ2
8XZF 8XZF-Apelin-WN561-Gi1/β1/γ2
8XZG 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
Net Summary
Imin 2.92
Number of Linked Nodes 884
Number of Links 1094
Number of Hubs 182
Number of Links mediated by Hubs 699
Number of Communities 24
Number of Nodes involved in Communities 253
Number of Links involved in Communities 377
Path Summary
Number Of Nodes in MetaPath 99
Number Of Links MetaPath 98
Number of Shortest Paths 2317617
Length Of Smallest Path 3
Average Path Length 33.544
Length of Longest Path 73
Minimum Path Strength 0.3
Average Path Strength 6.05209
Maximum Path Strength 23.182
Minimum Path Correlation 0.702
Average Path Correlation 0.981533
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.47059
Average % Of Corr. Nodes 35.3614
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 49.2087
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
gi_peptidegi_cck
gi_apelin
gi_compl-pept
gi_endothelin
gi_formylpeptide
gi_galanin
gi_ghrelin
gi_npy
gi_neurotensin
gi_opioid
gi_orexin
gi_relaxin
gi_somatostatin



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download gi_apelin.zip



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