Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.hfs2.07 2.77125409
2G.S2.05 8.583754153
3G.S2.08 8.6525475
4G.S3.03 6.54417677
5G.S3.04 8.3654156
6G.S3.06 10.72124155
7G.H2.06 6.59409
8G.H2.07 5.0885139
9G.H2.09 5.7675448
10G.H2.10 4.9675447
11G.h2s4.01 8.3045139
12G.S4.02 5.514208
13G.S4.04 7.9425409
14G.s4h3.04 11.1225498
15G.s4h3.05 11.2475499
16G.H3.06 4.46625466
17G.H3.09 5.48083609
18G.H3.17 8.19417645
19G.H3.18 5.9155209
20G.S5.05 4.58875409
21G.S5.07 4.5415219
22G.s5hg.01 5.10125409
23G.HG.04 6.87333699
24G.HG.07 5.25125499
25G.hgh4.02 5.42571767
26G.hgh4.05 11.2612467
27G.H4.05 5.8375464
28G.H4.15 4.95375408
29G.H4.16 4.988754243
30G.h4s6.02 5.2554238
31G.H5.03 6.0325408
32G.H5.08 5.91667678
33G.H5.20 3.31409
34G.H5.26 7.4325405
35b.1x15 2.6675407
36b.1x19 5.62436
37b.lh12x2 4.8975408
38b.lhb1x3 3.8425402
39b.lhb1x6 5.398754263
40b.l1x3 8.96417629
41b.b2x1 7.59667648
42b.b2x3 5.03125426
43b.b2x5 6.45583627
44b.b3x2 5.62375425
45b.l3x2 5.705429
46b.b4x2 5.1825408
47b.b4x6 11.669529
48b.b5x2 6.475407
49b.b5x3 7.48083629
50b.b5x7 8.14875407
51b.l5x1 5.4915168
52b.l5x5 9.47917609
53b.b6x5 3.86667606
54b.b7x1 6.68754284
55b.b8x3 3.746254286
56b.b8x4 6.60625406
57b.l8x3 3.57625403
58b.l9x3 7.7975119
59b.l9x6 5.8165138
60b.b10x5 5.066509
61b.l10x1 3.2875293
62b.b11x4 4.723754119
63b.b12x6 10.21586118
64b.b12x7 5.818754179
65b.b13x7 8.247557
66b.l13x3 8.461559
67b.l13x7 4.55125459
68b.b15x2 7.1725436
69b.l15x2 6.4375409
70b.b16x4 9.7425456
71b.b16x6 8.065658
72b.b17x7 9.13625438
73b.l17x3 8.6175639
74b.b18x3 5.469538
75b.b18x5 4.691535
76b.l18x1 7.181676126
77b.l18x2 6.023754127
78b.b19x2 7.371536
79b.b19x4 6.935438
80b.l19x2 7.25375439
81b.b20x4 12.0487438
82b.b20x6 8.79667636
83b.b20x7 5.65583609
84b.l20x2 10.8387409
85b.b21x1 8.45625437
86b.b21x7 4.93505
87b.l21x2 4.72125484
88b.l21x5 3.624584
89b.b22x5 5.9095127
90b.l22x5 9.19754269
91b.b23x2 5.7825406
92b.b23x6 6.14857787
93b.l23x1 7.79375406
94b.b24x2 3.94405
95b.b24x4 5.96486
96b.b24x6 6.76488
97b.l24x3 3.88125405
98b.l25x3 7.1775449
99b.b26x3 4.7675406
100b.l26x5 4.656525
101b.b27x3 5.035408
102b.l27x1 8.33357749
103b.l27x2 7.678549
104b.b28x4 5.63446
105b.b28x6 9.093549
106b.b28x7 6.719529
107g.h1x11 2.78625409
108g.l1x4 3.07438
109g.h2x11 7.94754126
110g.ctx3 5.66083609
111g.ctx14 4.6725629
112g.ctx16 4.83833628
113Lig 10.43881210
1141x35 11.439514
1151x39 8.785415
1161x50 6.2925409
1171x56 3.87875408
1182x40 6.795836149
1192x42 6.48875408
1202x46 6.68125419
1212x50 6.745519
1222x56 5.42625407
1232x57 5.1375406
1243x22 6.1775313
1253x33 4.83875414
1263x35 7.61125406
1273x37 4.66917616
1283x50 4.84419
1293x53 9.7025108
130I2x53 9.4815108
1314x50 3.595409
1324x60 6.17125415
133E2.N150 4.564315
134E2.T154 5.824322
135E2.V171 3.515405
136E2.M172 6.2575404
1375x39 9.7525416
1385x40 5.26625415
1395x411 5.001254183
1405x42 6.31415
1415x44 8.22375405
1425x461 6.50667615
1435x58 3.86509
1445x66 5.12625405
1456x48 7.98518
1466x51 4.20625416
1476x59 7.383754184
148E3.V259 3.95375404
1497x35 13.495414
1507x38 8.3375415
1517x39 5.42625415
1527x42 7.014517
1537x49 8.00375419
1547x53 5.701519
1558x50 6.345148
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1G.HN.40 b.b5x2 23.55788.195NoYes077
2G.HN.40 b.b5x3 23.75487.65NoYes079
3b.b4x6 b.b5x3 25.595311.02YesYes299
4b.b3x2 b.b4x6 33.55685.125YesYes259
5b.b2x3 b.b3x2 33.15195.65YesYes265
6b.b26x2 b.b2x3 45.77834.86NoYes076
7b.b26x1 b.b26x2 46.15013.44NoNo097
8b.b26x1 b.l27x1 46.33814.94NoYes099
9G.H3.17 b.l27x1 46.50264.215YesYes459
10G.H3.15 G.H3.17 62.07977.91NoYes085
11G.H3.15 G.H3.18 62.14354.23NoYes089
12G.H3.18 G.S4.02 62.33838.79YesYes2098
13G.S4.02 G.S5.02 87.69695.885YesNo086
14G.H3.09 G.S5.02 87.76523.14YesNo096
15G.H3.09 G.H4.15 88.33785.36YesYes098
16G.H4.15 G.S5.04 90.64575.48YesNo089
17G.S5.04 G.S5.06 91.16846.225NoNo098
18G.S5.06 G.s4h3.01 91.89669.685NoNo087
19G.HG.04 G.s4h3.01 91.849812.79YesNo997
20G.H4.03 G.HG.04 89.29233.61NoYes049
21G.H4.03 G.HG.01 89.47658.36NoNo045
22G.HG.01 G.s6h5.02 89.51326.47NoNo057
23G.s6h5.02 G.s6h5.04 89.55134.225NoNo078
24G.H5.03 G.s6h5.04 89.63045.85YesNo088
25G.H5.03 G.s6h5.01 89.826712.43YesNo089
26G.S5.05 G.s6h5.01 94.58224.54YesNo099
27G.S5.03 G.S5.05 99.93085.65NoYes089
28G.H5.10 G.S5.03 99.97724.06NoNo068
29G.H5.10 G.S6.02 1004.67NoNo067
30G.S6.02 G.h4s6.12 50.179411.22NoNo074
31G.H5.17 G.h4s6.12 49.9994.725NoNo054
32G.H5.17 G.H5.26 99.63927.445NoYes055
33G.H5.20 G.H5.26 98.8465.48YesYes095
34G.H5.20 G.H5.25 89.80132.77YesNo097
353x50 G.H5.25 89.44963.035YesNo097
363x46 3x50 14.44795.01NoYes189
372x42 3x46 16.72093.77YesNo088
38G.H5.13 G.S6.02 49.84419.77NoNo087
39G.H5.13 G.H5.17 49.7996.915NoNo085
40b.b2x1 b.l27x1 10.56248.2YesYes489
41G.H5.16 G.H5.20 12.23332.85NoYes069
42G.H5.16 I2x50 11.67668.36NoNo068
43I2x50 I2x51 11.39783.965NoNo086
44G.S1.05 G.h2s4.01 25.049614.615NoYes099
45G.S1.07 G.S4.02 25.40243.565NoYes098
46G.s1h1.05 G.s5hg.01 10.23844.59NoYes099
47G.s1h1.05 G.s1h1.06 10.45813.71NoNo099
48G.S5.07 G.s1h1.06 10.53195.09YesNo099
49G.H2.09 G.H2.10 10.33284.42YesYes487
50G.H2.10 b.l7x2 18.40723.97YesNo079
51G.H2.07 b.l7x2 18.81623.42YesNo099
52G.H2.07 b.l9x6 37.89115.79YesYes1398
53G.H2.06 b.l15x1 36.61364.85YesNo097
54b.l13x6 b.l15x1 36.89273.89NoNo097
55b.l13x6 b.l9x6 37.17154.6NoYes098
56G.H2.06 b.l17x6 35.49427.605YesNo099
572x39 G.H5.22 10.19695.78NoNo084
582x39 3x53 10.50567.115NoYes1088
593x49 3x53 11.05869.53NoYes1098
602x42 3x49 12.318113.135YesNo089
61b.l17x5 b.l17x6 34.65154.42NoNo069
62b.b19x6 b.l17x5 33.17454.075NoNo396
63b.b19x6 b.l17x3 32.9586.975NoYes399
64b.b20x6 b.l17x3 20.11043.96YesYes369
65b.b17x7 b.b20x6 13.865516.08YesYes386
66b.b17x7 b.b21x1 13.41436.57YesYes387
67b.b21x1 g.l1x4 10.37584.165YesYes378
68b.l23x1 b.l25x6 20.951217.865YesNo068
69b.l21x7 b.l23x1 19.2484.665NoYes056
70b.b23x6 b.l21x7 17.53064.03YesNo875
71b.b23x6 b.b24x6 14.55397.72YesYes878
72b.b21x7 b.b24x6 14.47177.235YesYes058
73b.b5x2 b.l4x3 22.841110.97YesNo076
74b.b4x7 b.l4x3 22.673210.12NoNo086
75b.l2x5 b.l4x2 10.241224.18NoNo054
76b.l26x5 g.ctx4 14.05135.87YesNo057
77g.ctx3 g.ctx4 13.5064.025YesNo097
78b.b3x1 b.b4x7 26.78054.07NoNo058
79b.b3x1 b.b6x5 31.04162.93NoYes056
80b.b2x4 b.b6x5 27.47483.27NoYes066
81b.b10x4 b.b2x4 27.17567.335NoNo066
82b.b2x5 b.l26x1 12.587810.31YesNo277
83b.l26x1 b.l26x3 12.01566.505NoNo277
84b.l26x3 b.l26x5 12.05743.465NoYes275
85b.b10x4 b.b14x5 17.54864.86NoNo065
86b.b14x5 b.l10x1 16.9264.845NoYes2953
87b.b11x1 b.l10x1 16.01992.66NoYes053
88b.b11x1 b.l10x2 13.42753.915NoNo055
89b.l10x2 b.l10x3 13.11392.66NoNo056
90b.l10x3 b.l6x3 12.80018.095NoNo066
91b.l6x3 b.l6x5 12.48598.195NoNo064
92b.b7x1 b.l6x5 11.85673.49YesNo044
93b.b19x4 b.l17x3 10.497410.95YesYes389
94b.b18x3 b.b19x4 10.21563.8YesYes388
95b.b21x7 b.b23x2 10.87584.685YesYes056
96b.b22x5 b.b23x2 10.499511.57YesYes076
97b.l25x5 b.l27x1 15.48657.345NoYes479
983x33 Lig 10.66074.835YesYes140
993x36 Lig 34.513512.165NoYes160
1003x36 6x48 54.31344.85NoYes168
1016x44 6x48 55.668814.53NoYes088
1025x54 6x44 57.71984.35NoNo088
1035x54 5x58 58.13324.79NoYes089
1043x50 5x58 59.36233.6YesYes099
1053x33 3x37 10.41353.215YesYes146
1063x36 3x37 19.57713.425NoYes166
107E2x52 Lig 10.665244.415NoYes150
1083x43 7x53 20.2025.275NoYes189
1093x50 7x53 19.20937.715YesYes199
1103x43 7x49 10.11244.12NoYes189
1112x50 7x46 12.18315.89YesNo099
1122x53 2x56 10.31434.81NoYes087
1132x53 7x46 11.2455.655NoNo089
1143x29 E2.V171 22.61843.175NoYes045
1153x29 E2.M172 23.42186.775NoYes044
1163x33 E2.M172 20.55964.945YesYes044
117E2.M172 E2x52 10.41499.955YesNo045
118G.S1.05 G.S1.07 25.14696.23NoNo099
119G.H2.07 G.h2s4.01 21.53374.01YesYes1399
120G.H3.17 b.l25x6 16.03046.5YesNo458
121b.b2x3 b.b2x5 12.25326.395YesYes267
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x33Lig4.8351YesYes4010
3x36Lig12.1651NoYes6010
3x37Lig3.261YesYes6010
E2x52Lig44.4151NoYes5010
E2.V169Lig5.6250NoYes0010
5x40Lig6.7651YesYes5010
6x51Lig4.91YesYes6010
6x55Lig4.381NoYes5010
7x34Lig11.8150NoYes4010
7x38Lig16.2351YesYes5010
7x42Lig7.391YesYes7010
1x351x3912.3451YesYes4522
1x357x385.441YesYes4521
1x397x4214.771YesYes5721
2x567x423.460YesYes7721
3x333x373.2151YesYes4611
3x33E2.M1724.9451YesYes4012
3x335x406.361YesYes4511
3x363x373.4251NoYes6611
3x366x484.851NoYes6812
3x374x567.611YesNo6412
3x375x436.2751YesNo6512
3x375x4614.231YesYes6512
4x565x46110.421NoYes4522
E2.M172E2x529.9550YesNo0521
5x40E2x523.731YesNo5511
5x376x556.310NoNo3521
5x376x583.6450NoNo3421
5x406x554.211YesNo5511
6x517x385.711YesYes6511
6x517x414.5051YesNo6712
6x58E3.V2596.140NoYes4012
7x387x425.9651YesYes5711
7x417x423.4850NoYes7721
6x58Lig3.480NoYes4010
6x517x371.711YesNo6612

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusa3_on_gpOrthosteric Liganda3a_on_gp
100.00Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
91.67Consensusa3_onOrthosteric Liganda3a_on
83.33Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
83.33Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
78.57Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
78.57Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
76.92Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
76.92Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
71.43Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
71.43Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
71.43Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
70.59Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
69.23Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
69.23Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
68.75Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
66.67Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
61.54Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
61.54Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
61.54Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
61.54Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
61.54Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
60.00Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
60.00Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
60.00Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
60.00Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
58.82Single7EZCUKA7EZC-A2A-UKA
57.89Single3QAKUK-4320973QAK-A2A-UK-432097
57.14Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
56.25Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
56.25Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
56.25Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
56.25Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
56.25Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
56.25Consensusa2_onOrthosteric Liganda2b_on
56.25Consensusa2_on_gpOrthosteric Liganda2b_on_gp
56.25Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
56.25Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
56.25Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
56.25Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
55.56Single3NY9ICI118-5513NY9-β2-ICI118-551
55.56Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
55.00Single5WF5UK-4320975WF5-A2A-UK-432097
55.00Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
53.85Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
53.85Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
53.85Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
53.33Single4EJ4Naltrindole4EJ4-δ-Naltrindole
53.33Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
53.33Single6PS1Timolol6PS1-β2-Timolol
53.33Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
53.33Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
53.33Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
53.33Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
53.33Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.33Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.33Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.33Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
53.33Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
53.33Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
53.33Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
52.94Single4RWADIPP-NH24RWA-δ-DIPP-NH2
52.94Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
52.94Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
52.94Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
52.94Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
52.94Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
52.63Single4IARErgotamine4IAR-5-HT1B-Ergotamine
52.63Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
52.63Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
52.63Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
52.63Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
50.00Single3PWHZM-2413853PWH-A2A-ZM-241385
50.00Single3RFMCaffeine3RFM-A2A-Caffeine
50.00Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
50.00Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
50.00Single5N2SPSB365N2S-A1-PSB36
50.00Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
50.00Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
50.00Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
50.00Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
50.00Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
50.00Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
50.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
50.00Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
50.00Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
50.00Single7C61Ergotamine7C61-5-HT1B-Ergotamine
50.00Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
50.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
50.00Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
50.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
50.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
50.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
50.00Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
50.00Single8GNEKW-63568GNE-A2A-KW-6356-Na
50.00Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
50.00Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
50.00Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
50.00Single8S4DCMF-0198S4D-Apelin-CMF-019
50.00Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
50.00Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
50.00Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
50.00Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
50.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
50.00Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
47.37Single4UG2CGS216804UG2-A2A-CGS21680
47.37Single5WF6UK-4320975WF6-A2A-UK-432097
47.37Single6PT3DPI-2876PT3-δ-DPI-287
47.37Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
47.37Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
47.37Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
47.06Single2YDVNECA2YDV-A2A-NECA
47.06Single4UHRCGS216804UHR-A2A-CGS21680
47.06Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
47.06Single5G53NECA5G53-A2A-NECA-Gs
47.06Single6J21Aprepitant6J21-NK1-Aprepitant
47.06Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
47.06Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
47.06Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
47.06Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
47.06Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
47.06Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
47.06Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
47.06Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
47.06Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
47.06Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
47.06Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
47.06Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
47.06Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
47.06Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
47.06Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
47.06Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
47.06Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
47.06Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
47.06Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
47.06Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
47.06Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
46.67Single2YDOAdenosine2YDO-A2A-Adenosine
46.67Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
46.67Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
46.67Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
46.67Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
46.67Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
46.67Single5IU7Q274563465IU7-A2A-Q27456346-Na
46.67Single5IUBQ274563445IUB-A2A-Q27456344-Na
46.67Single5JTBZM-2413855JTB-A2A-ZM-241385
46.67Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
46.67Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
46.67Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
46.67Single6AQFZM-2413856AQF-A2A-ZM-241385
46.67Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
46.67Single6MH8ZM-2413856MH8-A2A-ZM-241385
46.67Single6PS0S-Carazolol6PS0-β2-S-Carazolol
46.67Single6PS4ICI118-5516PS4-β2-ICI118-551
46.67Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
46.67Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
46.67Single7AROLUF58337ARO-A2A-LUF5833-Na
46.67Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
46.67Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
46.67Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
46.67Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
46.67Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
46.67Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
46.67Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
46.67Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
46.67Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
46.67Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
46.67Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
46.67Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
46.67Consensusa2_offOrthosteric Liganda2a_off
46.67Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
46.67Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
46.15Single3UZAGTPL92363UZA-A2A-GTPL9236
46.15Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
45.45Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
45.45Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
45.00Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
45.00Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
45.00Single8WDTphotoNECA8WDT-A2A-photoNECA
45.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
44.44Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
44.44Single3D4STimolol3D4S-β2-Timolol
44.44Single6MXTSalmeterol6MXT-β2-Salmeterol
44.44Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
44.44Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
44.44Single7YITNalfurafine7YIT-κ-Nalfurafine
44.44Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
44.44Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
44.44Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
44.44Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
44.44Single8JJ8Formoterol8JJ8-β2-Formoterol
44.44Single8JWY2-1188JWY-A2A-2-118
44.44Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
44.44Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
44.44Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
44.44Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
44.44Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
44.44Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
44.44Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
43.75Single3EMLZM-2413853EML-A2A-ZM-241385
43.75Single3NY8ICI118-5513NY8-β2-ICI118-551
43.75Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
43.75Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
43.75Single4GBRS-Carazolol4GBR-β2-S-Carazolol
43.75Single5IU8Q274563475IU8-A2A-Q27456347-Na
43.75Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
43.75Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
43.75Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
43.75Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
43.75Single5UENDU1725UEN-A1-DU172
43.75Single5UIGCmpd-15UIG-A2A-Cmpd-1
43.75Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
43.75Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
43.75Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
43.75Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
43.75Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
43.75Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
43.75Single6S0LZM-2413856S0L-A2A-ZM-241385
43.75Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
43.75Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
43.75Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
43.75Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
43.75Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
43.75Single7PYRPSB-21157PYR-A2A-PSB-2115
43.75Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
43.75Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
43.75Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
43.75Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
43.75Single8CU6LJ-45178CU6-A2A-LJ-4517
43.75Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
43.75Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
43.75Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
43.75Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
43.75Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
43.75Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
43.75Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
43.75Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
43.75Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
43.75Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
43.75Single8JJOAlprenolol8JJO-β2-Alprenolol
43.75Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
43.75Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
43.75Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
43.75Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
43.75Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
43.75Single9CHXS-Carazolol9CHX-β2-S-Carazolol
43.75Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
43.75Consensus5ht5_onOrthosteric Ligand5ht5a_on
43.75Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
43.75Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
43.75Consensusalpha2_onOrthosteric Ligandalpha2b_on
43.75Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
43.75Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
43.75Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
43.75Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
43.75Consensusdopamine_offOrthosteric Ligandd2_off d3_off
43.75Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
43.75Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
43.48Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
43.48Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
43.48Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
42.86Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
42.86Single7SRQLSD7SRQ-5-HT2B-LSD
42.86Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
42.86Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
42.86Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
42.86Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
42.86Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
42.86Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
42.86Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
42.11Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
42.11Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
42.11Single7UM4AS26747237UM4-5-HT5A-AS2674723
42.11Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
42.11Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.11Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
42.11Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
42.11Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
42.11Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.11Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
42.11Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
42.11Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
42.11Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
42.11Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
42.11Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
41.67Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
41.67Single8PWNTheophylline8PWN-A2A-Theophylline
41.67Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
41.18Single2RH1S-Carazolol2RH1-β2-S-Carazolol
41.18Single2YCWS-Carazolol2YCW-β1-S-Carazolol
41.18Single4NTJAZD12834NTJ-P2Y12-AZD1283
41.18Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
41.18Single5C1MBU725C1M-μ-BU72
41.18Single5D6LS-Carazolol5D6L-β2-S-Carazolol
41.18Single5IUAQ274563485IUA-A2A-Q27456348-Na
41.18Single5JQHS-Carazolol5JQH-β2-S-Carazolol
41.18Single5N2RPSB-365N2R-A2A-PSB-36-Na
41.18Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
41.18Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
41.18Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
41.18Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
41.18Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
41.18Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
41.18Single6PS6Timolol6PS6-β2-Timolol
41.18Single6S0QZM-2413856S0Q-A2A-ZM-241385
41.18Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
41.18Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
41.18Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
41.18Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
41.18Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
41.18Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
41.18Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
41.18Single7WC6LSD7WC6-5-HT2A-LSD
41.18Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
41.18Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
41.18Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
41.18Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
41.18Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
41.18Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
41.18Single8QOTNanobody-E8QOT-μ-Nanobody-E
41.18Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
41.18Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
41.18Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
41.18Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
41.18Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
41.18Consensusadenosine_offOrthosteric Liganda1_off a2_off
41.18Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
41.18Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
41.18Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
41.18Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
41.18Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
41.18Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
41.18Consensusamine_offonOrthosteric Ligandamine_off amine_on
41.18Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
41.18Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
41.18Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
41.18Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
41.18Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
41.18Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
41.18Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
41.18Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
41.18Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
41.18Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
41.18Consensustrace-amine_onOrthosteric Ligandta1_on
40.91Single6PT2KGCHM076PT2-δ-KGCHM07
40.91Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
40.91Consensusangiotensin_onOrthosteric Ligandat1_on
40.91Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
40.91Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
40.91Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
40.91Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
40.91Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
40.91Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
40.00Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
40.00Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
40.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
40.00Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
40.00Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
40.00Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
40.00Single7XN9L-054,5227XN9-SST2-L-054,522
40.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
40.00Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
40.00Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
40.00Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
40.00Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
40.00Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.00Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
40.00Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
40.00Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
40.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
40.00Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
40.00Single8IWESpermidine8IWE-TA9-Spermidine
40.00Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
40.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
40.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
40.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
40.00Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
40.00Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.00Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
40.00Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
40.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
40.00Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
40.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
40.00Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
40.00Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
40.00Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
40.00Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
39.13Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
39.13Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
39.13Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
39.13Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
39.13Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
38.89Single3P0GBI1671073P0G-β2-BI167107
38.89Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
38.89Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
38.89Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
38.89Single5D5AS-Carazolol5D5A-β2-S-Carazolol
38.89Single5D5BS-Carazolol5D5B-β2-S-Carazolol
38.89Single5V54Methiothepin5V54-5-HT1B-Methiothepin
38.89Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
38.89Single6H7JIsoprenaline6H7J-β1-Isoprenaline
38.89Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
38.89Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
38.89Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
38.89Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
38.89Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
38.89Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
38.89Single7PX4PSB-21137PX4-A2A-PSB-2113
38.89Single7TUYGSK682753A7TUY-GPR183-GSK682753A
38.89Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
38.89Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
38.89Single8E0GBU728E0G-μ-BU72
38.89Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
38.89Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
38.89Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
38.89Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
38.89Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
38.89Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
38.89Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
38.89Consensus5ht1_offOrthosteric Ligand5ht1b_off
38.89Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
38.89Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
38.89Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
38.89Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
38.89Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
38.89Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
38.46Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
38.46Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.46Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
38.46Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
38.46Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
38.46Consensusbradykinin_onOrthosteric Ligandbk2_on
38.46Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
38.46Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
38.10Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
38.10Single7F8XNN90567F8X-CCKA-NN9056
38.10Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
38.10Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
38.10Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
38.10Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
38.10Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
38.10Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
38.10Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
38.10Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
38.10Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
38.10Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
38.10Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
38.10Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
38.10Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
38.10Consensuslpl_onOrthosteric Ligands1p_on lpa_on
38.10Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
38.10Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
38.10Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
37.50Single3REYXAC3REY-A2A-XAC
37.50Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
37.50Single5UVIZM-2413855UVI-A2A-ZM-241385
37.50Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
37.50Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
37.50Single6PS5S-Propranolol6PS5-β2-S-Propranolol
37.50Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
37.50Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
37.50Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
37.50Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
37.50Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
37.50Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
37.50Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
37.50Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.50Single7T32ZM-2413857T32-A2A-ZM-241385
37.50Single7UL3Famotidine7UL3-H2-Famotidine
37.50Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
37.50Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
37.50Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
37.50Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
37.50Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
37.50Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
37.50Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
37.50Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
37.50Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
37.50Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
37.50Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
37.50Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
37.50Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.50Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
37.50Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
37.50Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
37.50Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
37.50Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
37.50Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
37.50Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
37.50Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
37.50Single9BJKNaloxone9BJK-μ-Naloxone-NAM
37.50Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
37.50Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
37.50Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
37.50Consensusalpha1_onOrthosteric Ligandalpha1a_on
37.50Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
37.50Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
37.50Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
37.50Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
37.50Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
37.50Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
37.50Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.84Single4AMIBucindolol4AMI-β1-Bucindolol
36.84Single4LDEBI1671074LDE-β2-BI167107
36.84Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
36.84Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
36.84Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
36.84Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
36.84Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
36.84Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
36.84Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
36.84Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
36.84Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
36.84Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
36.84Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.84Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
36.84Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
36.84Single8JJLOlodaterol8JJL-β2-Olodaterol
36.84Single8JWZAB9288JWZ-A2A-AB928-Na
36.84Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.84Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
36.84Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
36.84Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
36.84Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
36.84Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
36.84Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
36.84Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
36.84Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
36.84Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
36.84Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
36.84Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
36.84Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
36.84Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
36.84Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
36.84Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
36.36Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
36.36Single6HLOAprepitant6HLO-NK1-Aprepitant
36.36Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
36.36Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
36.36Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
36.36Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
36.36Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
36.36Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
36.36Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
36.00Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
36.00Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
36.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
35.71Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
35.71Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
35.71Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
35.71Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.71Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.71Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
35.71Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
35.71Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
35.71Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
35.71Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
35.71Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
35.71Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
35.71Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
35.71Consensus5ht2_onOrthosteric Ligand5ht2b_on
35.71Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.71Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
35.71Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
35.71Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
35.71Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
35.29Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
35.29Single2Y04Salbutamol2Y04-β1-Salbutamol
35.29Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
35.29Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
35.29Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
35.29Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
35.29Single4QKX35V4QKX-β2-35V
35.29Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
35.29Single6H7MSalbutamol6H7M-β1-Salbutamol
35.29Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
35.29Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
35.29Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.29Single7BU7BI1671077BU7-β1-BI167107
35.29Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
35.29Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
35.29Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
35.29Single7UL4Alvimopan7UL4-μ-Alvimopan
35.29Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
35.29Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
35.29Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
35.29Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
35.29Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
35.29Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
35.29Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
35.29Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
35.29Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
35.29Single8JXRLSD8JXR-D1-LSD
35.29Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
35.29Single8RLNLUF58348RLN-A2A-LUF5834
35.29Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
35.29Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
35.29Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
35.29Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
35.29Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
35.29Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
35.29Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
35.29Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
35.29Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
35.29Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
35.29Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
35.29Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
35.29Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
35.29Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
35.29Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
35.29Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
35.29Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
35.29Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
35.29Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
35.29Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
35.00Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
35.00Single6H7LDobutamine6H7L-β1-Dobutamine
35.00Single6IBLArformoterol6IBL-β1-Arformoterol
35.00Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
35.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
35.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
35.00Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
35.00Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
35.00Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
35.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
35.00Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
35.00Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
35.00Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
35.00Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
35.00Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
35.00Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
35.00Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
35.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
35.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
35.00Consensuscck_onOrthosteric Ligandccka_on cckb_on
35.00Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
35.00Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
35.00Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
35.00Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
35.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
35.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
35.00Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
34.78Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
34.78Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
34.78Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
34.78Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
34.62Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
34.62Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
34.62Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
34.62Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
34.62Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
34.62Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
34.62Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
34.48Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
33.33Single2Y03Isoprenaline2Y03-β1-Isoprenaline
33.33Single3PBLEticlopride3PBL-D3-Eticlopride
33.33Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
33.33Single5MZPCaffeine5MZP-A2A-Caffeine-Na
33.33Single5TVNLSD5TVN-5-HT2B-LSD
33.33Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
33.33Single6E67BI1671076E67-β2-BI167107-Gs (fused)
33.33Single6HLLCP999946HLL-NK1-CP99994
33.33Single6JODAngiotensin II6JOD-AT2-Angiotensin II
33.33Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
33.33Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
33.33Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
33.33Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
33.33Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
33.33Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
33.33Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
33.33Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
33.33Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
33.33Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
33.33Single7SINNPS-21437SIN-CaS-NPS-2143
33.33Single7SINNPS-21437SIN-CaS-NPS-2143
33.33Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
33.33Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
33.33Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
33.33Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
33.33Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
33.33Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
33.33Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
33.33Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
33.33Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
33.33Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
33.33Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
33.33Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
33.33Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
33.33Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
33.33Single8K5BNiacin8K5B-HCA2-Niacin
33.33Single8TF5Oleic acid8TF5-GPR6-Oleic acid
33.33Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
33.33Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
33.33Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
33.33Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
33.33Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
33.33Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
33.33Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
33.33Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
33.33Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
33.33Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
33.33Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
33.33Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
33.33Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
33.33Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
33.33Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
33.33Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
33.33Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
33.33Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
33.33Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
33.33Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
33.33Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
33.33Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
33.33Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
33.33Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
33.33Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
33.33Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
33.33Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
33.33Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
33.33Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
33.33Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
33.33Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
33.33Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
33.33Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
33.33Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
33.33Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
33.33Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
32.14Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
32.00Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
32.00Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
32.00Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
32.00Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
32.00Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
32.00Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
31.82Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
31.82Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
31.82Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
31.82Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
31.82Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
31.82Single8WKYPG-9348WKY-MC4-PG-934
31.82Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
31.82Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
31.82Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.58Single4U15Tiotropium4U15-M3-Tiotropium
31.58Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
31.58Single5TZRMK86665TZR-FFA1-MK8666
31.58Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
31.58Single6J20Aprepitant6J20-NK1-Aprepitant
31.58Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
31.58Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
31.58Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
31.58Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
31.58Single6OL9Tiotropium6OL9-M5-Tiotropium
31.58Single6TQ7SB-3348676TQ7-OX1-SB-334867
31.58Single6WGTLSD6WGT-5-HT2A-LSD
31.58Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
31.58Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
31.58Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
31.58Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
31.58Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
31.58Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
31.58Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
31.58Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
31.58Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
31.58Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
31.58Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
31.58Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
31.58Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
31.58Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
31.58Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.58Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
31.58Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
31.58Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
31.58Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
31.58Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
31.58Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
31.58Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
31.58Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
31.58Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
31.58Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
31.58Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.58Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
31.58Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
31.58Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
31.58Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
31.58Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
31.58Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
31.58Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
31.58Consensuslpa_onOrthosteric Ligandlpa1_on
31.58Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
31.58Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
31.58Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
31.58Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
31.58Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
31.58Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
31.58Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
31.58Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
31.58Consensustachykinin_offOrthosteric Ligandnk1_off
31.25Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
31.25Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
31.25Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
31.25Single6AKXA4R6AKX-CCR5-A4R
31.25Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
31.25Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
31.25Single6ME2Ramelteon6ME2-MT1-Ramelteon
31.25Single6ME9Ramelteon6ME9-MT2-Ramelteon
31.25Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
31.25Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
31.25Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
31.25Single6TODEMPA6TOD-OX1-EMPA-Na
31.25Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
31.25Single7F8ULintitript7F8U-CCKA-Lintitript
31.25Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
31.25Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
31.25Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
31.25Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
31.25Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
31.25Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
31.25Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
31.25Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
31.25Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
31.25Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
31.25Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
31.25Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
31.25Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
31.25Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
31.25Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
31.25Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
31.25Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
31.25Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.25Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.25Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
31.25Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
31.25Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
31.25Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
31.25Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
31.25Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
31.25Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
31.25Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
31.25Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
31.25Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
31.25Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
31.25Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
31.25Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
30.77Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
30.77Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
30.77Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
30.77Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
30.43Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
30.43Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
30.43Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
30.43Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
30.43Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
30.43Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
30.43Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
30.43Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
30.43Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
30.43Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
30.43Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
30.43Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
30.43Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
30.43Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
30.43Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
30.00Single4N4WSANT-14N4W-SMO-SANT-1
30.00Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
30.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
30.00Single5CXVTiotropium5CXV-M1-Tiotropium
30.00Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
30.00Single6A93Risperidone6A93-5-HT2A-Risperidone
30.00Single6CM4Risperidone6CM4-D2-Risperidone
30.00Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
30.00Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
30.00Single6ZG4HTL00099366ZG4-M1-HTL0009936
30.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
30.00Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
30.00Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
30.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
30.00Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
30.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
30.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
30.00Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
30.00Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
30.00Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
30.00Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
30.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
30.00Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
30.00Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
30.00Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
30.00Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
30.00Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
30.00Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.00Single8XYIVUF106618XYI-CXCR3-VUF10661
30.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
30.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
30.00Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
30.00Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
30.00Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
30.00Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
30.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
30.00Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
30.00Consensuslpa_offOrthosteric Ligandlpa1_off
30.00Consensuslpl_offOrthosteric Ligands1p_off lpa_off
30.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
30.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
30.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
30.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
30.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
30.00Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
29.63Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
29.63Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
29.63Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
29.63Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
29.41Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
29.41Single3RZECidoxepin3RZE-H1-Cidoxepin
29.41Single4MBSMaraviroc4MBS-CCR5-Maraviroc
29.41Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
29.41Single4ZJCSB-6740424ZJC-OX1-SB-674042
29.41Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
29.41Single6KUXRS-799486KUX-α2a-RS-79948
29.41Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
29.41Single6TPGEMPA6TPG-OX2-EMPA
29.41Single6V9SGTPL114036V9S-OX1-GTPL11403
29.41Single6VI4JDTic6VI4-κ-JDTic
29.41Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
29.41Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
29.41Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
29.41Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
29.41Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
29.41Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
29.41Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
29.41Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
29.41Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.41Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
29.41Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
29.41Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
29.41Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
29.41Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.41Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
29.41Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
29.41Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
29.41Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
29.41Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
29.41Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
29.41Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
29.41Single8K5CAcipimox8K5C-HCA2-Acipimox
29.41Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
29.41Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.41Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
29.41Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
29.41Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
29.41Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
29.41Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
29.41Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
29.41Consensushca_onOrthosteric Ligandhca2_on
29.41Consensusopsins_offOrthosteric Ligandrhodopsin_off
29.41Consensussensory_offOrthosteric Ligandopsins_off
29.17Single3OE0CVX153OE0-CXCR4-CVX15
29.17Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
29.17Single6W25SHU91196W25-MC4-SHU9119-Ca
29.17Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
29.17Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
29.17Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
29.17Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
29.17Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
29.17Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
29.17Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
28.57Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
28.57Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
28.57Single5X93K-87945X93-ETB-K-8794
28.57Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
28.57Single6IGLIRL16206IGL-ETB-IRL1620
28.57Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
28.57Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
28.57Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
28.57Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
28.57Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
28.57Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
28.57Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
28.57Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
28.57Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
28.57Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
28.57Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
28.57Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
28.57Single9CHUNoradrenaline9CHU-β2-Noradrenaline
28.57Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
28.57Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
28.57Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
28.57Consensuschemerin_onOrthosteric Ligandcml1_on
28.57Consensusendothelin_offOrthosteric Ligandetb_off
28.57Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
28.57Consensusprostanoid_offOrthosteric Ligandep_off dp_off
28.00Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
28.00Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.00Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
28.00Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
28.00Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
28.00Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
28.00Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
28.00Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
28.00Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.00Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.00Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.00Consensusvasop-oxy_onOrthosteric Ligandv2_on
28.00Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
27.78Single2Y01Dobutamine2Y01-β1-Dobutamine
27.78Single2Y02Carmoterol2Y02-β1-Carmoterol
27.78Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
27.78Single4MQSIperoxo4MQS-M2-Iperoxo
27.78Single4QIMANTA XV4QIM-SMO-ANTA XV
27.78Single4U14Tiotropium4U14-M3-Tiotropium
27.78Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
27.78Single5DHHSB-6121115DHH-NOP-SB-612111
27.78Single5DSGTiotropium5DSG-M4-Tiotropium
27.78Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
27.78Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
27.78Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
27.78Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
27.78Single6DRXLisuride6DRX-5-HT2B-Lisuride
27.78Single6TOTLemborexant6TOT-OX1-Lemborexant
27.78Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
27.78Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
27.78Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
27.78Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
27.78Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
27.78Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
27.78Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
27.78Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
27.78Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
27.78Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
27.78Single7WC7Lisuride7WC7-5-HT2A-Lisuride
27.78Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
27.78Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
27.78Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
27.78Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
27.78Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
27.78Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
27.78Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
27.78Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
27.78Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
27.78Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
27.78Single8T1WCVN4248T1W-GPR6-CVN424
27.78Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
27.78Single8X63Mepyramine8X63-H1-Mepyramine
27.78Single8X64Desloratadine8X64-H1-Desloratadine
27.78Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
27.78Single9IYAONO-97105319IYA-GPR55-ONO-9710531
27.78Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
27.78Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
27.78Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
27.78Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
27.78Consensusblt_onOrthosteric Ligandblt1_on
27.78Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
27.78Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
27.78Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
27.78Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
27.78Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
27.78Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
27.78Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
27.78Consensushca_on_gpOrthosteric Ligandhca2_on_gp
27.78Consensushistamine_offOrthosteric Ligandh1_off
27.78Consensusleukotriene_onOrthosteric Ligandblt_on
27.78Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
27.78Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
27.59Single5GLHEndothelin-15GLH-ETB-Endothelin-1
27.59Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
27.59Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
27.59Consensusbombesin_onOrthosteric Ligandbb2_on
27.59Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
27.59Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
27.59Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
27.59Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
27.59Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
27.27Single5ZTYAM102575ZTY-CB2-AM10257
27.27Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
27.27Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
27.27Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
27.27Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single7SK9CCX6627SK9-ACKR3-CCX662
27.27Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
27.27Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
27.27Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
27.27Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
27.27Single8X5YAstemizole8X5Y-H1-Astemizole
27.27Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
27.27Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
27.27Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
27.27Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
26.92Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
26.92Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
26.92Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
26.92Single8ZRTET-18ZRT-ETB-ET-1
26.92Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
26.92Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
26.67Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
26.67Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
26.67Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
26.67Single6ME5Agomelatine6ME5-MT1-Agomelatine
26.67Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
26.67Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
26.67Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
26.67Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
26.67Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
26.67Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
26.67Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
26.67Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
26.67Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
26.67Consensusgi_sensoryOrthosteric Ligandgi_opsins
26.67Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
26.67Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
26.67Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
26.67Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
26.67Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
26.67Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
26.67Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
26.32Single2Y00Dobutamine2Y00-β1-Dobutamine
26.32Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
26.32Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
26.32Single5WIUNemonapride5WIU-D4-Nemonapride
26.32Single5WIVNemonapride5WIV-D4-Nemonapride-Na
26.32Single5WQCEMPA5WQC-OX2-EMPA
26.32Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
26.32Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
26.32Single6D26Fevipiprant6D26-DP2-Fevipiprant
26.32Single6HLPNetupitant6HLP-NK1-Netupitant
26.32Single6LUQHaloperidol6LUQ-D2-Haloperidol
26.32Single6TP6Filorexant6TP6-OX1-Filorexant
26.32Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
26.32Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
26.32Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
26.32Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
26.32Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
26.32Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
26.32Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
26.32Single7W41PD1762527W41-BB2-PD176252
26.32Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
26.32Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.32Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
26.32Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.32Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
26.32Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
26.32Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
26.32Single8JXSPF-61428JXS-D1-PF-6142
26.32Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
26.32Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
26.32Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
26.32Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
26.32Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
26.32Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
26.32Single8ZMFA1L108ZMF-5-HT2C-A1L10
26.32Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
26.32Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
26.32Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
26.32Consensusbombesin_offOrthosteric Ligandbb2_off
26.32Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
26.32Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
26.32Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
26.32Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
26.32Consensusdp_offOrthosteric Liganddp2_off
26.32Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
26.32Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
26.32Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
26.32Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
26.32Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
26.32Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
26.09Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
26.09Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
26.09Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
26.09Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
26.09Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
26.09Single8IEBA1LYA8IEB-GPR156-A1LYA
26.09Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
26.09Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.09Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
26.09Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
26.09Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
26.09Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
26.09Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
25.93Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
25.93Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.93Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.93Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
25.93Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
25.81Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
25.00Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
25.00Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
25.00Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
25.00Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
25.00Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
25.00Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
25.00Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
25.00Single4DJHJDTic4DJH-κ-JDTic
25.00Single5L7IVismodegib5L7I-SMO-Vismodegib
25.00Single5XR8AM8415XR8-CB1-AM841
25.00Single5XRAAM115425XRA-CB1-AM11542
25.00Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
25.00Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
25.00Single6E59L-7607356E59-NK1-L-760735
25.00Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
25.00Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
25.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
25.00Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
25.00Single7B6WCyclazosin7B6W-α1b-Cyclazosin
25.00Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
25.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
25.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
25.00Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
25.00Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
25.00Single7FEECP559407FEE-CB1-CP55940-ZCZ011
25.00Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
25.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
25.00Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
25.00Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
25.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
25.00Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
25.00Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
25.00Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
25.00Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
25.00Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
25.00Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
25.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8EA0Iperoxo8EA0-M3-Iperoxo
25.00Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
25.00Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
25.00Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
25.00Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
25.00Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
25.00Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
25.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
25.00Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
25.00Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
25.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
25.00Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
25.00Single8XVLZibotentan8XVL-ETA-Zibotentan
25.00Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
25.00Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
25.00Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
25.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
25.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
25.00Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
25.00Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
25.00Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
25.00Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
25.00Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
25.00Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
25.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.00Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
25.00Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
25.00Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
25.00Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
25.00Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
25.00Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
25.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
25.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
24.14Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
24.14Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Consensusendothelin_onOrthosteric Ligandetb_on eta_on
24.14Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
24.00Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
24.00Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
24.00Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
24.00Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
24.00Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
24.00Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
24.00Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
24.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
24.00Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
23.81Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
23.81Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
23.81Single4PY02MeSATP4PY0-P2Y12-2MeSATP
23.81Single4XEENeurotensin4XEE-NTS1-Neurotensin
23.81Single4XESNeurotensin4XES-NTS1-Neurotensin
23.81Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
23.81Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
23.81Single6KQICP559406KQI-CB1-CP55940-Org27569
23.81Single6OS2TRV0266OS2-AT1-TRV026
23.81Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
23.81Single7DFPSpiperone7DFP-D2-Spiperone
23.81Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
23.81Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
23.81Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
23.81Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
23.81Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
23.81Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
23.81Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
23.81Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
23.81Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
23.81Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
23.81Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
23.81Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
23.81Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
23.81Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
23.81Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
23.81Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Consensusorexin_onOrthosteric Ligandox2_on
23.81Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
23.53Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
23.53Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
23.53Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
23.53Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
23.53Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
23.53Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
23.53Single4S0VSuvorexant4S0V-OX2-Suvorexant
23.53Single5WS3EMPA5WS3-OX2-EMPA
23.53Single6AKYMaraviroc6AKY-CCR5-Maraviroc
23.53Single6B73MP11046B73-κ-MP1104
23.53Single6DS0Ly2660976DS0-5-HT2B-Ly266097
23.53Single6TPJSuvorexant6TPJ-OX2-Suvorexant
23.53Single7BR3Elagolix7BR3-GnRH1-Elagolix
23.53Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
23.53Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
23.53Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
23.53Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
23.53Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
23.53Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
23.53Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.53Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
23.53Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
23.53Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
23.53Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
23.53Single8Y0HVUF114188Y0H-CXCR3-VUF11418
23.53Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
23.53Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
23.53Consensusangiotensin_offOrthosteric Ligandat1_off
23.53Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
23.53Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
23.53Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
23.53Consensusorexin_offOrthosteric Ligandox2_off ox1_off
23.53Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
23.53Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
23.53Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
23.53Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
23.53Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
23.33Single6IGKEndothelin-36IGK-ETB-Endothelin-3
23.33Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
23.33Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
23.08Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
23.08Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
23.08Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
23.08Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
23.08Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
23.08Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
23.08Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
23.08Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
23.08Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
23.08Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
23.08Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
23.08Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
23.08Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
23.08Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
23.08Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
22.73Single4BUONeurotensin4BUO-NTS1-Neurotensin
22.73Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
22.73Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
22.73Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
22.73Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
22.73Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
22.73Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
22.73Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
22.73Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
22.73Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
22.73Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
22.73Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single8XVJMacitentan8XVJ-ETA-Macitentan
22.73Single8XVUCXCL28XVU-CXCR2-CXCL2
22.73Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
22.73Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
22.73Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
22.58Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
22.58Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
22.22Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
22.22Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
22.22Single6A94Zotepine6A94-5-HT2A-Zotepine
22.22Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
22.22Single6IQLL7458706IQL-D4-L745870
22.22Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
22.22Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
22.22Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
22.22Single6TP3Nemorexant6TP3-OX1-Nemorexant
22.22Single6TPKRetosiban6TPK-OT-Retosiban
22.22Single6TPNHTL66416TPN-OX2-HTL6641
22.22Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
22.22Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
22.22Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
22.22Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
22.22Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
22.22Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
22.22Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
22.22Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
22.22Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
22.22Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
22.22Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
22.22Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
22.22Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
22.22Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
22.22Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
22.22Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
22.22Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
22.22Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
22.22Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
22.22Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
22.22Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
22.22Single8IHKAcifran8IHK-HCA3-Acifran
22.22Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
22.22Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.22Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
22.22Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
22.22Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
22.22Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
22.22Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
22.22Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
22.22Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
22.22Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Consensusgrh_offOrthosteric Ligandgnrh1_off
22.22Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
22.22Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
22.22Consensusvasop-oxy_offOrthosteric Ligandot_off
21.74Single5EE7MK08935EE7-Glucagon-MK0893
21.74Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
21.74Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
21.74Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
21.74Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
21.74Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
21.74Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
21.74Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
21.74Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single8XQJJN2418XQJ-Apelin-JN241
21.74Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
21.74Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
21.74Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
21.74Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
21.74Consensuskisspeptin_onOrthosteric Ligandkiss1_on
21.43Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
21.43Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
21.43Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
21.43Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
21.43Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
21.43Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
21.43Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
21.43Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
21.43Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
21.43Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
21.43Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
21.43Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
21.05Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
21.05Single4DAJTiotropium4DAJ-M3-Tiotropium
21.05Single4YAYZD-71554YAY-AT1-ZD-7155
21.05Single5DHGC-355DHG-NOP-C-35
21.05Single5TGZAM65385TGZ-CB1-AM6538
21.05Single6D27CAY104716D27-DP2-CAY10471
21.05Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
21.05Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
21.05Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
21.05Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
21.05Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
21.05Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
21.05Single7V3ZCP559407V3Z-CB1-CP55940
21.05Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
21.05Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
21.05Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.05Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
21.05Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
21.05Single8K5DGSK2560738K5D-HCA2-GSK256073
21.05Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
21.05Consensuscck_offOrthosteric Ligandccka_off
21.05Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
21.05Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
20.83Single4XT1Fractalkine4XT1-US28-Fractalkine
20.83Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
20.83Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
20.83Single7QA8Peptide7QA8-STE2-Peptide
20.83Single7QA8Peptide7QA8-STE2-Peptide
20.83Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
20.83Single8XWNCXCL88XWN-CXCR2-CXCL8
20.83Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.83Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.83Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.83Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
20.69Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
20.69Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
20.69Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
20.69Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
20.69Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
20.69Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
20.69Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
20.00Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
20.00Single5CGCHTL142425CGC-mGlu5-HTL14242
20.00Single5XPRBosentan5XPR-ETB-Bosentan
20.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
20.00Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
20.00Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
20.00Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.00Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
20.00Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
20.00Single6Z4SSR486926Z4S-NTS1-SR48692
20.00Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
20.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
20.00Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
20.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
20.00Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
20.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
20.00Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
20.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
20.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.00Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
20.00Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
20.00Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
20.00Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
20.00Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
20.00Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
20.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
20.00Single8IEBA1LYA8IEB-GPR156-A1LYA
20.00Single8IY6Endothelin-18IY6-ETB-Endothelin-1
20.00Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.00Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
20.00Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
20.00Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
20.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
20.00Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
20.00Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
20.00Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
20.00Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
20.00Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
20.00Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.00Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.00Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
20.00Consensusp2y_offOrthosteric Ligandp2y1_off
20.00Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
20.00Consensussensory_onOrthosteric Ligandopsins_on
20.00Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
19.35Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
19.23Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
19.23Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
19.23Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
19.23Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.23Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.23Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
19.23Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
19.05Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
19.05Single4BV0Neurotensin4BV0-NTS1-Neurotensin
19.05Single5V56TC1145V56-SMO-TC114
19.05Single6OS1TRV0266OS1-AT1-TRV026
19.05Single7F1TMIP-1a7F1T-CCR5-MIP-1a
19.05Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
19.05Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
19.05Single7P2L4YI7P2L-mGlu5-4YI
19.05Single7R0CAVP7R0C-V2-AVP-Arrestin2
19.05Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
19.05Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.05Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
19.05Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
19.05Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
19.05Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
19.05Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
19.05Consensusneurotensin_onOrthosteric Ligandnts1_on
19.05Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
18.75Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
18.75Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
18.75Single4XNWMRS25004XNW-P2Y1-MRS2500
18.75Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
18.75Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
18.75Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
18.75Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
18.75Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
18.75Single7WC5Psilocin7WC5-5-HT2A-Psilocin
18.75Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
18.75Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
18.75Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
18.75Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
18.75Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
18.75Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
18.75Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
18.52Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
18.52Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
18.52Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
18.52Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
18.18Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
18.18Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
18.18Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
18.18Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
18.18Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
18.18Single6YVRNTS8-136YVR-NTS1-NTS8-13
18.18Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
18.18Single7K15MKD0467K15-BLT1-MKD046-Na
18.18Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
18.18Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
18.18Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
18.18Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
18.18Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
18.18Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
18.18Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
18.18Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8XQJJN2418XQJ-Apelin-JN241
18.18Single8XWACXCL18XWA-CXCR2-CXCL1
18.18Single8XWMCXCL68XWM-CXCR2-CXCL6
18.18Single8XWSCXCL58XWS-CXCR2-CXCL5
18.18Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
18.18Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
18.18Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
18.18Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
18.18Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
18.18Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.86Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
17.86Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
17.86Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
17.86Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
17.86Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
17.65Single3OE9IT1t3OE9-CXCR4-IT1t
17.65Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
17.65Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
17.65Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
17.65Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.65Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
17.65Single7UL2SR486927UL2-NTS1-SR48692-Na
17.65Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
17.65Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
17.65Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
17.65Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
17.65Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
17.65Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
17.65Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
17.65Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
17.65Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
17.65Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
17.65Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
17.65Single9B9Y7DY9B9Y-CB1-7DY
17.65Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
17.65Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
17.65Consensusneurotensin_offOrthosteric Ligandnts1_off
17.65Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
17.39Single5CGDHTL142425CGD-mGlu5-HTL14242
17.39Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
17.39Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
17.39Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
17.39Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
17.39Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
17.39Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8XWFCXCL38XWF-CXCR2-CXCL3
17.39Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
17.39Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
17.39Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
17.39Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
17.39Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single4XT3Fractalkine4XT3-US28-Fractalkine
17.24Single6FJ3PTH6FJ3-PTH1-PTH
17.24Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
17.24Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
17.24Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
17.24Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
17.24Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
17.24Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
17.14Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.07Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
16.67Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
16.67Single5ZKQABT-4915ZKQ-PAF-ABT-491
16.67Single6KNMJN241-96KNM-Apelin-JN241-9
16.67Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
16.67Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
16.67Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
16.67Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
16.67Single7F8YDevazepide7F8Y-CCKA-Devazepide
16.67Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
16.67Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
16.67Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
16.67Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
16.67Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
16.67Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
16.67Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
16.67Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
16.67Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
16.67Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
16.67Single7XRRLemborexant7XRR-OX2-Lemborexant
16.67Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
16.67Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
16.67Single8IEIA1LYA8IEI-GPR156-A1LYA
16.67Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
16.67Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
16.67Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
16.67Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.67Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
16.67Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
16.22Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
16.13Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
16.13Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
16.13Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
16.13Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
16.13Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
16.13Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
16.13Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
16.00Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
16.00Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single8IEPA1LYA8IEP-GPR156-A1LYA
16.00Single8IEPA1LYA8IEP-GPR156-A1LYA
16.00Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
16.00Single8KIGSHU91198KIG-MC3-SHU9119-Ca
15.79Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
15.79Single6FFIMMPEP6FFI-mGlu5-MMPEP
15.79Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
15.79Single6ZG9GSK10347026ZG9-M1-GSK1034702
15.79Single6ZINSR486926ZIN-NTS1-SR48692
15.79Single7VV6C48/807VV6-MRGPRX2-C48/80
15.79Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.79Single8K2WAMG4878K2W-CXCR3-AMG487
15.79Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
15.79Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
15.79Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
15.79Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
15.79Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
15.79Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
15.79Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
15.79Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
15.79Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
15.79Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
15.79Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.62Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
15.62Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
15.62Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
15.62Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
15.38Single7SK5CXCL127SK5-ACKR3-CXCL12
15.38Single7XNACYN1548067XNA-SST2-CYN154806
15.38Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.38Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
15.38Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
15.15Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
15.15Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
15.00Single6FFHFenobam6FFH-mGlu5-Fenobam
15.00Single6GPSMK08126GPS-CCR2-MK0812
15.00Single6IIVDaltroban6IIV-TP-Daltroban
15.00Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
15.00Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
15.00Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
15.00Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
15.00Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
15.00Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
15.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
15.00Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
15.00Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
15.00Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
15.00Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
15.00Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.81Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
14.81Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
14.81Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
14.81Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
14.81Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
14.71Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
14.29Single4JKVTaladegib4JKV-SMO-Taladegib
14.29Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
14.29Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
14.29Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
14.29Single6GPXMK08126GPX-CCR2-MK0812
14.29Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
14.29Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
14.29Single7C4SS1P7C4S-S1P3-S1P
14.29Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
14.29Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
14.29Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
14.29Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
14.29Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
14.29Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
14.29Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
14.29Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
14.29Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
14.29Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
14.29Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
14.29Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
14.29Consensusblt_offOrthosteric Ligandblt1_off
14.29Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
14.29Consensusep_offOrthosteric Ligandep4_off
14.29Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
14.29Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
13.79Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
13.79Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
13.64Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
13.64Single5V57TC1145V57-SMO-TC114
13.64Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
13.64Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
13.64Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
13.64Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
13.64Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
13.64Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
13.33Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
13.33Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
13.33Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
13.33Single7SK3CXCL127SK3-ACKR3-CXCL12
13.33Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
13.33Single7WC4Serotonin7WC4-5-HT2A-Serotonin
13.33Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.33Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
13.33Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
13.33Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
13.04Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
13.04Single6IIURamatroban6IIU-TP-Ramatroban
13.04Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
13.04Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
13.04Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
12.90Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
12.90Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
12.90Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
12.90Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
12.90Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
12.82Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
12.50Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
12.50Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
12.50Single6K1QIRL25006K1Q-ETB-IRL2500
12.50Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
12.50Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
12.50Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
12.50Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
12.50Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
12.50Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
12.50Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
12.50Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
11.76Single3OE6IT1t3OE6-CXCR4-IT1t
11.76Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
11.76Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
11.76Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
11.76Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
11.76Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
11.76Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
11.76Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
11.54Single8IEIA1LYA8IEI-GPR156-A1LYA
11.54Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
11.54Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
11.54Consensussomatostatin_offOrthosteric Ligandsst2_off
11.11Single4O9RCyclopamine4O9R-SMO-Cyclopamine
11.11Single6LI0C176LI0-GPR52-C17
11.11Single6TP4ACT-4622066TP4-OX1-ACT-462206
11.11Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
11.11Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
11.11Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
11.11Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
11.11Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.11Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
11.11Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
11.11Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Consensusgq_nucleotideOrthosteric Ligandgq_p2y
11.11Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.53Single3ODUIT1t3ODU-CXCR4-IT1t
10.53Single4BWBNeurotensin4BWB-NTS1-Neurotensin
10.53Single4QINSAG1.54QIN-SMO-SAG1.5
10.53Single5U09Taranabant5U09-CB1-Taranabant
10.53Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
10.53Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
10.53Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
10.53Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
10.53Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
10.53Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
10.53Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.53Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
10.53Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
10.53Single9BA0A1AKN9BA0-CB1-A1AKN
10.53Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
10.53Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.53Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.53Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.34Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
10.34Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
10.00Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
10.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
10.00Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
10.00Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
10.00Single7VODCariprazine7VOD-5-HT2A-Cariprazine
10.00Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
10.00Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8IYXYL-3658IYX-GPR34-YL-365
10.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
9.52Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
9.52Single5T04Neurotensin5T04-NTS1-Neurotensin
9.52Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
9.52Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
9.52Single7YXAONO-54306087YXA-S1P5-ONO-5430608
9.52Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
9.52Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
9.52Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
9.52Single9B9ZA1AKO9B9Z-CB1-A1AKO
9.52Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
9.52Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
9.52Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
9.38Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
9.38Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
9.09Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
9.09Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
9.09Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
8.70Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
8.70Single9BJKNAM9BJK-μ-Naloxone-NAM
8.57Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
8.33Single5X33BIIL2605X33-BLT1-BIIL260
8.33Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
8.00Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
8.00Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
8.00Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
8.00Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
7.69Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
7.69Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
7.69Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
7.41Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
7.41Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
7.41Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.41Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
7.41Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.41Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.14Single7SHEPI; PE7SHE-GPR158-PI; PE
7.14Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
7.14Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
6.67Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
5.88Single3OE8IT1t3OE8-CXCR4-IT1t
5.88Single6TQ9SB-4081246TQ9-OX1-SB-408124
5.88Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
5.88Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
5.88Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
5.56Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
5.56Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
5.56Single8JPSCCL78JPS-ACKR1-CCL7
5.56Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
5.56Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.26Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
5.26Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
5.26Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
5.26Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
5.26Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
5.26Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
5.26Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
5.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
5.00Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.00Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
5.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
5.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
4.55Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
4.55Single7F83PF-051904577F83-Ghrelin-PF-05190457
4.55Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
4.35Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
4.17Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
4.00Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
4.00Single7SHEPI; PE7SHE-GPR158-PI; PE
3.57Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
3.45Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
3.45Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7

Consensus Members
Id Members
8X17 8X17-A3A-Namodenoson-Gi1/β1/γ2
8X16 8X16-A3A-Piclidenoson-Gi1/β1/γ2
Net Summary
Imin 3.12
Number of Linked Nodes 870
Number of Links 1017
Number of Hubs 155
Number of Links mediated by Hubs 585
Number of Communities 32
Number of Nodes involved in Communities 218
Number of Links involved in Communities 295
Path Summary
Number Of Nodes in MetaPath 122
Number Of Links MetaPath 121
Number of Shortest Paths 1110496
Length Of Smallest Path 3
Average Path Length 34.9613
Length of Longest Path 77
Minimum Path Strength 0.6875
Average Path Strength 6.22736
Maximum Path Strength 30.325
Minimum Path Correlation 0.7
Average Path Correlation 0.980732
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.12766
Average % Of Corr. Nodes 41.8726
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 43.2944
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
a3_on_gpa3a_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

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