Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.29 2.43859402
2G.HN.38 0.726604502
3G.S1.02 5.81648476
4G.s1h1.04 2.82049409
5G.H1.01 3.433964189
6G.S2.02 1.3581405
7G.S3.03 6.14866678
8G.S3.04 7.915234137
9G.S3.05 4.58698408
10G.S3.06 8.111255137
11G.H2.03 6.03596419
12G.H2.06 5.62325619
13G.H2.07 5.95951409
14G.H3.01 3.47925609
15G.H3.08 4.15695408
16G.H3.09 5.15386199
17G.H3.13 9.027775196
18G.H3.17 8.81188655
19G.S5.04 4.99143409
20G.S5.05 4.306695209
21G.S5.07 4.33651409
22G.HG.03 3.77875406
23G.HG.07 3.18159409
24G.hgh4.05 9.3681406
25G.hgh4.11 3.7971565
26G.hgh4.20 4.76854503
27G.hgh4.21 6.04924404
28G.H4.03 3.32745404
29G.H4.08 5.8234563
30G.H4.10 8.75621507
31G.H4.12 5.9935564
32G.H4.15 7.02737408
33G.h4s6.08 2.52352405
34G.h4s6.12 3.23615402
35G.h4s6.20 6.395494114
36G.S6.02 8.8645408
37G.S6.05 6.88169565
38G.H5.03 3.749144209
39G.H5.08 4.52929678
40G.H5.17 4.765336115
41G.H5.20 4.29555408
42b.1x4 2.56849408
43b.1x9 2.45555404
44b.1x11 3.07247408
45b.1x19 4.40806516
46b.lhb1x3 3.35432482
47b.lhb1x6 4.27198583
48b.b1x4 3.89374127
49b.l1x3 8.44681509
50b.l1x6 10.6403459
51b.b2x5 6.46723507
52b.l3x1 6.6032409
53b.l3x2 6.042965179
54b.b4x3 4.610424147
55b.b4x6 9.57225549
56b.b5x2 8.16799447
57b.b5x3 5.1272749
58b.b5x7 5.68974407
59b.l5x1 4.241485148
60b.l5x5 8.97658509
61b.b6x1 5.08836409
62b.b7x1 5.51964404
63b.b7x4 3.560684148
64b.l7x4 3.58141409
65b.b8x3 3.20875406
66b.b8x4 5.64855146
67b.l9x3 7.08525519
68b.l9x6 5.42615818
69b.b10x5 4.37346609
70b.l10x1 3.88555403
71b.b11x4 5.27633419
72b.l11x2 6.86175519
73b.b12x5 3.78081406
74b.b12x6 8.38849618
75b.b13x7 7.41617537
76b.l13x3 7.14141639
77b.l13x6 5.35581519
78b.b14x3 4.23375435
79b.b15x1 7.13318439
80b.l15x2 6.20448439
81b.b16x4 9.53148436
82b.b16x5 5.42034415
83b.b16x6 8.58087638
84b.b16x7 6.67456419
85b.b17x5 6.0676417
86b.b17x7 7.86044418
87b.l17x3 8.73481619
88b.l17x6 7.42637519
89b.b18x3 4.93083418
90b.l18x1 7.037227106
91b.l18x2 5.910344107
92b.l18x3 7.905734105
93b.b19x2 6.03316616
94b.b19x4 6.02615418
95b.l19x1 4.7806519
96b.l19x2 6.25221519
97b.b20x2 5.568416
98b.b20x4 10.0909518
99b.b20x6 6.78846516
100b.b21x1 6.94891417
101b.b21x3 5.17987416
102b.b21x5 5.6224404
103b.b21x7 6.6599505
104b.l21x2 5.90854404
105b.b22x5 5.304675107
106b.l22x5 7.13819589
107b.b23x6 6.986426157
108b.l23x1 7.67536456
109b.b24x4 6.826354156
110b.b24x6 6.626174158
111b.l25x3 8.9989599
112b.l25x6 12.8133558
113b.l27x1 9.89301759
114b.l27x2 8.25638499
115b.b28x3 4.19432407
116b.b28x4 7.70026496
117b.b28x6 8.48435599
118g.ntx8 1.42982404
119g.h1x5 1.38667406
120g.l1x4 4.81327518
121g.h2x9 1.86734484
122g.h2x11 9.044044106
123g.ctx3 6.88143409
124g.ctx6 3.22235586
125g.ctx14 5.65885409
126g.ctx15 5.87744129
127g.ctx16 5.234917128
128Lig 14.37843120
129NT 112.952725
1301x39 6.34752527
1311x43 5.66159727
1321x50 4.06578409
1331x60 4.348065227
134I1x50 3.505474229
1352x45 6.72064169
1362x47 3.41091408
1372x50 7.70735508
1382x53 5.75464628
1392x60 5.00669526
140E1 12.04191023
1413x32 4.57835526
1423x33 5.44786627
1433x34 3.98385409
1443x40 6.83815428
1453x42 9.373216169
1463x44 3.87753408
1473x46 8.13466409
1483x49 6.28567508
149I2 4.7462877
1504x46 4.01604407
1514x53 4.10137509
1524x60 7.9919428
1534x64 9.69943428
154E2 9.327691025
155E2x51 10.2945528
1565x40 3.19982424
1575x41 10.4989526
1586x29 2.64123505
1596x44 4.80891409
1606x47 7.00458408
1616x48 7.08682428
1626x51 4.84333527
163E3 3.97763824
1647x37 5.83904428
1658x53 7.022034228
166H.hahb.04 0.177135400
167H.HB.05 0.347313500
168H.hbhc.04 0.40401600
169H.HC.06 0.395495400
170H.hchd.01 0.192458500
171H.hdhe.01 0.224792500
172H.HE.04 0.493385400
173H.HE.05 0.256646500
174G.hfs2.03 0.242214400
175I3 5.24754110
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b4x4 b.l1x3 27.349512.1542NoYes089
2b.b3x6 b.l1x3 78.347910.9091NoYes099
3b.b3x6 b.l3x2 78.43697.29979NoYes099
4G.hns1.01 b.l3x2 82.4633.70073NoYes1749
5G.S1.03 G.hns1.01 82.944614.0089NoNo094
6G.S1.03 G.S3.06 83.03234.29677NoYes097
7G.S3.06 b.l5x5 83.908218.8227YesYes079
8b.l3x1 b.l5x5 84.69446.25281YesYes099
9G.H2.10 b.l3x1 40.80633.7374NoYes089
10G.H2.10 b.b6x1 40.84053.83063NoYes089
11b.b6x1 b.l9x6 89.04296.8601YesYes098
12G.H2.07 b.l9x6 99.02524.39062YesYes098
13G.H2.04 G.H2.07 99.03787.04167NoYes099
14G.H2.04 G.H3.08 99.03376.2749NoYes098
15G.H3.08 G.S4.04 99.04746.29344YesNo089
16G.S4.04 G.S5.04 98.46813.2999NoYes099
17G.S5.04 G.S5.06 99.99275.89469YesNo098
18G.S5.06 G.S6.05 1004.78167NoYes085
19G.H4.08 G.S6.05 66.3264.81302YesYes635
20G.H4.08 G.hgh4.11 66.51935.21292YesYes635
21G.hgh4.08 G.hgh4.11 33.39555.11115NoYes065
22G.H4.10 G.hgh4.08 66.550110.8314YesNo076
23G.H4.10 G.hgh4.05 66.034713.8998YesYes076
24G.HG.15 G.hgh4.05 98.92179.24927NoYes076
25G.HG.15 G.s4h3.04 98.82945.80583NoNo078
26G.HG.07 G.s4h3.04 98.73866.53104YesNo098
27G.HG.07 G.s4h3.02 98.27682.99625YesNo099
28G.HG.03 G.s4h3.02 98.18435.11448YesNo069
29G.HG.03 G.s5hg.01 97.72186.25688YesNo069
30G.S5.07 G.s5hg.01 86.11393.52833YesNo099
31G.S5.07 G.s6h5.01 85.53877.81427YesNo099
32G.S5.05 G.s6h5.01 84.81146.3501YesNo2099
33G.H5.07 G.S5.05 78.61943.13812NoYes099
34G.H5.07 G.S4.03 78.52184.01469NoNo097
35G.S1.04 G.S4.03 78.42424.84573NoNo077
36G.S1.04 G.S3.03 76.48934.04667NoYes078
37G.S1.02 G.S3.03 43.64847.80177YesYes768
38b.b2x1 b.l3x1 42.47068.23031NoYes089
39b.b2x1 b.b6x1 48.16876.1351NoYes089
40G.H4.12 G.S6.05 33.30175.53156YesYes645
41G.H4.12 G.H4.13 33.23464.28052YesNo043
42G.H4.13 G.hgh4.08 33.2127.25885NoNo036
43G.hgh4.10 G.hgh4.11 33.11733.28125NoYes015
44G.H4.05 G.hgh4.10 33.09453.94635NoNo051
45G.H4.05 G.hgh4.05 33.071912.517NoYes056
46G.H5.15 G.S1.02 11.82273.86687NoYes086
47G.S4.07 G.s1h1.04 13.70133.94698NoYes089
48G.S4.07 G.s5hg.01 13.81455.65521NoNo089
49G.S3.01 G.S3.03 31.72574.21677NoYes758
50G.S1.02 I2 31.63124.48YesYes767
51G.S3.01 I2 31.64955.04396NoYes757
52G.H2.06 b.l17x6 18.96258.22615YesYes199
53G.H2.06 b.l9x6 38.08073.34417YesYes198
54G.H2.06 b.l19x1 18.96343.38385YesYes199
55G.H5.15 G.H5.19 11.71863.49542NoNo088
563x53 G.H5.19 11.412313.8344NoNo088
573x49 3x53 11.31059.7326YesNo088
583x49 4x46 22.69955.70562YesYes087
594x42 4x46 61.54075.16094NoYes057
604x42 I2 62.78517.80406NoYes757
61I1x49 b.l25x4 15.90758.55937NoNo075
62b.l25x4 b.l27x2 16.50415.6526NoYes059
63b.l25x3 b.l27x2 18.82048.69219YesYes999
64b.b27x3 b.l25x3 24.11587.42885NoYes089
65b.b26x3 b.b27x3 31.80073.0101NoNo068
66b.b23x3 b.b26x3 32.99264.19583NoNo076
67b.b23x3 b.b24x5 35.37614.47NoNo075
68b.b23x1 b.b24x5 36.56775.23052NoNo055
69b.b23x1 b.l22x1 38.33683.36104NoNo059
70b.l22x1 g.ctx3 38.93247.68125NoYes099
71g.ctx3 g.ctx4 57.40765.08156YesNo097
72b.l26x5 g.ctx4 58.59743.68635NoNo057
73b.l26x5 g.ctx15 39.48264.75156NoYes059
74b.l17x5 b.l17x6 19.10994.6926NoYes169
75b.l17x5 b.l19x2 37.84312.46708NoYes169
76b.l17x3 b.l19x2 25.65984.86938YesYes199
77b.b19x4 b.l17x3 13.98429.26823YesYes189
78b.b19x4 b.b20x6 10.79226.34969YesYes186
79b.b17x7 b.b20x6 25.08759.54802YesYes186
80b.b17x7 b.b21x1 18.5734.82792YesYes187
81b.1x19 b.b21x1 15.8977.79208YesYes167
82b.l17x5 b.l19x1 18.85714.5701NoYes169
83b.b20x4 b.l17x3 11.172518.7129YesYes189
84b.b20x4 b.b20x6 21.57894.23281YesYes186
85b.b20x2 b.l19x2 11.80788.07073YesYes169
86b.b20x2 b.b20x4 11.17146.8176YesYes168
87g.ctx3 g.ctx6 17.29245.68219YesYes096
88b.b1x6 b.b4x6 26.213320.2046NoYes099
89b.b1x6 b.b28x5 52.01843.26885NoNo095
90b.b1x6 b.b28x3 26.20257.36615NoYes097
91b.b3x4 b.b4x6 24.03594.18385NoYes099
92b.b28x3 b.b3x4 13.29833.79958YesNo079
93b.l1x3 b.l1x7 13.39538.97521YesNo099
94b.b3x2 b.b4x6 21.68693.47771NoYes059
95b.b2x5 b.b3x2 21.48999.19406YesNo075
96b.b2x5 b.l26x1 20.304111.0306YesNo077
97b.l26x3 b.l26x5 19.71266.16562NoNo075
98b.l26x1 b.l26x3 19.90766.94208NoNo2177
993x45 4x46 38.32223.14167NoYes087
1003x42 3x45 37.68376.41052YesNo098
1012x49 3x42 33.00744.53062NoYes099
1022x49 3x39 32.79534.5476NoNo099
1032x53 3x39 26.51859.96375YesNo089
1042x53 Lig 19.83194.69677YesYes280
1051x50 2x50 11.29833.45312YesYes098
1062x46 3x46 10.13156.84781NoYes099
1072x42 3x46 24.09425.8349NoYes089
1082x42 3x49 24.41276.09469NoYes088
1093x46 6x43 10.99889.60958YesNo099
110G.s1h1.04 H.hehf.07 12.36350.404167YesNo090
111H.HF.03 H.hehf.07 12.2540.337396NoNo000
112H.HF.03 H.hehf.04 10.17520.263542NoNo000
113b.b28x5 g.ctx16 50.50293.2576NoYes1258
114b.b28x3 b.l1x7 13.29763.75906YesNo079
115g.ctx15 g.ctx16 42.58373.86719YesYes1298
116b.b3x4 b.l1x3 37.42628.52573NoYes099
117b.b4x4 b.b4x6 24.03469.53094NoYes489
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x33Lig7.263232YesYes7010
3x36Lig15.68642NoYes6010
5x41Lig8.934482YesYes6010
7x34Lig9.119170NoYes5010
7x37Lig6.932712YesYes8010
1x43Lig6.391772YesYes7010
2x53Lig4.696772YesYes8010
2x57Lig7.843542NoYes7010
3x32Lig4.028442YesYes6010
7x38Lig10.41912NoYes7010
E2Lig18.30542YesYes5010
7x30Lig8.763962NoYes5010
1x32Lig12.89010NoYes5010
1x35Lig4.29752NoYes6010
1x36Lig15.01132NoYes5010
1x39Lig10.1582YesYes7010
2x60Lig8.299792YesYes6010
2x64Lig3.390212NoYes7010
E2x52Lig10.64192NoYes5010
2x68Lig8.53250NoYes3010
1x29Lig8.103962NoYes2010
LigNT54.5122YesYes0501
E1Lig35.3072YesYes3010
NTNT356.1792YesYes5511
E1NT14.17632YesYes3511
1x357x356.021352NoNo6612
1x361x396.429692NoYes5711
1x362x617.039482NoNo5712
1x391x435.306562YesYes7711
1x392x616.36012YesNo7712
1x397x383.483232YesNo7711
1x432x535.655212YesYes7811
1x432x544.065942YesNo7712
1x432x579.416462YesNo7711
1x437x426.981562YesNo7912
2x533x366.999482YesNo8611
2x533x399.963752YesNo8912
2x533x404.791562YesYes8812
2x563x323.385830NoYes6621
2x602x613.51742YesNo6712
2x603x293.145832YesNo6512
2x603x328.724582YesYes6611
2x67E17.672080NoYes3321
E1E128.38782YesYes3311
3x26E211.0432NoYes8521
3x26E2x5121.43512NoYes8822
3x323x333.306672YesYes6711
3x323x363.446252YesNo6611
3x334x608.30992YesYes7812
3x335x413.665622YesYes7611
3x335x436.883332YesNo7712
3x406x486.859692YesYes8822
4x604x649.166352YesYes8822
4x605x4311.48412YesNo8722
4x644x686.944792YesNo8622
4x64E2x5118.04012YesYes8822
4x68E28.82012NoYes6521
E2E2x516.288852YesYes5812
E2E27.332192YesYes5511
E2x50E2x523.856870NoNo9521
5x41E220.7812YesYes6511
5x415x433.970942YesNo6712
5x415x4415.14222YesNo6612
5x44E34.506562NoYes6422
6x487x374.399372YesYes8821
6x517x336.106252YesNo7722
6x517x377.454272YesYes7821
E3E38.265942YesYes4422
7x30E33.288232NoYes5412
7x337x374.569792NoYes7821
E2NT5.976672YesYes5511
1x311x355.625210NoNo4621
2x64E13.165732NoYes7311
3x293x333.258440NoYes5721
4x64E24.646462YesYes8521
2x65Lig5.398962NoYes4010
2x64E2x526.016772NoNo7511
1x291x333.278442NoNo2311
1x25Lig5.938332NoYes0010
1x33Lig4.09252NoYes3010
5x40E22.750942YesYes4521
2x537x412.421042YesNo8612
6x56Lig2.409170NoYes0010
1x26NT2.17752NoYes0521
1x241x251.9850NoNo0021
1x432x581.813652YesNo7712
3x24E11.67242NoYes3321
1x22Lig1.566670NoYes0010
1x23NT1.46250NoYes0521
2x603x281.345832YesNo6712
1x37Lig0.9821880NoYes4010
2x66E10.8441670NoYes3321
2x622x650.750NoNo3421
3x21E10.4316670NoYes0321
2x69E10.3740620NoYes4321

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
96.55Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
79.31Consensusglp_onOrthosteric Ligandglp1_on glp2_on
79.31Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
75.00Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
73.33Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
70.97Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
70.97Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
70.00Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
69.70Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
68.97Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
68.97Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
68.75Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
67.74Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
66.67Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
65.62Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
65.62Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
65.62Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
64.71Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
64.71Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
64.52Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
64.52Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
64.52Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
64.52Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
64.10Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
63.64Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
63.33Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
63.33Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
63.33Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
62.86Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
62.50Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
62.50Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
62.16Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
61.76Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
61.76Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
61.29Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
61.29Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
60.61Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
60.61Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
59.38Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
59.38Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
59.38Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
58.33Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
58.06Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
58.06Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
58.06Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
57.89Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
57.58Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
57.58Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
57.58Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
57.58Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
57.14Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
56.67Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
56.25Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
56.25Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
56.25Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
56.25Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
55.88Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
55.56Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
55.56Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
54.55Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
54.55Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
54.55Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
54.05Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
54.05Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
54.05Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
53.33Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
53.12Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
52.78Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
52.63Consensuspth_onOrthosteric Ligandpth1_on pth2_on
51.72Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
51.52Consensuspac_onOrthosteric Ligandpac1_on
51.43Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
51.22Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
50.00Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
50.00Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
50.00Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
50.00Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
50.00Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
50.00Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
48.48Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
48.39Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
47.22Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
47.22Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
45.71Single6FJ3PTH6FJ3-PTH1-PTH
45.71Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
45.71Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
45.45Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
45.45Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
44.44Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
43.24Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
42.50Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
42.42Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
41.46Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
40.54Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
40.54Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
40.54Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
40.00Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
39.47Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
39.47Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
39.47Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
39.47Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
39.47Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
39.39Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
39.39Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
39.02Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
38.89Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
38.24Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
37.84Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
37.84Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
37.84Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
37.50Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
37.50Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
37.50Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
37.14Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
36.84Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
36.84Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
36.84Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
36.36Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
36.36Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
36.11Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
36.11Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
35.90Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
35.71Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
35.56Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
35.14Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
35.14Consensuscalcitonin_onOrthosteric Ligandctlike_on
35.14Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
35.00Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
35.00Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
35.00Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
34.38Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
34.21Single4XT3Fractalkine4XT3-US28-Fractalkine
34.21Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
34.21Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
34.21Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
34.21Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
34.21Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
34.15Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
34.09Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
33.33Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
33.33Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
33.33Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
33.33Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
33.33Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
33.33Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
33.33Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
32.50Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
32.50Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
32.50Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
32.50Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
32.43Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
32.43Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
32.43Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
31.91Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
31.82Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
31.71Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
31.71Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
31.58Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
31.58Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
31.58Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
31.43Single4XT1Fractalkine4XT1-US28-Fractalkine
31.25Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
30.77Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.77Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
30.77Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
30.56Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
30.56Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
30.30Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
30.30Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
30.30Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
30.23Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
30.23Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
30.23Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
30.00Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
30.00Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
30.00Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
29.41Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
29.41Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
29.27Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
29.27Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
29.03Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
29.03Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
28.95Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
28.95Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
28.95Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
28.95Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
28.95Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
28.57Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
28.57Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
28.21Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.21Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.12Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
28.12Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
28.12Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
28.12Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
28.12Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
27.91Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
27.78Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
27.78Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
27.78Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
27.78Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
27.50Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
27.50Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
27.50Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
27.27Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
27.03Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
27.03Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
27.03Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
27.03Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
26.83Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.83Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
26.83Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
26.83Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.83Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.47Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
26.47Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
26.47Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
26.47Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
26.47Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
26.47Consensuslpl_offOrthosteric Ligands1p_off lpa_off
26.32Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
26.32Consensusangiotensin_onOrthosteric Ligandat1_on
26.32Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
26.32Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
26.19Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
26.19Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
25.81Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
25.71Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
25.71Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
25.64Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
25.64Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.64Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
25.64Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
25.64Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
25.58Single6IGKEndothelin-36IGK-ETB-Endothelin-3
25.58Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.58Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.58Consensusbombesin_onOrthosteric Ligandbb2_on
25.58Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
25.58Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.00Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
25.00Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
25.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
25.00Single7V3ZCP559407V3Z-CB1-CP55940
25.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
25.00Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
25.00Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
25.00Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
25.00Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
25.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
25.00Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
25.00Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
25.00Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
25.00Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
25.00Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
25.00Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
25.00Consensushca_on_gpOrthosteric Ligandhca2_on_gp
25.00Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
25.00Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
24.39Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
24.39Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
24.32Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
24.32Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
24.32Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
24.32Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
24.32Consensuslpl_onOrthosteric Ligands1p_on lpa_on
24.32Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
24.32Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.24Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
24.24Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
24.24Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
24.24Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
24.24Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
24.24Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
24.24Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
24.24Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
24.24Single9B9ZA1AKO9B9Z-CB1-A1AKO
24.24Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
24.24Single9EHSLUF76029EHS-A3A-LUF7602
24.24Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
24.24Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
24.14Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
23.81Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
23.81Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
23.81Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
23.81Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
23.81Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
23.68Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
23.68Single7XNACYN1548067XNA-SST2-CYN154806
23.68Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
23.68Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
23.68Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
23.68Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
23.68Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
23.53Single5XR8AM8415XR8-CB1-AM841
23.53Single7TUYGSK682753A7TUY-GPR183-GSK682753A
23.53Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
23.53Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
23.53Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
23.53Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
23.53Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
23.33Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
23.33Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
23.33Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
23.33Single8K5BNiacin8K5B-HCA2-Niacin
23.33Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
23.08Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
23.08Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
23.08Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
22.92Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
22.92Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
22.86Single6KQICP559406KQI-CB1-CP55940-Org27569
22.86Single6OS2TRV0266OS2-AT1-TRV026
22.86Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
22.86Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
22.86Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
22.86Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.86Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
22.86Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
22.86Single8XYIVUF106618XYI-CXCR3-VUF10661
22.86Single9DGIZ85267113509DGI-CB1-Z8526711350
22.86Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
22.86Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
22.86Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
22.86Consensuslpa_offOrthosteric Ligandlpa1_off
22.86Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
22.86Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
22.73Single5GLHEndothelin-15GLH-ETB-Endothelin-1
22.73Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
22.73Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
22.73Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
22.58Single5U09Taranabant5U09-CB1-Taranabant
22.58Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
22.58Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
22.58Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
22.58Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.58Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.58Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.58Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.50Single6JODAngiotensin II6JOD-AT2-Angiotensin II
22.50Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
22.50Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
22.50Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
22.50Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.50Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
22.50Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
22.50Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
22.50Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
22.22Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
22.22Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
22.22Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
22.22Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
22.22Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
22.22Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
22.22Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
22.22Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
22.22Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
22.22Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
22.22Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
21.95Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
21.95Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
21.95Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
21.95Single8ZRTET-18ZRT-ETB-ET-1
21.95Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
21.95Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
21.95Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
21.95Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
21.88Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
21.88Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
21.88Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
21.88Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
21.88Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
21.88Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
21.88Single8K5CAcipimox8K5C-HCA2-Acipimox
21.88Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
21.88Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
21.88Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
21.88Consensushca_onOrthosteric Ligandhca2_on
21.74Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
21.74Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
21.62Single4UG2CGS216804UG2-A2A-CGS21680
21.62Single5ZTYAM102575ZTY-CB2-AM10257
21.62Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
21.62Single7SK9CCX6627SK9-ACKR3-CCX662
21.62Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
21.62Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
21.62Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
21.62Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
21.62Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
21.62Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
21.62Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
21.62Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
21.43Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
21.43Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
21.21Single4YAYZD-71554YAY-AT1-ZD-7155
21.21Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
21.21Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
21.21Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
21.21Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
21.21Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
21.21Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
21.21Single8K5DGSK2560738K5D-HCA2-GSK256073
21.21Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
21.21Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
21.21Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
21.21Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
21.21Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
21.21Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
21.05Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
21.05Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
21.05Single7QA8Peptide7QA8-STE2-Peptide
21.05Single7QA8Peptide7QA8-STE2-Peptide
21.05Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
21.05Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
21.05Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
21.05Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
21.05Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
21.05Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
21.05Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
21.05Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
21.05Consensussomatostatin_offOrthosteric Ligandsst2_off
20.93Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.93Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
20.93Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
20.93Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
20.59Single5C1MBU725C1M-μ-BU72
20.59Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
20.59Single7C4SS1P7C4S-S1P3-S1P
20.59Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
20.59Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.59Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
20.59Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
20.59Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
20.59Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
20.59Single8S4DCMF-0198S4D-Apelin-CMF-019
20.59Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
20.59Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
20.59Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
20.51Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
20.51Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
20.51Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
20.51Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
20.51Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
20.51Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
20.51Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
20.51Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.45Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
20.45Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
20.45Single8IY6Endothelin-18IY6-ETB-Endothelin-1
20.45Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
20.45Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
20.45Consensusbradykinin_onOrthosteric Ligandbk2_on
20.45Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
20.45Consensusendothelin_onOrthosteric Ligandetb_on eta_on
20.45Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
20.37Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.00Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
20.00Single5XRAAM115425XRA-CB1-AM11542
20.00Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
20.00Single6W25SHU91196W25-MC4-SHU9119-Ca
20.00Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
20.00Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
20.00Single7FEECP559407FEE-CB1-CP55940-ZCZ011
20.00Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
20.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
20.00Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
20.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
20.00Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
20.00Single8E0GBU728E0G-μ-BU72
20.00Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
20.00Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
20.00Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
20.00Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
20.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
20.00Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
20.00Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.00Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
20.00Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
20.00Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
20.00Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
20.00Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
20.00Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
20.00Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
20.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
20.00Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
20.00Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
20.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
20.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
20.00Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
20.00Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
20.00Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
20.00Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
20.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
20.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
19.57Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
19.57Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
19.57Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
19.51Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
19.51Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
19.51Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
19.51Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
19.51Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
19.51Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
19.51Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
19.51Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
19.51Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
19.51Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
19.51Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
19.51Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
19.51Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
19.51Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
19.51Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
19.51Consensusvasop-oxy_onOrthosteric Ligandv2_on
19.51Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
19.44Single4XEENeurotensin4XEE-NTS1-Neurotensin
19.44Single4XESNeurotensin4XES-NTS1-Neurotensin
19.44Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
19.44Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
19.44Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
19.44Single6IIURamatroban6IIU-TXA2-Ramatroban
19.44Single6YVRNTS8-136YVR-NTS1-NTS8-13
19.44Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
19.44Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
19.44Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
19.44Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
19.44Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
19.44Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
19.44Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
19.44Single8JWY2-1188JWY-A2A-2-118
19.44Single8JWZAB9288JWZ-A2A-AB928-Na
19.44Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
19.44Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
19.44Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.44Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
19.44Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
19.44Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
19.44Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
19.44Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
19.44Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
19.35Single6LI0C176LI0-GPR52-C17
19.35Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
19.35Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
19.35Single9B9Y7DY9B9Y-CB1-7DY
19.05Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
19.05Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
19.05Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
19.05Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
19.05Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
19.05Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
19.05Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
18.92Single4BUONeurotensin4BUO-NTS1-Neurotensin
18.92Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
18.92Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
18.92Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
18.92Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
18.92Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
18.92Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
18.92Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
18.92Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
18.92Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
18.92Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
18.92Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
18.92Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
18.92Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
18.92Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
18.92Consensuscck_onOrthosteric Ligandccka_on cckb_on
18.92Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
18.92Consensuschemerin_onOrthosteric Ligandcml1_on
18.92Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
18.92Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.92Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.92Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
18.92Consensusprostanoid_offOrthosteric Ligandep_off dp_off
18.75Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
18.75Single4BWBNeurotensin4BWB-NTS1-Neurotensin
18.75Single5ZKQABT-4915ZKQ-PAF-ABT-491
18.75Single6AKXA4R6AKX-CCR5-A4R
18.75Single6AKYMaraviroc6AKY-CCR5-Maraviroc
18.75Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
18.75Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
18.75Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
18.75Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
18.75Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
18.75Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
18.75Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
18.75Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
18.75Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
18.75Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
18.75Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
18.75Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
18.75Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
18.75Consensusangiotensin_offOrthosteric Ligandat1_off
18.75Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
18.75Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
18.60Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
18.60Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
18.60Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
18.60Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
18.60Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
18.60Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
18.60Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
18.42Single3NY9ICI118-5513NY9-β2-ICI118-551
18.42Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
18.42Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
18.42Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
18.42Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.42Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
18.42Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
18.42Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
18.42Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.42Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
18.42Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
18.42Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
18.42Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
18.42Single8QJ2pN1628QJ2-MC4-pN162-Gs
18.42Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
18.42Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
18.42Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
18.42Single9IPYJR14a9IPY-C3aB-JR14a
18.42Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
18.42Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
18.18Single4MBSMaraviroc4MBS-CCR5-Maraviroc
18.18Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
18.18Single7F61PF-036547467F61-H3-PF-03654746
18.18Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
18.18Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
18.18Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
18.18Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
18.18Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
18.18Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
18.18Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
18.18Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
18.18Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
18.18Single8RLNLUF58348RLN-A2A-LUF5834
18.18Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
18.18Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
18.18Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
18.18Single9BA0A1AKN9BA0-CB1-A1AKN
18.18Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
18.18Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
18.18Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
18.18Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
18.18Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
18.18Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
18.18Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
18.18Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
17.95Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
17.95Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
17.95Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
17.95Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
17.95Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
17.95Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
17.95Single8WDTphotoNECA8WDT-A2A-photoNECA
17.95Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.95Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
17.95Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
17.95Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
17.95Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
17.95Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
17.78Single6IGLIRL16206IGL-ETB-IRL1620
17.78Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
17.78Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
17.78Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
17.78Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
17.65Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
17.65Single5UENDU1725UEN-A1-DU172
17.65Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
17.65Single6PS1Timolol6PS1-β2-Timolol
17.65Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
17.65Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
17.65Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
17.65Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
17.65Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
17.65Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
17.65Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
17.65Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
17.65Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
17.65Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
17.65Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
17.65Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
17.65Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
17.65Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.65Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.65Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.65Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
17.65Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
17.65Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
17.65Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
17.65Single9CHXS-Carazolol9CHX-β2-S-Carazolol
17.65Consensusa3_onOrthosteric Liganda3a_on
17.65Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
17.65Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
17.65Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
17.50Single3QAKUK-4320973QAK-A2A-UK-432097
17.50Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
17.50Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
17.50Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
17.50Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
17.50Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
17.50Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
17.50Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
17.50Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
17.50Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
17.50Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
17.50Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
17.50Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
17.50Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
17.50Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
17.50Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
17.50Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
17.50Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
17.50Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
17.50Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
17.50Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
17.39Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
17.24Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
17.24Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
17.24Single8HS2Fab0468HS2-GPR20-Fab046
17.14Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
17.14Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
17.14Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
17.14Single6D26Fevipiprant6D26-DP2-Fevipiprant
17.14Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
17.14Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
17.14Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
17.14Single7C61Ergotamine7C61-5-HT1B-Ergotamine
17.14Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
17.14Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
17.14Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
17.14Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
17.14Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.14Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
17.14Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
17.14Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
17.14Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
17.14Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.14Single8JXSPF-61428JXS-D1-PF-6142
17.14Single8TF5Oleic acid8TF5-GPR6-Oleic acid
17.14Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
17.14Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.14Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.14Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
17.14Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
17.14Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
17.14Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
17.14Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
17.14Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
17.14Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
17.14Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
17.14Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
17.14Consensusa3_on_gpOrthosteric Liganda3a_on_gp
17.14Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.14Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.14Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
17.14Consensusblt_offOrthosteric Ligandblt1_off
17.14Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
17.14Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
17.14Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
17.14Consensusdp_offOrthosteric Liganddp2_off
17.14Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
17.14Consensusep_offOrthosteric Ligandep4_off
17.14Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
17.14Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
17.14Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
17.14Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.14Consensustrace-amine_onOrthosteric Ligandta1_on
17.07Single3OE0CVX153OE0-CXCR4-CVX15
17.07Single5WF5UK-4320975WF5-A2A-UK-432097
17.07Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
17.07Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
17.07Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
17.07Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
17.07Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
17.07Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.07Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
17.07Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
17.07Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
17.07Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
17.02Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
16.67Single2YDVNECA2YDV-A2A-NECA
16.67Single3P0GBI1671073P0G-β2-BI167107
16.67Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
16.67Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
16.67Single4BV0Neurotensin4BV0-NTS1-Neurotensin
16.67Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
16.67Single4UHRCGS216804UHR-A2A-CGS21680
16.67Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
16.67Single5G53NECA5G53-A2A-NECA-Gs
16.67Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
16.67Single6OS1TRV0266OS1-AT1-TRV026
16.67Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
16.67Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
16.67Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
16.67Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
16.67Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
16.67Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
16.67Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
16.67Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
16.67Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
16.67Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
16.67Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
16.67Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
16.67Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
16.67Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
16.67Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
16.67Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
16.67Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
16.67Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
16.67Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
16.67Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
16.67Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
16.67Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
16.67Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
16.67Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
16.67Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
16.67Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
16.67Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
16.67Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
16.67Single8ZWFJR14a8ZWF-C3aB-JR14a
16.67Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
16.67Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
16.67Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
16.67Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusa2_onOrthosteric Liganda2b_on
16.67Consensusa2_on_gpOrthosteric Liganda2b_on_gp
16.67Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
16.67Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
16.67Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
16.67Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
16.67Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
16.67Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
16.67Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
16.67Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
16.67Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
16.67Consensuslpa_onOrthosteric Ligandlpa1_on
16.67Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
16.67Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusneurotensin_onOrthosteric Ligandnts1_on
16.67Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
16.67Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
16.67Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
16.28Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
16.28Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
16.28Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
16.28Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
16.28Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.22Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
16.22Single6A93Risperidone6A93-5-HT2A-Risperidone
16.22Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
16.22Single6MXTSalmeterol6MXT-β2-Salmeterol
16.22Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
16.22Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
16.22Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
16.22Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
16.22Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
16.22Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
16.22Single7K15MKD0467K15-BLT1-MKD046-Na
16.22Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
16.22Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
16.22Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
16.22Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.22Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
16.22Single7YITNalfurafine7YIT-κ-Nalfurafine
16.22Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
16.22Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
16.22Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
16.22Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single8JJ8Formoterol8JJ8-β2-Formoterol
16.22Single8JJLOlodaterol8JJL-β2-Olodaterol
16.22Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
16.22Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
16.22Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
16.22Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
16.22Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
16.22Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
16.22Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
16.22Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
16.22Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.22Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.22Consensusalpha1_offOrthosteric Ligandalpha1a_off
16.22Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
16.22Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
16.22Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
16.22Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
16.22Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
16.22Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
16.22Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
16.22Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
16.22Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
16.22Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
16.22Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
16.22Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
16.22Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
16.22Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
16.22Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
16.22Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
16.13Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.13Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
16.13Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
16.13Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
15.91Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
15.91Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
15.91Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
15.91Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
15.91Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
15.91Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
15.79Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
15.79Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
15.79Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
15.79Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
15.79Single5X93K-87945X93-ETB-K-8794
15.79Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
15.79Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
15.79Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
15.79Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
15.79Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
15.79Single7EZCUKA7EZC-A2A-UKA
15.79Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
15.79Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
15.79Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
15.79Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
15.79Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
15.79Single7UM4AS26747237UM4-5-HT5A-AS2674723
15.79Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
15.79Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
15.79Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
15.79Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
15.79Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
15.79Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.79Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
15.79Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
15.79Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
15.79Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
15.79Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
15.79Consensusendothelin_offOrthosteric Ligandetb_off
15.79Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
15.79Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
15.79Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
15.62Single3OE9IT1t3OE9-CXCR4-IT1t
15.62Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
15.62Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
15.62Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
15.62Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
15.62Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
15.62Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
15.62Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
15.56Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
15.56Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
15.38Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
15.38Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
15.38Single6PT3DPI-2876PT3-δ-DPI-287
15.38Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
15.38Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
15.38Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
15.38Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
15.38Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
15.38Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
15.38Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
15.38Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
15.38Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
15.38Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
15.38Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.22Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
15.15Single3PWHZM-2413853PWH-A2A-ZM-241385
15.15Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
15.15Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
15.15Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
15.15Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
15.15Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
15.15Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
15.15Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
15.15Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
15.15Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.15Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
15.15Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
15.15Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
15.15Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
15.15Single8GNGIstradefylline8GNG-A2A-Istradefylline
15.15Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
15.15Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
15.15Single8IWESpermidine8IWE-TA9-Spermidine
15.15Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
15.15Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
15.15Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
15.15Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
15.15Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
15.15Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
15.15Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
15.15Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
15.15Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
15.15Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
15.15Consensusalpha2_offOrthosteric Ligandalpha2c_off
15.00Single4IARErgotamine4IAR-5-HT1B-Ergotamine
15.00Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
15.00Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
15.00Single7F8XNN90567F8X-CCKA-NN9056
15.00Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
15.00Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
15.00Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
15.00Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
15.00Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
15.00Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
15.00Single8KIGSHU91198KIG-MC3-SHU9119-Ca
15.00Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
15.00Single8WKYPG-9348WKY-MC4-PG-934
15.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.00Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
15.00Single9M4TSilodosin9M4T-Alpha1A-Silodosin
15.00Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
15.00Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
14.89Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
14.71Single2YDOAdenosine2YDO-A2A-Adenosine
14.71Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
14.71Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
14.71Single6PS0S-Carazolol6PS0-β2-S-Carazolol
14.71Single6PS4ICI118-5516PS4-β2-ICI118-551
14.71Single6PS5S-Propranolol6PS5-β2-S-Propranolol
14.71Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
14.71Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
14.71Single7AROLUF58337ARO-A2A-LUF5833-Na
14.71Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
14.71Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
14.71Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.71Single7T32ZM-2413857T32-A2A-ZM-241385
14.71Single7UL3Famotidine7UL3-H2-Famotidine
14.71Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.71Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
14.71Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
14.71Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
14.71Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
14.71Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
14.71Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
14.71Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
14.71Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
14.71Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.71Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.71Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
14.71Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
14.71Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
14.71Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
14.71Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
14.71Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
14.71Single8IHKAcifran8IHK-HCA3-Acifran
14.71Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
14.71Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
14.71Single8K2WAMG4878K2W-CXCR3-AMG487
14.71Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
14.71Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
14.71Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
14.71Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.71Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.71Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
14.71Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
14.71Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
14.71Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
14.71Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
14.71Single8ZPMAMD0708ZPM-CXCR4-AMD070
14.71Single9AS5Mescaline9AS5-5-HT2A-Mescaline
14.71Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
14.71Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
14.71Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
14.71Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
14.71Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
14.71Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
14.71Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.63Single6HLOAprepitant6HLO-NK1-Aprepitant
14.63Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
14.63Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
14.63Single7SK5CXCL127SK5-ACKR3-CXCL12
14.63Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.63Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
14.58Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
14.58Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
14.29Single2Y04Salbutamol2Y04-β1-Salbutamol
14.29Single3NY8ICI118-5513NY8-β2-ICI118-551
14.29Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
14.29Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
14.29Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
14.29Single4GBRS-Carazolol4GBR-β2-S-Carazolol
14.29Single4QKX35V4QKX-β2-35V
14.29Single5DHHSB-6121115DHH-NOP-SB-612111
14.29Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
14.29Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
14.29Single5T04Neurotensin5T04-NTS1-Neurotensin
14.29Single5TGZAM65385TGZ-CB1-AM6538
14.29Single5UIGCmpd-15UIG-A2A-Cmpd-1
14.29Single6D27CAY104716D27-DP2-CAY10471
14.29Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
14.29Single6GPSMK08126GPS-CCR2-MK0812
14.29Single6H7MSalbutamol6H7M-β1-Salbutamol
14.29Single6IIVDaltroban6IIV-TXA2-Daltroban
14.29Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
14.29Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
14.29Single6PT2KGCHM076PT2-δ-KGCHM07
14.29Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
14.29Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
14.29Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
14.29Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
14.29Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
14.29Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
14.29Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
14.29Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
14.29Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
14.29Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
14.29Single7UL4Alvimopan7UL4-μ-Alvimopan
14.29Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
14.29Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
14.29Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
14.29Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7WC7Lisuride7WC7-5-HT2A-Lisuride
14.29Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
14.29Single7YXAONO-54306087YXA-S1P5-ONO-5430608
14.29Single8CU6LJ-45178CU6-A2A-LJ-4517
14.29Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
14.29Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
14.29Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
14.29Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
14.29Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
14.29Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
14.29Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
14.29Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
14.29Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
14.29Single8JJOAlprenolol8JJO-β2-Alprenolol
14.29Single8JXRLSD8JXR-D1-LSD
14.29Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
14.29Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
14.29Single8T1WCVN4248T1W-GPR6-CVN424
14.29Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
14.29Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
14.29Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
14.29Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
14.29Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
14.29Single9AS1DMT9AS1-5-HT2A-DMT
14.29Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
14.29Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
14.29Single9H37A1IR09H37-A2A-A1IR0-Na
14.29Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
14.29Consensus5ht5_onOrthosteric Ligand5ht5a_on
14.29Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
14.29Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
14.29Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
14.29Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
14.29Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
14.29Consensusblt_onOrthosteric Ligandblt1_on
14.29Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
14.29Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
14.29Consensusdopamine_offOrthosteric Ligandd2_off d3_off
14.29Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
14.29Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
14.29Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
14.29Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
14.29Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
14.29Consensusleukotriene_onOrthosteric Ligandblt_on
14.29Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
14.29Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.29Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.29Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
13.95Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
13.95Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
13.95Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
13.95Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
13.95Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
13.89Single2RH1S-Carazolol2RH1-β2-S-Carazolol
13.89Single2Y03Isoprenaline2Y03-β1-Isoprenaline
13.89Single2YCWS-Carazolol2YCW-β1-S-Carazolol
13.89Single4JKVTaladegib4JKV-SMO-Taladegib
13.89Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
13.89Single5D6LS-Carazolol5D6L-β2-S-Carazolol
13.89Single5JQHS-Carazolol5JQH-β2-S-Carazolol
13.89Single5N2RPSB-365N2R-A2A-PSB-36-Na
13.89Single5N2SPSB365N2S-A1-PSB36
13.89Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
13.89Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
13.89Single5TVNLSD5TVN-5-HT2B-LSD
13.89Single5WIUNemonapride5WIU-D4-Nemonapride
13.89Single5WIVNemonapride5WIV-D4-Nemonapride-Na
13.89Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
13.89Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
13.89Single6E67BI1671076E67-β2-BI167107-Gs(CT)
13.89Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
13.89Single6GPXMK08126GPX-CCR2-MK0812
13.89Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
13.89Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
13.89Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
13.89Single6PS6Timolol6PS6-β2-Timolol
13.89Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
13.89Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
13.89Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.89Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
13.89Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
13.89Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
13.89Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
13.89Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
13.89Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
13.89Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
13.89Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.89Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.89Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
13.89Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
13.89Single8QOTNanobody-E8QOT-μ-Nanobody-E
13.89Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
13.89Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
13.89Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
13.89Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
13.89Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.89Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
13.89Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
13.89Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
13.89Consensusadenosine_offOrthosteric Liganda1_off a2_off
13.89Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
13.89Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
13.89Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
13.89Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
13.89Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
13.89Consensusamine_offonOrthosteric Ligandamine_off amine_on
13.89Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
13.89Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
13.89Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
13.89Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
13.89Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.89Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.89Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
13.89Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
13.89Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
13.89Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
13.79Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
13.64Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.64Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
13.64Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
13.64Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
13.51Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
13.51Single4DJHJDTic4DJH-κ-JDTic
13.51Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
13.51Single5D5AS-Carazolol5D5A-β2-S-Carazolol
13.51Single5D5BS-Carazolol5D5B-β2-S-Carazolol
13.51Single5V56TC1145V56-SMO-TC114
13.51Single5V57TC1145V57-SMO-TC114
13.51Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
13.51Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
13.51Single6H7JIsoprenaline6H7J-β1-Isoprenaline
13.51Single6J21Aprepitant6J21-NK1-Aprepitant
13.51Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
13.51Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
13.51Single6TQ7SB-3348676TQ7-OX1-SB-334867
13.51Single6WGTLSD6WGT-5-HT2A-LSD
13.51Single7B6WCyclazosin7B6W-α1b-Cyclazosin
13.51Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
13.51Single7F1TMIP-1a7F1T-CCR5-MIP-1a
13.51Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
13.51Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
13.51Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
13.51Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
13.51Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
13.51Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
13.51Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
13.51Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
13.51Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.51Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
13.51Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.51Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
13.51Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
13.51Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
13.51Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.51Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
13.51Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
13.51Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
13.51Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
13.51Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.51Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
13.51Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
13.51Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
13.51Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
13.51Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
13.51Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
13.51Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.51Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
13.51Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
13.51Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
13.51Single9BJKNaloxone9BJK-μ-Naloxone-NAM
13.51Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
13.51Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
13.51Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
13.51Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
13.51Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
13.51Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
13.51Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.51Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
13.51Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
13.51Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
13.51Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
13.51Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.51Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
13.51Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
13.51Consensusrelaxin_onOrthosteric Ligandrxfp4_on
13.51Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
13.33Single7SK3CXCL127SK3-ACKR3-CXCL12
13.16Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
13.16Single3D4STimolol3D4S-β2-Timolol
13.16Single4AMIBucindolol4AMI-β1-Bucindolol
13.16Single4LDEBI1671074LDE-β2-BI167107
13.16Single4N4WSANT-14N4W-SMO-SANT-1
13.16Single4RWADIPP-NH24RWA-δ-DIPP-NH2
13.16Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
13.16Single5X33BIIL2605X33-BLT1-BIIL260
13.16Single6CM4Risperidone6CM4-D2-Risperidone
13.16Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
13.16Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
13.16Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
13.16Single6ZG4HTL00099366ZG4-M1-HTL0009936
13.16Single7DFPSpiperone7DFP-D2-Spiperone
13.16Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.16Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
13.16Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.16Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
13.16Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
13.16Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.16Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
13.16Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
13.16Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
13.16Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
13.16Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
13.16Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
13.16Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.16Single9BJKNAM9BJK-μ-Naloxone-NAM
13.16Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.16Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
13.16Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
13.16Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
13.16Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
13.16Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
13.16Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
13.16Consensusorexin_onOrthosteric Ligandox2_on
13.16Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.16Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.04Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
13.04Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
13.04Single9KDFRES-701-39KDF-ETB-RES-701-3
12.90Single8A2OTheophylline8A2O-A2A-Theophylline-Na
12.90Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
12.90Single9CHUNoradrenaline9CHU-β2-Noradrenaline
12.90Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
12.82Single6H7LDobutamine6H7L-β1-Dobutamine
12.82Single6IBLArformoterol6IBL-β1-Arformoterol
12.82Single6K1QIRL25006K1Q-ETB-IRL2500
12.82Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
12.82Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
12.82Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.82Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
12.82Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
12.82Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
12.82Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
12.82Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
12.82Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
12.82Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
12.82Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
12.82Single8XVJMacitentan8XVJ-ETA-Macitentan
12.82Single8XVUCXCL28XVU-CXCR2-CXCL2
12.82Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
12.82Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
12.82Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
12.82Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
12.82Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
12.82Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
12.82Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
12.50Single3OE6IT1t3OE6-CXCR4-IT1t
12.50Single5WF6UK-4320975WF6-A2A-UK-432097
12.50Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
12.50Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
12.50Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
12.50Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
12.50Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
12.50Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
12.50Single7XN9L-054,5227XN9-SST2-L-054,522
12.50Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
12.50Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
12.50Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
12.50Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8X5YAstemizole8X5Y-H1-Astemizole
12.50Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
12.50Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
12.50Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
12.50Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
12.50Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
12.50Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
12.50Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9LRCHistamine9LRC-H4-Histamine
12.50Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
12.50Consensus5ht2_onOrthosteric Ligand5ht2b_on
12.50Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.50Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.50Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.50Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.20Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
12.20Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
12.20Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
12.20Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
12.20Single8XWNCXCL88XWN-CXCR2-CXCL8
12.20Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
12.20Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
12.20Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single7SRQLSD7SRQ-5-HT2B-LSD
12.12Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
12.12Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
12.12Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
12.12Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
12.12Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
12.12Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
12.12Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
12.12Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
12.12Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
12.12Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
12.12Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
12.12Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
12.12Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
12.12Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
12.12Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
12.12Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
12.12Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
12.12Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
12.12Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
12.12Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
12.12Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
12.12Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
12.12Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
12.12Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
12.12Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
12.12Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
12.12Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
12.12Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
11.90Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
11.90Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.90Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
11.90Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
11.90Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
11.90Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
11.90Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
11.76Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
11.76Single3ODUIT1t3ODU-CXCR4-IT1t
11.76Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
11.76Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
11.76Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
11.76Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
11.76Single6B73MP11046B73-κ-MP1104
11.76Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
11.76Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
11.76Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
11.76Single6ME2Ramelteon6ME2-MT1-Ramelteon
11.76Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
11.76Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
11.76Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
11.76Single7BR3Elagolix7BR3-GnRH1-Elagolix
11.76Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
11.76Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
11.76Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
11.76Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.76Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.76Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
11.76Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
11.76Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
11.76Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
11.76Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
11.76Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
11.76Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
11.76Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
11.76Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
11.76Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
11.76Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
11.76Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
11.76Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
11.76Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
11.76Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
11.76Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
11.76Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.76Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.76Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.76Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
11.76Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
11.76Single8Y0HVUF114188Y0H-CXCR3-VUF11418
11.76Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
11.76Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
11.76Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
11.76Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
11.76Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
11.76Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
11.76Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
11.76Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
11.76Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
11.76Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.76Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
11.76Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.76Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
11.76Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.76Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
11.76Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
11.76Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.76Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.76Consensusorexin_offOrthosteric Ligandox2_off ox1_off
11.76Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
11.76Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
11.76Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
11.63Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.63Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
11.63Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
11.63Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
11.63Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
11.63Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
11.43Single3REYXAC3REY-A2A-XAC
11.43Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
11.43Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
11.43Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
11.43Single4ZJCSB-6740424ZJC-OX1-SB-674042
11.43Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
11.43Single5IU7Q274563465IU7-A2A-Q27456346-Na
11.43Single5IUBQ274563445IUB-A2A-Q27456344-Na
11.43Single5JTBZM-2413855JTB-A2A-ZM-241385
11.43Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
11.43Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
11.43Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
11.43Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
11.43Single6A94Zotepine6A94-5-HT2A-Zotepine
11.43Single6AQFZM-2413856AQF-A2A-ZM-241385
11.43Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
11.43Single6KUXRS-799486KUX-α2a-RS-79948
11.43Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
11.43Single6MH8ZM-2413856MH8-A2A-ZM-241385
11.43Single6TPGEMPA6TPG-OX2-EMPA
11.43Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
11.43Single6V9SGTPL114036V9S-OX1-GTPL11403
11.43Single6VI4JDTic6VI4-κ-JDTic
11.43Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
11.43Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
11.43Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
11.43Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
11.43Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
11.43Single6ZG9GSK10347026ZG9-M1-GSK1034702
11.43Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
11.43Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
11.43Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
11.43Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
11.43Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
11.43Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
11.43Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.43Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
11.43Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
11.43Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
11.43Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
11.43Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
11.43Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
11.43Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
11.43Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.43Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
11.43Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
11.43Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
11.43Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
11.43Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.43Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.43Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.43Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.43Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
11.43Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
11.43Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
11.43Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Single8ZPNAMD31008ZPN-CXCR4-AMD3100
11.43Single9AS3LSD9AS3-5-HT2A-LSD
11.43Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
11.43Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
11.43Consensusa2_offOrthosteric Liganda2a_off
11.43Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
11.43Consensusalpha1_onOrthosteric Ligandalpha1a_on
11.43Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
11.43Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
11.43Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
11.43Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
11.43Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
11.43Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
11.43Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
11.43Consensusgrh_offOrthosteric Ligandgnrh1_off
11.43Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
11.36Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
11.36Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
11.36Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
11.11Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
11.11Single2Y01Dobutamine2Y01-β1-Dobutamine
11.11Single2Y02Carmoterol2Y02-β1-Carmoterol
11.11Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
11.11Single3EMLZM-2413853EML-A2A-ZM-241385
11.11Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
11.11Single4DAJTiotropium4DAJ-M3-Tiotropium
11.11Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
11.11Single4EJ4Naltrindole4EJ4-δ-Naltrindole
11.11Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
11.11Single4MQSIperoxo4MQS-M2-Iperoxo
11.11Single4QIMANTA XV4QIM-SMO-ANTA XV
11.11Single4U14Tiotropium4U14-M3-Tiotropium
11.11Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
11.11Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
11.11Single5DHGC-355DHG-NOP-C-35
11.11Single5IU8Q274563475IU8-A2A-Q27456347-Na
11.11Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
11.11Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
11.11Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
11.11Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
11.11Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
11.11Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
11.11Single6DRXLisuride6DRX-5-HT2B-Lisuride
11.11Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
11.11Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
11.11Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
11.11Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
11.11Single6S0LZM-2413856S0L-A2A-ZM-241385
11.11Single6TOTLemborexant6TOT-OX1-Lemborexant
11.11Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
11.11Single7BU7BI1671077BU7-β1-BI167107
11.11Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
11.11Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
11.11Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
11.11Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
11.11Single7PYRPSB-21157PYR-A2A-PSB-2115
11.11Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
11.11Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
11.11Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
11.11Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
11.11Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
11.11Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
11.11Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
11.11Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
11.11Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
11.11Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
11.11Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
11.11Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.11Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
11.11Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
11.11Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
11.11Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
11.11Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
11.11Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
11.11Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
11.11Single8X63Mepyramine8X63-H1-Mepyramine
11.11Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
11.11Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
11.11Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
11.11Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
11.11Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
11.11Single9JEAAtropine9JEA-M1-Atropine
11.11Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
11.11Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
11.11Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
11.11Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
11.11Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
11.11Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
11.11Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
11.11Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
11.11Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
11.11Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
11.11Consensusalpha2_onOrthosteric Ligandalpha2b_on
11.11Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
11.11Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
11.11Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
11.11Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
11.11Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.11Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
11.11Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
11.11Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
11.11Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
11.11Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
11.11Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
11.11Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
11.11Consensushistamine_offOrthosteric Ligandh1_off
11.11Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
11.11Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
10.81Single2Y00Dobutamine2Y00-β1-Dobutamine
10.81Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
10.81Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
10.81Single5CGCHTL142425CGC-mGlu5-HTL14242
10.81Single5IUAQ274563485IUA-A2A-Q27456348-Na
10.81Single5WQCEMPA5WQC-OX2-EMPA
10.81Single5XPRBosentan5XPR-ETB-Bosentan
10.81Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
10.81Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
10.81Single6LUQHaloperidol6LUQ-D2-Haloperidol
10.81Single6S0QZM-2413856S0Q-A2A-ZM-241385
10.81Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
10.81Single6TP6Filorexant6TP6-OX1-Filorexant
10.81Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
10.81Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
10.81Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
10.81Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
10.81Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
10.81Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
10.81Single7W41PD1762527W41-BB2-PD176252
10.81Single7WC6LSD7WC6-5-HT2A-LSD
10.81Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.81Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.81Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
10.81Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
10.81Single8GNEKW-63568GNE-A2A-KW-6356-Na
10.81Single8ZMFA1L108ZMF-5-HT2C-A1L10
10.81Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
10.81Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
10.81Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
10.81Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
10.81Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
10.81Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
10.81Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
10.81Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.81Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.81Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
10.81Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
10.81Consensusbombesin_offOrthosteric Ligandbb2_off
10.81Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
10.81Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
10.81Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
10.81Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.81Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
10.81Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.81Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
10.81Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.81Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
10.53Single4U15Tiotropium4U15-M3-Tiotropium
10.53Single5V54Methiothepin5V54-5-HT1B-Methiothepin
10.53Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
10.53Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
10.53Single6J20Aprepitant6J20-NK1-Aprepitant
10.53Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
10.53Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.53Single6OL9Tiotropium6OL9-M5-Tiotropium
10.53Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
10.53Single7PX4PSB-21137PX4-A2A-PSB-2113
10.53Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
10.53Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
10.53Single8EA0Iperoxo8EA0-M3-Iperoxo
10.53Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
10.53Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
10.53Single9AS9RS130-1809AS9-5-HT2A-RS130-180
10.53Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
10.53Consensus5ht1_offOrthosteric Ligand5ht1b_off
10.53Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
10.53Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
10.53Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
10.53Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
10.53Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.53Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
10.53Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
10.53Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
10.26Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
10.26Single5CXVTiotropium5CXV-M1-Tiotropium
10.26Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
10.26Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
10.26Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.26Single8XQJJN2418XQJ-Apelin-JN241
10.26Single8XWMCXCL68XWM-CXCR2-CXCL6
10.26Single8XWSCXCL58XWS-CXCR2-CXCL5
10.26Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
10.26Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
10.26Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
10.26Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
10.26Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
10.00Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
10.00Single5CGDHTL142425CGD-mGlu5-HTL14242
10.00Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
10.00Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
10.00Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
10.00Single8XWFCXCL38XWF-CXCR2-CXCL3
10.00Single8ZPLHF511168ZPL-CXCR4-HF51116
10.00Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
9.76Single6KNMJN241-96KNM-Apelin-JN241-9
9.76Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
9.76Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
9.76Single8XQJJN2418XQJ-Apelin-JN241
9.76Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
9.76Single9JF4PD1683689JF4-BB1-PD168368
9.68Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
9.68Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
9.68Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
9.68Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
9.68Single8PWNTheophylline8PWN-A2A-Theophylline
9.68Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
9.68Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
9.52Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
9.52Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.52Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
9.52Single8IEBA1LYA8IEB-GPR156-A1LYA
9.52Single8IEIA1LYA8IEI-GPR156-A1LYA
9.52Single8IEPA1LYA8IEP-GPR156-A1LYA
9.52Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
9.52Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
9.52Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.52Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.52Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
9.52Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
9.38Single3OE8IT1t3OE8-CXCR4-IT1t
9.38Single3RFMCaffeine3RFM-A2A-Caffeine
9.38Single6TQ9SB-4081246TQ9-OX1-SB-408124
9.38Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
9.38Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
9.38Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
9.38Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
9.38Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
9.38Consensusp2y_offOrthosteric Ligandp2y1_off
9.30Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
9.09Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
9.09Single4XNWMRS25004XNW-P2Y1-MRS2500
9.09Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
9.09Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
9.09Single6ME5Agomelatine6ME5-MT1-Agomelatine
9.09Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
9.09Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
9.09Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
9.09Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
9.09Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
9.09Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
9.09Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
9.09Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
9.09Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
9.09Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
9.09Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
9.09Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
8.89Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
8.89Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
8.89Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
8.82Single3PBLEticlopride3PBL-D3-Eticlopride
8.82Single4O9RCyclopamine4O9R-SMO-Cyclopamine
8.82Single5L7IVismodegib5L7I-SMO-Vismodegib
8.82Single6HLLCP999946HLL-NK1-CP99994
8.82Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
8.82Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
8.82Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
8.82Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
8.82Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
8.82Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
8.82Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
8.82Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.82Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.82Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
8.82Single9AS7Psilocin9AS7-5-HT2A-Psilocin
8.82Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
8.82Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
8.82Consensusgq_nucleotideOrthosteric Ligandgq_p2y
8.82Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
8.82Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
8.57Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
8.57Single4QINSAG1.54QIN-SMO-SAG1.5
8.57Single4S0VSuvorexant4S0V-OX2-Suvorexant
8.57Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
8.57Single5WS3EMPA5WS3-OX2-EMPA
8.57Single6DS0Ly2660976DS0-5-HT2B-Ly266097
8.57Single6ME9Ramelteon6ME9-MT2-Ramelteon
8.57Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
8.57Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
8.57Single6TODEMPA6TOD-OX1-EMPA-Na
8.57Single6TPJSuvorexant6TPJ-OX2-Suvorexant
8.57Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
8.57Single7F8ULintitript7F8U-CCKA-Lintitript
8.57Single7F8YDevazepide7F8Y-CCKA-Devazepide
8.57Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
8.57Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
8.57Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
8.57Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
8.57Single7XRRLemborexant7XRR-OX2-Lemborexant
8.57Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
8.57Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
8.57Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
8.57Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
8.57Single9H2XA1IR19H2X-A2A-A1IR1-Na
8.57Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
8.57Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.57Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.57Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
8.57Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
8.57Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
8.33Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
8.33Single3RZECidoxepin3RZE-H1-Cidoxepin
8.33Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
8.33Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
8.33Single5UVIZM-2413855UVI-A2A-ZM-241385
8.33Single6IQLL7458706IQL-D4-L745870
8.33Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
8.33Single6TP3Nemorexant6TP3-OX1-Nemorexant
8.33Single6TPNHTL66416TPN-OX2-HTL6641
8.33Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
8.33Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
8.33Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
8.33Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
8.33Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
8.33Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
8.33Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
8.33Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
8.33Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
8.33Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
8.33Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
8.33Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
8.33Single9ARXSerotonin9ARX-5-HT2A-Serotonin
8.33Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
8.33Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
8.33Consensusopsins_offOrthosteric Ligandrhodopsin_off
8.33Consensussensory_offOrthosteric Ligandopsins_off
8.11Single5DSGTiotropium5DSG-M4-Tiotropium
8.11Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.11Single7F83PF-051904577F83-Ghrelin-PF-05190457
8.11Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
8.11Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
8.11Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
8.11Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
8.11Single8X64Desloratadine8X64-H1-Desloratadine
8.11Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
8.11Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
8.11Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
8.11Single9IYAONO-97105319IYA-GPR55-ONO-9710531
8.11Consensuscck_offOrthosteric Ligandccka_off
8.11Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
8.11Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
7.89Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
7.89Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
7.89Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
7.89Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
7.89Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
7.89Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
7.89Single7SINNPS-21437SIN-CaS-NPS-2143
7.89Single7SINNPS-21437SIN-CaS-NPS-2143
7.89Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
7.89Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
7.89Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
7.89Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
7.89Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
7.89Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.89Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.89Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
7.89Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
7.89Single9HAPTolvaptan9HAP-V2-Tolvaptan
7.89Single9HC04YI9HC0-mGlu5-4YI
7.89Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
7.69Single5TZRMK86665TZR-FFA1-MK8666
7.69Single6E59L-7607356E59-NK1-L-760735
7.69Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
7.69Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
7.69Single7P2L4YI7P2L-mGlu5-4YI
7.69Single7R0CAVP7R0C-V2-AVP-Arrestin2
7.69Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
7.69Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
7.69Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
7.69Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
7.69Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
7.69Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
7.69Single8XVLZibotentan8XVL-ETA-Zibotentan
7.69Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
7.69Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.69Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
7.69Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
7.69Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
7.69Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
7.69Consensustachykinin_offOrthosteric Ligandnk1_off
7.50Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
7.50Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
7.50Single4PY02MeSATP4PY0-P2Y12-2MeSATP
7.50Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
7.50Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
7.50Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
7.50Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.50Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
7.50Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
7.50Single8XWACXCL18XWA-CXCR2-CXCL1
7.50Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
7.32Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
7.32Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
7.32Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
7.14Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
7.14Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
7.14Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
7.14Consensuskisspeptin_onOrthosteric Ligandkiss1_on
6.98Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.98Single8IEIA1LYA8IEI-GPR156-A1LYA
6.98Single8IEPA1LYA8IEP-GPR156-A1LYA
6.98Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
6.98Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
6.98Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
6.98Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
6.82Single8IEBA1LYA8IEB-GPR156-A1LYA
6.45Single5MZPCaffeine5MZP-A2A-Caffeine-Na
6.45Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
6.25Single7WC4Serotonin7WC4-5-HT2A-Serotonin
6.06Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
6.06Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
6.06Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
6.06Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
6.06Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
6.06Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
6.06Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
6.06Consensussensory_onOrthosteric Ligandopsins_on
5.88Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
5.88Single3UZAGTPL92363UZA-A2A-GTPL9236
5.88Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.88Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
5.88Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
5.88Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
5.88Single7WC5Psilocin7WC5-5-HT2A-Psilocin
5.88Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.88Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.88Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.88Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
5.88Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
5.88Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.88Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
5.88Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.88Consensusgi_sensoryOrthosteric Ligandgi_opsins
5.88Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.88Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
5.88Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
5.88Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
5.88Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
5.71Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
5.71Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
5.71Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
5.71Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
5.71Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
5.71Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
5.71Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
5.71Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
5.71Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.71Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
5.71Single7UL2SR486927UL2-NTS1-SR48692-Na
5.71Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
5.71Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
5.71Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
5.71Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
5.71Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.71Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.71Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.71Consensusneurotensin_offOrthosteric Ligandnts1_off
5.71Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
5.56Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
5.56Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
5.56Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
5.56Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
5.56Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
5.56Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
5.56Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.56Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.56Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.56Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
5.56Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
5.56Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
5.56Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
5.56Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
5.56Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.56Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
5.56Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.56Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
5.41Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
5.41Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
5.41Single6TPKRetosiban6TPK-OT-Retosiban
5.41Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
5.41Single7VODCariprazine7VOD-5-HT2A-Cariprazine
5.41Single7VV6C48/807VV6-MRGPRX2-C48/80
5.41Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
5.41Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
5.41Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
5.41Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
5.41Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
5.41Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.41Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.41Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
5.41Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.41Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.41Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.41Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.41Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
5.41Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
5.41Consensusvasop-oxy_offOrthosteric Ligandot_off
5.26Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
5.26Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
5.26Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
5.26Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
5.26Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
5.26Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
5.26Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.26Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
5.26Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
5.26Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
5.13Single4NTJAZD12834NTJ-P2Y12-AZD1283
5.13Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
5.13Single6HLPNetupitant6HLP-NK1-Netupitant
5.13Single6Z4SSR486926Z4S-NTS1-SR48692
5.13Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.13Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
5.13Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.13Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
5.13Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.13Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.13Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.13Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
5.00Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
4.88Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
4.88Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
4.88Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.88Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
4.88Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
4.76Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
4.76Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
4.65Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
4.65Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
4.55Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
3.45Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
3.45Single6D35Cholesterol6D35-SMO-Cholesterol
3.45Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
3.45Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
3.45Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
3.45Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
3.45Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
3.45Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
3.45Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
3.45Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
3.45Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
3.45Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
3.45Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.45Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.45Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.45Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.45Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
3.45Single7DTTCa7DTT-CaS-Ca-Ca
3.45Single7DTTCa7DTT-CaS-Ca-Ca
3.45Single7DTUTryptophan7DTU-CaS-Tryptophan
3.45Single7DTUTryptophan7DTU-CaS-Tryptophan
3.45Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
3.45Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
3.45Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
3.45Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
3.45Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.45Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.45Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.45Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.45Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
3.45Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
3.45Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
3.45Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
3.45Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
3.45Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
3.45Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
3.45Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
3.45Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
3.45Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
3.45Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
3.45Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
3.45Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
3.45Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.45Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.45Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
3.45Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
3.45Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.45Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.45Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.45Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.45Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
3.45Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
3.45Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
3.45Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
3.45Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
3.45Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
3.45Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.45Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.45Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.45Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.45Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.45Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.45Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.45Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.45Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
3.45Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
3.45Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
3.45Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
3.45Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
3.45Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
3.45Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
3.45Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
3.45Single7XW7K1-707XW7-TSH-K1-70
3.45Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
3.45Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
3.45Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
3.45Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
3.45Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
3.45Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
3.45Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
3.45Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
3.45Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
3.45Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
3.45Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
3.45Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
3.45Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
3.45Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
3.45Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
3.45Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
3.45Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
3.45Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
3.45Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
3.45Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
3.45Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
3.45Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.45Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.45Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.45Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.45Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.45Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.45Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
3.45Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
3.45Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
3.45Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
3.45Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
3.45Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.45Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.45Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
3.45Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
3.45Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
3.45Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
3.45Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
3.45Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
3.45Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
3.45Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
3.45Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
3.45Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
3.45Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
3.45Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
3.45Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
3.45Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
3.45Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
3.45Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
3.45Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.45Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.45Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.45Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.45Single8WVXNorrin8WVX-LGR4-Norrin
3.45Single8WVYNorrin8WVY-LGR4-Norrin
3.45Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.45Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.45Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.45Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.45Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.45Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.45Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
3.45Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
3.45Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.45Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.45Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
3.45Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
3.45Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
3.45Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
3.45Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
3.45Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.45Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.45Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.45Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.45Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.45Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.45Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.45Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.45Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.45Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.45Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.45Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.45Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.45Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.45Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.45Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.45Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
3.45Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
3.45Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
3.45Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
3.45Single9KHHNorrin9KHH-LGR4-Norrin
3.45Single9S37NB219S37-LGR4-NB21
3.45Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
3.33Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.33Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.33Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.33Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.33Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.33Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.33Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.33Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.33Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.33Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.33Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.33Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.33Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.33Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.33Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
3.33Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
3.23Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
3.23Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
3.23Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
3.12Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
3.12Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
3.12Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
3.12Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
3.12Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.03Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
3.03Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
3.03Single5L7DCholesterol5L7D-SMO-Cholesterol
3.03Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.03Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
2.94Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
2.94Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
2.86Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
2.86Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
2.86Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
2.86Single8JPSCCL78JPS-ACKR1-CCL7
2.86Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
2.78Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
2.78Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
2.78Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
2.78Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
2.78Single6TP4ACT-4622066TP4-OX1-ACT-462206
2.78Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.78Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
2.78Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
2.78Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
2.78Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
2.70Single4XNVBPTU4XNV-P2Y1-BPTU
2.70Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
2.70Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
2.70Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
2.63Single6FFIMMPEP6FFI-mGlu5-MMPEP
2.63Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
2.63Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
2.63Single6ZINSR486926ZIN-NTS1-SR48692
2.63Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
2.63Single8IYXYL-3658IYX-GPR34-YL-365
2.63Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
2.63Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
2.56Single6FFHFenobam6FFH-mGlu5-Fenobam
2.50Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
2.50Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
2.44Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
2.44Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
2.22Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.22Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.13Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.13Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.08Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
1.96Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
glp_on_gp glp1_on_gp
glp2_on_gp
gluc_on_gp 6LMK-Glucagon-Glucagon-Gs/β1/γ2
8JIT-Glucagon-MEDI0382-Gs/β1/γ2
7V35-Glucagon-Peptide-20-Gs/β1/γ2
secretin_on_gp 7D3S-Secretin-Secretin-Gs/β1/γ2
gip_on_gp 7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
7FIY-GIP-Tirzepatide-Gs/β1/γ2
7DTY-GIP-GIP-Gs/β1/γ2
Net Summary
Imin 3.12167
Number of Linked Nodes 1027
Number of Links 1188
Number of Hubs 175
Number of Links mediated by Hubs 703
Number of Communities 22
Number of Nodes involved in Communities 193
Number of Links involved in Communities 284
Path Summary
Number Of Nodes in MetaPath 118
Number Of Links MetaPath 117
Number of Shortest Paths 10233642
Length Of Smallest Path 3
Average Path Length 48.7131
Length of Longest Path 86
Minimum Path Strength 0.216354
Average Path Strength 6.18755
Maximum Path Strength 28.3447
Minimum Path Correlation 0.702604
Average Path Correlation 0.991432
Maximum Path Correlation 0.998854
Minimum % Of Corr. Nodes 1.28205
Average % Of Corr. Nodes 26.6101
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 50.5448
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
class-b1_on_gpglucagon_on_gp
vip-pacap_on_gp
pth_on_gp
crf_on_gp
calcitonin_on_gp



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Download glucagon_on_gp.zip



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