Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1NT 8.01813815
21x32 6.1825415
31x39 5.695416
41x43 4.57125407
51x56 4.44754208
61x57 4.96375407
72x40 6.555407
82x42 5.818597
92x50 6.4325409
102x57 4.12875408
11E1x50 7.77618
12E1x52 7.342507
133x42 9.581254168
143x43 4.936254108
153x49 9.4375498
163x51 5.835836178
17I2x51 5.4725405
18I2x57 6.46667696
194x50 5.4625169
20E2 16.46471613
21E2x52 8.03414
225x36 5.645414
235x40 6.16125415
245x47 5.1695108
255x53 3.8825406
265x60 5.273754174
275x71 5.614553
28I3 6.43753
296x41 4.5425407
306x44 4.886254109
316x48 6.53333609
326x51 6.94583616
336x62 8.92375413
347x35 5.74414
357x39 7.28615
367x42 7.566517
377x49 6.97754109
387x53 6.005509
398x50 4.786208
40Lig 12.29212610
41G.s1h1.10 6.9725127
42G.S2.04 7.813754237
43G.S2.08 4.945405
44G.S3.03 5.025607
45G.S3.04 9.28875407
46G.S3.07 7.241254239
47G.H2.04 5.87125409
48G.H2.06 6.14429
49G.H2.07 6.444509
50G.h2s4.01 6.25375429
51G.s4h3.03 5.5695247
52G.s4h3.04 7.339588
53G.s4h3.05 9.538589
54G.s4h3.08 3.37125408
55G.H3.01 8.78875409
56G.H3.06 6.1275407
57G.H3.09 7.62875409
58G.H3.15 4.776508
59G.H3.17 6.32375405
60G.H3.18 5.191509
61G.S5.05 5.064176129
62G.S5.07 3.605509
63G.HG.07 5.716589
64G.HG.08 1.78406
65G.HG.15 6.68625486
66G.hgh4.02 5.963508
67G.hgh4.05 9.135486
68G.H4.10 7.649587
69G.S6.02 7.84571758
70G.s6h5.01 4.574129
71G.s6h5.02 4.19625407
72G.H5.03 5.2945128
73G.H5.13 7.5875457
74G.H5.17 4.7825455
75G.H5.20 3.669558
76G.H5.22 3.52875404
77G.H5.23 7.308594
78G.H5.26 4.265508
79b.1x8 3.66125407
80b.1x12 6.27625446
81b.h2x1 3.95375405
82b.b1x3 5.27375477
83b.l1x3 9.66875409
84b.b2x1 8.7385188
85b.b2x5 6.24333607
86b.l3x2 7.785409
87b.b4x2 4.44375408
88b.b4x6 10.03676119
89b.b5x2 6.19125407
90b.b5x3 6.243577119
91b.l5x1 4.3025408
92b.l5x5 6.42829
93b.l7x2 4.3025429
94b.b8x4 5.72167606
95b.b9x3 4.84406
96b.l9x3 8.758529
97b.l9x6 4.89143728
98b.b10x5 4.742509
99b.l11x2 8.5775429
100b.b12x3 4.06438
101b.b12x6 8.5775628
102b.b13x7 7.045537
103b.l13x3 7.87833639
104b.l13x6 5.0525429
105b.l13x7 4.3375439
106b.b14x3 4.81625435
107b.b15x1 6.375639
108b.b15x3 4.565439
109b.l15x1 4.15375427
110b.l15x2 5.48625439
111b.b16x4 12.6075436
112b.b16x6 8.78167638
113b.b17x4 6.011254195
114b.b17x7 8.10125448
115b.l17x3 9.524549
116b.l17x6 6.958529
117b.l18x1 6.351676156
118b.l18x2 5.836254157
119b.b19x2 6.466546
120b.l19x2 6.7275409
121b.b20x4 10.681548
122b.b20x6 7.572546
123b.l20x2 7.745409
124b.b21x1 9.995447
125b.b21x3 7.6675446
126b.b21x7 7.826505
127b.b22x5 5.3195157
128b.l22x5 7.8575149
129b.b23x6 6.6356137
130b.l23x1 8.19875406
131b.b24x2 3.194135
132b.b24x4 7.6485136
133b.b24x5 3.4075405
134b.b24x7 8.3254149
135b.l25x3 9.50375469
136b.l27x1 13.37676189
137b.l27x2 8.2675469
138b.b28x3 4.96754117
139b.b28x4 7.99375466
140b.b28x6 7.62833669
141g.l1x4 5.023548
142g.h2x11 9.741254156
143g.ctx3 5.97167669
144g.ctx14 6.145479
145g.ctx16 5.79678
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
13x36 6x48 18.77435.125NoYes079
23x36 Lig 17.619610.35NoYes170
36x48 6x51 20.91324.01YesYes096
46x51 Lig 17.687815.785YesYes160
53x43 7x53 57.59696.45YesYes089
63x43 6x44 50.30333.655YesYes1089
76x44 6x48 40.75499.02YesYes099
83x50 7x53 62.92746.17NoYes099
93x50 G.H5.25 69.133511.54NoNo098
10G.H5.20 G.H5.25 69.29053.46YesNo588
11G.H5.06 G.S6.04 75.313316.405NoNo049
12G.H5.06 I3 75.12844.29NoYes043
13G.H5.17 I3 72.56825.425YesYes553
14G.H5.17 G.H5.20 71.70843.99YesYes558
15b.b4x6 b.b5x3 13.918412.18YesYes1199
16b.b3x2 b.b4x6 19.18385.125NoYes059
17b.b2x5 b.b3x2 19.393310.25YesNo075
18b.b2x3 b.b2x5 38.84964.65NoYes067
19b.b26x2 b.b2x3 39.0564.86NoNo076
20b.b26x1 b.b26x2 39.46884.3NoNo097
21b.b26x1 b.l27x1 39.67534.94NoYes099
22G.H2.09 b.l27x1 57.32996.35NoYes1889
23G.H2.09 G.H3.17 57.94017.41NoYes085
24G.H2.08 G.H3.17 29.60654.7NoYes085
25G.H2.04 G.H2.08 30.12535.01YesNo098
26G.H2.04 G.H3.12 99.82233.76YesNo097
27G.H3.12 G.S1.07 49.95465.71NoNo079
28G.S1.07 G.S4.04 49.99016.09NoNo099
29G.H3.09 G.S4.04 1009.11YesNo099
30G.H3.09 G.H4.15 50.05755.895YesNo099
31G.H3.06 G.H4.15 50.04563.72YesNo079
32G.H3.03 G.H3.06 34.353410.8NoYes047
33G.H3.03 G.hgh4.02 33.55575.245NoYes048
34G.HG.15 G.hgh4.02 63.09623.655YesYes068
35G.HG.15 G.s4h3.04 94.52874.69YesYes868
36G.HG.07 G.s4h3.04 92.95934.78YesYes898
37G.HG.07 G.s4h3.02 92.43364.59YesNo099
38G.s4h3.02 G.s5hg.01 92.07795.355NoNo099
39G.S5.07 G.s5hg.01 91.8964.2YesNo099
40G.S5.07 G.s6h5.01 83.83795.85YesYes099
41G.S6.04 G.s6h5.01 75.17953.425NoYes1299
42G.H3.15 G.H3.17 29.61573.375YesYes085
43G.H2.04 G.H3.15 30.34197.715YesYes098
44G.H3.08 G.H3.12 49.95463.565NoNo097
45G.H3.08 G.S4.04 49.99015.48NoNo099
46G.H3.09 G.h4s6.01 50.12026.09YesNo093
47G.H3.06 G.h4s6.01 50.09644.23YesNo073
48G.H3.06 G.H4.14 65.75275.76YesNo075
49G.H4.14 G.hgh4.02 33.5476.84NoYes058
50G.H4.10 G.H4.14 32.16489.33YesNo075
51G.H4.10 G.HG.15 31.57836.09YesYes876
52G.HN.47 b.b4x2 10.3592.82NoYes068
53G.HN.47 b.b5x3 10.56972.82NoYes069
54G.H2.07 b.l7x2 20.32023.99YesYes099
55G.H2.04 G.H2.07 39.5927YesYes099
56b.b11x6 b.l11x1 10.07062.785NoNo299
57b.l11x1 b.l9x6 10.18777.24NoYes298
58G.H2.02 b.l9x6 18.57215.725NoYes088
59G.H2.02 G.H2.07 18.68094.94NoYes089
60b.l7x2 b.l9x6 19.45443.52YesYes298
61G.H2.06 b.l9x6 26.13443.58YesYes298
62G.H2.06 b.l17x6 25.71698.3YesYes299
63b.l17x5 b.l17x6 25.18993.68NoYes069
64b.l17x5 b.l19x2 24.97985.155NoYes069
65b.b20x2 b.l19x2 23.28766.505NoYes069
66b.b20x2 b.b20x4 22.86727.115NoYes068
67b.b20x4 b.b20x6 22.02724.275YesYes486
68b.b17x7 b.b20x6 19.07188.575YesYes486
69b.b17x7 b.b21x1 18.24196.57YesYes487
70b.1x12 b.b21x1 17.394510.125YesYes467
71b.1x12 b.1x8 16.55563.76YesYes067
72b.1x8 g.h1x8 10.8544.78YesNo079
73b.l25x6 b.l27x1 18.242928.49NoYes089
74b.l23x1 b.l25x6 18.033219.655YesNo068
75b.l21x7 b.l23x1 17.40645.445NoYes056
76b.b23x6 b.l21x7 16.35874.03YesNo075
77b.b23x6 b.b24x6 13.84624.82YesNo1378
78b.b21x7 b.b24x6 13.653412.06YesNo058
79b.b2x5 b.l26x1 13.857810.92YesNo077
80b.l26x1 b.l26x3 13.43866.505NoNo2577
81b.l26x3 b.l26x5 13.23297.625NoNo075
82b.l26x5 g.ctx4 12.87116.71NoNo057
83g.ctx3 g.ctx4 12.66294.025YesNo097
84b.b17x6 g.h1x8 10.64218.47NoNo079
85b.b16x4 b.b17x6 10.430112.76YesNo067
86E2 Lig 10.101531.15YesYes130
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
NTNT12.5251YesYes5511
7x24NT7.280NoYes8521
7x28NT9.3650NoYes1521
E2NT3.951YesYes3511
1x30NT4.2951NoYes4521
7x32NT6.310NoYes2521
LigNT7.8951YesYes0501
1x311x353.3250NoNo3522
1x317x355.9850NoYes3421
1x322x677.4951YesNo5322
1x32E16.041YesNo5421
1x32E25.9151YesYes5321
1x327x355.281YesYes5421
1x351x393.991NoYes5622
1x357x399.371NoYes5521
1x392x573.461YesYes6822
1x397x3912.181YesYes6521
2x537x424.10NoYes7721
2x563x323.530NoNo6621
2x577x425.860YesYes8721
2x602x635.4551NoNo6512
2x603x296.781NoNo6512
2x60Lig14.191NoYes6010
2x63E1x504.850NoYes5822
2x647x395.0250NoYes5521
2x67E217.951NoYes3321
7x35E15.8551YesNo4411
E1Lig21.411NoYes4010
E1x49E27.290NoYes5321
E1x50E25.2351YesYes8321
3x22E25.471NoYes3321
3x294x6521.690NoNo5421
3x327x424.2351NoYes6711
3x32Lig3.3551NoYes6010
3x366x485.1251NoYes7912
3x36Lig10.351NoYes7010
4x61E2x523.6450NoYes4421
4x64E215.061NoYes4321
4x645x357.021NoNo4222
4x65E2x528.1451NoYes4411
4x65Lig4.51NoYes4010
E2E256.511YesYes3311
E2E2x5111.6451YesNo3411
E2Lig31.151YesYes3010
E2x51Lig7.921NoYes4010
E2E2x5215.111YesYes3411
E2x52Lig5.221YesYes4010
5x35E211.2851NoYes2321
5x36E210.11YesYes4311
5x39E29.3650NoYes5321
5x335x363.3150NoYes2421
5x366x625.2351YesYes4311
5x36Lig3.931YesYes4010
5x406x555.851YesNo5511
5x406x586.061YesNo5411
5x406x597.311YesNo5512
5x40Lig5.4251YesYes5010
5x436x514.871NoYes5611
5x43Lig4.8651NoYes5010
6x486x514.010YesYes9621
6x516x525.271YesNo6812
6x516x557.781YesNo6511
6x517x383.961YesNo6511
6x51Lig15.7851YesYes6010
6x547x345.60NoNo5521
6x55Lig13.5851NoYes5010
6x586x6213.6951NoYes4311
6x58Lig10.8151NoYes4010
6x616x625.641NoYes3311
6x617x2711.081NoNo3311
6x62Lig11.1251YesYes3010
7x31Lig15.1750NoYes3010
7x34Lig10.661NoYes5010
7x35Lig5.841YesYes4010
7x387x394.6251NoYes5511
7x38Lig12.211NoYes5010
7x397x426.7051YesYes5711
7x39Lig5.7751YesYes5010
7x42Lig16.931YesYes7010
3x363x373.5151NoNo7712
6x61Lig6.551NoYes3010
7x27Lig3.3751NoYes3010
5x32E20.891NoYes3321

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
100.00Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
100.00Consensusbradykinin_onOrthosteric Ligandbk2_on
100.00Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
87.50Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
87.50Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
68.00Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
66.67Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
64.29Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
64.29Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
62.96Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
62.96Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
62.96Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
62.07Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
61.54Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
61.54Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
60.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
59.26Consensusangiotensin_onOrthosteric Ligandat1_on
59.26Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
58.62Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
58.06Single5GLHEndothelin-15GLH-ETB-Endothelin-1
57.69Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
57.14Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
57.14Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
57.14Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
57.14Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
57.14Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
56.67Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
56.67Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
55.56Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
55.56Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
55.17Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
54.84Consensusendothelin_onOrthosteric Ligandetb_on eta_on
53.57Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
53.57Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
53.57Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
53.57Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
53.33Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
53.33Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
53.33Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
52.00Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
52.00Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
51.85Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
51.85Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
51.85Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
51.85Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
51.72Single6JODAngiotensin II6JOD-AT2-Angiotensin II
51.72Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
51.61Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
51.61Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
51.61Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
51.61Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
51.52Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
51.52Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
50.00Single6IGLIRL16206IGL-ETB-IRL1620
50.00Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
50.00Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
50.00Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
50.00Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
50.00Single8IY6Endothelin-18IY6-ETB-Endothelin-1
50.00Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
50.00Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
50.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
50.00Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
50.00Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
50.00Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
50.00Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
50.00Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
50.00Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
48.48Single6IGKEndothelin-36IGK-ETB-Endothelin-3
48.48Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
48.48Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
48.48Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
48.48Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
48.39Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
48.39Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
48.39Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
48.28Single3OE0CVX153OE0-CXCR4-CVX15
48.28Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
48.28Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
48.28Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
48.28Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
48.15Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
48.15Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
48.15Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
48.15Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
48.15Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
48.00Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
46.88Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
46.67Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
46.67Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
46.67Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
46.67Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
46.43Single4IARErgotamine4IAR-5-HT1B-Ergotamine
46.43Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
46.43Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
46.43Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
46.43Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
46.43Single8WDTphotoNECA8WDT-A2A-photoNECA
46.43Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
46.43Single8XWNCXCL88XWN-CXCR2-CXCL8
46.43Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
46.43Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
46.15Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
46.15Single6OS2TRV0266OS2-AT1-TRV026
46.15Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
45.83Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
45.83Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
45.83Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
45.83Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
45.16Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
45.16Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
45.16Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
45.16Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
45.16Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
45.16Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
45.16Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
45.16Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
45.16Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
45.16Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
44.83Single3QAKUK-4320973QAK-A2A-UK-432097
44.83Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
44.44Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
44.44Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
44.44Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
44.44Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
44.44Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
44.44Consensuschemerin_onOrthosteric Ligandcml1_on
44.44Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
44.44Consensusprostanoid_offOrthosteric Ligandep_off dp_off
44.12Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
44.00Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
44.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
43.75Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
43.75Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
43.75Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
43.75Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
43.33Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
43.33Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
43.33Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
43.33Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
42.86Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
42.86Single5WF6UK-4320975WF6-A2A-UK-432097
42.86Single6KNMJN241-96KNM-Apelin-JN241-9
42.86Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
42.86Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
42.86Single7XN9L-054,5227XN9-SST2-L-054,522
42.86Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
42.86Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
42.86Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
42.86Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
42.86Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
42.42Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
42.31Single6OS1TRV0266OS1-AT1-TRV026
42.31Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
42.31Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
42.31Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
42.31Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
42.31Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
42.31Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
41.94Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
41.94Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
41.94Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
41.94Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
41.94Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
41.94Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
41.94Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
41.94Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
41.94Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
41.94Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
41.94Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
41.94Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
41.94Consensusvasop-oxy_onOrthosteric Ligandv2_on
41.94Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
41.67Single7AROLUF58337ARO-A2A-LUF5833-Na
41.67Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
41.67Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
41.67Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
41.38Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
41.38Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
41.38Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
41.38Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
41.38Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
41.38Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
41.38Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.18Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
40.74Single4RWADIPP-NH24RWA-δ-DIPP-NH2
40.74Single6MXTSalmeterol6MXT-β2-Salmeterol
40.74Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
40.74Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
40.74Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
40.74Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
40.74Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.74Single8XWACXCL18XWA-CXCR2-CXCL1
40.74Single8XWMCXCL68XWM-CXCR2-CXCL6
40.74Single8XWSCXCL58XWS-CXCR2-CXCL5
40.74Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
40.74Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
40.74Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
40.74Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
40.62Single8ZRTET-18ZRT-ETB-ET-1
40.62Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
40.62Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
40.62Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
40.00Single6D27CAY104716D27-DP2-CAY10471
40.00Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
40.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
40.00Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
40.00Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
40.00Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
40.00Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
40.00Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
40.00Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
40.00Consensusa3_onOrthosteric Liganda3a_on
40.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
40.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
40.00Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
40.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
40.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
39.39Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
39.39Single7SK3CXCL127SK3-ACKR3-CXCL12
39.39Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
39.39Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
39.29Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
39.29Single6IBLArformoterol6IBL-β1-Arformoterol
39.29Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
39.29Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
39.29Single7EZCUKA7EZC-A2A-UKA
39.29Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
39.29Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
39.29Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
39.29Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
39.29Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
39.29Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
39.29Single8XVUCXCL28XVU-CXCR2-CXCL2
39.29Single8XWFCXCL38XWF-CXCR2-CXCL3
39.29Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
38.89Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
38.71Single5WF5UK-4320975WF5-A2A-UK-432097
38.71Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
38.71Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
38.71Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
38.71Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
38.71Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
38.71Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
38.71Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
38.71Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
38.71Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
38.71Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
38.46Single5C1MBU725C1M-μ-BU72
38.46Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
38.46Single6D26Fevipiprant6D26-DP2-Fevipiprant
38.46Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
38.46Single7C61Ergotamine7C61-5-HT1B-Ergotamine
38.46Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
38.46Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
38.46Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.46Single8S4DCMF-0198S4D-Apelin-CMF-019
38.46Single8TF5Oleic acid8TF5-GPR6-Oleic acid
38.46Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
38.46Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
38.46Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
38.46Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
38.46Consensusa3_on_gpOrthosteric Liganda3a_on_gp
38.46Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
38.46Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
38.46Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
38.46Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
38.46Consensusdp_offOrthosteric Liganddp2_off
38.24Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
38.24Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
38.24Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
38.24Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
38.24Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
38.24Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
37.93Single3NY9ICI118-5513NY9-β2-ICI118-551
37.93Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
37.93Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
37.93Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
37.93Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
37.93Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
37.93Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
37.93Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
37.93Single8XQJJN2418XQJ-Apelin-JN241
37.93Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
37.93Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
37.50Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
37.50Single8GNGIstradefylline8GNG-A2A-Istradefylline
37.50Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
37.50Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
37.50Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
37.50Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
37.50Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
37.50Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
37.50Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.50Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
37.50Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
37.50Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
37.50Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
37.14Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
37.04Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
37.04Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
37.04Single6J21Aprepitant6J21-NK1-Aprepitant
37.04Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
37.04Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
37.04Single8E0GBU728E0G-μ-BU72
37.04Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
37.04Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
37.04Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
37.04Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
37.04Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
37.04Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
37.04Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
37.04Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
37.04Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
37.04Consensusa2_onOrthosteric Liganda2b_on
37.04Consensusa2_on_gpOrthosteric Liganda2b_on_gp
37.04Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
37.04Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
37.04Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
37.04Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
37.04Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
37.04Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
37.04Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
37.04Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
36.67Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
36.67Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
36.67Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
36.67Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
36.67Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
36.67Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
36.67Consensuslpl_onOrthosteric Ligands1p_on lpa_on
36.67Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
36.36Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
36.36Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
36.36Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
36.36Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
36.36Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
36.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
36.00Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
36.00Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
36.00Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
36.00Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
36.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
36.00Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
36.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
36.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
35.71Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
35.71Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
35.71Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
35.71Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
35.71Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
35.71Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
35.71Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
35.71Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
35.71Single7YITNalfurafine7YIT-κ-Nalfurafine
35.71Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
35.71Single8JJ8Formoterol8JJ8-β2-Formoterol
35.71Single8JJLOlodaterol8JJL-β2-Olodaterol
35.71Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
35.71Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
35.71Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
35.71Single8XQJJN2418XQJ-Apelin-JN241
35.71Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
35.71Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
35.71Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
35.71Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
35.71Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
35.71Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
35.71Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
35.71Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
35.71Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
35.71Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
35.71Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
35.71Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
35.71Consensuslpa_offOrthosteric Ligandlpa1_off
35.71Consensuslpl_offOrthosteric Ligands1p_off lpa_off
35.71Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
35.71Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
35.71Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
35.48Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
35.48Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
35.48Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
35.48Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
35.48Single7XNACYN1548067XNA-SST2-CYN154806
35.48Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
35.48Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
35.48Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
35.48Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
35.48Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
35.29Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
34.62Single4EJ4Naltrindole4EJ4-δ-Naltrindole
34.62Single4QIMANTA XV4QIM-SMO-ANTA XV
34.62Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
34.62Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
34.62Single5UENDU1725UEN-A1-DU172
34.62Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
34.62Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
34.62Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
34.62Single7UL4Alvimopan7UL4-μ-Alvimopan
34.62Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
34.62Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
34.62Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
34.62Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
34.62Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
34.62Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
34.62Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.62Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.62Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.62Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.62Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.62Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
34.62Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
34.62Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
34.62Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
34.62Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
34.62Consensushca_on_gpOrthosteric Ligandhca2_on_gp
34.48Single4BUONeurotensin4BUO-NTS1-Neurotensin
34.48Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
34.48Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
34.48Single6H7LDobutamine6H7L-β1-Dobutamine
34.48Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
34.48Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
34.48Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
34.48Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
34.48Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
34.48Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
34.48Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.48Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
34.48Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
34.48Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
34.48Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
34.48Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
34.48Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
34.48Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
34.38Single6PT2KGCHM076PT2-δ-KGCHM07
34.38Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
34.38Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
34.38Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
34.38Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.38Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
34.38Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
34.38Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
33.33Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
33.33Single4UG2CGS216804UG2-A2A-CGS21680
33.33Single5IUAQ274563485IUA-A2A-Q27456348-Na
33.33Single5N2RPSB-365N2R-A2A-PSB-36-Na
33.33Single5N2SPSB365N2S-A1-PSB36
33.33Single5WQCEMPA5WQC-OX2-EMPA
33.33Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
33.33Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
33.33Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
33.33Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
33.33Single6PT3DPI-2876PT3-δ-DPI-287
33.33Single6S0QZM-2413856S0Q-A2A-ZM-241385
33.33Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
33.33Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
33.33Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
33.33Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
33.33Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
33.33Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
33.33Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
33.33Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
33.33Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
33.33Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
33.33Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
33.33Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
33.33Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
33.33Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
33.33Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
33.33Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
33.33Single8QJ2pN1628QJ2-MC4-pN162-Gs
33.33Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
33.33Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
33.33Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
33.33Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusadenosine_offOrthosteric Liganda1_off a2_off
33.33Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
33.33Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
33.33Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
33.33Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
33.33Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
33.33Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
33.33Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
33.33Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
33.33Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
33.33Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
32.43Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
32.43Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
32.43Consensusbombesin_onOrthosteric Ligandbb2_on
32.43Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
32.43Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
32.35Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
32.35Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
32.26Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
32.26Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
32.26Single7F8XNN90567F8X-CCKA-NN9056
32.26Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
32.26Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
32.26Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
32.26Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
32.26Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
32.26Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
32.26Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
32.26Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
32.26Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
32.26Consensussomatostatin_offOrthosteric Ligandsst2_off
32.14Single2YDVNECA2YDV-A2A-NECA
32.14Single3P0GBI1671073P0G-β2-BI167107
32.14Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
32.14Single4UHRCGS216804UHR-A2A-CGS21680
32.14Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
32.14Single5G53NECA5G53-A2A-NECA-Gs
32.14Single5V56TC1145V56-SMO-TC114
32.14Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
32.14Single7F1TMIP-1a7F1T-CCR5-MIP-1a
32.14Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
32.14Single7PX4PSB-21137PX4-A2A-PSB-2113
32.14Single7R0CAVP7R0C-V2-AVP-Arrestin2
32.14Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
32.14Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
32.14Single7TUYGSK682753A7TUY-GPR183-GSK682753A
32.14Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
32.14Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
32.14Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
32.14Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
32.14Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
32.14Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
32.14Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
32.14Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
32.14Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
32.14Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
32.14Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
32.14Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
32.14Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
32.14Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
32.14Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
32.14Consensuslpa_onOrthosteric Ligandlpa1_on
32.14Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
32.14Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Consensusneurotensin_onOrthosteric Ligandnts1_on
32.14Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
32.14Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
32.14Consensusrelaxin_onOrthosteric Ligandrxfp4_on
32.14Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
32.00Single3PWHZM-2413853PWH-A2A-ZM-241385
32.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
32.00Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
32.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
32.00Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
32.00Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
32.00Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
32.00Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
32.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
32.00Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
32.00Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
32.00Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
32.00Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
32.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
32.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
31.58Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
31.58Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
31.43Single4XT3Fractalkine4XT3-US28-Fractalkine
31.43Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
31.25Single6HLOAprepitant6HLO-NK1-Aprepitant
31.25Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
31.25Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
31.25Single7SK5CXCL127SK5-ACKR3-CXCL12
31.25Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
31.25Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
31.25Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
31.25Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
31.25Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
31.25Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
31.25Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
31.25Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
31.03Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
31.03Single4AMIBucindolol4AMI-β1-Bucindolol
31.03Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
31.03Single4LDEBI1671074LDE-β2-BI167107
31.03Single4N4WSANT-14N4W-SMO-SANT-1
31.03Single4XEENeurotensin4XEE-NTS1-Neurotensin
31.03Single4XESNeurotensin4XES-NTS1-Neurotensin
31.03Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
31.03Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
31.03Single6A93Risperidone6A93-5-HT2A-Risperidone
31.03Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
31.03Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
31.03Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
31.03Single6YVRNTS8-136YVR-NTS1-NTS8-13
31.03Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
31.03Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
31.03Single7K15MKD0467K15-BLT1-MKD046-Na
31.03Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
31.03Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
31.03Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
31.03Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
31.03Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
31.03Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
31.03Single8XYIVUF106618XYI-CXCR3-VUF10661
31.03Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
31.03Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
31.03Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
31.03Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
31.03Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
31.03Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
31.03Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
31.03Consensusorexin_onOrthosteric Ligandox2_on
30.77Single2YDOAdenosine2YDO-A2A-Adenosine
30.77Single3REYXAC3REY-A2A-XAC
30.77Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
30.77Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
30.77Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
30.77Single4MBSMaraviroc4MBS-CCR5-Maraviroc
30.77Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
30.77Single4ZJCSB-6740424ZJC-OX1-SB-674042
30.77Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
30.77Single5IUBQ274563445IUB-A2A-Q27456344-Na
30.77Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
30.77Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
30.77Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
30.77Single6AQFZM-2413856AQF-A2A-ZM-241385
30.77Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
30.77Single6PS0S-Carazolol6PS0-β2-S-Carazolol
30.77Single6PS4ICI118-5516PS4-β2-ICI118-551
30.77Single6TPGEMPA6TPG-OX2-EMPA
30.77Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
30.77Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
30.77Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
30.77Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
30.77Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
30.77Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.77Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
30.77Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
30.77Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
30.77Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
30.77Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
30.77Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
30.77Single8K5CAcipimox8K5C-HCA2-Acipimox
30.77Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
30.77Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.77Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.77Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
30.77Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
30.77Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
30.77Consensushca_onOrthosteric Ligandhca2_on
30.56Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
30.56Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
30.30Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
30.30Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
30.30Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
30.30Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
30.30Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
30.30Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
30.00Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
30.00Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
30.00Single5X93K-87945X93-ETB-K-8794
30.00Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
30.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
30.00Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
30.00Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
30.00Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
30.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
30.00Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
30.00Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
30.00Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
30.00Consensuscck_onOrthosteric Ligandccka_on cckb_on
30.00Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
30.00Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
30.00Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
30.00Consensusendothelin_offOrthosteric Ligandetb_off
30.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
30.00Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
30.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
30.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
29.73Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single2Y01Dobutamine2Y01-β1-Dobutamine
29.63Single3EMLZM-2413853EML-A2A-ZM-241385
29.63Single3NY8ICI118-5513NY8-β2-ICI118-551
29.63Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
29.63Single4GBRS-Carazolol4GBR-β2-S-Carazolol
29.63Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
29.63Single5IU8Q274563475IU8-A2A-Q27456347-Na
29.63Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
29.63Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
29.63Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
29.63Single6PS1Timolol6PS1-β2-Timolol
29.63Single6S0LZM-2413856S0L-A2A-ZM-241385
29.63Single6TOTLemborexant6TOT-OX1-Lemborexant
29.63Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
29.63Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
29.63Single7BU7BI1671077BU7-β1-BI167107
29.63Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
29.63Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
29.63Single7PYRPSB-21157PYR-A2A-PSB-2115
29.63Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
29.63Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
29.63Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
29.63Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
29.63Single8CU6LJ-45178CU6-A2A-LJ-4517
29.63Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
29.63Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
29.63Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
29.63Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
29.63Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
29.63Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
29.63Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.63Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.63Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.63Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.63Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.63Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.63Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.63Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.63Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.63Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.63Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
29.63Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
29.63Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
29.63Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
29.63Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
29.63Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
29.63Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
29.63Single8K5DGSK2560738K5D-HCA2-GSK256073
29.63Single8T1WCVN4248T1W-GPR6-CVN424
29.63Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
29.63Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.63Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.63Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
29.63Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
29.63Single9CHXS-Carazolol9CHX-β2-S-Carazolol
29.63Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
29.63Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
29.63Consensusdopamine_offOrthosteric Ligandd2_off d3_off
29.63Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
29.63Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
29.63Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
29.41Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
29.41Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
29.17Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
29.03Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
29.03Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
29.03Single7SK9CCX6627SK9-ACKR3-CCX662
29.03Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
29.03Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
29.03Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
29.03Single8X5YAstemizole8X5Y-H1-Astemizole
29.03Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
29.03Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
29.03Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
28.57Single2RH1S-Carazolol2RH1-β2-S-Carazolol
28.57Single2Y00Dobutamine2Y00-β1-Dobutamine
28.57Single2YCWS-Carazolol2YCW-β1-S-Carazolol
28.57Single4JKVTaladegib4JKV-SMO-Taladegib
28.57Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
28.57Single5D6LS-Carazolol5D6L-β2-S-Carazolol
28.57Single5JQHS-Carazolol5JQH-β2-S-Carazolol
28.57Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
28.57Single6E67BI1671076E67-β2-BI167107-Gs (fused)
28.57Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
28.57Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
28.57Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
28.57Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
28.57Single6TP6Filorexant6TP6-OX1-Filorexant
28.57Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
28.57Single6Z4SSR486926Z4S-NTS1-SR48692
28.57Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
28.57Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
28.57Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
28.57Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
28.57Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
28.57Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
28.57Single7WC6LSD7WC6-5-HT2A-LSD
28.57Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
28.57Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
28.57Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8GNEKW-63568GNE-A2A-KW-6356-Na
28.57Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
28.57Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
28.57Single8QOTNanobody-E8QOT-μ-Nanobody-E
28.57Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
28.57Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
28.57Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
28.57Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
28.57Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
28.57Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
28.57Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
28.57Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
28.57Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
28.57Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
28.57Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
28.57Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
28.57Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
28.57Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
28.57Consensusamine_offonOrthosteric Ligandamine_off amine_on
28.57Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
28.57Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
28.57Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
28.57Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
28.57Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
28.57Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.57Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
28.57Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
28.57Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
28.57Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
28.57Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
28.57Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
28.57Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
28.57Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
28.57Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
28.57Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
28.57Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Consensustrace-amine_onOrthosteric Ligandta1_on
28.12Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
28.12Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
28.12Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
28.12Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
28.12Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.12Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
28.12Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
28.12Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
28.12Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
28.12Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
28.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
28.00Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
28.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
28.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
28.00Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
28.00Single8K5BNiacin8K5B-HCA2-Niacin
28.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
28.00Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
28.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
27.78Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
27.59Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
27.59Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
27.59Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
27.59Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
27.59Single5D5AS-Carazolol5D5A-β2-S-Carazolol
27.59Single5D5BS-Carazolol5D5B-β2-S-Carazolol
27.59Single5V57TC1145V57-SMO-TC114
27.59Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
27.59Single6H7JIsoprenaline6H7J-β1-Isoprenaline
27.59Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
27.59Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
27.59Single6WGTLSD6WGT-5-HT2A-LSD
27.59Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
27.59Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
27.59Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
27.59Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
27.59Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
27.59Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
27.59Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
27.59Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
27.59Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
27.59Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
27.59Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.59Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
27.59Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.59Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
27.59Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
27.59Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
27.59Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
27.59Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
27.59Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
27.59Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
27.59Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
27.59Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
27.59Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
27.59Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
27.59Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
27.59Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
27.59Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
27.59Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
27.59Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
27.59Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
27.59Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
27.59Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.59Consensustachykinin_offOrthosteric Ligandnk1_off
27.59Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
27.27Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
27.27Single8IEBA1LYA8IEB-GPR156-A1LYA
27.27Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
27.27Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
26.92Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
26.92Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
26.92Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
26.92Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
26.92Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
26.92Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
26.92Single5WS3EMPA5WS3-OX2-EMPA
26.92Single6AKXA4R6AKX-CCR5-A4R
26.92Single6AKYMaraviroc6AKY-CCR5-Maraviroc
26.92Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
26.92Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
26.92Single6TODEMPA6TOD-OX1-EMPA-Na
26.92Single7BR3Elagolix7BR3-GnRH1-Elagolix
26.92Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
26.92Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
26.92Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
26.92Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
26.92Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
26.92Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
26.92Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
26.92Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
26.92Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
26.92Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
26.92Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
26.92Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
26.92Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
26.92Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
26.92Consensusalpha2_offOrthosteric Ligandalpha2c_off
26.92Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
26.92Consensusorexin_offOrthosteric Ligandox2_off ox1_off
26.92Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
26.92Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
26.67Single3D4STimolol3D4S-β2-Timolol
26.67Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
26.67Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
26.67Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
26.67Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
26.67Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
26.67Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
26.67Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
26.67Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.67Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
26.67Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.67Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
26.67Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
26.67Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
26.67Single8JWY2-1188JWY-A2A-2-118
26.67Single8JWZAB9288JWZ-A2A-AB928-Na
26.67Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
26.67Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
26.67Consensusalpha1_offOrthosteric Ligandalpha1a_off
26.67Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
26.67Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
26.67Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
26.67Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
26.67Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
26.67Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
26.67Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
26.67Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.67Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.47Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
26.47Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
26.47Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
26.47Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
26.32Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
25.93Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
25.93Single5IU7Q274563465IU7-A2A-Q27456346-Na
25.93Single5JTBZM-2413855JTB-A2A-ZM-241385
25.93Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
25.93Single5UVIZM-2413855UVI-A2A-ZM-241385
25.93Single6KUXRS-799486KUX-α2a-RS-79948
25.93Single6PS5S-Propranolol6PS5-β2-S-Propranolol
25.93Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
25.93Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
25.93Single6V9SGTPL114036V9S-OX1-GTPL11403
25.93Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
25.93Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
25.93Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
25.93Single6ZINSR486926ZIN-NTS1-SR48692
25.93Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
25.93Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
25.93Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
25.93Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
25.93Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
25.93Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
25.93Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
25.93Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.93Single7UL3Famotidine7UL3-H2-Famotidine
25.93Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
25.93Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
25.93Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
25.93Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.93Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
25.93Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
25.93Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
25.93Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
25.93Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
25.93Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
25.93Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.93Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.93Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
25.93Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
25.93Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
25.93Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
25.93Single8IHKAcifran8IHK-HCA3-Acifran
25.93Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
25.93Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
25.93Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.93Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.93Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
25.93Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
25.93Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
25.93Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
25.93Consensusa2_offOrthosteric Liganda2a_off
25.93Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
25.93Consensusalpha1_onOrthosteric Ligandalpha1a_on
25.93Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
25.93Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
25.93Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
25.93Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
25.93Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
25.93Consensusgrh_offOrthosteric Ligandgnrh1_off
25.93Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
25.81Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
25.81Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
25.81Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.81Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
25.81Single7UM4AS26747237UM4-5-HT5A-AS2674723
25.81Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
25.81Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
25.81Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.81Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
25.81Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
25.81Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.81Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
25.81Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
25.81Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
25.81Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
25.81Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
25.81Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
25.81Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
25.71Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
25.71Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
25.71Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
25.71Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
25.71Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
25.64Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
25.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
25.00Single2Y02Carmoterol2Y02-β1-Carmoterol
25.00Single2Y04Salbutamol2Y04-β1-Salbutamol
25.00Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
25.00Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
25.00Single3RFMCaffeine3RFM-A2A-Caffeine
25.00Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
25.00Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
25.00Single4QKX35V4QKX-β2-35V
25.00Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
25.00Single5TGZAM65385TGZ-CB1-AM6538
25.00Single5UIGCmpd-15UIG-A2A-Cmpd-1
25.00Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
25.00Single5ZTYAM102575ZTY-CB2-AM10257
25.00Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
25.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
25.00Single6H7MSalbutamol6H7M-β1-Salbutamol
25.00Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
25.00Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
25.00Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
25.00Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
25.00Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
25.00Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
25.00Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
25.00Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
25.00Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
25.00Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
25.00Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
25.00Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
25.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
25.00Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
25.00Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
25.00Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
25.00Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
25.00Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
25.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
25.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
25.00Single7YXAONO-54306087YXA-S1P5-ONO-5430608
25.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
25.00Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
25.00Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
25.00Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
25.00Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
25.00Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
25.00Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8JJOAlprenolol8JJO-β2-Alprenolol
25.00Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
25.00Single8JXRLSD8JXR-D1-LSD
25.00Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
25.00Single8RLNLUF58348RLN-A2A-LUF5834
25.00Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
25.00Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
25.00Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
25.00Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
25.00Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
25.00Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
25.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
25.00Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
25.00Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
25.00Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
25.00Consensus5ht5_onOrthosteric Ligand5ht5a_on
25.00Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
25.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
25.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
25.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
25.00Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
25.00Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
25.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
25.00Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
25.00Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
25.00Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
25.00Consensusp2y_offOrthosteric Ligandp2y1_off
24.32Single6FJ3PTH6FJ3-PTH1-PTH
24.32Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
24.32Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
24.24Single4XT1Fractalkine4XT1-US28-Fractalkine
24.24Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
24.24Single8IEBA1LYA8IEB-GPR156-A1LYA
24.24Single8IEPA1LYA8IEP-GPR156-A1LYA
24.24Single8IEPA1LYA8IEP-GPR156-A1LYA
24.24Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
24.24Single8WKYPG-9348WKY-MC4-PG-934
24.24Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
24.24Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
24.24Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single2Y03Isoprenaline2Y03-β1-Isoprenaline
24.14Single5TVNLSD5TVN-5-HT2B-LSD
24.14Single5WIUNemonapride5WIU-D4-Nemonapride
24.14Single5WIVNemonapride5WIV-D4-Nemonapride-Na
24.14Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
24.14Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
24.14Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
24.14Single6PS6Timolol6PS6-β2-Timolol
24.14Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
24.14Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
24.14Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
24.14Single7SINNPS-21437SIN-CaS-NPS-2143
24.14Single7SINNPS-21437SIN-CaS-NPS-2143
24.14Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
24.14Single7W41PD1762527W41-BB2-PD176252
24.14Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
24.14Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
24.14Single8JXSPF-61428JXS-D1-PF-6142
24.14Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
24.14Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
24.14Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
24.14Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
24.14Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
24.14Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
24.14Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
24.14Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
24.14Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
24.14Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
24.14Consensusblt_offOrthosteric Ligandblt1_off
24.14Consensusbombesin_offOrthosteric Ligandbb2_off
24.14Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
24.14Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
24.14Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
24.14Consensusep_offOrthosteric Ligandep4_off
24.14Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
24.00Single3UZAGTPL92363UZA-A2A-GTPL9236
24.00Single4XNWMRS25004XNW-P2Y1-MRS2500
24.00Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
24.00Single7V6A-7V6A-M4-PubChem 9864275-Gi1/β1/γ2
24.00Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
24.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
24.00Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
24.00Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
23.68Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
23.68Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
23.53Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
23.53Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
23.53Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
23.33Single4BV0Neurotensin4BV0-NTS1-Neurotensin
23.33Single4DJHJDTic4DJH-κ-JDTic
23.33Single5V54Methiothepin5V54-5-HT1B-Methiothepin
23.33Single6J20Aprepitant6J20-NK1-Aprepitant
23.33Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
23.33Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
23.33Single6TQ7SB-3348676TQ7-OX1-SB-334867
23.33Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
23.33Single7B6WCyclazosin7B6W-α1b-Cyclazosin
23.33Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
23.33Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
23.33Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
23.33Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
23.33Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
23.33Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
23.33Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.33Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
23.33Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
23.33Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
23.33Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
23.33Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
23.33Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
23.33Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
23.33Single8XVLZibotentan8XVL-ETA-Zibotentan
23.33Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
23.33Consensus5ht1_offOrthosteric Ligand5ht1b_off
23.33Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
23.33Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
23.33Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
23.33Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
23.33Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
23.33Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
23.33Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
23.33Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
23.33Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
23.08Single3OE9IT1t3OE9-CXCR4-IT1t
23.08Single3PBLEticlopride3PBL-D3-Eticlopride
23.08Single4O9RCyclopamine4O9R-SMO-Cyclopamine
23.08Single5L7IVismodegib5L7I-SMO-Vismodegib
23.08Single6HLLCP999946HLL-NK1-CP99994
23.08Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
23.08Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
23.08Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
23.08Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
23.08Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
23.08Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
23.08Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
23.08Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
23.08Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
23.08Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
23.08Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
23.08Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
23.08Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
23.08Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
23.08Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
23.08Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Single9B9Y7DY9B9Y-CB1-7DY
23.08Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
23.08Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
23.08Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
23.08Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
23.08Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
23.08Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
22.86Single6W25SHU91196W25-MC4-SHU9119-Ca
22.86Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
22.58Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
22.58Single4PY02MeSATP4PY0-P2Y12-2MeSATP
22.58Single6CM4Risperidone6CM4-D2-Risperidone
22.58Single7DFPSpiperone7DFP-D2-Spiperone
22.58Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
22.58Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
22.58Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
22.58Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
22.58Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
22.58Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
22.58Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
22.58Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
22.58Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
22.58Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
22.58Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
22.58Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
22.58Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
22.58Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
22.58Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
22.58Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
22.50Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
22.22Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
22.22Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
22.22Single4BWBNeurotensin4BWB-NTS1-Neurotensin
22.22Single4QINSAG1.54QIN-SMO-SAG1.5
22.22Single4S0VSuvorexant4S0V-OX2-Suvorexant
22.22Single5ZKQABT-4915ZKQ-PAF-ABT-491
22.22Single6B73MP11046B73-κ-MP1104
22.22Single6DS0Ly2660976DS0-5-HT2B-Ly266097
22.22Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
22.22Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
22.22Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
22.22Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
22.22Single6TPJSuvorexant6TPJ-OX2-Suvorexant
22.22Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
22.22Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
22.22Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
22.22Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
22.22Single7F8ULintitript7F8U-CCKA-Lintitript
22.22Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
22.22Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
22.22Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
22.22Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
22.22Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
22.22Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
22.22Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
22.22Single7XRRLemborexant7XRR-OX2-Lemborexant
22.22Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
22.22Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
22.22Single8IWESpermidine8IWE-TA9-Spermidine
22.22Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
22.22Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
22.22Single8Y0HVUF114188Y0H-CXCR3-VUF11418
22.22Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
22.22Single9BA0A1AKN9BA0-CB1-A1AKN
22.22Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
22.22Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
22.22Consensusangiotensin_offOrthosteric Ligandat1_off
22.22Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
22.22Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
22.22Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
22.22Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
22.22Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
22.22Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
21.95Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
21.88Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
21.88Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
21.88Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
21.88Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
21.88Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
21.88Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
21.88Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
21.88Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
21.88Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
21.88Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
21.88Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
21.62Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
21.62Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
21.43Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
21.43Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
21.43Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
21.43Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
21.43Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
21.43Single6TP3Nemorexant6TP3-OX1-Nemorexant
21.43Single6TPKRetosiban6TPK-OT-Retosiban
21.43Single6VI4JDTic6VI4-κ-JDTic
21.43Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
21.43Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
21.43Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
21.43Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
21.43Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
21.43Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
21.43Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
21.43Single7T32ZM-2413857T32-A2A-ZM-241385
21.43Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
21.43Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
21.43Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
21.43Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
21.43Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
21.43Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
21.43Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
21.43Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
21.43Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
21.43Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
21.43Single8K2WAMG4878K2W-CXCR3-AMG487
21.43Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
21.43Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
21.43Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
21.43Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
21.43Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
21.43Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
21.43Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
21.43Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single9BJKNaloxone9BJK-μ-Naloxone-NAM
21.43Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
21.43Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
21.43Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
21.43Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
21.43Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
21.43Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
21.43Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
21.43Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
21.43Consensusvasop-oxy_offOrthosteric Ligandot_off
21.21Single5EE7MK08935EE7-Glucagon-MK0893
21.21Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
21.21Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
21.21Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
21.21Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
21.21Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.21Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
21.21Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
21.21Single8IEIA1LYA8IEI-GPR156-A1LYA
21.21Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
21.21Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
21.21Consensuskisspeptin_onOrthosteric Ligandkiss1_on
21.05Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
21.05Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
21.05Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
21.05Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
20.83Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
20.83Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
20.83Single8PWNTheophylline8PWN-A2A-Theophylline
20.69Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
20.69Single4YAYZD-71554YAY-AT1-ZD-7155
20.69Single5DHHSB-6121115DHH-NOP-SB-612111
20.69Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
20.69Single5T04Neurotensin5T04-NTS1-Neurotensin
20.69Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
20.69Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
20.69Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
20.69Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.69Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
20.69Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
20.69Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
20.69Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
20.69Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
20.69Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
20.69Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
20.69Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
20.69Single7V3ZCP559407V3Z-CB1-CP55940
20.69Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
20.69Single7WC7Lisuride7WC7-5-HT2A-Lisuride
20.69Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
20.69Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
20.69Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
20.69Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
20.69Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
20.69Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
20.69Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
20.69Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
20.69Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
20.69Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
20.69Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
20.69Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
20.69Single8X64Desloratadine8X64-H1-Desloratadine
20.69Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
20.69Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
20.69Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
20.69Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
20.69Single9B9ZA1AKO9B9Z-CB1-A1AKO
20.69Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
20.69Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
20.69Consensusalpha2_onOrthosteric Ligandalpha2b_on
20.69Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
20.69Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
20.69Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
20.69Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
20.69Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
20.69Consensusblt_onOrthosteric Ligandblt1_on
20.69Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
20.69Consensuscck_offOrthosteric Ligandccka_off
20.69Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
20.69Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
20.69Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
20.69Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
20.69Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
20.69Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
20.69Consensusleukotriene_onOrthosteric Ligandblt_on
20.69Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
20.59Single7QA8Peptide7QA8-STE2-Peptide
20.59Single7QA8Peptide7QA8-STE2-Peptide
20.59Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
20.59Single8IEIA1LYA8IEI-GPR156-A1LYA
20.59Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.59Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.59Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.59Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
20.51Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
20.51Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
20.51Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
20.51Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
20.51Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
20.00Single4NTJAZD12834NTJ-P2Y12-AZD1283
20.00Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
20.00Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
20.00Single6GPXMK08126GPX-CCR2-MK0812
20.00Single6HLPNetupitant6HLP-NK1-Netupitant
20.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
20.00Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
20.00Single6LUQHaloperidol6LUQ-D2-Haloperidol
20.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
20.00Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
20.00Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
20.00Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
20.00Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
20.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
20.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.00Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
20.00Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
20.00Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
20.00Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
20.00Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.00Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
20.00Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
20.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
20.00Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
20.00Single8ZMFA1L108ZMF-5-HT2C-A1L10
20.00Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
20.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
20.00Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
20.00Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
20.00Consensussensory_onOrthosteric Ligandopsins_on
20.00Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
19.51Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
19.44Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
19.44Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
19.35Single4U15Tiotropium4U15-M3-Tiotropium
19.35Single5XR8AM8415XR8-CB1-AM841
19.35Single5XRAAM115425XRA-CB1-AM11542
19.35Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
19.35Single6E59L-7607356E59-NK1-L-760735
19.35Single6OL9Tiotropium6OL9-M5-Tiotropium
19.35Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
19.35Single7FEECP559407FEE-CB1-CP55940-ZCZ011
19.35Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
19.35Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
19.35Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
19.35Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
19.35Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
19.35Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
19.35Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
19.35Single9BJKNAM9BJK-μ-Naloxone-NAM
19.35Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
19.35Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
19.35Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
19.35Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
19.35Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
19.35Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
19.35Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
19.23Single3OE6IT1t3OE6-CXCR4-IT1t
19.23Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
19.23Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
19.23Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
19.23Single6ME5Agomelatine6ME5-MT1-Agomelatine
19.23Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
19.23Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
19.23Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
19.23Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
19.23Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
19.23Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
19.23Single7WC5Psilocin7WC5-5-HT2A-Psilocin
19.23Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
19.23Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
19.23Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
19.23Single8JPSCCL78JPS-ACKR1-CCL7
19.23Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
19.23Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
19.23Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
19.23Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
19.23Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
19.23Consensus5ht2_onOrthosteric Ligand5ht2b_on
19.23Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
19.23Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
19.23Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
19.23Consensusgi_sensoryOrthosteric Ligandgi_opsins
19.23Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
19.23Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
19.23Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
19.23Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
19.23Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
19.23Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
19.23Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
19.15Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
19.05Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
19.05Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
18.92Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
18.92Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
18.92Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
18.92Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
18.92Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
18.75Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
18.75Single5CXVTiotropium5CXV-M1-Tiotropium
18.75Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
18.75Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
18.75Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
18.75Single6KQICP559406KQI-CB1-CP55940-Org27569
18.75Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
18.75Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
18.75Single6ZG4HTL00099366ZG4-M1-HTL0009936
18.75Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
18.75Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
18.75Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
18.75Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
18.75Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
18.75Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
18.75Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
18.75Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
18.75Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
18.75Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
18.60Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
18.60Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
18.60Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
18.60Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
18.52Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
18.52Single7SRQLSD7SRQ-5-HT2B-LSD
18.52Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
18.52Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
18.52Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
18.52Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
18.52Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
18.52Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
18.52Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
18.52Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
18.52Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
18.52Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
18.52Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
18.52Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
18.52Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
18.52Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
18.52Consensusgq_nucleotideOrthosteric Ligandgq_p2y
18.52Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
18.42Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
18.42Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
18.42Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
18.18Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
18.18Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
18.18Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
18.18Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
18.18Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
18.18Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
18.18Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8XVJMacitentan8XVJ-ETA-Macitentan
18.18Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
18.18Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
18.18Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
18.18Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.95Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
17.95Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
17.95Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
17.95Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
17.86Single3ODUIT1t3ODU-CXCR4-IT1t
17.86Single5U09Taranabant5U09-CB1-Taranabant
17.86Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
17.86Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
17.86Single6ME2Ramelteon6ME2-MT1-Ramelteon
17.86Single6ME9Ramelteon6ME9-MT2-Ramelteon
17.86Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
17.86Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
17.86Single7F8YDevazepide7F8Y-CCKA-Devazepide
17.86Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
17.86Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
17.86Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
17.86Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
17.86Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
17.86Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
17.86Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
17.86Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
17.86Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
17.86Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
17.86Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
17.86Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
17.86Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
17.86Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
17.86Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
17.86Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
17.86Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
17.86Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
17.86Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
17.86Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
17.86Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
17.86Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
17.86Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
17.86Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
17.86Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
17.86Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
17.86Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
17.86Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
17.86Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
17.86Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
17.86Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
17.86Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
17.86Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
17.78Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.65Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
17.65Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
17.50Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
17.50Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
17.50Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
17.50Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
17.50Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
17.24Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
17.24Single6A94Zotepine6A94-5-HT2A-Zotepine
17.24Single6IQLL7458706IQL-D4-L745870
17.24Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
17.24Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
17.24Single6TPNHTL66416TPN-OX2-HTL6641
17.24Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
17.24Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
17.24Single6ZG9GSK10347026ZG9-M1-GSK1034702
17.24Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
17.24Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
17.24Single7VV6C48/807VV6-MRGPRX2-C48/80
17.24Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
17.24Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
17.24Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
17.24Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
17.24Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
17.24Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
17.24Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
17.24Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
17.24Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
17.24Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
17.14Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
17.14Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
17.14Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.14Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
17.14Single8KIGSHU91198KIG-MC3-SHU9119-Ca
17.07Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
17.07Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
17.07Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
17.07Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
16.67Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
16.67Single5DHGC-355DHG-NOP-C-35
16.67Single5MZPCaffeine5MZP-A2A-Caffeine-Na
16.67Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
16.67Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
16.67Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
16.67Single6DRXLisuride6DRX-5-HT2B-Lisuride
16.67Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
16.67Single6GPSMK08126GPS-CCR2-MK0812
16.67Single6IIVDaltroban6IIV-TP-Daltroban
16.67Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
16.67Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
16.67Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
16.67Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
16.67Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
16.67Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
16.67Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
16.67Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.67Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
16.67Single8X63Mepyramine8X63-H1-Mepyramine
16.67Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
16.67Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
16.67Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
16.67Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
16.67Consensushistamine_offOrthosteric Ligandh1_off
16.67Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
16.67Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
16.28Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
16.28Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
16.22Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
16.22Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.22Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.13Single5CGCHTL142425CGC-mGlu5-HTL14242
16.13Single5XPRBosentan5XPR-ETB-Bosentan
16.13Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
16.13Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
16.13Single7C4SS1P7C4S-S1P3-S1P
16.13Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
16.13Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
16.13Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
16.13Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
16.13Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
16.13Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
16.13Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
16.13Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
16.13Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
16.13Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.13Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.13Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
16.13Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
16.00Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
16.00Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
16.00Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
16.00Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
15.91Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
15.91Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.79Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
15.79Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
15.79Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
15.62Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
15.62Single5TZRMK86665TZR-FFA1-MK8666
15.62Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
15.62Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
15.62Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
15.62Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
15.62Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
15.62Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
15.62Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8EA0Iperoxo8EA0-M3-Iperoxo
15.62Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
15.62Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
15.62Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
15.62Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
15.62Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
15.62Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
15.62Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
15.62Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
15.56Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
15.56Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
15.56Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
15.56Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
15.38Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
15.38Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
15.38Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
15.38Single9CHUNoradrenaline9CHU-β2-Noradrenaline
15.38Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
15.38Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
15.38Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
15.15Single5X33BIIL2605X33-BLT1-BIIL260
15.15Single6IIURamatroban6IIU-TP-Ramatroban
15.15Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
15.15Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
15.15Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
15.00Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
15.00Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
14.81Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
14.81Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
14.81Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
14.81Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.81Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
14.81Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
14.81Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
14.81Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
14.81Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
14.71Single5CGDHTL142425CGD-mGlu5-HTL14242
14.71Single6K1QIRL25006K1Q-ETB-IRL2500
14.71Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
14.71Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
14.71Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
14.63Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
14.63Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
14.63Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
14.63Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
14.29Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
14.29Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
14.29Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
14.29Single6LI0C176LI0-GPR52-C17
14.29Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
14.29Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
14.29Single6TP4ACT-4622066TP4-OX1-ACT-462206
14.29Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
14.29Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
14.29Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
14.29Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
14.29Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
14.29Single7UL2SR486927UL2-NTS1-SR48692-Na
14.29Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
14.29Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
14.29Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
14.29Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
14.29Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
14.29Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
14.29Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
14.29Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
14.29Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
14.29Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
14.29Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
14.29Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
14.29Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
14.29Consensusneurotensin_offOrthosteric Ligandnts1_off
14.29Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
13.89Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
13.89Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
13.89Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
13.89Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.89Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
13.79Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
13.79Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
13.79Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
13.79Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
13.79Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
13.79Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
13.79Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
13.79Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
13.79Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
13.79Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
13.79Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
13.79Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
13.79Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
13.79Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
13.64Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
13.51Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
13.51Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
13.33Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
13.33Single3RZECidoxepin3RZE-H1-Cidoxepin
13.33Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
13.33Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
13.33Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
13.33Single7VODCariprazine7VOD-5-HT2A-Cariprazine
13.33Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
13.33Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
13.33Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
13.33Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
13.33Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
13.33Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
13.33Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
13.33Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
13.33Consensusopsins_offOrthosteric Ligandrhodopsin_off
13.33Consensussensory_offOrthosteric Ligandopsins_off
12.90Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
12.90Single4DAJTiotropium4DAJ-M3-Tiotropium
12.90Single4MQSIperoxo4MQS-M2-Iperoxo
12.90Single4U14Tiotropium4U14-M3-Tiotropium
12.90Single5DSGTiotropium5DSG-M4-Tiotropium
12.90Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
12.90Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.90Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
12.90Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
12.90Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
12.90Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
12.90Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
12.90Single9IYAONO-97105319IYA-GPR55-ONO-9710531
12.90Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
12.90Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
12.90Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
12.50Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
12.50Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
12.50Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
12.50Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
12.50Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
12.50Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
12.50Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
12.20Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
12.12Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
12.12Single7P2L4YI7P2L-mGlu5-4YI
12.12Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
12.12Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
12.00Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
12.00Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
12.00Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
12.00Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
11.90Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
11.76Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
11.76Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
11.76Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single7WC4Serotonin7WC4-5-HT2A-Serotonin
11.54Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
11.11Single3OE8IT1t3OE8-CXCR4-IT1t
11.11Single6TQ9SB-4081246TQ9-OX1-SB-408124
11.11Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
11.11Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
11.11Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
11.11Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
10.71Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
10.71Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
10.71Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
10.71Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
10.71Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
10.71Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
10.34Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
10.34Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
10.34Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
10.34Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
10.34Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
10.34Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
10.34Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
10.34Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
10.34Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
10.34Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.00Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
10.00Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
10.00Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
10.00Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
10.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
10.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
10.00Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
10.00Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
10.00Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
10.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
10.00Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
10.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
10.00Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
10.00Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
9.68Single6FFIMMPEP6FFI-mGlu5-MMPEP
9.68Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
9.68Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.68Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
9.38Single6FFHFenobam6FFH-mGlu5-Fenobam
9.38Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
9.38Single7F83PF-051904577F83-Ghrelin-PF-05190457
9.38Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
9.09Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
9.09Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
9.09Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
9.09Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
9.09Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
8.82Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
8.57Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
7.41Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
7.41Single8HS2Fab0468HS2-GPR20-Fab046
7.41Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
7.14Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
6.90Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
6.90Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
6.90Single7F61Cholesterol7F61-H3-PF-03654746-Cholesterol
6.90Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
6.90Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
6.67Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
6.67Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
6.67Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
6.67Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
6.67Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
6.67Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
6.67Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
6.45Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.88Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
5.88Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
5.88Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
5.71Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
4.17Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.17Single6D35Cholesterol6D35-SMO-Cholesterol
4.17Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.17Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.17Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.17Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.17Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
4.17Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
4.17Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
4.17Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
4.17Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.17Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
4.17Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.17Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.17Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.17Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.17Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.17Single7DTTCa7DTT-CaS-Ca-Ca
4.17Single7DTTCa7DTT-CaS-Ca-Ca
4.17Single7DTUTryptophan7DTU-CaS-Tryptophan
4.17Single7DTUTryptophan7DTU-CaS-Tryptophan
4.17Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.17Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.17Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.17Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.17Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.17Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.17Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.17Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.17Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.17Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.17Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.17Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.17Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.17Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.17Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.17Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.17Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.17Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.17Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.17Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.17Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.17Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.17Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.17Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.17Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.17Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.17Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.17Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.17Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.17Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.17Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
4.17Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.17Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.17Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.17Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.17Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.17Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.17Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.17Single7XW7K1-707XW7-TSH-K1-70
4.17Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.17Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.17Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.17Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.17Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.17Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.17Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.17Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.17Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.17Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.17Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.17Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.17Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.17Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.17Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.17Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.17Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.17Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
4.17Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
4.17Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.17Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.17Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
4.17Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
4.17Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.17Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.17Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.17Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.17Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.17Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
4.17Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
4.17Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
4.17Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
4.17Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
4.17Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
4.17Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.17Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.17Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.17Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.17Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.17Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.17Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.17Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.17Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.17Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.17Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.17Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.17Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.17Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.17Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.17Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.17Single8W8SAA-148W8S-GPR101-AA-14
4.17Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.17Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
4.17Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
4.17Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.17Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
4.17Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
4.17Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.17Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.17Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.17Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.17Single8WVXNorrin8WVX-LGR4-Norrin
4.17Single8WVYNorrin8WVY-LGR4-Norrin
4.17Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.17Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.17Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.17Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.17Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.17Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.17Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.17Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.17Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.17Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.17Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.17Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.17Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.17Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.17Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.17Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.17Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.17Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.17Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.17Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.17Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.17Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.17Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.17Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.17Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.17Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.17Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.00Single8W8RAA-148W8R-GPR101-AA-14-chim(NtGi1-Gs)/β1/γ2
4.00Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.00Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.85Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
3.85Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
3.85Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
3.70Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
3.70Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
3.70Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
3.70Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
3.70Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.70Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
3.57Single5L7DCholesterol5L7D-SMO-Cholesterol
3.57Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.57Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.57Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
3.45Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
3.33Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
3.12Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
2.70Single7SHEPI; PE7SHE-GPR158-PI; PE
2.63Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
2.50Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.50Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.44Single7SHEPI; PE7SHE-GPR158-PI; PE
2.44Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
2.38Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.38Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.33Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.17Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
7F6H 7F6H-BK2-Bradykinin-Gq/β1/γ2
7F6I 7F6I-BK2-Kallidin-Gq/β1/γ2
Net Summary
Imin 3.21
Number of Linked Nodes 861
Number of Links 1027
Number of Hubs 145
Number of Links mediated by Hubs 582
Number of Communities 25
Number of Nodes involved in Communities 202
Number of Links involved in Communities 287
Path Summary
Number Of Nodes in MetaPath 87
Number Of Links MetaPath 86
Number of Shortest Paths 6599745
Length Of Smallest Path 3
Average Path Length 39.4948
Length of Longest Path 61
Minimum Path Strength 0.6125
Average Path Strength 6.27101
Maximum Path Strength 26.43
Minimum Path Correlation 0.7
Average Path Correlation 0.992838
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.92308
Average % Of Corr. Nodes 27.9093
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 53.1229
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
gq_peptidegq_cck
gq_kisspeptin
gq_bradykinin
gq_bombesin
gq_angiotensin



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download gq_bradykinin.zip



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