Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1Lig 8.015362320
21x39 4.64917407
31x43 4.69875406
41x55 3.115834174
51x61 3.38167405
62x39 3.83708407
72x43 5.14333428
82x50 5.79875409
92x53 7.86667527
10E1x50 8.24194629
11E1x52 6.42111607
123x28 7.06125405
133x36 5.49875428
143x37 8.66208427
153x40 3.79292427
163x41 5.43625406
173x43 5.746528
183x46 5.04208429
193x50 7.785529
203x53 4.636254128
21I2x57 9.815424127
224x64 9.455425
23E2.T166 3.75792425
24E2x52 5.75625424
25E2.F180 5.276526
265x43 8.27133525
275x44 7.08917426
285x47 8.30792429
295x51 5.26583406
305x58 5.30143728
31I3.M233 4.314335203
326x40 3.78875428
336x44 5.76875429
346x48 5.48729
356x49 7.99958406
366x51 4.44083427
376x52 5.5725628
386x61 10.5496403
397x42 7.17542427
407x49 6.08458429
417x53 6.62133529
428x50 6.99528
43G.HN.30 2.16958407
44G.S1.02 5.38455
45G.S1.06 4.61458459
46G.H1.01 3.848559
47G.S2.06 7.80042458
48G.S2.08 8.493754135
49G.S3.01 5.56458404
50G.S3.03 7.88033557
51G.S3.04 7.6425417
52G.S3.05 3.96833457
53G.S3.06 8.76516
54G.S3.07 3.735459
55G.s3h2.03 4.64417419
56G.H2.02 4.65583418
57G.H2.06 5.70583819
58G.H2.07 4.85286719
59G.h2s4.01 7.21733519
60G.S4.02 4.87792417
61G.S4.03 3.94208408
62G.S4.04 6.16472649
63G.s4h3.04 5.82583668
64G.s4h3.05 7.07125469
65G.H3.09 6.30357749
66G.H3.17 7.92111615
67G.H3.18 7.23542419
68G.S5.03 3.55333408
69G.S5.04 4.87533549
70G.S5.07 6.11375409
71G.HG.04 4.96167668
72G.hgh4.02 6.156946118
73G.hgh4.05 9.47667406
74G.H4.10 10.61874116
75G.H4.11 3.433334117
76G.H4.15 5.94833448
77G.h4s6.02 5.07083447
78G.S6.02 6.09083408
79G.S6.04 8.42917409
80G.H5.08 7.664174138
81G.H5.26 5.102507
82b.lh12x2 4.92125408
83b.h2x5 3.56042475
84b.lhb1x3 3.22967572
85b.lhb1x6 3.4475473
86b.b1x4 5.27542437
87b.b1x6 8.85375439
88b.l1x3 9.13028639
89b.b2x1 9.29033518
90b.b2x5 6.91667637
91b.b3x2 6.12625435
92b.b3x3 3.88792408
93b.l3x2 5.34867539
94b.b4x3 5.06254147
95b.b4x4 9.785438
96b.b4x5 4.137084217
97b.b4x6 10.8942639
98b.b5x2 5.68458407
99b.b5x3 6.50306639
100b.b5x5 5.6054215
101b.b5x7 6.64417407
102b.l5x1 4.347675148
103b.l5x5 8.80262719
104b.b6x5 4.15767506
105b.l6x5 6.150834154
106b.b7x1 6.634675154
107b.l7x4 3.84625409
108b.b8x3 4.14625406
109b.b8x4 6.010335146
110b.l8x5 2.24583403
111b.l9x3 7.37722619
112b.l9x6 5.19708818
113b.b10x5 5.03556609
114b.l10x1 3.85583403
115b.b11x4 5.39625419
116b.l11x2 8.17833419
117b.b12x6 9.75139618
118b.b12x7 6.203334229
119b.b13x7 8.26567587
120b.l13x3 8.18833689
121b.l13x6 5.10667519
122b.l13x7 4.65767589
123b.b15x1 8.1425489
124b.b15x2 7.76833416
125b.l15x1 4.6075417
126b.l15x2 5.68458409
127b.b16x4 11.0958486
128b.b16x5 5.559515
129b.b16x6 8.00286788
130b.b17x5 6.11889617
131b.b17x7 8.785418
132b.l17x3 9.19944619
133b.l17x6 5.866519
134b.l17x7 5.43458417
135b.b18x3 5.03125418
136b.b18x5 5.89167405
137b.l18x1 7.014176106
138b.l18x2 5.893334107
139b.b19x2 7.05917616
140b.b19x4 6.21792418
141b.l19x1 5.84567519
142b.l19x2 6.32133519
143b.b20x4 11.3827518
144b.b20x6 7.10111616
145b.b21x1 7.46167517
146b.b21x2 3.47233506
147b.b21x7 6.23722605
148b.b22x5 5.7535107
149b.l22x5 7.07472679
150b.b23x1 4.12042405
151b.b23x6 6.35405717
152b.l23x1 7.705416
153b.b24x4 7.74125416
154b.b24x6 6.42292418
155b.l24x3 5.267575
156b.b25x3 8.14833415
157b.l25x3 8.46967599
158b.l25x6 10.7146418
159b.l27x1 10.9357719
160b.l27x2 8.47833499
161b.b28x4 8.29458496
162b.b28x6 9.221599
163g.h1x5 1.37333506
164g.h1x11 2.92708409
165g.l1x4 5.67833408
166g.h2x11 10.03834106
167g.ctx3 7.09033509
168g.ctx6 4.17676
169g.ctx14 6.675439
170g.ctx15 7.31458439
171g.ctx16 5.01278938
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
13x43 7x53 81.487910.0733YesYes289
23x43 6x44 73.60216.07YesYes289
33x40 6x44 32.15543.05667YesYes279
43x40 Lig 29.95743.41YesYes270
56x44 6x48 38.12568.35167YesYes299
66x48 Lig 29.99944.435YesYes290
77x54 8x50 96.88448.525NoYes278
82x43 7x54 97.07617.57167YesNo287
92x43 3x46 41.59163.42833YesYes289
103x46 7x53 41.43395.84167YesYes299
112x43 3x50 54.59875.82667YesYes289
123x50 7x53 41.42837.88667YesYes299
131x61 8x53 98.39516.615YesNo055
141x61 8x50 98.19434.14667YesYes058
153x29 E1x50 15.17444.05833NoYes269
163x29 Lig 15.91916.135NoYes260
17G.H5.17 G.H5.26 10.43183.30667NoYes057
18G.H5.20 G.H5.26 12.12828.93167NoYes087
19G.H5.20 G.H5.25 12.22765.99833NoNo087
206x37 G.H5.25 12.3274.84333NoNo087
215x58 6x37 12.62485.47167YesNo088
22b.b4x7 b.l2x5 48.922114.29NoNo085
23b.l2x5 b.l4x2 97.190122.295NoNo054
24b.l4x2 g.ctx15 95.981214.1417NoYes349
25b.l26x5 g.ctx15 98.29995.59167NoYes059
26b.l26x5 g.ctx4 99.99375.59NoNo057
27g.ctx3 g.ctx4 1004.29333YesNo097
28b.l22x1 g.ctx3 98.17138.83333NoYes099
29b.l22x1 g.ctx5 97.77895.00333NoNo099
30b.lhb1x11 g.ctx5 97.78225.89NoNo049
31b.b25x7 b.lhb1x11 99.65175.18333NoNo074
32b.b25x7 b.b28x6 99.659718.98NoYes079
33b.b27x3 b.b28x6 49.76679.09667NoYes089
34b.b27x3 b.l25x3 49.85047.53167NoYes089
35b.l25x3 b.l27x2 99.2647.77167YesYes999
36b.l25x4 b.l27x2 99.13726.20833NoYes059
378x53 b.l25x4 99.069710.52NoNo055
38b.b28x4 b.b28x6 49.85676.96YesYes969
39b.b28x4 b.l25x3 49.7048.95167YesYes969
40b.b3x1 b.b6x5 97.33393.32NoYes056
41b.b3x1 b.l2x3 48.22915.20333NoNo058
42b.l2x3 b.l2x5 48.25993.57167NoNo085
43b.b3x1 b.b4x7 49.18883.16667NoNo058
44G.H2.07 b.l9x6 44.9513.69833YesYes198
45G.H2.06 b.l9x6 58.87735.375YesYes198
46G.H2.06 b.l17x6 29.68438.75833YesYes199
47b.l17x5 b.l17x6 36.40774.17167NoYes169
48b.l17x5 b.l19x2 76.0123.435NoYes169
49b.l17x3 b.l19x2 75.54464.83YesYes199
50b.b19x4 b.l17x3 75.22768.44YesYes189
51b.b18x3 b.b19x4 75.10573.54667YesYes188
52b.b15x2 b.b18x3 75.2436.39833YesYes168
53b.b15x2 b.b18x5 83.21069.835YesYes065
54b.b18x5 b.l14x1 83.57085.77833YesNo054
55b.l14x1 b.l14x3 83.66083.08833NoNo045
56b.l14x3 b.l14x5 83.75076.94833NoNo055
57b.l14x5 b.l16x2 83.84066.93NoNo059
58b.l16x1 b.l16x2 83.93045.015NoNo049
59b.l10x1 b.l16x1 84.02023.47667YesNo034
60b.b14x5 b.l10x1 84.30884.61333NoYes053
61b.b10x4 b.b14x5 90.84833.64167NoNo065
62b.b10x4 b.b2x4 91.77113.5417NoNo066
63b.b2x4 b.b6x5 91.85763.27NoYes066
64G.H2.06 b.l19x1 29.83594.37833YesYes199
65b.l17x5 b.l19x1 39.5093.68NoYes169
66G.H3.08 G.S4.04 36.30596.90333NoYes099
67G.H2.04 G.H3.08 36.52185.465NoNo099
68G.H2.04 G.H2.07 36.96066.16667NoYes099
69G.H3.09 G.S4.04 10.064815.7183YesYes499
70G.S4.04 G.S5.04 17.63373.045YesYes499
71G.S5.04 G.S5.06 10.35473.92167YesNo099
72G.H3.06 G.hgh4.02 18.21735.25167NoYes068
73G.H3.06 G.H4.15 18.88915.6NoYes068
74b.l11x1 b.l9x6 12.2915.795NoYes198
75b.b11x6 b.l11x1 17.91663.09333NoNo199
76b.b11x6 b.l9x3 12.869315.11NoYes199
77b.b12x6 b.l9x3 10.17137.76YesYes189
783x50 5x58 13.01919.43167YesYes298
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x33Lig15.16332NoYes5010
3x36Lig5.571672YesYes8010
3x37Lig17.33832YesYes7010
3x40Lig3.412YesYes7010
5x39Lig12.29332NoYes5010
5x43Lig20.13832YesYes5010
6x48Lig4.4352YesYes9010
6x51Lig4.876672YesYes7010
6x52Lig3.231672YesYes8010
7x34Lig9.281670NoYes5010
5x36Lig4.0952NoYes4010
E1.E89Lig8.263332NoYes0010
E3.L272Lig3.756672NoYes0010
E2x52Lig4.581672YesYes4010
5x28Lig3.893332NoYes5010
2x533x368.323332YesYes7821
2x537x4213.932YesYes7722
3x29E1x504.058332NoYes6912
3x294x6562NoNo6512
3x334x576.023332NoNo5712
3x334x614.623332NoNo5412
3x366x483.226672YesYes8911
3x367x424.873332YesYes8712
3x373x416.786672YesYes7612
3x374x569.133332YesNo7512
3x405x504.4152YesNo7912
3x406x443.056672YesYes7912
4x614x654.221670NoNo4522
4x65E2x526.4950NoYes5421
5x39E2x528.196672NoYes5411
5x255x286.486670NoNo5521
5x36E3.L2685.0752NoNo4012
5x395x436.398332NoYes5511
5x405x433.50NoYes4521
5x436x527.42YesYes5811
5x436x553.922YesNo5512
5x445x474.288332YesYes6922
5x446x523.511672YesYes6821
5x476x5212.88332YesYes9821
6x446x488.351672YesYes9921
6x486x523.286672YesYes9811
6x487x416.483332YesNo9812
6x487x458.286672YesNo9912
6x516x523.121672YesYes7811
6x517x375.836672YesNo7712
6x517x413.928332YesNo7812
E3.L268E3.L2724.613330NoNo0021
7x30E3.M2713.160NoNo4021
7x31Lig3.3852NoYes4010
2x60Lig3.798330NoYes6010
3x29Lig6.1352NoYes6010
2x647x357.246670NoNo6421
3x406x484.292YesYes7911
E2.F180E2x523.751672YesYes0421
E2x51Lig3.333330NoYes3010
7x35Lig3.758332NoYes4010
1x357x352.4450NoNo5421
6x58E3.M2712.040NoNo4021
5x28E2.G18422NoNo5012
E3.M271Lig1.982NoYes0010
7x287x311.613330NoNo1421
3x374x531.392YesNo7812
2x67E1.E891.366670NoNo3021

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
95.00Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
90.48Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
72.73Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
72.00Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
71.43Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
63.64Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
60.87Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
57.14Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
56.00Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
56.00Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
54.17Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
52.17Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
47.62Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
46.15Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
46.15Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
45.83Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
45.83Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
45.45Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
45.45Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
45.45Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
45.00Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
44.44Consensusangiotensin_onOrthosteric Ligandat1_on
44.44Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
43.48Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
43.33Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
42.86Single6JODAngiotensin II6JOD-AT2-Angiotensin II
42.86Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
42.86Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
42.86Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.86Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
42.86Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
42.86Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
42.86Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
42.86Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
42.31Single4IARErgotamine4IAR-5-HT1B-Ergotamine
42.31Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
42.31Single8WDTphotoNECA8WDT-A2A-photoNECA
42.31Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
42.31Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
41.94Single6IGLIRL16206IGL-ETB-IRL1620
41.67Single6A93Risperidone6A93-5-HT2A-Risperidone
41.67Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
41.67Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
41.38Single8ZRTET-18ZRT-ETB-ET-1
40.74Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
40.74Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
40.74Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
40.62Single5GLHEndothelin-15GLH-ETB-Endothelin-1
40.62Single6IGKEndothelin-36IGK-ETB-Endothelin-3
40.00Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
40.00Single7EZCUKA7EZC-A2A-UKA
40.00Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
40.00Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
40.00Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
40.00Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
40.00Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
40.00Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
40.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
39.39Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
39.29Single5WF5UK-4320975WF5-A2A-UK-432097
39.29Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
39.29Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
39.29Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
39.29Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
39.29Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
39.29Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
39.29Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
39.29Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
39.13Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
38.71Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
38.71Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
38.71Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
38.71Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
38.46Single5WF6UK-4320975WF6-A2A-UK-432097
38.46Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
38.46Single7SK9CCX6627SK9-ACKR3-CCX662
38.46Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
38.46Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
38.46Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
38.46Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
38.24Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
37.50Single5V54Methiothepin5V54-5-HT1B-Methiothepin
37.50Single7B6WCyclazosin7B6W-α1b-Cyclazosin
37.50Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
37.50Single8IY6Endothelin-18IY6-ETB-Endothelin-1
37.50Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
37.50Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
37.50Consensus5ht1_offOrthosteric Ligand5ht1b_off
37.50Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
37.50Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
37.50Consensusendothelin_onOrthosteric Ligandetb_on eta_on
37.50Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
37.50Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
37.50Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
37.04Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
37.04Consensuslpl_onOrthosteric Ligands1p_on lpa_on
37.04Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
37.04Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
37.04Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
37.04Consensussomatostatin_offOrthosteric Ligandsst2_off
36.67Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
36.67Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
36.67Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
36.67Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
36.67Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
36.67Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
36.67Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.36Single7T32ZM-2413857T32-A2A-ZM-241385
36.36Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
36.36Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
36.36Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
36.00Single3D4STimolol3D4S-β2-Timolol
36.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
36.00Single6MXTSalmeterol6MXT-β2-Salmeterol
36.00Single7DFPSpiperone7DFP-D2-Spiperone
36.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
36.00Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
36.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
36.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
36.00Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
36.00Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
36.00Single7YITNalfurafine7YIT-κ-Nalfurafine
36.00Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
36.00Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
36.00Single8JJLOlodaterol8JJL-β2-Olodaterol
36.00Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
36.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
36.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
35.71Single3QAKUK-4320973QAK-A2A-UK-432097
35.71Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
35.71Single7XNACYN1548067XNA-SST2-CYN154806
35.71Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
35.71Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
35.71Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
35.48Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
35.48Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
35.48Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
35.48Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
35.48Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
35.48Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
35.29Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
35.29Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
34.78Single6DRXLisuride6DRX-5-HT2B-Lisuride
34.78Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
34.78Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
34.78Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
34.78Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
34.78Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
34.78Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
34.62Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
34.62Single6IBLArformoterol6IBL-β1-Arformoterol
34.62Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
34.62Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
34.62Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
34.62Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
34.62Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
34.62Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
34.62Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
34.62Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
34.48Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
34.48Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
34.48Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
34.38Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
34.38Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
34.38Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
34.38Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
34.29Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
33.33Single2YCWS-Carazolol2YCW-β1-S-Carazolol
33.33Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
33.33Single4UG2CGS216804UG2-A2A-CGS21680
33.33Single5D6LS-Carazolol5D6L-β2-S-Carazolol
33.33Single5IUAQ274563485IUA-A2A-Q27456348-Na
33.33Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
33.33Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
33.33Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
33.33Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
33.33Single6S0QZM-2413856S0Q-A2A-ZM-241385
33.33Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
33.33Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
33.33Single7C61Ergotamine7C61-5-HT1B-Ergotamine
33.33Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
33.33Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
33.33Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
33.33Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
33.33Single7XN9L-054,5227XN9-SST2-L-054,522
33.33Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
33.33Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
33.33Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
33.33Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
33.33Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
33.33Single8JXSPF-61428JXS-D1-PF-6142
33.33Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
33.33Single8X5YAstemizole8X5Y-H1-Astemizole
33.33Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
33.33Single8ZMFA1L108ZMF-5-HT2C-A1L10
33.33Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
33.33Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
33.33Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
33.33Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
33.33Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
33.33Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
33.33Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
33.33Consensusbradykinin_onOrthosteric Ligandbk2_on
33.33Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
33.33Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
33.33Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
33.33Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
33.33Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
33.33Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
33.33Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
33.33Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
33.33Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
33.33Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Consensusvasop-oxy_onOrthosteric Ligandv2_on
33.33Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
32.35Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
32.35Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
32.35Consensusbombesin_onOrthosteric Ligandbb2_on
32.35Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
32.35Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
32.35Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
32.26Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
32.26Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.26Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
32.26Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
32.26Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
32.26Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
32.26Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
32.26Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
32.26Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
32.26Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
32.14Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
32.14Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
32.14Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
32.14Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
32.14Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
32.14Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
32.14Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
32.14Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
32.14Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
32.14Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
32.14Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
32.14Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
32.14Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
32.14Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
32.14Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
32.14Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
32.00Single3P0GBI1671073P0G-β2-BI167107
32.00Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
32.00Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
32.00Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
32.00Single5D5AS-Carazolol5D5A-β2-S-Carazolol
32.00Single5D5BS-Carazolol5D5B-β2-S-Carazolol
32.00Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
32.00Single6J20Aprepitant6J20-NK1-Aprepitant
32.00Single6J21Aprepitant6J21-NK1-Aprepitant
32.00Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
32.00Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
32.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
32.00Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
32.00Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
32.00Single7PX4PSB-21137PX4-A2A-PSB-2113
32.00Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
32.00Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
32.00Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
32.00Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
32.00Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
32.00Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
32.00Single8E0GBU728E0G-μ-BU72
32.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
32.00Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
32.00Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
32.00Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
32.00Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
32.00Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
32.00Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
32.00Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
32.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
32.00Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
32.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
32.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
32.00Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
32.00Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
31.82Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
31.82Single6ME9Ramelteon6ME9-MT2-Ramelteon
31.82Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
31.43Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
31.03Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
31.03Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
31.03Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
31.03Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
31.03Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
31.03Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
31.03Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
31.03Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
31.03Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
31.03Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
31.03Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
31.03Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
30.77Single4AMIBucindolol4AMI-β1-Bucindolol
30.77Single4LDEBI1671074LDE-β2-BI167107
30.77Single4RWADIPP-NH24RWA-δ-DIPP-NH2
30.77Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
30.77Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
30.77Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
30.77Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
30.77Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
30.77Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
30.77Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
30.77Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
30.77Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
30.77Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
30.77Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
30.77Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
30.77Single8JJ8Formoterol8JJ8-β2-Formoterol
30.77Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
30.77Single8JWZAB9288JWZ-A2A-AB928-Na
30.77Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
30.77Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.77Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
30.77Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
30.77Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
30.77Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
30.77Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
30.77Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
30.77Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
30.77Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
30.77Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
30.77Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
30.77Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
30.77Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
30.77Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
30.77Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
30.77Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
30.77Consensuslpa_offOrthosteric Ligandlpa1_off
30.77Consensuslpl_offOrthosteric Ligands1p_off lpa_off
30.77Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
30.77Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
30.77Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
30.77Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
30.77Consensusorexin_onOrthosteric Ligandox2_on
30.43Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
30.43Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
30.43Single5UVIZM-2413855UVI-A2A-ZM-241385
30.43Single6A94Zotepine6A94-5-HT2A-Zotepine
30.43Single6TPNHTL66416TPN-OX2-HTL6641
30.43Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
30.43Single7UL3Famotidine7UL3-H2-Famotidine
30.43Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
30.43Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
30.43Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
30.43Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
30.43Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
30.43Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
30.43Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
30.43Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
30.43Single9BJKNaloxone9BJK-μ-Naloxone-NAM
30.30Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
30.00Single6PT2KGCHM076PT2-δ-KGCHM07
30.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
30.00Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
30.00Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.00Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
30.00Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
30.00Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
30.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
30.00Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
30.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
29.63Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
29.63Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
29.63Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
29.63Single5X93K-87945X93-ETB-K-8794
29.63Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
29.63Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
29.63Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
29.63Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.63Single7UM4AS26747237UM4-5-HT5A-AS2674723
29.63Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
29.63Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
29.63Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
29.63Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
29.63Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
29.63Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
29.63Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
29.63Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.63Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
29.63Consensuschemerin_onOrthosteric Ligandcml1_on
29.63Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
29.63Consensusendothelin_offOrthosteric Ligandetb_off
29.63Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
29.63Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
29.63Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
29.63Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
29.63Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
29.17Single2Y04Salbutamol2Y04-β1-Salbutamol
29.17Single3EMLZM-2413853EML-A2A-ZM-241385
29.17Single3NY8ICI118-5513NY8-β2-ICI118-551
29.17Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
29.17Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
29.17Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
29.17Single4GBRS-Carazolol4GBR-β2-S-Carazolol
29.17Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
29.17Single5IU8Q274563475IU8-A2A-Q27456347-Na
29.17Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
29.17Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
29.17Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
29.17Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
29.17Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
29.17Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
29.17Single6S0LZM-2413856S0L-A2A-ZM-241385
29.17Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
29.17Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
29.17Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
29.17Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
29.17Single7PYRPSB-21157PYR-A2A-PSB-2115
29.17Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
29.17Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
29.17Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
29.17Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
29.17Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
29.17Single7WC7Lisuride7WC7-5-HT2A-Lisuride
29.17Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
29.17Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
29.17Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
29.17Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
29.17Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
29.17Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
29.17Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
29.17Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
29.17Single8JXRLSD8JXR-D1-LSD
29.17Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
29.17Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.17Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.17Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.17Single8X64Desloratadine8X64-H1-Desloratadine
29.17Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
29.17Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
29.17Single9CHXS-Carazolol9CHX-β2-S-Carazolol
29.17Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
29.17Consensus5ht5_onOrthosteric Ligand5ht5a_on
29.17Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
29.17Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
29.17Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
29.17Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
29.17Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
29.17Consensusblt_onOrthosteric Ligandblt1_on
29.17Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
29.17Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
29.17Consensusdopamine_offOrthosteric Ligandd2_off d3_off
29.17Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
29.17Consensusleukotriene_onOrthosteric Ligandblt_on
29.17Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
29.03Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
29.03Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
29.03Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
29.03Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
29.03Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
29.03Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
29.03Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
29.03Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
28.57Single3NY9ICI118-5513NY9-β2-ICI118-551
28.57Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
28.57Single5ZTYAM102575ZTY-CB2-AM10257
28.57Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
28.57Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
28.57Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
28.57Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
28.57Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
28.57Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
28.57Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
28.57Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
28.57Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
28.57Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
28.57Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
28.57Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
28.57Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
28.57Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
28.57Consensuskisspeptin_onOrthosteric Ligandkiss1_on
28.57Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
28.57Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
28.57Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
28.12Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
28.12Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
28.12Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
28.12Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
28.12Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
28.12Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
28.12Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
28.12Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
28.00Single2RH1S-Carazolol2RH1-β2-S-Carazolol
28.00Single2Y03Isoprenaline2Y03-β1-Isoprenaline
28.00Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
28.00Single5C1MBU725C1M-μ-BU72
28.00Single5TVNLSD5TVN-5-HT2B-LSD
28.00Single5WIUNemonapride5WIU-D4-Nemonapride
28.00Single5WIVNemonapride5WIV-D4-Nemonapride-Na
28.00Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
28.00Single5XPRBosentan5XPR-ETB-Bosentan
28.00Single6D26Fevipiprant6D26-DP2-Fevipiprant
28.00Single6E67BI1671076E67-β2-BI167107-Gs (fused)
28.00Single6PS6Timolol6PS6-β2-Timolol
28.00Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
28.00Single7W41PD1762527W41-BB2-PD176252
28.00Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
28.00Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
28.00Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
28.00Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
28.00Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
28.00Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8QOTNanobody-E8QOT-μ-Nanobody-E
28.00Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
28.00Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
28.00Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
28.00Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
28.00Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
28.00Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
28.00Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
28.00Consensusadenosine_offOrthosteric Liganda1_off a2_off
28.00Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
28.00Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
28.00Consensusamine_offonOrthosteric Ligandamine_off amine_on
28.00Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
28.00Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
28.00Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
28.00Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
28.00Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
28.00Consensusbombesin_offOrthosteric Ligandbb2_off
28.00Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
28.00Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.00Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
28.00Consensusdp_offOrthosteric Liganddp2_off
28.00Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
28.00Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
28.00Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
28.00Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
28.00Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
28.00Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
28.00Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.00Consensustrace-amine_onOrthosteric Ligandta1_on
27.59Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
27.59Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
27.59Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
27.59Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
27.59Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
27.59Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
27.59Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
27.59Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
27.59Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
27.59Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
27.59Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
27.27Single4XT3Fractalkine4XT3-US28-Fractalkine
27.27Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
27.27Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
27.27Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
27.27Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
27.27Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
27.27Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
27.27Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
27.27Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
27.27Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
27.27Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
26.92Single2YDVNECA2YDV-A2A-NECA
26.92Single4U15Tiotropium4U15-M3-Tiotropium
26.92Single4UHRCGS216804UHR-A2A-CGS21680
26.92Single5G53NECA5G53-A2A-NECA-Gs
26.92Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
26.92Single6E59L-7607356E59-NK1-L-760735
26.92Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
26.92Single6H7JIsoprenaline6H7J-β1-Isoprenaline
26.92Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
26.92Single6OL9Tiotropium6OL9-M5-Tiotropium
26.92Single6OS1TRV0266OS1-AT1-TRV026
26.92Single6TQ7SB-3348676TQ7-OX1-SB-334867
26.92Single6WGTLSD6WGT-5-HT2A-LSD
26.92Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
26.92Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
26.92Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
26.92Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
26.92Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
26.92Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
26.92Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
26.92Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
26.92Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
26.92Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
26.92Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
26.92Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
26.92Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
26.92Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
26.92Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
26.92Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
26.92Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
26.92Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
26.92Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
26.92Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Consensusa2_onOrthosteric Liganda2b_on
26.92Consensusa2_on_gpOrthosteric Liganda2b_on_gp
26.92Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
26.92Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
26.92Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
26.92Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
26.92Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
26.92Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
26.92Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
26.92Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
26.92Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
26.92Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
26.92Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
26.92Consensustachykinin_offOrthosteric Ligandnk1_off
26.67Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
26.67Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
26.67Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
26.67Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
26.67Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
26.67Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
26.67Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
26.67Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
26.67Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
26.67Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
26.47Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.47Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
26.47Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
26.47Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.47Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.09Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
26.09Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
26.09Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
26.09Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
26.09Single6AKYMaraviroc6AKY-CCR5-Maraviroc
26.09Single6B73MP11046B73-κ-MP1104
26.09Single6ME2Ramelteon6ME2-MT1-Ramelteon
26.09Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
26.09Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
26.09Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
26.09Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
26.09Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
26.09Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
26.09Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
26.09Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
26.09Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
26.09Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
26.09Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
26.09Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
26.09Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
26.09Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
26.09Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
26.09Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
26.09Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
26.09Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
26.09Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
26.09Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
26.09Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
26.09Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
25.93Single5CXVTiotropium5CXV-M1-Tiotropium
25.93Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
25.93Single6CM4Risperidone6CM4-D2-Risperidone
25.93Single6OS2TRV0266OS2-AT1-TRV026
25.93Single6ZG4HTL00099366ZG4-M1-HTL0009936
25.93Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
25.93Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
25.93Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
25.93Single7K15MKD0467K15-BLT1-MKD046-Na
25.93Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
25.93Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
25.93Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.93Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
25.93Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
25.93Single8JWY2-1188JWY-A2A-2-118
25.93Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
25.93Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
25.93Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
25.93Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
25.93Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
25.93Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
25.93Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
25.93Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
25.93Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
25.93Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
25.93Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
25.93Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
25.93Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
25.93Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
25.93Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
25.93Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
25.93Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
25.93Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.93Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.81Single3OE0CVX153OE0-CXCR4-CVX15
25.81Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
25.81Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
25.81Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
25.71Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
25.71Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
25.71Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single3REYXAC3REY-A2A-XAC
25.00Single3RZECidoxepin3RZE-H1-Cidoxepin
25.00Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
25.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
25.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
25.00Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
25.00Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
25.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
25.00Single5IUBQ274563445IUB-A2A-Q27456344-Na
25.00Single5JTBZM-2413855JTB-A2A-ZM-241385
25.00Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
25.00Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
25.00Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
25.00Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
25.00Single6AQFZM-2413856AQF-A2A-ZM-241385
25.00Single6H7LDobutamine6H7L-β1-Dobutamine
25.00Single6KUXRS-799486KUX-α2a-RS-79948
25.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
25.00Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
25.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
25.00Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
25.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
25.00Single6PS4ICI118-5516PS4-β2-ICI118-551
25.00Single6PS5S-Propranolol6PS5-β2-S-Propranolol
25.00Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
25.00Single6TPGEMPA6TPG-OX2-EMPA
25.00Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
25.00Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
25.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
25.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
25.00Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
25.00Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
25.00Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
25.00Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
25.00Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
25.00Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
25.00Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
25.00Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
25.00Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
25.00Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.00Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
25.00Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
25.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
25.00Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
25.00Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
25.00Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
25.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
25.00Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
25.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
25.00Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
25.00Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
25.00Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
25.00Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
25.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
25.00Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
25.00Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
25.00Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
25.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
25.00Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
25.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
25.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
25.00Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
25.00Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
25.00Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
25.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
25.00Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
25.00Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
25.00Consensusa2_offOrthosteric Liganda2a_off
25.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
25.00Consensusalpha1_onOrthosteric Ligandalpha1a_on
25.00Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
25.00Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
25.00Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
25.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
25.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
25.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
25.00Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
25.00Consensusprostanoid_offOrthosteric Ligandep_off dp_off
24.24Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
24.24Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
24.24Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
24.14Single6PT3DPI-2876PT3-δ-DPI-287
24.14Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
24.14Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
24.14Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
24.14Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
24.14Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
24.14Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
24.14Single8XQJJN2418XQJ-Apelin-JN241
24.14Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
24.14Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
24.14Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
24.14Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
24.00Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
24.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
24.00Single2Y01Dobutamine2Y01-β1-Dobutamine
24.00Single2Y02Carmoterol2Y02-β1-Carmoterol
24.00Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
24.00Single4MQSIperoxo4MQS-M2-Iperoxo
24.00Single4U14Tiotropium4U14-M3-Tiotropium
24.00Single5UIGCmpd-15UIG-A2A-Cmpd-1
24.00Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
24.00Single6D27CAY104716D27-DP2-CAY10471
24.00Single6H7MSalbutamol6H7M-β1-Salbutamol
24.00Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
24.00Single6PS1Timolol6PS1-β2-Timolol
24.00Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
24.00Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
24.00Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
24.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
24.00Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
24.00Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
24.00Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
24.00Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
24.00Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
24.00Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
24.00Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
24.00Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
24.00Single7UL4Alvimopan7UL4-μ-Alvimopan
24.00Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
24.00Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
24.00Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
24.00Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
24.00Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
24.00Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
24.00Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
24.00Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
24.00Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
24.00Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
24.00Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
24.00Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
24.00Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
24.00Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
24.00Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
24.00Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
24.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
24.00Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
24.00Single8JJOAlprenolol8JJO-β2-Alprenolol
24.00Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
24.00Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
24.00Single8K5DGSK2560738K5D-HCA2-GSK256073
24.00Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
24.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
24.00Single8T1WCVN4248T1W-GPR6-CVN424
24.00Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
24.00Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
24.00Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
24.00Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
24.00Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
24.00Single8X63Mepyramine8X63-H1-Mepyramine
24.00Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
24.00Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
24.00Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
24.00Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
24.00Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
24.00Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
24.00Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
24.00Consensusalpha2_onOrthosteric Ligandalpha2b_on
24.00Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
24.00Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
24.00Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
24.00Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
24.00Consensuscck_offOrthosteric Ligandccka_off
24.00Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
24.00Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
24.00Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
24.00Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
24.00Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
24.00Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
24.00Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
24.00Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
24.00Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
24.00Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
24.00Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
24.00Consensushca_on_gpOrthosteric Ligandhca2_on_gp
24.00Consensushistamine_offOrthosteric Ligandh1_off
23.81Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
23.81Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
23.53Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
23.53Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
23.53Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
23.53Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
23.53Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
23.53Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
23.33Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
23.33Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
23.33Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
23.33Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
23.33Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
23.33Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.33Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
23.33Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
23.33Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
23.33Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single2Y00Dobutamine2Y00-β1-Dobutamine
23.08Single4NTJAZD12834NTJ-P2Y12-AZD1283
23.08Single5JQHS-Carazolol5JQH-β2-S-Carazolol
23.08Single5N2RPSB-365N2R-A2A-PSB-36-Na
23.08Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
23.08Single5WQCEMPA5WQC-OX2-EMPA
23.08Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
23.08Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
23.08Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
23.08Single6LUQHaloperidol6LUQ-D2-Haloperidol
23.08Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
23.08Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
23.08Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
23.08Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
23.08Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
23.08Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
23.08Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
23.08Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
23.08Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
23.08Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
23.08Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
23.08Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.08Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
23.08Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8GNEKW-63568GNE-A2A-KW-6356-Na
23.08Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
23.08Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
23.08Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
23.08Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
23.08Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
23.08Single8TF5Oleic acid8TF5-GPR6-Oleic acid
23.08Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
23.08Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
23.08Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
23.08Consensusa3_on_gpOrthosteric Liganda3a_on_gp
23.08Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.08Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.08Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
23.08Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
23.08Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
23.08Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
23.08Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
23.08Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
23.08Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
23.08Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
23.08Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
23.08Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
23.08Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.08Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.08Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
23.08Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
22.86Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
22.86Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
22.86Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
22.86Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
22.73Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
22.73Single6ME5Agomelatine6ME5-MT1-Agomelatine
22.73Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
22.73Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.73Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
22.73Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
22.73Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
22.73Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
22.73Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
22.58Single6HLOAprepitant6HLO-NK1-Aprepitant
22.58Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
22.58Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
22.22Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
22.22Single4DJHJDTic4DJH-κ-JDTic
22.22Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
22.22Single5TZRMK86665TZR-FFA1-MK8666
22.22Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
22.22Single5XR8AM8415XR8-CB1-AM841
22.22Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
22.22Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
22.22Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
22.22Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
22.22Single7F1TMIP-1a7F1T-CCR5-MIP-1a
22.22Single7FEECP559407FEE-CB1-CP55940-ZCZ011
22.22Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
22.22Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
22.22Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
22.22Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
22.22Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
22.22Single8EA0Iperoxo8EA0-M3-Iperoxo
22.22Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
22.22Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
22.22Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
22.22Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
22.22Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
22.22Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
22.22Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
22.22Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
22.22Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
22.22Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
22.22Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
22.22Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
22.22Single8XVLZibotentan8XVL-ETA-Zibotentan
22.22Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
22.22Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
22.22Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
22.22Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
22.22Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
22.22Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
22.22Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
22.22Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
22.22Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
22.22Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
22.22Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
22.22Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
22.22Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
22.22Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
22.22Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
22.22Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
22.22Consensuslpa_onOrthosteric Ligandlpa1_on
22.22Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
22.22Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
22.22Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
22.22Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
21.95Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
21.95Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
21.88Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
21.88Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
21.88Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
21.74Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
21.74Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
21.74Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
21.74Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
21.74Single3PBLEticlopride3PBL-D3-Eticlopride
21.74Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
21.74Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
21.74Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
21.74Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
21.74Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
21.74Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
21.74Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
21.74Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
21.74Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
21.74Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
21.74Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.74Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.74Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
21.74Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
21.74Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
21.74Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
21.74Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
21.74Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
21.74Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
21.62Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
21.62Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
21.43Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
21.43Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
21.43Single4PY02MeSATP4PY0-P2Y12-2MeSATP
21.43Single4XEENeurotensin4XEE-NTS1-Neurotensin
21.43Single4XESNeurotensin4XES-NTS1-Neurotensin
21.43Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
21.43Single6KQICP559406KQI-CB1-CP55940-Org27569
21.43Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
21.43Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
21.43Single6YVRNTS8-136YVR-NTS1-NTS8-13
21.43Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
21.43Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
21.43Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
21.43Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
21.43Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
21.43Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
21.43Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
21.43Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
21.43Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
21.43Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
21.43Single8XYIVUF106618XYI-CXCR3-VUF10661
21.43Consensusalpha1_offOrthosteric Ligandalpha1a_off
21.43Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
21.43Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
21.43Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
21.43Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
21.43Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
21.43Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
21.43Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
21.43Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
21.43Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
21.43Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
21.43Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
21.21Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
21.21Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
21.21Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
21.21Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
21.21Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
21.05Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
21.05Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
21.05Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
21.05Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
20.83Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
20.83Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
20.83Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
20.83Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
20.83Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
20.83Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
20.83Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
20.83Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
20.83Single6AKXA4R6AKX-CCR5-A4R
20.83Single6DS0Ly2660976DS0-5-HT2B-Ly266097
20.83Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
20.83Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
20.83Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.83Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
20.83Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
20.83Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
20.83Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
20.83Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
20.83Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
20.83Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
20.83Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
20.83Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
20.83Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
20.83Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
20.83Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
20.83Single8GNGIstradefylline8GNG-A2A-Istradefylline
20.83Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
20.83Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
20.83Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
20.83Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
20.83Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
20.83Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
20.83Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
20.83Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
20.83Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
20.83Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
20.83Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
20.83Single8Y0HVUF114188Y0H-CXCR3-VUF11418
20.83Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
20.83Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
20.83Consensusalpha2_offOrthosteric Ligandalpha2c_off
20.83Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
20.83Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
20.83Consensusorexin_offOrthosteric Ligandox2_off ox1_off
20.83Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
20.83Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
20.83Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.69Single4BUONeurotensin4BUO-NTS1-Neurotensin
20.69Single6K1QIRL25006K1Q-ETB-IRL2500
20.69Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
20.69Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
20.69Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
20.69Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
20.69Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
20.69Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.69Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
20.69Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
20.69Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
20.69Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
20.69Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
20.69Single8XWFCXCL38XWF-CXCR2-CXCL3
20.69Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
20.69Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
20.69Consensuscck_onOrthosteric Ligandccka_on cckb_on
20.69Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
20.69Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
20.69Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
20.69Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
20.69Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
20.59Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
20.59Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
20.59Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
20.59Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
20.59Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
20.59Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
20.59Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.59Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.00Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
20.00Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
20.00Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
20.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
20.00Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
20.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
20.00Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
20.00Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
20.00Single6IQLL7458706IQL-D4-L745870
20.00Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
20.00Single6KNMJN241-96KNM-Apelin-JN241-9
20.00Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
20.00Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
20.00Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
20.00Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
20.00Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
20.00Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
20.00Single7AROLUF58337ARO-A2A-LUF5833-Na
20.00Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
20.00Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
20.00Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
20.00Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
20.00Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
20.00Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
20.00Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
20.00Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
20.00Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
20.00Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
20.00Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
20.00Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
20.00Single7SK3CXCL127SK3-ACKR3-CXCL12
20.00Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
20.00Single7VODCariprazine7VOD-5-HT2A-Cariprazine
20.00Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
20.00Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
20.00Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
20.00Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
20.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
20.00Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
20.00Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
20.00Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
20.00Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
20.00Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
20.00Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
20.00Single8K5CAcipimox8K5C-HCA2-Acipimox
20.00Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
20.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
20.00Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
20.00Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
20.00Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
20.00Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
20.00Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
20.00Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
20.00Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
20.00Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
20.00Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
20.00Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
20.00Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
20.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
20.00Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
20.00Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
20.00Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
20.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
20.00Consensushca_onOrthosteric Ligandhca2_on
20.00Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
20.00Consensusopsins_offOrthosteric Ligandrhodopsin_off
20.00Consensussensory_offOrthosteric Ligandopsins_off
19.44Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
19.44Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
19.44Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
19.35Single4XT1Fractalkine4XT1-US28-Fractalkine
19.35Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
19.35Single7F8XNN90567F8X-CCKA-NN9056
19.35Single7QA8Peptide7QA8-STE2-Peptide
19.35Single7QA8Peptide7QA8-STE2-Peptide
19.35Single8IEBA1LYA8IEB-GPR156-A1LYA
19.35Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.35Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
19.35Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
19.35Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
19.35Single8XWNCXCL88XWN-CXCR2-CXCL8
19.35Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
19.23Single4DAJTiotropium4DAJ-M3-Tiotropium
19.23Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
19.23Single4EJ4Naltrindole4EJ4-δ-Naltrindole
19.23Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
19.23Single4QKX35V4QKX-β2-35V
19.23Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
19.23Single5DHGC-355DHG-NOP-C-35
19.23Single5DSGTiotropium5DSG-M4-Tiotropium
19.23Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
19.23Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
19.23Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
19.23Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
19.23Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
19.23Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
19.23Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
19.23Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
19.23Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
19.23Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
19.23Single6TOTLemborexant6TOT-OX1-Lemborexant
19.23Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7BU7BI1671077BU7-β1-BI167107
19.23Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
19.23Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
19.23Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
19.23Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
19.23Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
19.23Single7V3ZCP559407V3Z-CB1-CP55940
19.23Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
19.23Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
19.23Single8CU6LJ-45178CU6-A2A-LJ-4517
19.23Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
19.23Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.23Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
19.23Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
19.23Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
19.23Single8RLNLUF58348RLN-A2A-LUF5834
19.23Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
19.23Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
19.23Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
19.23Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
19.23Single9IYAONO-97105319IYA-GPR55-ONO-9710531
19.23Consensusa3_onOrthosteric Liganda3a_on
19.23Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
19.23Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
19.23Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
19.23Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
19.23Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
19.23Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
19.23Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
19.23Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
19.23Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
19.23Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
19.23Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
19.15Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
19.05Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
19.05Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
18.92Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
18.92Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
18.92Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
18.92Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
18.92Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
18.92Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
18.75Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
18.75Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
18.75Single7SK5CXCL127SK5-ACKR3-CXCL12
18.75Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
18.75Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
18.75Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
18.75Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.75Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
18.52Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
18.52Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
18.52Single5N2SPSB365N2S-A1-PSB36
18.52Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
18.52Single6HLPNetupitant6HLP-NK1-Netupitant
18.52Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
18.52Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
18.52Single6TP6Filorexant6TP6-OX1-Filorexant
18.52Single7C4SS1P7C4S-S1P3-S1P
18.52Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
18.52Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
18.52Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
18.52Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
18.52Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
18.52Single7WC6LSD7WC6-5-HT2A-LSD
18.52Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
18.52Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.52Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
18.52Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
18.52Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
18.52Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
18.52Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
18.52Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
18.52Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
18.52Consensusblt_offOrthosteric Ligandblt1_off
18.52Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
18.52Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
18.42Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
18.18Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
18.18Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
18.18Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
18.18Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
18.18Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
18.18Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
18.18Single9CHUNoradrenaline9CHU-β2-Noradrenaline
18.18Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
18.18Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.18Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
18.18Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
18.18Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
18.18Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
18.18Consensussensory_onOrthosteric Ligandopsins_on
17.95Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
17.95Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
17.86Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
17.86Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
17.86Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
17.86Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
17.86Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
17.86Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
17.86Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
17.86Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
17.86Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
17.86Single7R0CAVP7R0C-V2-AVP-Arrestin2
17.86Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
17.86Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
17.86Single7TUYGSK682753A7TUY-GPR183-GSK682753A
17.86Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
17.86Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
17.86Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
17.86Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
17.86Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
17.86Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
17.86Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
17.86Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
17.86Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
17.86Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
17.86Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
17.86Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensusneurotensin_onOrthosteric Ligandnts1_on
17.86Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
17.86Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.65Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
17.65Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
17.65Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
17.65Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
17.65Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
17.65Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
17.65Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
17.65Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
17.65Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
17.65Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
17.50Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
17.50Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
17.39Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
17.39Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
17.39Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
17.39Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
17.39Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
17.39Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
17.39Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
17.39Single7WC5Psilocin7WC5-5-HT2A-Psilocin
17.39Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
17.39Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
17.39Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
17.39Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
17.39Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
17.39Consensus5ht2_onOrthosteric Ligand5ht2b_on
17.39Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
17.39Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
17.24Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
17.24Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
17.24Single4N4WSANT-14N4W-SMO-SANT-1
17.24Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
17.24Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
17.24Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
17.24Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
17.24Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.24Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
17.24Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
17.24Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
17.24Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
17.24Single8XQJJN2418XQJ-Apelin-JN241
17.24Single8XWACXCL18XWA-CXCR2-CXCL1
17.24Single8XWMCXCL68XWM-CXCR2-CXCL6
17.24Single8XWSCXCL58XWS-CXCR2-CXCL5
17.24Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
17.24Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
17.24Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
17.14Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
17.07Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
17.07Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
17.07Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
16.67Single3OE9IT1t3OE9-CXCR4-IT1t
16.67Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
16.67Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
16.67Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
16.67Single6FJ3PTH6FJ3-PTH1-PTH
16.67Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
16.67Single6HLLCP999946HLL-NK1-CP99994
16.67Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
16.67Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
16.67Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
16.67Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
16.67Single6TP4ACT-4622066TP4-OX1-ACT-462206
16.67Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
16.67Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
16.67Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
16.67Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
16.67Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
16.67Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
16.67Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
16.67Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
16.67Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
16.67Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
16.67Single7SRQLSD7SRQ-5-HT2B-LSD
16.67Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
16.67Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
16.67Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
16.67Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
16.67Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
16.67Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
16.67Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
16.67Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
16.67Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
16.67Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
16.67Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
16.67Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
16.67Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
16.67Single8XVJMacitentan8XVJ-ETA-Macitentan
16.67Single8XVUCXCL28XVU-CXCR2-CXCL2
16.67Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
16.67Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
16.67Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
16.67Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
16.67Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
16.67Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
16.67Consensusgq_nucleotideOrthosteric Ligandgq_p2y
16.67Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
16.22Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
16.22Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
16.22Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
16.22Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
16.22Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
16.22Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
16.13Single5EE7MK08935EE7-Glucagon-MK0893
16.13Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
16.13Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
16.13Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
16.13Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
16.13Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
16.13Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
16.00Single3PWHZM-2413853PWH-A2A-ZM-241385
16.00Single4BWBNeurotensin4BWB-NTS1-Neurotensin
16.00Single5WS3EMPA5WS3-OX2-EMPA
16.00Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
16.00Single6TODEMPA6TOD-OX1-EMPA-Na
16.00Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
16.00Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
16.00Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
16.00Single7F8ULintitript7F8U-CCKA-Lintitript
16.00Single7F8YDevazepide7F8Y-CCKA-Devazepide
16.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
16.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
16.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
16.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
16.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
16.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
16.00Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
16.00Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
16.00Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
16.00Single7XRRLemborexant7XRR-OX2-Lemborexant
16.00Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
16.00Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
16.00Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
16.00Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
16.00Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
16.00Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
16.00Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
16.00Single8IWESpermidine8IWE-TA9-Spermidine
16.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
16.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
16.00Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
16.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
16.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
16.00Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
16.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
16.00Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
16.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
16.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
16.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
16.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
16.00Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
16.00Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
16.00Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
16.00Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
16.00Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
16.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
16.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
16.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.79Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
15.79Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
15.79Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
15.62Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
15.62Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8IEIA1LYA8IEI-GPR156-A1LYA
15.62Single8IEPA1LYA8IEP-GPR156-A1LYA
15.62Single8IEPA1LYA8IEP-GPR156-A1LYA
15.62Single8KIGSHU91198KIG-MC3-SHU9119-Ca
15.62Single8WKYPG-9348WKY-MC4-PG-934
15.62Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
15.62Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
15.62Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
15.62Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
15.62Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.56Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
15.38Single2YDOAdenosine2YDO-A2A-Adenosine
15.38Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
15.38Single6FFIMMPEP6FFI-mGlu5-MMPEP
15.38Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
15.38Single6TPKRetosiban6TPK-OT-Retosiban
15.38Single6V9SGTPL114036V9S-OX1-GTPL11403
15.38Single6ZG9GSK10347026ZG9-M1-GSK1034702
15.38Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
15.38Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
15.38Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
15.38Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
15.38Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
15.38Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.38Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
15.38Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
15.38Single8IHKAcifran8IHK-HCA3-Acifran
15.38Single8K2WAMG4878K2W-CXCR3-AMG487
15.38Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
15.38Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
15.38Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
15.38Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
15.38Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
15.38Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
15.38Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
15.38Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
15.38Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
15.38Consensusgrh_offOrthosteric Ligandgnrh1_off
15.38Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
15.38Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
15.38Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.38Consensusvasop-oxy_offOrthosteric Ligandot_off
15.22Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
15.15Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
15.15Single8IEBA1LYA8IEB-GPR156-A1LYA
15.15Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
15.15Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
15.00Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
15.00Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
14.81Single4YAYZD-71554YAY-AT1-ZD-7155
14.81Single5DHHSB-6121115DHH-NOP-SB-612111
14.81Single5UENDU1725UEN-A1-DU172
14.81Single6FFHFenobam6FFH-mGlu5-Fenobam
14.81Single6GPSMK08126GPS-CCR2-MK0812
14.81Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
14.81Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
14.81Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
14.81Single7F83PF-051904577F83-Ghrelin-PF-05190457
14.81Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
14.81Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
14.81Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
14.81Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
14.81Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
14.81Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
14.81Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
14.81Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
14.81Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
14.81Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
14.71Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
14.71Single6W25SHU91196W25-MC4-SHU9119-Ca
14.71Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.63Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
14.63Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
14.29Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
14.29Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
14.29Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
14.29Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
14.29Single6GPXMK08126GPX-CCR2-MK0812
14.29Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
14.29Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
14.29Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
14.29Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
14.29Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
14.29Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
14.29Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
14.29Single7SINNPS-21437SIN-CaS-NPS-2143
14.29Single7SINNPS-21437SIN-CaS-NPS-2143
14.29Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
14.29Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
14.29Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
14.29Single8S4DCMF-0198S4D-Apelin-CMF-019
14.29Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
14.29Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
14.29Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
14.29Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
14.29Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
14.29Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
14.29Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
14.29Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
14.29Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
13.95Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
13.89Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
13.89Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
13.79Single4BV0Neurotensin4BV0-NTS1-Neurotensin
13.79Single5XRAAM115425XRA-CB1-AM11542
13.79Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
13.79Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
13.79Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
13.79Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
13.79Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
13.79Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
13.79Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
13.79Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
13.79Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
13.79Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
13.79Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
13.79Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
13.79Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
13.64Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
13.64Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
13.64Single7WC4Serotonin7WC4-5-HT2A-Serotonin
13.64Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
13.64Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
13.51Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
13.51Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
13.33Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
13.33Single5X33BIIL2605X33-BLT1-BIIL260
13.33Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
13.33Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
13.33Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
13.16Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
13.16Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
13.16Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
13.16Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
13.04Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
13.04Single3RFMCaffeine3RFM-A2A-Caffeine
13.04Single6TQ9SB-4081246TQ9-OX1-SB-408124
13.04Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
13.04Single8A2OTheophylline8A2O-A2A-Theophylline-Na
13.04Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
13.04Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
12.90Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
12.90Single5CGDHTL142425CGD-mGlu5-HTL14242
12.90Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
12.90Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
12.82Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
12.82Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
12.82Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
12.82Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
12.82Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
12.50Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
12.50Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
12.50Single3OE6IT1t3OE6-CXCR4-IT1t
12.50Single3UZAGTPL92363UZA-A2A-GTPL9236
12.50Single4XNWMRS25004XNW-P2Y1-MRS2500
12.50Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
12.50Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
12.50Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
12.50Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
12.50Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
12.50Single8IEIA1LYA8IEI-GPR156-A1LYA
12.50Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
12.50Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
12.50Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
12.50Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
12.50Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
12.50Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
12.50Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
12.50Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
12.50Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
12.50Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Consensusgi_sensoryOrthosteric Ligandgi_opsins
12.50Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.50Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.50Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
12.20Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
12.12Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
12.12Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
12.00Single4O9RCyclopamine4O9R-SMO-Cyclopamine
12.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
12.00Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
12.00Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
12.00Single8K5BNiacin8K5B-HCA2-Niacin
12.00Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
12.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
12.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
12.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
12.00Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
12.00Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
12.00Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
12.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
12.00Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
11.90Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
11.90Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.76Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
11.76Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
11.63Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
11.54Single3ODUIT1t3ODU-CXCR4-IT1t
11.54Single4QINSAG1.54QIN-SMO-SAG1.5
11.54Single4S0VSuvorexant4S0V-OX2-Suvorexant
11.54Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
11.54Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
11.54Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
11.54Single6TPJSuvorexant6TPJ-OX2-Suvorexant
11.54Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
11.54Single7BR3Elagolix7BR3-GnRH1-Elagolix
11.54Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
11.54Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
11.54Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
11.54Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
11.54Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
11.54Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
11.54Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
11.54Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
11.54Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
11.54Consensusangiotensin_offOrthosteric Ligandat1_off
11.54Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
11.54Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
11.54Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.54Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
11.43Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.43Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.11Single6TP3Nemorexant6TP3-OX1-Nemorexant
11.11Single6VI4JDTic6VI4-κ-JDTic
11.11Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
11.11Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
11.11Single6ZINSR486926ZIN-NTS1-SR48692
11.11Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
11.11Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
11.11Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
11.11Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
11.11Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
11.11Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
11.11Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
11.11Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
10.81Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
10.81Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
10.81Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
10.71Single5T04Neurotensin5T04-NTS1-Neurotensin
10.71Single5TGZAM65385TGZ-CB1-AM6538
10.71Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
10.71Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
10.71Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
10.71Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
10.71Single7YXAONO-54306087YXA-S1P5-ONO-5430608
10.71Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
10.34Single4JKVTaladegib4JKV-SMO-Taladegib
10.34Single5CGCHTL142425CGC-mGlu5-HTL14242
10.34Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
10.34Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
10.34Single6Z4SSR486926Z4S-NTS1-SR48692
10.34Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
10.34Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
10.34Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
10.34Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
10.34Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
10.34Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
10.00Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
10.00Single5V56TC1145V56-SMO-TC114
10.00Single5V57TC1145V57-SMO-TC114
10.00Single7P2L4YI7P2L-mGlu5-4YI
10.00Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
10.00Single9BJKNAM9BJK-μ-Naloxone-NAM
9.68Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
9.68Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
9.52Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
9.38Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
9.38Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
9.38Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single5MZPCaffeine5MZP-A2A-Caffeine-Na
9.09Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
9.09Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
9.09Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
9.09Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
9.09Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
8.82Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.70Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
8.70Single8PWNTheophylline8PWN-A2A-Theophylline
8.70Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
8.57Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.33Single3OE8IT1t3OE8-CXCR4-IT1t
8.33Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
8.33Consensusp2y_offOrthosteric Ligandp2y1_off
8.11Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
8.11Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
8.11Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
8.00Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
8.00Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
8.00Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
8.00Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
8.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.69Single5L7IVismodegib5L7I-SMO-Vismodegib
7.69Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.69Single7UL2SR486927UL2-NTS1-SR48692-Na
7.69Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
7.69Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
7.69Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
7.69Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
7.69Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Consensusneurotensin_offOrthosteric Ligandnts1_off
7.69Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
7.50Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
7.41Single4K5YCP-3763954K5Y-CRF1-CP-376395
7.41Single5ZKQABT-4915ZKQ-PAF-ABT-491
7.41Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
7.41Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.41Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.41Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
7.41Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
7.41Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
7.41Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
7.14Single7VV6C48/807VV6-MRGPRX2-C48/80
7.14Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single8IYXYL-3658IYX-GPR34-YL-365
6.90Single4QIMANTA XV4QIM-SMO-ANTA XV
6.90Single4Z9GCP-3763954Z9G-CRF1-CP-376395
6.90Single8GTIBMK-C2058GTI-CRF1-BMK-C205
6.90Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.90Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
6.90Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
6.90Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
6.67Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
6.67Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
6.67Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
6.67Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
6.67Single8GTGBMK-I1528GTG-CRF1-BMK-I152
6.67Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
6.67Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.67Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
6.67Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
6.67Consensusep_offOrthosteric Ligandep4_off
6.45Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
6.25Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
6.25Single8GTMBMK-C2038GTM-CRF1-BMK-C203
6.25Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
6.06Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
6.06Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
6.06Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
5.88Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
5.88Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
5.71Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
5.71Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
5.56Single7SHEPI; PE7SHE-GPR158-PI; PE
4.35Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
4.17Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
4.17Single8HS2Fab0468HS2-GPR20-Fab046
4.17Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
4.00Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
4.00Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
4.00Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
4.00Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
4.00Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
3.85Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
3.85Single7F61Cholesterol7F61-H3-PF-03654746-Cholesterol
3.85Single8JPSCCL78JPS-ACKR1-CCL7
3.70Single6LI0C176LI0-GPR52-C17
3.70Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
3.70Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
3.70Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
3.70Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
3.70Single9B9Y7DY9B9Y-CB1-7DY
3.57Single6C1QNDT95137276C1Q-C5a1-PMX53-NDT9513727
3.57Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
3.57Single9BA0A1AKN9BA0-CB1-A1AKN
3.45Single8JD6N-(3-chlorophenyl)pyridine-2-carboxamide8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
3.45Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
3.33Single6IIVDaltroban6IIV-TP-Daltroban
3.33Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
3.33Single9B9ZA1AKO9B9Z-CB1-A1AKO
3.12Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
3.12Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
3.12Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
3.12Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
3.03Single6IIURamatroban6IIU-TP-Ramatroban
3.03Single7SHEPI; PE7SHE-GPR158-PI; PE
2.94Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
2.78Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
2.70Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
2.70Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7

Consensus Members
Id Members
7WVX 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
7T6U 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
7T6V 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
7WVY 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
7T6S 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
6OMM 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
Net Summary
Imin 3.04167
Number of Linked Nodes 912
Number of Links 1113
Number of Hubs 171
Number of Links mediated by Hubs 648
Number of Communities 22
Number of Nodes involved in Communities 246
Number of Links involved in Communities 358
Path Summary
Number Of Nodes in MetaPath 79
Number Of Links MetaPath 78
Number of Shortest Paths 5226197
Length Of Smallest Path 3
Average Path Length 49.0182
Length of Longest Path 78
Minimum Path Strength 0.29
Average Path Strength 6.63633
Maximum Path Strength 21.1917
Minimum Path Correlation 0.7
Average Path Correlation 0.991716
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.35135
Average % Of Corr. Nodes 26.7295
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 48.4578
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
formylpeptide_on_gpfpr2-alx_on_gp
fpr1-alx_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download fpr2-alx_on_gp.zip



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