Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1NT 6.123161215
21x39 3.95048407
31x59 2.21082405
41x60 1.92086605
52x40 2.55354408
62x41 2.20109405
72x42 4.21967507
82x46 4.22173419
92x50 5.69005519
102x53 3.41827407
11E1x50 6.39957418
12E1x52 4.17206407
133x30 2.84409406
143x50 5.47835519
15E2 8.567862214
165x47 5.50372408
175x58 4.70644619
185x62 2.30902405
196x32 1.28022407
206x44 4.56969419
216x48 6.27675518
226x49 2.79511406
236x51 4.38596516
246x59 2.1241404
25E3 2.62253812
267x34 3.36546414
277x38 3.948415
287x42 3.81502517
297x49 4.82081519
307x52 2.66031418
317x53 4.71464619
328x50 3.42634508
338x54 1.5864406
34Lig 7.62191910
35G.HN.33 2.21647404
36G.hns1.03 1.38244404
37G.S1.06 4.372134169
38G.s1h1.04 1.59042409
39G.H1.01 2.989485169
40G.S2.03 4.20941529
41G.S2.04 1.66407
42G.S2.06 4.55596508
43G.S2.08 4.927625105
44G.S3.03 6.578095147
45G.S3.04 8.19242427
46G.S3.06 7.44267526
47G.S3.07 3.022385169
48G.H2.03 4.25672429
49G.H2.06 4.83526729
50G.H2.07 5.01868629
51G.h2s4.01 6.19099529
52G.S4.04 5.45931409
53G.s4h3.04 4.94777678
54G.H3.01 4.07323509
55G.H3.09 4.89769769
56G.H3.13 3.78316665
57G.H3.14 4.23695408
58G.H3.17 6.63089624
59G.H3.18 5.551054159
60G.S5.04 3.93168469
61G.S5.05 3.137678179
62G.S5.07 3.76808409
63G.s5hg.01 3.59664479
64G.HG.04 5.08691409
65G.HG.13 2.32356476
66G.HG.14 2.75588405
67G.hgh4.02 4.805666189
68G.hgh4.05 8.39257407
69G.hgh4.08 2.689324193
70G.H4.05 2.984755194
71G.H4.10 8.455324187
72G.H4.13 0.853327403
73G.H4.15 5.41078468
74G.H4.16 2.58271563
75G.h4s6.02 4.13377467
76G.S6.02 4.831457138
77G.S6.05 4.41383505
78G.H5.03 3.499825178
79G.H5.08 5.696814108
80G.H5.17 2.42192506
81G.H5.20 3.10654408
82G.H5.26 3.30438605
83b.1x1 1.16612504
84b.1x3 1.16017401
85b.1x4 1.80309408
86b.1x11 2.17143508
87b.lh12x2 3.75808408
88b.h2x1 3.02802505
89b.lhb1x3 2.71578502
90b.lhb1x11 3.14604404
91b.b1x4 3.39363437
92b.b1x6 7.3881439
93b.l1x3 7.92191639
94b.b2x1 7.35114528
95b.b2x5 6.14722607
96b.b3x3 3.37994558
97b.l3x2 5.39565539
98b.b4x2 4.86139408
99b.b4x3 4.6181457
100b.b4x5 3.9595457
101b.b4x6 8.52214739
102b.l4x2 9.69454434
103b.b5x2 5.5192407
104b.b5x3 6.22979639
105b.b5x5 4.97372455
106b.b5x7 5.61158407
107b.l5x1 4.03251558
108b.l5x5 6.94268729
109b.b6x5 3.83676756
110b.l6x5 5.738474114
111b.b7x1 5.447255114
112b.b7x4 3.74498458
113b.l7x4 3.51591409
114b.b8x3 3.43463406
115b.b8x4 5.07971556
116b.l8x1 3.3952455
117b.l8x3 3.11636403
118b.b9x3 4.31554456
119b.l9x3 7.20166529
120b.l9x6 4.89388828
121b.b10x5 4.23059609
122b.b11x4 5.47753429
123b.l11x2 7.6186429
124b.b12x6 7.70879728
125b.b12x7 5.02267449
126b.b13x7 7.601547
127b.l13x3 7.42426649
128b.l13x6 4.97826429
129b.l13x7 4.43961449
130b.b14x3 4.31319445
131b.b15x1 6.36672549
132b.b15x2 6.22711426
133b.b15x3 4.41165449
134b.l15x1 5.22788427
135b.l15x2 5.25634549
136b.b16x4 10.4703446
137b.b16x5 4.42591405
138b.b16x6 8.31749648
139b.b17x5 7.00055427
140b.b17x7 8.24556428
141b.l17x3 8.64506629
142b.l17x6 6.23835529
143b.b18x3 4.78756428
144b.b18x5 4.8607405
145b.l18x1 5.28534896
146b.l18x2 5.25101497
147b.l18x3 6.51512495
148b.b19x2 7.34653526
149b.b19x4 5.89308428
150b.l19x2 6.21649529
151b.b20x4 9.96912528
152b.b20x6 7.40143526
153b.l20x2 4.1908609
154b.b21x1 6.9481527
155b.b21x2 3.05636406
156b.b21x5 5.0009404
157b.b21x7 5.60952605
158b.l21x2 4.71245404
159b.b22x5 5.37843597
160b.l22x5 5.612726209
161b.b23x6 6.940686127
162b.l23x1 7.2395426
163b.b24x4 7.457884126
164b.b24x6 6.547984128
165b.l24x2 3.41278506
166b.l24x3 4.43824405
167b.l25x3 8.45018589
168b.l25x6 12.0243428
169b.l26x5 4.43475405
170b.l27x1 10.0547729
171b.l27x2 7.94755489
172b.b28x2 4.45167404
173b.b28x3 3.92809537
174b.b28x4 7.52114486
175b.b28x6 8.2851589
176g.h2x5 1.2953405
177g.h2x11 7.86066499
178g.ctx3 6.04362404
179g.ctx6 2.95738405
180G.HN.11 0.994645600
181g.h1x1 1.00976600
182g.l1x4 3.50673500
183g.ctx14 4.50518430
184g.ctx15 5.44306430
185g.ctx16 3.99126830
186E1 0.423305500
187G.HN.29 0.205158400
188G.hgh4.13 0.14438400
189H.HA.16 0.0695807400
190H.HA.26 0.0813967400
191H.hahb.06 0.0846972400
192H.HB.02 0.0883463400
193H.HB.10 0.070955400
194H.HD.07 0.0934592500
195H.HE.02 0.0652575400
196H.HE.05 0.0654878400
197H.hehf.04 0.109597400
198H.HF.03 0.127776400
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1Lig NT 11.06194.13514YesYes105
22x42 3x49 10.30566.57408YesNo078
32x42 3x46 11.69433.74744YesNo079
47x49 7x53 32.18812.88YesYes199
57x45 7x49 22.16796.19735NoYes099
66x48 7x45 21.81688.33812YesNo089
73x36 6x48 42.87393.69395NoYes178
83x36 Lig 42.55344.50252NoYes170
96x44 6x48 21.76436.54846YesYes198
103x50 5x58 28.68685.17836YesYes199
115x54 5x58 25.8172.99235NoYes189
125x54 6x44 25.64264.24722NoYes189
133x50 7x53 35.59145.35579YesYes199
143x50 G.H5.25 78.33376.91573YesNo097
15G.H5.20 G.H5.25 78.50663.22294YesNo087
16G.S6.02 G.h4s6.12 42.90728.24416YesNo084
17G.H5.17 G.h4s6.12 42.67993.02642YesNo064
18G.H5.17 G.H5.26 84.61292.45894YesYes065
19G.H5.20 G.H5.26 82.62513.29696YesYes085
20G.H5.13 G.S6.02 43.02366.7442NoYes078
21G.H5.13 G.H5.17 42.68544.4844NoYes076
22b.b3x2 b.b4x6 17.38484.72526NoYes059
23b.b2x5 b.b3x2 17.61259.48354YesNo075
24b.b2x3 b.b2x5 44.96174.08209NoYes067
25b.b26x2 b.b2x3 45.18745.23871NoNo076
26b.b26x1 b.b26x2 45.41332.90047NoNo097
27b.b26x1 b.l27x1 45.63925.37968NoYes099
28b.b2x1 b.l27x1 24.18147.48204YesYes289
29b.b2x1 b.l3x1 24.538114.423YesNo289
30b.l3x1 b.l5x5 24.76616.48982NoYes299
31G.h2s4.01 b.l5x5 24.956210.1038YesYes299
32G.S1.05 G.h2s4.01 26.174811.0661NoYes099
33G.S1.05 G.S1.07 67.25685.53081NoNo099
34G.S1.07 G.S4.04 67.46742.90524NoYes099
35G.S4.04 G.S4.06 28.33582.87049YesNo097
36G.H4.15 G.S4.06 28.41386.39705YesNo087
37G.H3.06 G.H4.15 57.05875.46565NoYes068
38G.H3.06 G.hgh4.02 86.03143.67784NoYes069
39G.hgh4.01 G.hgh4.02 42.65478.11802NoYes059
40G.hgh4.01 G.s4h3.04 42.63784.40362NoYes058
41G.HG.07 G.s4h3.04 99.89055.47117NoYes798
42G.HG.07 G.s4h3.02 1002.42805NoNo799
43G.s4h3.02 G.s5hg.01 99.92933.54635NoYes799
44G.S5.07 G.s5hg.01 99.45022.8847YesYes099
45G.H1.04 G.S5.07 49.49033.48338NoYes079
46G.H1.04 G.S5.05 49.38372.98223NoYes079
47G.S5.03 G.S5.05 86.70663.50169NoYes099
48G.H5.10 G.S5.03 86.54434.69105NoNo069
49G.H5.10 G.S6.02 86.46317.06422NoYes068
50G.H3.17 b.l27x1 22.79293.09082YesYes249
51G.H3.15 G.H3.17 40.45114.64073NoYes084
52G.H3.15 G.H3.18 40.56185.51293NoYes089
53G.H3.18 G.S4.02 40.7816.57107YesNo1598
54G.S1.05 G.S4.02 41.00523.61038NoNo098
55G.H3.09 G.S4.04 70.92811.0729YesYes099
56G.H3.09 G.H4.15 28.62365.57983YesYes698
57G.H3.09 G.h4s6.01 28.62963.26466YesNo094
58G.H3.06 G.h4s6.01 28.95953.02304NoNo064
59G.HG.15 G.hgh4.02 43.0223.10402NoYes079
60G.HG.15 G.s4h3.04 42.93843.85228NoYes078
61G.H3.09 G.S5.04 14.29173.31161YesYes699
62G.S5.04 G.S5.06 14.363.61102YesNo098
63G.S5.06 G.s4h3.01 14.59496.03802NoNo087
64G.HG.04 G.s4h3.01 14.61428.19881YesNo097
65G.HG.04 G.s4h3.04 14.64315.06986YesYes098
66G.S5.07 G.s6h5.01 49.87646.31099YesNo099
67G.S5.05 G.s6h5.01 49.36814.85278YesNo1799
68G.S4.03 G.S5.05 13.31252.9739NoYes079
69G.S1.06 G.S4.03 10.59563.02229YesNo097
70G.H2.04 G.H2.07 31.42085.10819NoYes099
71G.H2.04 G.H3.08 31.58584.94761NoNo099
72G.H3.08 G.S4.04 31.69224.98861NoYes099
73G.H2.07 b.l9x6 31.73223.8366YesYes298
74G.H2.06 b.l9x6 24.97553.49987YesYes298
75G.H2.06 b.l17x6 24.16527.76438YesYes299
76b.l17x5 b.l17x6 24.05482.99688NoYes269
77b.l17x5 b.l19x2 23.9424.06153NoYes269
78b.l17x3 b.l19x2 16.43164.12217YesYes299
79b.b17x7 b.b20x6 18.68279.87499YesYes286
80b.b17x7 b.b21x1 17.63345.09138YesYes287
81b.1x19 b.b21x1 15.45427.65861NoYes067
82b.1x15 b.1x19 13.8343.82622NoNo076
83b.1x12 b.1x15 13.13131.75666NoNo067
84b.b20x4 b.b20x6 13.15694.22924YesYes286
85G.H3.17 b.l25x6 17.11585.84493YesYes248
86b.l23x1 b.l25x6 12.663118.3376YesYes268
87b.l21x7 b.l23x1 12.44964.40267NoYes056
88b.l21x7 b.l23x2 12.21766.51622NoNo058
89b.b23x6 b.l23x2 11.7533.80838YesNo078
90b.b23x6 b.b24x6 10.35646.68438YesYes1278
91b.b21x7 b.b24x6 10.13899.03457YesYes058
92b.b2x5 b.l4x1 21.64095.34984YesNo075
93b.l4x1 g.ctx16 21.41543.84668NoYes050
94b.l4x2 g.ctx16 17.07675.47037YesYes340
95b.l2x5 b.l4x2 16.830724.2267NoYes054
96b.l2x3 b.l2x5 16.1332.94035NoNo085
97b.b3x1 b.l2x3 15.90535.08359NoNo058
98b.b3x1 b.b6x5 15.67764.17053NoYes056
99b.b2x4 b.b6x5 12.62482.94971NoYes066
100b.b10x4 b.b2x4 12.395611.874NoNo066
101b.1x12 g.h1x11 10.67152.31756NoNo060
102E2 Lig 17.18739.56231YesYes140
1033x46 3x50 11.78474.55581NoYes199
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
NTNT21.75921YesYes5511
E2NT14.23511YesYes4511
1x397x423.640460YesYes7721
2x577x424.977090NoYes7721
3x25E22.787151NoYes9421
3x26E22.794221NoYes7421
3x32Lig5.732581NoYes5010
3x334x573.769721NoNo4712
3x33Lig6.120321NoYes4010
3x366x483.693951NoYes7812
3x36Lig4.502521NoYes7010
4x60E24.347321NoYes5421
4x605x395.707271NoNo5622
5x39E26.812241NoYes6421
5x36E28.713610NoYes4421
E2E251.56021YesYes4411
E2E2x525.455041YesNo4411
E2E2x518.132191YesNo4511
E2x52Lig6.361551NoYes4010
E2Lig9.562311YesYes4010
5x395x434.841011NoNo6521
5x43Lig4.145561NoYes5010
6x517x373.32291YesNo6612
6x517x382.963011YesYes6511
6x51Lig6.927941YesYes6010
6x547x343.468650NoYes5421
6x55Lig3.109251NoYes5010
6x587x343.156831NoYes4411
E3E34.497191YesYes2222
7x42Lig4.495931YesYes7010
2x537x423.109430YesYes7721
2x603x282.846931NoNo7512
3x223x262.864221NoNo3722
3x22E25.914931NoYes3421
3x375x433.678290NoNo6521
5x406x553.485810NoNo4521
6x547x373.530230NoNo5622
2x60Lig4.152481NoYes7010
2x64Lig2.791560NoYes5010
3x29Lig2.955341NoYes5010
7x38Lig6.796511YesYes5010
2x533x322.858570YesNo7521
2x563x323.792840NoNo6521
3x294x653.926481NoNo5012
4x64E26.784521NoYes0421
6x516x523.526841YesNo6712
6x516x555.189111YesNo6511
7x347x383.180281YesYes4511
7x387x422.852221YesYes5711
7x34Lig3.656081YesYes4010
E1x49E22.82031NoYes4421
E2x51Lig4.397331NoYes5010
6x58Lig2.90741NoYes4010
LigNT4.135141YesYes0501
E3NT2.577971YesYes2521
5x35E22.500661NoYes3421
7x31NT2.279220NoYes3521
1x32NT2.037481NoYes5521
6x587x301.823261NoNo4412
7x28NT1.739861NoYes0521
7x32NT1.678421NoYes1521
5x38E21.649120NoYes4421
6x62E21.224641NoYes0421
5x32E21.195521NoYes0421
7x24NT0.8674050NoYes0521
4x68E20.328780NoYes0421
E1x501NT0.2930320NoYes0521
E1x48NT0.1157861NoYes0521
5x27E20.0560871NoYes0421
5x28E20.03682191NoYes0421
3x29Ca50.0356461NoNo5012
4x69E20.02181550NoYes0421

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
88.24Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
85.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
73.91Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
70.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
69.57Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
66.67Single8E0GBU728E0G-μ-BU72
66.67Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
66.67Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
65.22Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
63.16Single4RWADIPP-NH24RWA-δ-DIPP-NH2
63.16Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
61.90Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
61.90Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
61.11Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
61.11Single5C1MBU725C1M-μ-BU72
61.11Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
61.11Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
61.11Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
60.87Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
60.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
59.09Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
59.09Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
58.82Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
58.82Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
58.82Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
58.82Consensushca_onOrthosteric Ligandhca2_on
58.33Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
58.33Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
58.33Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
58.33Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
57.89Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
57.89Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
57.89Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
57.89Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
57.89Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
57.89Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
57.89Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
57.89Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
57.14Single4UG2CGS216804UG2-A2A-CGS21680
57.14Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
57.14Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
57.14Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
56.52Consensusangiotensin_onOrthosteric Ligandat1_on
56.52Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
56.52Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
56.52Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
56.52Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
56.00Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
55.56Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
55.56Single7UL4Alvimopan7UL4-μ-Alvimopan
55.56Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
55.56Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
55.56Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
55.56Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
55.56Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
55.56Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
55.56Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
55.56Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
55.56Consensusa3_onOrthosteric Liganda3a_on
55.56Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
55.56Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
55.56Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
55.56Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
55.56Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
55.56Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
55.56Consensushca_on_gpOrthosteric Ligandhca2_on_gp
55.56Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
55.00Single6MXTSalmeterol6MXT-β2-Salmeterol
55.00Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
55.00Single7YITNalfurafine7YIT-κ-Nalfurafine
55.00Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
55.00Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
55.00Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
55.00Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
55.00Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
55.00Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
55.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
55.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
55.00Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
55.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
55.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
54.55Single4IARErgotamine4IAR-5-HT1B-Ergotamine
54.55Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
54.55Single8WDTphotoNECA8WDT-A2A-photoNECA
54.55Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
54.55Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
54.55Consensuslpl_onOrthosteric Ligands1p_on lpa_on
54.55Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
54.55Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
54.55Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
54.17Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
54.17Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
54.17Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
54.17Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
54.17Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
54.17Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
54.17Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
53.85Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
53.85Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
52.94Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
52.94Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
52.94Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
52.94Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
52.94Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
52.94Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
52.63Single7C61Ergotamine7C61-5-HT1B-Ergotamine
52.63Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
52.63Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
52.63Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
52.63Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
52.63Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
52.63Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
52.63Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
52.63Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
52.63Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
52.63Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
52.63Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
52.63Single8S4DCMF-0198S4D-Apelin-CMF-019
52.63Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
52.63Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
52.63Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
52.63Consensusa3_on_gpOrthosteric Liganda3a_on_gp
52.63Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
52.63Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
52.63Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
52.63Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
52.63Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
52.63Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
52.63Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
52.63Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
52.38Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
52.38Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
52.38Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
52.38Single7EZCUKA7EZC-A2A-UKA
52.38Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
52.38Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
52.38Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
52.38Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
52.38Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
52.38Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
52.38Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
52.17Single3QAKUK-4320973QAK-A2A-UK-432097
52.17Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
52.17Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
52.17Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
52.17Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
52.17Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
52.17Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
52.00Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
52.00Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
51.85Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
51.85Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
51.85Consensusbradykinin_onOrthosteric Ligandbk2_on
51.85Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
51.85Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
51.72Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
50.00Single2YDVNECA2YDV-A2A-NECA
50.00Single3NY9ICI118-5513NY9-β2-ICI118-551
50.00Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
50.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
50.00Single4UHRCGS216804UHR-A2A-CGS21680
50.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
50.00Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
50.00Single5G53NECA5G53-A2A-NECA-Gs
50.00Single5GLHEndothelin-15GLH-ETB-Endothelin-1
50.00Single5WF5UK-4320975WF5-A2A-UK-432097
50.00Single5WF6UK-4320975WF6-A2A-UK-432097
50.00Single5ZTYAM102575ZTY-CB2-AM10257
50.00Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
50.00Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
50.00Single6H7JIsoprenaline6H7J-β1-Isoprenaline
50.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
50.00Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
50.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
50.00Single6PS4ICI118-5516PS4-β2-ICI118-551
50.00Single6TPGEMPA6TPG-OX2-EMPA
50.00Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
50.00Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
50.00Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
50.00Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
50.00Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
50.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
50.00Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
50.00Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
50.00Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
50.00Single7XN9L-054,5227XN9-SST2-L-054,522
50.00Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
50.00Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
50.00Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
50.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
50.00Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
50.00Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
50.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
50.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
50.00Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
50.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
50.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
50.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
50.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
50.00Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
50.00Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
50.00Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
50.00Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
50.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
50.00Single8K5CAcipimox8K5C-HCA2-Acipimox
50.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
50.00Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
50.00Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
50.00Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
50.00Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
50.00Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
50.00Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
50.00Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
50.00Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
50.00Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
50.00Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
50.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
50.00Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
50.00Consensusa2_onOrthosteric Liganda2b_on
50.00Consensusa2_on_gpOrthosteric Liganda2b_on_gp
50.00Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
50.00Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
50.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
50.00Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
50.00Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
50.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
50.00Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
50.00Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
50.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
50.00Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
50.00Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
50.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
50.00Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
50.00Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
50.00Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
50.00Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
50.00Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
50.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
50.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
50.00Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
50.00Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
48.15Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
48.15Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
48.15Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
48.15Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
48.15Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
48.15Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
48.00Single6JODAngiotensin II6JOD-AT2-Angiotensin II
48.00Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
48.00Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
48.00Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
48.00Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
48.00Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
47.83Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
47.83Single4XT1Fractalkine4XT1-US28-Fractalkine
47.83Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
47.83Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
47.83Single7F8XNN90567F8X-CCKA-NN9056
47.83Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
47.83Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
47.83Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
47.83Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
47.83Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
47.83Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
47.83Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
47.83Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
47.83Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
47.83Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
47.62Single4AMIBucindolol4AMI-β1-Bucindolol
47.62Single4LDEBI1671074LDE-β2-BI167107
47.62Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
47.62Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
47.62Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
47.62Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
47.62Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
47.62Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
47.62Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
47.62Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
47.62Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
47.62Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
47.62Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
47.62Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
47.62Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
47.62Single8JJ8Formoterol8JJ8-β2-Formoterol
47.62Single8JJLOlodaterol8JJL-β2-Olodaterol
47.62Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
47.62Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
47.62Single8XYIVUF106618XYI-CXCR3-VUF10661
47.62Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
47.62Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
47.62Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
47.62Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
47.62Consensusalpha1_offOrthosteric Ligandalpha1a_off
47.62Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
47.62Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
47.62Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
47.62Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
47.62Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
47.62Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
47.62Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
47.62Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
47.62Consensuslpa_offOrthosteric Ligandlpa1_off
47.62Consensuslpl_offOrthosteric Ligands1p_off lpa_off
47.62Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
47.62Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
47.62Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
47.37Single2Y04Salbutamol2Y04-β1-Salbutamol
47.37Single3NY8ICI118-5513NY8-β2-ICI118-551
47.37Single4EJ4Naltrindole4EJ4-δ-Naltrindole
47.37Single4GBRS-Carazolol4GBR-β2-S-Carazolol
47.37Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
47.37Single6PS1Timolol6PS1-β2-Timolol
47.37Single6TOTLemborexant6TOT-OX1-Lemborexant
47.37Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
47.37Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
47.37Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
47.37Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
47.37Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
47.37Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
47.37Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
47.37Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
47.37Single7V3ZCP559407V3Z-CB1-CP55940
47.37Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
47.37Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
47.37Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
47.37Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
47.37Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
47.37Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
47.37Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
47.37Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
47.37Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
47.37Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
47.37Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
47.37Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
47.37Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
47.37Single8K5DGSK2560738K5D-HCA2-GSK256073
47.37Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
47.37Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
47.37Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.37Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
47.37Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
47.37Single9CHXS-Carazolol9CHX-β2-S-Carazolol
47.37Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
47.37Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
47.37Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
47.37Consensusdopamine_offOrthosteric Ligandd2_off d3_off
47.37Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
47.37Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
47.37Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
47.37Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
47.06Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
47.06Single8K5BNiacin8K5B-HCA2-Niacin
47.06Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
47.06Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
47.06Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
46.67Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
46.43Single6IGLIRL16206IGL-ETB-IRL1620
46.43Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
46.15Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
46.15Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
46.15Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
46.15Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
46.15Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
46.15Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
45.83Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
45.83Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
45.83Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
45.83Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
45.83Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
45.83Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
45.83Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
45.83Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
45.83Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
45.83Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
45.83Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
45.83Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
45.83Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
45.83Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
45.45Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
45.45Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
45.45Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
45.45Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
45.45Single5X93K-87945X93-ETB-K-8794
45.45Single6IBLArformoterol6IBL-β1-Arformoterol
45.45Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
45.45Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
45.45Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
45.45Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
45.45Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
45.45Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
45.45Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
45.45Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
45.45Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
45.45Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
45.45Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
45.45Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
45.45Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
45.45Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
45.45Consensuscck_onOrthosteric Ligandccka_on cckb_on
45.45Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
45.45Consensusendothelin_offOrthosteric Ligandetb_off
45.45Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
45.45Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
45.45Consensusprostanoid_offOrthosteric Ligandep_off dp_off
45.00Single2RH1S-Carazolol2RH1-β2-S-Carazolol
45.00Single2Y03Isoprenaline2Y03-β1-Isoprenaline
45.00Single2YCWS-Carazolol2YCW-β1-S-Carazolol
45.00Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
45.00Single5D6LS-Carazolol5D6L-β2-S-Carazolol
45.00Single5JQHS-Carazolol5JQH-β2-S-Carazolol
45.00Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
45.00Single5WQCEMPA5WQC-OX2-EMPA
45.00Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
45.00Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
45.00Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
45.00Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
45.00Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
45.00Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
45.00Single6TP6Filorexant6TP6-OX1-Filorexant
45.00Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
45.00Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
45.00Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
45.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
45.00Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
45.00Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
45.00Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
45.00Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
45.00Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
45.00Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
45.00Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
45.00Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
45.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
45.00Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
45.00Single8JXSPF-61428JXS-D1-PF-6142
45.00Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
45.00Single8TF5Oleic acid8TF5-GPR6-Oleic acid
45.00Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
45.00Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
45.00Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
45.00Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
45.00Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
45.00Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
45.00Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
45.00Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
45.00Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
45.00Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
45.00Consensusamine_offonOrthosteric Ligandamine_off amine_on
45.00Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
45.00Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
45.00Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
45.00Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
45.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
45.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
45.00Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
45.00Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
45.00Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
45.00Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
45.00Consensustrace-amine_onOrthosteric Ligandta1_on
44.83Single6IGKEndothelin-36IGK-ETB-Endothelin-3
44.83Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
44.83Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
44.83Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
44.83Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
44.44Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
44.44Single5WS3EMPA5WS3-OX2-EMPA
44.44Single6AKXA4R6AKX-CCR5-A4R
44.44Single6B73MP11046B73-κ-MP1104
44.44Single6TODEMPA6TOD-OX1-EMPA-Na
44.44Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
44.44Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
44.44Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
44.44Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
44.44Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
44.44Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
44.44Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
44.44Single8GNGIstradefylline8GNG-A2A-Istradefylline
44.44Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
44.44Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
44.44Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
44.44Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
44.44Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
44.44Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
44.44Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
44.44Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
44.44Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
44.44Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
44.44Consensusalpha2_offOrthosteric Ligandalpha2c_off
44.44Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
44.44Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
44.44Consensusorexin_offOrthosteric Ligandox2_off ox1_off
44.44Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
44.44Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
44.44Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
44.44Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
44.00Single6PT2KGCHM076PT2-δ-KGCHM07
44.00Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
44.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
44.00Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
44.00Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
44.00Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
44.00Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
44.00Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
44.00Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
44.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
44.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
43.48Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
43.48Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
43.48Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
43.48Single6PT3DPI-2876PT3-δ-DPI-287
43.48Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
43.48Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
43.48Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
43.48Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
43.48Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
43.48Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
43.48Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
43.48Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
43.33Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
43.33Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
42.86Single3P0GBI1671073P0G-β2-BI167107
42.86Single4DJHJDTic4DJH-κ-JDTic
42.86Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
42.86Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
42.86Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
42.86Single5D5AS-Carazolol5D5A-β2-S-Carazolol
42.86Single5D5BS-Carazolol5D5B-β2-S-Carazolol
42.86Single5XR8AM8415XR8-CB1-AM841
42.86Single5XRAAM115425XRA-CB1-AM11542
42.86Single6J21Aprepitant6J21-NK1-Aprepitant
42.86Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
42.86Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
42.86Single6TQ7SB-3348676TQ7-OX1-SB-334867
42.86Single6WGTLSD6WGT-5-HT2A-LSD
42.86Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
42.86Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
42.86Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
42.86Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
42.86Single7FEECP559407FEE-CB1-CP55940-ZCZ011
42.86Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
42.86Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
42.86Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
42.86Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
42.86Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
42.86Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
42.86Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
42.86Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
42.86Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
42.86Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
42.86Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
42.86Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
42.86Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
42.86Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
42.86Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
42.86Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
42.86Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
42.86Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
42.86Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
42.86Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
42.86Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
42.86Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
42.86Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.86Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
42.86Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
42.86Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
42.86Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
42.86Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
42.86Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
42.86Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
42.86Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
42.86Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
42.86Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
42.86Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
42.86Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
42.86Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
42.31Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
42.31Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
42.31Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
42.31Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
42.31Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
42.31Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.31Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
42.31Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
42.31Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
42.31Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
42.31Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
42.31Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
42.31Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
42.31Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
42.31Consensusvasop-oxy_onOrthosteric Ligandv2_on
42.31Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
42.11Single2YDOAdenosine2YDO-A2A-Adenosine
42.11Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
42.11Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
42.11Single4MBSMaraviroc4MBS-CCR5-Maraviroc
42.11Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
42.11Single6KUXRS-799486KUX-α2a-RS-79948
42.11Single6PS5S-Propranolol6PS5-β2-S-Propranolol
42.11Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
42.11Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
42.11Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
42.11Single6V9SGTPL114036V9S-OX1-GTPL11403
42.11Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
42.11Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
42.11Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
42.11Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
42.11Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
42.11Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
42.11Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
42.11Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.11Single7UL3Famotidine7UL3-H2-Famotidine
42.11Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
42.11Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
42.11Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
42.11Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
42.11Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
42.11Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
42.11Single8IHKAcifran8IHK-HCA3-Acifran
42.11Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
42.11Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
42.11Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
42.11Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.11Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
42.11Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
42.11Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
42.11Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
42.11Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
42.11Consensusalpha1_onOrthosteric Ligandalpha1a_on
42.11Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
42.11Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
42.11Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
42.11Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
42.11Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
42.11Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
41.67Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
41.67Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
41.67Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
41.67Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
41.67Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
41.67Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
41.67Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
41.67Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
41.67Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
41.67Single8WKYPG-9348WKY-MC4-PG-934
41.67Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
41.67Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
41.67Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
41.67Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
41.67Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
41.67Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.38Consensusendothelin_onOrthosteric Ligandetb_on eta_on
41.38Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
41.18Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
41.18Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
41.18Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
41.18Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
40.91Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
40.91Single3D4STimolol3D4S-β2-Timolol
40.91Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
40.91Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
40.91Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
40.91Single6A93Risperidone6A93-5-HT2A-Risperidone
40.91Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
40.91Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
40.91Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
40.91Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
40.91Single6KQICP559406KQI-CB1-CP55940-Org27569
40.91Single7DFPSpiperone7DFP-D2-Spiperone
40.91Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
40.91Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
40.91Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
40.91Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
40.91Single7K15MKD0467K15-BLT1-MKD046-Na
40.91Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
40.91Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
40.91Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
40.91Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
40.91Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
40.91Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
40.91Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
40.91Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.91Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
40.91Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
40.91Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
40.91Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
40.91Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
40.91Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
40.91Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
40.91Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
40.91Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
40.91Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
40.91Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
40.91Consensusorexin_onOrthosteric Ligandox2_on
40.91Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
40.74Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
40.74Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
40.74Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
40.74Single8ZRTET-18ZRT-ETB-ET-1
40.74Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
40.74Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
40.74Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
40.74Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
40.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
40.00Single2Y02Carmoterol2Y02-β1-Carmoterol
40.00Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
40.00Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
40.00Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
40.00Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
40.00Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
40.00Single4QKX35V4QKX-β2-35V
40.00Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
40.00Single4YAYZD-71554YAY-AT1-ZD-7155
40.00Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
40.00Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
40.00Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
40.00Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
40.00Single6H7MSalbutamol6H7M-β1-Salbutamol
40.00Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
40.00Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
40.00Single7BU7BI1671077BU7-β1-BI167107
40.00Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
40.00Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
40.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
40.00Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
40.00Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
40.00Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
40.00Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
40.00Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
40.00Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
40.00Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
40.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
40.00Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
40.00Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
40.00Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
40.00Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
40.00Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
40.00Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
40.00Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
40.00Single8JJOAlprenolol8JJO-β2-Alprenolol
40.00Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
40.00Single8JXRLSD8JXR-D1-LSD
40.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
40.00Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
40.00Single8T1WCVN4248T1W-GPR6-CVN424
40.00Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
40.00Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
40.00Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
40.00Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
40.00Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
40.00Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
40.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
40.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
40.00Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
40.00Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
40.00Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
40.00Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
40.00Consensus5ht5_onOrthosteric Ligand5ht5a_on
40.00Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
40.00Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
40.00Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
40.00Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
40.00Consensusbombesin_onOrthosteric Ligandbb2_on
40.00Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
40.00Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
40.00Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
40.00Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
40.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
40.00Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
40.00Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
40.00Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
40.00Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
39.29Single4XT3Fractalkine4XT3-US28-Fractalkine
39.29Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
39.29Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
39.29Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
39.13Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
39.13Single6H7LDobutamine6H7L-β1-Dobutamine
39.13Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
39.13Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
39.13Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
39.13Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Single7UM4AS26747237UM4-5-HT5A-AS2674723
39.13Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
39.13Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
39.13Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
39.13Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
39.13Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
39.13Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
39.13Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
39.13Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
39.13Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
39.13Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
39.13Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
39.13Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
39.13Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
39.13Consensuschemerin_onOrthosteric Ligandcml1_on
39.13Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
39.13Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
38.89Single3OE9IT1t3OE9-CXCR4-IT1t
38.89Single3PBLEticlopride3PBL-D3-Eticlopride
38.89Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
38.89Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
38.89Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
38.89Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
38.89Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
38.89Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
38.89Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
38.89Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
38.89Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
38.89Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
38.89Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
38.89Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
38.89Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
38.89Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
38.89Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
38.71Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
38.46Single3OE0CVX153OE0-CXCR4-CVX15
38.46Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
38.46Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
38.46Single6W25SHU91196W25-MC4-SHU9119-Ca
38.46Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
38.24Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
38.24Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
38.10Single5N2RPSB-365N2R-A2A-PSB-36-Na
38.10Single5N2SPSB365N2S-A1-PSB36
38.10Single5TVNLSD5TVN-5-HT2B-LSD
38.10Single5WIUNemonapride5WIU-D4-Nemonapride
38.10Single5WIVNemonapride5WIV-D4-Nemonapride-Na
38.10Single6D26Fevipiprant6D26-DP2-Fevipiprant
38.10Single6E67BI1671076E67-β2-BI167107-Gs (fused)
38.10Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
38.10Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
38.10Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
38.10Single6PS6Timolol6PS6-β2-Timolol
38.10Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
38.10Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
38.10Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
38.10Single7C4SS1P7C4S-S1P3-S1P
38.10Single7WC6LSD7WC6-5-HT2A-LSD
38.10Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.10Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
38.10Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
38.10Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
38.10Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
38.10Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
38.10Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
38.10Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
38.10Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
38.10Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
38.10Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
38.10Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
38.10Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
38.10Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
38.10Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
38.10Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
38.10Consensusdp_offOrthosteric Liganddp2_off
38.10Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
38.10Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
38.10Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
38.10Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
37.93Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.93Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
37.50Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
37.50Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
37.50Single7SK9CCX6627SK9-ACKR3-CCX662
37.50Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
37.50Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
37.50Single8X5YAstemizole8X5Y-H1-Astemizole
37.50Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
37.04Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
37.04Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
37.04Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
37.04Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
37.04Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
37.04Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
37.04Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
36.84Single3PWHZM-2413853PWH-A2A-ZM-241385
36.84Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
36.84Single4S0VSuvorexant4S0V-OX2-Suvorexant
36.84Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
36.84Single6AKYMaraviroc6AKY-CCR5-Maraviroc
36.84Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
36.84Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
36.84Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
36.84Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
36.84Single6TPJSuvorexant6TPJ-OX2-Suvorexant
36.84Single7BR3Elagolix7BR3-GnRH1-Elagolix
36.84Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
36.84Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
36.84Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
36.84Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
36.84Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
36.84Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
36.84Single7XRRLemborexant7XRR-OX2-Lemborexant
36.84Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
36.84Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
36.84Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
36.84Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
36.84Single8IWESpermidine8IWE-TA9-Spermidine
36.84Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
36.84Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
36.84Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
36.84Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
36.84Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
36.84Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
36.84Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
36.84Single8Y0HVUF114188Y0H-CXCR3-VUF11418
36.84Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
36.84Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
36.84Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
36.84Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
36.84Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
36.84Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
36.67Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
36.67Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
36.67Single8IY6Endothelin-18IY6-ETB-Endothelin-1
36.67Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
36.67Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
36.36Single7B6WCyclazosin7B6W-α1b-Cyclazosin
36.36Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
36.36Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
36.36Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
36.36Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
36.36Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
36.36Single7TUYGSK682753A7TUY-GPR183-GSK682753A
36.36Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
36.36Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.36Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
36.36Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
36.36Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
36.36Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
36.36Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
36.36Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
36.36Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
36.36Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
36.36Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
36.36Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
36.36Single8XVLZibotentan8XVL-ETA-Zibotentan
36.36Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
36.36Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
36.36Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
36.36Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
36.36Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
36.36Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
36.36Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
36.36Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
36.36Consensuslpa_onOrthosteric Ligandlpa1_on
36.36Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
36.36Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
36.36Consensusrelaxin_onOrthosteric Ligandrxfp4_on
36.36Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
36.00Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
36.00Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
36.00Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
36.00Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
36.00Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
35.71Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
35.71Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
35.71Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
35.71Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
35.71Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
35.71Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
35.71Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
35.48Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
35.29Single8A2OTheophylline8A2O-A2A-Theophylline-Na
35.29Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.29Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
35.29Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
35.00Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
35.00Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
35.00Single6IQLL7458706IQL-D4-L745870
35.00Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
35.00Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
35.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
35.00Single6TP3Nemorexant6TP3-OX1-Nemorexant
35.00Single6TPNHTL66416TPN-OX2-HTL6641
35.00Single6VI4JDTic6VI4-κ-JDTic
35.00Single7AROLUF58337ARO-A2A-LUF5833-Na
35.00Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
35.00Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
35.00Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
35.00Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
35.00Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
35.00Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
35.00Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
35.00Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
35.00Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
35.00Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
35.00Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
35.00Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
35.00Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
35.00Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
35.00Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
35.00Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
35.00Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.00Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
35.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
35.00Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
35.00Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
35.00Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
35.00Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
35.00Single9BJKNaloxone9BJK-μ-Naloxone-NAM
35.00Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
35.00Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
35.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
35.00Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
35.00Consensusgrh_offOrthosteric Ligandgnrh1_off
35.00Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
35.00Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
34.78Single4XEENeurotensin4XEE-NTS1-Neurotensin
34.78Single4XESNeurotensin4XES-NTS1-Neurotensin
34.78Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
34.78Single6OS2TRV0266OS2-AT1-TRV026
34.78Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
34.78Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
34.78Single6ZG4HTL00099366ZG4-M1-HTL0009936
34.78Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
34.78Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
34.78Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
34.78Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
34.78Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
34.78Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
34.78Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
34.78Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
34.78Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
34.78Single8JWY2-1188JWY-A2A-2-118
34.78Single8JWZAB9288JWZ-A2A-AB928-Na
34.78Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
34.78Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
34.78Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
34.78Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
34.78Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
34.78Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
34.78Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
34.78Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
34.78Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
34.62Single6HLOAprepitant6HLO-NK1-Aprepitant
34.62Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
34.62Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
34.62Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
34.62Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
34.48Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
34.48Single6FJ3PTH6FJ3-PTH1-PTH
34.48Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
34.48Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.48Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
34.48Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
34.48Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
34.38Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
34.38Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
33.33Single2Y01Dobutamine2Y01-β1-Dobutamine
33.33Single3OE6IT1t3OE6-CXCR4-IT1t
33.33Single4BUONeurotensin4BUO-NTS1-Neurotensin
33.33Single5DHGC-355DHG-NOP-C-35
33.33Single5DHHSB-6121115DHH-NOP-SB-612111
33.33Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
33.33Single5TGZAM65385TGZ-CB1-AM6538
33.33Single5UENDU1725UEN-A1-DU172
33.33Single5UIGCmpd-15UIG-A2A-Cmpd-1
33.33Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
33.33Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
33.33Single6D27CAY104716D27-DP2-CAY10471
33.33Single6DRXLisuride6DRX-5-HT2B-Lisuride
33.33Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
33.33Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
33.33Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
33.33Single6ME5Agomelatine6ME5-MT1-Agomelatine
33.33Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
33.33Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
33.33Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
33.33Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
33.33Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
33.33Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
33.33Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
33.33Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
33.33Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
33.33Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
33.33Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
33.33Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
33.33Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
33.33Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
33.33Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Single7WC7Lisuride7WC7-5-HT2A-Lisuride
33.33Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
33.33Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
33.33Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
33.33Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
33.33Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
33.33Single8CU6LJ-45178CU6-A2A-LJ-4517
33.33Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
33.33Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
33.33Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
33.33Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
33.33Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
33.33Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
33.33Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
33.33Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
33.33Single8RLNLUF58348RLN-A2A-LUF5834
33.33Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
33.33Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
33.33Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8X64Desloratadine8X64-H1-Desloratadine
33.33Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
33.33Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
33.33Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
33.33Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
33.33Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
33.33Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
33.33Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
33.33Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
33.33Consensus5ht2_onOrthosteric Ligand5ht2b_on
33.33Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
33.33Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
33.33Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
33.33Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
33.33Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
33.33Consensusalpha2_onOrthosteric Ligandalpha2b_on
33.33Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
33.33Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
33.33Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
33.33Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusblt_onOrthosteric Ligandblt1_on
33.33Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
33.33Consensuscck_offOrthosteric Ligandccka_off
33.33Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
33.33Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
33.33Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
33.33Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
33.33Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
33.33Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
33.33Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
33.33Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
33.33Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
33.33Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
33.33Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
33.33Consensusleukotriene_onOrthosteric Ligandblt_on
33.33Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
33.33Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
32.50Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
32.26Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
32.26Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
32.26Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
32.14Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
32.14Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
32.14Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
32.14Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
32.14Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
32.14Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
32.14Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
32.14Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
32.00Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
32.00Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
32.00Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
32.00Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
32.00Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
32.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
32.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
32.00Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
32.00Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Single2Y00Dobutamine2Y00-β1-Dobutamine
31.82Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
31.82Single5XPRBosentan5XPR-ETB-Bosentan
31.82Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
31.82Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
31.82Single7SINNPS-21437SIN-CaS-NPS-2143
31.82Single7SINNPS-21437SIN-CaS-NPS-2143
31.82Single7W41PD1762527W41-BB2-PD176252
31.82Single8GNEKW-63568GNE-A2A-KW-6356-Na
31.82Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
31.82Single8QOTNanobody-E8QOT-μ-Nanobody-E
31.82Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
31.82Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
31.82Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
31.82Single8ZMFA1L108ZMF-5-HT2C-A1L10
31.82Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
31.82Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
31.82Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
31.82Consensusadenosine_offOrthosteric Liganda1_off a2_off
31.82Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
31.82Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
31.82Consensusblt_offOrthosteric Ligandblt1_off
31.82Consensusbombesin_offOrthosteric Ligandbb2_off
31.82Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
31.82Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
31.82Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
31.82Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
31.58Single6HLLCP999946HLL-NK1-CP99994
31.58Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
31.58Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
31.58Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
31.58Single7SRQLSD7SRQ-5-HT2B-LSD
31.58Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
31.58Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
31.58Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
31.58Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
31.58Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
31.58Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
31.58Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
31.58Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
31.58Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
31.58Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
31.58Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
31.58Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
31.58Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
31.58Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
31.58Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
31.58Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
31.58Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
31.58Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
31.58Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
31.25Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
31.25Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
31.25Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
31.03Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
31.03Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
31.03Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
31.03Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
31.03Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
31.03Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
31.03Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.03Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
31.03Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
30.77Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
30.77Single7QA8Peptide7QA8-STE2-Peptide
30.77Single7QA8Peptide7QA8-STE2-Peptide
30.77Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
30.77Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
30.77Single8IEBA1LYA8IEB-GPR156-A1LYA
30.43Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
30.43Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
30.43Single4BV0Neurotensin4BV0-NTS1-Neurotensin
30.43Single4U15Tiotropium4U15-M3-Tiotropium
30.43Single5V54Methiothepin5V54-5-HT1B-Methiothepin
30.43Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
30.43Single6J20Aprepitant6J20-NK1-Aprepitant
30.43Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
30.43Single6OL9Tiotropium6OL9-M5-Tiotropium
30.43Single6OS1TRV0266OS1-AT1-TRV026
30.43Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
30.43Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
30.43Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
30.43Single7PX4PSB-21137PX4-A2A-PSB-2113
30.43Single7R0CAVP7R0C-V2-AVP-Arrestin2
30.43Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
30.43Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.43Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
30.43Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
30.43Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
30.43Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
30.43Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
30.43Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
30.43Consensus5ht1_offOrthosteric Ligand5ht1b_off
30.43Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
30.43Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
30.43Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
30.43Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
30.43Consensusneurotensin_onOrthosteric Ligandnts1_on
30.43Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
30.43Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
30.43Consensustachykinin_offOrthosteric Ligandnk1_off
30.30Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
30.30Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
30.30Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
30.00Single3ODUIT1t3ODU-CXCR4-IT1t
30.00Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
30.00Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
30.00Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
30.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
30.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
30.00Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
30.00Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
30.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
30.00Single6ME9Ramelteon6ME9-MT2-Ramelteon
30.00Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
30.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
30.00Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
30.00Single7F8ULintitript7F8U-CCKA-Lintitript
30.00Single7F8YDevazepide7F8Y-CCKA-Devazepide
30.00Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
30.00Single7SK3CXCL127SK3-ACKR3-CXCL12
30.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
30.00Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
30.00Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
30.00Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
30.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
30.00Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
30.00Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
30.00Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
30.00Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
30.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
30.00Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
30.00Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
30.00Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
30.00Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
30.00Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
30.00Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
30.00Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
30.00Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
30.00Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
30.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
30.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Consensusangiotensin_offOrthosteric Ligandat1_off
30.00Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
30.00Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
30.00Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
30.00Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
30.00Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
30.00Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
30.00Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
30.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
30.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
30.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
30.00Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
30.00Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
29.63Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
29.63Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
29.63Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
29.63Single7SK5CXCL127SK5-ACKR3-CXCL12
29.63Single7XNACYN1548067XNA-SST2-CYN154806
29.63Single8IEBA1LYA8IEB-GPR156-A1LYA
29.63Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
29.63Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
29.63Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
29.63Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
29.41Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
29.41Single8PWNTheophylline8PWN-A2A-Theophylline
29.41Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
29.17Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
29.17Single4N4WSANT-14N4W-SMO-SANT-1
29.17Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
29.17Single5CXVTiotropium5CXV-M1-Tiotropium
29.17Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
29.17Single6CM4Risperidone6CM4-D2-Risperidone
29.17Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
29.17Single6YVRNTS8-136YVR-NTS1-NTS8-13
29.17Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
29.17Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
29.17Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.17Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
29.17Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
29.17Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.17Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
29.17Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
29.17Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
29.17Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
29.17Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
29.17Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
29.03Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
29.03Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
29.03Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
28.57Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
28.57Single3REYXAC3REY-A2A-XAC
28.57Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
28.57Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
28.57Single5IU7Q274563465IU7-A2A-Q27456346-Na
28.57Single5IUBQ274563445IUB-A2A-Q27456344-Na
28.57Single5JTBZM-2413855JTB-A2A-ZM-241385
28.57Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
28.57Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
28.57Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
28.57Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
28.57Single6A94Zotepine6A94-5-HT2A-Zotepine
28.57Single6AQFZM-2413856AQF-A2A-ZM-241385
28.57Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
28.57Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
28.57Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
28.57Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
28.57Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
28.57Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
28.57Single6ZG9GSK10347026ZG9-M1-GSK1034702
28.57Single7T32ZM-2413857T32-A2A-ZM-241385
28.57Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
28.57Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
28.57Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
28.57Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
28.57Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
28.57Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
28.57Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
28.57Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
28.57Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
28.57Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
28.57Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
28.57Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
28.57Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
28.57Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
28.57Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
28.57Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
28.57Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
28.57Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
28.57Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
28.57Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
28.57Consensusa2_offOrthosteric Liganda2a_off
28.57Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
28.57Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
28.57Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
28.57Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
28.57Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
28.57Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
28.12Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
28.12Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
28.12Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
28.12Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
28.12Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
28.12Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
28.00Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
28.00Single6K1QIRL25006K1Q-ETB-IRL2500
28.00Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
28.00Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
28.00Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
28.00Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
28.00Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
28.00Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
28.00Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
28.00Single8XVJMacitentan8XVJ-ETA-Macitentan
28.00Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.00Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.00Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single3RFMCaffeine3RFM-A2A-Caffeine
27.78Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
27.78Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
27.78Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
27.78Single9CHUNoradrenaline9CHU-β2-Noradrenaline
27.78Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
27.78Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
27.78Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
27.78Consensussensory_onOrthosteric Ligandopsins_on
27.59Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
27.59Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
27.59Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
27.59Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
27.27Single3EMLZM-2413853EML-A2A-ZM-241385
27.27Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
27.27Single4QIMANTA XV4QIM-SMO-ANTA XV
27.27Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
27.27Single5IU8Q274563475IU8-A2A-Q27456347-Na
27.27Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
27.27Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
27.27Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
27.27Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
27.27Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
27.27Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
27.27Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
27.27Single6GPSMK08126GPS-CCR2-MK0812
27.27Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
27.27Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
27.27Single6S0LZM-2413856S0L-A2A-ZM-241385
27.27Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
27.27Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
27.27Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
27.27Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
27.27Single7PYRPSB-21157PYR-A2A-PSB-2115
27.27Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
27.27Single7YXAONO-54306087YXA-S1P5-ONO-5430608
27.27Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
27.27Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
27.27Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
27.27Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
27.27Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
27.27Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
27.27Single8X63Mepyramine8X63-H1-Mepyramine
27.27Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
27.27Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
27.27Single9IYAONO-97105319IYA-GPR55-ONO-9710531
27.27Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
27.27Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
27.27Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
27.27Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
27.27Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
27.27Consensushistamine_offOrthosteric Ligandh1_off
27.27Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
27.27Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
27.27Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
26.92Single5EE7MK08935EE7-Glucagon-MK0893
26.92Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
26.92Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
26.92Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
26.92Single8XQJJN2418XQJ-Apelin-JN241
26.92Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
26.92Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
26.92Consensuskisspeptin_onOrthosteric Ligandkiss1_on
26.67Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
26.67Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
26.47Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
26.32Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
26.32Single3UZAGTPL92363UZA-A2A-GTPL9236
26.32Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
26.32Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
26.32Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
26.32Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
26.32Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
26.32Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
26.32Single7WC5Psilocin7WC5-5-HT2A-Psilocin
26.32Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
26.32Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
26.32Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
26.32Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
26.32Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
26.32Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
26.32Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
26.32Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
26.32Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
26.32Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
26.09Single4NTJAZD12834NTJ-P2Y12-AZD1283
26.09Single5IUAQ274563485IUA-A2A-Q27456348-Na
26.09Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
26.09Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
26.09Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
26.09Single6GPXMK08126GPX-CCR2-MK0812
26.09Single6HLPNetupitant6HLP-NK1-Netupitant
26.09Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
26.09Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
26.09Single6LUQHaloperidol6LUQ-D2-Haloperidol
26.09Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
26.09Single6S0QZM-2413856S0Q-A2A-ZM-241385
26.09Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
26.09Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
26.09Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
26.09Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
26.09Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
26.09Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
26.09Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
26.09Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
26.09Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
26.09Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
26.09Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
26.09Consensusep_offOrthosteric Ligandep4_off
26.09Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
26.09Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
26.09Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
26.09Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
25.93Single8IEIA1LYA8IEI-GPR156-A1LYA
25.93Single8IEPA1LYA8IEP-GPR156-A1LYA
25.93Single8IEPA1LYA8IEP-GPR156-A1LYA
25.93Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
25.93Single8KIGSHU91198KIG-MC3-SHU9119-Ca
25.93Single8XWNCXCL88XWN-CXCR2-CXCL8
25.93Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
25.93Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
25.93Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
25.93Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
25.93Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
25.93Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
25.93Consensussomatostatin_offOrthosteric Ligandsst2_off
25.81Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
25.81Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
25.81Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
25.81Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
25.71Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
25.71Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
25.71Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
25.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
25.00Single5TZRMK86665TZR-FFA1-MK8666
25.00Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
25.00Single6E59L-7607356E59-NK1-L-760735
25.00Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
25.00Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
25.00Single6TP4ACT-4622066TP4-OX1-ACT-462206
25.00Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
25.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
25.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
25.00Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
25.00Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
25.00Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
25.00Single7F1TMIP-1a7F1T-CCR5-MIP-1a
25.00Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
25.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
25.00Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
25.00Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
25.00Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
25.00Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
25.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
25.00Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
25.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
25.00Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
25.00Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
25.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8EA0Iperoxo8EA0-M3-Iperoxo
25.00Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
25.00Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
25.00Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
25.00Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
25.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
25.00Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
25.00Single9B9Y7DY9B9Y-CB1-7DY
25.00Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
25.00Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
25.00Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
25.00Consensusgq_nucleotideOrthosteric Ligandgq_p2y
25.00Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
25.00Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
25.00Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
25.00Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
25.00Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
25.00Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
24.24Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
24.24Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
24.24Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
24.14Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
24.00Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
24.00Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
24.00Single4PY02MeSATP4PY0-P2Y12-2MeSATP
24.00Single5X33BIIL2605X33-BLT1-BIIL260
24.00Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
24.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
24.00Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
24.00Single8XQJJN2418XQJ-Apelin-JN241
24.00Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
23.81Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
23.81Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
23.81Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
23.81Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
23.81Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
23.81Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
23.81Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
23.81Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
23.81Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
23.81Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
23.81Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
23.81Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
23.81Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
23.81Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
23.81Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
23.81Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
23.81Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
23.81Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
23.81Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
23.81Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
23.81Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
23.81Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
23.53Single5MZPCaffeine5MZP-A2A-Caffeine-Na
23.53Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
23.53Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
23.53Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
23.33Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
23.33Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
23.33Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
23.33Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
23.08Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
23.08Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
23.08Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single8XVUCXCL28XVU-CXCR2-CXCL2
23.08Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
23.08Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
22.86Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
22.86Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
22.73Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
22.73Single3RZECidoxepin3RZE-H1-Cidoxepin
22.73Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
22.73Single5UVIZM-2413855UVI-A2A-ZM-241385
22.73Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
22.73Single6TPKRetosiban6TPK-OT-Retosiban
22.73Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
22.73Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
22.73Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
22.73Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
22.73Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
22.73Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
22.73Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
22.73Single8K2WAMG4878K2W-CXCR3-AMG487
22.73Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.73Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
22.73Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
22.73Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
22.73Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
22.73Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
22.73Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
22.73Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
22.73Consensusopsins_offOrthosteric Ligandrhodopsin_off
22.73Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
22.73Consensussensory_offOrthosteric Ligandopsins_off
22.73Consensusvasop-oxy_offOrthosteric Ligandot_off
22.58Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
22.22Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
22.22Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
22.22Single6KNMJN241-96KNM-Apelin-JN241-9
22.22Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
22.22Single7WC4Serotonin7WC4-5-HT2A-Serotonin
22.22Single8IEIA1LYA8IEI-GPR156-A1LYA
22.22Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
22.22Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
22.22Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
22.22Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
21.88Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
21.88Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
21.88Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
21.74Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
21.74Single4DAJTiotropium4DAJ-M3-Tiotropium
21.74Single4MQSIperoxo4MQS-M2-Iperoxo
21.74Single4U14Tiotropium4U14-M3-Tiotropium
21.74Single5DSGTiotropium5DSG-M4-Tiotropium
21.74Single5T04Neurotensin5T04-NTS1-Neurotensin
21.74Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
21.74Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
21.74Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
21.74Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
21.74Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
21.74Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
21.74Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
21.74Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
21.74Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.74Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
21.74Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
21.43Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
21.43Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
21.21Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
21.21Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
21.21Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
21.05Single3OE8IT1t3OE8-CXCR4-IT1t
21.05Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
21.05Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
21.05Single6TQ9SB-4081246TQ9-OX1-SB-408124
21.05Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
21.05Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
21.05Consensusp2y_offOrthosteric Ligandp2y1_off
20.83Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
20.83Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
20.83Single5CGCHTL142425CGC-mGlu5-HTL14242
20.83Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
20.83Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
20.83Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
20.83Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
20.83Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.83Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
20.83Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
20.83Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
20.83Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
20.83Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
20.83Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
20.69Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
20.69Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
20.59Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
20.59Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
20.59Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
20.59Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
20.00Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
20.00Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
20.00Single4XNWMRS25004XNW-P2Y1-MRS2500
20.00Single5V56TC1145V56-SMO-TC114
20.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
20.00Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
20.00Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
20.00Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
20.00Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
20.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
20.00Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
20.00Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
20.00Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
20.00Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
20.00Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
20.00Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
20.00Single9BJKNAM9BJK-μ-Naloxone-NAM
20.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
20.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
20.00Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
20.00Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
20.00Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
20.00Consensusgi_sensoryOrthosteric Ligandgi_opsins
20.00Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
20.00Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
20.00Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
20.00Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
19.51Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
19.44Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
19.35Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
19.35Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
19.35Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
19.23Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
19.23Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
19.23Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
19.23Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
19.23Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
19.23Single8XWACXCL18XWA-CXCR2-CXCL1
19.23Single8XWMCXCL68XWM-CXCR2-CXCL6
19.23Single8XWSCXCL58XWS-CXCR2-CXCL5
19.23Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
19.23Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
19.23Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
19.05Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
19.05Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
19.05Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
19.05Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
19.05Single5L7IVismodegib5L7I-SMO-Vismodegib
19.05Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
19.05Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
19.05Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
19.05Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
19.05Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
19.05Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
19.05Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.05Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.05Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
18.75Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
18.52Single5CGDHTL142425CGD-mGlu5-HTL14242
18.52Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
18.52Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single8XWFCXCL38XWF-CXCR2-CXCL3
18.52Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
18.52Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
18.52Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
18.52Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
18.42Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
18.42Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
18.18Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
18.18Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
18.18Single4BWBNeurotensin4BWB-NTS1-Neurotensin
18.18Single5U09Taranabant5U09-CB1-Taranabant
18.18Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
18.18Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
18.18Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
18.18Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
18.18Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
18.18Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
18.18Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
18.18Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
18.18Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
18.18Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
18.18Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
18.18Single9BA0A1AKN9BA0-CB1-A1AKN
18.18Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
17.86Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
17.86Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
17.86Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
17.86Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
17.65Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
17.65Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
17.39Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
17.39Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
17.39Single6ZINSR486926ZIN-NTS1-SR48692
17.39Single7VODCariprazine7VOD-5-HT2A-Cariprazine
17.24Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
17.24Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
17.24Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
17.24Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
17.24Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
17.14Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
17.14Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
16.67Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
16.67Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
16.67Single6IIVDaltroban6IIV-TP-Daltroban
16.67Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
16.67Single7F83PF-051904577F83-Ghrelin-PF-05190457
16.67Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
16.67Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
16.67Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
16.67Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
16.67Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9B9ZA1AKO9B9Z-CB1-A1AKO
16.22Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
16.00Single4JKVTaladegib4JKV-SMO-Taladegib
16.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
16.00Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
16.00Single6Z4SSR486926Z4S-NTS1-SR48692
16.00Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
16.00Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
16.00Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
16.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
16.00Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
15.79Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
15.79Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
15.38Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
15.38Single5V57TC1145V57-SMO-TC114
15.38Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
15.38Single7P2L4YI7P2L-mGlu5-4YI
15.38Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
15.38Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
15.38Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
15.15Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
15.00Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
15.00Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
14.81Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
14.81Single6IIURamatroban6IIU-TP-Ramatroban
14.81Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
14.81Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
14.29Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
14.29Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
14.29Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
14.29Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
14.29Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
14.29Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
14.29Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
13.79Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
13.64Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
13.64Single4O9RCyclopamine4O9R-SMO-Cyclopamine
13.64Single6LI0C176LI0-GPR52-C17
13.64Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
13.64Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
13.64Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
13.64Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
13.33Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
13.33Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single4QINSAG1.54QIN-SMO-SAG1.5
13.04Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
13.04Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
13.04Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
13.04Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
13.04Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
13.04Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
13.04Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
13.04Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
13.04Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
12.50Single6FFIMMPEP6FFI-mGlu5-MMPEP
12.50Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
12.50Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
12.50Single7VV6C48/807VV6-MRGPRX2-C48/80
12.50Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
12.50Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
12.12Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
12.00Single6FFHFenobam6FFH-mGlu5-Fenobam
12.00Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
11.76Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
11.54Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
11.54Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
11.54Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
11.54Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
11.54Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
11.11Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
11.11Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
10.71Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
10.34Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
10.34Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
10.00Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
10.00Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.00Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
10.00Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
10.00Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
10.00Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
9.68Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
9.52Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
9.52Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
9.09Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
9.09Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
9.09Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
9.09Single8JPSCCL78JPS-ACKR1-CCL7
8.70Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.70Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
8.70Single7UL2SR486927UL2-NTS1-SR48692-Na
8.70Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.70Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
8.70Consensusneurotensin_offOrthosteric Ligandnts1_off
8.70Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
8.00Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
7.69Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
7.69Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
7.41Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
7.41Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
7.41Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
7.14Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
6.06Single7SHEPI; PE7SHE-GPR158-PI; PE
5.88Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.88Single6D35Cholesterol6D35-SMO-Cholesterol
5.88Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.88Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.88Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
5.88Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
5.88Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
5.88Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
5.88Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
5.88Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
5.88Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
5.88Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
5.88Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.88Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.88Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.88Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.88Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
5.88Single7DTTCa7DTT-CaS-Ca-Ca
5.88Single7DTTCa7DTT-CaS-Ca-Ca
5.88Single7DTUTryptophan7DTU-CaS-Tryptophan
5.88Single7DTUTryptophan7DTU-CaS-Tryptophan
5.88Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.88Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.88Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.88Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.88Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.88Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.88Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.88Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.88Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
5.88Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.88Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.88Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.88Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.88Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.88Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.88Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
5.88Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
5.88Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.88Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.88Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.88Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.88Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.88Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.88Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.88Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.88Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.88Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.88Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.88Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.88Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.88Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.88Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.88Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.88Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.88Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.88Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.88Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
5.88Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.88Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.88Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.88Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.88Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.88Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.88Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
5.88Single7XW7K1-707XW7-TSH-K1-70
5.88Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.88Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.88Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.88Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.88Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.88Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.88Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.88Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.88Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.88Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.88Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.88Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.88Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
5.88Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.88Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.88Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.88Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.88Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
5.88Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
5.88Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.88Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.88Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
5.88Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
5.88Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
5.88Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
5.88Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.88Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.88Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.88Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
5.88Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
5.88Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
5.88Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
5.88Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.88Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.88Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.88Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.88Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.88Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.88Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.88Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.88Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.88Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.88Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.88Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.88Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.88Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.88Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.88Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.88Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.88Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.88Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
5.88Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
5.88Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
5.88Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
5.88Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
5.88Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
5.88Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.88Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.88Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8WVXNorrin8WVX-LGR4-Norrin
5.88Single8WVYNorrin8WVY-LGR4-Norrin
5.88Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.88Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.88Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.88Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.88Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.88Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.88Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
5.88Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.88Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.88Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.88Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.88Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.88Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.88Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.88Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.88Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.88Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.88Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.88Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.88Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.88Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.88Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.88Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.88Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.88Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.88Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.88Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.56Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.56Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.56Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.56Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.56Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.56Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.56Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.56Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.56Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.56Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.56Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
5.26Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
5.26Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
5.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
5.00Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
5.00Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
5.00Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
5.00Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
5.00Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
4.76Single5L7DCholesterol5L7D-SMO-Cholesterol
4.76Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.76Single8HS2Fab0468HS2-GPR20-Fab046
4.76Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.55Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
4.35Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
4.35Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
4.17Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.17Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
4.17Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.00Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
3.85Single8IYXYL-3658IYX-GPR34-YL-365
3.33Single7SHEPI; PE7SHE-GPR158-PI; PE
3.23Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
3.03Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
3.03Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.94Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
2.86Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.86Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.78Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.56Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
sensory_on_gp opsins_on_gp
alicarboxylic_on_gp succinate_on_gp
hca_on_gp
amine_on_gp 5ht_on_gp
adrenergic_on_gp
dopamine_on_gp
histamine_on_gp
muscarinic_on_gp
trace-amine_on_gp
lipid_on_gp cannabinoid_on_gp
ffa_on_gp
lpl_on_gp
prostanoid_on_gp
leukotriene_on_gp
nucleotide_on_gp adenosine_on_gp
p2y_on_gp
peptide_on_gp cck_on_gp
angiotensin_on_gp
apelin_on_gp
bombesin_on_gp
bradykinin_on_gp
compl-peptide_on_gp
endothelin_on_gp
formylpeptide_on_gp
galanin_on_gp
ghrelin_on_gp
kisspeptin_on_gp
melanocortin_on_gp
motilin_on_gp
neuromedin-u_on_gp
npy_on_gp
neurotensin_on_gp
opioid_on_gp
orexin_on_gp
relaxin_on_gp
somatostatin_on_gp
tachykinin_on_gp
trh_on_gp
vasop-oxy_on_gp
protein_on_gp chemokine_on_gp
chemerin_on_gp
Net Summary
Imin 2.7705
Number of Linked Nodes 1203
Number of Links 1376
Number of Hubs 198
Number of Links mediated by Hubs 799
Number of Communities 21
Number of Nodes involved in Communities 229
Number of Links involved in Communities 325
Path Summary
Number Of Nodes in MetaPath 104
Number Of Links MetaPath 103
Number of Shortest Paths 16851514
Length Of Smallest Path 3
Average Path Length 47.2058
Length of Longest Path 72
Minimum Path Strength 0.203775
Average Path Strength 4.75539
Maximum Path Strength 21.0844
Minimum Path Correlation 0.701431
Average Path Correlation 0.996289
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.49254
Average % Of Corr. Nodes 18.8168
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 57.5715
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following differences:
Id1st Network2nd Network
class-a_off_on_gpclass-a_on_gpclass-a_off



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