Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.34 2.01725404
2G.HN.37 3.43525403
3G.HN.40 6.78325427
4G.HN.43 3.48775409
5G.hns1.01 6.77254193
6G.S1.02 6.7075466
7G.H1.03 1.57425409
8G.H1.08 3.771509
9G.S3.03 5.40933668
10G.S3.04 7.03725457
11G.S3.05 5.425408
12G.S3.06 7.7124556
13G.H2.03 7.44425449
14G.H2.06 5.97717649
15G.H2.07 5.7365409
16G.S4.04 4.46867609
17G.H3.01 3.1882509
18G.H3.03 3.68825404
19G.H3.06 5.12125406
20G.H3.09 4.84383689
21G.H3.13 8.6476586
22G.H3.17 9.3394555
23G.S5.05 3.972676139
24G.s5hg.01 4.99625409
25G.HG.03 2.71525407
26G.hgh4.05 8.3944506
27G.hgh4.08 8.24725407
28G.hgh4.11 3.91675404
29G.hgh4.21 5.16825404
30G.H4.03 2.8055404
31G.H4.07 7.94325485
32G.H4.08 6.351483
33G.H4.10 10.5977406
34G.H4.12 5.5838585
35G.H4.15 6.1466508
36G.h4s6.02 3.9985488
37G.h4s6.08 3.108404
38G.h4s6.20 5.074254144
39G.S6.02 7.19185148
40G.S6.05 7.1114585
41G.s6h5.05 5.168254139
42G.H5.03 5.650754139
43G.H5.05 5.10725466
44G.H5.06 4.9864134
45G.H5.08 5.55429769
46G.H5.17 7.137836146
47G.H5.20 4.3195498
48G.H5.23 6.823404
49G.H5.25 3.522599
50b.1x4 2.1472508
51b.1x7 2.73925408
52b.h2x1 3.889405
53b.lhb1x6 4.65345113
54b.b1x6 7.6744529
55b.l1x3 7.61317629
56b.b2x1 5.77875458
57b.b2x5 6.4015627
58b.b3x2 5.1215425
59b.b3x3 4.27585168
60b.l3x1 6.18325459
61b.l3x2 7.220254199
62b.b4x3 3.5925407
63b.b4x6 7.75225829
64b.b4x7 7.5785428
65b.l4x2 9.79525424
66b.b5x3 6.92583629
67b.b5x7 5.66875407
68b.l5x1 4.037408
69b.l5x5 8.4035659
70b.b6x5 4.531254166
71b.l6x5 4.31254184
72b.b7x1 5.28965184
73b.b8x4 6.27975406
74b.l9x3 5.83817649
75b.l9x6 6.1845648
76b.b10x5 4.5798509
77b.l10x1 4.06225403
78b.b11x2 5.09775447
79b.b11x4 4.1782549
80b.b11x5 3.44925406
81b.l11x2 7.006549
82b.b12x6 8.72633648
83b.b13x7 6.605577
84b.l13x3 7.57833679
85b.l13x6 6.84549
86b.l13x7 5.39975479
87b.b15x1 5.90167679
88b.l15x1 5.1566547
89b.l15x2 5.3156579
90b.b16x4 7.2858576
91b.b16x6 8.54871778
92b.b16x7 8.12925439
93b.b17x5 6.2036537
94b.b17x7 8.057438
95b.l17x3 8.51143739
96b.l17x6 7.973549
97b.b18x3 4.6462538
98b.b18x5 6.029405
99b.l18x1 6.859717126
100b.l18x2 5.978754127
101b.l18x3 7.11065125
102b.b19x2 6.23133636
103b.b19x4 6.7855438
104b.l19x1 6.93175449
105b.l19x2 7.9604539
106b.b20x2 7.55025436
107b.b20x4 9.53883638
108b.b20x6 6.37243736
109b.b20x7 4.648409
110b.l20x2 6.20125409
111b.b21x1 6.7674537
112b.b21x5 5.77875404
113b.b21x7 5.4725605
114b.l21x2 7.466404
115b.l21x5 4.171254174
116b.l22x5 7.3895119
117b.b23x6 7.815676177
118b.l23x2 6.351754178
119b.b24x4 6.322254176
120b.b24x6 8.047254178
121b.l25x3 8.55345159
122b.l25x6 13.1062558
123b.l26x5 4.92225405
124b.l27x1 11.5793659
125b.b28x3 5.27925427
126b.b28x4 6.70954156
127b.b28x6 8.53865159
128g.h1x11 2.89875409
129g.h1x12 2.08775406
130g.l1x4 5.928438
131g.h2x9 1.879404
132g.h2x11 7.7614126
133g.ctx3 6.43185119
134g.ctx5 4.355754119
135g.ctx6 3.18185116
136g.ctx15 7.10675429
137g.ctx16 4.55138828
138NT 186.978715
1391x39 5.8735417
1401x43 6.2654517
1411x47 3.137407
1421x50 4.668409
1431x60 4.724676227
1442x38 3.5002567
1452x39 6.4134509
1462x45 7.8814108
1472x50 6.6275608
1482x53 7.0316518
1492x60 6.921417
1503x26 8.75125408
1513x32 8.7275417
1523x33 5.95025417
1533x34 5.72845109
1543x35 7.0035105
1553x38 4.84425108
1563x40 7.889517
1573x41 5.21685106
1583x42 9.11865109
1593x44 4.7865408
1603x46 8.022409
1613x49 7.3142568
1623x51 9.68425498
1633x53 7.3135468
164I2 6.768381367
1654x50 7.164109
1664x52 3.66954104
1674x53 3.80645109
1684x56 5.466254105
1694x60 6.5728518
1704x64 8.47375418
171E2 7.70833616
172E2x51 10.3073618
173E2x52 5.31025415
1745x41 6.6906517
1755x44 7.30275417
1765x58 8.7055499
1776x30 1.33725407
1786x40 5.05975499
1796x44 6.565699
1806x47 8.983418
1816x48 9.85417618
1826x51 4.899617
183E3 4.974815
1847x33 5.93325416
1857x37 6.59775417
1867x41 5.578416
1877x43 4.8396517
188Lig 14.44773510
189G.H1.11 0.88925400
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.l26x5 g.ctx15 11.38196.877YesYes059
2b.l26x5 g.ctx4 1003.019YesNo057
3g.ctx3 g.ctx4 99.94385.635YesNo097
4g.ctx3 g.ctx5 59.613.528YesYes1199
5b.lhb1x11 g.ctx5 58.46125.511NoYes049
6b.b25x7 b.lhb1x11 75.0275.792NoNo074
7b.b25x7 b.b28x6 74.051219.019NoYes079
8b.b28x4 b.b28x6 72.78424.988YesYes1569
9b.b1x5 b.b28x4 72.47156.905NoYes036
10b.b1x5 b.l1x1 72.3749.186NoNo037
11I1x48 b.l1x1 72.55529.699NoNo087
12I1x48 I1x51 72.45664.287NoNo088
132x41 I1x51 72.35783.484NoNo078
142x41 4x43 39.75564.1NoNo076
152x38 4x43 39.62374.423YesNo076
162x38 I2 25.66233.805YesYes677
17b.b2x5 b.l26x1 88.850110.798YesNo277
18b.l26x1 b.l26x3 88.73176.504NoNo277
19b.l26x3 b.l26x5 88.80475.684NoYes075
20G.S3.03 I2 15.13013.644YesYes687
21G.S2.06 G.S3.03 14.862511.041NoYes098
22G.H1.08 G.S2.06 14.68453.734YesNo099
23G.H1.08 G.H5.07 11.79264.092YesNo099
24G.H5.07 G.S5.05 11.61223.1NoYes099
25G.h2s4.01 b.l5x5 58.474312.427NoYes099
26G.S1.05 G.h2s4.01 57.903217.417NoNo099
27G.S1.05 G.S1.07 56.05573.181NoNo099
28G.S1.07 G.S4.04 55.79134.994NoYes099
29b.b26x2 b.b2x3 90.96944.86NoNo076
30b.b26x1 b.b26x2 90.97132.924NoNo097
31b.b26x1 b.l27x1 90.97375.931NoYes099
32b.b2x1 b.l27x1 71.156.753YesYes589
33b.b2x1 b.b6x1 31.85186.583YesNo089
34b.b6x1 b.l9x6 31.72584.909NoYes098
35G.H2.04 G.H2.07 20.5527.4NoYes099
36G.H2.04 G.H3.08 20.4649.443NoNo099
37G.H2.10 b.b2x1 19.68154.031NoYes588
38G.H2.10 b.l5x5 19.60373.133NoYes589
39b.l1x6 b.l27x1 19.744426.572NoYes599
40G.S4.04 G.S4.06 16.85333.537YesNo097
41G.H3.09 G.S4.04 31.13625.036YesYes099
42G.S4.04 G.S5.04 27.49412.924YesNo099
43G.H4.15 G.S4.06 16.1294.193YesNo087
44G.H3.09 G.H4.15 16.1786.322YesYes098
45G.H4.15 G.S5.04 16.12629.623YesNo089
46G.H4.15 G.S5.06 23.19073.166YesNo089
47G.H3.03 G.H3.06 11.78774.123YesYes046
48G.H3.06 G.H4.15 24.20037.429YesYes068
49G.H3.06 G.H4.14 19.01734.509YesNo066
50G.S5.04 G.S6.03 11.01832.952NoNo094
51G.S5.06 G.S6.05 18.78274.505NoYes095
52G.H4.12 G.S6.03 10.28375.472YesNo854
53G.H4.07 G.S6.05 22.152713.153YesYes855
54G.H4.03 G.H4.07 10.3431.976YesYes045
55G.H4.10 G.hgh4.05 10.212313.505YesYes066
56G.H4.10 G.H4.14 11.66036.648YesNo066
57G.H4.07 G.hgh4.20 10.3437.56YesNo053
583x53 I2 11.77663.724YesYes687
593x49 3x53 11.26969.496YesYes688
602x38 3x49 13.54324.995YesYes678
61G.H5.23 G.H5.25 15.15552.928YesYes049
623x53 G.H5.23 22.11253.05YesYes084
632x49 3x39 28.3845.662NoNo098
642x49 3x42 28.04774.696NoYes099
652x45 3x42 27.30814.707YesYes1089
662x41 2x45 33.31978.165NoYes078
67g.ctx3 g.ctx6 41.36994.886YesYes1196
68b.l22x5 g.ctx6 39.92814.13YesYes1196
69b.l22x5 b.lhb1x3 28.30314.26YesNo092
70b.h2x5 b.lhb1x3 27.47743.192NoNo052
71b.h2x1 b.h2x5 54.593.832YesNo055
72b.b21x4 b.h2x1 35.40143.185NoYes055
73b.b20x7 b.b21x4 34.83257.465YesNo095
74b.b20x7 b.l20x2 33.93433.097YesYes099
75b.l18x5 b.l20x2 32.43526.267NoYes029
76b.l18x3 b.l18x5 32.137611.169YesNo052
77b.l18x3 b.l18x4 29.81912.883YesNo057
78b.b18x5 b.l18x4 29.51593.011YesNo057
79b.b15x2 b.b18x5 28.30178.39NoYes065
80b.b15x2 b.b19x2 24.57267.869NoYes366
81b.b17x7 b.b19x2 15.87518.787YesYes386
82b.b17x7 b.b21x1 15.013.464YesYes387
83b.1x19 b.b21x1 12.56597.743NoYes067
84b.1x15 b.1x19 11.00625.636NoNo076
85b.1x15 g.h1x11 10.38121.714NoYes079
86b.l22x5 b.l24x2 27.54178.747YesNo096
87b.h2x5 b.l24x2 27.40414.866NoNo056
88b.b21x5 b.h2x1 18.626.644YesYes045
89b.lhb1x11 b.lhb1x9 17.10152.92NoNo043
90b.lhb1x6 b.lhb1x9 17.07223.378YesNo033
91b.l3x1 b.l5x5 39.22118.323YesYes599
92b.l1x6 b.l3x1 19.7187.456NoYes599
93b.b2x1 b.l3x1 19.69425.748YesYes589
94b.l11x1 b.l9x6 13.94295.647NoYes498
95b.b11x6 b.l11x1 13.95633.525NoNo499
96b.b11x6 b.l9x3 13.41213.248NoYes499
97b.b11x4 b.l9x3 12.21492.877YesYes499
98b.b21x5 b.b21x7 16.26910.776YesYes045
992x53 3x39 23.05710.485YesNo088
1002x53 Lig 19.10645.985YesYes180
101b.b2x3 b.b2x5 89.97556.746NoYes267
102G.H3.08 G.S4.04 20.38176.43NoYes099
103G.H2.07 b.l9x6 21.22156.173YesYes098
104b.l22x5 b.lhb1x6 16.42387.065YesYes1193
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
LigNT115.411YesYes0501
NTNT584.4741YesYes5511
1x21NT3.7531NoYes3511
1x28E33.1451NoYes3511
1x28Lig6.1371NoYes3010
1x291x333.2161NoNo3212
1x29Lig5.2471NoYes3010
1x32Lig19.5540NoYes6010
1x357x343.1110NoNo5621
1x357x384.3250NoNo5621
1x391x434.8631YesYes7721
1x392x616.8991YesNo7822
1x397x384.0441YesNo7621
1x432x537.9211YesYes7811
1x432x578.5821YesNo7711
1x437x423.8181YesNo7912
1x43Lig6.1431YesYes7010
2x533x365.831YesNo8611
2x533x3910.4851YesNo8812
2x533x404.9371YesYes8711
2x53Lig5.9851YesYes8010
2x573x323.0141NoYes7711
2x57Lig3.8931NoYes7010
2x60Lig9.7781YesYes7010
2x64E2x524.0031NoYes5511
2x64Lig4.1871NoYes5010
3x26E26.2580YesYes8621
3x29Lig2.8710NoYes6010
3x323x334.3211YesYes7711
3x32Lig15.1681YesYes7010
3x334x607.4131YesYes7812
3x335x437.0851YesNo7711
3x363x407.8541NoYes6711
3x36Lig6.0691NoYes6010
3x405x477.2561YesNo7711
3x406x4815.7881YesYes7812
3x40Lig3.611YesYes7010
4x604x646.41YesYes8822
4x605x438.5681YesNo8721
E2x50E2x523.2330NoYes9521
E2x52Lig10.1031YesYes5010
E2Lig16.7361YesYes6010
5x40E23.5190NoYes3621
5x415x427.1921YesNo7812
5x41E37.2851YesYes7511
5x41Lig8.3581YesYes7010
5x425x447.451NoYes8721
5x43Lig10.1091NoYes7010
5x44E33.2691YesYes7511
5x44Lig10.4891YesYes7010
5x47Lig4.8521NoYes7010
6x476x4818.4021YesYes8822
6x477x414.4631YesYes8621
6x487x419.5351YesYes8621
6x516x543.2041YesNo7522
6x517x337.4951YesYes7621
6x517x374.7821YesYes7721
6x54E34.3361NoYes5521
6x547x334.2531NoYes5621
E3Lig14.4191YesYes5010
7x30E34.8861NoYes5511
7x307x349.771NoNo5611
7x30Lig8.6451NoYes5010
7x337x378.961YesYes6711
7x33Lig3.0251YesYes6010
7x34Lig8.8261NoYes6010
7x377x414.8631YesYes7611
7x37Lig7.7861YesYes7010
7x38Lig8.1731NoYes6010
7x41Lig3.4511YesYes6010
3x33Lig4.9821YesYes7010
2x65Lig8.4161NoYes4010
1x25Lig5.0460NoYes1010
2x602x613.7331YesNo7812
2x603x3212.4071YesYes7711
2x642x652.9311NoNo5411
4x64E25.0981YesYes8621
E2E2x523.9021YesYes6511
5x48Lig2.9781NoYes4010
1x21Lig6.9591NoYes3010
5x415x448.0031YesYes7711
E2NT10.7371YesYes6511
E1NT8.1550NoYes4521
5x385x412.6150NoYes6721
1x261x292.4960NoNo3321
5x486x522.121NoNo4612
2x68Lig2.050NoYes0010
7x29E31.9160NoYes4521
1x22NT1.8430NoYes3521
2x603x281.7661YesNo7612
1x241x281.5860NoNo3321
2x622x650.5650NoNo4421
7x27E30.5360NoYes5521
1x23Lig0.5170NoYes1010

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
87.88Consensuspth_onOrthosteric Ligandpth1_on pth2_on
79.41Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
77.78Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
74.29Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
73.53Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
71.43Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
69.44Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
68.57Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
67.65Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
67.65Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
67.65Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
66.67Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
65.85Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
64.71Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
62.86Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
62.86Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
61.76Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
61.76Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
61.11Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
61.11Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
60.61Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
60.53Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
60.00Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
59.46Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
58.33Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
58.33Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
58.33Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
57.89Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
57.58Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
56.10Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
55.56Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
54.05Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
54.05Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
54.05Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
53.85Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
52.78Single6FJ3PTH6FJ3-PTH1-PTH
52.78Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
52.78Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
52.78Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
52.78Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
52.78Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
52.78Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
51.43Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
51.35Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
51.35Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
51.35Consensusglp_onOrthosteric Ligandglp1_on glp2_on
51.35Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
51.22Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
50.00Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
50.00Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
50.00Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
50.00Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
50.00Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
50.00Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
48.78Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
48.65Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
48.65Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
48.65Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
48.65Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
48.57Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
47.62Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
47.37Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
47.37Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
47.22Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
47.22Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
46.15Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
46.15Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
45.95Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
45.95Consensuspac_onOrthosteric Ligandpac1_on
45.95Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
45.71Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
45.24Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
45.00Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
44.74Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
44.74Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
44.44Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
44.44Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
43.59Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
43.59Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
43.59Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
43.24Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
43.24Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
43.24Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
43.24Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
42.86Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
42.50Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
42.50Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
42.11Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
41.86Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
41.86Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
41.67Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
41.46Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
41.18Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
41.03Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
40.54Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
40.48Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
40.00Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
40.00Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
39.53Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
39.53Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
39.53Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
39.47Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
39.47Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
39.02Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
38.89Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
38.64Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
38.46Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
37.50Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
37.21Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
37.21Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
36.84Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
36.59Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
36.59Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
35.90Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
35.71Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
35.71Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
35.14Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
35.00Consensuscalcitonin_onOrthosteric Ligandctlike_on
34.88Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
34.29Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
34.29Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
34.29Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
34.15Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
34.15Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
34.15Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
34.09Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
33.33Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
33.33Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
33.33Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
33.33Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
33.33Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
33.33Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
33.33Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
33.33Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
33.33Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
33.33Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
33.33Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
32.65Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
32.61Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
32.56Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
32.56Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
32.56Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
32.50Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
32.50Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
32.50Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
32.43Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
32.43Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
32.43Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
32.35Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
32.35Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
32.35Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
31.58Single4XT1Fractalkine4XT1-US28-Fractalkine
31.58Single7QA8Peptide7QA8-STE2-Peptide
31.58Single7QA8Peptide7QA8-STE2-Peptide
31.58Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
31.43Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
31.43Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
31.43Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
31.43Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
31.43Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
30.95Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
30.95Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
30.77Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
30.56Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
30.56Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
30.56Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
30.56Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
30.56Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
30.56Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
30.43Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
30.30Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
30.23Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
30.00Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
29.73Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
29.73Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
29.55Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
29.55Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
29.41Single7V3ZCP559407V3Z-CB1-CP55940
29.41Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
29.27Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
29.27Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
29.27Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
29.27Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
29.27Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
28.95Single4UG2CGS216804UG2-A2A-CGS21680
28.95Single5ZTYAM102575ZTY-CB2-AM10257
28.95Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
28.89Single6IGKEndothelin-36IGK-ETB-Endothelin-3
28.57Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
28.57Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
28.57Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
28.57Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
28.57Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
28.57Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
28.57Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
28.57Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
28.57Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.21Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
28.21Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
28.21Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
27.91Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
27.91Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
27.91Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
27.91Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
27.91Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
27.91Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
27.91Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
27.78Single5XR8AM8415XR8-CB1-AM841
27.78Single5XRAAM115425XRA-CB1-AM11542
27.78Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
27.78Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
27.50Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
27.50Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
27.50Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
27.27Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
27.27Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
27.27Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
27.27Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
27.27Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
27.27Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
27.03Single6KQICP559406KQI-CB1-CP55940-Org27569
27.03Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
27.03Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
27.03Single9DGIZ85267113509DGI-CB1-Z8526711350
27.03Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
27.03Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
27.03Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
26.83Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
26.83Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
26.83Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
26.83Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
26.67Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
26.67Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
26.47Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
26.47Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
26.32Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
26.32Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
26.32Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
26.19Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
26.19Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.19Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
26.09Single5GLHEndothelin-15GLH-ETB-Endothelin-1
26.09Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
26.09Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
26.09Consensusbombesin_onOrthosteric Ligandbb2_on
26.09Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
26.09Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
26.09Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.09Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
26.09Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
26.09Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
26.00Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
25.71Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
25.71Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
25.71Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
25.64Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
25.64Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
25.64Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
25.64Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
25.64Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
25.64Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
25.58Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
25.58Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
25.58Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
25.58Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
25.58Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
25.58Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
25.58Single8ZRTET-18ZRT-ETB-ET-1
25.58Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
25.58Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
25.58Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
25.58Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
25.00Single4XT3Fractalkine4XT3-US28-Fractalkine
25.00Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
25.00Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
25.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
25.00Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
25.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
25.00Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
25.00Single8TF5Oleic acid8TF5-GPR6-Oleic acid
25.00Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
25.00Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
25.00Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
25.00Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
25.00Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
25.00Consensuslpl_onOrthosteric Ligands1p_on lpa_on
25.00Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
25.00Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
25.00Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
25.00Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
24.44Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
24.44Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
24.44Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
24.44Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
24.44Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
24.44Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
24.44Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
24.44Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
24.44Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
24.39Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
24.39Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
24.39Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
24.39Single7XNACYN1548067XNA-SST2-CYN154806
24.39Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
24.39Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
24.39Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
24.39Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
24.39Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
24.32Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
24.32Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
24.32Single7FEECP559407FEE-CB1-CP55940-ZCZ011
24.32Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
24.32Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
24.32Single8E0GBU728E0G-μ-BU72
24.32Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
24.32Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
24.32Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
24.32Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
24.00Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
23.91Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
23.91Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
23.81Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
23.81Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
23.81Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
23.81Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
23.81Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
23.81Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.81Consensusangiotensin_onOrthosteric Ligandat1_on
23.81Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
23.81Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
23.81Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
23.81Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
23.81Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
23.81Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
23.68Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
23.68Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
23.68Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
23.68Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
23.68Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
23.68Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
23.68Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
23.68Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.68Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
23.68Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
23.68Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
23.68Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
23.68Consensuslpl_offOrthosteric Ligands1p_off lpa_off
23.68Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.68Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
23.53Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
23.53Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
23.40Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
23.40Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
23.40Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
23.26Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
23.26Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
23.26Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
23.26Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
23.26Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
23.26Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
23.26Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
23.26Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
23.26Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
23.26Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
23.26Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
23.26Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
23.26Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
23.26Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
23.26Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
23.26Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
23.26Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
23.26Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
23.26Consensusvasop-oxy_onOrthosteric Ligandv2_on
23.26Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
23.08Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
23.08Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
23.08Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
23.08Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
23.08Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
23.08Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
23.08Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
23.08Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
23.08Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
23.08Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
23.08Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
22.92Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
22.92Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
22.92Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
22.86Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
22.86Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
22.86Single8K5CAcipimox8K5C-HCA2-Acipimox
22.86Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
22.86Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
22.86Consensushca_onOrthosteric Ligandhca2_on
22.73Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
22.73Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
22.73Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
22.73Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
22.73Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
22.73Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
22.73Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
22.73Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
22.73Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
22.50Single3NY9ICI118-5513NY9-β2-ICI118-551
22.50Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
22.50Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
22.50Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
22.50Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
22.50Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
22.50Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
22.50Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
22.50Single8QJ2pN1628QJ2-MC4-pN162-Gs
22.50Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
22.50Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
22.50Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
22.50Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.50Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.45Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
22.22Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
22.22Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
22.22Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
22.22Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
22.22Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
22.22Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
22.22Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
22.22Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
22.22Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
22.22Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
22.22Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
22.22Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
22.22Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
22.22Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
22.22Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
22.22Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
22.22Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
22.22Consensushca_on_gpOrthosteric Ligandhca2_on_gp
22.22Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
22.00Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
21.95Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
21.95Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
21.95Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
21.95Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
21.95Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
21.95Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
21.95Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
21.95Single8WDTphotoNECA8WDT-A2A-photoNECA
21.95Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
21.95Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.95Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
21.95Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
21.95Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
21.95Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
21.95Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.95Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.95Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
21.95Consensussomatostatin_offOrthosteric Ligandsst2_off
21.95Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.74Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
21.74Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
21.62Single5C1MBU725C1M-μ-BU72
21.62Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
21.62Single7C4SS1P7C4S-S1P3-S1P
21.62Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
21.62Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
21.62Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
21.62Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
21.62Single8JXSPF-61428JXS-D1-PF-6142
21.62Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
21.62Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
21.62Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
21.62Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
21.62Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
21.43Single3QAKUK-4320973QAK-A2A-UK-432097
21.43Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
21.43Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
21.43Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
21.43Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
21.43Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
21.43Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
21.43Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
21.43Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
21.43Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
21.43Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
21.43Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
21.43Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
21.28Single6IGLIRL16206IGL-ETB-IRL1620
21.28Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
21.28Single8IY6Endothelin-18IY6-ETB-Endothelin-1
21.28Consensusendothelin_onOrthosteric Ligandetb_on eta_on
21.28Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
21.21Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.05Single2YDVNECA2YDV-A2A-NECA
21.05Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
21.05Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
21.05Single4UHRCGS216804UHR-A2A-CGS21680
21.05Single5G53NECA5G53-A2A-NECA-Gs
21.05Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
21.05Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
21.05Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
21.05Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
21.05Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
21.05Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
21.05Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
21.05Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
21.05Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
21.05Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
21.05Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
21.05Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
21.05Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.05Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
21.05Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
21.05Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
21.05Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
21.05Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
21.05Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
21.05Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
21.05Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
21.05Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
21.05Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.05Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
21.05Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
21.05Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
20.93Single5WF5UK-4320975WF5-A2A-UK-432097
20.93Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
20.93Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
20.93Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
20.93Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
20.93Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.93Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
20.93Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
20.93Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
20.93Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
20.59Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
20.59Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
20.59Single8K5BNiacin8K5B-HCA2-Niacin
20.59Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
20.51Single4XEENeurotensin4XEE-NTS1-Neurotensin
20.51Single4XESNeurotensin4XES-NTS1-Neurotensin
20.51Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
20.51Single6YVRNTS8-136YVR-NTS1-NTS8-13
20.51Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
20.51Single7DFPSpiperone7DFP-D2-Spiperone
20.51Single7K15MKD0467K15-BLT1-MKD046-Na
20.51Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
20.51Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
20.51Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
20.51Single7YITNalfurafine7YIT-κ-Nalfurafine
20.51Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
20.51Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
20.51Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
20.51Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
20.51Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
20.51Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
20.51Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
20.51Single8XYIVUF106618XYI-CXCR3-VUF10661
20.51Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
20.51Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
20.51Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
20.51Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
20.51Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
20.51Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
20.51Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
20.51Consensuslpa_offOrthosteric Ligandlpa1_off
20.51Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
20.51Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
20.51Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
20.51Consensusorexin_onOrthosteric Ligandox2_on
20.45Single6JODAngiotensin II6JOD-AT2-Angiotensin II
20.45Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
20.45Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
20.45Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
20.45Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
20.45Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
20.45Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
20.45Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
20.45Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
20.45Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
20.41Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
20.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
20.00Single4BUONeurotensin4BUO-NTS1-Neurotensin
20.00Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
20.00Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
20.00Single5U09Taranabant5U09-CB1-Taranabant
20.00Single5X93K-87945X93-ETB-K-8794
20.00Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
20.00Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
20.00Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
20.00Single7UM4AS26747237UM4-5-HT5A-AS2674723
20.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
20.00Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
20.00Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
20.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
20.00Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
20.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
20.00Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
20.00Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
20.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
20.00Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
20.00Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
20.00Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
20.00Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
20.00Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
20.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
20.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
20.00Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
20.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
20.00Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
20.00Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
20.00Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
20.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
20.00Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
20.00Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
20.00Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
20.00Consensuscck_onOrthosteric Ligandccka_on cckb_on
20.00Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
20.00Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
20.00Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
20.00Consensusendothelin_offOrthosteric Ligandetb_off
20.00Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
20.00Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
20.00Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
20.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
20.00Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
20.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
20.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.57Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
19.57Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
19.57Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
19.57Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
19.51Single5WF6UK-4320975WF6-A2A-UK-432097
19.51Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
19.51Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
19.51Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
19.51Single7SK9CCX6627SK9-ACKR3-CCX662
19.51Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
19.51Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
19.51Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
19.51Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
19.51Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
19.51Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
19.51Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.51Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
19.51Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
19.44Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.44Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
19.44Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
19.44Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
19.44Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
19.44Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
19.44Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
19.44Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
19.44Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.44Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
19.44Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
19.44Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
19.05Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
19.05Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
19.05Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
19.05Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
19.05Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
19.05Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
19.05Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
19.05Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
19.05Single8IEIA1LYA8IEI-GPR156-A1LYA
19.05Single8IEPA1LYA8IEP-GPR156-A1LYA
19.05Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.05Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
19.05Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
19.05Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
19.05Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
19.05Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
19.05Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
18.92Single2Y04Salbutamol2Y04-β1-Salbutamol
18.92Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
18.92Single4YAYZD-71554YAY-AT1-ZD-7155
18.92Single5TGZAM65385TGZ-CB1-AM6538
18.92Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
18.92Single6TOTLemborexant6TOT-OX1-Lemborexant
18.92Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
18.92Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
18.92Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
18.92Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
18.92Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
18.92Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
18.92Single7UL4Alvimopan7UL4-μ-Alvimopan
18.92Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
18.92Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
18.92Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
18.92Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
18.92Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
18.92Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
18.92Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
18.92Single8K5DGSK2560738K5D-HCA2-GSK256073
18.92Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
18.92Single8T1WCVN4248T1W-GPR6-CVN424
18.92Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.92Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.92Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.92Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
18.92Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
18.92Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
18.92Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
18.92Single9CHXS-Carazolol9CHX-β2-S-Carazolol
18.92Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
18.92Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
18.92Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
18.92Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
18.75Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
18.75Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
18.75Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
18.75Consensusbradykinin_onOrthosteric Ligandbk2_on
18.75Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
18.75Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
18.60Single6HLOAprepitant6HLO-NK1-Aprepitant
18.60Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
18.60Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
18.60Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
18.60Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
18.60Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
18.60Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
18.60Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
18.60Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
18.60Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.60Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
18.60Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
18.42Single2Y03Isoprenaline2Y03-β1-Isoprenaline
18.42Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
18.42Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
18.42Single5JQHS-Carazolol5JQH-β2-S-Carazolol
18.42Single5TVNLSD5TVN-5-HT2B-LSD
18.42Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
18.42Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
18.42Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
18.42Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
18.42Single6TP6Filorexant6TP6-OX1-Filorexant
18.42Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
18.42Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
18.42Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.42Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
18.42Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
18.42Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
18.42Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.42Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
18.42Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
18.42Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
18.42Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
18.42Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.42Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
18.42Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
18.42Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
18.42Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
18.42Single8S4DCMF-0198S4D-Apelin-CMF-019
18.42Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
18.42Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.42Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.42Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
18.42Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
18.42Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
18.42Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
18.42Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
18.42Single9B9ZA1AKO9B9Z-CB1-A1AKO
18.42Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
18.42Single9EHSLUF76029EHS-A3A-LUF7602
18.42Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
18.42Consensusblt_offOrthosteric Ligandblt1_off
18.42Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
18.42Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.42Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
18.42Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
18.42Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
18.42Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
18.42Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.42Consensustrace-amine_onOrthosteric Ligandta1_on
18.37Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
18.37Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
18.37Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
18.18Single3OE0CVX153OE0-CXCR4-CVX15
18.18Single6PT2KGCHM076PT2-δ-KGCHM07
18.18Single6W25SHU91196W25-MC4-SHU9119-Ca
18.18Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
18.18Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
18.18Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
18.18Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
18.18Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.18Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
18.00Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
18.00Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
18.00Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
17.95Single3P0GBI1671073P0G-β2-BI167107
17.95Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
17.95Single4BV0Neurotensin4BV0-NTS1-Neurotensin
17.95Single4DJHJDTic4DJH-κ-JDTic
17.95Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
17.95Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
17.95Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
17.95Single5V54Methiothepin5V54-5-HT1B-Methiothepin
17.95Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
17.95Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
17.95Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
17.95Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
17.95Single6H7JIsoprenaline6H7J-β1-Isoprenaline
17.95Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
17.95Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
17.95Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.95Single6WGTLSD6WGT-5-HT2A-LSD
17.95Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
17.95Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
17.95Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
17.95Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
17.95Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
17.95Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.95Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.95Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
17.95Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
17.95Single8EA0Iperoxo8EA0-M3-Iperoxo
17.95Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.95Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.95Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
17.95Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
17.95Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
17.95Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
17.95Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.95Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
17.95Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
17.95Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
17.95Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
17.95Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
17.95Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
17.95Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.95Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
17.95Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
17.95Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
17.95Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
17.95Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
17.95Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.95Consensus5ht1_offOrthosteric Ligand5ht1b_off
17.95Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
17.95Consensusa2_onOrthosteric Liganda2b_on
17.95Consensusa2_on_gpOrthosteric Liganda2b_on_gp
17.95Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.95Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.95Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
17.95Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.95Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
17.95Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
17.95Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
17.95Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
17.95Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
17.95Consensuslpa_onOrthosteric Ligandlpa1_on
17.95Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
17.95Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.95Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
17.95Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
17.95Consensusneurotensin_onOrthosteric Ligandnts1_on
17.95Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.95Consensusrelaxin_onOrthosteric Ligandrxfp4_on
17.95Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
17.95Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.95Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
17.78Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
17.78Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
17.78Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
17.78Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
17.78Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
17.78Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
17.65Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.65Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
17.65Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
17.65Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
17.50Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
17.50Single4LDEBI1671074LDE-β2-BI167107
17.50Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
17.50Single4RWADIPP-NH24RWA-δ-DIPP-NH2
17.50Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
17.50Single5CXVTiotropium5CXV-M1-Tiotropium
17.50Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
17.50Single6A93Risperidone6A93-5-HT2A-Risperidone
17.50Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
17.50Single6MXTSalmeterol6MXT-β2-Salmeterol
17.50Single6OS2TRV0266OS2-AT1-TRV026
17.50Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
17.50Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
17.50Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
17.50Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.50Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
17.50Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
17.50Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
17.50Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
17.50Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.50Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.50Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
17.50Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
17.50Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
17.50Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
17.50Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
17.50Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
17.50Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
17.50Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
17.50Single8JJ8Formoterol8JJ8-β2-Formoterol
17.50Single8JJLOlodaterol8JJL-β2-Olodaterol
17.50Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
17.50Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
17.50Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
17.50Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
17.50Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
17.50Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
17.50Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
17.50Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
17.50Consensusalpha1_offOrthosteric Ligandalpha1a_off
17.50Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
17.50Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
17.50Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
17.50Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
17.50Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
17.50Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.50Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
17.50Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
17.50Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
17.50Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
17.50Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
17.50Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.39Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
17.39Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
17.39Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
17.39Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
17.39Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
17.39Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
17.14Single3OE9IT1t3OE9-CXCR4-IT1t
17.14Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
17.14Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
17.14Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
17.14Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
17.07Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
17.07Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
17.07Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
17.07Single6K1QIRL25006K1Q-ETB-IRL2500
17.07Single7EZCUKA7EZC-A2A-UKA
17.07Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
17.07Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
17.07Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
17.07Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
17.07Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
17.07Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.07Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
17.07Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
17.07Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
17.07Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
17.07Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
17.07Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
17.07Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.07Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.07Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
17.07Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
17.07Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
17.07Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
17.07Consensuschemerin_onOrthosteric Ligandcml1_on
17.07Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.07Consensusprostanoid_offOrthosteric Ligandep_off dp_off
17.07Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
17.07Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
17.07Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.07Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.02Single7SK3CXCL127SK3-ACKR3-CXCL12
17.02Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
16.67Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
16.67Single4BWBNeurotensin4BWB-NTS1-Neurotensin
16.67Single6AKXA4R6AKX-CCR5-A4R
16.67Single6AKYMaraviroc6AKY-CCR5-Maraviroc
16.67Single6B73MP11046B73-κ-MP1104
16.67Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
16.67Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
16.67Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
16.67Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
16.67Single6PT3DPI-2876PT3-δ-DPI-287
16.67Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
16.67Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
16.67Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
16.67Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
16.67Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
16.67Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
16.67Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
16.67Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
16.67Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
16.67Single7XN9L-054,5227XN9-SST2-L-054,522
16.67Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
16.67Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
16.67Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
16.67Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
16.67Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
16.67Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
16.67Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
16.67Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
16.67Single8IWESpermidine8IWE-TA9-Spermidine
16.67Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
16.67Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
16.67Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
16.67Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
16.67Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
16.67Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
16.67Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
16.67Single8X5YAstemizole8X5Y-H1-Astemizole
16.67Single8Y0HVUF114188Y0H-CXCR3-VUF11418
16.67Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
16.67Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
16.67Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
16.67Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
16.67Single9IPYJR14a9IPY-C3aB-JR14a
16.67Single9KDFRES-701-39KDF-ETB-RES-701-3
16.67Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
16.67Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
16.67Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
16.67Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
16.67Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
16.67Consensusorexin_offOrthosteric Ligandox2_off ox1_off
16.67Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
16.67Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.67Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
16.67Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
16.33Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.33Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
16.28Single4IARErgotamine4IAR-5-HT1B-Ergotamine
16.28Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
16.28Single7F8XNN90567F8X-CCKA-NN9056
16.28Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
16.28Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.28Single8IEBA1LYA8IEB-GPR156-A1LYA
16.28Single8IEIA1LYA8IEI-GPR156-A1LYA
16.28Single8IEPA1LYA8IEP-GPR156-A1LYA
16.28Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
16.28Single8WKYPG-9348WKY-MC4-PG-934
16.28Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.28Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
16.28Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
16.28Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
16.28Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
16.28Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
16.28Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
16.22Single2YDOAdenosine2YDO-A2A-Adenosine
16.22Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
16.22Single4MBSMaraviroc4MBS-CCR5-Maraviroc
16.22Single4ZJCSB-6740424ZJC-OX1-SB-674042
16.22Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
16.22Single6PS0S-Carazolol6PS0-β2-S-Carazolol
16.22Single6PS4ICI118-5516PS4-β2-ICI118-551
16.22Single6PS5S-Propranolol6PS5-β2-S-Propranolol
16.22Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
16.22Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
16.22Single6TPGEMPA6TPG-OX2-EMPA
16.22Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
16.22Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
16.22Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
16.22Single7F61PF-036547467F61-H3-PF-03654746
16.22Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
16.22Single7T32ZM-2413857T32-A2A-ZM-241385
16.22Single7UL3Famotidine7UL3-H2-Famotidine
16.22Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
16.22Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
16.22Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
16.22Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
16.22Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
16.22Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
16.22Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
16.22Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
16.22Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
16.22Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
16.22Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.22Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.22Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
16.22Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
16.22Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
16.22Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
16.22Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
16.22Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
16.22Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
16.22Single8IHKAcifran8IHK-HCA3-Acifran
16.22Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
16.22Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
16.22Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
16.22Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
16.22Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
16.22Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.22Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.22Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
16.22Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
16.22Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
16.22Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
16.22Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.22Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
16.22Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
16.22Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
16.22Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
16.22Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
16.22Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
16.22Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
16.22Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
16.22Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
16.22Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
16.22Consensusgrh_offOrthosteric Ligandgnrh1_off
16.22Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.91Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
15.91Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
15.91Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
15.91Single7SK5CXCL127SK5-ACKR3-CXCL12
15.91Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.91Single8IEBA1LYA8IEB-GPR156-A1LYA
15.91Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
15.91Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
15.91Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
15.91Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
15.91Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
15.91Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
15.91Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
15.91Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
15.91Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
15.79Single3NY8ICI118-5513NY8-β2-ICI118-551
15.79Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
15.79Single4DAJTiotropium4DAJ-M3-Tiotropium
15.79Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
15.79Single4GBRS-Carazolol4GBR-β2-S-Carazolol
15.79Single4QKX35V4QKX-β2-35V
15.79Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
15.79Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
15.79Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
15.79Single5T04Neurotensin5T04-NTS1-Neurotensin
15.79Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
15.79Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
15.79Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
15.79Single6H7MSalbutamol6H7M-β1-Salbutamol
15.79Single6PS1Timolol6PS1-β2-Timolol
15.79Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
15.79Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
15.79Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
15.79Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
15.79Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
15.79Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
15.79Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
15.79Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
15.79Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
15.79Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
15.79Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
15.79Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
15.79Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
15.79Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
15.79Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
15.79Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
15.79Single7WC7Lisuride7WC7-5-HT2A-Lisuride
15.79Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
15.79Single7YXAONO-54306087YXA-S1P5-ONO-5430608
15.79Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
15.79Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
15.79Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
15.79Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
15.79Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
15.79Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
15.79Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
15.79Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
15.79Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
15.79Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
15.79Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
15.79Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
15.79Single8JXRLSD8JXR-D1-LSD
15.79Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
15.79Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
15.79Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
15.79Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
15.79Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
15.79Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
15.79Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
15.79Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
15.79Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
15.79Single9AS1DMT9AS1-5-HT2A-DMT
15.79Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
15.79Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
15.79Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
15.79Consensus5ht5_onOrthosteric Ligand5ht5a_on
15.79Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
15.79Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
15.79Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
15.79Consensusa3_onOrthosteric Liganda3a_on
15.79Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
15.79Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
15.79Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
15.79Consensusblt_onOrthosteric Ligandblt1_on
15.79Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
15.79Consensusdopamine_offOrthosteric Ligandd2_off d3_off
15.79Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
15.79Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
15.79Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
15.79Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
15.79Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
15.79Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
15.79Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
15.79Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
15.79Consensusleukotriene_onOrthosteric Ligandblt_on
15.79Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
15.79Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
15.79Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
15.56Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
15.56Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.56Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
15.56Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
15.56Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
15.56Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.56Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single2RH1S-Carazolol2RH1-β2-S-Carazolol
15.38Single2YCWS-Carazolol2YCW-β1-S-Carazolol
15.38Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
15.38Single5D6LS-Carazolol5D6L-β2-S-Carazolol
15.38Single5N2RPSB-365N2R-A2A-PSB-36-Na
15.38Single5N2SPSB365N2S-A1-PSB36
15.38Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
15.38Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
15.38Single5WIUNemonapride5WIU-D4-Nemonapride
15.38Single5WIVNemonapride5WIV-D4-Nemonapride-Na
15.38Single5WQCEMPA5WQC-OX2-EMPA
15.38Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
15.38Single5XPRBosentan5XPR-ETB-Bosentan
15.38Single6D26Fevipiprant6D26-DP2-Fevipiprant
15.38Single6E67BI1671076E67-β2-BI167107-Gs(CT)
15.38Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
15.38Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
15.38Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
15.38Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
15.38Single6PS6Timolol6PS6-β2-Timolol
15.38Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
15.38Single7C61Ergotamine7C61-5-HT1B-Ergotamine
15.38Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
15.38Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
15.38Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
15.38Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
15.38Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
15.38Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
15.38Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
15.38Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
15.38Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
15.38Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
15.38Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
15.38Single8QOTNanobody-E8QOT-μ-Nanobody-E
15.38Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
15.38Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
15.38Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
15.38Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
15.38Single8ZMFA1L108ZMF-5-HT2C-A1L10
15.38Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
15.38Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
15.38Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
15.38Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
15.38Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
15.38Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
15.38Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
15.38Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
15.38Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
15.38Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
15.38Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
15.38Consensusa3_on_gpOrthosteric Liganda3a_on_gp
15.38Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
15.38Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
15.38Consensusadenosine_offOrthosteric Liganda1_off a2_off
15.38Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
15.38Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
15.38Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
15.38Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
15.38Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
15.38Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
15.38Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
15.38Consensusamine_offonOrthosteric Ligandamine_off amine_on
15.38Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
15.38Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
15.38Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
15.38Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
15.38Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
15.38Consensusdp_offOrthosteric Liganddp2_off
15.38Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
15.38Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
15.38Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
15.38Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
15.38Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
15.38Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
15.38Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
15.38Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
15.38Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
15.38Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
15.22Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
15.22Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
15.22Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
15.22Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
15.22Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
15.00Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
15.00Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
15.00Single4U15Tiotropium4U15-M3-Tiotropium
15.00Single5D5AS-Carazolol5D5A-β2-S-Carazolol
15.00Single5D5BS-Carazolol5D5B-β2-S-Carazolol
15.00Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
15.00Single6J21Aprepitant6J21-NK1-Aprepitant
15.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
15.00Single6OL9Tiotropium6OL9-M5-Tiotropium
15.00Single6TQ7SB-3348676TQ7-OX1-SB-334867
15.00Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
15.00Single7B6WCyclazosin7B6W-α1b-Cyclazosin
15.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
15.00Single7F1TMIP-1a7F1T-CCR5-MIP-1a
15.00Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
15.00Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
15.00Single7PX4PSB-21137PX4-A2A-PSB-2113
15.00Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
15.00Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
15.00Single7TUYGSK682753A7TUY-GPR183-GSK682753A
15.00Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
15.00Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
15.00Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
15.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
15.00Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
15.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
15.00Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
15.00Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
15.00Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
15.00Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
15.00Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
15.00Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
15.00Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
15.00Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
15.00Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
15.00Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
15.00Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
15.00Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
15.00Single8ZWFJR14a8ZWF-C3aB-JR14a
15.00Single9AS9RS130-1809AS9-5-HT2A-RS130-180
15.00Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single9BJKNaloxone9BJK-μ-Naloxone-NAM
15.00Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
15.00Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
15.00Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
15.00Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
15.00Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
15.00Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
15.00Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
15.00Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
15.00Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
15.00Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
14.89Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
14.89Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
14.89Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
14.71Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
14.63Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
14.63Single3D4STimolol3D4S-β2-Timolol
14.63Single4AMIBucindolol4AMI-β1-Bucindolol
14.63Single4N4WSANT-14N4W-SMO-SANT-1
14.63Single5X33BIIL2605X33-BLT1-BIIL260
14.63Single6CM4Risperidone6CM4-D2-Risperidone
14.63Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
14.63Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
14.63Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
14.63Single6IIURamatroban6IIU-TXA2-Ramatroban
14.63Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
14.63Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
14.63Single6ZG4HTL00099366ZG4-M1-HTL0009936
14.63Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
14.63Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.63Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
14.63Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.63Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
14.63Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.63Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
14.63Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
14.63Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
14.63Single8JWY2-1188JWY-A2A-2-118
14.63Single8JWZAB9288JWZ-A2A-AB928-Na
14.63Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.63Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
14.63Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
14.63Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.63Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
14.63Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
14.63Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
14.63Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
14.63Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
14.63Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
14.63Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
14.63Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.63Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single3OE6IT1t3OE6-CXCR4-IT1t
14.29Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
14.29Single5CGDHTL142425CGD-mGlu5-HTL14242
14.29Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
14.29Single6H7LDobutamine6H7L-β1-Dobutamine
14.29Single6IBLArformoterol6IBL-β1-Arformoterol
14.29Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
14.29Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
14.29Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
14.29Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
14.29Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
14.29Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
14.29Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
14.29Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
14.29Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
14.29Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
14.29Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
14.29Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
14.29Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
14.29Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8XVJMacitentan8XVJ-ETA-Macitentan
14.29Single8XVUCXCL28XVU-CXCR2-CXCL2
14.29Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
14.29Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
14.29Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
14.29Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
14.29Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
14.29Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
14.29Single9LRCHistamine9LRC-H4-Histamine
14.29Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
14.29Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
14.29Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
14.29Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
14.29Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
13.95Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
13.95Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
13.95Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.95Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
13.95Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
13.95Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.95Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
13.95Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
13.95Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
13.95Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
13.95Consensuskisspeptin_onOrthosteric Ligandkiss1_on
13.89Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
13.89Single6LI0C176LI0-GPR52-C17
13.89Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
13.89Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
13.89Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
13.89Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
13.89Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
13.89Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.89Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
13.89Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
13.89Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
13.89Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
13.89Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
13.89Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
13.89Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
13.89Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
13.89Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.89Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
13.89Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
13.89Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
13.89Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
13.89Single9B9Y7DY9B9Y-CB1-7DY
13.89Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
13.89Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
13.89Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
13.89Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
13.89Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
13.89Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
13.89Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
13.89Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.64Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
13.64Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
13.64Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
13.64Single8KIGSHU91198KIG-MC3-SHU9119-Ca
13.64Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
13.64Single8XWNCXCL88XWN-CXCR2-CXCL8
13.64Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
13.64Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
13.64Single9M4TSilodosin9M4T-Alpha1A-Silodosin
13.64Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
13.64Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
13.64Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
13.51Single3ODUIT1t3ODU-CXCR4-IT1t
13.51Single3PWHZM-2413853PWH-A2A-ZM-241385
13.51Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
13.51Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
13.51Single4S0VSuvorexant4S0V-OX2-Suvorexant
13.51Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
13.51Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
13.51Single5WS3EMPA5WS3-OX2-EMPA
13.51Single5ZKQABT-4915ZKQ-PAF-ABT-491
13.51Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
13.51Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
13.51Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
13.51Single6ME2Ramelteon6ME2-MT1-Ramelteon
13.51Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
13.51Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
13.51Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
13.51Single6TODEMPA6TOD-OX1-EMPA-Na
13.51Single6TPJSuvorexant6TPJ-OX2-Suvorexant
13.51Single7BR3Elagolix7BR3-GnRH1-Elagolix
13.51Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
13.51Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
13.51Single7F8YDevazepide7F8Y-CCKA-Devazepide
13.51Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.51Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
13.51Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
13.51Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
13.51Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
13.51Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
13.51Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
13.51Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
13.51Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
13.51Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
13.51Single7XRRLemborexant7XRR-OX2-Lemborexant
13.51Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
13.51Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.51Single8GNGIstradefylline8GNG-A2A-Istradefylline
13.51Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
13.51Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
13.51Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
13.51Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.51Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.51Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.51Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
13.51Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
13.51Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
13.51Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
13.51Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
13.51Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
13.51Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
13.51Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
13.51Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
13.51Consensusalpha2_offOrthosteric Ligandalpha2c_off
13.51Consensusangiotensin_offOrthosteric Ligandat1_off
13.51Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
13.51Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
13.51Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
13.51Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
13.51Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
13.51Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
13.51Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
13.51Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
13.51Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
13.51Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
13.51Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
13.51Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
13.33Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
13.33Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
13.16Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
13.16Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
13.16Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
13.16Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
13.16Single5IU7Q274563465IU7-A2A-Q27456346-Na
13.16Single5IUBQ274563445IUB-A2A-Q27456344-Na
13.16Single5JTBZM-2413855JTB-A2A-ZM-241385
13.16Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
13.16Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
13.16Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
13.16Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
13.16Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
13.16Single6A94Zotepine6A94-5-HT2A-Zotepine
13.16Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
13.16Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
13.16Single6KUXRS-799486KUX-α2a-RS-79948
13.16Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
13.16Single6TP3Nemorexant6TP3-OX1-Nemorexant
13.16Single6TPNHTL66416TPN-OX2-HTL6641
13.16Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
13.16Single6V9SGTPL114036V9S-OX1-GTPL11403
13.16Single6VI4JDTic6VI4-κ-JDTic
13.16Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
13.16Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
13.16Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
13.16Single6ZG9GSK10347026ZG9-M1-GSK1034702
13.16Single7AROLUF58337ARO-A2A-LUF5833-Na
13.16Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
13.16Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
13.16Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
13.16Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
13.16Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
13.16Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
13.16Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
13.16Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.16Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
13.16Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
13.16Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
13.16Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
13.16Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
13.16Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
13.16Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
13.16Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.16Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
13.16Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.16Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
13.16Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
13.16Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
13.16Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.16Single8RLNLUF58348RLN-A2A-LUF5834
13.16Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
13.16Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.16Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.16Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
13.16Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.16Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.16Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
13.16Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
13.16Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
13.16Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
13.16Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
13.16Single9ARXSerotonin9ARX-5-HT2A-Serotonin
13.16Single9AS5Mescaline9AS5-5-HT2A-Mescaline
13.16Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single9BA0A1AKN9BA0-CB1-A1AKN
13.16Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
13.16Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
13.16Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
13.16Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
13.16Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
13.16Consensusa2_offOrthosteric Liganda2a_off
13.16Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
13.16Consensusalpha1_onOrthosteric Ligandalpha1a_on
13.16Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
13.16Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
13.16Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
13.16Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
13.16Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
13.16Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
13.16Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
13.16Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
13.04Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.04Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
13.04Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
13.04Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
13.04Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.04Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
12.82Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
12.82Single2Y01Dobutamine2Y01-β1-Dobutamine
12.82Single2Y02Carmoterol2Y02-β1-Carmoterol
12.82Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
12.82Single3EMLZM-2413853EML-A2A-ZM-241385
12.82Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
12.82Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
12.82Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
12.82Single4EJ4Naltrindole4EJ4-δ-Naltrindole
12.82Single4MQSIperoxo4MQS-M2-Iperoxo
12.82Single4U14Tiotropium4U14-M3-Tiotropium
12.82Single5DHGC-355DHG-NOP-C-35
12.82Single5DHHSB-6121115DHH-NOP-SB-612111
12.82Single5DSGTiotropium5DSG-M4-Tiotropium
12.82Single5IU8Q274563475IU8-A2A-Q27456347-Na
12.82Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
12.82Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
12.82Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
12.82Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
12.82Single5UENDU1725UEN-A1-DU172
12.82Single5UIGCmpd-15UIG-A2A-Cmpd-1
12.82Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
12.82Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
12.82Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
12.82Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
12.82Single6D27CAY104716D27-DP2-CAY10471
12.82Single6DRXLisuride6DRX-5-HT2B-Lisuride
12.82Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
12.82Single6GPSMK08126GPS-CCR2-MK0812
12.82Single6IIVDaltroban6IIV-TXA2-Daltroban
12.82Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
12.82Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
12.82Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
12.82Single6S0LZM-2413856S0L-A2A-ZM-241385
12.82Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
12.82Single7BU7BI1671077BU7-β1-BI167107
12.82Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
12.82Single7F83PF-051904577F83-Ghrelin-PF-05190457
12.82Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
12.82Single7PYRPSB-21157PYR-A2A-PSB-2115
12.82Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
12.82Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
12.82Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
12.82Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
12.82Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
12.82Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
12.82Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
12.82Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
12.82Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
12.82Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
12.82Single8CU6LJ-45178CU6-A2A-LJ-4517
12.82Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
12.82Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
12.82Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
12.82Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
12.82Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
12.82Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
12.82Single8JJOAlprenolol8JJO-β2-Alprenolol
12.82Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
12.82Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
12.82Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
12.82Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
12.82Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
12.82Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
12.82Single8X63Mepyramine8X63-H1-Mepyramine
12.82Single8X64Desloratadine8X64-H1-Desloratadine
12.82Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
12.82Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
12.82Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
12.82Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
12.82Single9H37A1IR09H37-A2A-A1IR0-Na
12.82Single9IYAONO-97105319IYA-GPR55-ONO-9710531
12.82Single9JEAAtropine9JEA-M1-Atropine
12.82Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
12.82Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
12.82Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
12.82Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
12.82Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
12.82Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
12.82Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
12.82Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
12.82Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
12.82Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
12.82Consensuscck_offOrthosteric Ligandccka_off
12.82Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
12.82Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
12.82Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
12.82Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
12.82Consensushistamine_offOrthosteric Ligandh1_off
12.82Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
12.82Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
12.82Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
12.82Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
12.77Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single2Y00Dobutamine2Y00-β1-Dobutamine
12.50Single4JKVTaladegib4JKV-SMO-Taladegib
12.50Single5CGCHTL142425CGC-mGlu5-HTL14242
12.50Single5IUAQ274563485IUA-A2A-Q27456348-Na
12.50Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
12.50Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
12.50Single6GPXMK08126GPX-CCR2-MK0812
12.50Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
12.50Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
12.50Single6LUQHaloperidol6LUQ-D2-Haloperidol
12.50Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
12.50Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
12.50Single6S0QZM-2413856S0Q-A2A-ZM-241385
12.50Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
12.50Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
12.50Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
12.50Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
12.50Single7SINNPS-21437SIN-CaS-NPS-2143
12.50Single7SINNPS-21437SIN-CaS-NPS-2143
12.50Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
12.50Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
12.50Single7W41PD1762527W41-BB2-PD176252
12.50Single7WC6LSD7WC6-5-HT2A-LSD
12.50Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
12.50Single8GNEKW-63568GNE-A2A-KW-6356-Na
12.50Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
12.50Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
12.50Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
12.50Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
12.50Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
12.50Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
12.50Single9HAPTolvaptan9HAP-V2-Tolvaptan
12.50Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
12.50Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
12.50Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
12.50Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
12.50Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
12.50Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
12.50Consensusbombesin_offOrthosteric Ligandbb2_off
12.50Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
12.50Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
12.50Consensusep_offOrthosteric Ligandep4_off
12.50Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.20Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
12.20Single5V56TC1145V56-SMO-TC114
12.20Single5V57TC1145V57-SMO-TC114
12.20Single6J20Aprepitant6J20-NK1-Aprepitant
12.20Single6OS1TRV0266OS1-AT1-TRV026
12.20Single7P2L4YI7P2L-mGlu5-4YI
12.20Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
12.20Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
12.20Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
12.20Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
12.20Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
12.20Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
12.20Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
12.20Single8XVLZibotentan8XVL-ETA-Zibotentan
12.20Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
12.20Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
12.20Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
12.20Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
12.12Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
11.90Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
11.90Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
11.90Single4PY02MeSATP4PY0-P2Y12-2MeSATP
11.90Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
11.90Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
11.90Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
11.90Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.90Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
11.90Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
11.90Single8XWMCXCL68XWM-CXCR2-CXCL6
11.90Single8XWSCXCL58XWS-CXCR2-CXCL5
11.90Single9BJKNAM9BJK-μ-Naloxone-NAM
11.90Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
11.90Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
11.76Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
11.76Single8HS2Fab0468HS2-GPR20-Fab046
11.76Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.63Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
11.63Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
11.63Single8XWFCXCL38XWF-CXCR2-CXCL3
11.63Single8ZPLHF511168ZPL-CXCR4-HF51116
11.63Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.43Single3OE8IT1t3OE8-CXCR4-IT1t
11.43Single6TQ9SB-4081246TQ9-OX1-SB-408124
11.43Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
11.43Single8A2OTheophylline8A2O-A2A-Theophylline-Na
11.43Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.43Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
11.43Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
11.43Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
11.43Single9CHUNoradrenaline9CHU-β2-Noradrenaline
11.43Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
11.43Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
11.43Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
11.36Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
11.36Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
11.36Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
11.36Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
11.36Single9JF4PD1683689JF4-BB1-PD168368
11.36Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.36Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single4XNWMRS25004XNW-P2Y1-MRS2500
11.11Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
11.11Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
11.11Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
11.11Single6ME5Agomelatine6ME5-MT1-Agomelatine
11.11Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
11.11Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
11.11Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
11.11Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
11.11Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
11.11Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
11.11Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
11.11Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.11Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
11.11Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
11.11Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
11.11Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
11.11Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
11.11Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
11.11Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
11.11Consensus5ht2_onOrthosteric Ligand5ht2b_on
11.11Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
11.11Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
10.87Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.87Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
10.81Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
10.81Single3PBLEticlopride3PBL-D3-Eticlopride
10.81Single5L7IVismodegib5L7I-SMO-Vismodegib
10.81Single6HLLCP999946HLL-NK1-CP99994
10.81Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
10.81Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
10.81Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
10.81Single7SRQLSD7SRQ-5-HT2B-LSD
10.81Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
10.81Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
10.81Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
10.81Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
10.81Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.81Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
10.81Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
10.81Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
10.81Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
10.81Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
10.81Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
10.81Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
10.81Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
10.81Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
10.81Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.81Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
10.81Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
10.81Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single9AS7Psilocin9AS7-5-HT2A-Psilocin
10.81Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
10.81Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
10.81Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
10.81Consensusgq_nucleotideOrthosteric Ligandgq_p2y
10.81Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.53Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
10.53Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
10.53Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
10.53Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
10.53Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
10.53Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
10.53Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
10.53Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
10.53Single6ME9Ramelteon6ME9-MT2-Ramelteon
10.53Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
10.53Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
10.53Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
10.53Single7F8ULintitript7F8U-CCKA-Lintitript
10.53Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.53Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.53Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
10.53Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
10.53Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
10.53Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
10.53Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
10.53Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
10.53Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
10.53Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
10.53Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
10.53Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
10.53Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
10.53Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
10.53Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
10.53Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
10.53Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
10.53Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
10.53Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
10.53Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
10.53Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
10.53Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
10.53Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
10.53Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
10.53Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
10.53Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
10.53Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
10.53Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.53Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.53Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.53Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.53Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.26Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
10.26Single3REYXAC3REY-A2A-XAC
10.26Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
10.26Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
10.26Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
10.26Single5UVIZM-2413855UVI-A2A-ZM-241385
10.26Single6AQFZM-2413856AQF-A2A-ZM-241385
10.26Single6IQLL7458706IQL-D4-L745870
10.26Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
10.26Single6MH8ZM-2413856MH8-A2A-ZM-241385
10.26Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
10.26Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
10.26Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
10.26Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
10.26Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
10.26Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
10.26Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
10.26Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
10.26Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
10.26Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
10.26Single8K2WAMG4878K2W-CXCR3-AMG487
10.26Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
10.26Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
10.26Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
10.26Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
10.26Single8ZPMAMD0708ZPM-CXCR4-AMD070
10.26Single8ZPNAMD31008ZPN-CXCR4-AMD3100
10.26Single9AS3LSD9AS3-5-HT2A-LSD
10.26Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
10.26Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
10.26Consensusopsins_offOrthosteric Ligandrhodopsin_off
10.26Consensussensory_offOrthosteric Ligandopsins_off
10.00Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
10.00Single4QIMANTA XV4QIM-SMO-ANTA XV
10.00Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.00Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
10.00Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
10.00Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
10.00Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.00Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
10.00Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.00Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
10.00Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
10.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
10.00Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
10.00Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
10.00Consensusalpha2_onOrthosteric Ligandalpha2b_on
10.00Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
10.00Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.00Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.00Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.00Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
9.76Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
9.76Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
9.76Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
9.76Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
9.76Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
9.76Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.76Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
9.76Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
9.76Single9HC04YI9HC0-mGlu5-4YI
9.76Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
9.52Single5TZRMK86665TZR-FFA1-MK8666
9.52Single6E59L-7607356E59-NK1-L-760735
9.52Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
9.52Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
9.52Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
9.52Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
9.52Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
9.52Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
9.52Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
9.52Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
9.52Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
9.52Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
9.52Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
9.52Consensustachykinin_offOrthosteric Ligandnk1_off
9.30Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
9.30Single8XWACXCL18XWA-CXCR2-CXCL1
9.30Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
9.30Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
9.09Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
9.09Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
9.09Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
9.09Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
8.89Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
8.89Single8XQJJN2418XQJ-Apelin-JN241
8.89Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
8.89Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
8.89Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
8.89Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
8.82Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
8.70Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
8.57Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
8.57Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
8.57Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.57Single8PWNTheophylline8PWN-A2A-Theophylline
8.57Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.33Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
8.33Single3RFMCaffeine3RFM-A2A-Caffeine
8.33Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
8.33Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
8.33Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
8.33Consensusp2y_offOrthosteric Ligandp2y1_off
8.33Consensussensory_onOrthosteric Ligandopsins_on
8.11Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
8.11Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
8.11Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
8.11Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.11Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.11Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
8.11Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
8.11Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
8.11Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
8.11Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
8.11Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.11Consensusgi_sensoryOrthosteric Ligandgi_opsins
8.11Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.11Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.11Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
8.11Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
8.11Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
7.89Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
7.89Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
7.89Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
7.89Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
7.89Single4O9RCyclopamine4O9R-SMO-Cyclopamine
7.89Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
7.89Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
7.89Single6TP4ACT-4622066TP4-OX1-ACT-462206
7.89Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.89Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.89Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
7.89Single7UL2SR486927UL2-NTS1-SR48692-Na
7.89Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
7.89Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.89Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
7.89Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.89Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.89Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.89Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
7.89Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
7.89Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.89Consensusneurotensin_offOrthosteric Ligandnts1_off
7.89Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
7.69Single4QINSAG1.54QIN-SMO-SAG1.5
7.69Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
7.69Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
7.69Single6DS0Ly2660976DS0-5-HT2B-Ly266097
7.69Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
7.69Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
7.69Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
7.69Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
7.69Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
7.69Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
7.69Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
7.69Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
7.69Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
7.69Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
7.69Single9H2XA1IR19H2X-A2A-A1IR1-Na
7.69Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
7.69Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
7.50Single3RZECidoxepin3RZE-H1-Cidoxepin
7.50Single6FFIMMPEP6FFI-mGlu5-MMPEP
7.50Single6TPKRetosiban6TPK-OT-Retosiban
7.50Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
7.50Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
7.50Single7VODCariprazine7VOD-5-HT2A-Cariprazine
7.50Single7VV6C48/807VV6-MRGPRX2-C48/80
7.50Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
7.50Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
7.50Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
7.50Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
7.50Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
7.50Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
7.50Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
7.50Consensusvasop-oxy_offOrthosteric Ligandot_off
7.32Single6FFHFenobam6FFH-mGlu5-Fenobam
7.32Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
7.32Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
7.14Single4NTJAZD12834NTJ-P2Y12-AZD1283
7.14Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
7.14Single6HLPNetupitant6HLP-NK1-Netupitant
7.14Single6Z4SSR486926Z4S-NTS1-SR48692
7.14Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
7.14Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
7.14Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
7.14Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
6.98Single7R0CAVP7R0C-V2-AVP-Arrestin2
6.98Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
6.82Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
6.82Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
6.82Single8XQJJN2418XQJ-Apelin-JN241
6.82Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.82Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
6.82Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
6.67Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
6.67Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
6.52Single6KNMJN241-96KNM-Apelin-JN241-9
6.52Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
5.88Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
5.71Single5MZPCaffeine5MZP-A2A-Caffeine-Na
5.71Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
5.56Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
5.56Single7WC4Serotonin7WC4-5-HT2A-Serotonin
5.56Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
5.56Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
5.41Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
5.41Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
5.41Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
5.41Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
5.41Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
5.26Single3UZAGTPL92363UZA-A2A-GTPL9236
5.26Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.26Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
5.26Single7WC5Psilocin7WC5-5-HT2A-Psilocin
5.26Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
5.26Single8JPSCCL78JPS-ACKR1-CCL7
5.13Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
5.13Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
4.88Single6ZINSR486926ZIN-NTS1-SR48692
4.88Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.88Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.65Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
4.55Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.35Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
3.03Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
3.03Single6D35Cholesterol6D35-SMO-Cholesterol
3.03Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
3.03Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
3.03Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
3.03Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
3.03Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
3.03Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
3.03Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
3.03Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
3.03Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
3.03Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
3.03Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.03Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.03Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.03Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.03Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
3.03Single7DTTCa7DTT-CaS-Ca-Ca
3.03Single7DTTCa7DTT-CaS-Ca-Ca
3.03Single7DTUTryptophan7DTU-CaS-Tryptophan
3.03Single7DTUTryptophan7DTU-CaS-Tryptophan
3.03Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
3.03Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
3.03Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
3.03Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
3.03Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.03Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.03Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.03Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.03Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
3.03Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
3.03Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
3.03Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
3.03Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
3.03Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
3.03Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
3.03Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
3.03Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
3.03Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
3.03Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
3.03Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
3.03Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
3.03Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.03Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.03Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
3.03Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
3.03Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.03Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.03Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.03Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.03Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
3.03Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
3.03Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
3.03Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
3.03Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
3.03Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
3.03Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.03Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.03Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.03Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.03Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.03Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.03Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.03Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.03Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
3.03Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
3.03Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
3.03Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
3.03Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
3.03Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
3.03Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
3.03Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
3.03Single7XW7K1-707XW7-TSH-K1-70
3.03Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
3.03Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
3.03Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
3.03Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
3.03Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
3.03Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
3.03Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
3.03Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
3.03Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
3.03Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
3.03Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
3.03Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
3.03Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
3.03Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
3.03Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
3.03Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
3.03Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
3.03Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
3.03Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
3.03Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
3.03Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
3.03Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.03Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.03Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.03Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.03Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.03Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.03Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
3.03Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
3.03Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
3.03Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
3.03Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
3.03Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.03Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.03Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
3.03Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
3.03Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
3.03Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
3.03Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
3.03Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
3.03Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
3.03Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
3.03Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
3.03Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
3.03Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
3.03Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
3.03Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
3.03Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
3.03Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
3.03Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
3.03Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.03Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.03Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.03Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.03Single8WVXNorrin8WVX-LGR4-Norrin
3.03Single8WVYNorrin8WVY-LGR4-Norrin
3.03Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.03Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.03Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.03Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.03Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.03Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.03Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
3.03Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
3.03Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.03Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.03Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
3.03Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
3.03Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
3.03Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
3.03Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
3.03Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.03Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.03Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.03Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.03Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.03Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.03Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.03Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.03Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.03Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.03Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.03Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.03Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.03Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.03Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.03Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.03Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.03Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.03Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.03Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.03Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.03Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.03Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
3.03Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
3.03Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
3.03Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
3.03Single9KHHNorrin9KHH-LGR4-Norrin
3.03Single9S37NB219S37-LGR4-NB21
3.03Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
2.94Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
2.94Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
2.94Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
2.94Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
2.94Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
2.94Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
2.94Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
2.94Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
2.94Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
2.94Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
2.94Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
2.94Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
2.94Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
2.94Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
2.94Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
2.94Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
2.94Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
2.94Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
2.86Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
2.86Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
2.86Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
2.78Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
2.78Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
2.78Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
2.78Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
2.78Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
2.78Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
2.78Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
2.70Single5L7DCholesterol5L7D-SMO-Cholesterol
2.70Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
2.70Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
2.70Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
2.63Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
2.63Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
2.56Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
2.50Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.50Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
2.50Single8HNNSCH5467388HNN-CXCR3-SCH546738
2.44Single4K5YCP-3763954K5Y-CRF1-CP-376395
2.44Single4XNVBPTU4XNV-P2Y1-BPTU
2.44Single6C1QNDT95137276C1Q-C5a1-PMX53-NDT9513727
2.38Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
2.38Single8IYXYL-3658IYX-GPR34-YL-365
2.33Single4Z9GCP-3763954Z9G-CRF1-CP-376395
2.33Single8GTIBMK-C2058GTI-CRF1-BMK-C205
2.27Single8GTGBMK-I1528GTG-CRF1-BMK-I152
2.17Single8GTMBMK-C2038GTM-CRF1-BMK-C203
2.04Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.04Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
1.96Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
1.96Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
1.92Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
1.82Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
pth1_on_gp 6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
7Y36-PTH1-Teriparatide-Gs/β1/γ2
7Y35-PTH1-Abaloparatide-Gs/β1/γ2
pth2_on_gp 7F16-PTH2-TIP39-Gs/β1/γ2
Net Summary
Imin 2.866
Number of Linked Nodes 896
Number of Links 1120
Number of Hubs 189
Number of Links mediated by Hubs 729
Number of Communities 22
Number of Nodes involved in Communities 255
Number of Links involved in Communities 398
Path Summary
Number Of Nodes in MetaPath 105
Number Of Links MetaPath 104
Number of Shortest Paths 1820581
Length Of Smallest Path 3
Average Path Length 32.2195
Length of Longest Path 59
Minimum Path Strength 0.1355
Average Path Strength 6.33257
Maximum Path Strength 58.6265
Minimum Path Correlation 0.7
Average Path Correlation 0.99056
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.38095
Average % Of Corr. Nodes 50.3196
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 47.0007
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
class-b1_on_gpglucagon_on_gp
vip-pacap_on_gp
pth_on_gp
crf_on_gp
calcitonin_on_gp



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