Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.40 5.37437457
2G.H1.01 3.2085509
3G.S3.03 6.18508
4G.S3.04 11.64884177
5G.S3.06 11.364177
6G.H2.01 5.73409
7G.H2.06 6.0055549
8G.H2.07 5.2025409
9G.h2s4.01 8.619509
10G.H3.01 3.25625409
11G.H3.09 5.0715199
12G.H3.13 8.82455196
13G.H3.17 10.1758665
14G.S5.05 5.145189
15G.S5.07 3.6875509
16G.s5hg.01 2.9175509
17G.HG.01 4.86812496
18G.hgh4.01 6.94875406
19G.hgh4.02 4.80254208
20G.hgh4.04 4.09254206
21G.hgh4.05 7.39506
22G.hgh4.08 8.05406
23G.hgh4.11 4.72125405
24G.hgh4.20 6.87438403
25G.H4.05 6.87188405
26G.H4.08 6.76125493
27G.H4.10 9.5765207
28G.H4.12 6.38937494
29G.H4.15 7.87125408
30G.h4s6.12 5.4975402
31G.S6.02 8.29875408
32G.S6.05 7.7035595
33G.s6h5.01 6.35754189
34G.H5.08 5.50417628
35G.H5.17 9.32875425
36G.H5.20 3.6325408
37G.H5.23 7.353754104
38b.1x3 2.14625408
39b.lh12x2 4.461874228
40b.lhb1x6 4.640624123
41b.l1x3 9.289559
42b.l1x6 9.5105569
43b.b2x1 6.51937468
44b.b2x5 6.92042607
45b.l3x2 7.47625409
46b.b4x6 10.0721659
47b.b4x7 8.09375458
48b.b5x2 8.66375457
49b.b5x3 6.936559
50b.l5x1 4.4575408
51b.l5x5 8.93917609
52b.b6x1 4.6625409
53b.l7x4 3.88625409
54b.b8x4 5.4515506
55b.l8x3 1.88188403
56b.l9x3 7.339549
57b.l9x6 6.01542648
58b.b10x5 4.91875609
59b.b12x6 8.43083648
60b.b13x7 9.535477
61b.l13x3 9.053579
62b.l13x6 6.67625449
63b.b15x2 7.23062436
64b.l15x1 5.08313447
65b.l15x2 6.52063479
66b.b16x4 9.839576
67b.b16x5 4.85625405
68b.b16x6 10.165578
69b.b16x7 7.828754139
70b.b17x5 7.86062437
71b.b17x7 8.97375438
72b.l17x3 8.67429739
73b.l17x6 8.38875449
74b.b18x3 5.185438
75b.l18x1 6.934586146
76b.l18x2 6.114384147
77b.b19x2 7.116536
78b.b19x4 5.37437438
79b.l19x1 6.72813449
80b.l19x2 7.9355539
81b.b20x2 7.19938436
82b.b20x4 9.50583638
83b.b20x6 7.1675536
84b.b21x1 6.806537
85b.b21x7 5.81917605
86b.b22x5 5.5855147
87b.l22x5 7.4375129
88b.b23x1 3.90625405
89b.b23x6 6.905836157
90b.l23x1 6.339566
91b.b24x6 7.286884158
92b.l25x3 7.785689
93b.l25x6 14.7775468
94b.l27x1 10.0271769
95b.l27x2 7.38938489
96b.b28x4 7.65375486
97b.b28x6 9.332589
98g.h1x8 3.295407
99g.ctx3 6.5975509
100g.ctx6 3.822926126
101g.ctx14 5.749374119
102g.ctx15 7.37754119
103g.ctx16 5.479297118
104Lig 21.37912610
105NT 187.545615
1061x29 3.6875412
1071x35 2.76187415
1081x39 6.54618
1091x43 6.11958618
1101x50 3.915409
1111x60 5.01562406
1122x39 6.2935109
1132x40 4.663134109
1142x43 6.595624109
1152x50 8.0815508
1162x53 7.29375618
1172x60 5.882517
118E1 22.1054614
1193x32 5.5495517
1203x33 5.0145517
1213x40 8.7555518
1223x41 4.90125415
1233x42 9.354586169
1243x46 8.97409
1253x49 6.1695508
1263x51 5.20312408
127I2 6.311226
1284x41 2.88063424
1294x46 4.997507
1304x50 8.07254168
1314x60 6.69518
1324x64 10.7094418
133E2 10.0112815
134E2x51 12.1565519
135E2x52 4.94625415
1365x41 8.3005517
1375x43 5.14687417
1385x51 3.01937417
1395x58 6.6454219
1405x68 6.88875429
141I3 5.3275725
1426x44 5.90455219
1436x48 7.19429718
1446x51 6.89875416
145E3 6.19964714
1467x33 6.27063418
1477x37 7.17563417
1487x45 6.3725419
1497x55 2.23563409
1508x58 3.5125406
151b.l11x2 6.9575440
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b4x6 b.l1x3 56.54684.76YesYes599
2b.b3x6 b.l1x3 57.551611.855NoYes099
3b.b3x6 b.l3x2 57.68467.7275NoYes099
4b.l1x4 b.l3x2 62.021311.8725NoYes069
5G.hns1.01 b.l1x4 62.50784.9825NoNo046
6G.S1.03 G.hns1.01 62.628720.835NoNo094
7G.S1.03 G.S3.06 62.74924.5425NoYes097
8G.S3.06 b.l5x5 63.702321.545YesYes079
9G.h2s4.01 b.l5x5 53.774911.7775YesYes099
10G.H2.07 G.h2s4.01 65.00593.7575YesYes099
11G.H2.04 G.H2.07 1006.75NoYes099
12G.H2.04 G.H3.08 99.8829.415NoNo098
13G.H3.08 G.S4.04 99.65886.7NoNo089
14G.H3.09 G.S4.04 99.43113.485YesNo099
15G.H3.09 G.H4.15 97.56478.3025YesYes098
16G.H4.15 G.S5.04 97.08578.22YesNo089
17G.S5.04 G.S6.03 84.41263.695NoNo095
18G.H4.16 G.S6.03 78.48924.105NoNo045
19G.H4.16 I3 78.35754.8025NoYes245
20G.H5.17 I3 77.33445.24YesYes255
215x68 G.H5.17 73.58267.735YesYes295
225x68 G.H5.16 77.72029.83YesNo296
23G.H5.16 I2 77.32964.995NoYes266
24G.S5.04 G.S5.06 12.67014.15NoNo098
25G.S5.06 G.S6.05 12.43914.2625NoYes085
26G.HG.01 G.S6.05 10.04345.27YesYes965
27G.S5.07 G.s6h5.01 10.382.925YesYes099
28G.H2.07 G.s3h2.03 36.2623.56YesNo099
29b.l5x5 b.l7x2 17.75375.41YesNo099
30b.l7x2 b.l9x6 17.72053.5175NoYes098
31G.s3h2.03 b.l9x6 36.19746.2NoYes098
32b.b14x1 b.l9x6 34.07314.4875NoYes088
33G.H2.06 b.b14x1 33.92287.2YesNo098
34G.H2.06 b.l19x1 36.35094.4925YesYes499
35G.H3.17 b.l27x1 33.81776.56YesYes659
36b.l1x6 b.l27x1 19.276419.725YesYes699
37b.l1x6 b.l3x1 19.65169.49YesNo699
38b.l3x1 b.l5x5 39.28245.2025NoYes099
39b.b2x1 b.l27x1 48.2884.34YesYes689
40b.b2x1 b.l3x1 19.534611.275YesNo689
41G.H2.10 G.h2s4.01 12.01293.49NoYes089
42G.H2.10 b.b6x1 11.94233.645NoYes089
43b.b2x1 b.b6x1 29.54625.6875YesYes089
44b.b6x1 b.l9x6 18.63965.39YesYes098
45G.H4.13 G.hgh4.08 10.56459.1975NoYes036
46G.H4.12 G.H4.13 10.82327.745YesNo043
47G.H4.12 G.S6.03 13.11795.04YesNo045
48G.H3.17 b.l23x1 30.94626.98YesYes656
49b.l25x6 b.l27x1 31.867121.99YesYes689
50b.l23x1 b.l25x6 30.896312.805YesYes668
513x49 4x46 16.84423.9725YesYes087
524x42 4x46 66.32424.09NoYes047
534x42 I2 66.683610.5125NoYes246
542x42 3x46 10.75766.1475NoYes099
552x42 3x49 11.10963.93NoYes098
56b.l17x5 b.l19x1 39.3023.3125NoYes069
57b.l17x5 b.l19x2 39.11794.415NoYes069
58b.l17x3 b.l19x2 31.72085.67YesYes399
59b.b19x4 b.l17x3 24.56187.19YesYes389
60b.b18x3 b.b19x4 18.84265.32YesYes388
61b.b15x2 b.b18x3 18.00946.1425YesYes368
62b.b15x2 b.b16x5 16.93584.0975YesYes065
63b.b16x5 b.l14x6 16.87014.4975YesNo053
64b.b16x7 b.l14x6 16.65935.09YesNo093
65b.b17x2 g.h1x13 14.72322.5275NoNo031
66g.h1x13 g.h1x9 13.83864.06NoNo016
67g.h1x8 g.h1x9 10.73271.7825YesNo076
68b.b17x7 b.b20x6 14.845811.255YesYes386
69b.b17x7 b.b21x1 12.85616.8675YesYes387
70b.b20x4 b.b20x6 11.23194.545YesYes386
71b.l21x7 b.l23x1 59.90725.0575NoYes056
72b.b23x6 b.l21x7 55.04034.03YesNo075
73b.b23x6 b.b24x6 43.27495.7875YesYes1578
74b.b21x7 b.b24x6 38.39338.44YesYes058
75b.l26x5 g.ctx4 44.04113.3525NoNo057
76g.ctx3 g.ctx4 43.71444.83YesNo097
77g.ctx3 g.ctx6 23.79878.48YesYes096
78b.l22x1 g.ctx3 19.43027.7275NoYes099
79b.b23x1 b.l22x1 19.24684.125YesNo059
80b.b23x1 b.b24x5 37.66024.8425YesNo055
81b.b23x3 b.b24x5 36.88625.215NoNo075
82b.b23x3 b.b27x1 36.49874.47NoNo076
83b.b27x1 g.ctx5 35.33442.98NoNo069
84b.lhb1x11 g.ctx5 34.94573.5325NoNo049
85b.b25x7 b.lhb1x11 34.55675.655NoNo074
86b.b23x1 g.ctx6 19.57913.805YesYes056
87b.b25x7 b.b28x6 33.777720.215NoYes079
88b.b28x4 b.b28x6 17.30696.96YesYes869
89b.b27x3 b.b28x6 15.29328.185NoYes089
90b.b27x3 b.l25x3 14.10137.19NoYes089
91b.l25x3 b.l27x2 24.17956.615YesYes899
92b.b28x4 b.l25x3 14.101712.7725YesYes869
93b.b3x2 b.b4x6 46.62285.125NoYes059
94b.b2x5 b.b3x2 46.47419.11YesNo075
95b.l11x1 b.l9x6 18.64366.155NoYes498
96b.b11x6 b.l11x1 24.11593.2475NoNo499
97b.b11x6 b.l9x3 22.860713.25NoYes499
98b.b11x4 b.l9x3 17.09155.8225NoYes499
99b.b10x3 b.b11x4 17.05232.9575NoNo089
100b.b10x3 b.b6x2 16.8045.07NoNo088
101b.b10x2 b.b6x2 16.55552.9575NoNo068
102b.b10x2 b.b14x3 16.30664.76NoNo065
103b.b11x3 b.b14x3 11.95874.0975NoNo055
104b.b2x5 b.l26x1 42.203114.5575YesNo077
105b.l26x3 b.l26x5 41.75217.275NoNo075
106b.l26x1 b.l26x3 41.85745.785NoNo2377
107b.b21x7 b.b23x2 25.65964.3975YesNo056
108b.b22x5 b.b23x2 24.67668.22YesNo076
109b.b22x5 b.l18x1 10.866210.1825YesYes1476
110b.l25x4 b.l27x2 21.78943.6575NoYes059
111I1x49 b.l25x4 10.492110.0225NoNo075
1128x56 b.l25x4 10.49215.3625NoNo075
1133x45 4x46 49.33384.915NoYes077
1143x42 3x45 48.92328.07YesNo097
1152x49 3x42 46.71274.6325NoYes099
1162x49 3x39 46.51437.45NoNo098
1172x53 3x39 42.578911.1475YesNo088
1182x53 Lig 32.44285.12YesYes180
1191x60 8x53 17.75119.6175YesNo067
1201x60 8x57 12.89625.8925YesNo065
1218x57 8x60 11.27731.1475NoNo057
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x32Lig3.91YesYes7010
3x33Lig6.49751YesYes7010
3x36Lig13.5051NoYes5010
3x40Lig5.47751YesYes8010
5x41Lig7.8051YesYes7010
7x34Lig8.830NoYes6010
7x37Lig6.351YesYes7010
7x38Lig11.89751NoYes7010
1x43Lig4.31251YesYes8010
2x53Lig5.121YesYes8010
E2Lig25.271YesYes5010
E3Lig5.12251YesYes4010
1x32Lig26.4951NoYes4010
1x35Lig4.4051YesYes5010
1x39Lig9.98251YesYes8010
2x60Lig9.00751YesYes7010
E1Lig40.1151YesYes4010
E2x52Lig8.40251YesYes5010
1x29Lig8.55251YesYes2010
LigNT89.4551YesYes0501
1x25Lig7.421NoYes1010
NTNT506.561YesYes5511
E1NT16.251YesYes4511
1x281x324.24250NoNo3421
1x361x395.67251NoYes5821
1x362x614.49251NoNo5722
1x391x403.74751YesNo8712
1x391x434.7151YesYes8811
1x392x616.03751YesNo8712
1x397x389.0851YesNo8711
1x432x536.94251YesYes8811
1x432x579.4651YesNo8712
1x437x427.94751YesNo8912
2x533x369.38251YesNo8511
2x533x3911.14751YesNo8812
2x533x407.56751YesYes8811
2x536x483.60251YesYes8812
2x563x325.07750NoYes6721
2x573x324.020NoYes7721
2x602x613.45751YesNo7712
2x602x643.87751YesNo7712
2x603x3210.4051YesYes7711
2x62E13.60NoYes2421
2x64E111.23251NoYes7421
E1E130.71751YesYes4411
3x26E27.00251NoYes8521
3x26E2x5122.04751NoYes8922
3x323x364.3451YesNo7511
3x334x606.72251YesYes7812
3x335x413.46751YesYes7711
3x335x436.071YesYes7712
3x405x4710.7051YesNo8712
3x405x514.62751YesYes8712
3x406x4815.41YesYes8812
4x60E2x513.751YesYes8922
4x605x436.16751YesYes8722
4x68E23.65751NoYes6521
E2E26.80751YesYes5511
E2E2x5110.051YesYes5912
E2E2x524.24751YesYes5511
5x41E216.24751YesYes7511
5x415x434.99251YesYes7712
5x415x448.991YesNo7712
5x516x483.631YesYes7822
6x487x376.7351YesYes8721
6x517x339.021YesYes6821
6x517x378.4551YesYes6721
6x54E36.48250NoYes5421
E3E39.151YesYes4411
7x31E33.481NoYes3421
7x32E35.770NoYes4421
7x33E34.24251YesYes8411
7x337x377.16251YesYes8711
7x33Lig4.65751YesYes8010
1x26Lig3.380NoYes2010
3x22NT5.26251NoYes3521
1x311x354.150NoYes5521
2x64E2x524.411NoYes7521
1x317x315.9150NoNo5322
1x432x543.3351YesNo8712
1x271x293.32750NoYes1221
7x30Lig3.03250NoYes5010
E2x50E2x522.7250NoYes9521
2x603x282.66251YesNo7512
1x291x332.491YesNo2312
3x293x332.3150NoYes5721
1x221x251.9950NoNo2121
1x357x391.281YesNo5512
1x341x351.21250NoYes4521
1x24NT1.18250NoYes2521
1x291x300.381YesNo2212

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
84.00Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
84.00Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
80.77Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
80.00Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
80.00Consensuspac_onOrthosteric Ligandpac1_on
80.00Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
77.78Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
77.78Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
77.78Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
76.92Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
75.00Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
74.07Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
74.07Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
73.08Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
73.08Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
72.41Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
70.37Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
70.37Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
69.23Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
68.97Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
68.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
67.86Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
67.86Consensusglp_onOrthosteric Ligandglp1_on glp2_on
67.86Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
66.67Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
66.67Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
65.52Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
65.38Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
64.52Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
64.52Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
64.29Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
64.29Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
64.29Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
64.29Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
64.29Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
64.29Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
62.96Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
62.96Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
62.96Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
62.96Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
62.50Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
62.07Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
61.29Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
60.71Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
60.61Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
60.00Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
60.00Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
59.46Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
58.62Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
58.62Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
58.62Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
58.62Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
57.58Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
57.58Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
57.58Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
57.58Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
57.14Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
57.14Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
57.14Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
56.67Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
56.67Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
56.00Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
54.84Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
54.84Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
54.84Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
54.55Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
54.05Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
53.57Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
53.12Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
52.78Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
52.78Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
51.85Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
51.72Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
51.61Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
51.43Consensuspth_onOrthosteric Ligandpth1_on pth2_on
50.00Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
50.00Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
50.00Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
50.00Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
50.00Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
50.00Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
48.28Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
46.88Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
46.67Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
45.45Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
44.44Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
44.44Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
44.44Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
43.75Single6FJ3PTH6FJ3-PTH1-PTH
43.33Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
43.33Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
43.33Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
43.24Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
42.86Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
42.42Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
41.67Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
41.18Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
41.18Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
41.18Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
41.18Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
41.18Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
40.62Consensuscalcitonin_onOrthosteric Ligandctlike_on
40.00Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
39.39Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
39.39Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
39.39Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
39.39Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
39.29Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
39.29Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
38.89Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
38.24Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
38.24Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
37.50Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
37.50Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
37.50Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
37.14Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
37.14Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
36.84Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
36.67Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
36.36Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
36.36Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
35.48Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
35.48Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
35.29Single4XT3Fractalkine4XT3-US28-Fractalkine
35.29Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
35.29Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
35.29Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
35.29Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
34.48Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
34.38Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
34.29Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
34.29Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
34.29Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
34.29Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
34.29Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
34.21Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
34.21Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
33.33Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
33.33Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
33.33Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
33.33Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
33.33Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
33.33Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
33.33Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
33.33Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
33.33Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
33.33Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
33.33Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
33.33Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
32.43Single6IGKEndothelin-36IGK-ETB-Endothelin-3
32.43Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
32.43Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
32.43Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
32.35Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
32.35Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
32.35Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
32.26Single4XT1Fractalkine4XT1-US28-Fractalkine
32.26Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
32.26Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
32.26Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
31.58Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
31.58Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
31.43Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
31.43Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
31.43Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
31.43Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
31.43Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
31.43Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
31.25Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
31.25Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
31.03Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
31.03Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
30.95Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
30.56Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
30.56Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
30.56Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
30.56Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
30.56Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
30.56Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
30.56Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
30.56Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
30.30Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
30.30Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
30.30Consensusangiotensin_onOrthosteric Ligandat1_on
30.30Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
30.00Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
30.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
30.00Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
29.73Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
29.73Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
29.63Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
29.63Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
29.55Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
29.41Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
29.41Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
29.41Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.41Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
29.03Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
29.03Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
29.03Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
29.03Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
28.95Single5GLHEndothelin-15GLH-ETB-Endothelin-1
28.95Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
28.95Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
28.95Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
28.95Consensusbombesin_onOrthosteric Ligandbb2_on
28.95Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
28.95Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
28.57Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
28.57Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
28.57Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
28.57Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
28.57Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8ZRTET-18ZRT-ETB-ET-1
28.57Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
28.57Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.57Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
28.21Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
28.12Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
28.12Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
28.12Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
28.12Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
28.12Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.12Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.12Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
28.12Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
27.78Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
27.59Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
27.59Single7TUYGSK682753A7TUY-GPR183-GSK682753A
27.59Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
27.59Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
27.50Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
27.27Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
27.27Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
27.27Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
27.27Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
27.27Single7XNACYN1548067XNA-SST2-CYN154806
27.27Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
27.27Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
27.27Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
27.27Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
27.27Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
27.27Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
27.27Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
27.27Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
27.03Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
27.03Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
27.03Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
27.03Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
27.03Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
26.92Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
26.67Single6OS2TRV0266OS2-AT1-TRV026
26.67Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
26.67Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
26.67Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
26.67Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
26.67Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
26.67Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
26.67Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
26.67Consensuslpa_offOrthosteric Ligandlpa1_off
26.67Consensuslpl_offOrthosteric Ligands1p_off lpa_off
26.47Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
26.47Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.47Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
26.47Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
26.47Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
26.47Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
26.47Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
26.47Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
26.32Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
26.32Single8IY6Endothelin-18IY6-ETB-Endothelin-1
26.32Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
26.32Consensusendothelin_onOrthosteric Ligandetb_on eta_on
25.93Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
25.81Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
25.81Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
25.81Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
25.81Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
25.81Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
25.81Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
25.71Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
25.71Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.71Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
25.71Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
25.71Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
25.71Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
25.71Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
25.71Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
25.71Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
25.71Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
25.71Consensusvasop-oxy_onOrthosteric Ligandv2_on
25.71Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
25.64Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
25.64Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
25.64Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
25.64Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
25.58Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
25.00Single4UG2CGS216804UG2-A2A-CGS21680
25.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
25.00Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
25.00Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
25.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
25.00Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.00Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
25.00Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
25.00Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
25.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
25.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
25.00Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
25.00Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
25.00Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
25.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
25.00Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
25.00Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
25.00Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
25.00Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
25.00Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
25.00Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
25.00Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
25.00Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
25.00Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
25.00Consensushca_on_gpOrthosteric Ligandhca2_on_gp
25.00Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
25.00Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
25.00Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
25.00Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
25.00Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
24.39Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
24.32Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
24.32Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
24.32Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
24.24Single7QA8Peptide7QA8-STE2-Peptide
24.24Single7QA8Peptide7QA8-STE2-Peptide
24.24Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
24.24Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
24.24Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
24.24Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
24.24Consensuslpl_onOrthosteric Ligands1p_on lpa_on
24.24Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
24.24Consensussomatostatin_offOrthosteric Ligandsst2_off
24.14Single5C1MBU725C1M-μ-BU72
24.14Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
24.14Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
24.14Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
24.14Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
24.14Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.14Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
24.14Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
24.14Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
24.14Single8S4DCMF-0198S4D-Apelin-CMF-019
24.14Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
24.14Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
24.14Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
24.14Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
24.14Single9B9ZA1AKO9B9Z-CB1-A1AKO
24.14Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
24.14Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
24.14Single9EHSLUF76029EHS-A3A-LUF7602
24.14Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
24.14Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
24.00Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
23.81Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
23.68Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
23.68Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
23.68Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
23.68Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
23.68Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
23.68Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
23.68Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
23.53Single3QAKUK-4320973QAK-A2A-UK-432097
23.53Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
23.53Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
23.53Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
23.53Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
23.53Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
23.53Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
23.53Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
23.33Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
23.33Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
23.33Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
23.33Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
23.33Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
23.33Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
23.33Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
23.33Single8E0GBU728E0G-μ-BU72
23.33Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
23.33Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
23.33Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
23.33Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
23.33Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
23.33Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
23.33Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
23.33Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
23.33Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
23.33Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
23.26Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
23.08Single6IGLIRL16206IGL-ETB-IRL1620
23.08Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
23.08Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
23.08Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
23.08Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
23.08Single8K5BNiacin8K5B-HCA2-Niacin
23.08Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
23.08Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
23.08Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
23.08Consensusbradykinin_onOrthosteric Ligandbk2_on
23.08Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
23.08Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
23.08Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
22.86Single3OE0CVX153OE0-CXCR4-CVX15
22.86Single5WF5UK-4320975WF5-A2A-UK-432097
22.86Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
22.86Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
22.86Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
22.86Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
22.86Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.86Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.86Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.86Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
22.86Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
22.86Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
22.86Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
22.86Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
22.86Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
22.86Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
22.86Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
22.58Single4XEENeurotensin4XEE-NTS1-Neurotensin
22.58Single4XESNeurotensin4XES-NTS1-Neurotensin
22.58Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
22.58Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
22.58Single6A93Risperidone6A93-5-HT2A-Risperidone
22.58Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
22.58Single6YVRNTS8-136YVR-NTS1-NTS8-13
22.58Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
22.58Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
22.58Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
22.58Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
22.58Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
22.58Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
22.58Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
22.58Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
22.58Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
22.58Single8XYIVUF106618XYI-CXCR3-VUF10661
22.58Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
22.58Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
22.58Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
22.58Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
22.58Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
22.58Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
22.58Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
22.58Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
22.58Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
22.58Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
22.58Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
22.58Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
22.58Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
22.50Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
22.50Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
22.22Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
22.22Single4BWBNeurotensin4BWB-NTS1-Neurotensin
22.22Single5U09Taranabant5U09-CB1-Taranabant
22.22Single6AKXA4R6AKX-CCR5-A4R
22.22Single6AKYMaraviroc6AKY-CCR5-Maraviroc
22.22Single6JODAngiotensin II6JOD-AT2-Angiotensin II
22.22Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
22.22Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
22.22Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
22.22Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
22.22Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
22.22Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
22.22Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
22.22Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
22.22Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
22.22Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
22.22Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
22.22Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
22.22Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.22Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
22.22Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
22.22Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
22.22Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
22.22Consensusangiotensin_offOrthosteric Ligandat1_off
22.22Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.22Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.22Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
22.22Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
22.22Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
22.22Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.22Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
22.22Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.22Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
21.95Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
21.95Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
21.95Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
21.88Single4BUONeurotensin4BUO-NTS1-Neurotensin
21.88Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
21.88Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
21.88Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
21.88Single7EZCUKA7EZC-A2A-UKA
21.88Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
21.88Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
21.88Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
21.88Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
21.88Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
21.88Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
21.88Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
21.88Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
21.88Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
21.88Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
21.88Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
21.88Consensuscck_onOrthosteric Ligandccka_on cckb_on
21.88Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
21.88Consensuschemerin_onOrthosteric Ligandcml1_on
21.88Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
21.88Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.88Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.88Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
21.88Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
21.62Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
21.62Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
21.62Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
21.62Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
21.62Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
21.62Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
21.62Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
21.43Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
21.43Single4MBSMaraviroc4MBS-CCR5-Maraviroc
21.43Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
21.43Single7F61PF-036547467F61-H3-PF-03654746
21.43Single7T32ZM-2413857T32-A2A-ZM-241385
21.43Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
21.43Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
21.43Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
21.43Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
21.43Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
21.43Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
21.43Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
21.43Single8K5CAcipimox8K5C-HCA2-Acipimox
21.43Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
21.43Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
21.43Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
21.43Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.43Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
21.43Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
21.43Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
21.43Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
21.43Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
21.43Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
21.43Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
21.43Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
21.43Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
21.43Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
21.43Consensushca_onOrthosteric Ligandhca2_on
21.21Single3NY9ICI118-5513NY9-β2-ICI118-551
21.21Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Single7SK9CCX6627SK9-ACKR3-CCX662
21.21Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
21.21Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
21.21Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
21.21Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
21.21Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
21.21Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
21.21Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
21.21Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
21.21Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
21.21Single9IPYJR14a9IPY-C3aB-JR14a
21.21Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
21.21Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
21.21Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
21.21Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
21.21Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
21.05Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
21.05Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
21.05Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
21.05Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
21.05Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
21.05Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
21.05Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
21.05Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
21.05Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
20.83Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
20.83Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
20.69Single4YAYZD-71554YAY-AT1-ZD-7155
20.69Single5UENDU1725UEN-A1-DU172
20.69Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
20.69Single6PS1Timolol6PS1-β2-Timolol
20.69Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
20.69Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
20.69Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
20.69Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
20.69Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
20.69Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
20.69Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
20.69Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
20.69Single7V3ZCP559407V3Z-CB1-CP55940
20.69Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
20.69Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
20.69Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
20.69Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
20.69Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
20.69Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
20.69Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
20.69Single8K5DGSK2560738K5D-HCA2-GSK256073
20.69Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
20.69Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.69Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.69Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.69Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
20.69Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
20.69Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
20.69Single9CHXS-Carazolol9CHX-β2-S-Carazolol
20.69Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
20.69Consensusa3_onOrthosteric Liganda3a_on
20.69Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
20.69Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
20.69Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
20.69Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
20.59Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
20.59Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.59Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
20.59Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
20.59Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
20.59Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
20.59Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
20.59Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
20.59Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
20.59Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
20.59Single8WDTphotoNECA8WDT-A2A-photoNECA
20.59Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
20.59Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.59Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
20.59Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
20.59Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
20.59Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
20.51Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
20.00Single5N2RPSB-365N2R-A2A-PSB-36-Na
20.00Single5N2SPSB365N2S-A1-PSB36
20.00Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
20.00Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
20.00Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
20.00Single6D26Fevipiprant6D26-DP2-Fevipiprant
20.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
20.00Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
20.00Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
20.00Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
20.00Single7C4SS1P7C4S-S1P3-S1P
20.00Single7C61Ergotamine7C61-5-HT1B-Ergotamine
20.00Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
20.00Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
20.00Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
20.00Single7SK5CXCL127SK5-ACKR3-CXCL12
20.00Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
20.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
20.00Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
20.00Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
20.00Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
20.00Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
20.00Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
20.00Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
20.00Single8JXSPF-61428JXS-D1-PF-6142
20.00Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
20.00Single8QOTNanobody-E8QOT-μ-Nanobody-E
20.00Single8TF5Oleic acid8TF5-GPR6-Oleic acid
20.00Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
20.00Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
20.00Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
20.00Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
20.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
20.00Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
20.00Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
20.00Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
20.00Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
20.00Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
20.00Consensusa3_on_gpOrthosteric Liganda3a_on_gp
20.00Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
20.00Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
20.00Consensusadenosine_offOrthosteric Liganda1_off a2_off
20.00Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
20.00Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
20.00Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
20.00Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
20.00Consensusdp_offOrthosteric Liganddp2_off
20.00Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
20.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
20.00Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
20.00Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
20.00Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
20.00Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
20.00Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.00Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.00Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
20.00Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.00Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
20.00Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Consensustrace-amine_onOrthosteric Ligandta1_on
19.51Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
19.44Single6PT2KGCHM076PT2-δ-KGCHM07
19.44Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
19.44Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
19.44Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
19.44Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
19.44Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
19.35Single2YDVNECA2YDV-A2A-NECA
19.35Single3P0GBI1671073P0G-β2-BI167107
19.35Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
19.35Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
19.35Single4BV0Neurotensin4BV0-NTS1-Neurotensin
19.35Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
19.35Single4UHRCGS216804UHR-A2A-CGS21680
19.35Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
19.35Single5G53NECA5G53-A2A-NECA-Gs
19.35Single5XR8AM8415XR8-CB1-AM841
19.35Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
19.35Single6OS1TRV0266OS1-AT1-TRV026
19.35Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
19.35Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
19.35Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
19.35Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
19.35Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
19.35Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
19.35Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
19.35Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
19.35Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
19.35Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
19.35Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
19.35Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
19.35Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
19.35Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
19.35Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
19.35Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
19.35Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
19.35Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
19.35Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
19.35Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
19.35Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
19.35Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
19.35Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
19.35Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
19.35Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
19.35Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
19.35Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
19.35Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.35Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
19.35Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
19.35Single8ZWFJR14a8ZWF-C3aB-JR14a
19.35Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
19.35Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
19.35Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
19.35Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
19.35Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
19.35Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
19.35Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
19.35Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
19.35Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
19.35Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
19.35Consensuslpa_onOrthosteric Ligandlpa1_on
19.35Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
19.35Consensusneurotensin_onOrthosteric Ligandnts1_on
19.35Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
19.35Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
19.35Consensusrelaxin_onOrthosteric Ligandrxfp4_on
19.35Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
19.35Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.35Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
19.23Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
19.23Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
19.05Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
19.05Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
18.92Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
18.92Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
18.92Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
18.92Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
18.92Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
18.75Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
18.75Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
18.75Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
18.75Single6MXTSalmeterol6MXT-β2-Salmeterol
18.75Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
18.75Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
18.75Single7DFPSpiperone7DFP-D2-Spiperone
18.75Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
18.75Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
18.75Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
18.75Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
18.75Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
18.75Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single7YITNalfurafine7YIT-κ-Nalfurafine
18.75Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
18.75Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
18.75Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
18.75Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
18.75Single8JJ8Formoterol8JJ8-β2-Formoterol
18.75Single8JJLOlodaterol8JJL-β2-Olodaterol
18.75Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
18.75Single8JWY2-1188JWY-A2A-2-118
18.75Single8JWZAB9288JWZ-A2A-AB928-Na
18.75Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
18.75Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
18.75Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
18.75Single9DGIZ85267113509DGI-CB1-Z8526711350
18.75Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
18.75Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
18.75Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
18.75Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
18.75Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
18.75Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
18.75Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
18.75Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
18.75Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
18.75Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
18.75Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
18.75Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
18.75Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
18.75Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
18.75Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
18.75Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
18.75Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
18.75Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
18.75Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
18.75Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
18.75Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
18.75Consensusorexin_onOrthosteric Ligandox2_on
18.75Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
18.52Single3OE9IT1t3OE9-CXCR4-IT1t
18.52Single6LI0C176LI0-GPR52-C17
18.52Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
18.52Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
18.52Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
18.52Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
18.52Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
18.52Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
18.52Single9B9Y7DY9B9Y-CB1-7DY
18.52Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
18.42Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
18.42Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
18.42Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
18.42Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
18.42Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
18.18Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
18.18Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
18.18Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
18.18Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
18.18Single5X93K-87945X93-ETB-K-8794
18.18Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
18.18Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
18.18Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
18.18Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
18.18Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
18.18Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
18.18Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
18.18Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
18.18Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
18.18Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
18.18Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
18.18Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
18.18Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
18.18Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
18.18Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
18.18Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
18.18Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
18.18Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
18.18Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
18.18Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
18.18Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
18.18Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.18Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8XVUCXCL28XVU-CXCR2-CXCL2
18.18Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
18.18Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
18.18Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
18.18Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
18.18Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
18.18Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
18.18Consensusendothelin_offOrthosteric Ligandetb_off
18.18Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
18.18Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
18.18Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
18.18Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
18.18Consensusprostanoid_offOrthosteric Ligandep_off dp_off
18.18Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
18.18Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
18.18Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.95Single7SK3CXCL127SK3-ACKR3-CXCL12
17.95Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
17.95Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
17.86Single3ODUIT1t3ODU-CXCR4-IT1t
17.86Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
17.86Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
17.86Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
17.86Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
17.86Single5ZKQABT-4915ZKQ-PAF-ABT-491
17.86Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
17.86Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
17.86Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
17.86Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
17.86Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
17.86Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
17.86Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
17.86Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
17.86Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
17.86Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
17.86Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
17.86Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
17.86Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
17.86Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
17.86Single8GNGIstradefylline8GNG-A2A-Istradefylline
17.86Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
17.86Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
17.86Single8IWESpermidine8IWE-TA9-Spermidine
17.86Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
17.86Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
17.86Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
17.86Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
17.86Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
17.86Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
17.86Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
17.86Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
17.86Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
17.86Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
17.86Consensusalpha2_offOrthosteric Ligandalpha2c_off
17.86Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
17.65Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
17.65Single5WF6UK-4320975WF6-A2A-UK-432097
17.65Single5ZTYAM102575ZTY-CB2-AM10257
17.65Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
17.65Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
17.65Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
17.65Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
17.65Single6PT3DPI-2876PT3-δ-DPI-287
17.65Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
17.65Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
17.65Single7XN9L-054,5227XN9-SST2-L-054,522
17.65Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
17.65Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
17.65Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
17.65Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
17.65Single8X5YAstemizole8X5Y-H1-Astemizole
17.65Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
17.65Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
17.65Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
17.65Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
17.65Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
17.65Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
17.65Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
17.65Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
17.50Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
17.24Single2YDOAdenosine2YDO-A2A-Adenosine
17.24Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
17.24Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
17.24Single5IU7Q274563465IU7-A2A-Q27456346-Na
17.24Single5IUBQ274563445IUB-A2A-Q27456344-Na
17.24Single5JTBZM-2413855JTB-A2A-ZM-241385
17.24Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
17.24Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
17.24Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
17.24Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
17.24Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
17.24Single6PS0S-Carazolol6PS0-β2-S-Carazolol
17.24Single6PS4ICI118-5516PS4-β2-ICI118-551
17.24Single6PS5S-Propranolol6PS5-β2-S-Propranolol
17.24Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
17.24Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
17.24Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
17.24Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
17.24Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
17.24Single7AROLUF58337ARO-A2A-LUF5833-Na
17.24Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
17.24Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
17.24Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.24Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
17.24Single7UL3Famotidine7UL3-H2-Famotidine
17.24Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
17.24Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
17.24Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
17.24Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
17.24Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
17.24Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
17.24Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
17.24Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
17.24Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
17.24Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
17.24Single8IHKAcifran8IHK-HCA3-Acifran
17.24Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
17.24Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
17.24Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
17.24Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
17.24Single8K2WAMG4878K2W-CXCR3-AMG487
17.24Single8RLNLUF58348RLN-A2A-LUF5834
17.24Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
17.24Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
17.24Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
17.24Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
17.24Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
17.24Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
17.24Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
17.24Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
17.24Single8ZPMAMD0708ZPM-CXCR4-AMD070
17.24Single9AS5Mescaline9AS5-5-HT2A-Mescaline
17.24Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single9BA0A1AKN9BA0-CB1-A1AKN
17.24Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
17.24Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
17.24Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
17.24Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
17.24Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
17.24Consensusa2_offOrthosteric Liganda2a_off
17.24Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
17.24Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
17.24Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
17.24Consensusgrh_offOrthosteric Ligandgnrh1_off
17.24Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
17.14Single4IARErgotamine4IAR-5-HT1B-Ergotamine
17.14Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
17.14Single7F8XNN90567F8X-CCKA-NN9056
17.14Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
17.14Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
17.14Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
17.14Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
17.14Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
17.14Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
17.14Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.14Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
17.14Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
17.14Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
17.07Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.67Single2Y04Salbutamol2Y04-β1-Salbutamol
16.67Single3EMLZM-2413853EML-A2A-ZM-241385
16.67Single3NY8ICI118-5513NY8-β2-ICI118-551
16.67Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
16.67Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
16.67Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
16.67Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
16.67Single4GBRS-Carazolol4GBR-β2-S-Carazolol
16.67Single4QKX35V4QKX-β2-35V
16.67Single5DHHSB-6121115DHH-NOP-SB-612111
16.67Single5IU8Q274563475IU8-A2A-Q27456347-Na
16.67Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
16.67Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
16.67Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
16.67Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
16.67Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
16.67Single5T04Neurotensin5T04-NTS1-Neurotensin
16.67Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
16.67Single6D27CAY104716D27-DP2-CAY10471
16.67Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
16.67Single6GPSMK08126GPS-CCR2-MK0812
16.67Single6H7MSalbutamol6H7M-β1-Salbutamol
16.67Single6HLOAprepitant6HLO-NK1-Aprepitant
16.67Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
16.67Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
16.67Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
16.67Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
16.67Single6S0LZM-2413856S0L-A2A-ZM-241385
16.67Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
16.67Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
16.67Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
16.67Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
16.67Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
16.67Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
16.67Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
16.67Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
16.67Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
16.67Single7PYRPSB-21157PYR-A2A-PSB-2115
16.67Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
16.67Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
16.67Single7UL4Alvimopan7UL4-μ-Alvimopan
16.67Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
16.67Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
16.67Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
16.67Single7WC7Lisuride7WC7-5-HT2A-Lisuride
16.67Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
16.67Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
16.67Single8CU6LJ-45178CU6-A2A-LJ-4517
16.67Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
16.67Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
16.67Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
16.67Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
16.67Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
16.67Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
16.67Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
16.67Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
16.67Single8JJOAlprenolol8JJO-β2-Alprenolol
16.67Single8JXRLSD8JXR-D1-LSD
16.67Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
16.67Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
16.67Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
16.67Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
16.67Single8T1WCVN4248T1W-GPR6-CVN424
16.67Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
16.67Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
16.67Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
16.67Single8X63Mepyramine8X63-H1-Mepyramine
16.67Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
16.67Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
16.67Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
16.67Single9AS1DMT9AS1-5-HT2A-DMT
16.67Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
16.67Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
16.67Single9H37A1IR09H37-A2A-A1IR0-Na
16.67Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
16.67Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
16.67Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
16.67Consensus5ht5_onOrthosteric Ligand5ht5a_on
16.67Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
16.67Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
16.67Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
16.67Consensusdopamine_offOrthosteric Ligandd2_off d3_off
16.67Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
16.67Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
16.67Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
16.67Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
16.67Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
16.67Consensushistamine_offOrthosteric Ligandh1_off
16.67Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
16.67Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
16.67Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
16.22Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
16.22Single6W25SHU91196W25-MC4-SHU9119-Ca
16.22Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
16.22Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
16.22Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
16.22Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single2RH1S-Carazolol2RH1-β2-S-Carazolol
16.13Single2Y03Isoprenaline2Y03-β1-Isoprenaline
16.13Single2YCWS-Carazolol2YCW-β1-S-Carazolol
16.13Single4JKVTaladegib4JKV-SMO-Taladegib
16.13Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
16.13Single5D6LS-Carazolol5D6L-β2-S-Carazolol
16.13Single5IUAQ274563485IUA-A2A-Q27456348-Na
16.13Single5JQHS-Carazolol5JQH-β2-S-Carazolol
16.13Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
16.13Single5TVNLSD5TVN-5-HT2B-LSD
16.13Single5WIUNemonapride5WIU-D4-Nemonapride
16.13Single5WIVNemonapride5WIV-D4-Nemonapride-Na
16.13Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
16.13Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
16.13Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
16.13Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
16.13Single6E67BI1671076E67-β2-BI167107-Gs(CT)
16.13Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
16.13Single6GPXMK08126GPX-CCR2-MK0812
16.13Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
16.13Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
16.13Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
16.13Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
16.13Single6PS6Timolol6PS6-β2-Timolol
16.13Single6S0QZM-2413856S0Q-A2A-ZM-241385
16.13Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
16.13Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
16.13Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
16.13Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
16.13Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
16.13Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
16.13Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
16.13Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
16.13Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
16.13Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
16.13Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
16.13Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
16.13Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
16.13Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
16.13Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.13Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.13Single8GNEKW-63568GNE-A2A-KW-6356-Na
16.13Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
16.13Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
16.13Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
16.13Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
16.13Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
16.13Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
16.13Single8ZMFA1L108ZMF-5-HT2C-A1L10
16.13Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
16.13Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
16.13Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
16.13Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
16.13Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
16.13Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
16.13Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
16.13Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
16.13Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
16.13Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
16.13Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
16.13Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
16.13Consensusamine_offonOrthosteric Ligandamine_off amine_on
16.13Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
16.13Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
16.13Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
16.13Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
16.13Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
16.13Consensusblt_offOrthosteric Ligandblt1_off
16.13Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
16.13Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.13Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
16.13Consensusep_offOrthosteric Ligandep4_off
16.13Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
16.13Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.13Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
16.13Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
16.13Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
16.13Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.13Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
16.13Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
16.13Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
15.79Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
15.79Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
15.79Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
15.62Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
15.62Single4DJHJDTic4DJH-κ-JDTic
15.62Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
15.62Single5D5AS-Carazolol5D5A-β2-S-Carazolol
15.62Single5D5BS-Carazolol5D5B-β2-S-Carazolol
15.62Single5V54Methiothepin5V54-5-HT1B-Methiothepin
15.62Single5V56TC1145V56-SMO-TC114
15.62Single5V57TC1145V57-SMO-TC114
15.62Single5XRAAM115425XRA-CB1-AM11542
15.62Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
15.62Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
15.62Single6H7JIsoprenaline6H7J-β1-Isoprenaline
15.62Single6J21Aprepitant6J21-NK1-Aprepitant
15.62Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
15.62Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
15.62Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
15.62Single6TQ7SB-3348676TQ7-OX1-SB-334867
15.62Single6WGTLSD6WGT-5-HT2A-LSD
15.62Single7B6WCyclazosin7B6W-α1b-Cyclazosin
15.62Single7F1TMIP-1a7F1T-CCR5-MIP-1a
15.62Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
15.62Single7FEECP559407FEE-CB1-CP55940-ZCZ011
15.62Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
15.62Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
15.62Single7PX4PSB-21137PX4-A2A-PSB-2113
15.62Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
15.62Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
15.62Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
15.62Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
15.62Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
15.62Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
15.62Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
15.62Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
15.62Single8EA0Iperoxo8EA0-M3-Iperoxo
15.62Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
15.62Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
15.62Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
15.62Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
15.62Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.62Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
15.62Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
15.62Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
15.62Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
15.62Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
15.62Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
15.62Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
15.62Single9BJKNaloxone9BJK-μ-Naloxone-NAM
15.62Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
15.62Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensus5ht1_offOrthosteric Ligand5ht1b_off
15.62Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
15.62Consensusa2_onOrthosteric Liganda2b_on
15.62Consensusa2_on_gpOrthosteric Liganda2b_on_gp
15.62Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
15.62Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
15.62Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
15.62Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
15.62Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
15.62Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
15.62Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.62Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
15.62Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
15.62Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
15.62Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
15.62Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
15.62Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
15.62Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
15.62Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
15.38Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
15.38Single8A2OTheophylline8A2O-A2A-Theophylline-Na
15.38Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single9CHUNoradrenaline9CHU-β2-Noradrenaline
15.38Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
15.38Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
15.15Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
15.15Single3D4STimolol3D4S-β2-Timolol
15.15Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
15.15Single4AMIBucindolol4AMI-β1-Bucindolol
15.15Single4LDEBI1671074LDE-β2-BI167107
15.15Single4N4WSANT-14N4W-SMO-SANT-1
15.15Single4RWADIPP-NH24RWA-δ-DIPP-NH2
15.15Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
15.15Single6CM4Risperidone6CM4-D2-Risperidone
15.15Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
15.15Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
15.15Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
15.15Single6IIURamatroban6IIU-TXA2-Ramatroban
15.15Single6KQICP559406KQI-CB1-CP55940-Org27569
15.15Single6ZG4HTL00099366ZG4-M1-HTL0009936
15.15Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
15.15Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
15.15Single7K15MKD0467K15-BLT1-MKD046-Na
15.15Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
15.15Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
15.15Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
15.15Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
15.15Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.15Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
15.15Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
15.15Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
15.15Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
15.15Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
15.15Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
15.15Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
15.15Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Single8XWMCXCL68XWM-CXCR2-CXCL6
15.15Single8XWSCXCL58XWS-CXCR2-CXCL5
15.15Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
15.15Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
15.15Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
15.15Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
15.15Consensusalpha1_offOrthosteric Ligandalpha1a_off
15.15Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
15.15Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
15.15Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
15.15Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
15.15Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.15Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.81Single3OE6IT1t3OE6-CXCR4-IT1t
14.81Single4XNWMRS25004XNW-P2Y1-MRS2500
14.81Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
14.81Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
14.81Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
14.81Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
14.81Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
14.81Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
14.81Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
14.81Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
14.81Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
14.81Single9LRCHistamine9LRC-H4-Histamine
14.81Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
14.81Consensus5ht2_onOrthosteric Ligand5ht2b_on
14.81Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
14.81Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
14.81Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
14.71Single5CGDHTL142425CGD-mGlu5-HTL14242
14.71Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
14.71Single6H7LDobutamine6H7L-β1-Dobutamine
14.71Single6IBLArformoterol6IBL-β1-Arformoterol
14.71Single6K1QIRL25006K1Q-ETB-IRL2500
14.71Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
14.71Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
14.71Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single7UM4AS26747237UM4-5-HT5A-AS2674723
14.71Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
14.71Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
14.71Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
14.71Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single8XVJMacitentan8XVJ-ETA-Macitentan
14.71Single8XWFCXCL38XWF-CXCR2-CXCL3
14.71Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
14.71Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
14.71Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
14.71Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
14.71Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
14.71Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
14.63Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
14.63Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
14.63Single9KDFRES-701-39KDF-ETB-RES-701-3
14.29Single4O9RCyclopamine4O9R-SMO-Cyclopamine
14.29Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
14.29Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7SRQLSD7SRQ-5-HT2B-LSD
14.29Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
14.29Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
14.29Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
14.29Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
14.29Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
14.29Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
14.29Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
14.29Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
14.29Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
14.29Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
14.29Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
14.29Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
14.29Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
14.29Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
14.29Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
14.29Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
14.29Single8XQJJN2418XQJ-Apelin-JN241
14.29Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
14.29Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
14.29Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
14.29Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
14.29Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
14.29Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
14.29Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
14.29Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
14.29Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
14.29Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
14.29Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
14.29Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
14.29Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
14.29Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
14.29Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
13.89Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
13.89Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
13.89Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
13.89Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
13.89Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
13.89Single8KIGSHU91198KIG-MC3-SHU9119-Ca
13.89Single8WKYPG-9348WKY-MC4-PG-934
13.89Single8XWNCXCL88XWN-CXCR2-CXCL8
13.89Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
13.89Single9M4TSilodosin9M4T-Alpha1A-Silodosin
13.89Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
13.89Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
13.79Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
13.79Single3PWHZM-2413853PWH-A2A-ZM-241385
13.79Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
13.79Single4QINSAG1.54QIN-SMO-SAG1.5
13.79Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
13.79Single6B73MP11046B73-κ-MP1104
13.79Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
13.79Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
13.79Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
13.79Single6ME2Ramelteon6ME2-MT1-Ramelteon
13.79Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
13.79Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
13.79Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
13.79Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
13.79Single7BR3Elagolix7BR3-GnRH1-Elagolix
13.79Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
13.79Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
13.79Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
13.79Single7F8ULintitript7F8U-CCKA-Lintitript
13.79Single7F8YDevazepide7F8Y-CCKA-Devazepide
13.79Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
13.79Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
13.79Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
13.79Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
13.79Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
13.79Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
13.79Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
13.79Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
13.79Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
13.79Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
13.79Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
13.79Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
13.79Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
13.79Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
13.79Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
13.79Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
13.79Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
13.79Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
13.79Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
13.79Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
13.79Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
13.79Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
13.79Single8Y0HVUF114188Y0H-CXCR3-VUF11418
13.79Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
13.79Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
13.79Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
13.79Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
13.79Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
13.79Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
13.79Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
13.79Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
13.79Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
13.79Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
13.79Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
13.79Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
13.79Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
13.79Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
13.79Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
13.79Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
13.79Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
13.79Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
13.79Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
13.79Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
13.79Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
13.79Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
13.79Consensusorexin_offOrthosteric Ligandox2_off ox1_off
13.79Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
13.79Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
13.51Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
13.51Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
13.51Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
13.51Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
13.51Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
13.33Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
13.33Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
13.33Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
13.33Single4ZJCSB-6740424ZJC-OX1-SB-674042
13.33Single5UVIZM-2413855UVI-A2A-ZM-241385
13.33Single6A94Zotepine6A94-5-HT2A-Zotepine
13.33Single6AQFZM-2413856AQF-A2A-ZM-241385
13.33Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
13.33Single6KUXRS-799486KUX-α2a-RS-79948
13.33Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
13.33Single6MH8ZM-2413856MH8-A2A-ZM-241385
13.33Single6TPGEMPA6TPG-OX2-EMPA
13.33Single6V9SGTPL114036V9S-OX1-GTPL11403
13.33Single6VI4JDTic6VI4-κ-JDTic
13.33Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
13.33Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
13.33Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
13.33Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
13.33Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
13.33Single6ZG9GSK10347026ZG9-M1-GSK1034702
13.33Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
13.33Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
13.33Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
13.33Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
13.33Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
13.33Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
13.33Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
13.33Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
13.33Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
13.33Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
13.33Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
13.33Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
13.33Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
13.33Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
13.33Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
13.33Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.33Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
13.33Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
13.33Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
13.33Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.33Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.33Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
13.33Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
13.33Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8ZPNAMD31008ZPN-CXCR4-AMD3100
13.33Single9AS3LSD9AS3-5-HT2A-LSD
13.33Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
13.33Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
13.33Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
13.33Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
13.33Consensusalpha1_onOrthosteric Ligandalpha1a_on
13.33Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
13.33Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
13.33Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
13.33Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
13.33Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
13.33Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
13.33Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
13.33Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
13.16Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.16Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.16Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
13.16Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
13.16Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
13.16Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.16Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
12.90Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
12.90Single2Y01Dobutamine2Y01-β1-Dobutamine
12.90Single2Y02Carmoterol2Y02-β1-Carmoterol
12.90Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
12.90Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
12.90Single4DAJTiotropium4DAJ-M3-Tiotropium
12.90Single4EJ4Naltrindole4EJ4-δ-Naltrindole
12.90Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
12.90Single4MQSIperoxo4MQS-M2-Iperoxo
12.90Single4U14Tiotropium4U14-M3-Tiotropium
12.90Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
12.90Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
12.90Single5DHGC-355DHG-NOP-C-35
12.90Single5TGZAM65385TGZ-CB1-AM6538
12.90Single5UIGCmpd-15UIG-A2A-Cmpd-1
12.90Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
12.90Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
12.90Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
12.90Single6DRXLisuride6DRX-5-HT2B-Lisuride
12.90Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
12.90Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
12.90Single6TOTLemborexant6TOT-OX1-Lemborexant
12.90Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
12.90Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
12.90Single7BU7BI1671077BU7-β1-BI167107
12.90Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
12.90Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
12.90Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
12.90Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
12.90Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
12.90Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
12.90Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
12.90Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
12.90Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
12.90Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
12.90Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
12.90Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
12.90Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
12.90Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
12.90Single7YXAONO-54306087YXA-S1P5-ONO-5430608
12.90Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
12.90Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
12.90Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
12.90Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
12.90Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
12.90Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
12.90Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
12.90Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
12.90Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
12.90Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
12.90Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
12.90Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
12.90Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
12.90Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
12.90Single8X64Desloratadine8X64-H1-Desloratadine
12.90Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
12.90Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
12.90Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
12.90Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
12.90Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
12.90Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
12.90Single9JEAAtropine9JEA-M1-Atropine
12.90Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
12.90Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
12.90Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
12.90Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
12.90Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
12.90Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
12.90Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
12.90Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
12.90Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
12.90Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
12.90Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
12.90Consensusalpha2_onOrthosteric Ligandalpha2b_on
12.90Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
12.90Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
12.90Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
12.90Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
12.90Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
12.90Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
12.90Consensusblt_onOrthosteric Ligandblt1_on
12.90Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
12.90Consensuscck_offOrthosteric Ligandccka_off
12.90Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
12.90Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
12.90Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
12.90Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
12.90Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
12.90Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
12.90Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
12.90Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
12.90Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
12.90Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
12.90Consensusleukotriene_onOrthosteric Ligandblt_on
12.90Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
12.90Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
12.90Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
12.90Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
12.82Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
12.82Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
12.82Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
12.50Single2Y00Dobutamine2Y00-β1-Dobutamine
12.50Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
12.50Single5CGCHTL142425CGC-mGlu5-HTL14242
12.50Single5WQCEMPA5WQC-OX2-EMPA
12.50Single5XPRBosentan5XPR-ETB-Bosentan
12.50Single6LUQHaloperidol6LUQ-D2-Haloperidol
12.50Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
12.50Single6TP6Filorexant6TP6-OX1-Filorexant
12.50Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
12.50Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
12.50Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
12.50Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
12.50Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
12.50Single7W41PD1762527W41-BB2-PD176252
12.50Single7WC6LSD7WC6-5-HT2A-LSD
12.50Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
12.50Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
12.50Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
12.50Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
12.50Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
12.50Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
12.50Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
12.50Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
12.50Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
12.50Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
12.50Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.50Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.50Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
12.50Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
12.50Consensusbombesin_offOrthosteric Ligandbb2_off
12.50Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
12.50Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
12.50Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
12.50Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
12.12Single4U15Tiotropium4U15-M3-Tiotropium
12.12Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
12.12Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
12.12Single6J20Aprepitant6J20-NK1-Aprepitant
12.12Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
12.12Single6OL9Tiotropium6OL9-M5-Tiotropium
12.12Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
12.12Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
12.12Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
12.12Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
12.12Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
12.12Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
12.12Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
12.12Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
12.12Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
12.12Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
12.12Single9AS9RS130-1809AS9-5-HT2A-RS130-180
12.12Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
12.12Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
12.12Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.12Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
12.12Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
12.12Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
12.12Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
12.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
11.76Single5CXVTiotropium5CXV-M1-Tiotropium
11.76Single5X33BIIL2605X33-BLT1-BIIL260
11.76Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
11.76Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
11.76Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
11.76Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
11.76Single8XQJJN2418XQJ-Apelin-JN241
11.76Single8XWACXCL18XWA-CXCR2-CXCL1
11.76Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
11.76Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
11.76Single9BJKNAM9BJK-μ-Naloxone-NAM
11.76Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
11.76Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
11.76Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
11.76Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
11.54Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
11.54Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
11.54Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
11.54Single8HS2Fab0468HS2-GPR20-Fab046
11.54Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
11.54Single8PWNTheophylline8PWN-A2A-Theophylline
11.54Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.54Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.43Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
11.43Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
11.43Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
11.43Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.43Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.43Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
11.43Single8ZPLHF511168ZPL-CXCR4-HF51116
11.43Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single3OE8IT1t3OE8-CXCR4-IT1t
11.11Single3RFMCaffeine3RFM-A2A-Caffeine
11.11Single6KNMJN241-96KNM-Apelin-JN241-9
11.11Single6TQ9SB-4081246TQ9-OX1-SB-408124
11.11Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
11.11Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
11.11Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
11.11Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
11.11Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
11.11Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
11.11Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
11.11Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
11.11Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
11.11Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
11.11Single9JF4PD1683689JF4-BB1-PD168368
11.11Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
11.11Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
11.11Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
11.11Consensuskisspeptin_onOrthosteric Ligandkiss1_on
11.11Consensusp2y_offOrthosteric Ligandp2y1_off
10.81Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
10.81Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.81Single8IEBA1LYA8IEB-GPR156-A1LYA
10.81Single8IEIA1LYA8IEI-GPR156-A1LYA
10.81Single8IEPA1LYA8IEP-GPR156-A1LYA
10.81Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.81Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
10.81Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.81Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
10.81Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.81Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.81Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
10.71Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
10.71Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
10.71Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
10.71Single6ME5Agomelatine6ME5-MT1-Agomelatine
10.71Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
10.71Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
10.71Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
10.71Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
10.71Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
10.71Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
10.71Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
10.71Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
10.71Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
10.71Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
10.71Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
10.71Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
10.53Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.53Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
10.53Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
10.34Single3PBLEticlopride3PBL-D3-Eticlopride
10.34Single5L7IVismodegib5L7I-SMO-Vismodegib
10.34Single6HLLCP999946HLL-NK1-CP99994
10.34Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
10.34Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
10.34Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.34Single7UL2SR486927UL2-NTS1-SR48692-Na
10.34Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
10.34Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
10.34Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
10.34Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
10.34Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
10.34Single9AS7Psilocin9AS7-5-HT2A-Psilocin
10.34Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
10.34Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
10.34Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
10.34Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
10.34Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
10.34Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.34Consensusneurotensin_offOrthosteric Ligandnts1_off
10.34Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
10.00Single4S0VSuvorexant4S0V-OX2-Suvorexant
10.00Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
10.00Single5WS3EMPA5WS3-OX2-EMPA
10.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
10.00Single6ME9Ramelteon6ME9-MT2-Ramelteon
10.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
10.00Single6TODEMPA6TOD-OX1-EMPA-Na
10.00Single6TPJSuvorexant6TPJ-OX2-Suvorexant
10.00Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
10.00Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
10.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
10.00Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
10.00Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
10.00Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
10.00Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
10.00Single7XRRLemborexant7XRR-OX2-Lemborexant
10.00Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
10.00Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
10.00Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
10.00Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
10.00Single9H2XA1IR19H2X-A2A-A1IR1-Na
10.00Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
10.00Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
10.00Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
10.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.00Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
10.00Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
9.68Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
9.68Single3REYXAC3REY-A2A-XAC
9.68Single3RZECidoxepin3RZE-H1-Cidoxepin
9.68Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
9.68Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
9.68Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
9.68Single6IQLL7458706IQL-D4-L745870
9.68Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
9.68Single6TP3Nemorexant6TP3-OX1-Nemorexant
9.68Single6TPNHTL66416TPN-OX2-HTL6641
9.68Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
9.68Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
9.68Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
9.68Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
9.68Single7VV6C48/807VV6-MRGPRX2-C48/80
9.68Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
9.68Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
9.68Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.68Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
9.68Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
9.68Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
9.68Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
9.68Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
9.68Single9ARXSerotonin9ARX-5-HT2A-Serotonin
9.68Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
9.68Consensusopsins_offOrthosteric Ligandrhodopsin_off
9.68Consensussensory_offOrthosteric Ligandopsins_off
9.38Single4QIMANTA XV4QIM-SMO-ANTA XV
9.38Single5DSGTiotropium5DSG-M4-Tiotropium
9.38Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
9.38Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
9.38Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
9.38Single6IIVDaltroban6IIV-TXA2-Daltroban
9.38Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
9.38Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Single7F83PF-051904577F83-Ghrelin-PF-05190457
9.38Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
9.38Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
9.38Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
9.38Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
9.38Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
9.38Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
9.38Single9IYAONO-97105319IYA-GPR55-ONO-9710531
9.38Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
9.09Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
9.09Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
9.09Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
9.09Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
9.09Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
9.09Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
9.09Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
9.09Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
9.09Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
9.09Single7SINNPS-21437SIN-CaS-NPS-2143
9.09Single7SINNPS-21437SIN-CaS-NPS-2143
9.09Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
9.09Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
9.09Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
9.09Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
9.09Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
9.09Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
9.09Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
9.09Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
9.09Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
9.09Single9HAPTolvaptan9HAP-V2-Tolvaptan
9.09Single9HC04YI9HC0-mGlu5-4YI
9.09Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
8.82Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
8.82Single5TZRMK86665TZR-FFA1-MK8666
8.82Single6E59L-7607356E59-NK1-L-760735
8.82Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
8.82Single7P2L4YI7P2L-mGlu5-4YI
8.82Single7R0CAVP7R0C-V2-AVP-Arrestin2
8.82Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
8.82Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
8.82Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
8.82Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
8.82Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
8.82Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
8.82Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
8.82Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
8.82Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
8.82Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
8.82Single8XVLZibotentan8XVL-ETA-Zibotentan
8.82Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
8.82Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
8.82Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
8.82Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
8.82Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
8.82Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
8.82Consensustachykinin_offOrthosteric Ligandnk1_off
8.57Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
8.57Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
8.57Single4PY02MeSATP4PY0-P2Y12-2MeSATP
8.57Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
8.57Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
8.57Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
8.57Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
8.33Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
8.33Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
8.33Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
8.11Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
8.11Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
7.89Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.89Single8IEIA1LYA8IEI-GPR156-A1LYA
7.89Single8IEPA1LYA8IEP-GPR156-A1LYA
7.89Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.89Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.69Single5MZPCaffeine5MZP-A2A-Caffeine-Na
7.69Single8IEBA1LYA8IEB-GPR156-A1LYA
7.69Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single7WC4Serotonin7WC4-5-HT2A-Serotonin
7.14Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
7.14Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
7.14Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.14Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
7.14Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
7.14Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
7.14Consensussensory_onOrthosteric Ligandopsins_on
6.90Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
6.90Single3UZAGTPL92363UZA-A2A-GTPL9236
6.90Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
6.90Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
6.90Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
6.90Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
6.90Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
6.90Single7WC5Psilocin7WC5-5-HT2A-Psilocin
6.90Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.90Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
6.90Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
6.90Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
6.90Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
6.90Single8JPSCCL78JPS-ACKR1-CCL7
6.90Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
6.90Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
6.90Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
6.90Consensusgi_sensoryOrthosteric Ligandgi_opsins
6.90Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
6.90Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
6.90Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
6.90Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
6.90Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
6.67Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
6.67Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
6.67Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
6.67Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
6.67Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
6.67Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
6.67Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
6.67Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
6.67Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
6.67Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
6.67Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
6.67Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
6.67Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
6.67Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
6.67Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
6.67Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
6.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
6.67Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.67Consensusgq_nucleotideOrthosteric Ligandgq_p2y
6.67Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
6.45Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
6.45Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
6.45Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
6.45Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
6.45Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
6.45Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
6.45Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
6.45Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
6.45Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
6.45Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
6.45Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.45Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.45Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
6.45Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
6.45Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
6.45Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.45Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
6.45Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.45Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.45Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
6.45Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
6.45Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.45Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.45Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
6.45Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
6.25Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
6.25Single6FFIMMPEP6FFI-mGlu5-MMPEP
6.25Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
6.25Single6TPKRetosiban6TPK-OT-Retosiban
6.25Single7VODCariprazine7VOD-5-HT2A-Cariprazine
6.25Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
6.25Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
6.25Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
6.25Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
6.25Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.25Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
6.25Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
6.25Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
6.25Consensusvasop-oxy_offOrthosteric Ligandot_off
6.06Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
6.06Single6FFHFenobam6FFH-mGlu5-Fenobam
6.06Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
6.06Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.06Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
6.06Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
5.88Single4NTJAZD12834NTJ-P2Y12-AZD1283
5.88Single6HLPNetupitant6HLP-NK1-Netupitant
5.88Single6Z4SSR486926Z4S-NTS1-SR48692
5.88Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
5.88Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.88Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
5.88Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
5.88Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
5.88Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
5.71Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.71Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.56Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
5.56Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.56Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.56Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.56Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.41Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
5.41Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
5.26Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
5.26Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
5.13Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
4.17Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.17Single6D35Cholesterol6D35-SMO-Cholesterol
4.17Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.17Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.17Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.17Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.17Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
4.17Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.17Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.17Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
4.17Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.17Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
4.17Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.17Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.17Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.17Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.17Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.17Single7DTTCa7DTT-CaS-Ca-Ca
4.17Single7DTTCa7DTT-CaS-Ca-Ca
4.17Single7DTUTryptophan7DTU-CaS-Tryptophan
4.17Single7DTUTryptophan7DTU-CaS-Tryptophan
4.17Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.17Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.17Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.17Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.17Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.17Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.17Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.17Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.17Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.17Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.17Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.17Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.17Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.17Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.17Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.17Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.17Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.17Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.17Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.17Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.17Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.17Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.17Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.17Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.17Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.17Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.17Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.17Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.17Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.17Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.17Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.17Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
4.17Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.17Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.17Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.17Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.17Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.17Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.17Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.17Single7XW7K1-707XW7-TSH-K1-70
4.17Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.17Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.17Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.17Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.17Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.17Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.17Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.17Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.17Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.17Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.17Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.17Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.17Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.17Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.17Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.17Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.17Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.17Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.17Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.17Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.17Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.17Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.17Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.17Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.17Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.17Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.17Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.17Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.17Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.17Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.17Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.17Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.17Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.17Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.17Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.17Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.17Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.17Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.17Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.17Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.17Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.17Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.17Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.17Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.17Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.17Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.17Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.17Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.17Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.17Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.17Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.17Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.17Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.17Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.17Single8WVXNorrin8WVX-LGR4-Norrin
4.17Single8WVYNorrin8WVY-LGR4-Norrin
4.17Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.17Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.17Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.17Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.17Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.17Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.17Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.17Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.17Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.17Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.17Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.17Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.17Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.17Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.17Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.17Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.17Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.17Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.17Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.17Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.17Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.17Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.17Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.17Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.17Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.17Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.17Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.17Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.17Single9KHHNorrin9KHH-LGR4-Norrin
4.17Single9S37NB219S37-LGR4-NB21
4.17Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.00Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.00Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.00Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.00Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.00Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
3.85Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
3.85Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
3.85Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
3.70Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
3.70Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
3.70Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
3.70Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
3.70Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.57Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
3.57Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
3.57Single5L7DCholesterol5L7D-SMO-Cholesterol
3.57Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.57Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.45Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
3.45Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
3.33Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
3.33Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
3.33Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.23Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
3.23Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
3.23Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
3.23Single6TP4ACT-4622066TP4-OX1-ACT-462206
3.23Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.23Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
3.23Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.23Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
3.12Single4K5YCP-3763954K5Y-CRF1-CP-376395
3.12Single4XNVBPTU4XNV-P2Y1-BPTU
3.12Single6C1QNDT95137276C1Q-C5a1-PMX53-NDT9513727
3.12Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
3.03Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
3.03Single6ZINSR486926ZIN-NTS1-SR48692
3.03Single8IYXYL-3658IYX-GPR34-YL-365
3.03Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.03Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
2.94Single4Z9GCP-3763954Z9G-CRF1-CP-376395
2.94Single8GTIBMK-C2058GTI-CRF1-BMK-C205
2.86Single8GTGBMK-I1528GTG-CRF1-BMK-I152
2.78Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
2.70Single8GTMBMK-C2038GTM-CRF1-BMK-C203
2.63Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
2.50Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.50Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.38Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.38Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.33Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.17Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
vpac_on_gp vpac1_on_gp
vpac2_on_gp
pac_on_gp pac1_on_gp
Net Summary
Imin 3.355
Number of Linked Nodes 874
Number of Links 1016
Number of Hubs 151
Number of Links mediated by Hubs 583
Number of Communities 24
Number of Nodes involved in Communities 183
Number of Links involved in Communities 259
Path Summary
Number Of Nodes in MetaPath 122
Number Of Links MetaPath 121
Number of Shortest Paths 1174337
Length Of Smallest Path 3
Average Path Length 31.3461
Length of Longest Path 69
Minimum Path Strength 0.5775
Average Path Strength 6.90162
Maximum Path Strength 41.5917
Minimum Path Correlation 0.7
Average Path Correlation 0.985609
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.66667
Average % Of Corr. Nodes 50.5025
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 48.8083
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
class-b1_on_gpglucagon_on_gp
vip-pacap_on_gp
pth_on_gp
crf_on_gp
calcitonin_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download vip-pacap_on_gp.zip



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You can also  read or  download a guide explaining the meaning of all files and numerical data.