Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.50 3.9975405
2G.hns1.01 5.54254154
3G.S1.02 6.71667406
4G.S3.03 6.16444658
5G.S3.04 8.218334137
6G.S3.05 3.66278658
7G.S3.06 8.3085137
8G.s3h2.03 5.07167409
9G.H2.04 4.275409
10G.H2.06 7.6125429
11G.H2.07 5.63667509
12G.h2s4.01 9.15917409
13G.S4.04 4.408509
14G.S4.06 3.50917407
15G.H3.01 2.168509
16G.H3.08 4.36167408
17G.H3.09 5.283896169
18G.H3.13 10.42334166
19G.H3.17 7.32167625
20G.S5.04 4.28417409
21G.S5.06 4.0275408
22G.S5.07 4.294509
23G.s5hg.01 3.589446179
24G.HG.03 3.309174176
25G.HG.15 4.17333407
26G.hgh4.02 5.095834218
27G.hgh4.04 2.660834216
28G.hgh4.11 4.39833435
29G.hgh4.20 4.104533
30G.hgh4.21 6.211674194
31G.H4.07 6.91167435
32G.H4.08 5.04933533
33G.H4.10 7.924675217
34G.H4.12 5.19067534
35G.H4.15 6.71833408
36G.h4s6.02 4.1975407
37G.h4s6.20 7.37083484
38G.S6.02 6.50889688
39G.H5.08 3.84267558
40G.H5.12 4.7925457
41G.H5.17 4.24762785
42G.H5.23 5.893334224
43b.1x3 2.59267501
44b.1x4 2.888508
45b.1x7 3.31267508
46b.1x11 2.7275408
47b.lhb1x6 4.1525143
48b.l1x3 9.34133549
49b.l1x6 9.91667429
50b.b2x1 4.73528
51b.b2x5 6.13722607
52b.l2x5 8.4575465
53b.b3x4 5.18333449
54b.l3x1 6.63083429
55b.l3x2 7.4954159
56b.b4x6 7.82875849
57b.b4x7 6.41167408
58b.b5x3 6.49067549
59b.l5x1 4.33267508
60b.b6x1 4.3775429
61b.b6x5 4.08867506
62b.b8x4 5.59733506
63b.l9x3 6.65286779
64b.l9x6 4.3525828
65b.b10x3 3.4075408
66b.b10x5 4.195609
67b.l10x1 4.3403
68b.b11x4 4.88583479
69b.l11x2 7.18583479
70b.b12x6 9.37945678
71b.b13x3 7.1275474
72b.b13x7 6.30611697
73b.l13x3 7.73867599
74b.b15x1 5.53599
75b.b15x2 7.37583426
76b.b16x4 10.3467496
77b.b16x5 4.62067505
78b.b16x6 8.12722698
79b.b17x5 6.188527
80b.b17x7 8.05417428
81b.l17x3 7.13476729
82b.l17x6 5.66067529
83b.b18x5 6.02333425
84b.l18x1 6.699527116
85b.l18x2 5.499174117
86b.l18x3 8.098334115
87b.b19x2 6.59733526
88b.b19x4 6.52417428
89b.l19x2 6.32267529
90b.b20x2 4.38583426
91b.b20x4 9.37528
92b.b20x6 5.26381726
93b.b20x7 4.27833409
94b.l20x2 7.82833409
95b.b21x1 8.71667527
96b.b21x2 4.87083406
97b.b21x5 4.79667404
98b.b21x7 6.24505
99b.l21x2 6.745834124
100b.b22x5 4.870566117
101b.l22x5 7.325566149
102b.b23x6 6.495127
103b.l23x1 8.11417426
104b.b24x4 7.144126
105b.b24x5 3.2575405
106b.b24x6 5.118675128
107b.l24x3 4.075405
108b.b25x7 8.0875407
109b.l25x3 7.434675109
110b.l25x6 14.2483428
111b.l26x1 6.601674237
112b.l27x1 9.73143729
113b.l27x2 8.015834109
114b.b28x3 3.41547
115b.b28x4 5.881674106
116b.b28x6 10.35424109
117g.h1x10 3.92083409
118g.h1x14 4.67467529
119g.h2x11 8.798334116
120g.ctx3 6.666509
121g.ctx6 3.766675146
122g.ctx14 3.26133509
123g.ctx15 5.55917469
124g.ctx16 5.47762768
125Lig 11.3464810
126NT.F33 6.03267514
127NT.W36 5.78056616
128NT.Y39 6.04857716
129NT.P53 2.9325403
130NT.R60 6.1225404
131NT.Y65 7.65933516
132NT.W68 6.5981719
133NT.P82 5.34167418
134NT.W83 5.67667402
135NT.Y84 6.56111615
136NT.L85 4.605416
137NT.P86 5.01833413
138NT.W87 7.72067513
139NT.K98 6.53933518
140NT.Q105 3.69167415
141NT.W106 7.19958819
142NT.R116 4.5075416
143NT.M123 5.26667513
144NT.D124 4.09667412
1451x30 2.956674262
1461x39 6.06583416
1471x40 11.5742415
1481x43 7.53933517
1491x47 5.068518
1501x61 2.76083408
151I1x49 5.80667408
1522x46 6.191674229
1532x47 4.96867509
1542x50 5.435834229
1552x53 4.1725409
1562x57 7.10733518
1572x60 4.77667418
1582x72 7.19267514
1592x74 7.854514
1602x75 8.89411
161E1.W215 11.288512
1623x36 5.27667406
1633x37 6.37417
1643x46 7.35333709
1653x50 4.72667409
1663x53 7.71533508
1674x46 5.12583407
1684x53 3.80111609
1694x60 7.88167419
1704x64 9.44417408
171E2x51 11.595409
172E2x52 3.8175415
173E2.F303 4.14167404
1745x37 11.3927516
1755x40 9.80833406
1765x53 4.03583408
1776x34 4.61889607
1786x48 6.125409
1796x52 5.32444608
1806x53 3.7125408
1816x61 6.23667414
1827x37 3.358517
1837x41 5.61417417
1847x47 4.85583407
1857x51 2.4225405
1867x56 2.79408
1878x53 5.1075408
1888x58 1.73333405
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1G.HN.40 b.b5x2 10.91688.62667NoNo077
2G.HN.40 b.b5x3 11.33445.59667NoYes079
3b.b3x6 b.l1x3 23.908210.6933NoYes099
4b.b3x6 b.l3x2 24.12467.85333NoYes099
5b.b4x6 b.l1x3 15.73455.99333YesYes499
6G.hns1.01 b.l3x2 26.03533.44667YesYes1549
7G.S1.03 G.hns1.01 28.024810.9767NoYes094
8G.S1.03 G.h2s4.03 30.25663.97NoNo096
9G.h2s4.03 b.l1x6 15.26075.53333NoYes269
10b.l1x6 b.l27x1 17.095318.5667YesYes299
11b.l25x6 b.l27x1 42.573621.99YesYes289
12b.l23x1 b.l25x6 42.560215.0867YesYes268
13b.l21x7 b.l23x1 85.64226.22NoYes056
14b.l21x7 b.l23x2 85.65924.15NoNo058
15b.b24x2 b.l23x2 85.66788.08NoNo058
16b.b24x2 b.b25x6 85.67754.43NoNo053
17b.b24x4 b.b25x6 85.71715.91YesNo063
18b.b24x4 b.b24x6 85.36054.52YesYes1268
19b.b21x7 b.b24x6 85.79728.68333YesYes058
20b.b21x5 b.b21x7 99.618111.1767YesYes045
21b.b21x5 b.h2x1 99.67043.76667YesNo045
22b.h2x1 b.h2x5 99.69223.44NoNo055
23b.h2x5 b.l24x2 99.31095.40333NoNo056
24b.l22x5 b.l24x2 99.281310.1233YesNo096
25b.l22x5 g.ctx6 99.4285.26333YesYes1496
26g.ctx3 g.ctx6 99.90219.04667YesYes096
27g.ctx3 g.ctx5 99.92623.16667YesNo099
28b.lhb1x11 g.ctx5 99.93224.71NoNo049
29b.b25x7 b.lhb1x11 99.93817.06667YesNo074
30b.b25x7 b.b28x6 10018.6YesYes079
31b.b27x3 b.b28x6 49.892510.9167NoYes089
32b.b27x3 b.l25x3 49.87316.84667NoYes089
33b.l25x3 b.l27x2 99.57977.56333YesYes1099
34b.l25x4 b.l27x2 99.46187.09333NoYes059
35I1x49 b.l25x4 99.39795.53YesNo085
362x47 I1x49 49.87724.19667YesYes098
372x46 2x47 48.05410.0433YesYes099
382x46 G.H5.23 22.54068.23YesYes2294
393x53 G.H5.23 22.02753.64333YesYes084
40G.h2s4.02 G.h2s4.03 15.22714.48667NoNo286
41G.h2s4.02 b.l27x1 15.34217.53333NoYes289
42G.H3.17 b.l27x1 42.61983.43667YesYes259
43G.H3.17 b.l23x1 42.97036.33YesYes256
44b.b28x4 b.b28x6 50.06895.02667YesYes1069
45b.b28x4 b.l25x3 49.92246.98667YesYes1069
468x49 I1x49 48.36689.45NoYes098
472x46 8x49 47.98333.48667YesNo099
483x53 3x57 19.858410.55YesNo088
493x57 G.H5.19 19.675211.57NoNo088
50G.H5.15 G.H5.19 19.12573.53667NoNo088
51G.H5.15 G.S1.02 18.94274.42NoYes086
52G.S1.02 G.S3.03 18.20588.29667YesYes068
53G.H2.04 G.H2.07 38.70597YesYes099
54G.H2.07 b.l9x6 38.69284.82333YesYes098
55b.b10x1 b.l9x6 14.39792.96667NoYes098
56b.b10x1 b.b11x5 14.29223.80333NoNo096
57b.b11x5 b.b14x3 14.08495.00333NoNo065
58b.b10x2 b.b14x3 12.50954.23NoNo065
59G.H2.04 G.S1.07 19.13643.24YesNo098
60G.S1.07 G.S4.04 19.02613.65333NoYes089
61G.H2.04 G.H3.08 19.3565.67YesYes098
62G.H3.08 G.S4.04 19.03296.49667YesYes089
63b.b6x1 b.l9x6 50.51455.58667YesYes298
64b.b2x1 b.b6x1 50.66655.19YesYes289
65b.b2x1 b.l27x1 52.58215.14333YesYes289
662x46 2x50 73.3263.00667YesYes2299
672x50 7x57 12.91055.08333YesNo098
686x45 7x57 11.39534.29667NoNo098
696x45 G.H5.25 10.4493.23NoNo098
70G.H5.20 G.H5.25 10.25974.15333NoNo088
71G.S4.04 G.S4.06 15.97233.49333YesYes097
72G.S4.04 G.S5.04 16.65594.46667YesYes099
73G.H1.04 G.S3.05 11.62970.973333NoYes078
74G.H1.03 G.H1.04 11.28221.01333NoNo097
75G.H1.03 G.S5.07 10.24240.973333NoYes099
76G.S4.06 G.S5.06 14.8573.47667YesYes078
77G.S5.04 G.S5.06 14.8873.69YesYes098
78G.H4.10 G.hgh4.08 12.54428.25YesNo076
79G.H4.13 G.hgh4.08 16.55546.13333NoNo036
80G.H4.12 G.H4.13 17.01333.17667YesNo043
81G.H4.12 G.S6.05 21.58564.27333YesNo045
82G.S5.06 G.S6.05 28.3746.09YesNo085
83b.1x19 b.b21x2 13.48666.62NoYes066
84b.b21x2 b.l20x3 13.51764.54667YesNo067
85b.b20x7 b.l20x3 13.5283.6YesNo097
86b.b20x7 b.l20x2 13.56096.35333YesYes099
87b.l18x5 b.l20x2 13.628815.2667NoYes029
88b.l18x3 b.l18x5 13.64899.53667YesNo052
89b.l18x1 b.l18x3 13.44726.85YesYes1165
90b.b22x5 b.l18x1 14.09569.29YesYes1176
91b.b21x7 b.b23x2 15.00214.69YesNo056
922x50 3x50 61.14278.20667YesYes099
932x53 3x50 60.33494.41667YesYes099
942x53 2x57 55.67386.09YesYes098
952x57 2x60 54.95592.89333YesYes188
962x60 3x40 54.83114.84667YesNo185
973x40 Lig 49.709111.2533NoYes150
98b.b22x5 b.b23x2 14.93538.93YesNo076
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x37Lig3.843331YesYes6010
3x40Lig11.25331NoYes8010
5x37Lig8.991YesYes0010
5x43Lig4.153331NoYes7010
7x38Lig13.02330NoYes7010
7x41Lig8.113331YesYes6010
1x43Lig12.55331YesYes8010
1x47Lig6.391YesYes6010
2x64Lig7.641NoYes6010
7x42Lig10.55671NoYes9010
6x61Lig9.636671YesYes0010
7x34Lig11.35331NoYes5010
7x37Lig3.031YesYes7010
1x36Lig18.97331NoYes5010
1x39Lig4.291YesYes7010
E2.N298Lig7.946671NoYes0010
1x40Lig26.371YesYes7010
E2x52Lig6.351YesYes5010
E2.S297Lig5.813331NoYes0010
LigNT.Q273.081YesNo0001
1x29Lig9.721NoYes3010
1x33Lig3.556670NoYes3010
2x75Lig20.711YesYes0010
LigNT.V287.896671YesNo0001
LigNT.M299.736671YesNo0001
E1.Q204Lig3.116671NoYes0010
E1.I206Lig10.751NoYes0010
E1.W215Lig17.231YesYes0010
LigNT.L327.353331YesNo0001
LigNT.W873.511YesYes0001
LigNT.M1235.616671YesYes0001
LigNT.W369.611YesYes0001
E1.V212Lig3.056671NoYes0010
LigNT.Y6513.911YesYes0001
LigNT.Y843.521YesYes0001
E2.D299NT.Q276.960NoNo0021
E1.W215NT.M293.103331YesNo0011
NT.L32NT.P864.381NoYes0011
NT.F33NT.W363.006671YesYes0021
NT.F33NT.K3713.64671YesNo0022
E1.V212NT.F333.056671NoYes0012
NT.K37NT.W366.186671NoYes0021
NT.W36NT.Y8410.611YesYes0011
E1.D209NT.W363.723331NoYes0021
E1.D209NT.K374.151NoNo0022
NT.P82NT.Y393.246671YesYes0022
NT.Y39NT.Y8410.261YesYes0021
NT.S66NT.Y657.630NoYes0021
NT.P82NT.Y656.956671YesYes0021
NT.Y65NT.Y843.971YesYes0011
NT.R116NT.Y655.831YesYes0011
NT.P82NT.Y847.881YesYes0021
NT.L85NT.P823.283331YesYes0022
NT.L85NT.Y843.126671YesYes0021
NT.L85NT.P863.281YesYes0021
NT.L85NT.W878.731YesYes0021
NT.P86NT.W879.461YesYes0011
NT.V91NT.W874.493330NoYes0021
NT.M123NT.W8712.411YesYes0011
NT.K98NT.R1164.541YesYes0021
NT.E127NT.M1233.156671NoYes0021
1x351x363.193330NoNo6521
1x351x398.293330NoYes6721
1x397x3910.361YesNo7512
1x401x437.513331YesYes7811
1x402x686.963331YesNo7112
1x402x725.451YesYes7011
1x431x475.293331YesYes8611
1x432x688.431YesNo8112
1x437x423.906671YesNo8911
1x472x613.113331YesNo6712
1x472x647.151YesNo6611
1x477x463.393331YesNo6912
2x603x404.846671YesNo6821
2x682x727.146671NoYes1021
2x692x7230NoYes4021
2x71E2x524.423330NoYes0521
2x742x753.431YesYes0021
2x74E1.W21523.32331YesYes0021
2x74E2.Q2938.571YesNo0022
2x75E1.W2158.036671YesYes0011
2x75E2.Q2933.383331YesNo0012
E1.Q204E1.W2154.746671NoYes0011
E1.I206E1.V2124.606671NoNo0011
3x363x376.346670YesYes5621
3x363x403.403330YesNo5821
3x374x607.303331YesYes6912
3x375x397.986671YesNo6012
3x445x4313.45670NoNo8721
3x446x525.806670NoYes8722
4x605x399.871YesNo9022
E2.S297E2.V2923.233331NoNo0012
5x37E2.N29818.83331YesNo0011
5x375x393.796671YesNo0012
5x375x4021.99331YesYes0012
5x376x613.351YesYes0011
6x527x415.880YesYes7621
6x557x373.540NoYes7721
6x567x373.306671NoYes4721
6x567x414.776671NoYes4621
6x617x348.733331YesNo0511
6x617x373.226671YesYes0711
7x377x413.686671YesYes7611
LigNT.P862.953331YesYes0001
LigNT.R1165.816671YesYes0001
1x37Lig7.580NoYes4010
1x41Lig3.760NoYes5010
1x44Lig4.183330NoYes7010
2x72Lig19.92671YesYes0010
E2x50E2x522.816670NoYes9521
NT.M123NT.Q1222.721YesNo0012
2x65Lig2.620NoYes4010
NT.I128NT.M1232.430NoYes0021
1x291x322.386671NoNo3512
1x48Lig2.366670NoYes4010
1x29NT.V1301.913331NoNo3012
1x45Lig1.880NoYes5010
7x34E3.A3731.843331NoNo5012
NT.A118NT.R1161.843330NoYes0021
3x33E2x521.680NoYes7521
E1.D208E1.G2071.676670NoNo0021
NT.K64NT.W361.546670NoYes0021
E1.G207Lig1.406671NoYes0010
E1.K205Lig1.383330NoYes0010
1x381x391.320NoYes6721
2x722x760.441YesNo0012

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
96.67Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
57.14Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
57.14Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
55.88Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
55.88Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
54.29Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
54.29Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
52.94Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
51.43Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
51.35Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
50.00Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
50.00Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
48.57Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
47.37Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
46.15Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
45.24Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
45.00Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
45.00Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
44.44Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
44.44Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
42.50Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
42.50Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
42.11Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
41.46Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
39.02Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
37.50Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
35.71Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
35.00Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
34.78Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
34.15Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
34.09Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
33.33Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
33.33Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
32.50Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
31.82Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
31.71Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
31.58Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
31.58Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
31.25Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
30.77Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
30.56Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
30.23Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
30.00Single6FJ3PTH6FJ3-PTH1-PTH
30.00Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
30.00Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
29.55Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
29.27Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
29.27Consensusglp_onOrthosteric Ligandglp1_on glp2_on
29.27Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
28.57Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
28.57Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
28.57Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
28.57Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
28.21Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
28.21Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
28.21Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
28.21Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
27.91Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
27.50Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
27.50Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
27.50Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
27.08Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
26.83Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
26.83Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
26.83Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
26.83Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
26.83Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
26.83Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
26.83Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
26.83Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
26.83Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
26.67Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
26.19Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
26.19Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
26.19Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
26.19Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
26.19Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
26.19Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
26.09Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
26.00Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
25.58Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
25.58Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
25.58Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
25.58Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
25.58Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
25.58Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
25.00Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
25.00Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
25.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
25.00Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
25.00Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
25.00Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
25.00Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
25.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
25.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
25.00Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
25.00Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
25.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
24.44Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
24.44Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
24.44Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
24.39Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
24.39Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
24.39Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
24.39Consensuscalcitonin_onOrthosteric Ligandctlike_on
24.39Consensuspac_onOrthosteric Ligandpac1_on
24.39Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
23.91Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
23.81Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
23.81Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
23.81Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
23.81Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
23.81Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
23.81Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
23.81Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
23.68Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
23.68Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
23.40Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
23.40Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
23.40Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.40Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
23.26Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
23.26Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
23.26Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
23.26Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
23.26Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
23.08Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
23.08Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
23.08Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
22.92Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
22.92Consensuspth_onOrthosteric Ligandpth1_on pth2_on
22.73Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
22.73Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
22.73Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
22.73Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
22.73Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
22.73Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
22.73Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
22.73Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
22.50Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
22.50Consensusangiotensin_onOrthosteric Ligandat1_on
22.50Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
22.50Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
22.50Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
22.22Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
22.22Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
22.22Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
22.22Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
22.00Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
21.95Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
21.95Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
21.95Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
21.74Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
21.74Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
21.62Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
21.62Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
21.43Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
21.43Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
21.05Single4UG2CGS216804UG2-A2A-CGS21680
21.05Single7SK9CCX6627SK9-ACKR3-CCX662
21.05Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
20.93Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
20.93Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
20.83Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
20.59Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
20.59Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
20.51Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
20.51Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
20.51Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
20.51Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
20.51Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
20.51Consensuslpl_onOrthosteric Ligands1p_on lpa_on
20.51Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
20.45Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
20.45Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
20.45Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
20.45Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
20.00Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
20.00Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
20.00Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
20.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
20.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
20.00Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
20.00Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
20.00Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
20.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
20.00Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
20.00Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
20.00Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
20.00Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
20.00Consensusbradykinin_onOrthosteric Ligandbk2_on
20.00Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
20.00Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
19.57Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
19.51Single5WF5UK-4320975WF5-A2A-UK-432097
19.51Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
19.51Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
19.51Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
19.44Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
19.44Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
19.44Consensusa2_onOrthosteric Liganda2b_on
19.44Consensusa2_on_gpOrthosteric Liganda2b_on_gp
19.44Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
19.44Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
19.44Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
19.44Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
19.05Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
19.05Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
19.05Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.05Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.05Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
19.05Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
19.05Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
19.05Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
18.92Single6OS2TRV0266OS2-AT1-TRV026
18.92Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
18.75Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
18.75Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.60Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
18.60Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
18.60Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
18.60Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
18.60Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
18.60Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
18.60Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.42Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
18.42Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
18.42Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
18.42Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
18.18Single4XT3Fractalkine4XT3-US28-Fractalkine
18.18Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
18.18Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
18.18Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
18.18Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
18.18Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
18.18Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
18.18Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
17.95Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
17.95Single5WF6UK-4320975WF6-A2A-UK-432097
17.95Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
17.95Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
17.95Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
17.95Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
17.78Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
17.78Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
17.78Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
17.78Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
17.65Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
17.50Single4XT1Fractalkine4XT1-US28-Fractalkine
17.50Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
17.50Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
17.50Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
17.50Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
17.50Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
17.50Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
17.50Single8WDTphotoNECA8WDT-A2A-photoNECA
17.50Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.50Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
17.50Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
17.50Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
17.50Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
17.14Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
17.14Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
17.14Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
17.14Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
17.14Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
17.14Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
17.14Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
17.14Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
17.14Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
17.14Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
17.14Consensushca_on_gpOrthosteric Ligandhca2_on_gp
17.07Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
17.07Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
17.07Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
17.07Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
17.07Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
17.07Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
17.07Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
17.07Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
17.07Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
17.07Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
16.67Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
16.67Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
16.67Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
16.67Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
16.67Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
16.67Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
16.67Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
16.67Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
16.67Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
16.67Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
16.67Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
16.67Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
16.67Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
16.67Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
16.67Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
16.67Consensusa3_on_gpOrthosteric Liganda3a_on_gp
16.67Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
16.67Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
16.67Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
16.67Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
16.67Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
16.67Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
16.67Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
16.28Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
16.28Single6JODAngiotensin II6JOD-AT2-Angiotensin II
16.28Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
16.28Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
16.28Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
16.28Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
16.22Single2YDVNECA2YDV-A2A-NECA
16.22Single4UHRCGS216804UHR-A2A-CGS21680
16.22Single5G53NECA5G53-A2A-NECA-Gs
16.22Single5XRAAM115425XRA-CB1-AM11542
16.22Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
16.22Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
16.22Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
16.22Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
16.22Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
16.22Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
16.22Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
16.22Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
16.22Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
16.22Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
16.22Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
16.22Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
16.22Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
16.22Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
16.22Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
16.22Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
16.22Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
16.22Consensuslpa_onOrthosteric Ligandlpa1_on
16.22Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
16.22Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Consensusrelaxin_onOrthosteric Ligandrxfp4_on
16.22Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
16.22Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
16.22Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
16.22Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.22Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
16.13Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
15.91Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
15.91Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
15.91Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
15.91Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
15.91Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
15.91Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
15.91Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
15.91Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
15.91Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
15.91Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
15.91Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
15.79Single4XEENeurotensin4XEE-NTS1-Neurotensin
15.79Single4XESNeurotensin4XES-NTS1-Neurotensin
15.79Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
15.79Single6IIURamatroban6IIU-TXA2-Ramatroban
15.79Single6KQICP559406KQI-CB1-CP55940-Org27569
15.79Single6YVRNTS8-136YVR-NTS1-NTS8-13
15.79Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
15.79Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
15.79Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
15.79Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
15.79Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
15.79Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
15.79Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
15.79Single8XYIVUF106618XYI-CXCR3-VUF10661
15.79Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
15.79Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
15.79Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
15.79Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
15.79Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
15.79Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
15.79Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
15.79Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
15.79Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
15.79Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
15.79Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
15.79Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
15.79Consensuslpa_offOrthosteric Ligandlpa1_off
15.79Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
15.56Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.56Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
15.56Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
15.56Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
15.38Single4BUONeurotensin4BUO-NTS1-Neurotensin
15.38Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
15.38Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
15.38Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
15.38Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
15.38Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
15.38Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
15.38Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
15.38Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
15.38Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
15.38Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
15.38Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
15.38Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
15.38Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
15.38Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
15.38Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
15.38Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
15.38Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
15.38Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
15.38Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
15.38Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
15.38Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
15.38Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
15.38Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.38Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.38Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
15.38Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
15.38Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.22Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.22Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
15.22Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
15.22Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
15.22Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
15.22Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
15.15Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
15.15Single8K5BNiacin8K5B-HCA2-Niacin
15.15Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
15.00Single3NY9ICI118-5513NY9-β2-ICI118-551
15.00Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
15.00Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
15.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
15.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
15.00Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
15.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
15.00Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
15.00Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
15.00Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
15.00Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
15.00Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
15.00Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
15.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
15.00Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
14.89Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
14.89Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
14.71Single3PWHZM-2413853PWH-A2A-ZM-241385
14.71Single4BWBNeurotensin4BWB-NTS1-Neurotensin
14.71Single5U09Taranabant5U09-CB1-Taranabant
14.71Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
14.71Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
14.71Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.71Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
14.71Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
14.71Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
14.71Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
14.71Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
14.71Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
14.71Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
14.71Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
14.63Single4IARErgotamine4IAR-5-HT1B-Ergotamine
14.63Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
14.63Single7F8XNN90567F8X-CCKA-NN9056
14.63Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
14.63Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
14.63Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
14.63Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
14.63Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
14.63Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
14.63Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
14.63Single8XWNCXCL88XWN-CXCR2-CXCL8
14.63Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
14.63Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
14.63Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
14.63Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
14.63Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
14.63Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
14.63Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.58Single5GLHEndothelin-15GLH-ETB-Endothelin-1
14.58Single6IGKEndothelin-36IGK-ETB-Endothelin-3
14.58Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
14.58Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
14.58Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
14.29Single2YDOAdenosine2YDO-A2A-Adenosine
14.29Single3QAKUK-4320973QAK-A2A-UK-432097
14.29Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
14.29Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
14.29Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
14.29Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
14.29Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
14.29Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
14.29Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
14.29Single7XNACYN1548067XNA-SST2-CYN154806
14.29Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.29Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
14.29Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
14.29Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
14.29Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
14.29Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
14.29Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
14.29Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
14.29Single8K5CAcipimox8K5C-HCA2-Acipimox
14.29Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
14.29Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
14.29Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
14.29Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
14.29Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
14.29Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
14.29Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
14.29Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
14.29Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
14.29Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
14.29Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
14.29Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
14.29Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.29Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
14.29Consensushca_onOrthosteric Ligandhca2_on
14.29Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
14.29Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
14.29Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
14.29Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.29Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
14.29Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
14.00Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
14.00Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
13.95Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
13.95Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
13.95Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.95Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
13.95Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
13.95Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.95Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
13.95Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
13.95Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
13.95Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
13.95Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
13.95Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
13.95Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
13.95Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
13.89Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
13.89Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
13.89Single4YAYZD-71554YAY-AT1-ZD-7155
13.89Single5TGZAM65385TGZ-CB1-AM6538
13.89Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
13.89Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
13.89Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
13.89Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
13.89Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
13.89Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
13.89Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
13.89Single7V3ZCP559407V3Z-CB1-CP55940
13.89Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
13.89Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
13.89Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
13.89Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
13.89Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
13.89Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
13.89Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
13.89Single8K5DGSK2560738K5D-HCA2-GSK256073
13.89Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
13.89Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
13.89Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.89Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.89Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.89Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.89Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.89Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
13.89Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
13.89Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
13.89Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
13.89Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
13.89Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
13.89Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
13.89Consensusa3_onOrthosteric Liganda3a_on
13.89Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
13.89Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
13.89Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
13.89Consensusblt_onOrthosteric Ligandblt1_on
13.89Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
13.89Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
13.89Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
13.89Consensusleukotriene_onOrthosteric Ligandblt_on
13.89Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
13.89Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
13.89Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
13.79Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
13.64Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
13.64Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
13.64Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
13.64Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
13.64Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
13.64Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
13.64Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
13.64Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
13.64Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
13.51Single5C1MBU725C1M-μ-BU72
13.51Single5N2RPSB-365N2R-A2A-PSB-36-Na
13.51Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
13.51Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
13.51Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
13.51Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
13.51Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
13.51Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
13.51Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
13.51Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
13.51Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
13.51Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
13.51Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.51Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.51Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.51Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
13.51Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
13.51Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.51Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.51Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
13.51Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
13.51Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
13.51Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
13.51Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
13.51Single9B9ZA1AKO9B9Z-CB1-A1AKO
13.51Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
13.51Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
13.51Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
13.51Single9EHSLUF76029EHS-A3A-LUF7602
13.51Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
13.51Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
13.51Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
13.51Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
13.51Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
13.51Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
13.51Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
13.51Consensusep_offOrthosteric Ligandep4_off
13.51Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.51Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
13.51Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
13.51Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
13.51Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
13.51Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
13.51Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.51Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
13.51Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.51Consensustrace-amine_onOrthosteric Ligandta1_on
13.33Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
13.33Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
13.33Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
13.33Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
13.33Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
13.33Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
13.33Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
13.33Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
13.33Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
13.16Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
13.16Single4BV0Neurotensin4BV0-NTS1-Neurotensin
13.16Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
13.16Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
13.16Single4U15Tiotropium4U15-M3-Tiotropium
13.16Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
13.16Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
13.16Single5V54Methiothepin5V54-5-HT1B-Methiothepin
13.16Single5XR8AM8415XR8-CB1-AM841
13.16Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
13.16Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
13.16Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
13.16Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.16Single6OL9Tiotropium6OL9-M5-Tiotropium
13.16Single6OS1TRV0266OS1-AT1-TRV026
13.16Single7F1TMIP-1a7F1T-CCR5-MIP-1a
13.16Single7FEECP559407FEE-CB1-CP55940-ZCZ011
13.16Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
13.16Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
13.16Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
13.16Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
13.16Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
13.16Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
13.16Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
13.16Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
13.16Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
13.16Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
13.16Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
13.16Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.16Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
13.16Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
13.16Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
13.16Single8E0GBU728E0G-μ-BU72
13.16Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
13.16Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
13.16Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
13.16Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
13.16Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
13.16Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.16Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
13.16Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
13.16Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
13.16Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
13.16Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
13.16Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
13.16Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
13.16Consensus5ht1_offOrthosteric Ligand5ht1b_off
13.16Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
13.16Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
13.16Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
13.16Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
13.16Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
13.16Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
13.16Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
13.16Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
13.16Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
13.16Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
13.16Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.16Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.16Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
13.16Consensusneurotensin_onOrthosteric Ligandnts1_on
13.16Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.16Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
13.04Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
13.04Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
13.04Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
13.04Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
13.04Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
13.04Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
12.90Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.90Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
12.90Single8HS2Fab0468HS2-GPR20-Fab046
12.82Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
12.82Single3D4STimolol3D4S-β2-Timolol
12.82Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
12.82Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
12.82Single5CXVTiotropium5CXV-M1-Tiotropium
12.82Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
12.82Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
12.82Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
12.82Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
12.82Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
12.82Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
12.82Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
12.82Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
12.82Single7K15MKD0467K15-BLT1-MKD046-Na
12.82Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
12.82Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
12.82Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
12.82Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
12.82Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
12.82Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
12.82Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
12.82Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.82Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
12.82Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
12.82Single8JJ8Formoterol8JJ8-β2-Formoterol
12.82Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
12.82Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
12.82Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
12.82Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.82Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
12.82Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.82Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
12.82Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
12.82Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
12.82Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
12.82Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
12.82Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
12.82Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
12.82Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
12.82Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.82Consensuslpl_offOrthosteric Ligands1p_off lpa_off
12.82Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
12.82Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
12.82Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.82Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
12.82Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
12.77Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
12.77Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
12.77Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
12.77Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
12.77Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
12.77Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
12.77Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
12.77Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
12.50Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
12.50Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
12.50Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
12.50Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
12.50Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
12.50Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
12.50Single7EZCUKA7EZC-A2A-UKA
12.50Single7UM4AS26747237UM4-5-HT5A-AS2674723
12.50Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
12.50Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
12.50Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
12.50Single8A2OTheophylline8A2O-A2A-Theophylline-Na
12.50Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
12.50Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
12.50Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
12.50Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
12.50Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
12.50Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
12.50Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
12.50Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
12.50Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
12.50Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
12.50Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
12.50Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
12.50Consensuscck_onOrthosteric Ligandccka_on cckb_on
12.50Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
12.50Consensuschemerin_onOrthosteric Ligandcml1_on
12.50Consensusendothelin_onOrthosteric Ligandetb_on eta_on
12.50Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Consensusprostanoid_offOrthosteric Ligandep_off dp_off
12.24Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
12.24Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
12.24Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
12.24Consensusbombesin_onOrthosteric Ligandbb2_on
12.24Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
12.24Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
12.24Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
12.20Single5ZTYAM102575ZTY-CB2-AM10257
12.20Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
12.20Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
12.20Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
12.20Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
12.20Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
12.20Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
12.20Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
12.20Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
12.20Single7XN9L-054,5227XN9-SST2-L-054,522
12.20Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
12.20Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
12.20Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
12.20Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
12.20Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.20Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
12.20Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
12.20Single9IPYJR14a9IPY-C3aB-JR14a
12.20Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
12.20Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
12.20Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
12.12Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
12.12Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
12.12Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
12.12Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.12Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
12.12Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
12.12Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
12.12Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
12.12Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
12.12Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
12.12Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.12Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
12.00Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
12.00Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
11.90Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
11.90Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
11.90Single7QA8Peptide7QA8-STE2-Peptide
11.90Single7QA8Peptide7QA8-STE2-Peptide
11.90Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.90Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
11.90Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
11.90Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
11.90Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
11.90Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
11.90Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.90Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.90Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
11.90Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.90Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.90Consensussomatostatin_offOrthosteric Ligandsst2_off
11.76Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
11.76Single6LI0C176LI0-GPR52-C17
11.76Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.76Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
11.76Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
11.76Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
11.76Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
11.76Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
11.76Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
11.76Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
11.76Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
11.76Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
11.76Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
11.76Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
11.76Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
11.63Single6HLOAprepitant6HLO-NK1-Aprepitant
11.63Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
11.63Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
11.63Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
11.63Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
11.63Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.63Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
11.63Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
11.63Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
11.63Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
11.63Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
11.63Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
11.63Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
11.63Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
11.63Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
11.54Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
11.43Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
11.43Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
11.43Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
11.43Single5ZKQABT-4915ZKQ-PAF-ABT-491
11.43Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
11.43Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
11.43Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
11.43Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
11.43Single6ME9Ramelteon6ME9-MT2-Ramelteon
11.43Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
11.43Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
11.43Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
11.43Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
11.43Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
11.43Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
11.43Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
11.43Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
11.43Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.43Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
11.43Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
11.43Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
11.43Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
11.43Single8GNGIstradefylline8GNG-A2A-Istradefylline
11.43Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
11.43Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
11.43Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
11.43Single8IWESpermidine8IWE-TA9-Spermidine
11.43Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
11.43Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
11.43Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
11.43Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
11.43Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
11.43Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
11.43Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
11.43Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.43Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
11.43Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
11.43Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
11.43Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
11.43Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
11.43Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
11.43Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
11.43Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
11.43Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
11.43Consensusangiotensin_offOrthosteric Ligandat1_off
11.43Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.43Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
11.43Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
11.43Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
11.43Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
11.36Single3OE0CVX153OE0-CXCR4-CVX15
11.36Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
11.36Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.36Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
11.36Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
11.36Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
11.36Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
11.36Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
11.36Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.36Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.36Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.36Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
11.11Single3REYXAC3REY-A2A-XAC
11.11Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
11.11Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
11.11Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
11.11Single5IU7Q274563465IU7-A2A-Q27456346-Na
11.11Single5IUBQ274563445IUB-A2A-Q27456344-Na
11.11Single5JTBZM-2413855JTB-A2A-ZM-241385
11.11Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
11.11Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
11.11Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
11.11Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
11.11Single6AQFZM-2413856AQF-A2A-ZM-241385
11.11Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
11.11Single6KUXRS-799486KUX-α2a-RS-79948
11.11Single6MH8ZM-2413856MH8-A2A-ZM-241385
11.11Single6PS0S-Carazolol6PS0-β2-S-Carazolol
11.11Single6PS4ICI118-5516PS4-β2-ICI118-551
11.11Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
11.11Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
11.11Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
11.11Single7AROLUF58337ARO-A2A-LUF5833-Na
11.11Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
11.11Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
11.11Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
11.11Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
11.11Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
11.11Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
11.11Single7T32ZM-2413857T32-A2A-ZM-241385
11.11Single7UL3Famotidine7UL3-H2-Famotidine
11.11Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
11.11Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
11.11Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
11.11Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
11.11Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
11.11Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
11.11Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
11.11Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
11.11Single8K2WAMG4878K2W-CXCR3-AMG487
11.11Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
11.11Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
11.11Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
11.11Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
11.11Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
11.11Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
11.11Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
11.11Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
11.11Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
11.11Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
11.11Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
11.11Single8ZPMAMD0708ZPM-CXCR4-AMD070
11.11Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
11.11Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
11.11Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
11.11Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
11.11Consensusa2_offOrthosteric Liganda2a_off
11.11Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
11.11Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
11.11Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
11.11Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
11.11Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
10.87Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
10.87Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.87Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
10.87Single8ZRTET-18ZRT-ETB-ET-1
10.87Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
10.87Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
10.81Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
10.81Single2Y01Dobutamine2Y01-β1-Dobutamine
10.81Single2Y04Salbutamol2Y04-β1-Salbutamol
10.81Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
10.81Single3EMLZM-2413853EML-A2A-ZM-241385
10.81Single3NY8ICI118-5513NY8-β2-ICI118-551
10.81Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
10.81Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
10.81Single4GBRS-Carazolol4GBR-β2-S-Carazolol
10.81Single4QKX35V4QKX-β2-35V
10.81Single5IU8Q274563475IU8-A2A-Q27456347-Na
10.81Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
10.81Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
10.81Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
10.81Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
10.81Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
10.81Single5T04Neurotensin5T04-NTS1-Neurotensin
10.81Single5UENDU1725UEN-A1-DU172
10.81Single5UIGCmpd-15UIG-A2A-Cmpd-1
10.81Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
10.81Single6D27CAY104716D27-DP2-CAY10471
10.81Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
10.81Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
10.81Single6H7MSalbutamol6H7M-β1-Salbutamol
10.81Single6IIVDaltroban6IIV-TXA2-Daltroban
10.81Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
10.81Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
10.81Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
10.81Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
10.81Single6PS1Timolol6PS1-β2-Timolol
10.81Single6S0LZM-2413856S0L-A2A-ZM-241385
10.81Single6TOTLemborexant6TOT-OX1-Lemborexant
10.81Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.81Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
10.81Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
10.81Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
10.81Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
10.81Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
10.81Single7BU7BI1671077BU7-β1-BI167107
10.81Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
10.81Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
10.81Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
10.81Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
10.81Single7PYRPSB-21157PYR-A2A-PSB-2115
10.81Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
10.81Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
10.81Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
10.81Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
10.81Single7UL4Alvimopan7UL4-μ-Alvimopan
10.81Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
10.81Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
10.81Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
10.81Single8CU6LJ-45178CU6-A2A-LJ-4517
10.81Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
10.81Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
10.81Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
10.81Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
10.81Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
10.81Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.81Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.81Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.81Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.81Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.81Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.81Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.81Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.81Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.81Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.81Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
10.81Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
10.81Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
10.81Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
10.81Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
10.81Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
10.81Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.81Single8JXRLSD8JXR-D1-LSD
10.81Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
10.81Single8T1WCVN4248T1W-GPR6-CVN424
10.81Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
10.81Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.81Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.81Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
10.81Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
10.81Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
10.81Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
10.81Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
10.81Single9CHXS-Carazolol9CHX-β2-S-Carazolol
10.81Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
10.81Single9H37A1IR09H37-A2A-A1IR0-Na
10.81Single9IYAONO-97105319IYA-GPR55-ONO-9710531
10.81Single9JEAAtropine9JEA-M1-Atropine
10.81Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
10.81Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
10.81Consensus5ht5_onOrthosteric Ligand5ht5a_on
10.81Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
10.81Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
10.81Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
10.81Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.81Consensusdopamine_offOrthosteric Ligandd2_off d3_off
10.81Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
10.81Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
10.81Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
10.81Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
10.81Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
10.81Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
10.81Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
10.81Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
10.64Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
10.64Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
10.64Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
10.53Single2RH1S-Carazolol2RH1-β2-S-Carazolol
10.53Single2Y00Dobutamine2Y00-β1-Dobutamine
10.53Single2Y03Isoprenaline2Y03-β1-Isoprenaline
10.53Single2YCWS-Carazolol2YCW-β1-S-Carazolol
10.53Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
10.53Single5D6LS-Carazolol5D6L-β2-S-Carazolol
10.53Single5IUAQ274563485IUA-A2A-Q27456348-Na
10.53Single5JQHS-Carazolol5JQH-β2-S-Carazolol
10.53Single5N2SPSB365N2S-A1-PSB36
10.53Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
10.53Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
10.53Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
10.53Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
10.53Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
10.53Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
10.53Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
10.53Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
10.53Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
10.53Single6S0QZM-2413856S0Q-A2A-ZM-241385
10.53Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
10.53Single6TP6Filorexant6TP6-OX1-Filorexant
10.53Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
10.53Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
10.53Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
10.53Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
10.53Single7C61Ergotamine7C61-5-HT1B-Ergotamine
10.53Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
10.53Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
10.53Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
10.53Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
10.53Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
10.53Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
10.53Single7SINNPS-21437SIN-CaS-NPS-2143
10.53Single7SINNPS-21437SIN-CaS-NPS-2143
10.53Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
10.53Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
10.53Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
10.53Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
10.53Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
10.53Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
10.53Single8GNEKW-63568GNE-A2A-KW-6356-Na
10.53Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
10.53Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
10.53Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
10.53Single8S4DCMF-0198S4D-Apelin-CMF-019
10.53Single8TF5Oleic acid8TF5-GPR6-Oleic acid
10.53Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
10.53Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
10.53Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
10.53Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
10.53Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
10.53Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
10.53Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
10.53Single8ZMFA1L108ZMF-5-HT2C-A1L10
10.53Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
10.53Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
10.53Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
10.53Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
10.53Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
10.53Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
10.53Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
10.53Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
10.53Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
10.53Consensusadenosine_offOrthosteric Liganda1_off a2_off
10.53Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
10.53Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
10.53Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
10.53Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
10.53Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
10.53Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
10.53Consensusamine_offonOrthosteric Ligandamine_off amine_on
10.53Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
10.53Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
10.53Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
10.53Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
10.53Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
10.53Consensusblt_offOrthosteric Ligandblt1_off
10.53Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
10.53Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
10.53Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
10.53Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
10.53Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
10.53Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
10.53Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
10.53Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
10.42Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
10.42Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
10.26Single3P0GBI1671073P0G-β2-BI167107
10.26Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
10.26Single5D5AS-Carazolol5D5A-β2-S-Carazolol
10.26Single5D5BS-Carazolol5D5B-β2-S-Carazolol
10.26Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
10.26Single6H7JIsoprenaline6H7J-β1-Isoprenaline
10.26Single6J21Aprepitant6J21-NK1-Aprepitant
10.26Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
10.26Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
10.26Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
10.26Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
10.26Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
10.26Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
10.26Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
10.26Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
10.26Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
10.26Single7P2L4YI7P2L-mGlu5-4YI
10.26Single7PX4PSB-21137PX4-A2A-PSB-2113
10.26Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
10.26Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
10.26Single7TUYGSK682753A7TUY-GPR183-GSK682753A
10.26Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.26Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
10.26Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
10.26Single8EA0Iperoxo8EA0-M3-Iperoxo
10.26Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
10.26Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.26Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
10.26Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
10.26Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
10.26Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
10.26Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
10.26Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
10.26Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
10.26Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
10.26Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
10.26Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
10.26Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
10.26Single9BJKNaloxone9BJK-μ-Naloxone-NAM
10.26Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
10.26Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
10.26Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
10.26Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
10.26Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
10.26Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
10.26Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
10.26Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
10.26Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
10.20Single6IGLIRL16206IGL-ETB-IRL1620
10.20Single8IY6Endothelin-18IY6-ETB-Endothelin-1
10.20Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single4AMIBucindolol4AMI-β1-Bucindolol
10.00Single4LDEBI1671074LDE-β2-BI167107
10.00Single4N4WSANT-14N4W-SMO-SANT-1
10.00Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
10.00Single4RWADIPP-NH24RWA-δ-DIPP-NH2
10.00Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
10.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
10.00Single6A93Risperidone6A93-5-HT2A-Risperidone
10.00Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
10.00Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
10.00Single6MXTSalmeterol6MXT-β2-Salmeterol
10.00Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
10.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
10.00Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
10.00Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
10.00Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
10.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
10.00Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
10.00Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
10.00Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
10.00Single7YITNalfurafine7YIT-κ-Nalfurafine
10.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
10.00Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
10.00Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
10.00Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
10.00Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
10.00Single8JJLOlodaterol8JJL-β2-Olodaterol
10.00Single8JWY2-1188JWY-A2A-2-118
10.00Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
10.00Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
10.00Single8XQJJN2418XQJ-Apelin-JN241
10.00Single8XWACXCL18XWA-CXCR2-CXCL1
10.00Single8XWMCXCL68XWM-CXCR2-CXCL6
10.00Single8XWSCXCL58XWS-CXCR2-CXCL5
10.00Single9BJKNAM9BJK-μ-Naloxone-NAM
10.00Single9DGIZ85267113509DGI-CB1-Z8526711350
10.00Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
10.00Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
10.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
10.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
10.00Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
10.00Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
10.00Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
10.00Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
10.00Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
10.00Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
10.00Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
10.00Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
10.00Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
10.00Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
10.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
10.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
10.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
10.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
10.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
10.00Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
10.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
9.80Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
9.76Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
9.76Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
9.76Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
9.76Single6H7LDobutamine6H7L-β1-Dobutamine
9.76Single6IBLArformoterol6IBL-β1-Arformoterol
9.76Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
9.76Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
9.76Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
9.76Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
9.76Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
9.76Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
9.76Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
9.76Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.76Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
9.76Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
9.76Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
9.76Single8XVUCXCL28XVU-CXCR2-CXCL2
9.76Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
9.76Single8ZPLHF511168ZPL-CXCR4-HF51116
9.76Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
9.76Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
9.76Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.76Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
9.76Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
9.76Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
9.76Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
9.76Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
9.76Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
9.76Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
9.76Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
9.76Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
9.76Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Single6KNMJN241-96KNM-Apelin-JN241-9
9.52Single6PT3DPI-2876PT3-δ-DPI-287
9.52Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
9.52Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
9.52Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
9.52Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
9.52Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
9.52Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
9.52Single8QJ2pN1628QJ2-MC4-pN162-Gs
9.52Single8X5YAstemizole8X5Y-H1-Astemizole
9.52Single8XQJJN2418XQJ-Apelin-JN241
9.52Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
9.52Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
9.52Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
9.52Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
9.52Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
9.52Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
9.52Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
9.38Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
9.38Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
9.38Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
9.38Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
9.38Single8PWNTheophylline8PWN-A2A-Theophylline
9.38Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
9.30Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
9.30Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
9.30Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
9.30Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
9.30Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
9.30Single8KIGSHU91198KIG-MC3-SHU9119-Ca
9.30Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
9.30Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
9.30Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
9.30Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
9.30Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
9.30Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
9.30Single9M4TSilodosin9M4T-Alpha1A-Silodosin
9.30Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
9.30Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single3RFMCaffeine3RFM-A2A-Caffeine
9.09Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
9.09Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
9.09Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
9.09Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
9.09Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
9.09Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
9.09Single7SK5CXCL127SK5-ACKR3-CXCL12
9.09Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
9.09Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
9.09Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
9.09Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
9.09Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
9.09Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
9.09Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
9.09Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
9.09Consensusp2y_offOrthosteric Ligandp2y1_off
9.09Consensussensory_onOrthosteric Ligandopsins_on
9.09Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
8.89Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
8.89Single6PT2KGCHM076PT2-δ-KGCHM07
8.89Single6W25SHU91196W25-MC4-SHU9119-Ca
8.89Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
8.89Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
8.89Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.89Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
8.89Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
8.89Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
8.89Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
8.82Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
8.82Single3UZAGTPL92363UZA-A2A-GTPL9236
8.82Single4XNWMRS25004XNW-P2Y1-MRS2500
8.82Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
8.82Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
8.82Single6ME5Agomelatine6ME5-MT1-Agomelatine
8.82Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
8.82Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
8.82Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
8.82Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
8.82Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.82Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
8.82Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
8.82Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
8.82Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
8.82Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
8.82Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
8.82Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
8.82Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.82Single9LRCHistamine9LRC-H4-Histamine
8.82Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
8.82Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
8.82Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
8.82Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
8.70Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
8.70Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
8.70Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
8.70Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
8.70Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
8.70Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
8.70Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
8.70Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
8.70Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
8.70Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
8.70Consensusvasop-oxy_onOrthosteric Ligandv2_on
8.70Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
8.57Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
8.57Single3OE9IT1t3OE9-CXCR4-IT1t
8.57Single3PBLEticlopride3PBL-D3-Eticlopride
8.57Single4O9RCyclopamine4O9R-SMO-Cyclopamine
8.57Single5L7IVismodegib5L7I-SMO-Vismodegib
8.57Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
8.57Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
8.57Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
8.57Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
8.57Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
8.57Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
8.57Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
8.57Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
8.57Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
8.57Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
8.57Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
8.57Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
8.57Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
8.57Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
8.57Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
8.57Single9B9Y7DY9B9Y-CB1-7DY
8.57Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
8.57Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
8.57Consensusgq_nucleotideOrthosteric Ligandgq_p2y
8.57Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
8.57Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
8.51Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
8.51Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
8.51Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
8.51Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
8.33Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
8.33Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
8.33Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
8.33Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
8.33Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
8.33Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
8.33Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
8.33Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
8.33Single4QINSAG1.54QIN-SMO-SAG1.5
8.33Single4S0VSuvorexant4S0V-OX2-Suvorexant
8.33Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
8.33Single5WS3EMPA5WS3-OX2-EMPA
8.33Single6AKXA4R6AKX-CCR5-A4R
8.33Single6AKYMaraviroc6AKY-CCR5-Maraviroc
8.33Single6ME2Ramelteon6ME2-MT1-Ramelteon
8.33Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
8.33Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
8.33Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
8.33Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
8.33Single6TODEMPA6TOD-OX1-EMPA-Na
8.33Single6TPJSuvorexant6TPJ-OX2-Suvorexant
8.33Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
8.33Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
8.33Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
8.33Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
8.33Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
8.33Single7SK3CXCL127SK3-ACKR3-CXCL12
8.33Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
8.33Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
8.33Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
8.33Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
8.33Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
8.33Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
8.33Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
8.33Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
8.33Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
8.33Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
8.33Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
8.33Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
8.33Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
8.33Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.33Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
8.33Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
8.33Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
8.33Single8Y0HVUF114188Y0H-CXCR3-VUF11418
8.33Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
8.33Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
8.33Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
8.33Single9H2XA1IR19H2X-A2A-A1IR1-Na
8.33Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
8.33Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
8.33Consensusalpha2_offOrthosteric Ligandalpha2c_off
8.33Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.33Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.33Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
8.33Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
8.33Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
8.33Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
8.33Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
8.33Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
8.33Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
8.16Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
8.16Single9KDFRES-701-39KDF-ETB-RES-701-3
8.11Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
8.11Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
8.11Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
8.11Single4MBSMaraviroc4MBS-CCR5-Maraviroc
8.11Single4ZJCSB-6740424ZJC-OX1-SB-674042
8.11Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
8.11Single5UVIZM-2413855UVI-A2A-ZM-241385
8.11Single6FFIMMPEP6FFI-mGlu5-MMPEP
8.11Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
8.11Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
8.11Single6PS5S-Propranolol6PS5-β2-S-Propranolol
8.11Single6TP3Nemorexant6TP3-OX1-Nemorexant
8.11Single6TPGEMPA6TPG-OX2-EMPA
8.11Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
8.11Single6V9SGTPL114036V9S-OX1-GTPL11403
8.11Single6VI4JDTic6VI4-κ-JDTic
8.11Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
8.11Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
8.11Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
8.11Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
8.11Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
8.11Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
8.11Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
8.11Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
8.11Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.11Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
8.11Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
8.11Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
8.11Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
8.11Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
8.11Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
8.11Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
8.11Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
8.11Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
8.11Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.11Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
8.11Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.11Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
8.11Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
8.11Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
8.11Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
8.11Single8IHKAcifran8IHK-HCA3-Acifran
8.11Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
8.11Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
8.11Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
8.11Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
8.11Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.11Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
8.11Single8RLNLUF58348RLN-A2A-LUF5834
8.11Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.11Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.11Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
8.11Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.11Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
8.11Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
8.11Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
8.11Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
8.11Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
8.11Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
8.11Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
8.11Single8ZPNAMD31008ZPN-CXCR4-AMD3100
8.11Single9AS5Mescaline9AS5-5-HT2A-Mescaline
8.11Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
8.11Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
8.11Single9BA0A1AKN9BA0-CB1-A1AKN
8.11Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
8.11Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
8.11Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
8.11Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
8.11Consensusalpha1_onOrthosteric Ligandalpha1a_on
8.11Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
8.11Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
8.11Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
8.11Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
8.11Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
8.11Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
8.11Consensusopsins_offOrthosteric Ligandrhodopsin_off
8.11Consensussensory_offOrthosteric Ligandopsins_off
8.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
8.00Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
8.00Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
7.89Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
7.89Single2Y02Carmoterol2Y02-β1-Carmoterol
7.89Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
7.89Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
7.89Single4EJ4Naltrindole4EJ4-δ-Naltrindole
7.89Single4MQSIperoxo4MQS-M2-Iperoxo
7.89Single4QIMANTA XV4QIM-SMO-ANTA XV
7.89Single4U14Tiotropium4U14-M3-Tiotropium
7.89Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
7.89Single5DSGTiotropium5DSG-M4-Tiotropium
7.89Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
7.89Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
7.89Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
7.89Single6FFHFenobam6FFH-mGlu5-Fenobam
7.89Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
7.89Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
7.89Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
7.89Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
7.89Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
7.89Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
7.89Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
7.89Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
7.89Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
7.89Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
7.89Single7WC7Lisuride7WC7-5-HT2A-Lisuride
7.89Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.89Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
7.89Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
7.89Single7YXAONO-54306087YXA-S1P5-ONO-5430608
7.89Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
7.89Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
7.89Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.89Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
7.89Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
7.89Single8JJOAlprenolol8JJO-β2-Alprenolol
7.89Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
7.89Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
7.89Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
7.89Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
7.89Single8X64Desloratadine8X64-H1-Desloratadine
7.89Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
7.89Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
7.89Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
7.89Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
7.89Single9AS1DMT9AS1-5-HT2A-DMT
7.89Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
7.89Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
7.89Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
7.89Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
7.89Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
7.89Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
7.89Consensusalpha2_onOrthosteric Ligandalpha2b_on
7.89Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
7.89Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
7.89Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
7.89Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
7.89Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
7.89Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.89Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.89Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.89Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
7.89Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
7.84Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
7.69Single4JKVTaladegib4JKV-SMO-Taladegib
7.69Single4NTJAZD12834NTJ-P2Y12-AZD1283
7.69Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
7.69Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
7.69Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
7.69Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
7.69Single5TVNLSD5TVN-5-HT2B-LSD
7.69Single5WIUNemonapride5WIU-D4-Nemonapride
7.69Single5WIVNemonapride5WIV-D4-Nemonapride-Na
7.69Single5WQCEMPA5WQC-OX2-EMPA
7.69Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
7.69Single6D26Fevipiprant6D26-DP2-Fevipiprant
7.69Single6E67BI1671076E67-β2-BI167107-Gs(CT)
7.69Single6LUQHaloperidol6LUQ-D2-Haloperidol
7.69Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
7.69Single6PS6Timolol6PS6-β2-Timolol
7.69Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
7.69Single7C4SS1P7C4S-S1P3-S1P
7.69Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
7.69Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
7.69Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
7.69Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
7.69Single7W41PD1762527W41-BB2-PD176252
7.69Single7WC6LSD7WC6-5-HT2A-LSD
7.69Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
7.69Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
7.69Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
7.69Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
7.69Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
7.69Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
7.69Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
7.69Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
7.69Single8JXSPF-61428JXS-D1-PF-6142
7.69Single8QOTNanobody-E8QOT-μ-Nanobody-E
7.69Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
7.69Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
7.69Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
7.69Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
7.69Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
7.69Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
7.69Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.69Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
7.69Single9HAPTolvaptan9HAP-V2-Tolvaptan
7.69Single9HC04YI9HC0-mGlu5-4YI
7.69Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
7.69Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
7.69Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
7.69Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
7.69Consensusbombesin_offOrthosteric Ligandbb2_off
7.69Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
7.69Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
7.69Consensusdp_offOrthosteric Liganddp2_off
7.69Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
7.69Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
7.50Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
7.50Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
7.50Single4DJHJDTic4DJH-κ-JDTic
7.50Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
7.50Single5TZRMK86665TZR-FFA1-MK8666
7.50Single5V56TC1145V56-SMO-TC114
7.50Single5V57TC1145V57-SMO-TC114
7.50Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
7.50Single6WGTLSD6WGT-5-HT2A-LSD
7.50Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
7.50Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
7.50Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
7.50Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
7.50Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
7.50Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
7.50Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
7.50Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.50Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
7.50Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
7.50Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
7.50Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
7.50Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
7.50Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
7.50Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
7.50Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
7.50Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
7.50Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
7.50Single8XVLZibotentan8XVL-ETA-Zibotentan
7.50Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
7.50Single8ZWFJR14a8ZWF-C3aB-JR14a
7.50Single9AS9RS130-1809AS9-5-HT2A-RS130-180
7.50Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
7.50Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
7.50Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
7.50Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
7.50Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
7.50Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
7.50Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
7.50Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
7.50Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
7.50Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
7.50Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
7.50Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.50Consensustachykinin_offOrthosteric Ligandnk1_off
7.32Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
7.32Single4PY02MeSATP4PY0-P2Y12-2MeSATP
7.32Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
7.32Single5X33BIIL2605X33-BLT1-BIIL260
7.32Single6CM4Risperidone6CM4-D2-Risperidone
7.32Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
7.32Single6ZG4HTL00099366ZG4-M1-HTL0009936
7.32Single7DFPSpiperone7DFP-D2-Spiperone
7.32Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
7.32Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
7.32Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
7.32Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
7.32Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
7.32Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
7.32Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.32Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
7.32Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
7.32Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
7.32Single8JWZAB9288JWZ-A2A-AB928-Na
7.32Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.32Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
7.32Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
7.32Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
7.32Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
7.32Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
7.32Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
7.32Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.32Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
7.14Single5CGDHTL142425CGD-mGlu5-HTL14242
7.14Single5X93K-87945X93-ETB-K-8794
7.14Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
7.14Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
7.14Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
7.14Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
7.14Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
7.14Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
7.14Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
7.14Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
7.14Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
7.14Single8XVJMacitentan8XVJ-ETA-Macitentan
7.14Single8XWFCXCL38XWF-CXCR2-CXCL3
7.14Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
7.14Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
7.14Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
7.14Consensusendothelin_offOrthosteric Ligandetb_off
7.14Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
6.98Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.98Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
6.98Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
6.98Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.98Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.82Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
6.82Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
6.82Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
6.82Single8WKYPG-9348WKY-MC4-PG-934
6.82Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.82Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
6.67Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
6.67Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
6.52Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
6.52Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
6.52Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
6.52Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
6.52Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
6.25Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
6.25Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
6.25Single5MZPCaffeine5MZP-A2A-Caffeine-Na
6.25Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
6.06Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
6.06Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
6.06Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
6.06Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
5.88Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
5.88Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
5.88Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
5.88Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
5.88Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
5.71Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
5.71Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
5.71Single3OE6IT1t3OE6-CXCR4-IT1t
5.71Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.71Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
5.71Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
5.71Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
5.71Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.71Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.71Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
5.71Single8JPSCCL78JPS-ACKR1-CCL7
5.71Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
5.71Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
5.71Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.71Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.71Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.71Consensusgi_sensoryOrthosteric Ligandgi_opsins
5.71Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.71Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.56Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
5.56Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
5.56Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
5.56Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
5.56Single6HLLCP999946HLL-NK1-CP99994
5.56Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
5.56Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
5.56Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
5.56Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
5.56Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
5.56Single7SRQLSD7SRQ-5-HT2B-LSD
5.56Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
5.56Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
5.56Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
5.56Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
5.56Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
5.56Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
5.56Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
5.56Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
5.56Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
5.56Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
5.56Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
5.56Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.56Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
5.56Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
5.56Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.56Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
5.56Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
5.56Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
5.56Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
5.56Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
5.56Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
5.41Single3ODUIT1t3ODU-CXCR4-IT1t
5.41Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
5.41Single4XNVBPTU4XNV-P2Y1-BPTU
5.41Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
5.41Single6B73MP11046B73-κ-MP1104
5.41Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
5.41Single7BR3Elagolix7BR3-GnRH1-Elagolix
5.41Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
5.41Single7F8ULintitript7F8U-CCKA-Lintitript
5.41Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.41Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
5.41Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
5.41Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
5.41Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
5.41Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
5.41Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
5.41Single7XRRLemborexant7XRR-OX2-Lemborexant
5.41Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
5.41Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
5.41Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
5.41Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
5.41Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
5.41Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
5.41Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.41Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
5.41Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
5.41Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
5.41Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
5.41Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.41Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
5.41Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
5.41Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
5.41Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
5.41Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
5.41Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
5.41Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
5.41Consensusorexin_offOrthosteric Ligandox2_off ox1_off
5.41Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
5.41Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
5.41Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
5.26Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
5.26Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
5.26Single6A94Zotepine6A94-5-HT2A-Zotepine
5.26Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
5.26Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
5.26Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
5.26Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
5.26Single6ZG9GSK10347026ZG9-M1-GSK1034702
5.26Single6ZINSR486926ZIN-NTS1-SR48692
5.26Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
5.26Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
5.26Single7F61PF-036547467F61-H3-PF-03654746
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.26Single7VV6C48/807VV6-MRGPRX2-C48/80
5.26Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
5.26Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
5.26Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.26Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
5.26Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
5.26Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
5.26Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.26Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AS3LSD9AS3-5-HT2A-LSD
5.26Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
5.26Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
5.26Consensusgrh_offOrthosteric Ligandgnrh1_off
5.13Single4DAJTiotropium4DAJ-M3-Tiotropium
5.13Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
5.13Single5DHHSB-6121115DHH-NOP-SB-612111
5.13Single6DRXLisuride6DRX-5-HT2B-Lisuride
5.13Single6GPSMK08126GPS-CCR2-MK0812
5.13Single7F83PF-051904577F83-Ghrelin-PF-05190457
5.13Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
5.13Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
5.13Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
5.13Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
5.13Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
5.13Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
5.13Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
5.13Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
5.13Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
5.13Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
5.13Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
5.13Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
5.13Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
5.13Single8X63Mepyramine8X63-H1-Mepyramine
5.13Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
5.13Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
5.13Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
5.13Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
5.13Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
5.13Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
5.13Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
5.13Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
5.13Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
5.13Consensushistamine_offOrthosteric Ligandh1_off
5.00Single5CGCHTL142425CGC-mGlu5-HTL14242
5.00Single5XPRBosentan5XPR-ETB-Bosentan
5.00Single6GPXMK08126GPX-CCR2-MK0812
5.00Single6HLPNetupitant6HLP-NK1-Netupitant
5.00Single6Z4SSR486926Z4S-NTS1-SR48692
5.00Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
5.00Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.00Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
5.00Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
5.00Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
4.88Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
4.88Single6TQ7SB-3348676TQ7-OX1-SB-334867
4.88Single7B6WCyclazosin7B6W-α1b-Cyclazosin
4.88Single7R0CAVP7R0C-V2-AVP-Arrestin2
4.88Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
4.88Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
4.88Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.88Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
4.88Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
4.88Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
4.88Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
4.88Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
4.88Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
4.76Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
4.76Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
4.76Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.76Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
4.76Consensusorexin_onOrthosteric Ligandox2_on
4.76Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
4.65Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.65Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.65Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
4.65Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
4.65Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
4.55Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
4.55Single9JF4PD1683689JF4-BB1-PD168368
4.55Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
4.55Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
4.55Consensuskisspeptin_onOrthosteric Ligandkiss1_on
4.44Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.44Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
4.44Single8IEIA1LYA8IEI-GPR156-A1LYA
4.44Single8IEIA1LYA8IEI-GPR156-A1LYA
4.44Single8IEPA1LYA8IEP-GPR156-A1LYA
4.44Single8IEPA1LYA8IEP-GPR156-A1LYA
4.44Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
4.44Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
4.44Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
4.44Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
4.44Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
4.44Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
4.35Single8IEBA1LYA8IEB-GPR156-A1LYA
4.35Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
4.17Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
4.17Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
3.33Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
3.33Single6D35Cholesterol6D35-SMO-Cholesterol
3.33Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
3.33Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
3.33Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
3.33Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
3.33Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
3.33Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
3.33Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
3.33Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
3.33Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
3.33Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
3.33Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.33Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.33Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.33Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.33Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
3.33Single7DTTCa7DTT-CaS-Ca-Ca
3.33Single7DTTCa7DTT-CaS-Ca-Ca
3.33Single7DTUTryptophan7DTU-CaS-Tryptophan
3.33Single7DTUTryptophan7DTU-CaS-Tryptophan
3.33Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
3.33Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
3.33Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
3.33Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
3.33Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.33Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.33Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.33Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.33Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
3.33Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
3.33Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
3.33Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
3.33Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
3.33Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
3.33Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
3.33Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
3.33Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
3.33Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
3.33Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
3.33Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
3.33Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
3.33Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.33Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.33Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
3.33Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
3.33Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.33Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.33Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.33Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.33Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
3.33Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
3.33Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
3.33Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
3.33Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
3.33Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
3.33Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.33Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.33Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.33Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.33Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.33Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.33Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.33Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.33Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
3.33Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
3.33Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
3.33Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
3.33Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
3.33Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
3.33Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
3.33Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
3.33Single7XW7K1-707XW7-TSH-K1-70
3.33Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
3.33Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
3.33Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
3.33Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
3.33Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
3.33Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
3.33Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
3.33Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
3.33Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
3.33Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
3.33Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
3.33Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
3.33Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
3.33Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
3.33Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
3.33Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
3.33Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
3.33Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
3.33Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
3.33Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
3.33Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
3.33Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.33Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.33Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.33Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.33Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.33Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.33Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
3.33Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
3.33Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
3.33Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
3.33Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
3.33Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.33Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.33Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
3.33Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
3.33Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
3.33Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
3.33Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
3.33Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
3.33Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
3.33Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
3.33Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
3.33Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
3.33Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
3.33Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
3.33Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
3.33Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
3.33Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
3.33Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
3.33Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.33Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.33Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.33Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.33Single8WVXNorrin8WVX-LGR4-Norrin
3.33Single8WVYNorrin8WVY-LGR4-Norrin
3.33Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
3.33Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
3.33Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
3.33Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
3.33Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
3.33Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
3.33Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
3.33Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.33Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.33Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.33Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.33Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.33Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.33Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.33Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.33Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.33Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.33Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.33Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.33Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.33Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.33Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.33Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.33Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
3.33Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
3.33Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
3.33Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
3.33Single9KHHNorrin9KHH-LGR4-Norrin
3.33Single9S37NB219S37-LGR4-NB21
3.33Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
3.23Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.23Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.23Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.23Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.23Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.23Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.23Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.23Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.23Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.23Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.23Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.23Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.23Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.23Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.12Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
3.12Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
3.12Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
3.03Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
3.03Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
3.03Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
3.03Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
3.03Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.03Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
3.03Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
2.94Single5L7DCholesterol5L7D-SMO-Cholesterol
2.94Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
2.94Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
2.86Single3OE8IT1t3OE8-CXCR4-IT1t
2.86Single6TQ9SB-4081246TQ9-OX1-SB-408124
2.86Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
2.86Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
2.86Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
2.86Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
2.86Single9CHUNoradrenaline9CHU-β2-Noradrenaline
2.86Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
2.86Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
2.78Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
2.78Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
2.78Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
2.78Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
2.78Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
2.78Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
2.78Consensus5ht2_onOrthosteric Ligand5ht2b_on
2.78Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.78Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
2.70Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
2.70Single6TP4ACT-4622066TP4-OX1-ACT-462206
2.70Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
2.70Single7LD3MIPS5217LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
2.70Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.70Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
2.70Single7UL2SR486927UL2-NTS1-SR48692-Na
2.70Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
2.70Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
2.70Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
2.70Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.70Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
2.70Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
2.70Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
2.70Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
2.70Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
2.70Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
2.70Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
2.70Consensusneurotensin_offOrthosteric Ligandnts1_off
2.70Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
2.63Single4K5YCP-3763954K5Y-CRF1-CP-376395
2.63Single6C1QNDT95137276C1Q-C5a1-PMX53-NDT9513727
2.63Single6DS0Ly2660976DS0-5-HT2B-Ly266097
2.63Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
2.63Single7F8YDevazepide7F8Y-CCKA-Devazepide
2.63Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
2.63Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
2.63Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
2.63Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.63Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
2.63Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
2.63Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.63Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
2.63Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.63Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.63Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
2.63Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
2.63Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
2.63Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.56Single3RZECidoxepin3RZE-H1-Cidoxepin
2.56Single6IQLL7458706IQL-D4-L745870
2.56Single6TPNHTL66416TPN-OX2-HTL6641
2.56Single8IYXYL-3658IYX-GPR34-YL-365
2.56Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
2.56Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
2.56Single9ARXSerotonin9ARX-5-HT2A-Serotonin
2.56Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
2.56Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
2.56Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
2.56Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
2.50Single4Z9GCP-3763954Z9G-CRF1-CP-376395
2.50Single5DHGC-355DHG-NOP-C-35
2.50Single8GTIBMK-C2058GTI-CRF1-BMK-C205
2.50Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
2.50Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
2.50Consensuscck_offOrthosteric Ligandccka_off
2.50Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
2.44Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
2.44Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
2.44Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
2.44Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
2.44Single8GTGBMK-I1528GTG-CRF1-BMK-I152
2.44Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
2.38Single6J20Aprepitant6J20-NK1-Aprepitant
2.38Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
2.38Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
2.38Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
2.33Single8GTMBMK-C2038GTM-CRF1-BMK-C203
2.27Single6K1QIRL25006K1Q-ETB-IRL2500
2.27Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
2.17Single8IEBA1LYA8IEB-GPR156-A1LYA
2.17Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.17Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.08Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.08Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.04Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
1.92Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
6LMK 6LMK-Glucagon-Glucagon-Gs/β1/γ2
8JIT 8JIT-Glucagon-MEDI0382-Gs/β1/γ2
7V35 7V35-Glucagon-Peptide-20-Gs/β1/γ2
Net Summary
Imin 2.89333
Number of Linked Nodes 1009
Number of Links 1200
Number of Hubs 188
Number of Links mediated by Hubs 733
Number of Communities 28
Number of Nodes involved in Communities 224
Number of Links involved in Communities 323
Path Summary
Number Of Nodes in MetaPath 99
Number Of Links MetaPath 98
Number of Shortest Paths 5342878
Length Of Smallest Path 3
Average Path Length 44.4397
Length of Longest Path 69
Minimum Path Strength 0.511667
Average Path Strength 6.44494
Maximum Path Strength 22.3078
Minimum Path Correlation 0.7
Average Path Correlation 0.992084
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.75439
Average % Of Corr. Nodes 37.0347
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 59.3203
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
glucagon_on_gpglp_on_gp
gluc_on_gp
secretin_on_gp
gip_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download gluc_on_gp.zip



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