Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 2.30583603
2G.HN.37 2.96712402
3G.HN.52 1.19519404
4G.S1.02 6.09423454
5G.S1.05 5.62894409
6G.S1.06 3.58106458
7G.S2.08 7.42096455
8G.S3.01 4.96856454
9G.S3.03 7.90962557
10G.S3.04 8.33019416
11G.S3.05 3.53238556
12G.S3.06 7.879516
13G.S3.07 3.4624459
14G.s3h2.03 5.22315519
15G.H2.04 4.42327409
16G.H2.06 5.92775719
17G.H2.07 5.45814619
18G.h2s4.01 7.96663419
19G.s4h3.02 4.99288409
20G.s4h3.03 5.56014158
21G.s4h3.04 5.15104798
22G.H3.09 5.91742779
23G.H3.13 4.02442475
24G.H3.17 7.51564614
25G.H3.18 6.33038419
26G.S5.05 4.00064689
27G.S5.07 4.13375489
28G.HG.04 5.37223598
29G.hgh4.02 5.261327168
30G.hgh4.05 8.85317406
31G.H4.03 7.40933403
32G.H4.10 8.99264166
33G.H4.12 7.23413475
34G.H4.15 5.04048478
35G.h4s6.02 5.30404477
36G.h4s6.11 4.48106478
37G.S6.02 8.05125408
38G.S6.04 8.81923488
39G.s6h5.01 5.97779489
40G.H5.08 5.72836458
41G.H5.15 3.32875408
42G.H5.20 3.39962408
43G.H5.26 7.01173405
44b.1x4 1.58238508
45b.h2x1 3.48529405
46b.lhb1x6 3.822625133
47b.lhb1x9 3.61673403
48b.b1x4 4.81635447
49b.b1x6 8.11519449
50b.l1x3 8.79808649
51b.b2x1 9.06915518
52b.b2x5 6.97546507
53b.b3x3 4.32942468
54b.l3x2 5.62808549
55b.b4x2 5.58442408
56b.b4x3 5.75183467
57b.b4x4 9.08067448
58b.b4x5 4.62029467
59b.b4x6 8.98857749
60b.b5x2 6.16231407
61b.b5x3 7.01692649
62b.b5x5 5.78125465
63b.b5x7 5.72788407
64b.l5x1 4.35815568
65b.l5x5 8.05719
66b.b6x5 4.0526866
67b.l6x5 6.571544144
68b.b7x1 5.899545144
69b.l7x2 4.74135419
70b.l7x4 3.71971409
71b.b8x3 4.31404406
72b.b8x4 5.15123566
73b.l8x1 4.03683465
74b.l8x3 3.58433403
75b.l9x3 7.692519
76b.l9x6 5.91668818
77b.b10x5 4.98859609
78b.b11x2 4.67971407
79b.l11x2 8.49692419
80b.b12x3 3.62106438
81b.b12x6 8.08841718
82b.b12x7 5.80173439
83b.b13x7 8.25661537
84b.l13x3 9.01815539
85b.l13x6 5.95106419
86b.l13x7 4.77279439
87b.b14x3 4.80269405
88b.b15x1 7.43654539
89b.b15x3 4.8051439
90b.l15x2 6.66942439
91b.b16x4 9.19331536
92b.b16x5 4.46769405
93b.b16x6 9.937538
94b.b17x5 7.19952417
95b.b17x7 9.23615418
96b.l17x3 8.3189719
97b.l17x6 7.486519
98b.b18x3 5.42625418
99b.b18x5 5.69192405
100b.l18x1 5.262268116
101b.l18x3 5.861544115
102b.b19x2 8.39662516
103b.b19x4 6.12135418
104b.l19x2 6.39946519
105b.b20x2 6.10519416
106b.b20x4 10.4531518
107b.b20x6 7.93408516
108b.b20x7 4.3601409
109b.l20x2 4.91854509
110b.b21x1 6.91585517
111b.b21x2 3.32394406
112b.b21x5 6.13462404
113b.b21x7 5.58192605
114b.l22x5 5.548656139
115b.b23x1 4.45635405
116b.b23x6 6.8794717
117b.l23x1 7.99894416
118b.b24x4 7.40577416
119b.b24x6 6.10452418
120b.l24x2 4.24279406
121b.l25x3 8.825395109
122b.l25x4 3.41962405
123b.l25x6 11.9926418
124b.b27x1 2.90048406
125b.l27x1 11.1443719
126b.l27x2 8.281834109
127b.b28x3 4.89029447
128b.b28x4 8.625394106
129b.b28x6 8.890925109
130g.h1x11 2.6049409
131g.l1x4 4508
132g.h2x11 9.514524116
133g.ctx3 6.66087409
134g.ctx4 3.95221407
135g.ctx6 3.819746136
136g.ctx15 7.04125449
137g.ctx16 5.37956748
138Lig 19.64972420
139NT 9.20163423
1401x29 1.75038404
1411x35 3.68317405
1421x39 4.79721408
1432x42 5.70538607
1442x46 5.159044129
1452x50 6.015925129
1462x53 5.38692506
147E1x50 7.96212628
148E1x52 6.46408507
1493x33 4.52654425
1503x37 4.26087407
1513x50 7.0475409
1524x54 3.0125404
153E2 13.51631524
1545x35 3.59446522
1555x50 3.32885409
1565x58 7.52398629
1575x64 3.02769405
1586x44 5.033529
1596x48 7.36185529
1606x51 5.39215527
1616x59 4.22923405
162E3 4.47269504
1637x26 2.08067401
1647x42 4.87592507
1657x49 5.463086129
1667x53 5.300456129
1677x55 2.29269406
1688x50 3.4351408
169G.H1.08 4.22029450
170I2x57 7.641634190
171g.ntx4 0.860673400
172I1 5.67400
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.l2x3 b.l2x5 18.70583.75308NoNo085
2b.b3x1 b.l2x3 18.64445.95308NoNo058
3b.b3x1 b.b6x5 18.63654.19308NoYes056
4b.b3x2 b.b4x6 80.14676.26192NoYes059
5b.b2x5 b.b3x2 80.22738.40808YesNo075
6b.b2x3 b.b2x5 86.13215.05731NoYes067
7b.b26x2 b.b2x3 86.18485.91923NoNo076
8b.b26x1 b.b26x2 86.2143.24154NoNo097
9b.b26x1 b.l27x1 86.24565.03538NoYes099
10b.b2x1 b.l27x1 49.69149.53462YesYes189
11b.b2x1 b.l3x1 49.70916.8669YesNo189
12b.l3x1 b.l5x5 49.80196.53154NoYes199
13b.l1x3 b.l3x2 88.35756.15462YesYes499
14b.l1x4 b.l3x2 1003.70731NoYes069
15I1 b.l1x4 99.72464.23YesNo006
168x48 I1 96.40848.155NoYes050
177x56 8x48 96.28714.135NoNo075
187x56 8x47 96.00533.03846NoNo078
198x47 8x50 95.86423.01NoYes088
207x54 8x50 93.76833.57308NoYes068
212x43 7x54 93.33493.82538NoNo086
222x43 7x53 93.192.65038NoYes089
233x46 7x53 44.88775.92423NoYes099
242x42 3x46 44.6894.48115YesNo079
252x42 3x49 21.44478.77923YesNo078
263x49 I2x57 21.01410.1519NoYes1980
273x53 I2x57 41.60624.53885NoYes080
283x53 G.H5.19 40.74355.84346NoNo088
29G.H5.15 G.H5.19 40.31192.66808YesNo088
30G.H5.11 G.H5.15 38.58332.71615NoYes088
31b.b4x6 b.l1x3 87.17633.62YesYes499
322x38 2x42 21.22474.56038NoYes067
332x38 I2x57 21.01419.80462NoYes060
34G.H5.11 G.S3.03 32.85654.28269NoYes587
35G.S1.04 G.S3.03 20.69925.24808NoYes077
36G.S1.04 G.S4.03 15.51385.49NoNo077
37G.h2s4.01 b.l5x5 16.327511.7204YesYes199
38G.H3.17 b.l27x1 29.9953.35308YesYes149
39G.H3.15 G.H3.17 36.13177.48154NoYes184
40G.S4.03 G.S5.05 15.07263.52692NoYes079
41b.l5x5 b.l7x2 32.61056.30808YesYes199
42G.s3h2.03 b.l7x2 16.64494.195YesYes199
433x50 7x53 13.60416.845YesYes099
44G.H2.04 G.H2.07 23.21226YesYes099
45G.H2.04 G.H2.08 35.43973.80538YesNo098
46G.H2.08 G.H3.15 35.40443.37846NoNo188
47G.H2.07 b.l7x2 15.98164.51077YesYes199
48G.H2.07 G.h2s4.01 16.63873.855YesYes199
49G.H2.07 b.l9x6 53.99713.67346YesYes198
50G.s3h2.03 b.l9x6 15.8526.50269YesYes198
51G.H2.06 b.l9x6 51.39093.39654YesYes198
52G.H2.04 G.H3.08 20.28884.94615YesNo099
53G.H2.06 b.l17x6 49.29099.35962YesYes199
54G.H3.08 G.S4.04 20.18685.89962NoNo099
55G.H3.09 G.S4.04 20.082614.1812YesNo099
56G.H3.06 G.hgh4.02 13.38034.92846NoYes078
57b.b2x4 b.b6x5 29.03913.14423NoYes066
58b.b10x4 b.b2x4 28.802416.9238NoNo066
59b.b10x2 b.b10x4 28.56684.28654NoNo066
60b.b10x2 b.b14x3 28.33115.49462NoYes065
61b.b14x3 b.b15x1 25.14254.215YesYes059
62b.b15x1 b.b16x6 20.219314.8023YesYes398
63b.b16x4 b.b16x6 10.07687.89692YesYes368
64g.h1x11 g.h1x14 18.19971.17577YesNo099
65b.1x11 g.h1x11 16.70675.27269NoYes089
66b.1x11 g.h1x12 12.71683.14538NoNo086
67b.1x7 g.h1x12 10.21681.76538NoNo086
68b.l17x5 b.l17x6 48.68644.305NoYes169
69b.l17x5 b.l19x2 48.36522.26346NoYes169
70b.l17x3 b.l19x2 32.6225.76731YesYes199
71b.b19x4 b.l17x3 17.23028.00077YesYes189
72b.b19x4 b.b20x6 12.90337.48154YesYes186
73b.b17x7 b.b20x6 35.444111.1696YesYes186
74b.b17x7 b.b21x1 17.13934.36462YesYes187
75b.b20x4 b.l17x3 13.976517.1831YesYes189
76b.b20x4 b.b20x6 25.78984.68885YesYes186
77b.b20x2 b.l19x2 14.68637.78192YesYes169
78b.b20x2 b.b20x4 13.97297.41231YesYes168
79b.l2x5 b.l4x2 19.218528.0981NoNo054
80b.l26x5 g.ctx15 16.45077.73923NoYes059
81b.l26x5 g.ctx4 28.74576.775NoYes057
82g.ctx3 g.ctx4 27.30643.59154YesYes097
83g.ctx3 g.ctx6 19.37797.87731YesYes096
84b.b23x1 b.lhb1x9 11.47164.88731YesYes053
85b.lhb1x11 b.lhb1x9 17.42263.58808NoYes043
86b.b25x7 b.lhb1x11 16.90626.46769NoNo074
87b.l4x2 g.ctx16 14.47796.90269NoYes448
88b.b25x7 b.b28x6 18.470218.3108NoYes079
89b.b1x6 b.b4x6 12.558817.3442YesYes499
90b.b1x6 b.b28x5 12.12854.28231YesNo495
91b.b2x5 b.l4x1 15.65556.27038YesNo075
92b.l4x1 g.ctx16 15.52783.70692NoYes058
93b.b2x5 b.l26x1 12.981811.1515YesNo077
94b.l26x1 b.l26x3 12.67357.11808NoNo1877
95b.l26x3 b.l26x5 12.59455.33231NoNo075
96b.b4x2 b.b5x8 20.63863.41308YesNo085
97b.b5x7 b.b5x8 20.30313.39YesNo075
98b.l11x1 b.l9x6 16.98058.24577NoYes198
99b.b11x6 b.l11x1 16.63323.42538NoNo199
100b.b11x6 b.l9x3 14.049515.2877NoYes199
101b.b12x6 b.l9x3 12.96764.31154YesYes189
102b.b17x5 b.b17x7 17.25729.91038YesYes178
103b.b16x5 b.b17x5 15.22765.73YesYes057
104b.b16x5 b.b17x4 11.96772.66192YesNo055
1057x49 7x53 39.3853.80385YesYes1299
1067x45 7x49 26.92013.32962NoYes099
1076x48 7x45 26.513212.57YesNo099
1083x36 6x48 25.50615.80577NoYes279
1093x36 Lig 25.42053.74154NoYes270
1102x50 7x49 10.17598.28539YesYes1299
111b.b4x2 b.l3x2 18.10717.18154YesYes089
112b.b28x5 g.ctx16 11.98115.16846NoYes458
113g.ctx15 g.ctx16 11.77733.94231YesYes498
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
7x34Lig4.294622NoYes5010
LigNT20.48042YesYes0301
E2Lig23.80152YesYes4010
E2x51Lig17.89272NoYes3010
NTNT6.833082YesYes3311
2x533x328.336150YesNo6721
2x533x363.498460YesNo6721
2x537x425.300770YesYes6722
2x63E1x509.075772NoYes5822
E1x49E26.091150NoYes4421
E1x50E23.558462YesYes8421
3x22E24.357692NoYes4421
3x334x574.443082YesNo5612
3x334x614.306542YesNo5411
3x374x573.198080YesNo7622
4x614x653.239622NoNo4512
4x64E215.22082NoYes4421
4x645x354.727312NoYes4222
4x65E2x527.0150NoNo5521
E2E248.37152YesYes4411
E2E2x5110.83732YesNo4311
E2E2x528.623852YesNo4511
5x35E25.7052YesYes2421
5x36E210.92732NoYes4411
5x39E25.947692NoYes5421
5x32E23.908460NoYes2421
6x516x524.708082YesNo7812
6x517x373.519622YesNo7612
6x517x384.081542YesNo7611
6x547x346.627310NoNo5521
6x61E34.982NoYes4412
7x387x423.891922NoYes6712
2x60Lig9.230382NoYes6010
2x63E24.257312NoYes5421
3x32Lig8.213462NoYes7010
3x335x434.010772YesNo5511
3x33Lig5.345772YesYes5010
3x366x485.805772NoYes7912
3x36Lig3.741542NoYes7010
3x375x435.346540YesNo7521
E2x52Lig4.554232NoYes5010
5x36Lig3.6652NoYes4010
5x43Lig5.754622NoYes5010
6x516x559.535772YesNo7612
6x51Lig5.115772YesYes7010
6x587x305.039622NoNo4411
6x58Lig9.306542NoYes4010
7x27Lig3.291540NoYes4010
7x30Lig6.775382NoYes4010
7x38Lig5.742692NoYes6010
2x602x633.608082NoNo6512
6x61Lig8.150772NoYes4010
5x366x593.793852NoYes4512
4x61Lig3.367312NoYes4010
E1Lig4.642NoYes0010
7x31Lig3.129622NoYes5010
2x67E22.7652NoYes4421
7x24NT2.660NoYes7321
2x64E120NoNo5021
7x317x321.836152NoNo5212
1x28Lig1.808850NoYes4010
6x62Lig1.278080NoYes5010
1x247x310.9269230NoNo0521

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
90.91Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
75.00Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
75.00Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
69.57Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
69.57Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
69.57Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
69.23Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
65.38Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
64.29Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
64.29Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
64.29Consensusbradykinin_onOrthosteric Ligandbk2_on
64.29Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
64.29Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
64.00Consensusangiotensin_onOrthosteric Ligandat1_on
64.00Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
62.50Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
61.54Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
61.54Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
61.54Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
61.54Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
60.87Consensuschemerin_onOrthosteric Ligandcml1_on
60.71Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
60.71Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
60.71Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
60.00Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
60.00Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
57.14Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
56.52Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
56.52Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
55.56Single6JODAngiotensin II6JOD-AT2-Angiotensin II
55.56Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
55.56Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
55.17Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
55.17Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
53.85Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
53.85Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
53.85Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
53.57Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
53.57Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
53.57Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
53.57Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
53.33Single8IY6Endothelin-18IY6-ETB-Endothelin-1
53.33Consensusendothelin_onOrthosteric Ligandetb_on eta_on
52.00Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
52.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
51.85Single3OE0CVX153OE0-CXCR4-CVX15
51.85Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
51.61Single5GLHEndothelin-15GLH-ETB-Endothelin-1
51.61Single6IGKEndothelin-36IGK-ETB-Endothelin-3
51.61Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
51.61Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
51.61Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
50.00Single6OS2TRV0266OS2-AT1-TRV026
50.00Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
50.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
50.00Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
50.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
50.00Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
50.00Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
48.48Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
48.39Single6IGLIRL16206IGL-ETB-IRL1620
48.39Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
48.28Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
48.28Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
48.28Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
48.28Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
48.28Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
48.28Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
48.28Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
48.15Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
48.15Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
48.15Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
48.00Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
48.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
47.06Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
46.88Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
46.67Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
46.67Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
46.67Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
46.43Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
46.43Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
46.43Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
46.43Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
46.43Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
46.43Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
46.43Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
46.43Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
45.83Single6OS1TRV0266OS1-AT1-TRV026
45.16Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
45.16Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
45.16Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
45.16Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
45.16Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
44.83Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
44.83Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
44.83Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
44.44Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
44.44Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
44.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
44.00Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
44.00Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
44.00Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
44.00Single8XWSCXCL58XWS-CXCR2-CXCL5
43.48Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
43.48Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
43.33Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
43.33Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
43.33Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
43.33Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
43.33Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
43.33Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
43.33Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.86Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
42.86Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
42.86Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
42.86Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
42.86Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
42.42Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
42.31Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
42.31Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
42.31Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
41.94Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
41.94Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
41.67Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
41.67Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
41.67Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
41.67Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
41.38Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.38Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
41.38Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
41.38Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
41.38Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
41.38Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
41.18Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
40.74Single6KNMJN241-96KNM-Apelin-JN241-9
40.74Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
40.74Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
40.74Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
40.74Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
40.74Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
40.74Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
40.74Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
40.74Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
40.74Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
40.74Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
40.62Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
40.00Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
40.00Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
40.00Single7F1TMIP-1a7F1T-CCR5-MIP-1a
40.00Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
40.00Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
40.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
40.00Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
40.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
40.00Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
40.00Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
40.00Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
40.00Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
40.00Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
40.00Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
40.00Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
40.00Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
40.00Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
40.00Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
40.00Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
40.00Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
40.00Consensusvasop-oxy_onOrthosteric Ligandv2_on
40.00Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
39.39Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
39.39Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
39.29Single4IARErgotamine4IAR-5-HT1B-Ergotamine
39.29Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
39.29Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
39.29Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
39.29Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
39.29Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
39.29Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
39.29Single8WDTphotoNECA8WDT-A2A-photoNECA
39.29Single8XWNCXCL88XWN-CXCR2-CXCL8
39.29Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
39.29Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
39.29Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
39.13Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
39.13Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
38.71Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.71Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
38.71Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
38.71Single8ZRTET-18ZRT-ETB-ET-1
38.71Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
38.46Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
38.46Single6MXTSalmeterol6MXT-β2-Salmeterol
38.46Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
38.46Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
38.46Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
38.46Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
38.46Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
38.46Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
38.46Single8XWACXCL18XWA-CXCR2-CXCL1
38.46Single8XWMCXCL68XWM-CXCR2-CXCL6
38.46Consensusorexin_onOrthosteric Ligandox2_on
38.24Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
37.93Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
37.93Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
37.93Single7XNACYN1548067XNA-SST2-CYN154806
37.93Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
37.93Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
37.93Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
37.93Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
37.93Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
37.93Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
37.93Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
37.93Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
37.93Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
37.50Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
37.50Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
37.50Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
37.50Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
37.50Single7SK3CXCL127SK3-ACKR3-CXCL12
37.50Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
37.50Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
37.50Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
37.50Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
37.50Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
37.50Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
37.50Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
37.50Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
37.14Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
37.14Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
37.04Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
37.04Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
37.04Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
37.04Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
37.04Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
37.04Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
37.04Single8XVUCXCL28XVU-CXCR2-CXCL2
37.04Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
37.04Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
37.04Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
36.67Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
36.67Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
36.67Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
36.67Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
36.67Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
36.36Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
36.00Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
36.00Single5C1MBU725C1M-μ-BU72
36.00Single6D26Fevipiprant6D26-DP2-Fevipiprant
36.00Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
36.00Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
36.00Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
36.00Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.00Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
36.00Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
36.00Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
36.00Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
36.00Consensusdp_offOrthosteric Liganddp2_off
35.71Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
35.71Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
35.71Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
35.71Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
35.71Single7XN9L-054,5227XN9-SST2-L-054,522
35.71Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
35.71Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
35.71Single8XQJJN2418XQJ-Apelin-JN241
35.71Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
35.48Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
35.48Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
35.48Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
35.48Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
35.48Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
35.48Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
35.48Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
35.29Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
35.29Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Single6AKYMaraviroc6AKY-CCR5-Maraviroc
34.78Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
34.78Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
34.78Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GNGIstradefylline8GNG-A2A-Istradefylline
34.78Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
34.78Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
34.62Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
34.62Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
34.62Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
34.62Single8E0GBU728E0G-μ-BU72
34.62Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
34.62Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
34.62Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
34.62Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
34.62Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
34.62Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
34.62Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
34.62Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
34.62Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
34.62Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
34.62Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
34.48Single4XT1Fractalkine4XT1-US28-Fractalkine
34.48Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
34.48Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
34.48Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
34.48Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
34.48Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
34.48Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.48Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
34.48Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
34.48Consensuslpl_onOrthosteric Ligands1p_on lpa_on
34.48Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
34.48Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
34.48Consensussomatostatin_offOrthosteric Ligandsst2_off
34.38Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
34.38Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
34.38Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
34.38Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
34.38Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
34.38Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
34.29Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.29Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
34.29Consensusbombesin_onOrthosteric Ligandbb2_on
34.29Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
34.29Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
33.33Single3QAKUK-4320973QAK-A2A-UK-432097
33.33Single4MBSMaraviroc4MBS-CCR5-Maraviroc
33.33Single4RWADIPP-NH24RWA-δ-DIPP-NH2
33.33Single4XEENeurotensin4XEE-NTS1-Neurotensin
33.33Single4XESNeurotensin4XES-NTS1-Neurotensin
33.33Single4XT3Fractalkine4XT3-US28-Fractalkine
33.33Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
33.33Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
33.33Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
33.33Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
33.33Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
33.33Single6YVRNTS8-136YVR-NTS1-NTS8-13
33.33Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
33.33Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
33.33Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
33.33Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
33.33Single7SK5CXCL127SK5-ACKR3-CXCL12
33.33Single7UL3Famotidine7UL3-H2-Famotidine
33.33Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
33.33Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
33.33Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
33.33Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
33.33Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
33.33Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8JJLOlodaterol8JJL-β2-Olodaterol
33.33Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
33.33Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
33.33Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
33.33Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
33.33Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8XQJJN2418XQJ-Apelin-JN241
33.33Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
33.33Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
33.33Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
33.33Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
33.33Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
33.33Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
33.33Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
33.33Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
33.33Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
33.33Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
33.33Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
33.33Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
33.33Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
33.33Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
33.33Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
33.33Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
33.33Consensuslpa_offOrthosteric Ligandlpa1_off
33.33Consensuslpl_offOrthosteric Ligands1p_off lpa_off
33.33Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
33.33Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
33.33Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
32.50Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
32.35Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
32.35Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
32.35Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
32.35Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
32.35Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
32.26Single5WF5UK-4320975WF5-A2A-UK-432097
32.26Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
32.26Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
32.26Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
32.26Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
32.26Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
32.26Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
32.26Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
32.26Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
32.26Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
32.26Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
32.14Single4BUONeurotensin4BUO-NTS1-Neurotensin
32.14Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
32.14Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
32.14Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
32.14Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
32.14Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
32.14Single6IBLArformoterol6IBL-β1-Arformoterol
32.14Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
32.14Single7EZCUKA7EZC-A2A-UKA
32.14Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
32.14Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
32.14Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
32.14Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
32.14Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
32.14Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
32.14Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
32.14Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
32.14Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
32.14Single8XWFCXCL38XWF-CXCR2-CXCL3
32.14Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
32.14Consensuscck_onOrthosteric Ligandccka_on cckb_on
32.14Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
32.14Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.14Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.14Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
32.14Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
32.14Consensusprostanoid_offOrthosteric Ligandep_off dp_off
32.00Single6D27CAY104716D27-DP2-CAY10471
32.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
32.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
32.00Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
32.00Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
32.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
32.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
32.00Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
32.00Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
32.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
32.00Single9CHXS-Carazolol9CHX-β2-S-Carazolol
32.00Consensusa3_onOrthosteric Liganda3a_on
32.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
32.00Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
32.00Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
32.00Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
32.00Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
32.00Consensushca_on_gpOrthosteric Ligandhca2_on_gp
31.82Single6ME5Agomelatine6ME5-MT1-Agomelatine
31.82Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.43Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
31.43Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
31.43Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
31.25Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
31.25Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
31.25Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
31.25Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.03Single3NY9ICI118-5513NY9-β2-ICI118-551
31.03Single4UG2CGS216804UG2-A2A-CGS21680
31.03Single5WF6UK-4320975WF6-A2A-UK-432097
31.03Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
31.03Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
31.03Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
31.03Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
31.03Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
31.03Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
31.03Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
31.03Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
31.03Single8QJ2pN1628QJ2-MC4-pN162-Gs
31.03Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
31.03Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
31.03Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
31.03Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
31.03Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
30.77Single7C61Ergotamine7C61-5-HT1B-Ergotamine
30.77Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
30.77Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
30.77Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
30.77Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
30.77Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
30.77Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
30.77Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
30.77Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
30.77Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
30.77Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
30.77Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
30.77Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
30.77Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.77Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
30.77Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
30.77Single8JXSPF-61428JXS-D1-PF-6142
30.77Single8S4DCMF-0198S4D-Apelin-CMF-019
30.77Single8TF5Oleic acid8TF5-GPR6-Oleic acid
30.77Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.77Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.77Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
30.77Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
30.77Consensusa3_on_gpOrthosteric Liganda3a_on_gp
30.77Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
30.77Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
30.77Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
30.77Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
30.77Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
30.77Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
30.77Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
30.77Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
30.77Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
30.77Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
30.77Consensustrace-amine_onOrthosteric Ligandta1_on
30.56Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
30.43Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
30.43Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
30.30Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
30.30Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
30.30Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
30.30Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
30.30Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
30.30Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
30.00Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
30.00Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
30.00Single7F8XNN90567F8X-CCKA-NN9056
30.00Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
30.00Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
30.00Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
30.00Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
30.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
30.00Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
30.00Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
30.00Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
30.00Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
30.00Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
30.00Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
30.00Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
29.73Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
29.73Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
29.73Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
29.63Single2YDVNECA2YDV-A2A-NECA
29.63Single3P0GBI1671073P0G-β2-BI167107
29.63Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
29.63Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
29.63Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
29.63Single4UHRCGS216804UHR-A2A-CGS21680
29.63Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
29.63Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
29.63Single5G53NECA5G53-A2A-NECA-Gs
29.63Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
29.63Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
29.63Single6J21Aprepitant6J21-NK1-Aprepitant
29.63Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
29.63Single6WGTLSD6WGT-5-HT2A-LSD
29.63Single7B6WCyclazosin7B6W-α1b-Cyclazosin
29.63Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
29.63Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
29.63Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
29.63Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
29.63Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
29.63Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
29.63Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
29.63Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
29.63Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
29.63Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
29.63Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
29.63Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
29.63Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
29.63Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
29.63Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
29.63Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
29.63Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
29.63Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
29.63Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
29.63Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
29.63Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
29.63Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
29.63Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensusneurotensin_onOrthosteric Ligandnts1_on
29.63Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
29.63Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.63Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
29.41Single6FJ3PTH6FJ3-PTH1-PTH
29.41Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
29.41Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
29.41Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
29.41Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
29.41Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
29.17Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
29.17Single4BWBNeurotensin4BWB-NTS1-Neurotensin
29.17Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
29.17Single6AKXA4R6AKX-CCR5-A4R
29.17Single6ME2Ramelteon6ME2-MT1-Ramelteon
29.17Single6ME9Ramelteon6ME9-MT2-Ramelteon
29.17Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
29.17Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
29.17Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
29.17Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
29.17Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.17Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
29.17Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
29.17Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
29.17Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
29.17Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
29.17Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
29.17Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
29.17Single8IWESpermidine8IWE-TA9-Spermidine
29.17Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
29.17Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
29.17Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
29.17Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
29.17Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
29.17Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
29.17Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
29.17Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
29.17Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
29.17Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
29.17Consensusorexin_offOrthosteric Ligandox2_off ox1_off
29.17Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
29.03Single6HLOAprepitant6HLO-NK1-Aprepitant
29.03Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
29.03Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
29.03Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
29.03Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
29.03Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
29.03Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
29.03Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
29.03Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
29.03Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
29.03Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
28.95Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
28.95Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
28.57Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
28.57Single4AMIBucindolol4AMI-β1-Bucindolol
28.57Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
28.57Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
28.57Single6A93Risperidone6A93-5-HT2A-Risperidone
28.57Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
28.57Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
28.57Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
28.57Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
28.57Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
28.57Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
28.57Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
28.57Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
28.57Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
28.57Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
28.57Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single7YITNalfurafine7YIT-κ-Nalfurafine
28.57Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
28.57Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
28.57Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
28.57Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
28.57Single8JJ8Formoterol8JJ8-β2-Formoterol
28.57Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
28.57Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
28.57Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
28.57Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
28.57Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
28.57Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
28.57Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
28.57Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
28.57Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
28.57Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
28.57Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
28.57Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
28.57Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
28.57Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
28.57Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
28.57Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
28.57Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
28.57Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
28.57Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
28.57Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
28.57Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
28.57Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
28.57Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
28.21Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
28.21Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
28.12Single6PT2KGCHM076PT2-δ-KGCHM07
28.12Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
28.12Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.12Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
28.12Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.12Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
28.12Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
28.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
28.00Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
28.00Single6KUXRS-799486KUX-α2a-RS-79948
28.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
28.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
28.00Single6PS4ICI118-5516PS4-β2-ICI118-551
28.00Single6PS5S-Propranolol6PS5-β2-S-Propranolol
28.00Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
28.00Single7AROLUF58337ARO-A2A-LUF5833-Na
28.00Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
28.00Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.00Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
28.00Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
28.00Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
28.00Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
28.00Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
28.00Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
28.00Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
28.00Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
28.00Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
28.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
28.00Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
28.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
28.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
28.00Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
28.00Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
28.00Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
28.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
28.00Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
28.00Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
28.00Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
28.00Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.00Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
28.00Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
28.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
28.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
28.00Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
28.00Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
28.00Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
28.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
28.00Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
28.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
28.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
28.00Consensushca_onOrthosteric Ligandhca2_on
28.00Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
27.78Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
27.78Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
27.78Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
27.78Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
27.78Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
27.78Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
27.78Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
27.78Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
27.59Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
27.59Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
27.59Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
27.59Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
27.59Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
27.59Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
27.59Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.59Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
27.59Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
27.59Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
27.59Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.59Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
27.59Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
27.59Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
27.59Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
27.59Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.59Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
27.59Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
27.59Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
27.59Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
27.59Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
27.59Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
27.59Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
27.59Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
27.27Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
27.27Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
27.27Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
27.27Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
27.27Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
27.27Consensusp2y_offOrthosteric Ligandp2y1_off
27.27Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
27.03Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
26.92Single2Y02Carmoterol2Y02-β1-Carmoterol
26.92Single2Y04Salbutamol2Y04-β1-Salbutamol
26.92Single3NY8ICI118-5513NY8-β2-ICI118-551
26.92Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
26.92Single4EJ4Naltrindole4EJ4-δ-Naltrindole
26.92Single4GBRS-Carazolol4GBR-β2-S-Carazolol
26.92Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
26.92Single4QKX35V4QKX-β2-35V
26.92Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
26.92Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
26.92Single6H7MSalbutamol6H7M-β1-Salbutamol
26.92Single6PS1Timolol6PS1-β2-Timolol
26.92Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
26.92Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
26.92Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
26.92Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
26.92Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
26.92Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
26.92Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
26.92Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
26.92Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
26.92Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
26.92Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
26.92Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
26.92Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
26.92Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
26.92Single7UL4Alvimopan7UL4-μ-Alvimopan
26.92Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
26.92Single7V3ZCP559407V3Z-CB1-CP55940
26.92Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
26.92Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
26.92Single7WC7Lisuride7WC7-5-HT2A-Lisuride
26.92Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
26.92Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
26.92Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
26.92Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
26.92Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
26.92Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
26.92Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
26.92Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
26.92Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
26.92Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
26.92Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
26.92Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
26.92Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
26.92Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
26.92Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
26.92Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
26.92Single8JXRLSD8JXR-D1-LSD
26.92Single8K5DGSK2560738K5D-HCA2-GSK256073
26.92Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
26.92Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
26.92Single8T1WCVN4248T1W-GPR6-CVN424
26.92Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
26.92Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.92Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
26.92Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
26.92Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
26.92Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
26.92Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
26.92Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
26.92Consensus5ht5_onOrthosteric Ligand5ht5a_on
26.92Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
26.92Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
26.92Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
26.92Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
26.92Consensusdopamine_offOrthosteric Ligandd2_off d3_off
26.92Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
26.92Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
26.92Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
26.92Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
26.92Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
26.92Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
26.67Single5ZTYAM102575ZTY-CB2-AM10257
26.67Single6PT3DPI-2876PT3-δ-DPI-287
26.67Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
26.67Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
26.67Single7SK9CCX6627SK9-ACKR3-CCX662
26.67Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
26.67Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
26.67Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
26.67Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
26.67Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
26.67Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
26.47Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
26.47Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
26.47Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
26.47Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
26.47Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
26.32Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
26.09Single4XNWMRS25004XNW-P2Y1-MRS2500
26.09Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
26.09Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
26.09Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
26.09Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
26.09Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
26.09Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
25.93Single2RH1S-Carazolol2RH1-β2-S-Carazolol
25.93Single2Y03Isoprenaline2Y03-β1-Isoprenaline
25.93Single2YCWS-Carazolol2YCW-β1-S-Carazolol
25.93Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
25.93Single5D6LS-Carazolol5D6L-β2-S-Carazolol
25.93Single5JQHS-Carazolol5JQH-β2-S-Carazolol
25.93Single5N2RPSB-365N2R-A2A-PSB-36-Na
25.93Single5N2SPSB365N2S-A1-PSB36
25.93Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
25.93Single5TVNLSD5TVN-5-HT2B-LSD
25.93Single5WIUNemonapride5WIU-D4-Nemonapride
25.93Single5WIVNemonapride5WIV-D4-Nemonapride-Na
25.93Single5WQCEMPA5WQC-OX2-EMPA
25.93Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
25.93Single6E67BI1671076E67-β2-BI167107-Gs (fused)
25.93Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
25.93Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
25.93Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
25.93Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
25.93Single6TP6Filorexant6TP6-OX1-Filorexant
25.93Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
25.93Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
25.93Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
25.93Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
25.93Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
25.93Single7W41PD1762527W41-BB2-PD176252
25.93Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
25.93Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.93Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
25.93Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.93Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.93Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
25.93Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
25.93Single8QOTNanobody-E8QOT-μ-Nanobody-E
25.93Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
25.93Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
25.93Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
25.93Single8ZMFA1L108ZMF-5-HT2C-A1L10
25.93Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
25.93Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
25.93Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
25.93Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
25.93Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
25.93Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
25.93Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
25.93Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
25.93Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
25.93Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
25.93Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
25.93Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
25.93Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
25.93Consensusamine_offonOrthosteric Ligandamine_off amine_on
25.93Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
25.93Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
25.93Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
25.93Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
25.93Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
25.93Consensusbombesin_offOrthosteric Ligandbb2_off
25.93Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.93Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
25.93Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
25.93Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
25.93Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.93Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.81Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
25.81Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
25.81Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
25.81Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
25.81Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
25.81Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
25.81Single8WKYPG-9348WKY-MC4-PG-934
25.81Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
25.81Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
25.71Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
25.71Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
25.71Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
25.64Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
25.64Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
25.64Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single3OE9IT1t3OE9-CXCR4-IT1t
25.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
25.00Single4BV0Neurotensin4BV0-NTS1-Neurotensin
25.00Single5D5AS-Carazolol5D5A-β2-S-Carazolol
25.00Single5D5BS-Carazolol5D5B-β2-S-Carazolol
25.00Single5XR8AM8415XR8-CB1-AM841
25.00Single6H7JIsoprenaline6H7J-β1-Isoprenaline
25.00Single6HLLCP999946HLL-NK1-CP99994
25.00Single6J20Aprepitant6J20-NK1-Aprepitant
25.00Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
25.00Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
25.00Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
25.00Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
25.00Single6TQ7SB-3348676TQ7-OX1-SB-334867
25.00Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
25.00Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
25.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
25.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
25.00Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
25.00Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
25.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
25.00Single7PX4PSB-21137PX4-A2A-PSB-2113
25.00Single7R0CAVP7R0C-V2-AVP-Arrestin2
25.00Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
25.00Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
25.00Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
25.00Single7TUYGSK682753A7TUY-GPR183-GSK682753A
25.00Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
25.00Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
25.00Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
25.00Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
25.00Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
25.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
25.00Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
25.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
25.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
25.00Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
25.00Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
25.00Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
25.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
25.00Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
25.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
25.00Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
25.00Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
25.00Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
25.00Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
25.00Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
25.00Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
25.00Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
25.00Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
25.00Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
25.00Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
25.00Single8K5BNiacin8K5B-HCA2-Niacin
25.00Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
25.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
25.00Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
25.00Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
25.00Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
25.00Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
25.00Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
25.00Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
25.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
25.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
25.00Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
25.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
25.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
25.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
25.00Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
25.00Consensusa2_onOrthosteric Liganda2b_on
25.00Consensusa2_on_gpOrthosteric Liganda2b_on_gp
25.00Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
25.00Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
25.00Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
25.00Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
25.00Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
25.00Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
25.00Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
25.00Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
25.00Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.00Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
25.00Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
25.00Consensuslpa_onOrthosteric Ligandlpa1_on
25.00Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
25.00Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
25.00Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
25.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
25.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
25.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
25.00Consensustachykinin_offOrthosteric Ligandnk1_off
24.39Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
24.32Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
24.32Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
24.24Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
24.24Single6W25SHU91196W25-MC4-SHU9119-Ca
24.24Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
24.24Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
24.24Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
24.14Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
24.14Single3D4STimolol3D4S-β2-Timolol
24.14Single4LDEBI1671074LDE-β2-BI167107
24.14Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
24.14Single4PY02MeSATP4PY0-P2Y12-2MeSATP
24.14Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
24.14Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
24.14Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
24.14Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
24.14Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
24.14Single7DFPSpiperone7DFP-D2-Spiperone
24.14Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
24.14Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
24.14Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
24.14Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
24.14Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
24.14Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
24.14Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
24.14Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
24.14Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
24.14Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.14Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
24.14Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
24.14Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
24.14Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
24.14Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
24.14Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
24.14Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
24.14Single8XYIVUF106618XYI-CXCR3-VUF10661
24.14Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
24.14Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
24.14Consensusalpha1_offOrthosteric Ligandalpha1a_off
24.14Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
24.14Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
24.14Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.14Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
24.00Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
24.00Single5WS3EMPA5WS3-OX2-EMPA
24.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
24.00Single6TODEMPA6TOD-OX1-EMPA-Na
24.00Single7BR3Elagolix7BR3-GnRH1-Elagolix
24.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
24.00Single7F8ULintitript7F8U-CCKA-Lintitript
24.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
24.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
24.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
24.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
24.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
24.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
24.00Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
24.00Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
24.00Single7XRRLemborexant7XRR-OX2-Lemborexant
24.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
24.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
24.00Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
24.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
24.00Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
24.00Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
24.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
24.00Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
24.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
24.00Consensusangiotensin_offOrthosteric Ligandat1_off
24.00Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
24.00Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
24.00Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
24.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
24.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
23.68Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
23.68Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
23.53Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
23.53Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
23.53Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
23.53Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
23.53Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
23.33Single5X93K-87945X93-ETB-K-8794
23.33Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
23.33Single6H7LDobutamine6H7L-β1-Dobutamine
23.33Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
23.33Single7UM4AS26747237UM4-5-HT5A-AS2674723
23.33Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
23.33Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
23.33Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
23.33Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
23.33Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
23.33Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
23.33Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
23.33Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
23.33Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
23.33Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
23.33Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
23.33Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
23.33Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
23.33Consensusendothelin_offOrthosteric Ligandetb_off
23.33Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
23.33Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single2YDOAdenosine2YDO-A2A-Adenosine
23.08Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
23.08Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
23.08Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
23.08Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
23.08Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
23.08Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
23.08Single6A94Zotepine6A94-5-HT2A-Zotepine
23.08Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
23.08Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
23.08Single6TPGEMPA6TPG-OX2-EMPA
23.08Single6TPNHTL66416TPN-OX2-HTL6641
23.08Single6V9SGTPL114036V9S-OX1-GTPL11403
23.08Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
23.08Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
23.08Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
23.08Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
23.08Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
23.08Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
23.08Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
23.08Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
23.08Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single7T32ZM-2413857T32-A2A-ZM-241385
23.08Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
23.08Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
23.08Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
23.08Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
23.08Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
23.08Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
23.08Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single8IHKAcifran8IHK-HCA3-Acifran
23.08Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
23.08Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
23.08Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
23.08Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
23.08Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
23.08Single8K5CAcipimox8K5C-HCA2-Acipimox
23.08Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
23.08Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
23.08Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
23.08Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
23.08Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
23.08Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
23.08Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
23.08Consensusalpha1_onOrthosteric Ligandalpha1a_on
23.08Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
23.08Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
23.08Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
23.08Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
23.08Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
23.08Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
23.08Consensusgrh_offOrthosteric Ligandgnrh1_off
22.86Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
22.86Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
22.73Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
22.73Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
22.58Single5EE7MK08935EE7-Glucagon-MK0893
22.58Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
22.58Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
22.58Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
22.58Single8X5YAstemizole8X5Y-H1-Astemizole
22.50Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
22.22Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
22.22Single2Y01Dobutamine2Y01-β1-Dobutamine
22.22Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
22.22Single3EMLZM-2413853EML-A2A-ZM-241385
22.22Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
22.22Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
22.22Single4QIMANTA XV4QIM-SMO-ANTA XV
22.22Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
22.22Single4YAYZD-71554YAY-AT1-ZD-7155
22.22Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
22.22Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
22.22Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
22.22Single5T04Neurotensin5T04-NTS1-Neurotensin
22.22Single5UENDU1725UEN-A1-DU172
22.22Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
22.22Single6DRXLisuride6DRX-5-HT2B-Lisuride
22.22Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
22.22Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
22.22Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
22.22Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
22.22Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
22.22Single6S0LZM-2413856S0L-A2A-ZM-241385
22.22Single6TOTLemborexant6TOT-OX1-Lemborexant
22.22Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
22.22Single7BU7BI1671077BU7-β1-BI167107
22.22Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
22.22Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
22.22Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
22.22Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
22.22Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
22.22Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
22.22Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
22.22Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
22.22Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
22.22Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.22Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
22.22Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
22.22Single8CU6LJ-45178CU6-A2A-LJ-4517
22.22Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
22.22Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
22.22Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
22.22Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
22.22Single8JJOAlprenolol8JJO-β2-Alprenolol
22.22Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
22.22Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
22.22Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
22.22Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
22.22Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
22.22Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
22.22Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
22.22Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
22.22Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
22.22Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
22.22Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
22.22Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
22.22Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
22.22Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
22.22Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
22.22Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
22.22Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Consensusblt_onOrthosteric Ligandblt1_on
22.22Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
22.22Consensuscck_offOrthosteric Ligandccka_off
22.22Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
22.22Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.22Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.22Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
22.22Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Consensusleukotriene_onOrthosteric Ligandblt_on
22.22Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
21.95Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.88Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
21.88Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
21.88Single8IEBA1LYA8IEB-GPR156-A1LYA
21.88Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
21.74Single6TQ9SB-4081246TQ9-OX1-SB-408124
21.74Single8A2OTheophylline8A2O-A2A-Theophylline-Na
21.74Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
21.74Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
21.74Single9CHUNoradrenaline9CHU-β2-Noradrenaline
21.74Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
21.74Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
21.62Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
21.62Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
21.43Single2Y00Dobutamine2Y00-β1-Dobutamine
21.43Single5IUAQ274563485IUA-A2A-Q27456348-Na
21.43Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
21.43Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
21.43Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
21.43Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
21.43Single6PS6Timolol6PS6-β2-Timolol
21.43Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
21.43Single6S0QZM-2413856S0Q-A2A-ZM-241385
21.43Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
21.43Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
21.43Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
21.43Single6Z4SSR486926Z4S-NTS1-SR48692
21.43Single7C4SS1P7C4S-S1P3-S1P
21.43Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
21.43Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
21.43Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
21.43Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
21.43Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
21.43Single7WC6LSD7WC6-5-HT2A-LSD
21.43Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
21.43Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
21.43Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
21.43Single8GNEKW-63568GNE-A2A-KW-6356-Na
21.43Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
21.43Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
21.43Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
21.43Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
21.43Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
21.43Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
21.43Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
21.43Consensusadenosine_offOrthosteric Liganda1_off a2_off
21.43Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
21.43Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
21.43Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
21.43Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
21.21Single8IEBA1LYA8IEB-GPR156-A1LYA
21.21Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
21.21Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
21.05Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
21.05Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
20.83Single3OE6IT1t3OE6-CXCR4-IT1t
20.83Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
20.83Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
20.83Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
20.83Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
20.83Single7V6A-7V6A-M4-PubChem 9864275-Gi1/β1/γ2
20.83Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.83Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
20.83Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
20.83Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
20.83Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
20.83Single8JPSCCL78JPS-ACKR1-CCL7
20.83Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
20.83Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
20.83Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
20.83Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
20.83Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
20.83Consensus5ht2_onOrthosteric Ligand5ht2b_on
20.83Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
20.83Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
20.83Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
20.69Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
20.69Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
20.69Single4DJHJDTic4DJH-κ-JDTic
20.69Single4U15Tiotropium4U15-M3-Tiotropium
20.69Single5TZRMK86665TZR-FFA1-MK8666
20.69Single5V54Methiothepin5V54-5-HT1B-Methiothepin
20.69Single5XRAAM115425XRA-CB1-AM11542
20.69Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
20.69Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
20.69Single6E59L-7607356E59-NK1-L-760735
20.69Single6OL9Tiotropium6OL9-M5-Tiotropium
20.69Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
20.69Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
20.69Single7FEECP559407FEE-CB1-CP55940-ZCZ011
20.69Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
20.69Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
20.69Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
20.69Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
20.69Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
20.69Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
20.69Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.69Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
20.69Consensus5ht1_offOrthosteric Ligand5ht1b_off
20.69Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
20.69Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
20.69Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
20.69Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
20.69Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.69Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
20.69Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
20.69Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
20.69Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
20.69Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
20.59Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
20.59Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
20.59Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
20.51Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
20.00Single3PBLEticlopride3PBL-D3-Eticlopride
20.00Single4O9RCyclopamine4O9R-SMO-Cyclopamine
20.00Single5CXVTiotropium5CXV-M1-Tiotropium
20.00Single6CM4Risperidone6CM4-D2-Risperidone
20.00Single6KQICP559406KQI-CB1-CP55940-Org27569
20.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
20.00Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
20.00Single6ZG4HTL00099366ZG4-M1-HTL0009936
20.00Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
20.00Single7K15MKD0467K15-BLT1-MKD046-Na
20.00Single7SRQLSD7SRQ-5-HT2B-LSD
20.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
20.00Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
20.00Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
20.00Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
20.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
20.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
20.00Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
20.00Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
20.00Single8JWY2-1188JWY-A2A-2-118
20.00Single8JWZAB9288JWZ-A2A-AB928-Na
20.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
20.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
20.00Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
20.00Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
20.00Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
20.00Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
20.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
20.00Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
20.00Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
20.00Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
20.00Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
20.00Single9B9Y7DY9B9Y-CB1-7DY
20.00Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
20.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
20.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
20.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
20.00Consensusgq_nucleotideOrthosteric Ligandgq_p2y
20.00Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
20.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
20.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
20.00Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
20.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
19.57Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
19.44Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
19.44Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
19.44Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
19.35Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
19.35Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
19.35Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
19.35Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
19.23Single3ODUIT1t3ODU-CXCR4-IT1t
19.23Single3PWHZM-2413853PWH-A2A-ZM-241385
19.23Single4QINSAG1.54QIN-SMO-SAG1.5
19.23Single4S0VSuvorexant4S0V-OX2-Suvorexant
19.23Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
19.23Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
19.23Single5ZKQABT-4915ZKQ-PAF-ABT-491
19.23Single6B73MP11046B73-κ-MP1104
19.23Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
19.23Single6DS0Ly2660976DS0-5-HT2B-Ly266097
19.23Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
19.23Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
19.23Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
19.23Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
19.23Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
19.23Single6TPJSuvorexant6TPJ-OX2-Suvorexant
19.23Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
19.23Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
19.23Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
19.23Single7F8YDevazepide7F8Y-CCKA-Devazepide
19.23Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
19.23Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
19.23Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.23Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.23Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
19.23Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
19.23Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
19.23Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
19.23Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
19.23Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
19.23Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
19.23Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
19.23Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
19.23Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
19.23Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
19.23Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
19.23Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
19.23Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
19.23Single8Y0HVUF114188Y0H-CXCR3-VUF11418
19.23Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.23Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
19.23Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
19.23Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
19.23Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
19.23Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.23Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
19.23Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
19.23Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
19.23Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
19.23Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.23Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.23Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
19.23Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
19.23Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
19.23Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
19.23Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.23Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.05Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
19.05Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
18.92Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
18.92Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
18.75Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
18.75Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
18.75Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.75Consensuskisspeptin_onOrthosteric Ligandkiss1_on
18.52Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
18.52Single3REYXAC3REY-A2A-XAC
18.52Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
18.52Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
18.52Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
18.52Single5IU7Q274563465IU7-A2A-Q27456346-Na
18.52Single5IUBQ274563445IUB-A2A-Q27456344-Na
18.52Single5JTBZM-2413855JTB-A2A-ZM-241385
18.52Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
18.52Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
18.52Single5UVIZM-2413855UVI-A2A-ZM-241385
18.52Single6AQFZM-2413856AQF-A2A-ZM-241385
18.52Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
18.52Single6TP3Nemorexant6TP3-OX1-Nemorexant
18.52Single6VI4JDTic6VI4-κ-JDTic
18.52Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
18.52Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
18.52Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
18.52Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
18.52Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
18.52Single6ZINSR486926ZIN-NTS1-SR48692
18.52Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
18.52Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
18.52Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
18.52Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
18.52Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
18.52Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
18.52Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
18.52Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
18.52Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
18.52Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
18.52Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
18.52Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
18.52Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
18.52Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
18.52Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
18.52Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
18.52Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
18.52Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
18.52Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
18.52Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
18.52Single9BJKNaloxone9BJK-μ-Naloxone-NAM
18.52Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
18.52Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
18.52Consensusa2_offOrthosteric Liganda2a_off
18.52Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
18.52Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
18.42Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
18.42Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
18.18Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
18.18Single7QA8Peptide7QA8-STE2-Peptide
18.18Single7QA8Peptide7QA8-STE2-Peptide
18.18Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
18.18Single8IEIA1LYA8IEI-GPR156-A1LYA
18.18Single8IEPA1LYA8IEP-GPR156-A1LYA
18.18Single8IEPA1LYA8IEP-GPR156-A1LYA
18.18Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
18.18Single8KIGSHU91198KIG-MC3-SHU9119-Ca
18.18Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
18.18Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.18Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.18Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.18Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
17.95Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
17.95Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
17.95Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
17.86Single4DAJTiotropium4DAJ-M3-Tiotropium
17.86Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
17.86Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
17.86Single4MQSIperoxo4MQS-M2-Iperoxo
17.86Single4U14Tiotropium4U14-M3-Tiotropium
17.86Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
17.86Single5DHHSB-6121115DHH-NOP-SB-612111
17.86Single5IU8Q274563475IU8-A2A-Q27456347-Na
17.86Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
17.86Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
17.86Single5TGZAM65385TGZ-CB1-AM6538
17.86Single5UIGCmpd-15UIG-A2A-Cmpd-1
17.86Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
17.86Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
17.86Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
17.86Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
17.86Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
17.86Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
17.86Single7PYRPSB-21157PYR-A2A-PSB-2115
17.86Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
17.86Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
17.86Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
17.86Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
17.86Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
17.86Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
17.86Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
17.86Single8RLNLUF58348RLN-A2A-LUF5834
17.86Single8X63Mepyramine8X63-H1-Mepyramine
17.86Single8X64Desloratadine8X64-H1-Desloratadine
17.86Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
17.86Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
17.86Single9IYAONO-97105319IYA-GPR55-ONO-9710531
17.86Consensusalpha2_onOrthosteric Ligandalpha2b_on
17.86Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
17.86Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
17.86Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
17.86Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
17.86Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
17.86Consensushistamine_offOrthosteric Ligandh1_off
17.86Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
17.86Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
17.65Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
17.65Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
17.65Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
17.65Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.39Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
17.39Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
17.39Single7WC4Serotonin7WC4-5-HT2A-Serotonin
17.39Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
17.39Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
17.39Single8PWNTheophylline8PWN-A2A-Theophylline
17.24Single4JKVTaladegib4JKV-SMO-Taladegib
17.24Single4NTJAZD12834NTJ-P2Y12-AZD1283
17.24Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
17.24Single5XPRBosentan5XPR-ETB-Bosentan
17.24Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
17.24Single6HLPNetupitant6HLP-NK1-Netupitant
17.24Single6LUQHaloperidol6LUQ-D2-Haloperidol
17.24Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
17.24Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.24Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
17.24Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
17.24Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
17.24Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
17.24Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.24Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.24Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
17.24Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
16.67Single3RFMCaffeine3RFM-A2A-Caffeine
16.67Single5V56TC1145V56-SMO-TC114
16.67Single5V57TC1145V57-SMO-TC114
16.67Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
16.67Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
16.67Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.67Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
16.67Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
16.67Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
16.67Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
16.67Single8EA0Iperoxo8EA0-M3-Iperoxo
16.67Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
16.67Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
16.67Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
16.67Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
16.67Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
16.67Single8XVLZibotentan8XVL-ETA-Zibotentan
16.67Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
16.67Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
16.67Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
16.67Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
16.67Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
16.67Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.67Consensussensory_onOrthosteric Ligandopsins_on
16.28Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
16.22Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
16.13Single4N4WSANT-14N4W-SMO-SANT-1
16.13Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
16.13Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
16.13Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
16.13Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.13Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
16.13Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
16.13Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
16.13Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.13Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.00Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
16.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
16.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
16.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
16.00Single7WC5Psilocin7WC5-5-HT2A-Psilocin
16.00Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
16.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
16.00Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
16.00Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
16.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
16.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
16.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
16.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
16.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
15.79Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
15.62Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
15.62Single6K1QIRL25006K1Q-ETB-IRL2500
15.62Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
15.62Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
15.62Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8XVJMacitentan8XVJ-ETA-Macitentan
15.62Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
15.62Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single5L7IVismodegib5L7I-SMO-Vismodegib
15.38Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
15.38Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
15.38Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
15.38Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
15.38Single6TP4ACT-4622066TP4-OX1-ACT-462206
15.38Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
15.38Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
15.38Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
15.38Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
15.38Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
15.38Single7UL2SR486927UL2-NTS1-SR48692-Na
15.38Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
15.38Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
15.38Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
15.38Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
15.38Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
15.38Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
15.38Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
15.38Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
15.38Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
15.38Consensusneurotensin_offOrthosteric Ligandnts1_off
15.38Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
15.15Single8IEIA1LYA8IEI-GPR156-A1LYA
15.15Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
15.15Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
15.15Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
15.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
14.81Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
14.81Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
14.81Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
14.81Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
14.81Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
14.81Single5U09Taranabant5U09-CB1-Taranabant
14.81Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
14.81Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
14.81Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
14.81Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
14.81Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
14.81Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single9BA0A1AKN9BA0-CB1-A1AKN
14.81Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
14.81Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
14.81Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
14.71Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
14.71Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
14.71Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.71Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.71Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
14.29Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
14.29Single3RZECidoxepin3RZE-H1-Cidoxepin
14.29Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
14.29Single6IQLL7458706IQL-D4-L745870
14.29Single6TPKRetosiban6TPK-OT-Retosiban
14.29Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
14.29Single6ZG9GSK10347026ZG9-M1-GSK1034702
14.29Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
14.29Single7VODCariprazine7VOD-5-HT2A-Cariprazine
14.29Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
14.29Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
14.29Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
14.29Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
14.29Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
14.29Consensusopsins_offOrthosteric Ligandrhodopsin_off
14.29Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
14.29Consensussensory_offOrthosteric Ligandopsins_off
14.29Consensusvasop-oxy_offOrthosteric Ligandot_off
13.79Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
13.79Single5DHGC-355DHG-NOP-C-35
13.79Single5DSGTiotropium5DSG-M4-Tiotropium
13.79Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
13.79Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
13.79Single6GPSMK08126GPS-CCR2-MK0812
13.79Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
13.79Single7YXAONO-54306087YXA-S1P5-ONO-5430608
13.79Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
13.79Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
13.79Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
13.79Single9B9ZA1AKO9B9Z-CB1-A1AKO
13.79Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
13.79Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
13.64Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
13.51Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
13.51Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
13.51Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
13.33Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
13.33Single5CGCHTL142425CGC-mGlu5-HTL14242
13.33Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
13.33Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
13.33Single6GPXMK08126GPX-CCR2-MK0812
13.33Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
13.33Single7SINNPS-21437SIN-CaS-NPS-2143
13.33Single7SINNPS-21437SIN-CaS-NPS-2143
13.33Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
13.33Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
13.33Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
13.33Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
13.33Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
13.33Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
13.33Consensusblt_offOrthosteric Ligandblt1_off
13.33Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
13.33Consensusep_offOrthosteric Ligandep4_off
13.16Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.04Single5MZPCaffeine5MZP-A2A-Caffeine-Na
13.04Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
12.90Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
12.50Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
12.50Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
12.50Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
12.50Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
12.50Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
12.50Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
12.50Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
12.50Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single5CGDHTL142425CGD-mGlu5-HTL14242
12.12Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
12.12Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
12.12Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
12.12Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single3OE8IT1t3OE8-CXCR4-IT1t
12.00Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
12.00Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
12.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.00Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
11.76Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
11.76Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
11.54Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
11.54Single3UZAGTPL92363UZA-A2A-GTPL9236
11.54Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
11.54Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
11.54Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.54Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.54Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
11.54Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
11.54Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
11.54Consensusgi_sensoryOrthosteric Ligandgi_opsins
11.54Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
11.54Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
11.43Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
11.11Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
11.11Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
11.11Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
11.11Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
11.11Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
11.11Single6LI0C176LI0-GPR52-C17
11.11Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
11.11Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
11.11Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
11.11Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
11.11Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.11Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
11.11Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
11.11Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
11.11Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
10.71Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
10.71Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
10.71Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
10.71Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
10.71Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.71Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
10.71Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
10.71Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
10.71Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
10.71Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
10.71Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
10.71Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
10.71Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
10.71Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
10.71Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
10.71Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.71Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
10.71Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
10.53Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
10.34Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
10.34Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
10.34Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
10.34Single7VV6C48/807VV6-MRGPRX2-C48/80
10.34Single8K2WAMG4878K2W-CXCR3-AMG487
10.34Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.34Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
10.34Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
10.34Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
10.00Single6IIVDaltroban6IIV-TP-Daltroban
10.00Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
10.00Single7F83PF-051904577F83-Ghrelin-PF-05190457
10.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
10.00Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
10.00Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
10.00Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
10.00Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
10.00Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
10.00Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
10.00Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
9.68Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
9.68Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
9.68Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
9.68Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
9.68Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
9.68Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
9.68Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
9.68Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
9.68Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
9.68Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
9.68Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
9.68Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
9.38Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
9.38Single9BJKNAM9BJK-μ-Naloxone-NAM
9.09Single5X33BIIL2605X33-BLT1-BIIL260
9.09Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
9.09Single6IIURamatroban6IIU-TP-Ramatroban
8.33Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
8.33Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
8.00Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.00Single8HS2Fab0468HS2-GPR20-Fab046
8.00Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
7.69Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
7.69Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
7.69Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
7.69Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
7.41Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
7.41Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
7.41Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.41Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.14Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
7.14Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
7.14Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.14Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
7.14Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.14Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
6.90Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.90Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.90Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.67Single6FFIMMPEP6FFI-mGlu5-MMPEP
6.67Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
6.45Single6FFHFenobam6FFH-mGlu5-Fenobam
6.25Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Single7P2L4YI7P2L-mGlu5-4YI
6.06Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
6.06Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
6.06Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.06Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
5.71Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
5.56Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
5.41Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
5.26Single7SHEPI; PE7SHE-GPR158-PI; PE
4.55Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.55Single6D35Cholesterol6D35-SMO-Cholesterol
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.55Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.55Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
4.55Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
4.55Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.55Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.55Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.55Single7XW7K1-707XW7-TSH-K1-70
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.55Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
4.55Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
4.55Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
4.55Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
4.55Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
4.55Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
4.55Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.55Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
4.55Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WVXNorrin8WVX-LGR4-Norrin
4.55Single8WVYNorrin8WVY-LGR4-Norrin
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.55Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.55Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.55Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.17Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.17Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.17Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.00Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.00Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
4.00Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.00Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.85Single5L7DCholesterol5L7D-SMO-Cholesterol
3.85Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.85Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.85Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
3.85Single9GE2Cholesterol9GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
3.57Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
3.57Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
3.45Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
3.45Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
3.33Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
3.33Single8G94CD698G94-S1P1-CD69-Gi1/β1/γ2
3.23Single8IYXYL-3658IYX-GPR34-YL-365
3.03Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
3.03Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.03Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
2.94Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
2.86Single7SHEPI; PE7SHE-GPR158-PI; PE
2.78Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
2.63Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.63Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.56Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
2.50Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.50Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.44Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.27Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
gi_chemokine 6WWZ-CCR6-CCL20-Go/β1/γ2
8HNK-CXCR3-CXCL11-Gi1/β1/γ2
8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
8KFX-CCR8-LMD-009-Gi1/β1/γ2
7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
8HNL-CXCR3-PS372424-Gi1/β1/γ2
8KFY-CCR8-ZK-756326-Gi1/β1/γ2
7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
8U1U-CCR8-CCL1-Gi1/β1/γ2
7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7XA3-CCR2-CCL2-Gi1/β1/γ2
gi_chemerin 7YKD-CML1-Chemerin-9-Gi1/β1/γ2
Net Summary
Imin 3.16769
Number of Linked Nodes 949
Number of Links 1127
Number of Hubs 172
Number of Links mediated by Hubs 678
Number of Communities 20
Number of Nodes involved in Communities 221
Number of Links involved in Communities 317
Path Summary
Number Of Nodes in MetaPath 114
Number Of Links MetaPath 113
Number of Shortest Paths 1705284
Length Of Smallest Path 3
Average Path Length 31.519
Length of Longest Path 58
Minimum Path Strength 0.242885
Average Path Strength 5.8005
Maximum Path Strength 22.9627
Minimum Path Correlation 0.700385
Average Path Correlation 0.971116
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.96078
Average % Of Corr. Nodes 39.3302
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 50.6579
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
gi_class-agi_peptide
gi_sensory
gi_alicarboxylic
gi_amine
gi_lipid
gi_nucleotide
gi_protein



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

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