Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.33 1.0715604
2G.S1.06 4.50238468
3G.s1h1.04 2.86411409
4G.H1.01 2.78548569
5G.S2.02 1.34508405
6G.S2.04 2.26299407
7G.S2.08 3.82162436
8G.S3.03 5.15352608
9G.S3.04 8.281444127
10G.S3.06 8.666814127
11G.H2.06 5.1317519
12G.H2.07 4.36243719
13G.h2s4.01 8.49626409
14G.S4.03 3.43118467
15G.S4.04 4.51892409
16G.s4h3.04 2.93576408
17G.s4h3.14 0.278912406
18G.H3.01 2.08476709
19G.H3.09 5.076946169
20G.H3.13 6.964015166
21G.H3.17 7.13115515
22G.H3.18 4.8642419
23G.S5.05 4.41847669
24G.hgh4.05 6.18552606
25G.hgh4.20 3.05912503
26G.hgh4.21 3.77785404
27G.H4.03 2.48284404
28G.H4.08 5.50587483
29G.H4.10 9.14116407
30G.H4.12 5.67497484
31G.H4.15 7.19239408
32G.h4s6.12 3.03551402
33G.h4s6.20 4.64047434
34G.S6.02 7.6824408
35G.S6.05 6.56946585
36G.s6h5.01 4.83161469
37G.s6h5.05 2.83133569
38G.H5.03 4.12572569
39G.H5.08 6.24402438
40G.H5.17 5.03759535
41G.H5.20 3.35057408
42G.H5.22 1.70559404
43b.1x4 1.47507408
44b.lh12x2 4.14057408
45b.h2x1 4.13107405
46b.lhb1x6 3.974275133
47b.l1x3 8.90435549
48b.l1x6 9.14515519
49b.b2x1 5.45314518
50b.b2x5 6.23421647
51b.b3x3 3.64309408
52b.l3x2 6.46615409
53b.b4x3 3.73794147
54b.b4x6 9.03045649
55b.b5x2 6.30127407
56b.b5x3 6.13518649
57b.b5x5 4.90708405
58b.b5x7 4.89541407
59b.l5x1 3.751785148
60b.l5x5 9.46812509
61b.b6x1 3.90489419
62b.b6x5 3.73473506
63b.b7x1 5.19925504
64b.b8x4 5.424745146
65b.l8x5 2.20756403
66b.l9x3 6.45289619
67b.l9x6 5.06195718
68b.b10x5 4.70366509
69b.b11x4 5.10235419
70b.l11x2 6.91096519
71b.b12x6 8.53209618
72b.b13x7 7.54842557
73b.l13x3 7.32361659
74b.l13x6 5.14383519
75b.l13x7 4.49972459
76b.b14x3 4.06042455
77b.b15x1 6.75089559
78b.l15x2 5.69206459
79b.b16x4 9.91932456
80b.b16x6 7.5743758
81b.b17x5 6.93448417
82b.b17x7 7.99806418
83b.l17x3 8.70133619
84b.l17x6 6.35505519
85b.b18x3 5.23392418
86b.l18x1 6.40157116
87b.l18x3 7.887914115
88b.b19x2 6.42881616
89b.b19x4 6.09579418
90b.l19x2 6.84297519
91b.b20x4 10.47518
92b.b20x6 6.22196616
93b.b21x1 6.50065517
94b.b21x5 5.14957404
95b.b21x7 5.43358605
96b.l21x2 5.39408404
97b.b22x5 5.250385117
98b.l22x5 6.93215139
99b.b23x6 7.104616157
100b.l23x1 6.38525416
101b.b24x4 7.430964156
102b.b24x6 6.573764158
103b.b25x3 4.691875155
104b.l25x3 8.73005579
105b.l25x4 3.31063405
106b.l25x6 11.4781518
107b.l27x1 10.1293719
108b.l27x2 7.72375479
109b.b28x3 4.1656407
110b.b28x4 6.33243576
111b.b28x6 8.60322579
112g.h1x5 1.43828506
113g.l1x4 3.55239508
114g.h2x11 8.506034116
115g.ctx3 6.01977509
116g.ctx6 3.19185136
117g.ctx14 5.27406499
118g.ctx15 6.51685499
119g.ctx16 4.93134898
120Lig 9.031452120
121NT 27.18712025
1221x43 4.80603407
1231x50 3.715409
1241x60 3.71473507
125I1x50 2.28996509
1262x38 3.8191437
1272x39 5.30745509
1282x40 3.97305409
1292x50 5.82031408
1302x57 4.4951427
131E1 5.156251023
1323x32 4.26905426
1333x34 4.197246109
1343x36 4.65124426
1353x42 9.371745109
1363x44 3.48267408
1373x46 7.33694409
1383x49 4.84702508
1393x53 5.29019408
140I2 5.272481637
1414x50 6.486194109
1424x53 3.639165109
1434x60 4.13378428
144E2 7.386921625
145E2x51 5.42875728
146E2x52 3.84483425
1475x40 1.44237404
1485x58 4.65557409
1495x68 3.40053539
1506x47 4.66562428
1516x48 7.77097628
152E3 2.73815724
1537x33 3.41603427
1547x37 4.86913628
1557x45 4.92477429
1567x50 4.02344408
1577x52 3.08414408
1587x53 5.7197408
1598x58 1.10348405
160H.hahb.04 0.0177135400
161H.HB.05 0.0347313500
162H.hbhc.04 0.040401600
163H.HC.06 0.0395495400
164H.hchd.01 0.0192458500
165H.hdhe.01 0.0224792500
166H.HE.04 0.0493385400
167H.HE.05 0.0256646500
168G.hfs2.03 0.0242214400
169I3 2.74881530
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1G.HN.36 b.b5x2 13.13235.36579NoYes047
2G.HN.40 b.b5x2 25.13187.73719NoYes077
3G.HN.40 b.b5x3 25.15144.19306NoYes479
4b.b4x4 b.b5x3 12.78934.10028NoYes489
5b.b4x4 b.l1x3 12.836211.2192NoYes489
6b.b3x6 b.l1x3 90.392711.8323NoYes099
7b.b3x6 b.l3x2 90.34438.04758NoYes099
8b.b4x6 b.b5x3 13.275411.3743YesYes499
9b.b4x6 b.l1x3 77.34213.45015YesYes499
10b.l1x4 b.l3x2 89.91398.47664NoYes069
11G.HN.51 b.l1x4 89.76986.10333NoNo046
12G.HN.51 G.hns1.02 89.67384.16495NoNo044
13G.HN.36 b.b4x7 13.09793.21233NoNo048
14b.b4x7 b.l2x5 26.048314.9909NoNo085
15b.l2x5 b.l4x2 22.385119.156NoNo054
16b.l4x2 g.ctx15 10.812411.9389NoYes949
17b.l26x5 g.ctx15 13.34.97911NoYes059
18b.l26x5 g.ctx4 65.00874.76637NoNo057
19g.ctx3 g.ctx4 65.03874.72099YesNo097
20g.ctx3 g.ctx6 99.71965.78357YesYes096
21b.l22x5 g.ctx6 99.18524.69523YesYes1396
22b.l22x5 b.l24x2 99.57447.7131YesNo096
23b.h2x5 b.l24x2 99.58874.43862NoNo056
24b.h2x1 b.h2x5 99.59573.76285YesNo055
25b.b21x5 b.h2x1 99.2956.81112YesYes045
26b.b21x5 b.b21x7 99.32588.55578YesYes045
27b.b21x7 b.b24x6 99.62368.64313YesYes058
28b.b23x6 b.b24x6 99.17847.59333YesYes1578
29b.b23x6 b.l23x2 99.90823.8434YesNo078
30b.l21x7 b.l23x2 99.99836.66913NoNo058
31b.l21x7 b.l23x1 1003.45849NoYes056
32G.H3.17 b.l23x1 49.98755.8221YesYes156
33G.H3.17 b.l27x1 49.91053.17874YesYes159
34b.l1x6 b.l27x1 19.193521.4991YesYes199
35b.l1x6 b.l3x1 18.94387.90416YesNo199
36b.l3x1 b.l5x5 37.61128.62208NoYes099
37b.l23x1 b.l25x6 50.013813.7469YesYes168
38b.l25x6 b.l27x1 49.913122.2605YesYes189
39b.b2x1 b.l27x1 79.96815.51186YesYes189
40b.b2x1 b.l3x1 18.94569.76641YesNo189
41G.hns1.02 I2 89.62593.16457NoYes347
42G.S1.02 I2 24.27335.6295NoYes367
43G.S3.01 I2 24.13619.93206NoYes357
44G.S3.01 G.S3.03 24.01514.27399NoYes058
45G.S1.02 G.S3.03 24.0245.80638NoYes068
46G.H5.08 I2 25.05586.51313YesYes387
47G.H5.08 G.S3.03 24.06363.91191YesYes088
48G.S1.04 G.S3.03 62.58773.64732NoYes078
49G.S1.04 G.S4.03 62.18823.72587NoYes077
50G.h2s4.01 b.l5x5 34.105211.6517YesYes099
51G.S1.05 G.h2s4.01 33.408315.7489NoYes099
52G.S1.05 G.S1.07 32.59153.60918NoNo098
53G.S1.07 G.S4.04 32.31063.33365NoYes089
54b.b2x1 b.b6x1 60.85454.38431YesYes189
55b.b6x1 b.l9x6 60.64374.92833YesYes198
56G.H2.07 b.l9x6 19.79383.40353YesYes198
57G.H2.04 G.H2.07 18.54336.16067NoYes099
58G.H2.04 G.H3.08 18.39646.06054NoNo098
59G.H3.08 G.S4.04 17.98226.09068NoYes089
60G.S4.07 G.s1h1.04 45.0532.65456NoYes089
61G.S4.07 G.s5hg.01 45.45977.24299NoNo089
62G.S5.07 G.s5hg.01 47.08583.59182NoNo099
63G.S5.07 G.s6h5.01 48.71044.44883NoYes099
64G.S5.05 G.s6h5.01 51.11955.14581YesYes699
65G.S4.03 G.S5.05 56.89933.46161YesYes679
66G.H2.06 b.l17x6 36.98467.29035YesYes199
67G.H2.06 b.l9x6 37.48593.05033YesYes198
68G.H3.09 G.S4.04 23.61855.42072YesYes099
69G.S4.04 G.S5.04 26.3063.23064YesNo099
70G.H3.09 G.H4.15 15.36377.0742YesYes098
71G.H4.15 G.S5.04 15.37627.97946YesNo089
72G.S5.04 G.S5.06 10.64823.094NoNo098
73G.H3.06 G.H4.15 28.15448.27258NoYes068
74G.H4.10 G.H4.14 18.11137.86131YesNo075
75G.H3.06 G.H4.14 19.80433.70554NoNo065
762x38 3x49 32.48425.64552YesYes078
772x38 I2 33.08663.27279YesYes377
782x40 I1x50 33.58044.04402YesYes099
792x39 2x40 33.60323.86451YesYes099
80b.l17x5 b.l17x6 37.19843.37194NoYes169
81b.l17x5 b.l19x2 37.08483.16759NoYes169
82b.l17x3 b.l19x2 25.32994.90324YesYes199
83b.b19x4 b.l17x3 13.71228.04877YesYes189
84b.b19x4 b.b20x6 10.61656.41132YesYes186
85b.b17x7 b.b20x6 26.07099.63787YesYes186
86b.b17x7 b.b21x1 21.21534.09361YesYes187
87b.1x19 b.b21x1 18.30126.09876NoYes067
88b.1x15 b.1x19 14.75043.10165NoNo076
89b.1x12 b.1x15 13.86181.62683NoNo067
90b.b20x4 b.l17x3 11.050517.9437YesYes189
91b.b20x4 b.b20x6 21.21684.2437YesYes186
92b.b20x2 b.l19x2 11.335510.5674NoYes069
93b.b20x2 b.b20x4 11.04767.54506NoYes068
94b.l4x2 g.ctx16 11.75567.21073NoYes948
95b.l22x1 g.ctx3 35.89537.66394NoYes099
96b.b23x1 b.l22x1 35.80733.35804NoNo059
97b.b23x1 b.b24x5 35.74775.28857NoNo055
98b.b23x3 b.b24x5 35.68374.47993NoNo075
99b.b23x3 b.b26x3 35.55533.55598NoNo076
100b.b26x3 b.b27x3 35.49113.53589NoNo068
101b.b27x3 b.l25x3 34.76667.32579NoYes089
102b.l25x3 b.l27x2 34.60277.99342YesYes799
103b.b3x2 b.b4x6 58.30774.56085NoYes459
104b.b2x5 b.b3x2 58.21349.63521YesNo475
105b.l2x3 b.l2x5 42.23274.08411NoNo085
106b.b3x1 b.l2x3 41.8233.98737NoNo058
107b.b3x1 b.b6x5 41.41322.95458NoYes056
108b.b2x4 b.b6x5 21.2293.24003NoYes066
109b.b10x4 b.b2x4 20.814913.189NoNo066
110b.l26x3 b.l26x5 51.73256.86821NoNo075
111b.l26x1 b.l26x3 51.62486.28378NoNo477
112b.b2x5 b.l26x1 51.666111.2203YesNo477
113b.b3x3 b.b6x5 19.15773.93188YesYes086
114b.b3x3 b.b4x3 15.0033.34474YesYes087
115b.b4x7 b.l4x3 13.09797.2705NoNo086
116b.b5x2 b.l4x3 13.13239.27744YesNo076
117b.b10x2 b.b10x4 14.57563.77441NoNo066
118b.b10x2 b.b14x3 14.16024.16402NoYes065
119b.l25x4 b.l27x2 34.54854.31653YesYes059
120I1x49 b.l25x4 34.39164.46767NoYes075
1213x42 4x50 14.782613.2377YesYes1099
1223x34 4x50 11.32733.60674YesYes1099
1232x42 3x49 27.32923.64005NoYes088
1242x42 3x46 17.67315.63034NoYes089
1252x46 3x46 41.92424.7324NoYes099
1262x46 2x50 22.7774.46579NoYes098
1272x50 7x45 18.82955.26801YesYes089
1286x48 7x45 35.62337.00441YesYes289
1292x46 3x43 19.02453.17423NoNo099
1303x43 7x45 18.75553.68859NoYes099
1316x48 NT 27.16523.94167YesYes285
1321x60 I1x50 33.6353.09632YesYes079
1331x60 8x53 34.3446.18167YesNo078
1348x53 I1x49 34.37254.49236NoNo087
1352x39 2x43 25.48525.00362YesNo099
136G.s1h1.04 H.hehf.07 40.16420.0404167YesNo090
137H.HF.03 H.hehf.07 39.80870.0337396NoNo000
138H.HF.03 H.hehf.04 33.05550.0263542NoNo000
139H.HE.12 H.hehf.04 28.43480.0276979NoNo000
140H.HC.04 H.HE.12 28.07940.0126042NoNo000
141H.HC.03 H.HC.04 26.30220.0365312NoNo000
142H.HC.03 H.hbhc.04 25.94680.0502292NoYes000
143H.HB.12 H.hbhc.04 20.25980.0341354NoYes000
144H.HB.08 H.HB.12 19.54890.0381146NoNo000
145H.HB.08 H.HC.06 18.48260.0442396NoYes000
146H.HB.05 H.HC.06 17.06090.0658229YesYes000
147H.HB.05 H.HC.10 14.92830.0392187YesNo000
148H.HB.06 H.HC.10 14.57280.0217292NoNo000
149H.HB.02 H.HB.06 12.44020.0354062NoNo000
150H.HB.02 H.hchd.01 12.08480.0154271NoYes000
151H.hahb.06 H.hchd.01 10.66310.0268646NoYes000
1522x43 3x46 24.4329.9029NoYes099
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x36Lig4.574952YesYes6010
7x34Lig3.551182NoYes5010
7x37Lig4.374292YesYes8010
3x32Lig3.974642YesYes6010
7x38Lig4.847122NoYes7010
E2Lig9.291392YesYes5010
1x32Lig7.565332NoYes5010
E2x52Lig5.247992YesYes5010
1x29Lig3.823352NoYes2010
LigNT38.76422YesYes0501
E1Lig9.88072YesYes3010
NTNT223.8632YesYes5511
E1NT4.713122YesYes3511
1x357x383.678420NoNo6721
1x397x383.457812NoNo7721
2x533x366.585110NoYes8621
2x563x323.812670NoYes6621
2x603x324.958830NoYes6621
E1E113.75642YesYes3311
3x26E24.674352NoYes8521
3x26E2x5111.87932NoYes8822
3x363x403.38642YesNo6812
3x406x4812.37560NoYes8822
4x64E2x518.903362NoYes8822
4x68E25.531060NoYes6521
E2E2x513.920392YesYes5812
E2E226.01812YesYes5511
E2E2x523.292352YesYes5511
5x41E23.920952NoYes6521
5x415x446.903192NoNo6621
5x425x443.37830NoNo7621
6x487x374.148842YesYes8821
6x487x4112.6472YesNo8622
6x517x333.191462NoYes7722
6x517x374.735542NoYes7821
E3E35.727332YesYes4422
7x337x373.992982YesYes7821
E2NT9.067952YesYes5511
2x573x324.330072YesYes7621
E1E24.015932YesYes3511
4x64E26.03772NoYes8521
7x377x417.715982YesNo8612
1x32NT3.929542NoYes5511
5x44Lig4.836322NoYes6010
5x39E25.531830NoYes3521
3x33E23.4122NoYes7521
1x39NT3.481172NoYes7521
2x57NT4.420672YesYes7521
6x48NT3.941672YesYes8521
7x37NT4.247172YesYes8511
7x34NT4.143172NoYes5511
E2x51NT4.5182YesYes8521
3x36NT4.05852YesYes6511
E3NT4.302832YesYes4521
E2x51E2x525.2422YesYes8521
3x30E22.961172NoYes5521
3x29E22.841830NoYes5521
E1E2x502.620192YesNo3912
1x25Lig2.202930NoYes0010
1x28NT2.196330NoYes0521
1x291x332.172942NoNo2312
1x30NT1.683710NoYes2521
5x38E21.655660NoYes5521
2x64E2x521.596980NoYes7521
3x24E11.407492NoYes3321
2x65Lig1.38150NoYes4010
1x24NT1.173252NoYes0521
2x68Lig1.058250NoYes3010
1x21Lig1.05290NoYes0010
6x55NT0.9262NoYes7521
1x26Lig0.8539170NoYes0010
2x67E10.7672080NoYes3321
2x66E10.607750NoYes3321
1x22Lig0.5470170NoYes0010
1x23Lig0.30320NoYes0010
6x58NT0.2303330NoYes0521
1x19NT0.21750NoYes0521
2x69E10.03740620NoYes4321

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
69.23Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
62.07Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
61.29Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
55.56Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
54.29Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
50.00Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
50.00Consensuspth_onOrthosteric Ligandpth1_on pth2_on
48.39Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
48.28Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
46.88Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
46.43Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
45.45Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
44.83Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
44.83Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
44.83Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
44.83Consensusglp_onOrthosteric Ligandglp1_on glp2_on
44.83Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
44.44Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
44.44Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
44.44Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
44.44Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
44.00Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
43.33Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
43.33Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
43.33Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
43.33Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
42.86Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
42.86Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
42.86Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
42.86Consensuscalcitonin_onOrthosteric Ligandctlike_on
42.86Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
42.42Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
42.31Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
42.31Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
41.67Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
41.67Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
41.38Single6FJ3PTH6FJ3-PTH1-PTH
41.38Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
41.38Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
41.38Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
41.18Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
40.62Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
40.00Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
40.00Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
40.00Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
40.00Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
39.39Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
39.39Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
39.39Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
39.29Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
39.29Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
39.29Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
39.29Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
39.29Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
39.29Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
38.71Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
38.71Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
38.71Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
38.71Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
38.71Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
38.71Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
38.71Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
38.71Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
38.24Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
38.24Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
38.24Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.93Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
37.93Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
37.93Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
37.93Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
37.93Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
37.93Consensuspac_onOrthosteric Ligandpac1_on
37.50Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
37.50Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
37.50Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
36.67Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
36.67Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
36.67Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
36.67Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
36.67Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
36.67Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
36.67Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
36.67Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
36.36Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
36.36Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
36.36Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
36.00Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
35.71Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
35.71Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
35.48Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
35.48Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
35.29Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
35.29Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.48Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
34.48Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
34.48Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
34.38Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
34.38Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
34.29Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
34.29Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
34.29Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
33.33Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
33.33Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
32.26Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
32.26Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
32.26Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
32.26Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
32.26Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
32.26Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
32.14Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
31.43Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
31.25Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
31.25Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
31.25Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
31.03Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
31.03Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
30.30Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
30.30Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
30.30Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
30.30Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
30.30Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
30.00Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
30.00Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
30.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
29.41Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
29.03Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
29.03Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
29.03Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
28.57Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
28.57Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
28.57Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
28.57Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
28.21Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
28.12Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
28.12Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
28.12Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
27.59Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
27.59Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
27.59Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
27.59Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
27.50Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
27.27Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
27.27Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
27.27Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
27.27Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
27.27Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
27.27Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
27.03Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
26.92Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
26.92Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
26.92Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
26.83Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
26.67Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
26.67Consensusangiotensin_onOrthosteric Ligandat1_on
26.67Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
26.67Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
26.47Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
26.47Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
26.47Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
26.47Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
26.47Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
26.32Single8HS2Fab0468HS2-GPR20-Fab046
25.93Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
25.81Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
25.81Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
25.81Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
25.81Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
25.81Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
25.81Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
25.71Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
25.00Single3NY9ICI118-5513NY9-β2-ICI118-551
25.00Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
25.00Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
25.00Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
25.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
25.00Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
25.00Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
25.00Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
25.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
25.00Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
25.00Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
25.00Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
25.00Consensushca_on_gpOrthosteric Ligandhca2_on_gp
24.32Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
24.32Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
24.24Single4XT3Fractalkine4XT3-US28-Fractalkine
24.24Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
24.24Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
24.24Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
24.24Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
24.24Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
24.14Single4XT1Fractalkine4XT1-US28-Fractalkine
24.14Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
24.14Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
24.14Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
24.14Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
24.00Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
24.00Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
24.00Single8TF5Oleic acid8TF5-GPR6-Oleic acid
24.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
24.00Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
24.00Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
24.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
23.81Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.81Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
23.81Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
23.81Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
23.53Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
23.53Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
23.53Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
23.53Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
23.53Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
23.53Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
23.33Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
23.33Single7XNACYN1548067XNA-SST2-CYN154806
23.33Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
23.33Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
23.33Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
23.33Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
23.33Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
23.08Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
23.08Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
23.08Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
23.08Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
23.08Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
23.08Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
23.08Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
23.08Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
23.08Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
22.86Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
22.86Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
22.86Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
22.86Consensusbradykinin_onOrthosteric Ligandbk2_on
22.86Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
22.86Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
22.73Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
22.73Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
22.73Single8K5BNiacin8K5B-HCA2-Niacin
22.73Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
22.58Single3OE0CVX153OE0-CXCR4-CVX15
22.58Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
22.58Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
22.50Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
22.22Single5GLHEndothelin-15GLH-ETB-Endothelin-1
22.22Single6IGKEndothelin-36IGK-ETB-Endothelin-3
22.22Single6OS2TRV0266OS2-AT1-TRV026
22.22Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
22.22Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
22.22Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
22.22Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
22.22Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
22.22Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
22.22Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
22.22Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
22.22Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
22.22Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
22.22Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
22.22Consensuslpa_offOrthosteric Ligandlpa1_off
22.22Consensuslpl_offOrthosteric Ligands1p_off lpa_off
21.88Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
21.88Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
21.88Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.88Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.88Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
21.88Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
21.88Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
21.88Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
21.74Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
21.74Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8GNGIstradefylline8GNG-A2A-Istradefylline
21.74Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
21.74Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
21.74Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
21.74Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
21.74Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
21.43Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
21.43Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
21.43Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
21.43Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
21.43Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
21.43Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
21.43Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
21.43Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
21.43Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
21.43Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
21.43Consensuscck_onOrthosteric Ligandccka_on cckb_on
21.43Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
21.21Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
21.21Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
21.21Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
21.21Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
21.21Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
21.21Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
21.21Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Single8ZRTET-18ZRT-ETB-ET-1
21.21Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
21.21Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
21.21Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
21.21Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.21Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
21.05Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
21.05Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
20.83Single2YDOAdenosine2YDO-A2A-Adenosine
20.83Single7AROLUF58337ARO-A2A-LUF5833-Na
20.83Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
20.83Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
20.83Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
20.83Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
20.83Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
20.83Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
20.83Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
20.83Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
20.83Single8K5CAcipimox8K5C-HCA2-Acipimox
20.83Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
20.83Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
20.83Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
20.83Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
20.83Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
20.83Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
20.83Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
20.83Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
20.83Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
20.83Consensushca_onOrthosteric Ligandhca2_on
20.83Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
20.69Single4UG2CGS216804UG2-A2A-CGS21680
20.69Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
20.69Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
20.69Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
20.69Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
20.69Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
20.69Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
20.69Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
20.69Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
20.69Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
20.69Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
20.69Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
20.69Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
20.59Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
20.59Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
20.59Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
20.59Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
20.59Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
20.59Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
20.00Single5UENDU1725UEN-A1-DU172
20.00Single6D27CAY104716D27-DP2-CAY10471
20.00Single6PS1Timolol6PS1-β2-Timolol
20.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
20.00Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
20.00Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
20.00Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
20.00Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
20.00Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.00Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
20.00Single8CU6LJ-45178CU6-A2A-LJ-4517
20.00Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
20.00Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
20.00Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
20.00Single8K5DGSK2560738K5D-HCA2-GSK256073
20.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
20.00Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
20.00Single8T1WCVN4248T1W-GPR6-CVN424
20.00Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
20.00Single8WDTphotoNECA8WDT-A2A-photoNECA
20.00Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
20.00Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
20.00Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
20.00Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
20.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
20.00Single9AS1DMT9AS1-5-HT2A-DMT
20.00Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
20.00Single9CHXS-Carazolol9CHX-β2-S-Carazolol
20.00Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
20.00Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
20.00Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
20.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
20.00Consensusa3_onOrthosteric Liganda3a_on
20.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
20.00Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
20.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
20.00Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
20.00Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
20.00Consensuslpl_onOrthosteric Ligands1p_on lpa_on
20.00Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
20.00Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
20.00Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.00Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
20.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
20.00Consensussomatostatin_offOrthosteric Ligandsst2_off
20.00Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.44Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
19.44Consensusendothelin_onOrthosteric Ligandetb_on eta_on
19.35Single3QAKUK-4320973QAK-A2A-UK-432097
19.35Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
19.35Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
19.35Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
19.35Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
19.35Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
19.35Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
19.35Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
19.35Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
19.35Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
19.23Single5C1MBU725C1M-μ-BU72
19.23Single5JQHS-Carazolol5JQH-β2-S-Carazolol
19.23Single5N2RPSB-365N2R-A2A-PSB-36-Na
19.23Single5N2SPSB365N2S-A1-PSB36
19.23Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
19.23Single5TVNLSD5TVN-5-HT2B-LSD
19.23Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
19.23Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
19.23Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
19.23Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
19.23Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
19.23Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
19.23Single6PS6Timolol6PS6-β2-Timolol
19.23Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
19.23Single7C61Ergotamine7C61-5-HT1B-Ergotamine
19.23Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
19.23Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
19.23Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
19.23Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
19.23Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
19.23Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
19.23Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
19.23Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
19.23Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
19.23Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
19.23Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
19.23Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
19.23Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
19.23Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
19.23Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
19.23Single9EHSLUF76029EHS-A3A-LUF7602
19.23Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
19.23Consensusa3_on_gpOrthosteric Liganda3a_on_gp
19.23Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
19.23Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
19.23Consensusadenosine_offOrthosteric Liganda1_off a2_off
19.23Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
19.23Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
19.23Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
19.23Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
19.23Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
19.23Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
19.23Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.23Consensustrace-amine_onOrthosteric Ligandta1_on
19.05Single8A2OTheophylline8A2O-A2A-Theophylline-Na
19.05Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
18.92Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
18.92Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
18.92Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
18.92Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
18.75Single5WF5UK-4320975WF5-A2A-UK-432097
18.75Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
18.75Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
18.75Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
18.75Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.75Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.75Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
18.75Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.75Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
18.75Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.75Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
18.75Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
18.75Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
18.75Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
18.75Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
18.75Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
18.75Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
18.52Single2YDVNECA2YDV-A2A-NECA
18.52Single3P0GBI1671073P0G-β2-BI167107
18.52Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
18.52Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
18.52Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
18.52Single4UHRCGS216804UHR-A2A-CGS21680
18.52Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
18.52Single5G53NECA5G53-A2A-NECA-Gs
18.52Single5XR8AM8415XR8-CB1-AM841
18.52Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
18.52Single6WGTLSD6WGT-5-HT2A-LSD
18.52Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
18.52Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
18.52Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
18.52Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
18.52Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
18.52Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
18.52Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
18.52Single8E0GBU728E0G-μ-BU72
18.52Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
18.52Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
18.52Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
18.52Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
18.52Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
18.52Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
18.52Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
18.52Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
18.52Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
18.52Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
18.52Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
18.52Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
18.52Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
18.52Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
18.52Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
18.52Consensusa2_onOrthosteric Liganda2b_on
18.52Consensusa2_on_gpOrthosteric Liganda2b_on_gp
18.52Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
18.52Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
18.52Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
18.52Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
18.52Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
18.52Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
18.52Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
18.52Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
18.52Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
18.52Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
18.52Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
18.52Consensuslpa_onOrthosteric Ligandlpa1_on
18.52Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
18.52Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
18.52Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
18.52Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.52Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
18.42Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
18.18Single6JODAngiotensin II6JOD-AT2-Angiotensin II
18.18Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
18.18Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
18.18Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
18.18Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
18.18Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
18.18Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.18Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.18Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
18.18Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
17.95Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
17.86Single4XEENeurotensin4XEE-NTS1-Neurotensin
17.86Single4XESNeurotensin4XES-NTS1-Neurotensin
17.86Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
17.86Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
17.86Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
17.86Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
17.86Single6MXTSalmeterol6MXT-β2-Salmeterol
17.86Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
17.86Single6YVRNTS8-136YVR-NTS1-NTS8-13
17.86Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
17.86Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
17.86Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
17.86Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
17.86Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
17.86Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
17.86Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
17.86Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
17.86Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
17.86Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
17.86Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
17.86Single8JJ8Formoterol8JJ8-β2-Formoterol
17.86Single8JJLOlodaterol8JJL-β2-Olodaterol
17.86Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
17.86Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
17.86Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
17.86Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
17.86Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.86Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
17.86Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
17.86Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
17.86Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
17.86Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
17.86Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
17.86Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
17.86Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
17.86Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
17.86Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
17.86Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
17.86Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
17.86Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
17.86Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
17.86Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
17.86Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
17.86Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
17.65Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
17.65Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
17.65Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
17.65Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
17.65Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
17.65Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
17.65Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
17.65Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
17.50Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
17.39Single3OE9IT1t3OE9-CXCR4-IT1t
17.39Single6LI0C176LI0-GPR52-C17
17.39Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
17.39Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
17.39Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
17.39Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
17.39Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
17.39Single9B9Y7DY9B9Y-CB1-7DY
17.39Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
17.39Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
17.24Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
17.24Single4BUONeurotensin4BUO-NTS1-Neurotensin
17.24Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
17.24Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
17.24Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
17.24Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
17.24Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
17.24Single7EZCUKA7EZC-A2A-UKA
17.24Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
17.24Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
17.24Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
17.24Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
17.24Single7UM4AS26747237UM4-5-HT5A-AS2674723
17.24Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
17.24Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
17.24Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
17.24Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
17.24Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
17.24Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
17.24Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
17.24Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
17.24Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
17.24Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
17.24Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8XVUCXCL28XVU-CXCR2-CXCL2
17.24Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
17.24Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
17.24Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
17.24Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
17.24Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
17.24Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
17.24Consensuschemerin_onOrthosteric Ligandcml1_on
17.24Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
17.24Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
17.24Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
17.24Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
17.24Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
17.24Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
17.14Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.14Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
17.14Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
17.14Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
17.14Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
17.14Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
17.14Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
16.67Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
16.67Single3ODUIT1t3ODU-CXCR4-IT1t
16.67Single3PWHZM-2413853PWH-A2A-ZM-241385
16.67Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
16.67Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
16.67Single4BWBNeurotensin4BWB-NTS1-Neurotensin
16.67Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
16.67Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
16.67Single5U09Taranabant5U09-CB1-Taranabant
16.67Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
16.67Single5WF6UK-4320975WF6-A2A-UK-432097
16.67Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
16.67Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
16.67Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
16.67Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
16.67Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
16.67Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
16.67Single7BR3Elagolix7BR3-GnRH1-Elagolix
16.67Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
16.67Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
16.67Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
16.67Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
16.67Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
16.67Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
16.67Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
16.67Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
16.67Single7XN9L-054,5227XN9-SST2-L-054,522
16.67Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
16.67Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
16.67Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
16.67Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
16.67Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
16.67Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
16.67Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
16.67Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
16.67Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
16.67Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
16.67Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
16.67Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
16.67Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
16.67Single8IWESpermidine8IWE-TA9-Spermidine
16.67Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
16.67Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
16.67Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
16.67Single8QJ2pN1628QJ2-MC4-pN162-Gs
16.67Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
16.67Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
16.67Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
16.67Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
16.67Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
16.67Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
16.67Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
16.67Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
16.67Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
16.67Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
16.67Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
16.67Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
16.67Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
16.67Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
16.67Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
16.67Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
16.67Consensusalpha2_offOrthosteric Ligandalpha2c_off
16.67Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
16.67Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
16.67Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
16.67Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
16.67Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
16.67Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
16.67Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
16.67Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
16.67Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
16.22Single6IGLIRL16206IGL-ETB-IRL1620
16.22Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
16.22Single8IY6Endothelin-18IY6-ETB-Endothelin-1
16.13Single4IARErgotamine4IAR-5-HT1B-Ergotamine
16.13Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
16.13Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
16.13Single7F8XNN90567F8X-CCKA-NN9056
16.13Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
16.13Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
16.13Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
16.13Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
16.13Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
16.13Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
16.13Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
16.13Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.13Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
16.13Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
16.13Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
16.00Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
16.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
16.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
16.00Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
16.00Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
16.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
16.00Single5IUBQ274563445IUB-A2A-Q27456344-Na
16.00Single5JTBZM-2413855JTB-A2A-ZM-241385
16.00Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
16.00Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
16.00Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
16.00Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
16.00Single6AQFZM-2413856AQF-A2A-ZM-241385
16.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
16.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
16.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
16.00Single6PS4ICI118-5516PS4-β2-ICI118-551
16.00Single6PS5S-Propranolol6PS5-β2-S-Propranolol
16.00Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
16.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
16.00Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
16.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
16.00Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
16.00Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
16.00Single7F61PF-036547467F61-H3-PF-03654746
16.00Single7T32ZM-2413857T32-A2A-ZM-241385
16.00Single7UL3Famotidine7UL3-H2-Famotidine
16.00Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
16.00Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
16.00Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
16.00Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
16.00Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
16.00Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
16.00Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
16.00Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
16.00Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
16.00Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
16.00Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.00Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
16.00Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
16.00Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
16.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
16.00Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
16.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
16.00Single8IHKAcifran8IHK-HCA3-Acifran
16.00Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
16.00Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
16.00Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
16.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
16.00Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
16.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
16.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
16.00Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.00Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.00Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.00Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
16.00Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
16.00Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
16.00Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
16.00Single9AS5Mescaline9AS5-5-HT2A-Mescaline
16.00Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single9BA0A1AKN9BA0-CB1-A1AKN
16.00Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
16.00Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
16.00Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
16.00Consensusa2_offOrthosteric Liganda2a_off
16.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
16.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
16.00Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
16.00Consensusgrh_offOrthosteric Ligandgnrh1_off
16.00Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.79Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
15.79Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
15.79Consensusbombesin_onOrthosteric Ligandbb2_on
15.79Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
15.79Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
15.79Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
15.62Single6HLOAprepitant6HLO-NK1-Aprepitant
15.62Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
15.62Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
15.62Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
15.62Single7SK5CXCL127SK5-ACKR3-CXCL12
15.62Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
15.62Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
15.62Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
15.62Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
15.62Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
15.62Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
15.62Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
15.62Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
15.62Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
15.62Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
15.62Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
15.62Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
15.38Single2Y04Salbutamol2Y04-β1-Salbutamol
15.38Single3EMLZM-2413853EML-A2A-ZM-241385
15.38Single3NY8ICI118-5513NY8-β2-ICI118-551
15.38Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
15.38Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
15.38Single4DAJTiotropium4DAJ-M3-Tiotropium
15.38Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
15.38Single4GBRS-Carazolol4GBR-β2-S-Carazolol
15.38Single4QKX35V4QKX-β2-35V
15.38Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
15.38Single5IU8Q274563475IU8-A2A-Q27456347-Na
15.38Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
15.38Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
15.38Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
15.38Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
15.38Single5TGZAM65385TGZ-CB1-AM6538
15.38Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
15.38Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
15.38Single6H7MSalbutamol6H7M-β1-Salbutamol
15.38Single6IIVDaltroban6IIV-TXA2-Daltroban
15.38Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
15.38Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
15.38Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
15.38Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
15.38Single6S0LZM-2413856S0L-A2A-ZM-241385
15.38Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
15.38Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
15.38Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
15.38Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
15.38Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
15.38Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
15.38Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
15.38Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
15.38Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
15.38Single7PYRPSB-21157PYR-A2A-PSB-2115
15.38Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
15.38Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
15.38Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
15.38Single7UL4Alvimopan7UL4-μ-Alvimopan
15.38Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
15.38Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
15.38Single7V3ZCP559407V3Z-CB1-CP55940
15.38Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
15.38Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
15.38Single7WC7Lisuride7WC7-5-HT2A-Lisuride
15.38Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
15.38Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
15.38Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
15.38Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
15.38Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
15.38Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
15.38Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
15.38Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
15.38Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
15.38Single8JJOAlprenolol8JJO-β2-Alprenolol
15.38Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
15.38Single8JXRLSD8JXR-D1-LSD
15.38Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
15.38Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
15.38Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
15.38Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
15.38Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
15.38Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
15.38Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
15.38Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
15.38Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
15.38Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
15.38Single9H37A1IR09H37-A2A-A1IR0-Na
15.38Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
15.38Consensus5ht5_onOrthosteric Ligand5ht5a_on
15.38Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
15.38Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
15.38Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
15.38Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
15.38Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
15.38Consensusdopamine_offOrthosteric Ligandd2_off d3_off
15.38Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
15.38Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
15.38Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
15.38Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
15.38Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
15.38Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
15.15Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
15.15Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
15.15Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
15.15Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
15.15Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
15.15Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
15.15Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
15.00Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
14.81Single2RH1S-Carazolol2RH1-β2-S-Carazolol
14.81Single2Y03Isoprenaline2Y03-β1-Isoprenaline
14.81Single2YCWS-Carazolol2YCW-β1-S-Carazolol
14.81Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
14.81Single5CGCHTL142425CGC-mGlu5-HTL14242
14.81Single5D6LS-Carazolol5D6L-β2-S-Carazolol
14.81Single5IUAQ274563485IUA-A2A-Q27456348-Na
14.81Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
14.81Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
14.81Single6D26Fevipiprant6D26-DP2-Fevipiprant
14.81Single6E67BI1671076E67-β2-BI167107-Gs(CT)
14.81Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
14.81Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
14.81Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
14.81Single6LUQHaloperidol6LUQ-D2-Haloperidol
14.81Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
14.81Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
14.81Single6S0QZM-2413856S0Q-A2A-ZM-241385
14.81Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
14.81Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
14.81Single7C4SS1P7C4S-S1P3-S1P
14.81Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
14.81Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
14.81Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
14.81Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
14.81Single7SINNPS-21437SIN-CaS-NPS-2143
14.81Single7SINNPS-21437SIN-CaS-NPS-2143
14.81Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
14.81Single7W41PD1762527W41-BB2-PD176252
14.81Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
14.81Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
14.81Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
14.81Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
14.81Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
14.81Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
14.81Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GNEKW-63568GNE-A2A-KW-6356-Na
14.81Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
14.81Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
14.81Single8JXSPF-61428JXS-D1-PF-6142
14.81Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
14.81Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
14.81Single8QOTNanobody-E8QOT-μ-Nanobody-E
14.81Single8S4DCMF-0198S4D-Apelin-CMF-019
14.81Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
14.81Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
14.81Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
14.81Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
14.81Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
14.81Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
14.81Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single9B9ZA1AKO9B9Z-CB1-A1AKO
14.81Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
14.81Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
14.81Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
14.81Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
14.81Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
14.81Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
14.81Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
14.81Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
14.81Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
14.81Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
14.81Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
14.81Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
14.81Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
14.81Consensusamine_offonOrthosteric Ligandamine_off amine_on
14.81Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
14.81Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
14.81Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
14.81Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
14.81Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
14.81Consensusbombesin_offOrthosteric Ligandbb2_off
14.81Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
14.81Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
14.81Consensusdp_offOrthosteric Liganddp2_off
14.81Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
14.81Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
14.81Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
14.81Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
14.81Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
14.81Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
14.81Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
14.81Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
14.81Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
14.81Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
14.71Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
14.71Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
14.71Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
14.71Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
14.71Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
14.71Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
14.71Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
14.71Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
14.71Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
14.71Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
14.71Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
14.71Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
14.71Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
14.71Consensusvasop-oxy_onOrthosteric Ligandv2_on
14.71Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
14.29Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
14.29Single4BV0Neurotensin4BV0-NTS1-Neurotensin
14.29Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
14.29Single5D5AS-Carazolol5D5A-β2-S-Carazolol
14.29Single5D5BS-Carazolol5D5B-β2-S-Carazolol
14.29Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
14.29Single5V54Methiothepin5V54-5-HT1B-Methiothepin
14.29Single5XRAAM115425XRA-CB1-AM11542
14.29Single6H7JIsoprenaline6H7J-β1-Isoprenaline
14.29Single6J21Aprepitant6J21-NK1-Aprepitant
14.29Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
14.29Single6OS1TRV0266OS1-AT1-TRV026
14.29Single7B6WCyclazosin7B6W-α1b-Cyclazosin
14.29Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
14.29Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
14.29Single7F1TMIP-1a7F1T-CCR5-MIP-1a
14.29Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
14.29Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
14.29Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
14.29Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
14.29Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
14.29Single7PX4PSB-21137PX4-A2A-PSB-2113
14.29Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
14.29Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
14.29Single7TUYGSK682753A7TUY-GPR183-GSK682753A
14.29Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
14.29Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
14.29Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
14.29Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
14.29Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
14.29Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
14.29Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
14.29Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
14.29Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
14.29Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
14.29Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
14.29Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
14.29Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
14.29Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
14.29Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.29Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
14.29Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
14.29Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
14.29Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
14.29Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
14.29Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
14.29Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
14.29Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
14.29Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
14.29Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
14.29Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
14.29Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
14.29Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
14.29Single8PWNTheophylline8PWN-A2A-Theophylline
14.29Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
14.29Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
14.29Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
14.29Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
14.29Single8ZWFJR14a8ZWF-C3aB-JR14a
14.29Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
14.29Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
14.29Single9BJKNaloxone9BJK-μ-Naloxone-NAM
14.29Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
14.29Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
14.29Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
14.29Consensus5ht1_offOrthosteric Ligand5ht1b_off
14.29Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
14.29Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
14.29Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
14.29Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
14.29Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
14.29Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
14.29Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
14.29Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
14.29Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
14.29Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
14.29Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
14.29Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
14.29Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
14.29Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
14.29Consensusneurotensin_onOrthosteric Ligandnts1_on
14.29Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
14.29Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
14.29Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
14.29Consensusrelaxin_onOrthosteric Ligandrxfp4_on
14.29Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
13.89Single7SK3CXCL127SK3-ACKR3-CXCL12
13.89Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
13.89Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.89Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.79Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
13.79Single3D4STimolol3D4S-β2-Timolol
13.79Single4AMIBucindolol4AMI-β1-Bucindolol
13.79Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
13.79Single4LDEBI1671074LDE-β2-BI167107
13.79Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
13.79Single4RWADIPP-NH24RWA-δ-DIPP-NH2
13.79Single5CXVTiotropium5CXV-M1-Tiotropium
13.79Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
13.79Single6A93Risperidone6A93-5-HT2A-Risperidone
13.79Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
13.79Single6CM4Risperidone6CM4-D2-Risperidone
13.79Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
13.79Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
13.79Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
13.79Single6IIURamatroban6IIU-TXA2-Ramatroban
13.79Single6KQICP559406KQI-CB1-CP55940-Org27569
13.79Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
13.79Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
13.79Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
13.79Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.79Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.79Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
13.79Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
13.79Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.79Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
13.79Single7YITNalfurafine7YIT-κ-Nalfurafine
13.79Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
13.79Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
13.79Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
13.79Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
13.79Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
13.79Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
13.79Single8JWY2-1188JWY-A2A-2-118
13.79Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
13.79Single8XQJJN2418XQJ-Apelin-JN241
13.79Single8XWMCXCL68XWM-CXCR2-CXCL6
13.79Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
13.79Single8XYIVUF106618XYI-CXCR3-VUF10661
13.79Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
13.79Single9DGIZ85267113509DGI-CB1-Z8526711350
13.79Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
13.79Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
13.79Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
13.79Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
13.79Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.79Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.79Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
13.79Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
13.79Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
13.79Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.79Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
13.79Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
13.79Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
13.79Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
13.79Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
13.79Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
13.79Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
13.79Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.79Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
13.79Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
13.79Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.79Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.64Single3RFMCaffeine3RFM-A2A-Caffeine
13.64Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
13.64Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
13.64Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
13.64Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
13.64Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
13.64Single9CHUNoradrenaline9CHU-β2-Noradrenaline
13.64Consensusp2y_offOrthosteric Ligandp2y1_off
13.51Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
13.51Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
13.51Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
13.51Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
13.51Single9KDFRES-701-39KDF-ETB-RES-701-3
13.33Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
13.33Single5CGDHTL142425CGD-mGlu5-HTL14242
13.33Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
13.33Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
13.33Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
13.33Single6H7LDobutamine6H7L-β1-Dobutamine
13.33Single6IBLArformoterol6IBL-β1-Arformoterol
13.33Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
13.33Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
13.33Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
13.33Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
13.33Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
13.33Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
13.33Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
13.33Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
13.33Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
13.33Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
13.33Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
13.33Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
13.33Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
13.33Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
13.33Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.33Single8XWFCXCL38XWF-CXCR2-CXCL3
13.33Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
13.33Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
13.33Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
13.33Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
13.33Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.33Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.33Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
13.33Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
13.33Consensusprostanoid_offOrthosteric Ligandep_off dp_off
13.16Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
13.16Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
13.04Single3OE6IT1t3OE6-CXCR4-IT1t
13.04Single4XNWMRS25004XNW-P2Y1-MRS2500
13.04Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
13.04Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
13.04Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
13.04Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
13.04Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
13.04Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
13.04Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
13.04Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
13.04Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
13.04Single9LRCHistamine9LRC-H4-Histamine
13.04Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
13.04Consensus5ht2_onOrthosteric Ligand5ht2b_on
13.04Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
13.04Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
13.04Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
12.90Single5ZTYAM102575ZTY-CB2-AM10257
12.90Single6KNMJN241-96KNM-Apelin-JN241-9
12.90Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
12.90Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
12.90Single6PT3DPI-2876PT3-δ-DPI-287
12.90Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
12.90Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
12.90Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
12.90Single7SK9CCX6627SK9-ACKR3-CCX662
12.90Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
12.90Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
12.90Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8XQJJN2418XQJ-Apelin-JN241
12.90Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
12.90Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
12.90Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
12.90Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
12.90Single9IPYJR14a9IPY-C3aB-JR14a
12.90Single9JF4PD1683689JF4-BB1-PD168368
12.90Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
12.90Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
12.90Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.90Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.82Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
12.82Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
12.50Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
12.50Single4O9RCyclopamine4O9R-SMO-Cyclopamine
12.50Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
12.50Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.50Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
12.50Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
12.50Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
12.50Single7QA8Peptide7QA8-STE2-Peptide
12.50Single7QA8Peptide7QA8-STE2-Peptide
12.50Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
12.50Single7SRQLSD7SRQ-5-HT2B-LSD
12.50Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
12.50Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
12.50Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
12.50Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.50Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
12.50Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
12.50Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
12.50Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
12.50Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
12.50Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
12.50Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
12.50Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
12.50Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
12.50Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
12.50Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
12.50Single8IEBA1LYA8IEB-GPR156-A1LYA
12.50Single8IEIA1LYA8IEI-GPR156-A1LYA
12.50Single8IEIA1LYA8IEI-GPR156-A1LYA
12.50Single8IEPA1LYA8IEP-GPR156-A1LYA
12.50Single8IEPA1LYA8IEP-GPR156-A1LYA
12.50Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
12.50Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
12.50Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
12.50Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
12.50Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
12.50Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
12.50Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
12.50Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
12.50Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
12.50Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8XWNCXCL88XWN-CXCR2-CXCL8
12.50Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
12.50Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
12.50Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
12.50Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
12.50Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
12.50Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9AS7Psilocin9AS7-5-HT2A-Psilocin
12.50Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
12.50Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
12.50Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
12.50Single9M4TSilodosin9M4T-Alpha1A-Silodosin
12.50Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
12.50Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
12.50Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
12.50Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
12.50Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
12.50Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
12.50Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
12.50Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
12.12Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
12.12Single8IEBA1LYA8IEB-GPR156-A1LYA
12.12Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
12.12Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
12.12Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
12.12Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
12.12Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
12.12Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
12.12Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
12.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
12.00Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
12.00Single4QINSAG1.54QIN-SMO-SAG1.5
12.00Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
12.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
12.00Single6AKXA4R6AKX-CCR5-A4R
12.00Single6AKYMaraviroc6AKY-CCR5-Maraviroc
12.00Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
12.00Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
12.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
12.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
12.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.00Single6TODEMPA6TOD-OX1-EMPA-Na
12.00Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
12.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
12.00Single7F8ULintitript7F8U-CCKA-Lintitript
12.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
12.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
12.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
12.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
12.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
12.00Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
12.00Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
12.00Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
12.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
12.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
12.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
12.00Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
12.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
12.00Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
12.00Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
12.00Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
12.00Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
12.00Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
12.00Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
12.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
12.00Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
12.00Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
12.00Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
12.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
12.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
12.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
12.00Single8Y0HVUF114188Y0H-CXCR3-VUF11418
12.00Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
12.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
12.00Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
12.00Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
12.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
12.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
12.00Single9H2XA1IR19H2X-A2A-A1IR1-Na
12.00Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
12.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
12.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
12.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
12.00Consensusangiotensin_offOrthosteric Ligandat1_off
12.00Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
12.00Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
12.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
12.00Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
12.00Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
12.00Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
12.00Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
12.00Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
12.00Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
12.00Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
12.00Consensusorexin_offOrthosteric Ligandox2_off ox1_off
12.00Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
12.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
12.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
12.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
12.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
11.76Single6PT2KGCHM076PT2-δ-KGCHM07
11.76Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
11.76Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
11.76Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
11.76Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
11.76Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
11.76Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
11.76Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
11.76Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
11.76Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single3REYXAC3REY-A2A-XAC
11.54Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
11.54Single4MBSMaraviroc4MBS-CCR5-Maraviroc
11.54Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
11.54Single4ZJCSB-6740424ZJC-OX1-SB-674042
11.54Single5UVIZM-2413855UVI-A2A-ZM-241385
11.54Single6A94Zotepine6A94-5-HT2A-Zotepine
11.54Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
11.54Single6KUXRS-799486KUX-α2a-RS-79948
11.54Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
11.54Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
11.54Single6TPGEMPA6TPG-OX2-EMPA
11.54Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
11.54Single6V9SGTPL114036V9S-OX1-GTPL11403
11.54Single6VI4JDTic6VI4-κ-JDTic
11.54Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
11.54Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
11.54Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
11.54Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
11.54Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
11.54Single6ZG9GSK10347026ZG9-M1-GSK1034702
11.54Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
11.54Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
11.54Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
11.54Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
11.54Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
11.54Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
11.54Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.54Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
11.54Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
11.54Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
11.54Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
11.54Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
11.54Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
11.54Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
11.54Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
11.54Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
11.54Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
11.54Single8RLNLUF58348RLN-A2A-LUF5834
11.54Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
11.54Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
11.54Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
11.54Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
11.54Single8ZPMAMD0708ZPM-CXCR4-AMD070
11.54Single8ZPNAMD31008ZPN-CXCR4-AMD3100
11.54Single9ARXSerotonin9ARX-5-HT2A-Serotonin
11.54Single9AS3LSD9AS3-5-HT2A-LSD
11.54Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
11.54Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
11.54Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
11.54Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
11.54Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
11.54Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
11.54Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
11.54Consensusalpha1_onOrthosteric Ligandalpha1a_on
11.54Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
11.54Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
11.54Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
11.54Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
11.54Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
11.54Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
11.54Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
11.43Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
11.43Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
11.43Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
11.43Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
11.43Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
11.43Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
11.36Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
11.36Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
11.11Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
11.11Single2Y01Dobutamine2Y01-β1-Dobutamine
11.11Single2Y02Carmoterol2Y02-β1-Carmoterol
11.11Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
11.11Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
11.11Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
11.11Single4EJ4Naltrindole4EJ4-δ-Naltrindole
11.11Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
11.11Single4MQSIperoxo4MQS-M2-Iperoxo
11.11Single4QIMANTA XV4QIM-SMO-ANTA XV
11.11Single4U14Tiotropium4U14-M3-Tiotropium
11.11Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
11.11Single4YAYZD-71554YAY-AT1-ZD-7155
11.11Single5DHHSB-6121115DHH-NOP-SB-612111
11.11Single5DSGTiotropium5DSG-M4-Tiotropium
11.11Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
11.11Single5T04Neurotensin5T04-NTS1-Neurotensin
11.11Single5UIGCmpd-15UIG-A2A-Cmpd-1
11.11Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
11.11Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
11.11Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
11.11Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
11.11Single6DRXLisuride6DRX-5-HT2B-Lisuride
11.11Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
11.11Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
11.11Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
11.11Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
11.11Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
11.11Single6TOTLemborexant6TOT-OX1-Lemborexant
11.11Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
11.11Single7BU7BI1671077BU7-β1-BI167107
11.11Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
11.11Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
11.11Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
11.11Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
11.11Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
11.11Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
11.11Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
11.11Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
11.11Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
11.11Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
11.11Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
11.11Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
11.11Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
11.11Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
11.11Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
11.11Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
11.11Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
11.11Single7YXAONO-54306087YXA-S1P5-ONO-5430608
11.11Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
11.11Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
11.11Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
11.11Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
11.11Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
11.11Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
11.11Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
11.11Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
11.11Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
11.11Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
11.11Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
11.11Single8X63Mepyramine8X63-H1-Mepyramine
11.11Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
11.11Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
11.11Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
11.11Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
11.11Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
11.11Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
11.11Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
11.11Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
11.11Single9JEAAtropine9JEA-M1-Atropine
11.11Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
11.11Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
11.11Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
11.11Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
11.11Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
11.11Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
11.11Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
11.11Consensusalpha2_onOrthosteric Ligandalpha2b_on
11.11Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
11.11Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
11.11Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
11.11Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
11.11Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
11.11Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
11.11Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
11.11Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
11.11Consensushistamine_offOrthosteric Ligandh1_off
11.11Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
11.11Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
11.11Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
10.81Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
10.81Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
10.71Single2Y00Dobutamine2Y00-β1-Dobutamine
10.71Single4JKVTaladegib4JKV-SMO-Taladegib
10.71Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
10.71Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
10.71Single5WIUNemonapride5WIU-D4-Nemonapride
10.71Single5WIVNemonapride5WIV-D4-Nemonapride-Na
10.71Single5WQCEMPA5WQC-OX2-EMPA
10.71Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
10.71Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
10.71Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
10.71Single6TP6Filorexant6TP6-OX1-Filorexant
10.71Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
10.71Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
10.71Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
10.71Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
10.71Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
10.71Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
10.71Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
10.71Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
10.71Single7WC6LSD7WC6-5-HT2A-LSD
10.71Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
10.71Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
10.71Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
10.71Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
10.71Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
10.71Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
10.71Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
10.71Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
10.71Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
10.71Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
10.71Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
10.71Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
10.71Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
10.71Single8ZMFA1L108ZMF-5-HT2C-A1L10
10.71Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
10.71Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
10.71Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
10.71Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
10.71Single9HC04YI9HC0-mGlu5-4YI
10.71Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
10.71Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
10.71Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
10.71Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
10.71Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
10.71Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
10.71Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
10.71Consensusblt_offOrthosteric Ligandblt1_off
10.71Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
10.71Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
10.71Consensusep_offOrthosteric Ligandep4_off
10.71Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
10.71Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
10.71Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.71Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
10.71Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.71Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
10.53Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
10.53Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
10.34Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
10.34Single4DJHJDTic4DJH-κ-JDTic
10.34Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
10.34Single4U15Tiotropium4U15-M3-Tiotropium
10.34Single5V56TC1145V56-SMO-TC114
10.34Single5V57TC1145V57-SMO-TC114
10.34Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
10.34Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
10.34Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
10.34Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
10.34Single6J20Aprepitant6J20-NK1-Aprepitant
10.34Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
10.34Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
10.34Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.34Single6OL9Tiotropium6OL9-M5-Tiotropium
10.34Single6TQ7SB-3348676TQ7-OX1-SB-334867
10.34Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
10.34Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
10.34Single7FEECP559407FEE-CB1-CP55940-ZCZ011
10.34Single7P2L4YI7P2L-mGlu5-4YI
10.34Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
10.34Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
10.34Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
10.34Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
10.34Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
10.34Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8EA0Iperoxo8EA0-M3-Iperoxo
10.34Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
10.34Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
10.34Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
10.34Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
10.34Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
10.34Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
10.34Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
10.34Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
10.34Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
10.34Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
10.34Single9AS9RS130-1809AS9-5-HT2A-RS130-180
10.34Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
10.34Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
10.34Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
10.34Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
10.34Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
10.34Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.34Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
10.26Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
10.00Single4N4WSANT-14N4W-SMO-SANT-1
10.00Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
10.00Single6ZG4HTL00099366ZG4-M1-HTL0009936
10.00Single7DFPSpiperone7DFP-D2-Spiperone
10.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
10.00Single7K15MKD0467K15-BLT1-MKD046-Na
10.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
10.00Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
10.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
10.00Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
10.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
10.00Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
10.00Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
10.00Single8JWZAB9288JWZ-A2A-AB928-Na
10.00Single8XWACXCL18XWA-CXCR2-CXCL1
10.00Single8XWSCXCL58XWS-CXCR2-CXCL5
10.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
10.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
10.00Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
10.00Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
10.00Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
10.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
10.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
10.00Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
10.00Consensusorexin_onOrthosteric Ligandox2_on
9.68Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
9.68Single5X93K-87945X93-ETB-K-8794
9.68Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
9.68Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
9.68Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.68Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
9.68Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
9.68Single8XVJMacitentan8XVJ-ETA-Macitentan
9.68Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
9.68Single8ZPLHF511168ZPL-CXCR4-HF51116
9.68Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
9.68Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
9.68Consensusendothelin_offOrthosteric Ligandetb_off
9.68Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
9.68Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
9.52Single5MZPCaffeine5MZP-A2A-Caffeine-Na
9.52Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
9.38Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
9.38Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
9.38Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
9.38Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
9.38Single8X5YAstemizole8X5Y-H1-Astemizole
9.38Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
9.09Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
9.09Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
9.09Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
9.09Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.09Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
9.09Single8KIGSHU91198KIG-MC3-SHU9119-Ca
9.09Single8WKYPG-9348WKY-MC4-PG-934
9.09Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
9.09Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
9.09Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
9.09Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
9.09Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.09Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.82Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
8.82Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.82Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
8.82Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
8.82Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
8.82Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
8.70Single3OE8IT1t3OE8-CXCR4-IT1t
8.70Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
8.70Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
8.70Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
8.70Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
8.70Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
8.70Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
8.70Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
8.70Consensussensory_onOrthosteric Ligandopsins_on
8.57Single6W25SHU91196W25-MC4-SHU9119-Ca
8.57Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
8.57Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
8.57Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.57Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.57Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
8.57Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
8.33Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
8.33Single3UZAGTPL92363UZA-A2A-GTPL9236
8.33Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
8.33Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
8.33Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
8.33Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
8.33Single6ME5Agomelatine6ME5-MT1-Agomelatine
8.33Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
8.33Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
8.33Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
8.33Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
8.33Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
8.33Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
8.33Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
8.33Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.33Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
8.33Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
8.33Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
8.33Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
8.33Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
8.33Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
8.33Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
8.33Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.33Consensusgi_sensoryOrthosteric Ligandgi_opsins
8.33Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
8.33Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
8.33Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.33Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.33Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
8.33Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
8.33Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
8.00Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
8.00Single3PBLEticlopride3PBL-D3-Eticlopride
8.00Single5L7IVismodegib5L7I-SMO-Vismodegib
8.00Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
8.00Single6HLLCP999946HLL-NK1-CP99994
8.00Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
8.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
8.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
8.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
8.00Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
8.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
8.00Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
8.00Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
8.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
8.00Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
8.00Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
8.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
8.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
8.00Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.00Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.00Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
8.00Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
8.00Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
8.00Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
8.00Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
8.00Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
8.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
8.00Consensusgq_nucleotideOrthosteric Ligandgq_p2y
8.00Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
8.00Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.69Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
7.69Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
7.69Single4S0VSuvorexant4S0V-OX2-Suvorexant
7.69Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
7.69Single5WS3EMPA5WS3-OX2-EMPA
7.69Single6B73MP11046B73-κ-MP1104
7.69Single6DS0Ly2660976DS0-5-HT2B-Ly266097
7.69Single6ME9Ramelteon6ME9-MT2-Ramelteon
7.69Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
7.69Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
7.69Single6TPJSuvorexant6TPJ-OX2-Suvorexant
7.69Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
7.69Single7F8YDevazepide7F8Y-CCKA-Devazepide
7.69Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
7.69Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.69Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
7.69Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
7.69Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
7.69Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
7.69Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
7.69Single7XRRLemborexant7XRR-OX2-Lemborexant
7.69Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
7.69Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
7.69Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
7.69Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
7.69Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.69Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
7.69Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
7.69Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
7.69Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
7.69Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
7.69Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
7.69Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
7.50Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
7.41Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
7.41Single3RZECidoxepin3RZE-H1-Cidoxepin
7.41Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
7.41Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
7.41Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
7.41Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
7.41Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
7.41Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
7.41Single6TP3Nemorexant6TP3-OX1-Nemorexant
7.41Single6TPKRetosiban6TPK-OT-Retosiban
7.41Single6TPNHTL66416TPN-OX2-HTL6641
7.41Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
7.41Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
7.41Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
7.41Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
7.41Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
7.41Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
7.41Single7VODCariprazine7VOD-5-HT2A-Cariprazine
7.41Single7VV6C48/807VV6-MRGPRX2-C48/80
7.41Single8K2WAMG4878K2W-CXCR3-AMG487
7.41Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
7.41Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
7.41Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
7.41Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
7.41Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
7.41Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
7.41Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
7.41Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
7.41Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
7.41Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
7.41Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
7.41Consensusopsins_offOrthosteric Ligandrhodopsin_off
7.41Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
7.41Consensussensory_offOrthosteric Ligandopsins_off
7.41Consensusvasop-oxy_offOrthosteric Ligandot_off
7.14Single5DHGC-355DHG-NOP-C-35
7.14Single6GPSMK08126GPS-CCR2-MK0812
7.14Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
7.14Single7F83PF-051904577F83-Ghrelin-PF-05190457
7.14Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
7.14Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
7.14Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
7.14Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.14Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
7.14Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
7.14Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
7.14Single8X64Desloratadine8X64-H1-Desloratadine
7.14Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
7.14Single9IYAONO-97105319IYA-GPR55-ONO-9710531
7.14Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
7.14Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
7.14Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
7.14Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
7.14Consensusblt_onOrthosteric Ligandblt1_on
7.14Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
7.14Consensuscck_offOrthosteric Ligandccka_off
7.14Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
7.14Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
7.14Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.14Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.14Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.14Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
7.14Consensusleukotriene_onOrthosteric Ligandblt_on
7.14Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
7.14Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
6.90Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
6.90Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
6.90Single5XPRBosentan5XPR-ETB-Bosentan
6.90Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
6.90Single6GPXMK08126GPX-CCR2-MK0812
6.90Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
6.90Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
6.90Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
6.90Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.90Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
6.90Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.90Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.90Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
6.90Single9HAPTolvaptan9HAP-V2-Tolvaptan
6.90Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
6.67Single5TZRMK86665TZR-FFA1-MK8666
6.67Single6E59L-7607356E59-NK1-L-760735
6.67Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
6.67Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
6.67Single7R0CAVP7R0C-V2-AVP-Arrestin2
6.67Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
6.67Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.67Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
6.67Single8XVLZibotentan8XVL-ETA-Zibotentan
6.67Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
6.67Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
6.67Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
6.67Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
6.67Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
6.67Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Consensustachykinin_offOrthosteric Ligandnk1_off
6.45Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
6.45Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
6.45Single4PY02MeSATP4PY0-P2Y12-2MeSATP
6.45Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
6.45Single5X33BIIL2605X33-BLT1-BIIL260
6.45Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
6.45Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.45Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
6.45Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.45Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
6.45Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
6.45Single9BJKNAM9BJK-μ-Naloxone-NAM
6.25Single6K1QIRL25006K1Q-ETB-IRL2500
6.25Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
6.25Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
6.06Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
6.06Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
6.06Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
6.06Consensuskisspeptin_onOrthosteric Ligandkiss1_on
5.88Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
5.88Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
5.88Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
5.88Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
5.88Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
5.88Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
5.88Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
5.88Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
5.88Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
5.71Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
5.41Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
5.26Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.26Single6D35Cholesterol6D35-SMO-Cholesterol
5.26Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.26Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.26Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
5.26Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
5.26Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
5.26Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
5.26Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
5.26Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
5.26Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
5.26Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
5.26Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
5.26Single7DTTCa7DTT-CaS-Ca-Ca
5.26Single7DTTCa7DTT-CaS-Ca-Ca
5.26Single7DTUTryptophan7DTU-CaS-Tryptophan
5.26Single7DTUTryptophan7DTU-CaS-Tryptophan
5.26Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.26Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.26Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.26Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.26Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.26Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.26Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.26Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.26Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
5.26Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.26Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.26Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.26Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.26Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.26Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.26Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
5.26Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
5.26Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.26Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.26Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.26Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.26Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.26Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.26Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.26Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.26Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.26Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.26Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.26Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.26Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.26Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
5.26Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.26Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.26Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.26Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.26Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.26Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.26Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
5.26Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
5.26Single7XW7K1-707XW7-TSH-K1-70
5.26Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.26Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.26Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.26Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.26Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.26Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.26Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.26Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.26Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.26Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.26Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.26Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.26Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
5.26Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.26Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.26Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.26Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.26Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.26Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.26Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.26Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.26Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.26Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.26Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.26Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.26Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.26Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.26Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
5.26Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.26Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.26Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.26Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.26Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.26Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.26Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.26Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.26Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.26Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.26Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.26Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.26Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.26Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.26Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.26Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.26Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
5.26Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
5.26Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
5.26Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
5.26Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
5.26Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
5.26Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.26Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.26Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.26Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.26Single8WVXNorrin8WVX-LGR4-Norrin
5.26Single8WVYNorrin8WVY-LGR4-Norrin
5.26Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.26Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.26Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.26Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.26Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.26Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.26Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
5.26Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.26Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.26Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.26Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.26Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.26Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.26Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.26Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.26Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.26Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.26Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.26Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.26Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.26Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.26Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.26Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.26Single9KHHNorrin9KHH-LGR4-Norrin
5.26Single9S37NB219S37-LGR4-NB21
5.26Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
5.26Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
5.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.00Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.00Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.00Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
5.00Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.76Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.76Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.76Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.55Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.55Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.55Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.55Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.55Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.35Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
4.35Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
4.35Single5L7DCholesterol5L7D-SMO-Cholesterol
4.35Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
4.35Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.35Single7WC4Serotonin7WC4-5-HT2A-Serotonin
4.35Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.17Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
4.17Single6TQ9SB-4081246TQ9-OX1-SB-408124
4.17Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
4.17Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
4.00Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
4.00Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
4.00Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
4.00Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
4.00Single7WC5Psilocin7WC5-5-HT2A-Psilocin
4.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
4.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
4.00Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
4.00Single8JPSCCL78JPS-ACKR1-CCL7
4.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
4.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
3.85Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
3.85Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
3.85Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
3.85Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
3.85Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
3.85Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
3.85Single6TP4ACT-4622066TP4-OX1-ACT-462206
3.85Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.85Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
3.85Single7UL2SR486927UL2-NTS1-SR48692-Na
3.85Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
3.85Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.85Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
3.85Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.85Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
3.85Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
3.85Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
3.85Consensusneurotensin_offOrthosteric Ligandnts1_off
3.85Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
3.70Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
3.70Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
3.70Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
3.70Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
3.70Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
3.70Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
3.70Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
3.70Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
3.70Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
3.70Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
3.70Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
3.57Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
3.57Single6FFIMMPEP6FFI-mGlu5-MMPEP
3.57Single6IQLL7458706IQL-D4-L745870
3.57Single6ZINSR486926ZIN-NTS1-SR48692
3.57Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
3.57Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
3.57Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
3.57Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
3.57Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
3.57Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.57Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
3.57Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.57Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
3.45Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
3.45Single6FFHFenobam6FFH-mGlu5-Fenobam
3.45Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
3.45Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
3.45Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.45Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
3.45Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
3.33Single4NTJAZD12834NTJ-P2Y12-AZD1283
3.33Single6HLPNetupitant6HLP-NK1-Netupitant
3.33Single6Z4SSR486926Z4S-NTS1-SR48692
3.33Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.33Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
3.33Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
3.33Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
3.33Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
3.23Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.23Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
3.12Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
3.12Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
3.12Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.12Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
3.12Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
3.03Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
3.03Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
3.03Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
2.94Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
2.94Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
2.86Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
2.86Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.86Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.70Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.70Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.63Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.44Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
class-b1_on_gp glucagon_on_gp
vip-pacap_on_gp
pth_on_gp
crf_on_gp
calcitonin_on_gp
class-b2_on_gp adgrg_on_gp
adgrf_on_gp
adgrl_on_gp
adgre_on_gp
adgrd_on_gp
Net Summary
Imin 3.04735
Number of Linked Nodes 1061
Number of Links 1215
Number of Hubs 169
Number of Links mediated by Hubs 703
Number of Communities 17
Number of Nodes involved in Communities 195
Number of Links involved in Communities 284
Path Summary
Number Of Nodes in MetaPath 153
Number Of Links MetaPath 152
Number of Shortest Paths 4037629
Length Of Smallest Path 3
Average Path Length 40.4594
Length of Longest Path 90
Minimum Path Strength 0.121796
Average Path Strength 5.59812
Maximum Path Strength 21.8798
Minimum Path Correlation 0.701146
Average Path Correlation 0.964209
Maximum Path Correlation 0.997885
Minimum % Of Corr. Nodes 1.21951
Average % Of Corr. Nodes 25.814
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 50.8642
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .




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