Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 2.1575402
2G.HN.45 2.47958404
3G.S1.06 4.412924218
4G.H1.01 4.84655219
5G.H1.03 2.04271409
6G.S2.03 4.77667429
7G.S2.08 8.208964185
8G.s2s3.01 5.440634184
9G.S3.03 7.771335207
10G.S3.04 8.23646426
11G.S3.06 7.69933525
12G.S3.07 3.797924219
13G.s3h2.03 5.02167429
14G.H2.02 4.43583428
15G.H2.04 3.17267509
16G.H2.06 5.70083729
17G.H2.07 5.20917629
18G.H2.09 5.76271428
19G.H2.10 4.36292427
20G.h2s4.01 6.04933529
21G.S4.04 5.30521479
22G.s4h3.04 6.67229485
23G.s4h3.05 4.03604403
24G.s4h3.08 1.53375408
25G.H3.01 5.82729409
26G.H3.09 4.73976779
27G.H3.13 3.91479475
28G.H3.14 5.51583478
29G.H3.17 6.46833625
30G.H3.18 5.996044229
31G.S5.03 3.01271408
32G.S5.04 3.94125479
33G.S5.05 4.265836179
34G.HG.04 5.71633509
35G.HG.15 5.6575487
36G.hgh4.02 6.30403687
37G.hgh4.05 8.84104487
38G.H4.03 4.76625404
39G.H4.10 6.308586
40G.H4.12 5.86475
41G.h4s6.02 4.65542478
42G.S6.02 6.68271407
43G.H5.03 4.56667508
44G.H5.08 5.750335188
45G.H5.17 6.280834195
46G.H5.25 5.60792407
47G.H5.26 4.70083505
48b.1x1 2.11896404
49b.1x4 3.34604408
50b.1x11 3.23033508
51b.h2x1 3.92208405
52b.lhb1x3 2.91667502
53b.lhb1x6 4.568754163
54b.lhb1x9 3.50437403
55b.lhb1x11 4.13937494
56b.b1x3 5.94437
57b.l1x3 9.45217539
58b.b2x1 8.3125528
59b.b2x5 5.55988737
60b.b3x3 3.37458468
61b.l3x2 4.98067539
62b.b4x2 4.86562408
63b.b4x3 4.87854467
64b.b4x4 9.26792438
65b.b4x5 4.19313467
66b.b4x6 10.0732639
67b.b5x2 5.69896407
68b.b5x3 6.68306639
69b.b5x5 5.67063465
70b.b5x7 5.31063467
71b.l5x1 4.33683568
72b.l5x5 7.58476729
73b.b6x1 3.51562409
74b.b6x5 4.14889666
75b.l6x5 6.894114
76b.b7x1 5.648335114
77b.b7x2 3.73896468
78b.b7x4 4.28625468
79b.l7x4 4.50125409
80b.b8x3 3.88979406
81b.b8x4 4.54083766
82b.l8x3 3.820424113
83b.l8x8 5.38125464
84b.b9x4 6.46896409
85b.l9x3 6.99805629
86b.l9x6 5.67306928
87b.b10x5 4.5175609
88b.b11x4 5.5655529
89b.l11x2 8.57292429
90b.b12x3 3.72479458
91b.b12x5 3.9275456
92b.b12x6 9.09167628
93b.b13x7 8.26267557
94b.l13x3 7.12194659
95b.l13x6 5.68229429
96b.l13x7 4.685459
97b.b14x3 4.89479455
98b.b15x1 7.62267559
99b.b15x3 4.67125459
100b.l15x1 5.27427
101b.l15x2 5.484559
102b.b16x4 8.23333556
103b.b16x5 4.68563405
104b.b16x6 8.47403658
105b.b17x5 7.08563447
106b.b17x7 8.39125448
107b.l17x3 9.41889649
108b.l17x6 6.032529
109b.b18x3 5.16979448
110b.b18x5 4.53688405
111b.l18x1 5.903457136
112b.l18x2 6.052924137
113b.b19x2 8.44267546
114b.b19x4 6.38312448
115b.l19x2 6.8495549
116b.b20x2 6.25917446
117b.b20x4 10.7563548
118b.b20x6 8.1075546
119b.b21x1 8.1225447
120b.b21x5 4.75688404
121b.b21x7 5.66625605
122b.b22x5 6.425624137
123b.l22x5 6.574586169
124b.b23x6 7.255836147
125b.l23x1 7.70729406
126b.b24x2 5.134584145
127b.b24x4 7.2195146
128b.b24x6 6.832294148
129b.l25x3 8.75017599
130b.b26x3 3.99917406
131b.l27x1 11.4323729
132b.l27x2 8.82479499
133b.b28x3 4.71583437
134b.b28x4 8.03854496
135b.b28x6 7.61153699
136g.h1x1 2.18267502
137g.l1x4 4.257508
138g.l1x6 3.752294244
139g.h2x11 8.191464136
140g.ctx3 5.40556609
141g.ctx6 3.37667406
142g.ctx14 3.9495539
143g.ctx15 6.28896439
144g.ctx16 4.62802838
145NT 13.0609815
1461x35 5.51188415
1471x39 5.13083618
1481x57 5.36254277
1492x42 4.47754287
1502x43 3.515834278
1512x44 4.73917406
1522x50 7.26479409
1532x53 5.66813417
1542x64 5.534516
155E1x50 6.766816109
156E1x52 6.5775107
1573x30 4.46767516
1583x32 5.34417416
1593x37 4.83125617
1603x42 8.766884158
1613x50 6.84417409
1623x51 6.217335127
1633x52 3.319584125
1643x53 5.70312408
1653x56 6.128754127
166I2x51 4.34021406
167I2x52 4.808134124
1684x50 5.261674159
169E2 7.467241613
1705x39 4.311464295
1715x44 3.97771416
1725x47 7.09278618
1735x51 4.00958417
1745x54 4.32229418
1755x58 4.007518
176I3 6.068066193
1776x36 4.06292407
1786x44 6.06183519
1796x48 7.266518
1806x51 4.87458416
1816x52 6.515518
1826x55 5.16824915
1836x59 4.42708415
184E3 4.94736614
1857x28 3.04813411
1867x34 7.6315514
1877x39 4.76896416
1887x42 5.83633517
1897x43 3.51521415
1907x47 3.55917418
1917x49 6.00125409
1927x53 4.91514609
1937x54 4.640127277
194Lig 6.922951110
1951x27 2.46400
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.l2x3 b.l2x5 11.18123.2725NoNo085
2b.b3x1 b.l2x3 11.28537.23917NoNo058
3b.b3x1 b.b6x5 11.39262.92917NoYes056
4b.b2x4 b.b6x5 23.84353.90583NoYes066
5b.b10x4 b.b2x4 23.928816.0792NoNo066
6b.b10x2 b.b10x4 24.48383.48083NoNo066
7b.b10x2 b.b14x3 24.60165.02417NoYes065
8b.b11x5 b.b14x3 23.44215.505NoYes065
9b.b10x1 b.b11x5 33.89513.6675NoNo096
10b.b10x1 b.l9x6 34.00913.39NoYes098
11G.H2.07 b.l9x6 56.90984.42167YesYes298
12b.b6x1 b.l9x6 11.63964.69083YesYes098
13G.H2.04 G.H2.07 59.64845YesYes099
14G.H2.04 G.H3.08 77.37673.74417YesNo099
15G.H3.08 G.S4.04 77.41945.37917NoYes099
16G.S4.04 G.s1h1.01 99.98332.25917YesNo099
17G.H1.01 G.s1h1.01 1003.05167YesNo099
18G.H1.01 G.S4.05 98.36283.635YesNo097
19G.H1.04 G.S4.05 98.3764.36333NoNo077
20G.H1.04 G.S5.05 97.44724.91833NoYes1779
21G.S5.03 G.S5.05 97.76863.55917YesYes089
22G.H2.06 b.l9x6 29.04223.58YesYes298
23G.H2.04 G.H2.08 18.14712.92167YesNo098
24G.H2.06 b.l17x6 14.23618.5275YesYes299
25G.H2.06 b.b18x1 14.23643.96667YesNo299
26G.H2.08 G.H3.18 18.0325.44NoYes089
27G.H2.10 b.b6x1 11.00153.105YesYes079
28G.H3.18 G.S4.02 19.41037.42917YesNo2298
29G.S4.02 G.S5.02 19.54483.06583NoNo086
30G.H3.09 G.S4.04 25.958210.5383YesYes799
31G.H3.09 G.S5.02 19.54443.14YesNo096
32G.H3.15 G.H3.17 36.83466.02667NoYes085
33G.H3.15 G.H3.18 36.99533.22333NoYes089
34g.ctx3 g.ctx5 10.13232.94YesNo099
35b.b22x2 b.b26x3 23.76496.00667NoYes086
36b.b22x1 b.b22x2 23.99863.6NoNo088
37b.b22x1 b.l23x1 24.25083.9775NoYes086
38b.l23x1 b.l25x6 45.093618.165YesNo068
39b.b26x3 b.b27x3 11.64533.685YesNo068
40G.H5.10 G.S5.03 99.97223.25NoYes068
41G.H5.10 G.S6.02 99.97876.00583NoYes067
42G.S6.02 G.h4s6.12 50.00188.88583YesNo074
43G.H5.17 G.h4s6.12 49.66025.9625YesNo1954
44G.H5.13 G.H5.17 49.66028.52667NoYes1985
45G.H5.13 G.S6.02 50.00187.27833NoYes087
462x37 I2x52 17.33097.23NoYes074
472x37 2x40 18.01835.35583NoNo077
481x57 2x40 18.36182.94667YesNo077
491x57 2x43 20.36793.45083YesYes2778
502x43 3x46 11.56243.38167YesNo089
513x46 3x50 11.72525.76NoYes099
523x50 G.H5.25 68.75611.8442YesYes097
53G.H5.20 G.H5.25 98.44584.5NoYes097
54G.H5.20 G.H5.26 98.564.2625NoYes095
55G.H5.17 G.H5.26 99.36374.65YesYes055
562x43 7x53 13.90633.51833YesYes089
573x50 7x53 28.36755.6575YesYes099
586x37 G.H5.25 29.60383.035NoYes077
59b.b11x5 b.l13x7 10.67435.65333NoYes069
60b.l17x6 b.l19x1 14.46956.43YesNo299
61b.l17x5 b.l19x1 28.27463.67833NoNo069
62b.l17x5 b.l19x2 27.98363.80167NoYes069
63b.l17x3 b.l19x2 18.96375.88YesYes499
64b.b19x4 b.l17x3 10.54779.355YesYes489
65b.b18x1 b.l19x1 14.09711.6683NoNo299
66b.b17x7 b.b20x6 17.602810.3617YesYes486
67b.b21x7 b.b24x6 13.33658.28YesYes058
68b.b23x6 b.b24x6 14.4616.83417YesYes1478
69b.l21x7 b.l23x1 20.64715.05417NoYes056
70b.l21x7 b.l23x2 20.06676.74083NoNo058
71b.b23x6 b.l23x2 17.63274.3125YesNo078
723x50 5x58 28.98954.115YesYes098
735x54 5x58 56.82073.17YesYes188
745x54 6x44 55.29767.48583YesYes189
755x47 6x44 50.64645.0925YesYes189
765x47 6x52 49.830614.5067YesYes188
775x44 6x52 19.86274.99333YesYes168
785x44 E2 19.24334.28667YesYes163
79E2 NT 15.106427.2083YesYes135
805x58 6x37 28.91285.52YesNo087
816x52 6x55 23.29824.2325YesYes185
826x55 E2 19.68365.88833YesYes153
832x53 7x46 10.05274.59833YesNo078
842x50 7x46 10.20019.32417YesNo098
852x50 7x49 11.55247.81167YesYes099
867x49 7x53 17.19064.52917YesYes099
87G.H3.17 b.l25x6 38.21165.25YesNo258
88b.b20x4 b.b20x6 13.28584.81167YesYes486
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
NTNT24.26671YesYes5522
E2NT27.20831YesYes3512
1x311x353.041671NoYes5522
1x312x646.125831NoYes5621
1x351x397.024171YesYes5821
1x352x648.499171YesYes5621
1x357x393.48251YesYes5622
1x392x613.345831YesNo8712
1x397x395.771YesYes8612
1x397x425.651671YesYes8711
1x427x424.565831NoYes7721
2x533x325.225831YesYes7621
2x563x325.5650NoYes6621
2x602x644.004171NoYes6611
2x64Lig7.479171YesYes6010
3x29E2x523.16251NoNo5411
3x29Lig6.924171NoYes5010
3x327x423.391YesYes6711
3x32Lig7.195831YesYes6010
3x33Lig4.3551NoYes4010
3x36Lig5.604170NoYes8010
E2E213.71421YesYes3311
E2E2x519.206671YesNo3412
E2x52Lig7.33251NoYes4010
5x44E24.286671YesYes6321
6x55E25.888331YesYes5321
7x34E26.868331YesYes4321
E2Lig4.119171YesYes3010
6x58E26.34751NoYes4321
6x62E25.015831NoYes3321
6x557x3410.78671YesYes5422
7x347x3811.69671YesNo4521
7x38Lig15.37671NoYes5010
7x42Lig6.754171YesYes7010
2x60Lig5.924171NoYes6010
1x392x573.905831YesNo8812
2x537x428.821YesYes7721
3x22E23.488331NoYes3321
5x40E24.8551NoYes5321
4x64E23.460831NoYes4321
5x446x552.975831YesYes6522
1x39Lig5.08751YesYes8010
3x33E25.091NoYes4311
3x363x373.810NoYes8712
3x376x553.0851YesYes7522
4x61E25.02251NoYes5321
7x38E2x522.97751NoNo5411
5x406x554.28251NoYes5522
1x362x641.561670NoYes6621
4x68E21.190NoYes0321

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
81.82Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
81.82Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
81.82Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
81.82Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
81.82Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
81.82Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
76.92Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
75.00Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
75.00Single8K5CAcipimox8K5C-HCA2-Acipimox
75.00Consensushca_onOrthosteric Ligandhca2_on
72.73Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
72.73Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
72.73Single8K5BNiacin8K5B-HCA2-Niacin
72.73Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
72.73Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
69.23Single4YAYZD-71554YAY-AT1-ZD-7155
69.23Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
69.23Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
69.23Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
69.23Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
69.23Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
69.23Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
69.23Consensushca_on_gpOrthosteric Ligandhca2_on_gp
64.29Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
64.29Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
63.64Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
62.50Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
62.50Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
61.54Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
61.54Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
61.54Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
61.54Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
61.54Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
60.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
60.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
58.33Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
57.14Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
57.14Single8K5DGSK2560738K5D-HCA2-GSK256073
57.14Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
56.25Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
56.25Single8XYIVUF106618XYI-CXCR3-VUF10661
55.56Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
55.56Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
55.00Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
53.85Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
53.85Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
53.85Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
53.85Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
53.85Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
53.85Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
53.85Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
53.85Consensusangiotensin_offOrthosteric Ligandat1_off
53.33Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
53.33Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
53.33Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
53.33Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
53.33Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
53.33Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
53.33Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
53.33Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
52.94Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
52.94Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
52.63Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
50.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
50.00Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
50.00Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
50.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
50.00Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
50.00Single8IHKAcifran8IHK-HCA3-Acifran
50.00Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
50.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
50.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
50.00Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
50.00Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
50.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
50.00Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
50.00Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
50.00Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
50.00Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
47.62Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
47.62Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
47.37Single4XT1Fractalkine4XT1-US28-Fractalkine
47.37Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
47.06Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
47.06Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
47.06Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
47.06Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
47.06Single9DGIZ85267113509DGI-CB1-Z8526711350
47.06Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
47.06Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
47.06Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
47.06Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
47.06Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
47.06Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
46.67Single2Y04Salbutamol2Y04-β1-Salbutamol
46.67Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
46.67Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
46.67Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
46.67Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
46.67Single7UL4Alvimopan7UL4-μ-Alvimopan
46.67Single7V3ZCP559407V3Z-CB1-CP55940
46.67Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
46.67Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
46.67Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
46.67Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
46.67Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
46.67Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
46.67Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
46.67Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
46.67Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
46.67Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
46.15Single3OE9IT1t3OE9-CXCR4-IT1t
46.15Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
46.15Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
46.15Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
45.45Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
45.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
45.00Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
44.44Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
44.44Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
44.44Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
44.44Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
44.44Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
44.44Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
44.44Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
44.44Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
44.44Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
44.44Consensusprostanoid_offOrthosteric Ligandep_off dp_off
43.75Single2Y03Isoprenaline2Y03-β1-Isoprenaline
43.75Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
43.75Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
43.75Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
43.75Single7C4SS1P7C4S-S1P3-S1P
43.75Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
43.75Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
43.75Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
43.75Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
43.75Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
43.75Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
43.75Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
43.75Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
43.75Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
43.75Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
43.75Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
43.75Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
43.75Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
43.75Consensusblt_offOrthosteric Ligandblt1_off
43.75Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
43.75Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
43.75Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
43.75Consensusep_offOrthosteric Ligandep4_off
43.75Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
43.75Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
43.75Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
43.75Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
43.75Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
43.75Consensustrace-amine_onOrthosteric Ligandta1_on
42.86Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
42.86Single5ZKQABT-4915ZKQ-PAF-ABT-491
42.86Single6AKXA4R6AKX-CCR5-A4R
42.86Single6AKYMaraviroc6AKY-CCR5-Maraviroc
42.86Single6B73MP11046B73-κ-MP1104
42.86Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
42.86Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
42.86Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
42.86Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
42.86Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.86Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.86Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
42.86Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
42.86Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
42.86Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
42.86Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
42.86Single8IWESpermidine8IWE-TA9-Spermidine
42.86Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
42.86Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
42.86Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
42.86Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.86Single8Y0HVUF114188Y0H-CXCR3-VUF11418
42.86Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
42.86Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
42.86Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
42.86Consensusalpha2_offOrthosteric Ligandalpha2c_off
42.86Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
42.86Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
42.11Single4UG2CGS216804UG2-A2A-CGS21680
42.11Single5ZTYAM102575ZTY-CB2-AM10257
42.11Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
42.11Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
42.11Single7SK9CCX6627SK9-ACKR3-CCX662
42.11Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
42.11Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
42.11Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
42.11Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
42.11Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
42.11Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
41.67Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
41.67Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
41.67Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
41.18Single2YDVNECA2YDV-A2A-NECA
41.18Single4DJHJDTic4DJH-κ-JDTic
41.18Single4UHRCGS216804UHR-A2A-CGS21680
41.18Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
41.18Single5G53NECA5G53-A2A-NECA-Gs
41.18Single5XR8AM8415XR8-CB1-AM841
41.18Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
41.18Single6H7JIsoprenaline6H7J-β1-Isoprenaline
41.18Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
41.18Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
41.18Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
41.18Single6TQ7SB-3348676TQ7-OX1-SB-334867
41.18Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
41.18Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
41.18Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
41.18Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
41.18Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
41.18Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
41.18Single7TUYGSK682753A7TUY-GPR183-GSK682753A
41.18Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
41.18Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
41.18Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
41.18Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
41.18Single8E0GBU728E0G-μ-BU72
41.18Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
41.18Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.18Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
41.18Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
41.18Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
41.18Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
41.18Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
41.18Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
41.18Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
41.18Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
41.18Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.18Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
41.18Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
41.18Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
41.18Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
40.91Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
40.91Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
40.91Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
40.00Single2YDOAdenosine2YDO-A2A-Adenosine
40.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
40.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
40.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
40.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
40.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
40.00Single6PS4ICI118-5516PS4-β2-ICI118-551
40.00Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
40.00Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
40.00Single6TPGEMPA6TPG-OX2-EMPA
40.00Single6V9SGTPL114036V9S-OX1-GTPL11403
40.00Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
40.00Single6ZG9GSK10347026ZG9-M1-GSK1034702
40.00Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
40.00Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
40.00Single7F61PF-036547467F61-H3-PF-03654746
40.00Single7QA8Peptide7QA8-STE2-Peptide
40.00Single7QA8Peptide7QA8-STE2-Peptide
40.00Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
40.00Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
40.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
40.00Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
40.00Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
40.00Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
40.00Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
40.00Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
40.00Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
40.00Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
40.00Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
40.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
40.00Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
40.00Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
40.00Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
40.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
40.00Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
40.00Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
40.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
40.00Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
40.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
40.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
40.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
40.00Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
40.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
40.00Single9AS5Mescaline9AS5-5-HT2A-Mescaline
40.00Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
40.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
40.00Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
40.00Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
40.00Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
40.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
40.00Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
40.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
40.00Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
40.00Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
40.00Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
39.13Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
39.13Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
39.13Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
39.13Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
38.89Single4LDEBI1671074LDE-β2-BI167107
38.89Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
38.89Single6ZG4HTL00099366ZG4-M1-HTL0009936
38.89Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
38.89Single7DFPSpiperone7DFP-D2-Spiperone
38.89Single7K15MKD0467K15-BLT1-MKD046-Na
38.89Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
38.89Single7YITNalfurafine7YIT-κ-Nalfurafine
38.89Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
38.89Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
38.89Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
38.89Single9BJKNAM9BJK-μ-Naloxone-NAM
38.89Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
38.89Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
38.89Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
38.89Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
38.89Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
38.89Consensusalpha1_offOrthosteric Ligandalpha1a_off
38.89Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
38.89Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
38.89Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
38.89Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
38.89Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
38.89Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
38.89Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
38.89Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
38.89Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
38.89Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
38.89Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
38.89Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
38.89Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
38.46Single3OE6IT1t3OE6-CXCR4-IT1t
38.46Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
38.46Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
38.46Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.46Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
38.46Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
38.46Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
38.46Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
38.46Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
38.46Single9LRCHistamine9LRC-H4-Histamine
38.46Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
38.46Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
38.46Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
38.46Consensusbombesin_onOrthosteric Ligandbb2_on
38.46Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
38.46Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
38.46Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
38.46Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
38.10Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
38.10Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
38.10Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
37.50Single3NY8ICI118-5513NY8-β2-ICI118-551
37.50Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
37.50Single4GBRS-Carazolol4GBR-β2-S-Carazolol
37.50Single4QKX35V4QKX-β2-35V
37.50Single4XT3Fractalkine4XT3-US28-Fractalkine
37.50Single5DHGC-355DHG-NOP-C-35
37.50Single5DHHSB-6121115DHH-NOP-SB-612111
37.50Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
37.50Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
37.50Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
37.50Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
37.50Single6GPSMK08126GPS-CCR2-MK0812
37.50Single6H7MSalbutamol6H7M-β1-Salbutamol
37.50Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
37.50Single6PS1Timolol6PS1-β2-Timolol
37.50Single6TOTLemborexant6TOT-OX1-Lemborexant
37.50Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
37.50Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
37.50Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
37.50Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
37.50Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
37.50Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
37.50Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
37.50Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
37.50Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
37.50Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
37.50Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
37.50Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
37.50Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
37.50Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
37.50Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
37.50Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
37.50Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
37.50Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
37.50Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
37.50Single8JJOAlprenolol8JJO-β2-Alprenolol
37.50Single8T1WCVN4248T1W-GPR6-CVN424
37.50Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
37.50Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
37.50Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
37.50Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
37.50Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
37.50Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
37.50Single9CHXS-Carazolol9CHX-β2-S-Carazolol
37.50Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
37.50Consensusa3_onOrthosteric Liganda3a_on
37.50Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
37.50Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
37.50Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
37.50Consensusblt_onOrthosteric Ligandblt1_on
37.50Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
37.50Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
37.50Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
37.50Consensusdopamine_offOrthosteric Ligandd2_off d3_off
37.50Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
37.50Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
37.50Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
37.50Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
37.50Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
37.50Consensusleukotriene_onOrthosteric Ligandblt_on
37.50Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
36.84Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
36.84Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
36.84Single5X93K-87945X93-ETB-K-8794
36.84Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
36.84Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
36.84Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
36.84Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
36.84Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.84Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
36.84Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
36.84Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
36.84Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
36.84Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
36.84Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
36.84Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
36.84Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
36.84Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
36.84Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
36.84Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
36.84Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
36.84Consensusendothelin_offOrthosteric Ligandetb_off
36.84Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
36.84Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
36.36Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
36.36Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
36.36Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
36.36Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
36.36Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
36.36Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
36.36Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
36.00Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
36.00Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
36.00Consensusglp_onOrthosteric Ligandglp1_on glp2_on
36.00Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
36.00Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
36.00Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
35.71Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
35.71Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
35.71Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
35.71Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
35.71Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
35.71Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
35.71Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
35.71Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
35.71Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
35.71Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
35.71Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
35.71Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
35.71Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
35.29Single2RH1S-Carazolol2RH1-β2-S-Carazolol
35.29Single2YCWS-Carazolol2YCW-β1-S-Carazolol
35.29Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
35.29Single5C1MBU725C1M-μ-BU72
35.29Single5D6LS-Carazolol5D6L-β2-S-Carazolol
35.29Single5JQHS-Carazolol5JQH-β2-S-Carazolol
35.29Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
35.29Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
35.29Single5WIUNemonapride5WIU-D4-Nemonapride
35.29Single5WIVNemonapride5WIV-D4-Nemonapride-Na
35.29Single5WQCEMPA5WQC-OX2-EMPA
35.29Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
35.29Single6D26Fevipiprant6D26-DP2-Fevipiprant
35.29Single6GPXMK08126GPX-CCR2-MK0812
35.29Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
35.29Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
35.29Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
35.29Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
35.29Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
35.29Single6PS6Timolol6PS6-β2-Timolol
35.29Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
35.29Single6TP6Filorexant6TP6-OX1-Filorexant
35.29Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
35.29Single7C61Ergotamine7C61-5-HT1B-Ergotamine
35.29Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
35.29Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
35.29Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
35.29Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
35.29Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
35.29Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
35.29Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
35.29Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
35.29Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
35.29Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.29Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.29Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.29Single8JXSPF-61428JXS-D1-PF-6142
35.29Single8S4DCMF-0198S4D-Apelin-CMF-019
35.29Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.29Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.29Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
35.29Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
35.29Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
35.29Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
35.29Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
35.29Single9EHSLUF76029EHS-A3A-LUF7602
35.29Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
35.29Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
35.29Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
35.29Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
35.29Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
35.29Consensusa3_on_gpOrthosteric Liganda3a_on_gp
35.29Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
35.29Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
35.29Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
35.29Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
35.29Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
35.29Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
35.29Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
35.29Consensusamine_offonOrthosteric Ligandamine_off amine_on
35.29Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
35.29Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
35.29Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
35.29Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
35.29Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
35.29Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
35.29Consensusdp_offOrthosteric Liganddp2_off
35.29Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
35.29Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
35.29Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
35.29Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
35.00Single3NY9ICI118-5513NY9-β2-ICI118-551
35.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
35.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
35.00Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
35.00Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
35.00Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
35.00Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
35.00Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
35.00Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
35.00Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
35.00Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
34.78Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
34.78Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
34.78Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
34.78Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
34.78Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
34.78Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
34.78Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
34.78Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
34.78Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
34.78Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
34.62Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
34.62Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
34.62Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
34.62Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
33.33Single3ODUIT1t3ODU-CXCR4-IT1t
33.33Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
33.33Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
33.33Single4S0VSuvorexant4S0V-OX2-Suvorexant
33.33Single5D5AS-Carazolol5D5A-β2-S-Carazolol
33.33Single5D5BS-Carazolol5D5B-β2-S-Carazolol
33.33Single5WS3EMPA5WS3-OX2-EMPA
33.33Single5XRAAM115425XRA-CB1-AM11542
33.33Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
33.33Single6J21Aprepitant6J21-NK1-Aprepitant
33.33Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
33.33Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
33.33Single6TODEMPA6TOD-OX1-EMPA-Na
33.33Single6TPJSuvorexant6TPJ-OX2-Suvorexant
33.33Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
33.33Single7B6WCyclazosin7B6W-α1b-Cyclazosin
33.33Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
33.33Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
33.33Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
33.33Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
33.33Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
33.33Single7FEECP559407FEE-CB1-CP55940-ZCZ011
33.33Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
33.33Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
33.33Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
33.33Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
33.33Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
33.33Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
33.33Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
33.33Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
33.33Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
33.33Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
33.33Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
33.33Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
33.33Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
33.33Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
33.33Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
33.33Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
33.33Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
33.33Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
33.33Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
33.33Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
33.33Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
33.33Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
33.33Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
33.33Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
33.33Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
33.33Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
33.33Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
33.33Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
33.33Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
33.33Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
33.33Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
33.33Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
33.33Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
33.33Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
33.33Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
33.33Single8WDTphotoNECA8WDT-A2A-photoNECA
33.33Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
33.33Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
33.33Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
33.33Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
33.33Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
33.33Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
33.33Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
33.33Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
33.33Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
33.33Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
33.33Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
33.33Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
33.33Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
33.33Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
33.33Single9M4TSilodosin9M4T-Alpha1A-Silodosin
33.33Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
33.33Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
33.33Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
33.33Consensusa2_onOrthosteric Liganda2b_on
33.33Consensusa2_on_gpOrthosteric Liganda2b_on_gp
33.33Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
33.33Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
33.33Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
33.33Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
33.33Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
33.33Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
33.33Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
33.33Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
33.33Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
33.33Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
33.33Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
33.33Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
33.33Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
33.33Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
33.33Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
33.33Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
33.33Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
33.33Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
33.33Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
33.33Consensuslpl_onOrthosteric Ligands1p_on lpa_on
33.33Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
33.33Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
33.33Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
33.33Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
33.33Consensusorexin_offOrthosteric Ligandox2_off ox1_off
33.33Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
33.33Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
33.33Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
33.33Consensusrelaxin_onOrthosteric Ligandrxfp4_on
33.33Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
33.33Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
33.33Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
33.33Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
32.00Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
32.00Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
32.00Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
32.00Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
32.00Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
32.00Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
32.00Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
32.00Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
32.00Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
32.00Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
32.00Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
31.82Single3QAKUK-4320973QAK-A2A-UK-432097
31.82Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
31.82Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
31.82Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
31.82Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
31.82Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
31.82Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
31.82Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
31.82Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
31.82Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
31.82Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
31.82Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
31.58Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
31.58Single3D4STimolol3D4S-β2-Timolol
31.58Single4AMIBucindolol4AMI-β1-Bucindolol
31.58Single4RWADIPP-NH24RWA-δ-DIPP-NH2
31.58Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
31.58Single5X33BIIL2605X33-BLT1-BIIL260
31.58Single6A93Risperidone6A93-5-HT2A-Risperidone
31.58Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
31.58Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
31.58Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
31.58Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
31.58Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
31.58Single6KQICP559406KQI-CB1-CP55940-Org27569
31.58Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
31.58Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
31.58Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
31.58Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
31.58Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
31.58Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
31.58Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
31.58Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
31.58Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
31.58Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
31.58Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.58Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
31.58Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
31.58Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
31.58Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single8JJ8Formoterol8JJ8-β2-Formoterol
31.58Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
31.58Single8JWY2-1188JWY-A2A-2-118
31.58Single8JWZAB9288JWZ-A2A-AB928-Na
31.58Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.58Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.58Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
31.58Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
31.58Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
31.58Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
31.58Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
31.58Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
31.58Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
31.58Consensuslpl_offOrthosteric Ligands1p_off lpa_off
31.58Consensusorexin_onOrthosteric Ligandox2_on
31.58Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.58Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.25Single6IQLL7458706IQL-D4-L745870
31.25Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
31.25Single6KUXRS-799486KUX-α2a-RS-79948
31.25Single6PS5S-Propranolol6PS5-β2-S-Propranolol
31.25Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
31.25Single6TP3Nemorexant6TP3-OX1-Nemorexant
31.25Single6VI4JDTic6VI4-κ-JDTic
31.25Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
31.25Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
31.25Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
31.25Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
31.25Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
31.25Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
31.25Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
31.25Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
31.25Single7UL3Famotidine7UL3-H2-Famotidine
31.25Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
31.25Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
31.25Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
31.25Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
31.25Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.25Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.25Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.25Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
31.25Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
31.25Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
31.25Single8K2WAMG4878K2W-CXCR3-AMG487
31.25Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
31.25Single8RLNLUF58348RLN-A2A-LUF5834
31.25Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
31.25Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.25Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.25Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.25Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.25Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
31.25Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
31.25Single8ZPMAMD0708ZPM-CXCR4-AMD070
31.25Single9AS3LSD9AS3-5-HT2A-LSD
31.25Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
31.25Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
31.25Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
31.25Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
31.25Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
31.25Consensusalpha1_onOrthosteric Ligandalpha1a_on
31.25Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
31.25Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
31.25Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
31.25Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
31.25Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
31.25Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
31.25Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
30.77Single3OE8IT1t3OE8-CXCR4-IT1t
30.77Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
30.77Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
30.77Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
30.77Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
30.77Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
30.77Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
30.77Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
30.77Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
30.77Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
30.77Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
30.77Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
30.77Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
30.77Single9CHUNoradrenaline9CHU-β2-Noradrenaline
30.77Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
30.77Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
30.77Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
30.77Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
30.43Single5WF5UK-4320975WF5-A2A-UK-432097
30.43Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
30.43Single6W25SHU91196W25-MC4-SHU9119-Ca
30.43Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
30.43Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
30.43Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
30.43Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
30.43Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.43Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
30.43Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
30.43Consensusangiotensin_onOrthosteric Ligandat1_on
30.43Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
30.43Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
30.43Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
30.43Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
30.43Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
30.43Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
30.43Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
30.00Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
30.00Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
30.00Single6H7LDobutamine6H7L-β1-Dobutamine
30.00Single6IBLArformoterol6IBL-β1-Arformoterol
30.00Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
30.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
30.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
30.00Single7EZCUKA7EZC-A2A-UKA
30.00Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
30.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
30.00Single7UM4AS26747237UM4-5-HT5A-AS2674723
30.00Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
30.00Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
30.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
30.00Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
30.00Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
30.00Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
30.00Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
30.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
30.00Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
30.00Consensuscck_onOrthosteric Ligandccka_on cckb_on
30.00Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
30.00Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
30.00Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
30.00Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
30.00Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
30.00Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
30.00Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
29.63Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
29.63Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
29.63Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
29.63Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
29.63Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
29.41Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
29.41Single2Y01Dobutamine2Y01-β1-Dobutamine
29.41Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
29.41Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
29.41Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
29.41Single4EJ4Naltrindole4EJ4-δ-Naltrindole
29.41Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
29.41Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
29.41Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
29.41Single5TGZAM65385TGZ-CB1-AM6538
29.41Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
29.41Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
29.41Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
29.41Single6DRXLisuride6DRX-5-HT2B-Lisuride
29.41Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
29.41Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
29.41Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
29.41Single7BU7BI1671077BU7-β1-BI167107
29.41Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
29.41Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
29.41Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
29.41Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
29.41Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
29.41Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
29.41Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
29.41Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
29.41Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
29.41Single7WC7Lisuride7WC7-5-HT2A-Lisuride
29.41Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
29.41Single7YXAONO-54306087YXA-S1P5-ONO-5430608
29.41Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
29.41Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
29.41Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
29.41Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
29.41Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
29.41Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
29.41Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
29.41Single8JXRLSD8JXR-D1-LSD
29.41Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
29.41Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
29.41Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
29.41Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
29.41Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
29.41Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
29.41Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
29.41Single9AS1DMT9AS1-5-HT2A-DMT
29.41Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
29.41Single9JEAAtropine9JEA-M1-Atropine
29.41Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
29.41Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
29.41Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
29.41Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
29.41Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
29.41Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
29.41Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
29.41Consensus5ht5_onOrthosteric Ligand5ht5a_on
29.41Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
29.41Consensusalpha2_onOrthosteric Ligandalpha2b_on
29.41Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
29.41Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
29.41Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
29.41Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
29.41Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
29.41Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
29.41Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
29.41Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
29.41Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
29.41Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
29.17Single6JODAngiotensin II6JOD-AT2-Angiotensin II
29.17Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
29.17Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
29.17Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
29.17Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.17Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
29.17Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
29.17Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
29.17Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
29.17Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
29.17Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
29.17Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
29.17Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
29.17Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
29.03Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
29.03Consensuspth_onOrthosteric Ligandpth1_on pth2_on
28.57Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
28.57Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
28.57Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
28.57Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
28.57Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
28.57Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
28.57Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
28.57Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
28.57Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
28.57Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
28.57Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
28.57Single8QJ2pN1628QJ2-MC4-pN162-Gs
28.57Single8X5YAstemizole8X5Y-H1-Astemizole
28.57Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
28.57Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
28.57Single9IPYJR14a9IPY-C3aB-JR14a
28.57Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
28.57Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensus5ht2_onOrthosteric Ligand5ht2b_on
28.57Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
28.57Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
28.57Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
28.00Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
28.00Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
28.00Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
28.00Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
28.00Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
28.00Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
28.00Single8ZRTET-18ZRT-ETB-ET-1
28.00Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.00Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
28.00Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
28.00Consensuspac_onOrthosteric Ligandpac1_on
28.00Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
27.78Single2Y00Dobutamine2Y00-β1-Dobutamine
27.78Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
27.78Single5TVNLSD5TVN-5-HT2B-LSD
27.78Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
27.78Single6E67BI1671076E67-β2-BI167107-Gs(CT)
27.78Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
27.78Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
27.78Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
27.78Single7SINNPS-21437SIN-CaS-NPS-2143
27.78Single7SINNPS-21437SIN-CaS-NPS-2143
27.78Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
27.78Single7W41PD1762527W41-BB2-PD176252
27.78Single7WC6LSD7WC6-5-HT2A-LSD
27.78Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
27.78Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
27.78Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.78Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
27.78Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
27.78Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
27.78Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
27.78Single8TF5Oleic acid8TF5-GPR6-Oleic acid
27.78Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
27.78Single8ZMFA1L108ZMF-5-HT2C-A1L10
27.78Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
27.78Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
27.78Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
27.78Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
27.78Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
27.78Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
27.78Single9HAPTolvaptan9HAP-V2-Tolvaptan
27.78Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
27.78Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.78Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
27.78Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
27.78Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
27.78Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
27.78Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
27.78Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
27.78Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
27.78Consensusbombesin_offOrthosteric Ligandbb2_off
27.78Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
27.78Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
27.78Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
27.78Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.78Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.78Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
27.59Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
27.59Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
27.59Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
27.59Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
27.27Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
27.27Single4IARErgotamine4IAR-5-HT1B-Ergotamine
27.27Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
27.27Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
27.27Single7F8XNN90567F8X-CCKA-NN9056
27.27Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
27.27Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
27.27Single8KIGSHU91198KIG-MC3-SHU9119-Ca
27.27Single8WKYPG-9348WKY-MC4-PG-934
27.27Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
27.27Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
27.27Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
27.27Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
27.27Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
27.27Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
27.27Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
26.92Single6FJ3PTH6FJ3-PTH1-PTH
26.92Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
26.92Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
26.92Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
26.92Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
26.92Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
26.92Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
26.92Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
26.92Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
26.92Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
26.92Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
26.92Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
26.92Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
26.92Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
26.92Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
26.92Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
26.92Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
26.92Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
26.92Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
26.67Single3PBLEticlopride3PBL-D3-Eticlopride
26.67Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
26.67Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
26.67Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
26.67Single7SRQLSD7SRQ-5-HT2B-LSD
26.67Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
26.67Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
26.67Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
26.67Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.67Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
26.67Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
26.67Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.67Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
26.67Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
26.67Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
26.67Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
26.67Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
26.67Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
26.67Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
26.67Consensusgq_nucleotideOrthosteric Ligandgq_p2y
26.67Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
26.67Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
26.32Single3P0GBI1671073P0G-β2-BI167107
26.32Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
26.32Single4U15Tiotropium4U15-M3-Tiotropium
26.32Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
26.32Single5V54Methiothepin5V54-5-HT1B-Methiothepin
26.32Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
26.32Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
26.32Single6J20Aprepitant6J20-NK1-Aprepitant
26.32Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
26.32Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
26.32Single6OL9Tiotropium6OL9-M5-Tiotropium
26.32Single6WGTLSD6WGT-5-HT2A-LSD
26.32Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
26.32Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
26.32Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.32Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
26.32Single8EA0Iperoxo8EA0-M3-Iperoxo
26.32Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
26.32Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
26.32Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
26.32Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
26.32Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
26.32Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
26.32Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
26.32Single8XVLZibotentan8XVL-ETA-Zibotentan
26.32Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
26.32Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
26.32Single8ZWFJR14a8ZWF-C3aB-JR14a
26.32Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
26.32Single9BJKNaloxone9BJK-μ-Naloxone-NAM
26.32Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
26.32Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Consensus5ht1_offOrthosteric Ligand5ht1b_off
26.32Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
26.32Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
26.32Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
26.32Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
26.32Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
26.32Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
26.09Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
26.09Single6HLOAprepitant6HLO-NK1-Aprepitant
26.09Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
26.09Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
26.09Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
26.09Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
26.09Single7XNACYN1548067XNA-SST2-CYN154806
26.09Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
26.09Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
26.09Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
26.09Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
26.09Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
26.09Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
26.09Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
26.09Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
26.09Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
26.09Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
26.09Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
26.09Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
26.09Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
26.09Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
25.93Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
25.93Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
25.93Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
25.93Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
25.93Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
25.93Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
25.93Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
25.93Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
25.93Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
25.93Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
25.93Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
25.93Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
25.81Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
25.81Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
25.81Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.81Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
25.71Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
25.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
25.00Single3OE0CVX153OE0-CXCR4-CVX15
25.00Single3PWHZM-2413853PWH-A2A-ZM-241385
25.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
25.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
25.00Single5CXVTiotropium5CXV-M1-Tiotropium
25.00Single5U09Taranabant5U09-CB1-Taranabant
25.00Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
25.00Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
25.00Single6CM4Risperidone6CM4-D2-Risperidone
25.00Single6IGLIRL16206IGL-ETB-IRL1620
25.00Single6IIURamatroban6IIU-TXA2-Ramatroban
25.00Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
25.00Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
25.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
25.00Single6MXTSalmeterol6MXT-β2-Salmeterol
25.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
25.00Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
25.00Single6PT2KGCHM076PT2-δ-KGCHM07
25.00Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
25.00Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
25.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
25.00Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
25.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
25.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
25.00Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
25.00Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
25.00Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
25.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
25.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
25.00Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
25.00Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
25.00Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
25.00Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
25.00Single7XRRLemborexant7XRR-OX2-Lemborexant
25.00Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
25.00Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
25.00Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
25.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
25.00Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
25.00Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
25.00Single8JJLOlodaterol8JJL-β2-Olodaterol
25.00Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
25.00Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
25.00Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
25.00Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
25.00Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
25.00Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
25.00Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
25.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
25.00Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
25.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
25.00Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
25.00Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
25.00Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
25.00Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
25.00Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
25.00Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
25.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
25.00Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
25.00Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
25.00Consensusbradykinin_onOrthosteric Ligandbk2_on
25.00Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
25.00Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.00Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
25.00Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
25.00Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
25.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
25.00Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
25.00Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
25.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
25.00Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
25.00Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
25.00Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
25.00Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
25.00Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
25.00Consensuslpa_offOrthosteric Ligandlpa1_off
25.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
25.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
25.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
25.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
25.00Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
25.00Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
25.00Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
25.00Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
24.24Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
24.24Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
24.14Single5GLHEndothelin-15GLH-ETB-Endothelin-1
24.14Single6IGKEndothelin-36IGK-ETB-Endothelin-3
24.14Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
24.14Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
24.14Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
24.14Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
24.14Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
24.14Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
24.14Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
24.00Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
24.00Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
24.00Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
24.00Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
24.00Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
24.00Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
24.00Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
24.00Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
24.00Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
24.00Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
24.00Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
24.00Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
24.00Consensusvasop-oxy_onOrthosteric Ligandv2_on
24.00Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
23.81Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
23.81Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
23.81Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
23.81Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
23.81Single6K1QIRL25006K1Q-ETB-IRL2500
23.81Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
23.81Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
23.81Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
23.81Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
23.81Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
23.81Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
23.81Single8XVJMacitentan8XVJ-ETA-Macitentan
23.81Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
23.81Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
23.81Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
23.81Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
23.81Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
23.81Consensuschemerin_onOrthosteric Ligandcml1_on
23.81Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.53Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
23.53Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
23.53Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
23.53Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
23.53Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
23.53Single6A94Zotepine6A94-5-HT2A-Zotepine
23.53Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
23.53Single6TPNHTL66416TPN-OX2-HTL6641
23.53Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
23.53Single7AROLUF58337ARO-A2A-LUF5833-Na
23.53Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
23.53Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
23.53Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
23.53Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
23.53Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
23.53Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
23.53Single7T32ZM-2413857T32-A2A-ZM-241385
23.53Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.53Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
23.53Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
23.53Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
23.53Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
23.53Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
23.53Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
23.53Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
23.53Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
23.53Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
23.53Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
23.53Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
23.53Single8ZPNAMD31008ZPN-CXCR4-AMD3100
23.53Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
23.53Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
23.53Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
23.53Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
23.53Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
23.53Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
23.53Consensusopsins_offOrthosteric Ligandrhodopsin_off
23.53Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
23.53Consensussensory_offOrthosteric Ligandopsins_off
23.33Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
23.33Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
23.33Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
23.33Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
23.08Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
23.08Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
23.08Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
23.08Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
23.08Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
23.08Single8PWNTheophylline8PWN-A2A-Theophylline
23.08Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
23.08Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
23.08Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
23.08Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
23.08Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
22.73Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
22.73Single5WF6UK-4320975WF6-A2A-UK-432097
22.73Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
22.73Single6PT3DPI-2876PT3-δ-DPI-287
22.73Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
22.73Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
22.73Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
22.73Single7XN9L-054,5227XN9-SST2-L-054,522
22.73Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
22.73Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
22.73Single9JF4PD1683689JF4-BB1-PD168368
22.73Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
22.73Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
22.73Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
22.73Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
22.58Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
22.58Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
22.58Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
22.58Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
22.58Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
22.58Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.58Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
22.58Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
22.58Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
22.22Single2Y02Carmoterol2Y02-β1-Carmoterol
22.22Single4DAJTiotropium4DAJ-M3-Tiotropium
22.22Single4MQSIperoxo4MQS-M2-Iperoxo
22.22Single4U14Tiotropium4U14-M3-Tiotropium
22.22Single5DSGTiotropium5DSG-M4-Tiotropium
22.22Single5UENDU1725UEN-A1-DU172
22.22Single5UIGCmpd-15UIG-A2A-Cmpd-1
22.22Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
22.22Single6IIVDaltroban6IIV-TXA2-Daltroban
22.22Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
22.22Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
22.22Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
22.22Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
22.22Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
22.22Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
22.22Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
22.22Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
22.22Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
22.22Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
22.22Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
22.22Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.22Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
22.22Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
22.22Single8CU6LJ-45178CU6-A2A-LJ-4517
22.22Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
22.22Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
22.22Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
22.22Single8X63Mepyramine8X63-H1-Mepyramine
22.22Single8X64Desloratadine8X64-H1-Desloratadine
22.22Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
22.22Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
22.22Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
22.22Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
22.22Single9H37A1IR09H37-A2A-A1IR0-Na
22.22Single9IYAONO-97105319IYA-GPR55-ONO-9710531
22.22Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
22.22Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
22.22Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
22.22Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
22.22Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
22.22Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
22.22Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.22Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.22Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.22Consensushistamine_offOrthosteric Ligandh1_off
22.22Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
22.22Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
22.22Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
22.22Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
22.22Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
21.88Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
21.74Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
21.74Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
21.74Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
21.74Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
21.74Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
21.74Single8IEBA1LYA8IEB-GPR156-A1LYA
21.74Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
21.74Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
21.74Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
21.74Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
21.74Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
21.74Consensussomatostatin_offOrthosteric Ligandsst2_off
21.43Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
21.43Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
21.43Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
21.43Single6TQ9SB-4081246TQ9-OX1-SB-408124
21.43Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
21.43Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
21.43Single8A2OTheophylline8A2O-A2A-Theophylline-Na
21.43Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
21.43Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
21.43Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
21.43Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
21.43Single9KDFRES-701-39KDF-ETB-RES-701-3
21.43Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
21.43Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
21.43Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
21.43Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
21.43Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
21.43Consensussensory_onOrthosteric Ligandopsins_on
21.05Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
21.05Single5CGCHTL142425CGC-mGlu5-HTL14242
21.05Single5N2RPSB-365N2R-A2A-PSB-36-Na
21.05Single5N2SPSB365N2S-A1-PSB36
21.05Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
21.05Single5XPRBosentan5XPR-ETB-Bosentan
21.05Single6LUQHaloperidol6LUQ-D2-Haloperidol
21.05Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
21.05Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
21.05Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
21.05Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
21.05Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
21.05Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
21.05Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
21.05Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.05Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
21.05Single8QOTNanobody-E8QOT-μ-Nanobody-E
21.05Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
21.05Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single9B9ZA1AKO9B9Z-CB1-A1AKO
21.05Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
21.05Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
21.05Consensusadenosine_offOrthosteric Liganda1_off a2_off
21.05Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
21.05Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
21.05Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
21.05Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
20.83Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
20.83Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
20.83Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
20.83Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
20.83Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
20.83Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
20.83Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
20.83Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
20.83Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
20.69Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
20.69Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
20.69Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
20.69Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
20.51Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.00Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
20.00Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
20.00Single3UZAGTPL92363UZA-A2A-GTPL9236
20.00Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
20.00Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
20.00Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
20.00Single6E59L-7607356E59-NK1-L-760735
20.00Single6ME5Agomelatine6ME5-MT1-Agomelatine
20.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
20.00Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
20.00Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
20.00Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
20.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
20.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
20.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
20.00Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
20.00Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
20.00Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
20.00Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
20.00Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
20.00Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
20.00Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
20.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
20.00Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
20.00Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
20.00Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
20.00Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
20.00Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
20.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
20.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
20.00Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
20.00Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
20.00Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
20.00Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
20.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
20.00Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
20.00Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
20.00Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
20.00Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
20.00Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
20.00Single9AS9RS130-1809AS9-5-HT2A-RS130-180
20.00Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
20.00Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
20.00Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
20.00Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
20.00Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
20.00Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
20.00Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
20.00Consensusgi_sensoryOrthosteric Ligandgi_opsins
20.00Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
20.00Consensuslpa_onOrthosteric Ligandlpa1_on
20.00Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
20.00Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
20.00Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
20.00Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
20.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
20.00Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
20.00Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
20.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
20.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
20.00Consensustachykinin_offOrthosteric Ligandnk1_off
19.44Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
19.35Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
19.23Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
19.23Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
19.23Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
19.23Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
19.23Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
19.23Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
19.23Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
19.23Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
19.23Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
19.23Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
19.23Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
19.23Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
19.05Single4N4WSANT-14N4W-SMO-SANT-1
19.05Single4XEENeurotensin4XEE-NTS1-Neurotensin
19.05Single4XESNeurotensin4XES-NTS1-Neurotensin
19.05Single6OS2TRV0266OS2-AT1-TRV026
19.05Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
19.05Single6YVRNTS8-136YVR-NTS1-NTS8-13
19.05Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
19.05Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.05Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
19.05Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
19.05Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
19.05Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
19.05Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.05Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
19.05Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
19.05Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
19.05Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
19.05Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
19.05Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
18.92Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
18.75Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
18.75Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
18.75Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
18.75Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
18.75Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
18.75Single5L7IVismodegib5L7I-SMO-Vismodegib
18.75Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
18.75Single6HLLCP999946HLL-NK1-CP99994
18.75Single6LI0C176LI0-GPR52-C17
18.75Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
18.75Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
18.75Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
18.75Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
18.75Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
18.75Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
18.75Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
18.75Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
18.75Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
18.75Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
18.75Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
18.75Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
18.75Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
18.75Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.75Single9AS7Psilocin9AS7-5-HT2A-Psilocin
18.75Single9B9Y7DY9B9Y-CB1-7DY
18.75Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
18.52Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
18.52Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
18.52Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
18.52Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Consensuscalcitonin_onOrthosteric Ligandctlike_on
18.52Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single4BUONeurotensin4BUO-NTS1-Neurotensin
18.18Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
18.18Single5CGDHTL142425CGD-mGlu5-HTL14242
18.18Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
18.18Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
18.18Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
18.18Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
18.18Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
18.18Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
18.18Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
18.18Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8ZPLHF511168ZPL-CXCR4-HF51116
18.18Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
18.18Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
18.18Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
18.18Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single7SK3CXCL127SK3-ACKR3-CXCL12
17.86Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
17.86Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
17.86Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
17.86Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
17.65Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
17.65Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
17.65Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
17.65Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
17.65Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
17.65Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
17.65Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
17.65Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
17.65Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
17.65Single6DS0Ly2660976DS0-5-HT2B-Ly266097
17.65Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.65Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
17.65Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
17.65Single6ME9Ramelteon6ME9-MT2-Ramelteon
17.65Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
17.65Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
17.65Single7F8YDevazepide7F8Y-CCKA-Devazepide
17.65Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
17.65Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
17.65Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
17.65Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
17.65Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.65Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
17.65Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
17.65Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
17.65Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
17.65Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
17.65Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
17.65Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
17.65Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
17.65Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
17.65Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
17.65Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
17.65Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
17.65Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
17.65Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.65Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.65Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
17.65Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
17.65Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
17.65Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
17.65Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
17.65Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
17.65Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
17.65Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
17.65Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
17.65Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
17.65Single9H2XA1IR19H2X-A2A-A1IR1-Na
17.65Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
17.65Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
17.65Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
17.39Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
17.39Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
17.39Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
17.39Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
17.39Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
17.39Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
17.39Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
17.39Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
17.39Consensuskisspeptin_onOrthosteric Ligandkiss1_on
17.39Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
17.24Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
17.14Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
16.67Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
16.67Single3REYXAC3REY-A2A-XAC
16.67Single3RZECidoxepin3RZE-H1-Cidoxepin
16.67Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
16.67Single5IU7Q274563465IU7-A2A-Q27456346-Na
16.67Single5IUBQ274563445IUB-A2A-Q27456344-Na
16.67Single5JTBZM-2413855JTB-A2A-ZM-241385
16.67Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
16.67Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
16.67Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
16.67Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
16.67Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
16.67Single6AQFZM-2413856AQF-A2A-ZM-241385
16.67Single6MH8ZM-2413856MH8-A2A-ZM-241385
16.67Single6TPKRetosiban6TPK-OT-Retosiban
16.67Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
16.67Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
16.67Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
16.67Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
16.67Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
16.67Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
16.67Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
16.67Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
16.67Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
16.67Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
16.67Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
16.67Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
16.67Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
16.67Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
16.67Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
16.67Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
16.67Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
16.67Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
16.67Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
16.67Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
16.67Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
16.67Single8IEIA1LYA8IEI-GPR156-A1LYA
16.67Single8IEIA1LYA8IEI-GPR156-A1LYA
16.67Single8IEPA1LYA8IEP-GPR156-A1LYA
16.67Single8IEPA1LYA8IEP-GPR156-A1LYA
16.67Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.67Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
16.67Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
16.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
16.67Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
16.67Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
16.67Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
16.67Single9ARXSerotonin9ARX-5-HT2A-Serotonin
16.67Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
16.67Single9BA0A1AKN9BA0-CB1-A1AKN
16.67Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
16.67Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
16.67Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
16.67Consensusa2_offOrthosteric Liganda2a_off
16.67Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
16.67Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
16.67Consensusendothelin_onOrthosteric Ligandetb_on eta_on
16.67Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
16.67Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
16.67Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
16.67Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
16.67Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
16.67Consensusvasop-oxy_offOrthosteric Ligandot_off
16.13Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
16.13Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
16.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
16.00Single7SK5CXCL127SK5-ACKR3-CXCL12
16.00Single8IEBA1LYA8IEB-GPR156-A1LYA
16.00Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.00Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
15.79Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
15.79Single3EMLZM-2413853EML-A2A-ZM-241385
15.79Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
15.79Single5IU8Q274563475IU8-A2A-Q27456347-Na
15.79Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
15.79Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
15.79Single5T04Neurotensin5T04-NTS1-Neurotensin
15.79Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
15.79Single6D27CAY104716D27-DP2-CAY10471
15.79Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
15.79Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
15.79Single6S0LZM-2413856S0L-A2A-ZM-241385
15.79Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
15.79Single7F83PF-051904577F83-Ghrelin-PF-05190457
15.79Single7PYRPSB-21157PYR-A2A-PSB-2115
15.79Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
15.79Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
15.79Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
15.79Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
15.79Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.79Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
15.79Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
15.79Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
15.79Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
15.79Consensuscck_offOrthosteric Ligandccka_off
15.79Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
15.62Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
15.62Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
15.62Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
15.62Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
15.38Single5MZPCaffeine5MZP-A2A-Caffeine-Na
15.38Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
15.38Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
15.00Single5IUAQ274563485IUA-A2A-Q27456348-Na
15.00Single6HLPNetupitant6HLP-NK1-Netupitant
15.00Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
15.00Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
15.00Single6S0QZM-2413856S0Q-A2A-ZM-241385
15.00Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
15.00Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
15.00Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
15.00Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
15.00Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
15.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.00Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.00Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
15.00Single8GNEKW-63568GNE-A2A-KW-6356-Na
15.00Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
15.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
15.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
15.00Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
15.00Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
15.00Single9HC04YI9HC0-mGlu5-4YI
15.00Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
15.00Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
15.00Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
15.00Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
14.81Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
14.81Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
14.81Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
14.81Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
14.71Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
14.29Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
14.29Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
14.29Single4BV0Neurotensin4BV0-NTS1-Neurotensin
14.29Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
14.29Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
14.29Single5TZRMK86665TZR-FFA1-MK8666
14.29Single6OS1TRV0266OS1-AT1-TRV026
14.29Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
14.29Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
14.29Single7F1TMIP-1a7F1T-CCR5-MIP-1a
14.29Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
14.29Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
14.29Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
14.29Single7P2L4YI7P2L-mGlu5-4YI
14.29Single7PX4PSB-21137PX4-A2A-PSB-2113
14.29Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
14.29Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
14.29Single7WC4Serotonin7WC4-5-HT2A-Serotonin
14.29Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
14.29Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
14.29Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
14.29Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
14.29Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
14.29Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
14.29Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
14.29Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
14.29Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
14.29Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
14.29Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
14.29Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
14.29Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
14.29Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
14.29Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
14.29Consensusneurotensin_onOrthosteric Ligandnts1_on
14.29Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
14.29Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.79Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
13.79Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
13.79Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
13.64Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
13.64Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
13.64Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
13.64Single4PY02MeSATP4PY0-P2Y12-2MeSATP
13.64Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
13.64Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
13.64Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.64Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
13.64Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
13.64Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
13.64Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.64Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.64Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
13.64Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.33Single3RFMCaffeine3RFM-A2A-Caffeine
13.33Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
13.33Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
13.33Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
13.04Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
13.04Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
13.04Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
13.04Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
12.90Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
12.90Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
12.90Single8IY6Endothelin-18IY6-ETB-Endothelin-1
12.90Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
12.90Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
12.90Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
12.90Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
12.50Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
12.50Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
12.50Single7WC5Psilocin7WC5-5-HT2A-Psilocin
12.50Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
12.50Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
12.50Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
12.50Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.50Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
12.50Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
12.50Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
12.50Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
12.12Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
12.00Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
12.00Single8XWNCXCL88XWN-CXCR2-CXCL8
12.00Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
11.76Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
11.76Single6TP4ACT-4622066TP4-OX1-ACT-462206
11.76Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
11.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
11.76Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
11.76Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
11.76Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
11.76Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
11.76Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
11.76Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
11.76Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
11.76Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
11.54Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
11.54Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
11.54Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
11.54Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
11.54Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
11.43Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
11.11Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
11.11Single4BWBNeurotensin4BWB-NTS1-Neurotensin
11.11Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
11.11Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
11.11Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
11.11Single7BR3Elagolix7BR3-GnRH1-Elagolix
11.11Single7F8ULintitript7F8U-CCKA-Lintitript
11.11Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
11.11Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
11.11Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
11.11Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
11.11Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.11Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
11.11Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
11.11Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
10.53Single5UVIZM-2413855UVI-A2A-ZM-241385
10.53Single6FFIMMPEP6FFI-mGlu5-MMPEP
10.53Single7VODCariprazine7VOD-5-HT2A-Cariprazine
10.53Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
10.53Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
10.53Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.53Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
10.53Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
10.53Consensusgrh_offOrthosteric Ligandgnrh1_off
10.34Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
10.34Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single4QIMANTA XV4QIM-SMO-ANTA XV
10.00Single6FFHFenobam6FFH-mGlu5-Fenobam
10.00Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
10.00Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.00Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
10.00Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
9.52Single4JKVTaladegib4JKV-SMO-Taladegib
9.52Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
9.52Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
9.52Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
9.52Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
9.52Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
9.52Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
9.52Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
9.52Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
9.52Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
9.52Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
9.52Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
9.09Single5V56TC1145V56-SMO-TC114
9.09Single5V57TC1145V57-SMO-TC114
9.09Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
9.09Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
9.09Single7R0CAVP7R0C-V2-AVP-Arrestin2
9.09Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
9.09Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
9.09Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
9.09Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
9.09Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
9.09Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
9.09Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
9.09Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
8.70Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
8.70Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
8.70Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
8.70Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
8.70Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
8.70Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.70Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
8.70Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
8.70Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
8.70Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
8.33Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
8.33Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
8.33Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
8.33Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
8.33Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
8.33Single8XVUCXCL28XVU-CXCR2-CXCL2
8.33Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
8.33Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
8.33Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
8.33Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
8.00Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
8.00Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
8.00Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
8.00Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
7.69Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.69Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
7.69Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.69Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.14Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
7.14Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
6.67Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
6.67Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
6.25Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
6.25Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
6.25Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
6.25Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
6.25Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
6.25Consensusp2y_offOrthosteric Ligandp2y1_off
5.88Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
5.88Single4XNWMRS25004XNW-P2Y1-MRS2500
5.88Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.88Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
5.88Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
5.88Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.88Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.88Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
5.88Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
5.88Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
5.88Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.88Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.88Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
5.56Single4O9RCyclopamine4O9R-SMO-Cyclopamine
5.56Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
5.56Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
5.56Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
5.56Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
5.56Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
5.56Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
5.56Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
5.56Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
5.56Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
5.56Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
5.56Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.26Single4QINSAG1.54QIN-SMO-SAG1.5
5.26Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
5.26Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
5.26Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
5.26Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
5.26Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
5.26Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.26Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
5.26Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
5.26Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
5.26Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
5.26Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
5.26Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
5.00Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
5.00Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
5.00Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
5.00Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
5.00Single6ZINSR486926ZIN-NTS1-SR48692
5.00Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
5.00Single7VV6C48/807VV6-MRGPRX2-C48/80
5.00Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
5.00Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single8IYXYL-3658IYX-GPR34-YL-365
5.00Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
4.76Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
4.76Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
4.76Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
4.76Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
4.76Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
4.76Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
4.76Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
4.76Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
4.76Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
4.55Single4NTJAZD12834NTJ-P2Y12-AZD1283
4.55Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
4.55Single6Z4SSR486926Z4S-NTS1-SR48692
4.55Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
4.55Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
4.55Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
4.35Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
4.35Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.35Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
4.35Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.17Single8XQJJN2418XQJ-Apelin-JN241
4.17Single8XWACXCL18XWA-CXCR2-CXCL1
4.17Single8XWMCXCL68XWM-CXCR2-CXCL6
4.17Single8XWSCXCL58XWS-CXCR2-CXCL5
4.17Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
4.17Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.00Single8XWFCXCL38XWF-CXCR2-CXCL3
4.00Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
3.85Single6KNMJN241-96KNM-Apelin-JN241-9
3.85Single8XQJJN2418XQJ-Apelin-JN241
3.85Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2

Consensus Members
Id Members
gi_hca 8J6R-HCA2-MK6892-Gi1/β1/γ2
8JIM-HCA2-MMF-Gi1/β1/γ2
8IHI-HCA2-Acifran-Gi1/β1/γ2
8IHH-HCA2-LUF6283-Gi1/β1/γ2
8I7V-HCA2-Acipimox-Gi1/β1/γ2
8I7W-HCA2-GSK256073-Gi1/β1/γ2
gi_succinate 8YKW-Succinate-Succinic acid-Gi1/β1/γ1
8YKX-Succinate-Maleic acid-Gi1/β1/γ1
Net Summary
Imin 2.90583
Number of Linked Nodes 901
Number of Links 1115
Number of Hubs 195
Number of Links mediated by Hubs 725
Number of Communities 29
Number of Nodes involved in Communities 277
Number of Links involved in Communities 403
Path Summary
Number Of Nodes in MetaPath 89
Number Of Links MetaPath 88
Number of Shortest Paths 2231501
Length Of Smallest Path 3
Average Path Length 31.3966
Length of Longest Path 54
Minimum Path Strength 0.339583
Average Path Strength 5.61612
Maximum Path Strength 25.3375
Minimum Path Correlation 0.701667
Average Path Correlation 0.978221
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.17391
Average % Of Corr. Nodes 36.7795
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 57.072
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
gi_class-agi_peptide
gi_sensory
gi_alicarboxylic
gi_amine
gi_lipid
gi_nucleotide
gi_protein



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download gi_alicarboxylic.zip



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You can also  read or  download a guide explaining the meaning of all files and numerical data.