Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 1.10049602
2G.HN.45 1.87456404
3G.HN.48 2.26044403
4G.S1.02 5.11529495
5G.S1.06 5.45059448
6G.H1.01 4.74485449
7G.H1.07 2.62603409
8G.S2.01 3.34618419
9G.S2.04 1.96485406
10G.S2.08 8.90412495
11G.S3.01 5.16368494
12G.S3.03 7.76741597
13G.S3.04 6.39103416
14G.S3.06 6.56343615
15G.s3h2.03 5.01779419
16G.H2.02 4.09706418
17G.H2.04 4.46282509
18G.H2.06 5.71306519
19G.H2.07 5.10865719
20G.H2.09 5.98574418
21G.h2s4.01 6.554519
22G.S4.02 4.25435518
23G.S4.03 3.56794447
24G.S4.04 6.00221409
25G.s4h3.04 5.71284668
26G.s4h3.05 6.27647469
27G.s4h3.10 1.28471409
28G.H3.01 6.93941469
29G.H3.09 5.90922619
30G.H3.13 4.16265415
31G.H3.15 4.64544418
32G.H3.17 7.09539615
33G.H3.18 6.45544419
34G.S5.02 3.91426416
35G.S5.03 3.264548
36G.S5.05 3.79566849
37G.HG.03 2.5025466
38G.HG.04 5.19047569
39G.hgh4.02 4.421186167
40G.hgh4.05 8.37735407
41G.H4.03 5.84897404
42G.H4.10 8.907654166
43G.H4.15 3.53226608
44G.h4s6.02 5.74838418
45G.S6.02 5.42286747
46G.H5.03 4.69206448
47G.H5.08 7.38382498
48G.H5.15 2.79353407
49G.H5.19 3.060294188
50G.H5.26 4.31506505
51b.1x15 2.27574407
52b.h2x1 3.79441405
53b.lhb1x11 3.75838404
54b.b1x3 5.06044457
55b.b1x4 3.18676457
56b.l1x3 7.76804679
57b.b2x1 7.73318518
58b.b2x5 6.17441607
59b.l3x2 4.52929579
60b.b4x2 5.74177408
61b.b4x6 8.5637779
62b.l4x2 10.2001454
63b.b5x2 5.96544407
64b.b5x3 5.90008779
65b.b5x5 5.29191405
66b.b5x7 6.00147487
67b.l5x1 4.07624588
68b.l5x5 7.44833619
69b.b6x5 3.79333606
70b.l6x5 6.214564134
71b.b7x1 5.590715134
72b.l7x2 4.52574419
73b.b8x4 5.05157686
74b.l8x8 4.82912484
75b.b9x3 4.08868486
76b.l9x3 7.79388519
77b.l9x6 4.81779818
78b.b10x5 4.07814609
79b.l10x1 3.66662403
80b.b11x4 5.50485419
81b.l11x2 6.78235519
82b.b12x6 10.2538518
83b.b12x7 5.65765439
84b.b13x7 7.74141537
85b.l13x3 7.44186639
86b.l13x6 4.59906519
87b.l13x7 4.64662439
88b.b14x3 4.03471435
89b.b15x1 5.48775639
90b.b15x2 6.55838416
91b.b15x3 4.38529439
92b.l15x1 4.69941517
93b.l15x2 4.91553539
94b.b16x4 8.25894536
95b.b16x5 4.94471515
96b.b16x6 8.66598638
97b.l16x3 5.70324413
98b.b17x5 6.07129517
99b.b17x7 8.84559418
100b.l17x3 8.07748719
101b.l17x6 6.34309419
102b.b18x3 4.83118418
103b.l18x1 6.235977106
104b.l18x2 5.523684107
105b.l18x3 7.324124105
106b.b19x2 5.95118716
107b.b19x4 5.35988518
108b.l19x2 5.2619
109b.b20x2 5.84573416
110b.b20x4 9.02686618
111b.b20x6 7.19755616
112b.b21x1 7.12412517
113b.b21x5 5.27956404
114b.b21x7 4.61118605
115b.b22x5 5.096945107
116b.l22x5 6.696235199
117b.b23x1 3.68691405
118b.b23x6 6.393436127
119b.l23x1 8.07426406
120b.b24x3 3.24985405
121b.b24x4 7.014126
122b.b24x6 6.017944128
123b.b25x3 6.306184125
124b.l25x3 8.047295119
125b.b26x3 3.60941406
126b.l27x1 10.352719
127b.l27x2 7.663974119
128b.b28x3 4.23271577
129b.b28x4 4.720475116
130b.b28x6 9.502354119
131b.b28x7 5.14588459
132g.h1x5 1.2802606
133g.h1x8 2.20456407
134g.h1x12 1.82988506
135g.l1x4 3.75108618
136g.h2x11 8.043824106
137g.ctx3 5.82833609
138g.ctx6 4.03071506
139g.ctx14 4.35823559
140g.ctx15 6.61426459
141g.ctx16 4.57824958
142Lig 6.100491920
1431x35 4.68735426
1441x39 5.81809407
1451x43 3.13265406
1461x53 2.98544409
1472x42 5.86282507
1482x44 5.30176406
1492x46 4.27847529
1502x50 6.34894529
1512x57 5.21794407
152E1x50 7.41731728
153E1x52 8.39965526
1543x29 3.50147424
1553x32 6.82265425
1563x34 4.486186145
1573x35 5.16691408
1583x37 4.60306506
1593x38 6.746474147
1603x50 5.24471409
1613x51 7.059274228
162I2x57 5.814026187
1634x50 8.883974149
164E2 10.04451423
165E2x50 6.65853429
166E2x52 2.95382424
1675x44 5.66897426
1685x47 5.49953528
1695x58 6.40659509
170I3 6.3711843
1716x44 4.20024529
1726x48 5.5605728
1736x49 4.15735405
1746x52 5.89662427
175E3 4.752354232
1767x34 6.26623524
1777x35 7.18988524
1787x42 7.85441427
1797x45 7.05221429
1807x49 5.67059529
1817x53 4.7402629
1828x50 3.773826218
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1G.HN.47 b.b5x3 10.1132.65412NoYes069
2b.b4x6 b.b5x3 22.271411.3953YesYes799
3b.b3x2 b.b4x6 36.46214.42176NoYes059
4b.b2x5 b.b3x2 36.81966.02941YesNo075
5b.b2x3 b.b2x5 44.58055.95294NoYes067
6b.b26x2 b.b2x3 44.94534.47882NoNo076
7b.b26x1 b.b26x2 45.37172.93412NoNo097
8b.b26x1 b.l27x1 45.84275.16NoYes099
9b.b2x1 b.l27x1 19.69766.86529YesYes189
10b.b2x1 b.l3x1 20.759612.4018YesNo089
11b.l3x1 b.l5x5 21.20118.05353NoYes099
12G.H3.17 b.l27x1 26.08783.97059YesYes159
13G.H3.15 G.H3.17 60.29747.17882YesYes185
14G.H2.08 G.H3.15 53.02383.74941NoYes188
15G.H2.04 G.H2.08 53.58292.87412YesNo098
16G.H2.04 G.H3.08 96.70763.28471YesNo099
17G.H3.08 G.S4.04 96.68436.01882NoYes099
18G.S4.04 G.s1h1.01 1003.01235YesNo099
19G.H1.01 G.s1h1.01 99.88383.07824YesNo099
20G.H1.01 G.S1.06 99.08976.80118YesYes498
21G.S1.06 G.S4.03 98.58882.76706YesYes487
22G.S1.04 G.S4.03 36.56735.03765NoYes077
23G.S1.04 G.S3.03 36.39693.72529NoYes077
24G.H5.11 G.S3.03 32.91535.70588NoYes987
25G.HG.04 G.s4h3.04 28.78356.00882YesYes698
26G.HG.04 G.s4h3.01 33.62179.31471YesNo097
27G.H4.11 G.s4h3.01 33.9683.35588NoNo077
28G.H4.11 G.H4.15 34.44532.80647NoYes078
29G.H3.09 G.H4.15 23.05412.96294YesYes098
30b.b4x2 b.b5x8 16.77373.34529YesNo085
31b.b5x7 b.b5x8 16.52153.39YesNo075
32b.l8x1 b.l8x8 10.72453.33059NoYes054
33b.b7x2 b.l8x1 10.30374.64529NoNo085
34b.b6x5 b.b7x2 10.48563.26353YesNo068
35b.b2x4 b.b6x5 13.9283.71882NoYes066
36b.b10x4 b.b2x4 14.17359.95765NoNo066
37b.b10x2 b.b10x4 13.62555.81529NoNo066
38b.b10x2 b.b6x2 30.57512.88294NoNo068
39b.b10x3 b.b6x2 30.85393.97647NoNo088
40b.b10x3 b.b11x4 44.00682.68412NoYes089
41b.b11x4 b.l9x3 43.91476.44412YesYes199
42G.H2.04 G.H2.07 82.35455.29412YesYes099
43G.H2.07 b.l9x6 93.6143.74471YesYes198
44b.l11x1 b.l9x6 42.06525.36882NoYes198
45b.b11x6 b.l11x1 50.53453.38353NoNo199
46G.H2.07 G.h2s4.01 11.13683.89177YesYes199
47b.l5x5 b.l7x2 13.68545.82765YesYes199
48G.H2.06 b.l9x6 73.50123.44YesYes198
49G.H2.06 b.l17x6 72.30167.80941YesYes199
50G.S4.03 G.S5.03 57.70053.80824YesYes478
51G.S4.04 G.S4.06 16.75233.31353YesNo097
52G.S5.03 G.S6.02 58.52732.98882YesYes487
53G.S6.02 I3 57.423910.0118YesYes473
54G.H5.11 G.H5.15 33.06852.88941NoYes087
55G.H5.15 G.H5.19 31.03873.24824YesYes078
56G.H5.19 I2x57 30.47163.47529YesYes1887
575x65 I3 51.21663.66353NoYes083
583x50 G.H5.23 13.25392.70294YesNo094
59G.H5.23 I2x57 13.42934.83412NoYes047
603x50 5x58 13.09617.98882YesYes099
615x58 5x61 51.93523.37824YesNo098
623x54 5x61 52.11286.96412NoNo088
633x54 5x65 52.29663.58588NoNo088
64b.l17x5 b.l17x6 80.55633.63588NoYes169
65b.l17x5 b.l19x2 80.33452.68412NoYes169
66b.b20x4 b.l19x2 30.94232.94294YesYes189
67b.b20x4 b.b20x6 29.88744.52823YesYes186
68b.b17x7 b.b20x6 40.104412.9865YesYes186
69b.b17x7 b.b21x1 31.1126.32177YesYes187
70b.1x19 b.b21x1 25.95144.27412NoYes167
71b.1x15 b.1x19 25.23743.75471YesNo076
72b.1x15 g.h1x11 19.88831.67706YesNo079
73b.1x11 g.h1x11 18.35564.08882NoNo089
74b.l17x3 b.l19x2 47.22783.18706YesYes199
75b.b20x6 b.l17x3 29.88694.39471YesYes169
76b.1x11 g.h1x12 17.58852.73706NoYes086
77b.b4x6 b.l1x3 11.63675.41471YesYes799
78b.l1x3 b.l3x2 10.68382.74294YesYes799
79b.b10x3 b.b11x2 16.14422.50412NoNo087
80b.b7x1 b.b8x3 11.06963.91471YesNo046
81b.b10x2 b.b14x3 17.22845.04059NoYes065
82b.b19x4 b.l17x3 15.9399.98412YesYes189
83b.b19x2 b.b20x6 18.99759.70765YesYes166
84b.b15x2 b.b19x2 16.01799.87059YesYes166
85b.b15x2 b.b16x5 12.23582.71706YesYes165
86b.b19x2 b.l20x1 10.27043.15353YesNo166
87b.b16x5 b.b17x4 20.61994.07176YesNo155
88b.b17x4 b.l16x3 13.75173.07824NoYes153
89b.l23x1 b.l25x6 36.636220.3894YesNo068
90b.l21x7 b.l23x1 22.23855.30706NoYes056
91b.l21x7 b.l23x2 21.9656.03941NoNo058
92b.b23x6 b.l23x2 19.99163.92353YesNo078
93b.b23x6 b.b24x6 16.05247.60471YesYes1278
94b.b22x1 b.l23x1 15.11343.74118NoYes086
95b.b22x2 b.b26x3 14.62184.15NoYes086
96b.b22x1 b.b22x2 14.84733.2NoNo088
97g.h1x12 g.h1x9 12.20531.03235YesNo066
98g.h1x5 g.h1x9 10.66293.35235YesNo066
993x47 5x58 38.31589.60823NoYes099
1003x47 5x54 38.17826.04471NoNo098
1015x54 6x44 37.95463.99NoYes089
1026x44 6x48 29.35518.31353YesYes298
1036x48 Lig 30.68273.03YesYes280
1042x42 3x49 11.67476.83176YesNo078
1053x49 I2x57 12.649312.2612NoYes087
1061x50 2x50 11.7036.19706NoYes099
1073x50 7x53 22.80964.35765YesYes099
1087x49 7x53 11.22664.17176YesYes299
109b.b2x5 b.l4x1 12.74524.36059YesNo075
110b.l4x1 g.ctx16 10.06364.81471NoYes558
111b.b21x7 b.b24x6 15.18796.52471YesYes058
112b.b11x6 b.l9x3 46.649912.7159NoYes199
113b.b14x3 b.b15x1 10.14082.65059YesYes359
114G.H3.09 G.S4.04 19.987911.6641YesYes099
115G.H4.15 G.S4.06 16.21715.47412YesNo087
116G.H3.17 b.l25x6 33.29473.52941YesNo158
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x33Lig9.292352NoYes4010
3x36Lig7.847652NoYes7010
5x43Lig4.322NoYes5010
6x52Lig3.664122YesYes7010
6x55Lig4.914122NoYes5010
6x51Lig4.021182NoYes6010
7x34Lig4.378822YesYes4010
7x38Lig5.753532NoYes5010
2x60Lig12.41822NoYes6010
2x63Lig4.151762NoYes4010
3x29Lig5.772352YesYes4010
3x32Lig10.69712YesYes5010
E2x50Lig2.682YesYes9010
1x392x574.211180YesYes7722
1x397x3510.30240YesYes7422
1x397x385.905880YesNo7521
2x563x325.867650NoYes6521
2x577x429.749410YesYes7721
2x603x323.152NoYes6511
2x607x427.427062NoYes6711
2x63E1x506.802942NoYes4812
E1x49E26.439410NoYes5321
3x25E1x505.761182NoYes9822
E1x50E2x5013.82712YesYes8921
3x22E28.758232NoYes3321
3x25E23.402942NoYes9321
3x25E2x506.958822NoYes9921
3x29E2x503.168242YesYes4911
3x29E2x522.767062YesYes4412
3x327x427.575882YesYes5711
3x334x605.165292NoNo4512
3x33E2x522.837652NoYes4412
3x363x373.512352NoYes7612
3x366x485.406472NoYes7811
3x375x434.621760YesNo6521
3x406x442.881762NoYes7922
3x406x485.527652NoYes7821
4x60E2x522.987652NoYes5422
4x63E23.614710NoYes5321
E2E239.79592YesYes3311
E2E2x515.597062YesNo3412
E2E2x523.222942YesYes3412
5x32E23.076470NoYes3321
5x35E27.337062NoYes1321
5x36E28.170592NoYes4321
5x39E23.403530NoYes6321
5x31E23.872NoYes4321
5x315x352.752942NoNo4122
5x365x406.552NoNo4422
5x445x474.602352YesYes6822
5x446x525.540592YesYes6721
5x476x528.532YesYes8721
6x446x488.313532YesYes9821
6x447x453.054712YesYes9922
6x486x525.851762YesYes8711
6x487x458.973532YesYes8912
6x517x373.367652NoNo6612
6x547x348.142940NoYes5421
6x587x348.188820NoYes3421
7x347x353.948822YesYes4412
7x347x386.671762YesNo4511
5x406x552.648820NoNo4521
6x48Lig3.032YesYes8010
7x42Lig6.665292YesYes7010
E2Lig4.138242YesYes3010
3x294x642.298242YesNo4512
6x487x411.820592YesNo8712
LigNT0.2094122YesNo0701

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
82.35Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
82.35Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
76.47Single8E0GBU728E0G-μ-BU72
72.73Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
72.22Single7YITNalfurafine7YIT-κ-Nalfurafine
72.22Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
72.22Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
70.59Single5C1MBU725C1M-μ-BU72
70.59Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
70.59Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
69.57Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
68.42Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
68.42Consensusendothelin_offOrthosteric Ligandetb_off
68.42Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
66.67Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
66.67Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
64.71Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
63.64Single6PT2KGCHM076PT2-δ-KGCHM07
61.90Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
61.90Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
61.90Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
61.90Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
61.11Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
61.11Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
61.11Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
60.00Single5X93K-87945X93-ETB-K-8794
60.00Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
60.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
60.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
60.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
59.09Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
59.09Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
58.82Single6TPGEMPA6TPG-OX2-EMPA
58.82Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
58.82Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
58.82Consensusalpha1_onOrthosteric Ligandalpha1a_on
58.82Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
58.82Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
58.82Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
57.89Single2YDVNECA2YDV-A2A-NECA
57.89Single4DJHJDTic4DJH-κ-JDTic
57.89Single4UHRCGS216804UHR-A2A-CGS21680
57.89Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
57.89Single5G53NECA5G53-A2A-NECA-Gs
57.89Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
57.89Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
57.89Single6TQ7SB-3348676TQ7-OX1-SB-334867
57.89Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
57.89Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
57.89Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
57.89Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
57.89Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
57.89Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
57.89Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
57.89Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
57.89Single8XVLZibotentan8XVL-ETA-Zibotentan
57.89Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
57.89Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
57.89Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
57.89Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
57.89Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
57.89Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
57.14Single3NY9ICI118-5513NY9-β2-ICI118-551
57.14Single4UG2CGS216804UG2-A2A-CGS21680
57.14Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
57.14Single8X5YAstemizole8X5Y-H1-Astemizole
57.14Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
57.14Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
57.14Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
55.56Single3NY8ICI118-5513NY8-β2-ICI118-551
55.56Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
55.56Single4GBRS-Carazolol4GBR-β2-S-Carazolol
55.56Single5DHHSB-6121115DHH-NOP-SB-612111
55.56Single6TOTLemborexant6TOT-OX1-Lemborexant
55.56Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
55.56Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
55.56Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
55.56Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
55.56Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
55.56Single8JXRLSD8JXR-D1-LSD
55.56Single8T1WCVN4248T1W-GPR6-CVN424
55.56Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
55.56Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
55.56Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
55.56Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
55.56Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
55.56Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
55.56Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
55.56Single9CHXS-Carazolol9CHX-β2-S-Carazolol
55.56Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
55.56Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
55.56Consensusdopamine_offOrthosteric Ligandd2_off d3_off
55.56Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
55.00Single4RWADIPP-NH24RWA-δ-DIPP-NH2
55.00Single7DFPSpiperone7DFP-D2-Spiperone
55.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
55.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
55.00Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
55.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
55.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
55.00Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
55.00Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
55.00Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
55.00Consensuslpa_offOrthosteric Ligandlpa1_off
55.00Consensuslpl_offOrthosteric Ligands1p_off lpa_off
55.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
55.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
54.55Single8WDTphotoNECA8WDT-A2A-photoNECA
54.17Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
54.17Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
53.85Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
53.85Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
52.94Single6B73MP11046B73-κ-MP1104
52.94Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
52.94Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
52.94Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
52.94Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
52.63Single2RH1S-Carazolol2RH1-β2-S-Carazolol
52.63Single2YCWS-Carazolol2YCW-β1-S-Carazolol
52.63Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
52.63Single5D6LS-Carazolol5D6L-β2-S-Carazolol
52.63Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
52.63Single5WQCEMPA5WQC-OX2-EMPA
52.63Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
52.63Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
52.63Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
52.63Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
52.63Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
52.63Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
52.63Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
52.63Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
52.63Single8JXSPF-61428JXS-D1-PF-6142
52.63Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
52.63Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
52.63Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
52.63Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
52.63Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
52.63Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
52.63Consensusamine_offonOrthosteric Ligandamine_off amine_on
52.63Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
52.63Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
52.63Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
52.63Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
52.63Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
52.63Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
52.63Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
52.63Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
52.63Consensustrace-amine_onOrthosteric Ligandta1_on
52.38Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
52.38Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
52.38Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
52.38Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
52.38Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
52.38Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
52.38Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
52.38Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
52.38Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
52.38Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
52.38Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
52.17Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
52.17Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
52.00Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
50.00Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
50.00Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
50.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
50.00Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
50.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
50.00Single5D5AS-Carazolol5D5A-β2-S-Carazolol
50.00Single5D5BS-Carazolol5D5B-β2-S-Carazolol
50.00Single5ZTYAM102575ZTY-CB2-AM10257
50.00Single6H7JIsoprenaline6H7J-β1-Isoprenaline
50.00Single6IQLL7458706IQL-D4-L745870
50.00Single6J21Aprepitant6J21-NK1-Aprepitant
50.00Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
50.00Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
50.00Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
50.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
50.00Single6PS4ICI118-5516PS4-β2-ICI118-551
50.00Single6PT3DPI-2876PT3-δ-DPI-287
50.00Single6TPNHTL66416TPN-OX2-HTL6641
50.00Single6ZG9GSK10347026ZG9-M1-GSK1034702
50.00Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
50.00Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
50.00Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
50.00Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
50.00Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
50.00Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
50.00Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
50.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
50.00Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
50.00Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
50.00Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
50.00Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
50.00Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
50.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
50.00Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
50.00Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
50.00Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
50.00Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
50.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
50.00Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
50.00Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
50.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
50.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
50.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
50.00Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
50.00Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
50.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
50.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
50.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
50.00Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
50.00Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
50.00Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
50.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
50.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
50.00Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
50.00Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
50.00Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
50.00Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
50.00Single9BJKNaloxone9BJK-μ-Naloxone-NAM
50.00Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
50.00Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
50.00Consensusa2_onOrthosteric Liganda2b_on
50.00Consensusa2_on_gpOrthosteric Liganda2b_on_gp
50.00Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
50.00Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
50.00Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
50.00Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
50.00Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
50.00Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
50.00Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
50.00Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
50.00Consensusbombesin_onOrthosteric Ligandbb2_on
50.00Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
50.00Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
50.00Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
50.00Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
50.00Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
50.00Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
50.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
50.00Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
50.00Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
50.00Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
50.00Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
50.00Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
50.00Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
50.00Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
50.00Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
50.00Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
48.15Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
48.15Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
48.15Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
48.15Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
48.00Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
48.00Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
47.83Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
47.83Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
47.83Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
47.83Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
47.83Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
47.83Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
47.83Consensuslpl_onOrthosteric Ligands1p_on lpa_on
47.83Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
47.83Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
47.83Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
47.62Single3D4STimolol3D4S-β2-Timolol
47.62Single4AMIBucindolol4AMI-β1-Bucindolol
47.62Single4LDEBI1671074LDE-β2-BI167107
47.62Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
47.62Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
47.62Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
47.62Single6A93Risperidone6A93-5-HT2A-Risperidone
47.62Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
47.62Single6ZG4HTL00099366ZG4-M1-HTL0009936
47.62Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
47.62Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
47.62Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
47.62Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
47.62Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
47.62Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
47.62Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
47.62Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
47.62Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
47.62Single8JJ8Formoterol8JJ8-β2-Formoterol
47.62Single8JJLOlodaterol8JJL-β2-Olodaterol
47.62Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
47.62Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
47.62Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
47.62Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
47.62Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
47.62Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
47.62Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
47.62Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
47.62Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
47.62Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
47.62Consensusorexin_onOrthosteric Ligandox2_on
47.37Single2Y04Salbutamol2Y04-β1-Salbutamol
47.37Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
47.37Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
47.37Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
47.37Single4EJ4Naltrindole4EJ4-δ-Naltrindole
47.37Single5DHGC-355DHG-NOP-C-35
47.37Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
47.37Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
47.37Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
47.37Single6PS1Timolol6PS1-β2-Timolol
47.37Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
47.37Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
47.37Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
47.37Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
47.37Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
47.37Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
47.37Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
47.37Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
47.37Single7UL4Alvimopan7UL4-μ-Alvimopan
47.37Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
47.37Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
47.37Single8CU6LJ-45178CU6-A2A-LJ-4517
47.37Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
47.37Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
47.37Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
47.37Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
47.37Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
47.37Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
47.37Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
47.37Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
47.37Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
47.37Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
47.37Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
47.37Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
47.37Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
47.37Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
47.37Single8JJOAlprenolol8JJO-β2-Alprenolol
47.37Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
47.37Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
47.37Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
47.37Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
47.37Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
47.37Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
47.37Single8X64Desloratadine8X64-H1-Desloratadine
47.37Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
47.37Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
47.37Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
47.37Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
47.37Consensusalpha2_onOrthosteric Ligandalpha2b_on
47.37Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
47.37Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
47.37Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
47.37Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
47.37Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
47.37Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
47.37Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
47.37Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
47.06Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
47.06Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
47.06Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
47.06Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
47.06Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
47.06Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
47.06Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
47.06Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
47.06Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
46.43Single6IGLIRL16206IGL-ETB-IRL1620
46.15Single8ZRTET-18ZRT-ETB-ET-1
45.83Single3QAKUK-4320973QAK-A2A-UK-432097
45.83Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
45.83Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
45.83Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
45.45Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
45.45Single6H7LDobutamine6H7L-β1-Dobutamine
45.45Single7EZCUKA7EZC-A2A-UKA
45.45Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
45.45Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
45.45Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
45.45Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
45.45Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
45.45Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
45.45Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
45.45Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
45.45Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
45.45Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
45.45Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
45.45Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
45.45Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
45.00Single2Y03Isoprenaline2Y03-β1-Isoprenaline
45.00Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
45.00Single5JQHS-Carazolol5JQH-β2-S-Carazolol
45.00Single5WIUNemonapride5WIU-D4-Nemonapride
45.00Single5WIVNemonapride5WIV-D4-Nemonapride-Na
45.00Single5XPRBosentan5XPR-ETB-Bosentan
45.00Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
45.00Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
45.00Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
45.00Single6PS6Timolol6PS6-β2-Timolol
45.00Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
45.00Single6TP6Filorexant6TP6-OX1-Filorexant
45.00Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
45.00Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
45.00Single7C61Ergotamine7C61-5-HT1B-Ergotamine
45.00Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
45.00Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
45.00Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
45.00Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
45.00Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
45.00Single7WC6LSD7WC6-5-HT2A-LSD
45.00Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
45.00Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
45.00Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
45.00Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
45.00Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
45.00Single8S4DCMF-0198S4D-Apelin-CMF-019
45.00Single8TF5Oleic acid8TF5-GPR6-Oleic acid
45.00Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
45.00Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
45.00Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
45.00Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
45.00Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
45.00Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
45.00Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
45.00Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
45.00Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
45.00Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
45.00Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
45.00Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
45.00Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
45.00Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
44.83Single6IGKEndothelin-36IGK-ETB-Endothelin-3
44.44Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
44.44Single5WS3EMPA5WS3-OX2-EMPA
44.44Single6AKXA4R6AKX-CCR5-A4R
44.44Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
44.44Single6TODEMPA6TOD-OX1-EMPA-Na
44.44Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
44.44Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
44.44Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
44.44Single7XRRLemborexant7XRR-OX2-Lemborexant
44.44Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
44.44Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
44.44Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
44.44Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
44.44Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
44.44Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
44.44Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
44.44Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
44.44Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
44.44Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
44.44Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
44.44Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
44.44Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
44.44Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
44.44Single8Y0HVUF114188Y0H-CXCR3-VUF11418
44.44Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
44.44Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
44.44Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
44.44Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
44.44Consensusalpha2_offOrthosteric Ligandalpha2c_off
44.44Consensusorexin_offOrthosteric Ligandox2_off ox1_off
44.44Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
44.44Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
44.44Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
44.00Single5WF5UK-4320975WF5-A2A-UK-432097
44.00Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
44.00Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
44.00Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
44.00Consensusangiotensin_onOrthosteric Ligandat1_on
44.00Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
44.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
44.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
44.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
44.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
43.48Single5WF6UK-4320975WF6-A2A-UK-432097
43.48Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
43.48Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
43.48Single7SK9CCX6627SK9-ACKR3-CCX662
43.48Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
43.48Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
43.48Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
43.48Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
43.48Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
42.86Single3P0GBI1671073P0G-β2-BI167107
42.86Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
42.86Single4U15Tiotropium4U15-M3-Tiotropium
42.86Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
42.86Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
42.86Single6OL9Tiotropium6OL9-M5-Tiotropium
42.86Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
42.86Single7FEECP559407FEE-CB1-CP55940-ZCZ011
42.86Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
42.86Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
42.86Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
42.86Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
42.86Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
42.86Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
42.86Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
42.86Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
42.86Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
42.86Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
42.86Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
42.86Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
42.86Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
42.86Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
42.86Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
42.86Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
42.86Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
42.86Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
42.86Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
42.31Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
42.31Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
42.31Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
42.31Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
42.31Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
42.31Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
42.31Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
42.11Single2YDOAdenosine2YDO-A2A-Adenosine
42.11Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
42.11Single4MBSMaraviroc4MBS-CCR5-Maraviroc
42.11Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
42.11Single6PS5S-Propranolol6PS5-β2-S-Propranolol
42.11Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
42.11Single6VI4JDTic6VI4-κ-JDTic
42.11Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
42.11Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
42.11Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
42.11Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
42.11Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
42.11Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
42.11Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
42.11Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
42.11Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
42.11Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
42.11Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
42.11Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
42.11Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
42.11Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
42.11Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
42.11Single8IHKAcifran8IHK-HCA3-Acifran
42.11Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
42.11Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
42.11Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
42.11Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
42.11Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
42.11Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
42.11Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
42.11Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
42.11Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
42.11Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
42.11Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
41.67Single4IARErgotamine4IAR-5-HT1B-Ergotamine
41.67Single4XT1Fractalkine4XT1-US28-Fractalkine
41.67Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
41.67Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
41.67Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
41.67Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
41.67Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
41.67Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
41.67Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
41.18Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
41.18Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
41.18Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
41.18Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
41.18Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
40.91Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
40.91Single5CXVTiotropium5CXV-M1-Tiotropium
40.91Single6CM4Risperidone6CM4-D2-Risperidone
40.91Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
40.91Single6KQICP559406KQI-CB1-CP55940-Org27569
40.91Single6MXTSalmeterol6MXT-β2-Salmeterol
40.91Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
40.91Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
40.91Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
40.91Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
40.91Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
40.91Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
40.91Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.91Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
40.91Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
40.91Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
40.91Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
40.91Single8JWY2-1188JWY-A2A-2-118
40.91Single8JWZAB9288JWZ-A2A-AB928-Na
40.91Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
40.91Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
40.91Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
40.91Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
40.91Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
40.91Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
40.91Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
40.91Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
40.91Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
40.91Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
40.91Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
40.91Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
40.91Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
40.91Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
40.91Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
40.74Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
40.74Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
40.74Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
40.74Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
40.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
40.00Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
40.00Single4QKX35V4QKX-β2-35V
40.00Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
40.00Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
40.00Single5GLHEndothelin-15GLH-ETB-Endothelin-1
40.00Single5TGZAM65385TGZ-CB1-AM6538
40.00Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
40.00Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
40.00Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
40.00Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
40.00Single6H7MSalbutamol6H7M-β1-Salbutamol
40.00Single6HLOAprepitant6HLO-NK1-Aprepitant
40.00Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
40.00Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
40.00Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
40.00Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
40.00Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
40.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
40.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
40.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
40.00Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
40.00Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
40.00Single7V3ZCP559407V3Z-CB1-CP55940
40.00Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
40.00Single7WC7Lisuride7WC7-5-HT2A-Lisuride
40.00Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
40.00Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
40.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
40.00Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
40.00Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
40.00Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
40.00Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
40.00Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
40.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
40.00Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
40.00Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
40.00Single8X63Mepyramine8X63-H1-Mepyramine
40.00Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
40.00Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
40.00Consensus5ht5_onOrthosteric Ligand5ht5a_on
40.00Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
40.00Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
40.00Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
40.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
40.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
40.00Consensusa3_onOrthosteric Liganda3a_on
40.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
40.00Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
40.00Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
40.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
40.00Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
40.00Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
40.00Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
40.00Consensushistamine_offOrthosteric Ligandh1_off
40.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
40.00Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
40.00Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
40.00Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
39.29Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
39.13Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
39.13Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
39.13Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
39.13Single6IBLArformoterol6IBL-β1-Arformoterol
39.13Single6K1QIRL25006K1Q-ETB-IRL2500
39.13Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
39.13Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
39.13Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
39.13Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
39.13Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
39.13Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
39.13Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
39.13Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
39.13Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
39.13Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
39.13Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
39.13Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
39.13Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
39.13Consensuscck_onOrthosteric Ligandccka_on cckb_on
39.13Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
39.13Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
38.89Single3PBLEticlopride3PBL-D3-Eticlopride
38.89Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
38.89Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
38.89Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
38.89Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
38.89Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
38.89Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
38.89Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
38.89Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
38.89Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
38.89Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
38.89Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
38.71Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
38.71Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
38.71Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
38.71Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
38.71Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
38.46Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
38.46Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
38.46Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
38.46Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
38.10Single2Y00Dobutamine2Y00-β1-Dobutamine
38.10Single5N2SPSB365N2S-A1-PSB36
38.10Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
38.10Single5TVNLSD5TVN-5-HT2B-LSD
38.10Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
38.10Single6E67BI1671076E67-β2-BI167107-Gs (fused)
38.10Single6HLPNetupitant6HLP-NK1-Netupitant
38.10Single6LUQHaloperidol6LUQ-D2-Haloperidol
38.10Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
38.10Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
38.10Single7C4SS1P7C4S-S1P3-S1P
38.10Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
38.10Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
38.10Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
38.10Single7W41PD1762527W41-BB2-PD176252
38.10Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
38.10Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
38.10Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
38.10Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.10Single8GNEKW-63568GNE-A2A-KW-6356-Na
38.10Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
38.10Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
38.10Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
38.10Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
38.10Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
38.10Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
38.10Single8ZMFA1L108ZMF-5-HT2C-A1L10
38.10Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
38.10Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
38.10Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
38.10Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
38.10Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
38.10Consensusa3_on_gpOrthosteric Liganda3a_on_gp
38.10Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
38.10Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
38.10Consensusadenosine_offOrthosteric Liganda1_off a2_off
38.10Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
38.10Consensusbombesin_offOrthosteric Ligandbb2_off
38.10Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
38.10Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
38.10Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
38.10Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.10Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.93Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
37.93Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
37.93Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
37.50Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
37.50Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
37.50Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
37.50Single7XN9L-054,5227XN9-SST2-L-054,522
37.50Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
37.50Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
37.50Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
37.50Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
37.50Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
37.04Single6JODAngiotensin II6JOD-AT2-Angiotensin II
37.04Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
37.04Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
37.04Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
36.84Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
36.84Single3ODUIT1t3ODU-CXCR4-IT1t
36.84Single4S0VSuvorexant4S0V-OX2-Suvorexant
36.84Single6AKYMaraviroc6AKY-CCR5-Maraviroc
36.84Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
36.84Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
36.84Single6TPJSuvorexant6TPJ-OX2-Suvorexant
36.84Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
36.84Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
36.84Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
36.84Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
36.84Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
36.84Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
36.84Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
36.84Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
36.84Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
36.84Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
36.84Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
36.84Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
36.84Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
36.84Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
36.84Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
36.84Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
36.84Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
36.84Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
36.84Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
36.84Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
36.84Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
36.84Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
36.84Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
36.84Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
36.84Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
36.84Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
36.84Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
36.84Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
36.84Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
36.84Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
36.84Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
36.84Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
36.67Single8IY6Endothelin-18IY6-ETB-Endothelin-1
36.67Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
36.67Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
36.67Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
36.67Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
36.67Consensusbradykinin_onOrthosteric Ligandbk2_on
36.67Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
36.67Consensusendothelin_onOrthosteric Ligandetb_on eta_on
36.67Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
36.67Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
36.67Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
36.36Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
36.36Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
36.36Single5V54Methiothepin5V54-5-HT1B-Methiothepin
36.36Single5XR8AM8415XR8-CB1-AM841
36.36Single5XRAAM115425XRA-CB1-AM11542
36.36Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
36.36Single6E59L-7607356E59-NK1-L-760735
36.36Single6J20Aprepitant6J20-NK1-Aprepitant
36.36Single6WGTLSD6WGT-5-HT2A-LSD
36.36Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
36.36Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
36.36Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
36.36Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
36.36Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
36.36Single7TUYGSK682753A7TUY-GPR183-GSK682753A
36.36Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
36.36Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
36.36Single8EA0Iperoxo8EA0-M3-Iperoxo
36.36Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
36.36Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
36.36Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
36.36Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
36.36Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
36.36Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
36.36Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
36.36Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.36Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
36.36Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
36.36Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
36.36Consensus5ht1_offOrthosteric Ligand5ht1b_off
36.36Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
36.36Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
36.36Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
36.36Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
36.36Consensuslpa_onOrthosteric Ligandlpa1_on
36.36Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
36.36Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
36.36Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
36.36Consensustachykinin_offOrthosteric Ligandnk1_off
36.00Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
36.00Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
36.00Single7F8XNN90567F8X-CCKA-NN9056
36.00Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
36.00Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
36.00Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
36.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
36.00Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
36.00Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
36.00Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
35.71Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
35.71Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
35.71Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
35.71Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
35.71Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.71Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
35.71Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
35.71Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
35.71Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
35.48Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
35.48Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
35.29Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
35.29Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.29Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
35.29Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
35.29Single9CHUNoradrenaline9CHU-β2-Noradrenaline
35.29Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
35.29Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
35.00Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
35.00Single3RZECidoxepin3RZE-H1-Cidoxepin
35.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
35.00Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
35.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
35.00Single5JTBZM-2413855JTB-A2A-ZM-241385
35.00Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
35.00Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
35.00Single6A94Zotepine6A94-5-HT2A-Zotepine
35.00Single6AQFZM-2413856AQF-A2A-ZM-241385
35.00Single6KUXRS-799486KUX-α2a-RS-79948
35.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
35.00Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
35.00Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
35.00Single6TP3Nemorexant6TP3-OX1-Nemorexant
35.00Single6V9SGTPL114036V9S-OX1-GTPL11403
35.00Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
35.00Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
35.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
35.00Single7T32ZM-2413857T32-A2A-ZM-241385
35.00Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
35.00Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
35.00Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
35.00Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
35.00Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
35.00Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
35.00Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
35.00Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
35.00Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
35.00Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
35.00Single8K5CAcipimox8K5C-HCA2-Acipimox
35.00Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
35.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
35.00Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
35.00Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
35.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
35.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.00Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
35.00Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
35.00Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
35.00Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
35.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
35.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
35.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
35.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
35.00Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
35.00Consensusa2_offOrthosteric Liganda2a_off
35.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
35.00Consensushca_onOrthosteric Ligandhca2_on
35.00Consensusopsins_offOrthosteric Ligandrhodopsin_off
35.00Consensussensory_offOrthosteric Ligandopsins_off
34.78Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
34.78Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
34.78Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
34.78Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
34.78Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
34.78Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
34.78Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
34.78Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
34.78Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.78Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
34.78Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
34.78Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
34.78Single8XYIVUF106618XYI-CXCR3-VUF10661
34.78Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
34.78Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.78Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.62Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
34.62Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
34.62Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
34.62Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
34.62Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
34.62Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
34.62Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
34.48Single4XT3Fractalkine4XT3-US28-Fractalkine
34.48Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.48Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
34.48Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
34.48Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
34.48Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
34.48Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
34.48Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
34.29Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
34.29Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
33.33Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
33.33Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
33.33Single2Y01Dobutamine2Y01-β1-Dobutamine
33.33Single2Y02Carmoterol2Y02-β1-Carmoterol
33.33Single3EMLZM-2413853EML-A2A-ZM-241385
33.33Single3OE6IT1t3OE6-CXCR4-IT1t
33.33Single4DAJTiotropium4DAJ-M3-Tiotropium
33.33Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
33.33Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
33.33Single4MQSIperoxo4MQS-M2-Iperoxo
33.33Single4U14Tiotropium4U14-M3-Tiotropium
33.33Single5DSGTiotropium5DSG-M4-Tiotropium
33.33Single5IU8Q274563475IU8-A2A-Q27456347-Na
33.33Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
33.33Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
33.33Single5UIGCmpd-15UIG-A2A-Cmpd-1
33.33Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
33.33Single6DRXLisuride6DRX-5-HT2B-Lisuride
33.33Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
33.33Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
33.33Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
33.33Single6S0LZM-2413856S0L-A2A-ZM-241385
33.33Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
33.33Single7BU7BI1671077BU7-β1-BI167107
33.33Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
33.33Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
33.33Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
33.33Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
33.33Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
33.33Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
33.33Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
33.33Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
33.33Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
33.33Single7PYRPSB-21157PYR-A2A-PSB-2115
33.33Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
33.33Single7UM4AS26747237UM4-5-HT5A-AS2674723
33.33Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
33.33Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
33.33Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
33.33Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
33.33Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
33.33Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
33.33Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
33.33Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
33.33Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
33.33Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
33.33Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
33.33Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
33.33Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
33.33Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
33.33Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
33.33Single8K5DGSK2560738K5D-HCA2-GSK256073
33.33Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
33.33Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
33.33Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
33.33Single8XVJMacitentan8XVJ-ETA-Macitentan
33.33Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
33.33Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
33.33Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
33.33Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
33.33Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
33.33Consensus5ht2_onOrthosteric Ligand5ht2b_on
33.33Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
33.33Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusblt_onOrthosteric Ligandblt1_on
33.33Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
33.33Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
33.33Consensuscck_offOrthosteric Ligandccka_off
33.33Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
33.33Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
33.33Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
33.33Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
33.33Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
33.33Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
33.33Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
33.33Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
33.33Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
33.33Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
33.33Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
33.33Consensushca_on_gpOrthosteric Ligandhca2_on_gp
33.33Consensusleukotriene_onOrthosteric Ligandblt_on
33.33Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
33.33Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
33.33Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
33.33Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
33.33Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
33.33Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
33.33Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
33.33Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
33.33Consensusprostanoid_offOrthosteric Ligandep_off dp_off
32.26Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
32.26Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
32.14Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
32.14Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
32.14Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.14Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.14Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
32.14Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
32.14Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
32.14Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
32.14Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
32.14Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
32.14Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
32.14Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
32.14Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.14Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
32.14Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.14Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.14Consensusvasop-oxy_onOrthosteric Ligandv2_on
32.14Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
32.00Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
32.00Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
32.00Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
32.00Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
32.00Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
32.00Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
32.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
32.00Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
32.00Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
31.82Single5IUAQ274563485IUA-A2A-Q27456348-Na
31.82Single5N2RPSB-365N2R-A2A-PSB-36-Na
31.82Single6D26Fevipiprant6D26-DP2-Fevipiprant
31.82Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
31.82Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
31.82Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
31.82Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
31.82Single6S0QZM-2413856S0Q-A2A-ZM-241385
31.82Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
31.82Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
31.82Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
31.82Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
31.82Single7SINNPS-21437SIN-CaS-NPS-2143
31.82Single7SINNPS-21437SIN-CaS-NPS-2143
31.82Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
31.82Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
31.82Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
31.82Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
31.82Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
31.82Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
31.82Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
31.82Single8QOTNanobody-E8QOT-μ-Nanobody-E
31.82Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
31.82Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
31.82Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
31.82Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
31.82Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
31.82Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
31.82Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
31.82Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
31.82Consensusdp_offOrthosteric Liganddp2_off
31.82Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
31.82Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
31.82Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
31.82Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
31.82Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
31.82Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
31.82Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
31.82Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
31.58Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
31.58Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
31.58Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
31.58Single3OE9IT1t3OE9-CXCR4-IT1t
31.58Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
31.58Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
31.58Single6TP4ACT-4622066TP4-OX1-ACT-462206
31.58Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
31.58Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
31.58Single7SRQLSD7SRQ-5-HT2B-LSD
31.58Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
31.58Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.58Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
31.58Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
31.58Single8K5BNiacin8K5B-HCA2-Niacin
31.58Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
31.58Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
31.58Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
31.58Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
31.58Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
31.58Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
31.58Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
31.58Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
31.58Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
31.58Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
31.25Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
31.25Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
31.25Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
31.03Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
31.03Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
31.03Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
31.03Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
31.03Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
31.03Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
31.03Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
31.03Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
31.03Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
31.03Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
31.03Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
31.03Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
31.03Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
30.77Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
30.77Single7QA8Peptide7QA8-STE2-Peptide
30.77Single7QA8Peptide7QA8-STE2-Peptide
30.77Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
30.77Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
30.77Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
30.77Single8WKYPG-9348WKY-MC4-PG-934
30.77Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
30.77Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
30.77Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
30.77Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
30.77Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.77Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.77Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
30.77Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
30.77Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
30.77Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
30.77Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
30.43Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
30.43Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
30.43Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
30.43Single7B6WCyclazosin7B6W-α1b-Cyclazosin
30.43Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
30.43Single7PX4PSB-21137PX4-A2A-PSB-2113
30.43Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
30.43Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
30.43Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
30.43Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
30.43Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
30.43Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
30.43Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
30.43Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
30.43Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
30.43Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
30.43Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
30.43Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
30.43Consensusrelaxin_onOrthosteric Ligandrxfp4_on
30.43Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
30.00Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
30.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
30.00Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
30.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
30.00Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
30.00Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
30.00Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
30.00Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
30.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
30.00Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
30.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
30.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
30.00Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
30.00Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
30.00Single7BR3Elagolix7BR3-GnRH1-Elagolix
30.00Single7F8ULintitript7F8U-CCKA-Lintitript
30.00Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
30.00Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
30.00Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
30.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
30.00Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
30.00Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
30.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
30.00Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
30.00Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
30.00Single8IWESpermidine8IWE-TA9-Spermidine
30.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
30.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
30.00Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
30.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
30.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
30.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
30.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
30.00Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
30.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
30.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
30.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
30.00Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
30.00Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
30.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
30.00Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
30.00Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
30.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
30.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
29.63Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
29.63Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
29.63Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
29.63Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
29.63Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
29.63Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
29.41Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
29.41Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
29.27Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
29.17Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
29.17Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
29.17Single7K15MKD0467K15-BLT1-MKD046-Na
29.17Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
29.17Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
29.17Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
29.17Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
29.17Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
29.17Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
29.17Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
29.17Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
29.17Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
29.17Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
29.17Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
29.17Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
29.03Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
29.03Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
28.57Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
28.57Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
28.57Single5IUBQ274563445IUB-A2A-Q27456344-Na
28.57Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
28.57Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
28.57Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
28.57Single5UVIZM-2413855UVI-A2A-ZM-241385
28.57Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
28.57Single6MH8ZM-2413856MH8-A2A-ZM-241385
28.57Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
28.57Single6TPKRetosiban6TPK-OT-Retosiban
28.57Single6W25SHU91196W25-MC4-SHU9119-Ca
28.57Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
28.57Single7AROLUF58337ARO-A2A-LUF5833-Na
28.57Single7UL3Famotidine7UL3-H2-Famotidine
28.57Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
28.57Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
28.57Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
28.57Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
28.57Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
28.57Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
28.57Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
28.57Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
28.57Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
28.57Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
28.57Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
28.57Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
28.57Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
28.57Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
28.57Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
28.57Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
28.57Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
28.57Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
28.57Consensusgrh_offOrthosteric Ligandgnrh1_off
28.57Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
28.57Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
28.57Consensusvasop-oxy_offOrthosteric Ligandot_off
28.12Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
28.12Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
28.00Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
28.00Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
28.00Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
28.00Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.00Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
28.00Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
28.00Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
28.00Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
28.00Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single3OE8IT1t3OE8-CXCR4-IT1t
27.78Single6TQ9SB-4081246TQ9-OX1-SB-408124
27.78Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
27.78Single8A2OTheophylline8A2O-A2A-Theophylline-Na
27.78Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
27.78Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
27.78Consensussensory_onOrthosteric Ligandopsins_on
27.59Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
27.59Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
27.59Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
27.59Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
27.59Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
27.59Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.59Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
27.59Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
27.59Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
27.59Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
27.59Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
27.59Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
27.27Single4YAYZD-71554YAY-AT1-ZD-7155
27.27Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
27.27Single5UENDU1725UEN-A1-DU172
27.27Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
27.27Single6D27CAY104716D27-DP2-CAY10471
27.27Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
27.27Single6GPSMK08126GPS-CCR2-MK0812
27.27Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
27.27Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
27.27Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
27.27Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
27.27Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
27.27Single7F83PF-051904577F83-Ghrelin-PF-05190457
27.27Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
27.27Single7YXAONO-54306087YXA-S1P5-ONO-5430608
27.27Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
27.27Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
27.27Single8RLNLUF58348RLN-A2A-LUF5834
27.27Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
27.27Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
27.27Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
27.27Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
27.27Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
27.27Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
27.27Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
27.27Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
26.92Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
26.92Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
26.92Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
26.92Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
26.92Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
26.92Consensuskisspeptin_onOrthosteric Ligandkiss1_on
26.92Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
26.67Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
26.67Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
26.67Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
26.67Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
26.67Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
26.47Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
26.47Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
26.47Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
26.32Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
26.32Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
26.32Single3UZAGTPL92363UZA-A2A-GTPL9236
26.32Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
26.32Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
26.32Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
26.32Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
26.32Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
26.32Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.32Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
26.32Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
26.32Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
26.32Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
26.32Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
26.32Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
26.32Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
26.32Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
26.32Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
26.32Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
26.32Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
26.32Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
26.32Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
26.09Single5CGCHTL142425CGC-mGlu5-HTL14242
26.09Single6GPXMK08126GPX-CCR2-MK0812
26.09Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
26.09Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
26.09Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
26.09Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
26.09Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
26.09Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
26.09Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
26.09Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
26.09Consensusblt_offOrthosteric Ligandblt1_off
26.09Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
26.09Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.93Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single8IEBA1LYA8IEB-GPR156-A1LYA
25.93Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
25.93Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
25.93Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
25.93Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
25.93Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Single7SK3CXCL127SK3-ACKR3-CXCL12
25.81Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
25.81Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
25.81Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
25.81Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
25.00Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
25.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
25.00Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
25.00Single6HLLCP999946HLL-NK1-CP99994
25.00Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
25.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
25.00Single6OS1TRV0266OS1-AT1-TRV026
25.00Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
25.00Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
25.00Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
25.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
25.00Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
25.00Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
25.00Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7R0CAVP7R0C-V2-AVP-Arrestin2
25.00Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
25.00Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
25.00Single7SK5CXCL127SK5-ACKR3-CXCL12
25.00Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
25.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
25.00Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
25.00Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
25.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
25.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
25.00Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
25.00Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
25.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
25.00Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
25.00Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
25.00Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
25.00Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
25.00Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
25.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
25.00Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
25.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
25.00Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
25.00Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
25.00Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
25.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
25.00Single9B9Y7DY9B9Y-CB1-7DY
25.00Single9BJKNAM9BJK-μ-Naloxone-NAM
25.00Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
25.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
25.00Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
25.00Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
25.00Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
25.00Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
25.00Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
24.24Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
24.24Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
24.24Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
24.24Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
24.24Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
24.24Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
24.24Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
24.14Single3OE0CVX153OE0-CXCR4-CVX15
24.14Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.14Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
24.14Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
24.14Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
24.14Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
24.00Single4N4WSANT-14N4W-SMO-SANT-1
24.00Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
24.00Single4PY02MeSATP4PY0-P2Y12-2MeSATP
24.00Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
24.00Single5X33BIIL2605X33-BLT1-BIIL260
24.00Single6OS2TRV0266OS2-AT1-TRV026
24.00Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
24.00Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
24.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
24.00Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
24.00Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single3PWHZM-2413853PWH-A2A-ZM-241385
23.81Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
23.81Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
23.81Single6DS0Ly2660976DS0-5-HT2B-Ly266097
23.81Single7F8YDevazepide7F8Y-CCKA-Devazepide
23.81Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
23.81Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
23.81Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
23.81Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
23.81Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
23.81Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
23.81Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
23.81Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
23.81Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
23.81Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
23.81Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
23.81Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
23.81Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
23.81Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
23.81Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
23.81Consensusangiotensin_offOrthosteric Ligandat1_off
23.53Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
23.53Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
23.53Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
23.53Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
23.33Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
23.33Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
23.33Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
23.33Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
23.33Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
23.33Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
23.33Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
23.08Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
23.08Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
23.08Single5CGDHTL142425CGD-mGlu5-HTL14242
23.08Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
23.08Consensuschemerin_onOrthosteric Ligandcml1_on
23.08Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
23.08Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
23.08Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
22.86Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
22.86Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
22.73Single3REYXAC3REY-A2A-XAC
22.73Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
22.73Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
22.73Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
22.73Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
22.73Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
22.73Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
22.73Single7VODCariprazine7VOD-5-HT2A-Cariprazine
22.73Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
22.73Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
22.73Single8K2WAMG4878K2W-CXCR3-AMG487
22.73Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.73Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
22.73Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
22.73Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
22.73Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
22.73Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
22.73Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
22.58Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
22.58Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
22.58Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
22.58Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
22.22Single5EE7MK08935EE7-Glucagon-MK0893
22.22Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
22.22Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
22.22Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
22.22Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
22.22Single8IEIA1LYA8IEI-GPR156-A1LYA
22.22Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8PWNTheophylline8PWN-A2A-Theophylline
22.22Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
22.22Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.88Single6FJ3PTH6FJ3-PTH1-PTH
21.88Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
21.88Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
21.88Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
21.88Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
21.74Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
21.74Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
21.74Single6IIVDaltroban6IIV-TP-Daltroban
21.74Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
21.74Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
21.74Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
21.74Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
21.74Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
21.74Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
21.74Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
21.74Single9IYAONO-97105319IYA-GPR55-ONO-9710531
21.74Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
21.74Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
21.74Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
21.43Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
21.43Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
21.43Single8IEIA1LYA8IEI-GPR156-A1LYA
21.43Single8IEPA1LYA8IEP-GPR156-A1LYA
21.43Single8IEPA1LYA8IEP-GPR156-A1LYA
21.43Single8KIGSHU91198KIG-MC3-SHU9119-Ca
21.21Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
21.21Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
21.21Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
21.21Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
21.21Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
21.21Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
21.21Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
21.21Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
21.05Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
21.05Single3RFMCaffeine3RFM-A2A-Caffeine
21.05Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
21.05Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
21.05Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
20.83Single4NTJAZD12834NTJ-P2Y12-AZD1283
20.83Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
20.83Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
20.83Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
20.83Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
20.83Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
20.83Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
20.83Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
20.83Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
20.83Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
20.83Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
20.83Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
20.83Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
20.83Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
20.83Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
20.83Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
20.83Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
20.83Consensusep_offOrthosteric Ligandep4_off
20.69Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
20.69Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
20.69Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.69Single8IEBA1LYA8IEB-GPR156-A1LYA
20.69Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
20.69Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
20.59Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
20.59Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
20.59Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
20.59Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
20.59Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
20.59Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
20.59Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
20.00Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
20.00Single4BV0Neurotensin4BV0-NTS1-Neurotensin
20.00Single5TZRMK86665TZR-FFA1-MK8666
20.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
20.00Single6ME5Agomelatine6ME5-MT1-Agomelatine
20.00Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
20.00Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
20.00Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
20.00Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
20.00Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
20.00Single7P2L4YI7P2L-mGlu5-4YI
20.00Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
20.00Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
20.00Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7WC5Psilocin7WC5-5-HT2A-Psilocin
20.00Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
20.00Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
20.00Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
20.00Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
20.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
20.00Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
20.00Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
20.00Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
20.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
20.00Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
20.00Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
20.00Consensusgi_sensoryOrthosteric Ligandgi_opsins
20.00Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
20.00Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
20.00Consensusneurotensin_onOrthosteric Ligandnts1_on
20.00Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
20.00Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.00Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
20.00Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
20.00Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
19.51Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
19.44Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
19.44Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
19.35Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
19.35Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
19.35Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
19.23Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
19.23Single4XEENeurotensin4XEE-NTS1-Neurotensin
19.23Single4XESNeurotensin4XES-NTS1-Neurotensin
19.23Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
19.23Single6IIURamatroban6IIU-TP-Ramatroban
19.23Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
19.23Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
19.23Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
19.23Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
19.23Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
19.23Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
19.23Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
19.23Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
19.23Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
19.23Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
19.23Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
19.23Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
19.23Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
19.23Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
19.23Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
19.23Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
19.23Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
19.05Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
19.05Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
19.05Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
19.05Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
19.05Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
19.05Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
19.05Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
18.92Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
18.92Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
18.92Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
18.75Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
18.52Single4BUONeurotensin4BUO-NTS1-Neurotensin
18.52Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
18.52Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
18.52Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
18.52Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
18.52Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
18.52Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
18.52Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
18.52Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
18.52Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.42Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
18.18Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
18.18Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
18.18Single5U09Taranabant5U09-CB1-Taranabant
18.18Single5ZKQABT-4915ZKQ-PAF-ABT-491
18.18Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
18.18Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
18.18Single6ME9Ramelteon6ME9-MT2-Ramelteon
18.18Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
18.18Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
18.18Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
18.18Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
18.18Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
18.18Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
18.18Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
18.18Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
18.18Single9BA0A1AKN9BA0-CB1-A1AKN
18.18Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
18.18Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
18.18Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
17.95Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.86Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
17.86Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
17.86Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
17.86Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
17.86Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
17.86Single8XQJJN2418XQJ-Apelin-JN241
17.86Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
17.86Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
17.86Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
17.86Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
17.65Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
17.65Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
17.65Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
17.65Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
17.39Single6FFIMMPEP6FFI-mGlu5-MMPEP
17.39Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
17.39Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
17.39Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
17.39Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
17.39Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
17.39Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
17.24Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
17.24Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
17.24Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
17.24Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.14Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
16.67Single4QIMANTA XV4QIM-SMO-ANTA XV
16.67Single5MZPCaffeine5MZP-A2A-Caffeine-Na
16.67Single6FFHFenobam6FFH-mGlu5-Fenobam
16.67Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
16.67Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
16.67Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
16.67Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
16.67Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
16.67Single7XNACYN1548067XNA-SST2-CYN154806
16.67Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
16.67Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
16.67Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.67Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
16.67Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
16.67Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
16.67Single9B9ZA1AKO9B9Z-CB1-A1AKO
16.67Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
16.67Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
16.22Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
16.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
16.00Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
16.00Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.00Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
16.00Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
15.79Single7WC4Serotonin7WC4-5-HT2A-Serotonin
15.79Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
15.79Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
15.62Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
15.62Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
15.38Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
15.38Single5V56TC1145V56-SMO-TC114
15.38Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
15.38Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
15.38Single7F1TMIP-1a7F1T-CCR5-MIP-1a
15.38Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
15.38Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
15.38Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
15.38Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
15.38Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
15.15Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
15.15Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
15.15Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
15.00Consensusp2y_offOrthosteric Ligandp2y1_off
14.81Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
14.81Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
14.81Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
14.81Single6YVRNTS8-136YVR-NTS1-NTS8-13
14.81Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
14.81Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
14.81Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
14.81Single8XQJJN2418XQJ-Apelin-JN241
14.81Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
14.71Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
14.71Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
14.71Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
14.29Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
14.29Single4XNWMRS25004XNW-P2Y1-MRS2500
14.29Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
14.29Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
14.29Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
14.29Single7V6A-7V6A-M4-PubChem 9864275-Gi1/β1/γ2
14.29Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
14.29Single8XVUCXCL28XVU-CXCR2-CXCL2
14.29Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
14.29Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
14.29Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
13.89Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
13.79Single6KNMJN241-96KNM-Apelin-JN241-9
13.79Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
13.79Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
13.79Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
13.79Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single5L7IVismodegib5L7I-SMO-Vismodegib
13.64Single6LI0C176LI0-GPR52-C17
13.64Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
13.64Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
13.64Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.64Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
13.64Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Consensusgq_nucleotideOrthosteric Ligandgq_p2y
13.64Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
13.33Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
13.33Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
13.33Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8XWNCXCL88XWN-CXCR2-CXCL8
13.33Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
13.33Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
13.33Consensussomatostatin_offOrthosteric Ligandsst2_off
13.04Single4BWBNeurotensin4BWB-NTS1-Neurotensin
13.04Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
13.04Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
13.04Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
13.04Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
13.04Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
13.04Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
13.04Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
13.04Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
12.90Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
12.50Single6ZINSR486926ZIN-NTS1-SR48692
12.50Single7VV6C48/807VV6-MRGPRX2-C48/80
12.50Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
12.50Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
12.00Single5T04Neurotensin5T04-NTS1-Neurotensin
12.00Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
12.00Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
12.00Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
11.76Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
11.54Single4JKVTaladegib4JKV-SMO-Taladegib
11.54Single6Z4SSR486926Z4S-NTS1-SR48692
11.54Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
11.54Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
11.54Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
11.11Single5V57TC1145V57-SMO-TC114
11.11Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
11.11Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
11.11Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
11.11Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
10.71Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8XWACXCL18XWA-CXCR2-CXCL1
10.71Single8XWMCXCL68XWM-CXCR2-CXCL6
10.71Single8XWSCXCL58XWS-CXCR2-CXCL5
10.71Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
10.53Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
10.34Single8XWFCXCL38XWF-CXCR2-CXCL3
10.34Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
10.00Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
10.00Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
10.00Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
9.68Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
9.68Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
9.52Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
9.52Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
9.52Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
9.09Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
9.09Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
9.09Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
9.09Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
9.09Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
8.82Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
8.70Single4O9RCyclopamine4O9R-SMO-Cyclopamine
8.70Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.70Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
8.33Single4QINSAG1.54QIN-SMO-SAG1.5
8.33Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
8.33Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
8.33Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
8.33Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
8.33Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
8.00Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
8.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
8.00Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
8.00Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
7.69Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
7.69Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
7.41Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
7.41Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
7.41Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
7.41Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
7.41Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
7.14Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
6.06Single7SHEPI; PE7SHE-GPR158-PI; PE
5.88Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.88Single6D35Cholesterol6D35-SMO-Cholesterol
5.88Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.88Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.88Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
5.88Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
5.88Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
5.88Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
5.88Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
5.88Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
5.88Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
5.88Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
5.88Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.88Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.88Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.88Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.88Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
5.88Single7DTTCa7DTT-CaS-Ca-Ca
5.88Single7DTTCa7DTT-CaS-Ca-Ca
5.88Single7DTUTryptophan7DTU-CaS-Tryptophan
5.88Single7DTUTryptophan7DTU-CaS-Tryptophan
5.88Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.88Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.88Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.88Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.88Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.88Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.88Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.88Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.88Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
5.88Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.88Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.88Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.88Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.88Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.88Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.88Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
5.88Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
5.88Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.88Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.88Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.88Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.88Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.88Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.88Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.88Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.88Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.88Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.88Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.88Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.88Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.88Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.88Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.88Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.88Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.88Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.88Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
5.88Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.88Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.88Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.88Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.88Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.88Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.88Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
5.88Single7XW7K1-707XW7-TSH-K1-70
5.88Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.88Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.88Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.88Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.88Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.88Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.88Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.88Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.88Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.88Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.88Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.88Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.88Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
5.88Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.88Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.88Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.88Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.88Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
5.88Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
5.88Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.88Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.88Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
5.88Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
5.88Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
5.88Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
5.88Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.88Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.88Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.88Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
5.88Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
5.88Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
5.88Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
5.88Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.88Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.88Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.88Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.88Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.88Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.88Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.88Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.88Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.88Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.88Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.88Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.88Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.88Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.88Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.88Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.88Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.88Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.88Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
5.88Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
5.88Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
5.88Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
5.88Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
5.88Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
5.88Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.88Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.88Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8WVXNorrin8WVX-LGR4-Norrin
5.88Single8WVYNorrin8WVY-LGR4-Norrin
5.88Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.88Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.88Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.88Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.88Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.88Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.88Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
5.88Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.88Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.88Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.88Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.88Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.88Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.88Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.88Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.88Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.88Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.88Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.88Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.88Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.88Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.88Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.88Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.88Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.88Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.88Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.88Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.56Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.56Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.56Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.56Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.56Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.56Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.56Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.56Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.56Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.56Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.56Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
5.26Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
5.26Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
5.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
5.00Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
5.00Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
5.00Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
5.00Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
5.00Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
4.76Single5L7DCholesterol5L7D-SMO-Cholesterol
4.76Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.76Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
4.76Single8HS2Fab0468HS2-GPR20-Fab046
4.76Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
4.76Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.76Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
4.55Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
4.35Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
4.35Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
4.35Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
4.35Single8JPSCCL78JPS-ACKR1-CCL7
4.17Single7UL2SR486927UL2-NTS1-SR48692-Na
4.17Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
4.17Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.17Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
4.17Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.17Consensusneurotensin_offOrthosteric Ligandnts1_off
4.17Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
4.00Single4K5YCP-3763954K5Y-CRF1-CP-376395
3.85Single8IYXYL-3658IYX-GPR34-YL-365
3.85Single8JD6N-(3-chlorophenyl)pyridine-2-carboxamide8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
3.70Single4Z9GCP-3763954Z9G-CRF1-CP-376395
3.70Single8GTIBMK-C2058GTI-CRF1-BMK-C205
3.57Single8GTGBMK-I1528GTG-CRF1-BMK-I152
3.57Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
3.45Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
3.33Single7SHEPI; PE7SHE-GPR158-PI; PE
3.33Single8GTMBMK-C2038GTM-CRF1-BMK-C203
3.23Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
3.03Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
3.03Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.94Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
2.86Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.86Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.78Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.56Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
8F7R 8F7R-μ-Endomorphin-Gi1/β1/γ2
8EF5 8EF5-μ-Fentanyl-Gi1/β1/γ2
7SCG 7SCG-μ-FH210-Gi1/β1/γ2
7T2H 7T2H-μ-Lofentanil-Gi1/β1/γ2
7T2G 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
8DZP 8DZP-κ-momSalB-Gi1/β1/γ2
8EF6 8EF6-μ-Morphine-Gi1/β1/γ2
8F7X 8F7X-NOP-Nociceptin-Gi1/β1/γ2
8EFB 8EFB-μ-Oliceridine-Gi1/β1/γ2
7U2L 7U2L-μ-PubChem 163201242-Gi1/β1/γ2
8EFO 8EFO-μ-PZM21-Gi1/β1/γ2
8EFL 8EFL-μ-SR17018-Gi1/β1/γ2
8F7Q 8F7Q-μ-β-Endorphin-Gi1/β1/γ2
7U2K 7U2K-μ-C6-guano-Gi1/β1/γ2
8EFQ 8EFQ-μ-Damgo-Gi1/β1/γ2
8F7S 8F7S-δ-Deltorphin-Gi1/β1/γ2
8F7W 8F7W-κ-Dynorphin-Gi1/β1/γ2
Net Summary
Imin 2.64176
Number of Linked Nodes 889
Number of Links 1105
Number of Hubs 182
Number of Links mediated by Hubs 708
Number of Communities 23
Number of Nodes involved in Communities 252
Number of Links involved in Communities 380
Path Summary
Number Of Nodes in MetaPath 117
Number Of Links MetaPath 116
Number of Shortest Paths 963922
Length Of Smallest Path 3
Average Path Length 23.8133
Length of Longest Path 49
Minimum Path Strength 0.289706
Average Path Strength 5.13547
Maximum Path Strength 20.8097
Minimum Path Correlation 0.701176
Average Path Correlation 0.974063
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.32558
Average % Of Corr. Nodes 48.3587
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 56.8467
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
gi_peptidegi_cck
gi_apelin
gi_compl-pept
gi_endothelin
gi_formylpeptide
gi_galanin
gi_ghrelin
gi_npy
gi_neurotensin
gi_opioid
gi_orexin
gi_relaxin
gi_somatostatin



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download gi_opioid.zip



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