Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg Int. Strength Num Of Links Community ConSurf
1A:A:E27 7.3725406
2A:A:Y37 9.1575404
3A:A:L44 9.7025419
4A:A:L46 5.1375418
5A:A:K53 6.98754159
6A:A:I207 5.242519
7A:A:E209 7.3225419
8A:A:V214 5.4325466
9A:A:F219 5.52429768
10A:A:F222 9.195617
11A:A:Q227 6.592519
12A:A:R231 4.6025409
13A:A:K233 6.51519
14A:A:F238 10.522519
15A:A:I244 4.2075418
16A:A:F246 5.958519
17A:A:S250 5.274166
18A:A:L270 7.2075416
19A:A:F273 10.936519
20A:A:W277 10.8117616
21A:A:W281 10.672515
22A:A:L289 4.75419
23A:A:N292 5.885409
24A:A:Q294 9.78254166
25A:A:F312 4.422508
26A:A:F315 10.2775406
27A:A:F345 9.125418
28A:A:I348 6.1975414
29A:A:C359 4.635415
30A:A:Y360 8.444178
31A:A:T364 8.3854119
32A:A:D368 5.684119
33A:A:F376 7.16833668
34A:A:D378 11.1054177
35A:A:N387 3.79428
36A:A:L388 5.0025408
37A:A:Y391 6.436524
38B:B:V40 3.44403
39B:B:M45 5.51254184
40B:B:L51 8.292519
41B:B:H54 9.84519
42B:B:K57 18.72419
43B:B:W63 6.54833607
44B:B:L70 6.63415
45B:B:Q75 16.2925419
46B:B:L79 4.7325407
47B:B:I80 9.2925418
48B:B:W82 11.6667619
49B:B:Y85 11.9975414
50B:B:N88 7.3975407
51B:B:K89 9.645409
52B:B:H91 6.9725405
53B:B:I93 6.1475407
54B:B:L95 4.556578
55B:B:W99 8.84143719
56B:B:Y105 4.396576
57B:B:N110 6.8925454
58B:B:Y111 6.96833654
59B:B:I123 4.10833656
60B:B:Y124 6.28676
61B:B:L126 5.3025475
62B:B:E130 2.426503
63B:B:H142 8.906549
64B:B:Y145 8.37429718
65B:B:C148 4.2875406
66B:B:F151 4.8425859
67B:B:T159 5.546549
68B:B:S160 3.862516
69B:B:D163 7.424549
70B:B:C166 3.736518
71B:B:W169 10.472548
72B:B:F180 8.448517
73B:B:H183 10.8519
74B:B:V187 5.256519
75B:B:M188 5.852518
76B:B:L190 5.108515
77B:B:F199 7.84667619
78B:B:S201 3.68333619
79B:B:C204 4.02507
80B:B:D205 8.355419
81B:B:K209 11.825416
82B:B:L210 7.4175435
83B:B:W211 9.50833618
84B:B:Q220 7.546537
85B:B:F222 8.4025438
86B:B:H225 10.87539
87B:B:D228 8.43419
88B:B:I229 4.5025437
89B:B:I232 5.4825438
90B:B:F234 3.83833605
91B:B:F235 6.2265196
92B:B:F241 9.14636
93B:B:T243 6.62438
94B:B:D247 9.0825409
95B:B:T249 8.37436
96B:B:R251 13.148538
97B:B:F253 7.628536
98B:B:D258 12.1725437
99B:B:L261 4.52405
100B:B:Y264 19.084505
101B:B:I273 5.74406
102B:B:F278 6.622507
103B:B:R283 6.136589
104B:B:Y289 7.725127
105B:B:D290 8.475416
106B:B:N295 7.92754126
107B:B:W297 19.1054128
108B:B:K301 7.3675485
109B:B:H311 9.6056139
110B:B:R314 15.528518
111B:B:C317 3.3225417
112B:B:T321 9.17417
113B:B:M325 8.59167615
114B:B:W332 13.228519
115B:B:D333 8.6254139
116B:B:K337 9.76406
117B:B:I338 5.1325415
118B:B:W339 8.7045189
119G:G:Q18 7.8725409
120G:G:L19 3.912509
121G:G:E22 6.6725409
122G:G:R27 6.925438
123G:G:D48 6.942509
124G:G:L51 4.914506
125G:G:N59 5.5875409
126G:G:F61 8.06571718
127L:L:?1 9.88254200
128R:R:N40 6.42409
129R:R:I47 6.6625148
130R:R:W59 11.925144
131R:R:M64 6.6125429
132R:R:M76 5.7065217
133R:R:W88 8.16407
134R:R:H98 6.1175405
135R:R:H112 7.42528
136R:R:R120 6.074529
137R:R:L128 6.935407
138R:R:R129 7.5154105
139R:R:Y130 6.6627
140R:R:W147 5.31629
141R:R:Y171 12.475493
142R:R:F184 7.335492
143R:R:P201 4.4075408
144R:R:Y209 5.2254229
145R:R:V254 2.0375408
146R:R:W261 9.59407
147R:R:F264 8.165206
148R:R:F265 65206
149R:R:P279 3.8675401
150R:R:Y301 6.766529
151R:R:Y305 5.504528
152R:R:W307 4.886526
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Int. Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.

Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1B:B:K57 B:B:W332 17.155534.81YesYes199
2B:B:K57 B:B:Q75 15.787720.34YesYes199
3B:B:Q75 B:B:W99 15.877110.95YesYes199
4A:A:F238 B:B:W99 16.002614.03YesYes199
5A:A:F238 A:A:L44 17.464323.14YesYes199
6A:A:I244 A:A:L44 17.61994.28YesYes189
7A:A:I244 A:A:V287 35.62893.07YesNo186
8A:A:V287 A:A:W277 54.485712.26NoYes166
9A:A:T350 A:A:W277 79.96289.7NoYes146
10A:A:I358 A:A:T350 1003.04NoNo044
11A:A:I358 A:A:Y360 99.99754.84NoYes048
12A:A:D381 A:A:Y360 97.98266.9NoYes088
13A:A:D381 A:A:Q385 97.97466.53NoNo085
14A:A:Q385 R:R:Q219 97.96746.4NoNo057
15A:A:L384 R:R:Q219 97.95383.99NoNo067
16A:A:L384 R:R:P127 96.74176.57NoNo068
17A:A:N387 R:R:P127 98.61913.26YesNo088
18A:A:N387 R:R:Y130 49.85945.81YesYes287
19A:A:L46 A:A:R231 18.74463.64YesYes089
20A:A:Q227 A:A:W234 74.29825.48YesNo099
21A:A:R231 A:A:W234 74.7835YesNo099
22A:A:Q227 B:B:N119 13.079710.56YesNo199
23A:A:I276 A:A:R231 56.84325.01NoYes089
24A:A:F246 A:A:I276 57.19718.79YesNo098
25A:A:F246 A:A:F273 20.17299.65YesYes199
26A:A:F246 A:A:L289 19.21983.65YesYes199
27A:A:C359 A:A:L289 19.56243.17YesYes159
28A:A:N387 R:R:A123 48.73564.69YesNo288
29A:A:Y391 R:R:A123 48.69255.34YesNo248
30A:A:Y391 R:R:Y130 49.35744.96YesYes247
31A:A:Y391 R:R:R120 95.46978.23YesYes249
32B:B:H62 B:B:Y105 10.66613.27NoYes066
33B:B:H62 B:B:R150 10.944212.41NoNo066
34B:B:C148 B:B:R150 12.33545.57YesNo066
35B:B:C148 B:B:L190 20.46394.76YesYes065
36B:B:K209 B:B:T221 10.191813.51YesNo067
37B:B:S201 B:B:W211 13.34863.71YesYes198
38B:B:C271 B:B:D290 10.45244.67NoYes056
39B:B:C271 B:B:D291 10.27786.22NoNo058
40B:B:D291 B:B:Y289 10.10313.45NoYes087
41R:R:R120 R:R:Y301 94.04074.12YesYes299
42R:R:L113 R:R:Y301 46.91077.03NoYes289
43R:R:L113 R:R:M64 46.77515.65NoYes289
44R:R:H112 R:R:M64 92.97999.19YesYes289
45R:R:H112 R:R:W147 85.48334.23YesYes289
46R:R:L70 R:R:W147 84.37033.42NoYes069
47R:R:L105 R:R:L70 84.08259.69NoNo076
48R:R:L105 R:R:L71 83.21824.15NoNo077
49R:R:L71 R:R:S294 82.64163NoNo079
50R:R:D68 R:R:S294 82.353210.31NoNo099
51R:R:D68 R:R:N40 45.305412.12NoYes099
52R:R:A65 R:R:N40 42.90586.25NoYes099
53R:R:A65 R:R:V43 42.60555.09NoNo099
54R:R:I47 R:R:V43 40.49463.07YesNo089
55R:R:I47 R:R:W59 38.6933.52YesYes1484
56R:R:H54 R:R:W59 37.809715.87NoYes074
57R:R:H54 R:R:K51 37.50779.17NoNo076
58B:B:R52 R:R:K51 37.20558.66NoNo076
59B:B:R52 B:B:T50 16.29979.06NoNo073
60B:B:K337 B:B:T50 15.99479.01YesNo063
61B:B:K337 B:B:W339 28.32829.28YesYes069
62B:B:M45 B:B:W339 24.04164.65YesYes1849
63B:B:M45 G:G:L50 18.5134.24YesNo049
64G:G:D48 G:G:L50 17.89724.07YesNo099
65G:G:D48 G:G:L51 12.35088.14YesYes096
66R:R:N297 R:R:Y301 46.910712.79NoYes299
67R:R:M64 R:R:N297 46.77517.01YesNo299
68B:B:F335 B:B:R52 20.605110.69NoNo047
69B:B:F335 B:B:K337 16.00563.72NoYes046
70B:B:G144 B:B:N119 12.79623.39NoNo089
71B:B:D163 B:B:G144 12.51823.35YesNo098
72B:B:S147 B:B:Y145 49.74893.82NoYes198
73B:B:L190 B:B:S160 20.35064.5YesYes156
74B:B:S160 B:B:V187 11.82864.85YesYes169
75R:R:D68 R:R:T36 38.392314.45NoNo097
76R:R:A295 R:R:T36 38.09063.36NoNo067
77R:R:A295 R:R:I32 37.78894.87NoNo067
78R:R:I32 R:R:M76 37.4878.75NoYes077
79R:R:M76 R:R:Y291 32.64564.79YesNo077
80R:R:D102 R:R:Y291 27.11975.75NoNo067
81L:L:?1 R:R:D102 23.78568.34YesNo006
82L:L:?1 R:R:F264 10.848716.22YesYes2006
83B:B:S147 B:B:S160 49.58613.26NoYes196
84B:B:D163 B:B:H142 10.60247.56YesYes499
85A:A:Q227 B:B:Y145 61.7485.64YesYes198
86B:B:S160 B:B:S201 13.57773.26YesYes169
87A:A:I244 A:A:L46 18.84725.71YesYes188
88A:A:F246 A:A:V287 18.82543.93YesNo196
89A:A:F273 A:A:W277 22.439415.03YesYes196
90A:A:C359 A:A:T350 20.03955.07YesNo154
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1 Node2 LinkStrength Comm IsNode1Hub? IsNode2Hub? Node1Cons Node2Cons Node1Shell Node2Shell
L:L:?1 R:R:D102 8.34 20 Yes No 0 6 0 1
L:L:?1 R:R:F185 4.99 20 Yes No 0 2 0 1
L:L:?1 R:R:F264 16.22 20 Yes Yes 0 6 0 1
L:L:?1 R:R:F265 9.98 20 Yes Yes 0 6 0 1
R:R:D102 R:R:I75 4.2 0 No No 6 6 1 2
R:R:D102 R:R:Y291 5.75 0 No No 6 7 1 2
R:R:F185 R:R:N163 7.25 0 No No 2 4 1 2
R:R:A193 R:R:F185 6.93 0 No No 4 2 2 1
R:R:F194 R:R:F265 5.36 0 No Yes 5 6 2 1
R:R:F194 R:R:T268 5.19 0 No No 5 4 2 2
R:R:F198 R:R:F265 4.29 0 No Yes 7 6 2 1
R:R:F265 R:R:W261 5.01 20 Yes Yes 6 7 1 2
R:R:F264 R:R:F265 5.36 20 Yes Yes 6 6 1 1
R:R:F264 R:R:T268 7.78 20 Yes No 6 4 1 2
R:R:F264 R:R:L286 7.31 20 Yes No 6 5 1 2
R:R:F264 R:R:Y287 4.13 20 Yes No 6 5 1 2

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
60.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
57.14Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
50.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
50.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
50.00Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
50.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
50.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
50.00Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
50.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
50.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
50.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
44.44Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
44.44Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
44.44Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
44.44Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
44.44Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
42.86Single9CHUNoradrenaline9CHU-β2-Noradrenaline
42.86Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
42.86Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
40.00Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
40.00Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
40.00Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
40.00Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
40.00Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
40.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
40.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
40.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
40.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
40.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
40.00Consensusopsins_offOrthosteric Ligandrhodopsin_off
40.00Consensussensory_offOrthosteric Ligandopsins_off
37.50Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
37.50Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
37.50Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
37.50Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.50Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
37.50Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
36.36Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
36.36Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
36.36Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
36.36Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
36.36Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
36.36Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
36.36Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
36.36Single8CU6LJ-45178CU6-A2A-LJ-4517
36.36Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
36.36Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
36.36Single8T1WCVN4248T1W-GPR6-CVN424
36.36Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
36.36Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
36.36Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
36.36Single9CHXS-Carazolol9CHX-β2-S-Carazolol
36.36Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
36.36Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
36.36Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
33.33Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
33.33Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
33.33Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
33.33Single3PBLEticlopride3PBL-D3-Eticlopride
33.33Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
33.33Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
33.33Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
33.33Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
33.33Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
33.33Single6TP4ACT-4622066TP4-OX1-ACT-462206
33.33Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
33.33Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
33.33Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
33.33Single7W41PD1762527W41-BB2-PD176252
33.33Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
33.33Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
33.33Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
33.33Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
33.33Single8JXSPF-61428JXS-D1-PF-6142
33.33Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single9B9Y7DY9B9Y-CB1-7DY
33.33Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
33.33Consensusadenosine_offOrthosteric Liganda1_off a2_off
33.33Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
33.33Consensusbombesin_offOrthosteric Ligandbb2_off
33.33Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
33.33Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
33.33Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
33.33Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
33.33Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Consensustrace-amine_onOrthosteric Ligandta1_on
30.77Single2YDVNECA2YDV-A2A-NECA
30.77Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
30.77Single4UHRCGS216804UHR-A2A-CGS21680
30.77Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
30.77Single5G53NECA5G53-A2A-NECA-Gs
30.77Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
30.77Single6J21Aprepitant6J21-NK1-Aprepitant
30.77Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
30.77Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
30.77Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
30.77Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
30.77Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
30.77Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
30.77Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
30.77Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
30.77Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
30.00Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
30.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
30.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
30.00Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
30.00Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
30.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
30.00Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
30.00Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
30.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
30.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
30.00Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
30.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
30.00Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
30.00Single7F8ULintitript7F8U-CCKA-Lintitript
30.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
30.00Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
30.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
30.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
30.00Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
30.00Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
30.00Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
30.00Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
30.00Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
30.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
30.00Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
30.00Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.00Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
30.00Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
30.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
30.00Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
30.00Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
30.00Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
30.00Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.00Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.00Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.00Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
30.00Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
30.00Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
30.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
30.00Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
30.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
30.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
30.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
30.00Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
30.00Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
30.00Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
30.00Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
30.00Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
30.00Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
30.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
28.57Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
28.57Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
28.57Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
28.57Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
28.57Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
28.57Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
28.57Single7WC4Serotonin7WC4-5-HT2A-Serotonin
28.57Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
28.57Single8PWNTheophylline8PWN-A2A-Theophylline
28.57Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
28.57Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
28.57Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
28.57Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
28.57Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
28.57Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
27.27Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
27.27Single2YDOAdenosine2YDO-A2A-Adenosine
27.27Single3RZECidoxepin3RZE-H1-Cidoxepin
27.27Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
27.27Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
27.27Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
27.27Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
27.27Single5IU7Q274563465IU7-A2A-Q27456346-Na
27.27Single5IUBQ274563445IUB-A2A-Q27456344-Na
27.27Single5JTBZM-2413855JTB-A2A-ZM-241385
27.27Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
27.27Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
27.27Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
27.27Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
27.27Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
27.27Single5UVIZM-2413855UVI-A2A-ZM-241385
27.27Single6A94Zotepine6A94-5-HT2A-Zotepine
27.27Single6AQFZM-2413856AQF-A2A-ZM-241385
27.27Single6IQLL7458706IQL-D4-L745870
27.27Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
27.27Single6KUXRS-799486KUX-α2a-RS-79948
27.27Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
27.27Single6PS0S-Carazolol6PS0-β2-S-Carazolol
27.27Single6PS4ICI118-5516PS4-β2-ICI118-551
27.27Single6PS5S-Propranolol6PS5-β2-S-Propranolol
27.27Single6TPGEMPA6TPG-OX2-EMPA
27.27Single6TPNHTL66416TPN-OX2-HTL6641
27.27Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
27.27Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
27.27Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
27.27Single7AROLUF58337ARO-A2A-LUF5833-Na
27.27Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
27.27Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
27.27Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
27.27Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
27.27Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
27.27Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
27.27Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
27.27Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single7T32ZM-2413857T32-A2A-ZM-241385
27.27Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
27.27Single7VODCariprazine7VOD-5-HT2A-Cariprazine
27.27Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
27.27Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
27.27Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
27.27Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
27.27Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.27Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.27Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
27.27Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
27.27Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
27.27Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
27.27Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
27.27Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
27.27Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
27.27Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
27.27Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
27.27Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
27.27Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
27.27Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
27.27Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
27.27Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
27.27Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
27.27Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.27Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.27Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.27Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.27Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
27.27Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
27.27Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
27.27Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
27.27Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
27.27Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
27.27Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
27.27Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
27.27Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
27.27Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
27.27Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
27.27Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
27.27Consensusa2_offOrthosteric Liganda2a_off
27.27Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
27.27Consensusalpha1_onOrthosteric Ligandalpha1a_on
27.27Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
27.27Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
27.27Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
27.27Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
27.27Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
27.27Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
26.67Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
26.67Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
26.67Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
26.67Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
26.67Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
26.67Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
26.67Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
26.67Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
25.00Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
25.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
25.00Single2Y01Dobutamine2Y01-β1-Dobutamine
25.00Single2Y02Carmoterol2Y02-β1-Carmoterol
25.00Single2Y04Salbutamol2Y04-β1-Salbutamol
25.00Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
25.00Single3EMLZM-2413853EML-A2A-ZM-241385
25.00Single3NY8ICI118-5513NY8-β2-ICI118-551
25.00Single3NY9ICI118-5513NY9-β2-ICI118-551
25.00Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
25.00Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
25.00Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
25.00Single4DAJTiotropium4DAJ-M3-Tiotropium
25.00Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
25.00Single4GBRS-Carazolol4GBR-β2-S-Carazolol
25.00Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
25.00Single4MQSIperoxo4MQS-M2-Iperoxo
25.00Single4U14Tiotropium4U14-M3-Tiotropium
25.00Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
25.00Single4UG2CGS216804UG2-A2A-CGS21680
25.00Single5IU8Q274563475IU8-A2A-Q27456347-Na
25.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
25.00Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
25.00Single5TGZAM65385TGZ-CB1-AM6538
25.00Single5UENDU1725UEN-A1-DU172
25.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
25.00Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
25.00Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
25.00Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
25.00Single6DRXLisuride6DRX-5-HT2B-Lisuride
25.00Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
25.00Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
25.00Single6H7MSalbutamol6H7M-β1-Salbutamol
25.00Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
25.00Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
25.00Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
25.00Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
25.00Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
25.00Single6PS1Timolol6PS1-β2-Timolol
25.00Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
25.00Single6S0LZM-2413856S0L-A2A-ZM-241385
25.00Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
25.00Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
25.00Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
25.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
25.00Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
25.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
25.00Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7PYRPSB-21157PYR-A2A-PSB-2115
25.00Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
25.00Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
25.00Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
25.00Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
25.00Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
25.00Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
25.00Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
25.00Single7WC7Lisuride7WC7-5-HT2A-Lisuride
25.00Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
25.00Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
25.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
25.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
25.00Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
25.00Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
25.00Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
25.00Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
25.00Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
25.00Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
25.00Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
25.00Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
25.00Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
25.00Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
25.00Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
25.00Single8JJOAlprenolol8JJO-β2-Alprenolol
25.00Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
25.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
25.00Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
25.00Single8JXRLSD8JXR-D1-LSD
25.00Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
25.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
25.00Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
25.00Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
25.00Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
25.00Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
25.00Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
25.00Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
25.00Single8X63Mepyramine8X63-H1-Mepyramine
25.00Single8X64Desloratadine8X64-H1-Desloratadine
25.00Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
25.00Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
25.00Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
25.00Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
25.00Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
25.00Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
25.00Consensus5ht5_onOrthosteric Ligand5ht5a_on
25.00Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
25.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
25.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
25.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
25.00Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
25.00Consensusalpha2_onOrthosteric Ligandalpha2b_on
25.00Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
25.00Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
25.00Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
25.00Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
25.00Consensuscck_offOrthosteric Ligandccka_off
25.00Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
25.00Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
25.00Consensusdopamine_offOrthosteric Ligandd2_off d3_off
25.00Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
25.00Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
25.00Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
25.00Consensushistamine_offOrthosteric Ligandh1_off
25.00Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
25.00Consensussensory_onOrthosteric Ligandopsins_on
23.53Single7F8XNN90567F8X-CCKA-NN9056
23.53Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
23.53Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
23.53Single8WDTphotoNECA8WDT-A2A-photoNECA
23.53Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.53Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
23.53Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
23.08Single2RH1S-Carazolol2RH1-β2-S-Carazolol
23.08Single2Y00Dobutamine2Y00-β1-Dobutamine
23.08Single2Y03Isoprenaline2Y03-β1-Isoprenaline
23.08Single2YCWS-Carazolol2YCW-β1-S-Carazolol
23.08Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
23.08Single5C1MBU725C1M-μ-BU72
23.08Single5D6LS-Carazolol5D6L-β2-S-Carazolol
23.08Single5IUAQ274563485IUA-A2A-Q27456348-Na
23.08Single5JQHS-Carazolol5JQH-β2-S-Carazolol
23.08Single5N2RPSB-365N2R-A2A-PSB-36-Na
23.08Single5N2SPSB365N2S-A1-PSB36
23.08Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
23.08Single5TVNLSD5TVN-5-HT2B-LSD
23.08Single5WIUNemonapride5WIU-D4-Nemonapride
23.08Single5WIVNemonapride5WIV-D4-Nemonapride-Na
23.08Single5WQCEMPA5WQC-OX2-EMPA
23.08Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
23.08Single5XPRBosentan5XPR-ETB-Bosentan
23.08Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
23.08Single6D26Fevipiprant6D26-DP2-Fevipiprant
23.08Single6E67BI1671076E67-β2-BI167107-Gs (fused)
23.08Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
23.08Single6HLPNetupitant6HLP-NK1-Netupitant
23.08Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
23.08Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
23.08Single6LUQHaloperidol6LUQ-D2-Haloperidol
23.08Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
23.08Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
23.08Single6PS6Timolol6PS6-β2-Timolol
23.08Single6S0QZM-2413856S0Q-A2A-ZM-241385
23.08Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
23.08Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
23.08Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
23.08Single7C61Ergotamine7C61-5-HT1B-Ergotamine
23.08Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
23.08Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
23.08Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
23.08Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
23.08Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
23.08Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
23.08Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
23.08Single7WC6LSD7WC6-5-HT2A-LSD
23.08Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
23.08Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
23.08Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
23.08Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
23.08Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
23.08Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
23.08Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
23.08Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
23.08Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
23.08Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GNEKW-63568GNE-A2A-KW-6356-Na
23.08Single8QOTNanobody-E8QOT-μ-Nanobody-E
23.08Single8S4DCMF-0198S4D-Apelin-CMF-019
23.08Single8TF5Oleic acid8TF5-GPR6-Oleic acid
23.08Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
23.08Single8ZMFA1L108ZMF-5-HT2C-A1L10
23.08Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
23.08Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
23.08Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
23.08Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
23.08Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
23.08Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
23.08Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
23.08Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
23.08Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
23.08Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
23.08Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
23.08Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
23.08Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
23.08Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
23.08Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
23.08Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
23.08Consensusamine_offonOrthosteric Ligandamine_off amine_on
23.08Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
23.08Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
23.08Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
23.08Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
23.08Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
23.08Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
23.08Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
23.08Consensusdp_offOrthosteric Liganddp2_off
23.08Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
23.08Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
23.08Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
23.08Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
22.22Single3OE6IT1t3OE6-CXCR4-IT1t
22.22Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
22.22Single3QAKUK-4320973QAK-A2A-UK-432097
22.22Single3UZAGTPL92363UZA-A2A-GTPL9236
22.22Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
22.22Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
22.22Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
22.22Single6HLOAprepitant6HLO-NK1-Aprepitant
22.22Single6ME5Agomelatine6ME5-MT1-Agomelatine
22.22Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
22.22Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
22.22Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
22.22Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
22.22Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
22.22Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
22.22Single7WC5Psilocin7WC5-5-HT2A-Psilocin
22.22Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
22.22Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
22.22Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
22.22Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
22.22Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
22.22Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
22.22Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
22.22Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
22.22Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
22.22Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
22.22Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
22.22Consensus5ht2_onOrthosteric Ligand5ht2b_on
22.22Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
22.22Consensusgi_sensoryOrthosteric Ligandgi_opsins
22.22Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
22.22Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
22.22Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
22.22Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
22.22Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
22.22Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
22.22Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
22.22Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
21.43Single3P0GBI1671073P0G-β2-BI167107
21.43Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
21.43Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
21.43Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
21.43Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
21.43Single4U15Tiotropium4U15-M3-Tiotropium
21.43Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
21.43Single5D5AS-Carazolol5D5A-β2-S-Carazolol
21.43Single5D5BS-Carazolol5D5B-β2-S-Carazolol
21.43Single5V54Methiothepin5V54-5-HT1B-Methiothepin
21.43Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
21.43Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
21.43Single6E59L-7607356E59-NK1-L-760735
21.43Single6H7JIsoprenaline6H7J-β1-Isoprenaline
21.43Single6J20Aprepitant6J20-NK1-Aprepitant
21.43Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
21.43Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
21.43Single6OL9Tiotropium6OL9-M5-Tiotropium
21.43Single6TQ7SB-3348676TQ7-OX1-SB-334867
21.43Single6WGTLSD6WGT-5-HT2A-LSD
21.43Single7B6WCyclazosin7B6W-α1b-Cyclazosin
21.43Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
21.43Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
21.43Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
21.43Single7PX4PSB-21137PX4-A2A-PSB-2113
21.43Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
21.43Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
21.43Single7TUYGSK682753A7TUY-GPR183-GSK682753A
21.43Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
21.43Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
21.43Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
21.43Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
21.43Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
21.43Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
21.43Single8E0GBU728E0G-μ-BU72
21.43Single8EA0Iperoxo8EA0-M3-Iperoxo
21.43Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
21.43Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
21.43Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
21.43Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
21.43Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
21.43Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
21.43Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.43Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
21.43Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
21.43Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
21.43Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
21.43Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
21.43Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
21.43Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
21.43Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
21.43Single8XVLZibotentan8XVL-ETA-Zibotentan
21.43Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
21.43Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
21.43Consensus5ht1_offOrthosteric Ligand5ht1b_off
21.43Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
21.43Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
21.43Consensusa2_onOrthosteric Liganda2b_on
21.43Consensusa2_on_gpOrthosteric Liganda2b_on_gp
21.43Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
21.43Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
21.43Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
21.43Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
21.43Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
21.43Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
21.43Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
21.43Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.43Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
21.43Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
21.43Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
21.43Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
21.43Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
21.43Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
21.43Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
21.43Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
21.43Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
21.43Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
21.43Consensustachykinin_offOrthosteric Ligandnk1_off
21.05Single5WF5UK-4320975WF5-A2A-UK-432097
21.05Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
21.05Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
20.00Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
20.00Single3D4STimolol3D4S-β2-Timolol
20.00Single3OE9IT1t3OE9-CXCR4-IT1t
20.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
20.00Single4AMIBucindolol4AMI-β1-Bucindolol
20.00Single4LDEBI1671074LDE-β2-BI167107
20.00Single4RWADIPP-NH24RWA-δ-DIPP-NH2
20.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
20.00Single5CXVTiotropium5CXV-M1-Tiotropium
20.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
20.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
20.00Single6A93Risperidone6A93-5-HT2A-Risperidone
20.00Single6CM4Risperidone6CM4-D2-Risperidone
20.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
20.00Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
20.00Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
20.00Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
20.00Single6HLLCP999946HLL-NK1-CP99994
20.00Single6MXTSalmeterol6MXT-β2-Salmeterol
20.00Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
20.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
20.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
20.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
20.00Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
20.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
20.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
20.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
20.00Single7DFPSpiperone7DFP-D2-Spiperone
20.00Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
20.00Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
20.00Single7SRQLSD7SRQ-5-HT2B-LSD
20.00Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
20.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
20.00Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
20.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
20.00Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
20.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7YITNalfurafine7YIT-κ-Nalfurafine
20.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
20.00Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
20.00Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
20.00Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
20.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
20.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
20.00Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
20.00Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
20.00Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
20.00Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
20.00Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
20.00Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
20.00Single8JJ8Formoterol8JJ8-β2-Formoterol
20.00Single8JJLOlodaterol8JJL-β2-Olodaterol
20.00Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
20.00Single8JWY2-1188JWY-A2A-2-118
20.00Single8K5BNiacin8K5B-HCA2-Niacin
20.00Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
20.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
20.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
20.00Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.00Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
20.00Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
20.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
20.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
20.00Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
20.00Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
20.00Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
20.00Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
20.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
20.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
20.00Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
20.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
20.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
20.00Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
20.00Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
20.00Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
20.00Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
20.00Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
20.00Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
20.00Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
20.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
20.00Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
20.00Consensuslpa_offOrthosteric Ligandlpa1_off
20.00Consensuslpl_offOrthosteric Ligands1p_off lpa_off
20.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
20.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
20.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
20.00Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
20.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
20.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
19.05Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.05Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
18.75Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
18.75Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
18.75Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
18.75Single5X93K-87945X93-ETB-K-8794
18.75Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
18.75Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
18.75Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
18.75Single6H7LDobutamine6H7L-β1-Dobutamine
18.75Single6IBLArformoterol6IBL-β1-Arformoterol
18.75Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
18.75Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
18.75Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
18.75Single7EZCUKA7EZC-A2A-UKA
18.75Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
18.75Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
18.75Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
18.75Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
18.75Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
18.75Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
18.75Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
18.75Single7UM4AS26747237UM4-5-HT5A-AS2674723
18.75Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
18.75Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
18.75Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
18.75Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
18.75Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
18.75Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
18.75Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
18.75Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
18.75Consensuscck_onOrthosteric Ligandccka_on cckb_on
18.75Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
18.75Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
18.75Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
18.75Consensuschemerin_onOrthosteric Ligandcml1_on
18.75Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
18.75Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
18.75Consensusendothelin_offOrthosteric Ligandetb_off
18.75Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
18.75Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
18.75Consensusprostanoid_offOrthosteric Ligandep_off dp_off
18.18Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
18.18Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
18.18Single3ODUIT1t3ODU-CXCR4-IT1t
18.18Single3PWHZM-2413853PWH-A2A-ZM-241385
18.18Single4S0VSuvorexant4S0V-OX2-Suvorexant
18.18Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
18.18Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
18.18Single5U09Taranabant5U09-CB1-Taranabant
18.18Single5WS3EMPA5WS3-OX2-EMPA
18.18Single5ZKQABT-4915ZKQ-PAF-ABT-491
18.18Single6AKXA4R6AKX-CCR5-A4R
18.18Single6AKYMaraviroc6AKY-CCR5-Maraviroc
18.18Single6DS0Ly2660976DS0-5-HT2B-Ly266097
18.18Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
18.18Single6ME9Ramelteon6ME9-MT2-Ramelteon
18.18Single6TODEMPA6TOD-OX1-EMPA-Na
18.18Single6TPJSuvorexant6TPJ-OX2-Suvorexant
18.18Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
18.18Single7BR3Elagolix7BR3-GnRH1-Elagolix
18.18Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
18.18Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
18.18Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
18.18Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
18.18Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
18.18Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
18.18Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
18.18Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
18.18Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
18.18Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
18.18Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
18.18Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
18.18Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
18.18Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
18.18Single7XRRLemborexant7XRR-OX2-Lemborexant
18.18Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
18.18Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
18.18Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
18.18Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
18.18Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
18.18Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
18.18Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
18.18Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
18.18Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
18.18Single8IWESpermidine8IWE-TA9-Spermidine
18.18Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
18.18Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
18.18Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
18.18Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
18.18Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
18.18Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
18.18Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
18.18Single8Y0HVUF114188Y0H-CXCR3-VUF11418
18.18Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
18.18Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
18.18Single9BA0A1AKN9BA0-CB1-A1AKN
18.18Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
18.18Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
18.18Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
18.18Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
18.18Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
18.18Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
18.18Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
18.18Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
18.18Consensusorexin_offOrthosteric Ligandox2_off ox1_off
18.18Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
18.18Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
18.18Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
18.18Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
18.18Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
17.65Single5EE7MK08935EE7-Glucagon-MK0893
17.65Single5WF6UK-4320975WF6-A2A-UK-432097
17.65Single5ZTYAM102575ZTY-CB2-AM10257
17.65Single6PT3DPI-2876PT3-δ-DPI-287
17.65Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
17.65Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
17.65Single7SK9CCX6627SK9-ACKR3-CCX662
17.65Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
17.65Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
17.65Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
17.65Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
17.65Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
17.65Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single8QJ2pN1628QJ2-MC4-pN162-Gs
17.65Single8X5YAstemizole8X5Y-H1-Astemizole
17.65Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
17.65Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
17.65Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
17.65Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
17.65Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
17.65Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
17.65Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
17.39Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
17.39Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
16.67Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
16.67Single3REYXAC3REY-A2A-XAC
16.67Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
16.67Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
16.67Single4IARErgotamine4IAR-5-HT1B-Ergotamine
16.67Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
16.67Single4MBSMaraviroc4MBS-CCR5-Maraviroc
16.67Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
16.67Single4ZJCSB-6740424ZJC-OX1-SB-674042
16.67Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
16.67Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
16.67Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
16.67Single6MH8ZM-2413856MH8-A2A-ZM-241385
16.67Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
16.67Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
16.67Single6TP3Nemorexant6TP3-OX1-Nemorexant
16.67Single6TPKRetosiban6TPK-OT-Retosiban
16.67Single6V9SGTPL114036V9S-OX1-GTPL11403
16.67Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
16.67Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
16.67Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
16.67Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
16.67Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
16.67Single7UL3Famotidine7UL3-H2-Famotidine
16.67Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
16.67Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
16.67Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
16.67Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
16.67Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
16.67Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
16.67Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
16.67Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.67Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
16.67Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
16.67Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
16.67Single8IEBA1LYA8IEB-GPR156-A1LYA
16.67Single8IHKAcifran8IHK-HCA3-Acifran
16.67Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
16.67Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
16.67Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
16.67Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
16.67Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
16.67Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
16.67Single8K5CAcipimox8K5C-HCA2-Acipimox
16.67Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
16.67Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
16.67Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
16.67Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
16.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
16.67Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
16.67Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
16.67Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
16.67Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
16.67Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
16.67Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
16.67Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9BJKNaloxone9BJK-μ-Naloxone-NAM
16.67Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
16.67Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
16.67Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
16.67Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
16.67Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
16.67Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
16.67Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
16.67Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
16.67Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
16.67Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
16.67Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
16.67Consensusgrh_offOrthosteric Ligandgnrh1_off
16.67Consensushca_onOrthosteric Ligandhca2_on
16.67Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
16.67Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
16.67Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
16.67Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
16.67Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
16.67Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Consensusvasop-oxy_offOrthosteric Ligandot_off
16.00Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
16.00Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
16.00Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
16.00Consensusbombesin_onOrthosteric Ligandbb2_on
16.00Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
16.00Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
16.00Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
15.79Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
15.79Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
15.79Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
15.79Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
15.79Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.79Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
15.79Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
15.79Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.79Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
15.79Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
15.79Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
15.79Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
15.38Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
15.38Single4EJ4Naltrindole4EJ4-δ-Naltrindole
15.38Single4QKX35V4QKX-β2-35V
15.38Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
15.38Single5DHGC-355DHG-NOP-C-35
15.38Single5DHHSB-6121115DHH-NOP-SB-612111
15.38Single5DSGTiotropium5DSG-M4-Tiotropium
15.38Single5UIGCmpd-15UIG-A2A-Cmpd-1
15.38Single6D27CAY104716D27-DP2-CAY10471
15.38Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
15.38Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
15.38Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
15.38Single6IIVDaltroban6IIV-TP-Daltroban
15.38Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
15.38Single6TOTLemborexant6TOT-OX1-Lemborexant
15.38Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
15.38Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
15.38Single7BU7BI1671077BU7-β1-BI167107
15.38Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
15.38Single7F83PF-051904577F83-Ghrelin-PF-05190457
15.38Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
15.38Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
15.38Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
15.38Single7UL4Alvimopan7UL4-μ-Alvimopan
15.38Single7V3ZCP559407V3Z-CB1-CP55940
15.38Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
15.38Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
15.38Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
15.38Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
15.38Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
15.38Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
15.38Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
15.38Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
15.38Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
15.38Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
15.38Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
15.38Single8RLNLUF58348RLN-A2A-LUF5834
15.38Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
15.38Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
15.38Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
15.38Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
15.38Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
15.38Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
15.38Single9B9ZA1AKO9B9Z-CB1-A1AKO
15.38Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
15.38Consensusa3_onOrthosteric Liganda3a_on
15.38Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
15.38Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
15.38Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
15.38Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
15.38Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
15.38Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
15.38Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
15.38Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
15.38Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
15.38Consensushca_on_gpOrthosteric Ligandhca2_on_gp
15.38Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
15.38Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
15.38Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
15.38Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
15.38Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
15.38Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
15.00Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
15.00Single6PT2KGCHM076PT2-δ-KGCHM07
15.00Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
15.00Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
15.00Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
15.00Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
15.00Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.00Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.00Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
15.00Consensusangiotensin_onOrthosteric Ligandat1_on
15.00Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
15.00Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
15.00Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
15.00Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
15.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
15.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
15.00Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
15.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
15.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
14.29Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
14.29Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
14.29Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
14.29Single5CGCHTL142425CGC-mGlu5-HTL14242
14.29Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
14.29Single5MZPCaffeine5MZP-A2A-Caffeine-Na
14.29Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
14.29Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
14.29Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
14.29Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
14.29Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
14.29Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
14.29Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
14.29Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
14.29Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
14.29Single6TP6Filorexant6TP6-OX1-Filorexant
14.29Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
14.29Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
14.29Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
14.29Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
14.29Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
14.29Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
14.29Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
14.29Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
14.29Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
14.29Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
14.29Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
14.29Single7SINNPS-21437SIN-CaS-NPS-2143
14.29Single7SINNPS-21437SIN-CaS-NPS-2143
14.29Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
14.29Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
14.29Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
14.29Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
14.29Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
14.29Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
14.29Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
14.29Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
14.29Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
14.29Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
14.29Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
14.29Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
14.29Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
14.29Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
14.29Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
14.29Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
14.29Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
14.29Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
14.29Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
14.29Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
14.29Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
14.29Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
14.29Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
14.29Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
14.29Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusa3_on_gpOrthosteric Liganda3a_on_gp
14.29Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.29Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.29Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
14.29Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
14.29Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
14.29Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
14.29Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
14.29Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
14.29Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
14.29Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
14.29Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
14.29Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
14.29Consensusep_offOrthosteric Ligandep4_off
14.29Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
14.29Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
14.29Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
14.29Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
14.29Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
14.29Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
14.29Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
14.29Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
14.29Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
14.29Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
14.29Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
13.64Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
13.64Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
13.64Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.64Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
13.64Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
13.64Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
13.64Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
13.64Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
13.64Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
13.64Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
13.64Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
13.64Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
13.64Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
13.64Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
13.64Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
13.64Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
13.64Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
13.64Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.33Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
13.33Single5TZRMK86665TZR-FFA1-MK8666
13.33Single5XR8AM8415XR8-CB1-AM841
13.33Single5XRAAM115425XRA-CB1-AM11542
13.33Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
13.33Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
13.33Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
13.33Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
13.33Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.33Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
13.33Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
13.33Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
13.33Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
13.33Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
13.33Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
13.33Single7R0CAVP7R0C-V2-AVP-Arrestin2
13.33Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
13.33Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
13.33Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
13.33Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
13.33Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
13.33Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
13.33Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
13.33Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
13.33Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
13.33Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
13.33Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
13.33Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
13.33Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
13.33Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
13.33Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
13.33Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.33Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
13.33Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
13.33Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
13.33Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
13.33Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
13.33Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
13.33Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
13.33Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
13.33Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
13.33Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
13.33Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
13.33Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.33Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
13.33Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
13.33Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
13.33Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.33Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.33Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.33Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
13.33Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
13.33Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
13.33Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
13.04Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
13.04Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
13.04Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
13.04Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
13.04Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
13.04Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
13.04Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
13.04Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.04Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.04Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
12.50Single4N4WSANT-14N4W-SMO-SANT-1
12.50Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
12.50Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
12.50Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
12.50Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
12.50Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
12.50Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
12.50Single6IIURamatroban6IIU-TP-Ramatroban
12.50Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
12.50Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
12.50Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
12.50Single6ZG4HTL00099366ZG4-M1-HTL0009936
12.50Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
12.50Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
12.50Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
12.50Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
12.50Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
12.50Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
12.50Single7K15MKD0467K15-BLT1-MKD046-Na
12.50Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
12.50Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
12.50Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
12.50Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
12.50Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
12.50Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.50Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
12.50Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
12.50Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
12.50Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
12.50Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
12.50Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
12.50Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
12.50Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
12.50Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
12.50Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
12.50Single8JWZAB9288JWZ-A2A-AB928-Na
12.50Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
12.50Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
12.50Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
12.50Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
12.50Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
12.50Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
12.50Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.50Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
12.50Single8XYIVUF106618XYI-CXCR3-VUF10661
12.50Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
12.50Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
12.50Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
12.50Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
12.50Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
12.50Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
12.50Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
12.50Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.50Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
12.50Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
12.50Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
12.50Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
12.50Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
12.50Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
12.50Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
12.50Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
12.50Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
12.50Consensusorexin_onOrthosteric Ligandox2_on
12.50Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
12.50Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
12.50Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
12.50Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.00Single6IGLIRL16206IGL-ETB-IRL1620
12.00Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
12.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
12.00Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
12.00Single8IY6Endothelin-18IY6-ETB-Endothelin-1
12.00Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
12.00Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
12.00Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
12.00Consensusbradykinin_onOrthosteric Ligandbk2_on
12.00Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
12.00Consensusendothelin_onOrthosteric Ligandetb_on eta_on
12.00Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
12.00Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
11.76Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
11.76Single5CGDHTL142425CGD-mGlu5-HTL14242
11.76Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
11.76Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
11.76Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
11.76Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
11.76Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
11.76Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
11.76Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
11.76Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
11.76Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
11.76Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
11.76Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
11.76Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
11.76Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
11.76Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
11.76Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
11.76Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
11.76Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
11.76Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
11.76Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
11.76Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
11.76Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
11.76Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
11.76Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
11.76Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
11.76Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
11.76Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
11.76Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single5GLHEndothelin-15GLH-ETB-Endothelin-1
11.54Single6IGKEndothelin-36IGK-ETB-Endothelin-3
11.54Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
11.54Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
11.11Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
11.11Single3OE8IT1t3OE8-CXCR4-IT1t
11.11Single3RFMCaffeine3RFM-A2A-Caffeine
11.11Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
11.11Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
11.11Single6KNMJN241-96KNM-Apelin-JN241-9
11.11Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
11.11Single6TQ9SB-4081246TQ9-OX1-SB-408124
11.11Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
11.11Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
11.11Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
11.11Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
11.11Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
11.11Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
11.11Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
11.11Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
11.11Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
11.11Single7XN9L-054,5227XN9-SST2-L-054,522
11.11Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
11.11Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
11.11Single8IEIA1LYA8IEI-GPR156-A1LYA
11.11Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
11.11Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
11.11Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
11.11Single8XQJJN2418XQJ-Apelin-JN241
11.11Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
11.11Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
11.11Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
11.11Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
11.11Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
11.11Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
11.11Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
11.11Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
11.11Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
11.11Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
11.11Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
11.11Consensuskisspeptin_onOrthosteric Ligandkiss1_on
11.11Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
11.11Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
11.11Consensusp2y_offOrthosteric Ligandp2y1_off
11.11Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
11.11Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
10.71Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
10.71Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
10.53Single4XT1Fractalkine4XT1-US28-Fractalkine
10.53Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
10.53Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
10.53Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
10.53Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
10.53Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
10.53Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
10.53Single7QA8Peptide7QA8-STE2-Peptide
10.53Single7QA8Peptide7QA8-STE2-Peptide
10.53Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
10.53Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
10.53Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
10.53Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
10.53Single8IEIA1LYA8IEI-GPR156-A1LYA
10.53Single8IEPA1LYA8IEP-GPR156-A1LYA
10.53Single8IEPA1LYA8IEP-GPR156-A1LYA
10.53Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
10.53Single8KIGSHU91198KIG-MC3-SHU9119-Ca
10.53Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
10.53Single8WKYPG-9348WKY-MC4-PG-934
10.53Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.53Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
10.53Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
10.53Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.53Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.53Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
10.53Consensuslpl_onOrthosteric Ligands1p_on lpa_on
10.53Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
10.53Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
10.53Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
10.00Single4XNWMRS25004XNW-P2Y1-MRS2500
10.00Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
10.00Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
10.00Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
10.00Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
10.00Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
10.00Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
10.00Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
10.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
10.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
10.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
10.00Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
10.00Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
10.00Single7V6A-7V6A-M4-PubChem 9864275-Gi1/β1/γ2
10.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
10.00Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
10.00Single7XNACYN1548067XNA-SST2-CYN154806
10.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.00Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
10.00Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
10.00Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
10.00Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
10.00Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8IEBA1LYA8IEB-GPR156-A1LYA
10.00Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
10.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
10.00Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
10.00Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
10.00Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
10.00Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
10.00Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
10.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
10.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
10.00Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
10.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
10.00Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
10.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
10.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
10.00Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
10.00Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
10.00Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
10.00Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
10.00Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
10.00Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
10.00Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
10.00Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
10.00Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
9.68Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
9.68Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
9.52Single3OE0CVX153OE0-CXCR4-CVX15
9.52Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
9.52Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
9.52Single6W25SHU91196W25-MC4-SHU9119-Ca
9.52Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
9.52Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
9.52Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
9.52Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
9.52Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
9.52Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
9.52Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
9.52Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
9.52Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
9.52Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
9.52Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
9.52Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
9.52Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
9.52Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
9.52Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
9.52Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
9.52Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
9.09Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
9.09Single4O9RCyclopamine4O9R-SMO-Cyclopamine
9.09Single5L7IVismodegib5L7I-SMO-Vismodegib
9.09Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
9.09Single6JODAngiotensin II6JOD-AT2-Angiotensin II
9.09Single6LI0C176LI0-GPR52-C17
9.09Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
9.09Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
9.09Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
9.09Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
9.09Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
9.09Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
9.09Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
9.09Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
9.09Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
9.09Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
9.09Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
9.09Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
9.09Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
9.09Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
9.09Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
9.09Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
9.09Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
9.09Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
9.09Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
9.09Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
9.09Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
9.09Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
9.09Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
9.09Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
9.09Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
9.09Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
9.09Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
9.09Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.09Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
9.09Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
9.09Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
9.09Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
9.09Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
9.09Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
9.09Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
9.09Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
9.09Consensusgq_nucleotideOrthosteric Ligandgq_p2y
9.09Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.09Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
9.09Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
9.09Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
9.09Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
9.09Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
9.09Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
9.09Consensusvasop-oxy_onOrthosteric Ligandv2_on
9.09Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
8.70Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
8.70Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
8.70Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
8.70Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
8.70Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
8.70Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
8.70Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
8.70Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
8.70Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
8.70Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
8.70Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
8.70Single8ZRTET-18ZRT-ETB-ET-1
8.70Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
8.70Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
8.70Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
8.70Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
8.33Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
8.33Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
8.33Single4BWBNeurotensin4BWB-NTS1-Neurotensin
8.33Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
8.33Single4QINSAG1.54QIN-SMO-SAG1.5
8.33Single4XT3Fractalkine4XT3-US28-Fractalkine
8.33Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
8.33Single6B73MP11046B73-κ-MP1104
8.33Single6FJ3PTH6FJ3-PTH1-PTH
8.33Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
8.33Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
8.33Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
8.33Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
8.33Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
8.33Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
8.33Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
8.33Single7F8YDevazepide7F8Y-CCKA-Devazepide
8.33Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
8.33Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
8.33Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
8.33Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
8.33Single7SK3CXCL127SK3-ACKR3-CXCL12
8.33Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
8.33Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
8.33Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
8.33Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
8.33Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
8.33Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
8.33Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
8.33Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
8.33Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
8.33Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
8.33Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
8.33Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
8.33Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
8.33Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
8.33Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
8.33Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
8.33Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
8.33Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
8.33Consensusangiotensin_offOrthosteric Ligandat1_off
8.33Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
8.33Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
8.33Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.33Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.33Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
8.33Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
8.33Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
8.33Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
8.33Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
8.33Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
8.33Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
8.11Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
8.00Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
8.00Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
8.00Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
8.00Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
8.00Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
8.00Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
8.00Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
8.00Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
8.00Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
8.00Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
8.00Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
7.69Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
7.69Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
7.69Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
7.69Single6FFIMMPEP6FFI-mGlu5-MMPEP
7.69Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
7.69Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
7.69Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
7.69Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
7.69Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
7.69Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
7.69Single6VI4JDTic6VI4-κ-JDTic
7.69Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
7.69Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
7.69Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
7.69Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
7.69Single6ZG9GSK10347026ZG9-M1-GSK1034702
7.69Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
7.69Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
7.69Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
7.69Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
7.69Single7VV6C48/807VV6-MRGPRX2-C48/80
7.69Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
7.69Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
7.69Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
7.69Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
7.69Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
7.69Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
7.69Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
7.69Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
7.69Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
7.69Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8JD6N-(3-chlorophenyl)pyridine-2-carboxamide8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
7.69Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
7.69Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
7.69Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
7.69Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
7.69Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
7.69Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
7.69Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
7.69Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
7.69Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
7.69Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
7.41Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
7.41Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
7.41Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
7.41Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
7.41Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
7.14Single4QIMANTA XV4QIM-SMO-ANTA XV
7.14Single4YAYZD-71554YAY-AT1-ZD-7155
7.14Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
7.14Single5T04Neurotensin5T04-NTS1-Neurotensin
7.14Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
7.14Single6FFHFenobam6FFH-mGlu5-Fenobam
7.14Single6GPSMK08126GPS-CCR2-MK0812
7.14Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
7.14Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
7.14Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
7.14Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
7.14Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
7.14Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
7.14Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
7.14Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
7.14Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
7.14Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
7.14Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.14Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
7.14Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
7.14Single7YXAONO-54306087YXA-S1P5-ONO-5430608
7.14Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
7.14Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
7.14Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
7.14Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
7.14Single8K5DGSK2560738K5D-HCA2-GSK256073
7.14Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
7.14Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
7.14Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
7.14Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
7.14Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
7.14Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
7.14Single9IYAONO-97105319IYA-GPR55-ONO-9710531
7.14Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
7.14Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
7.14Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
7.14Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.14Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.14Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
7.14Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
6.90Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
6.90Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
6.90Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.67Single4JKVTaladegib4JKV-SMO-Taladegib
6.67Single4NTJAZD12834NTJ-P2Y12-AZD1283
6.67Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
6.67Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
6.67Single6GPXMK08126GPX-CCR2-MK0812
6.67Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
6.67Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
6.67Single7C4SS1P7C4S-S1P3-S1P
6.67Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.67Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
6.67Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
6.67Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
6.67Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
6.67Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
6.67Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
6.67Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
6.67Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
6.67Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
6.67Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
6.67Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
6.67Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
6.67Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
6.67Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
6.67Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
6.67Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
6.67Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
6.67Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.67Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
6.67Consensusblt_offOrthosteric Ligandblt1_off
6.67Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
6.67Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
6.67Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
6.67Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
6.67Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
6.67Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
6.67Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
6.45Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
6.25Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
6.25Single4BV0Neurotensin4BV0-NTS1-Neurotensin
6.25Single4DJHJDTic4DJH-κ-JDTic
6.25Single5V56TC1145V56-SMO-TC114
6.25Single5V57TC1145V57-SMO-TC114
6.25Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
6.25Single6OS1TRV0266OS1-AT1-TRV026
6.25Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
6.25Single7F1TMIP-1a7F1T-CCR5-MIP-1a
6.25Single7FEECP559407FEE-CB1-CP55940-ZCZ011
6.25Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
6.25Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
6.25Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
6.25Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
6.25Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
6.25Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
6.25Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
6.25Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
6.25Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
6.25Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
6.25Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
6.25Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.25Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
6.25Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
6.25Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
6.25Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
6.25Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
6.25Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
6.25Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
6.25Single9BJKNAM9BJK-μ-Naloxone-NAM
6.25Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
6.25Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
6.25Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
6.25Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
6.25Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
6.25Consensuslpa_onOrthosteric Ligandlpa1_on
6.25Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
6.25Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusneurotensin_onOrthosteric Ligandnts1_on
6.25Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
6.25Consensusrelaxin_onOrthosteric Ligandrxfp4_on
6.25Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
6.06Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
5.88Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
5.88Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
5.88Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
5.88Single4PY02MeSATP4PY0-P2Y12-2MeSATP
5.88Single4XEENeurotensin4XEE-NTS1-Neurotensin
5.88Single4XESNeurotensin4XES-NTS1-Neurotensin
5.88Single5X33BIIL2605X33-BLT1-BIIL260
5.88Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
5.88Single6KQICP559406KQI-CB1-CP55940-Org27569
5.88Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
5.88Single6OS2TRV0266OS2-AT1-TRV026
5.88Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
5.88Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
5.88Single6YVRNTS8-136YVR-NTS1-NTS8-13
5.88Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
5.88Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
5.88Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
5.88Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
5.88Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
5.88Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
5.88Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
5.88Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
5.88Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
5.88Single8XQJJN2418XQJ-Apelin-JN241
5.88Single8XWACXCL18XWA-CXCR2-CXCL1
5.88Single8XWMCXCL68XWM-CXCR2-CXCL6
5.88Single8XWSCXCL58XWS-CXCR2-CXCL5
5.88Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
5.88Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
5.88Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
5.88Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
5.88Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
5.88Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
5.88Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
5.71Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
5.56Single4BUONeurotensin4BUO-NTS1-Neurotensin
5.56Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
5.56Single6K1QIRL25006K1Q-ETB-IRL2500
5.56Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
5.56Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
5.56Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
5.56Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.56Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
5.56Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
5.56Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
5.56Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
5.56Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
5.56Single8XVJMacitentan8XVJ-ETA-Macitentan
5.56Single8XVUCXCL28XVU-CXCR2-CXCL2
5.56Single8XWFCXCL38XWF-CXCR2-CXCL3
5.56Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
5.56Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
5.56Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
5.56Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
5.56Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
5.56Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
5.56Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
5.56Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.26Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
5.26Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
5.26Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
5.26Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
5.26Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
5.26Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
5.26Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
5.26Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
5.26Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
5.26Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
5.00Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
5.00Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
5.00Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
5.00Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
5.00Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
5.00Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
5.00Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.00Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
5.00Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
5.00Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
5.00Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
5.00Single8XWNCXCL88XWN-CXCR2-CXCL8
5.00Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
5.00Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
5.00Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
5.00Consensussomatostatin_offOrthosteric Ligandsst2_off
4.76Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
4.76Single7SK5CXCL127SK5-ACKR3-CXCL12
4.76Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
4.76Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
4.76Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
4.55Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
4.55Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
4.55Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
4.55Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
4.35Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
4.35Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
4.35Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
4.35Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
4.35Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
4.17Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
4.17Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
4.17Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
4.17Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
4.17Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
4.17Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
4.17Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
4.00Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
4.00Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
4.00Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
4.00Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
4.00Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
4.00Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
4.00Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
4.00Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
4.00Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
3.85Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
3.85Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
3.85Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
3.85Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
3.85Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
3.85Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
3.85Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
3.85Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
3.70Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
3.70Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
3.70Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
3.70Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
3.57Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
3.57Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
3.45Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
3.33Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
3.33Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
3.33Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
3.23Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
3.23Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
3.23Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2

PDB Summary
PDB 8WCB
Class A
SubFamily Amine
Type Trace Amine Receptors
SubType TA1
Species Mus Musculus
Ligand Cyclohexylammonium Ion
Other Ligand(s) -
Protein Partners chim(NtGi1-Gs-CtGq)/Beta1/Gamma2
PDB Resolution 3.1
Date 2023-12-27
D.O.I. 10.1016/j.cell.2023.10.014
Net Summary
Imin 3.04
Number of Linked Nodes 797
Number of Links 970
Number of Hubs 152
Number of Links mediated by Hubs 555
Number of Communities 22
Number of Nodes involved in Communities 210
Number of Links involved in Communities 313
Path Summary
Number Of Nodes in MetaPath 91
Number Of Links MetaPath 90
Number of Shortest Paths 2742980
Length Of Smallest Path 3
Average Path Length 40.2561
Length of Longest Path 65
Minimum Path Strength 1.16
Average Path Strength 6.74574
Maximum Path Strength 37.66
Minimum Path Correlation 0.7
Average Path Correlation 0.987464
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.22222
Average % Of Corr. Nodes 31.4939
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 46.499
Maximum Path Hubs % 100
AnnotationTypeLinks
Gene OntologyMolecular Function• D2 dopamine receptor binding   • protein binding   • binding   • signaling receptor binding   • G protein-coupled receptor binding   • dopamine receptor binding   • phosphorus-oxygen lyase activity   • enzyme regulator activity   • cyclase regulator activity   • molecular function regulator activity   • cyclase activity   • adenylate cyclase regulator activity   • lyase activity   • catalytic activity   • adenylate cyclase activity   • guanyl nucleotide binding   • GTP binding   • nucleotide binding   • guanyl ribonucleotide binding   • purine ribonucleotide binding   • purine ribonucleoside triphosphate binding   • nucleoside phosphate binding   • ion binding   • purine nucleotide binding   • anion binding   • heterocyclic compound binding   • carbohydrate derivative binding   • ribonucleotide binding   • small molecule binding   • cation binding   • magnesium ion binding   • metal ion binding   • GDP binding   • G protein-coupled serotonin receptor binding   • protein-containing complex binding   • G-protein beta/gamma-subunit complex binding   • pyrophosphatase activity   • GTPase activity   • G protein activity   • ribonucleoside triphosphate phosphatase activity   • hydrolase activity, acting on acid anhydrides, in phosphorus-containing anhydrides   • hydrolase activity   • hydrolase activity, acting on acid anhydrides   • D1 dopamine receptor binding   • molecular function activator activity   • enzyme activator activity   • cyclase activator activity   • adenylate cyclase activator activity   • cellular response to stimulus   • regulation of biological process   • regulation of cellular process   • response to stimulus   • signaling   • biological regulation   • adenylate cyclase-inhibiting serotonin receptor signaling pathway   • G protein-coupled serotonin receptor signaling pathway   • cell communication   • adenylate cyclase-inhibiting G protein-coupled receptor signaling pathway   • adenylate cyclase-modulating G protein-coupled receptor signaling pathway   • G protein-coupled receptor signaling pathway   • cellular process   • signal transduction
Gene OntologyBiological Process• cellular response to stimulus   • regulation of biological process   • regulation of cellular process   • response to stimulus   • signaling   • biological regulation   • adenylate cyclase-inhibiting serotonin receptor signaling pathway   • G protein-coupled serotonin receptor signaling pathway   • cell communication   • adenylate cyclase-inhibiting G protein-coupled receptor signaling pathway   • adenylate cyclase-modulating G protein-coupled receptor signaling pathway   • G protein-coupled receptor signaling pathway   • cellular process   • signal transduction   • response to hormone   • response to chemical   • response to endogenous stimulus   • response to peptide hormone   • response to oxygen-containing compound   • response to nitrogen compound   • cell division   • leukocyte migration   • immune system process   • mononuclear cell migration   • lymphocyte migration   • cell migration   • T cell migration   • cell motility   • regulation of steroid biosynthetic process   • regulation of cholesterol biosynthetic process   • regulation of cholesterol metabolic process   • steroid metabolic process   • regulation of lipid metabolic process   • sterol metabolic process   • positive regulation of biological process   • cholesterol metabolic process   • lipid biosynthetic process   • alcohol metabolic process   • regulation of primary metabolic process   • positive regulation of metabolic process   • regulation of small molecule metabolic process   • positive regulation of biosynthetic process   • positive regulation of lipid metabolic process   • small molecule metabolic process   • steroid biosynthetic process   • positive regulation of cellular process   • regulation of biosynthetic process   • secondary alcohol biosynthetic process   • regulation of alcohol biosynthetic process   • small molecule biosynthetic process   • regulation of steroid metabolic process   • cholesterol biosynthetic process   • positive regulation of cholesterol biosynthetic process   • primary metabolic process   • secondary alcohol metabolic process   • positive regulation of steroid biosynthetic process   • biosynthetic process   • sterol biosynthetic process   • positive regulation of lipid biosynthetic process   • regulation of sterol biosynthetic process   • alcohol biosynthetic process   • positive regulation of cholesterol metabolic process   • positive regulation of steroid metabolic process   • metabolic process   • regulation of lipid biosynthetic process   • positive regulation of small molecule metabolic process   • regulation of metabolic process   • positive regulation of alcohol biosynthetic process   • positive regulation of sterol biosynthetic process   • lipid metabolic process   • regulation of cytoskeleton organization   • regulation of cellular component organization   • microtubule cytoskeleton organization   • regulation of mitotic spindle organization   • mitotic cell cycle   • cellular component organization   • cell cycle   • cellular component organization or biogenesis   • regulation of cell cycle   • microtubule cytoskeleton organization involved in mitosis   • spindle organization   • cell cycle process   • regulation of cell cycle process   • regulation of microtubule-based process   • regulation of spindle organization   • regulation of organelle organization   • mitotic spindle organization   • organelle organization   • mitotic cell cycle process   • microtubule-based process   • cytoskeleton organization   • regulation of microtubule cytoskeleton organization   • protein localization   • positive regulation of protein localization to cell periphery   • regulation of localization   • protein localization to cell periphery   • cellular localization   • regulation of protein localization   • positive regulation of protein localization to cell cortex   • regulation of protein localization to cell periphery   • localization   • regulation of cellular localization   • regulation of protein localization to cell cortex   • cellular macromolecule localization   • macromolecule localization   • positive regulation of protein localization   • protein localization to cell cortex   • response to ketone   • response to prostaglandin   • response to lipid   • response to alcohol   • response to prostaglandin E   • cellular response to forskolin   • cellular response to oxygen-containing compound   • cellular response to chemical stimulus   • cellular response to alcohol   • response to forskolin   • cellular response to lipid   • cellular response to ketone   • developmental process   • multicellular organismal process   • epithelium development   • ectodermal placode morphogenesis   • epidermis development   • molting cycle process   • hair cycle   • animal organ development   • hair follicle placode formation   • tissue development   • ectodermal placode formation   • anatomical structure morphogenesis   • skin development   • skin epidermis development   • hair follicle development   • molting cycle   • anatomical structure development   • anatomical structure formation involved in morphogenesis   • ectodermal placode development   • hair cycle process   • system process   • sensory perception of chemical stimulus   • sensory perception   • nervous system process   • sensory perception of smell   • cellular response to nitrogen compound   • cellular response to peptide hormone stimulus   • response to glucagon   • cellular response to glucagon stimulus   • cellular response to endogenous stimulus   • cellular response to hormone stimulus   • multicellular organism development   • skeletal system development   • bone development   • system development   • regulation of body fluid levels   • wound healing   • homotypic cell-cell adhesion   • cell activation   • hemostasis   • platelet aggregation   • blood coagulation   • cell adhesion   • cell-cell adhesion   • response to stress   • coagulation   • regulation of biological quality   • response to wounding   • platelet activation   • response to fluid shear stress   • vascular endothelial cell response to laminar fluid shear stress   • response to laminar fluid shear stress   • cellular response to stress   • cellular response to laminar fluid shear stress   • vascular endothelial cell response to fluid shear stress   • cellular response to fluid shear stress   • cognition   • developmental growth   • growth   • cellular response to prostaglandin stimulus   • cellular response to prostaglandin E stimulus   • adenylate cyclase-activating G protein-coupled receptor signaling pathway   • homeostatic process   • adaptive thermogenesis   • multicellular organismal-level homeostasis   • regulation of cold-induced thermogenesis   • cold-induced thermogenesis   • temperature homeostasis   • positive regulation of cold-induced thermogenesis   • positive regulation of multicellular organismal process   • regulation of multicellular organismal process   • establishment of protein localization   • nitrogen compound transport   • regulation of peptide hormone secretion   • regulation of hormone levels   • establishment of protein localization to extracellular region   • protein secretion   • establishment of localization   • regulation of protein secretion   • regulation of secretion   • regulation of hormone secretion   • regulation of peptide secretion   • transport   • hormone secretion   • protein localization to extracellular region   • peptide secretion   • regulation of secretion by cell   • secretion by cell   • amide transport   • signal release   • regulation of signaling   • regulation of transport   • secretion   • regulation of peptide transport   • regulation of establishment of protein localization   • export from cell   • cell-cell signaling   • regulation of protein transport   • peptide transport   • protein transport   • regulation of insulin secretion   • peptide hormone secretion   • hormone transport   • regulation of cell communication   • insulin secretion   • adenylate cyclase-activating adrenergic receptor signaling pathway   • adrenergic receptor signaling pathway   • establishment of localization in cell   • intracellular transport   • regulation of defense response   • regulation of response to external stimulus   • negative regulation of inflammatory response   • negative regulation of biological process   • inflammatory response to antigenic stimulus   • regulation of response to stress   • regulation of immune system process   • negative regulation of inflammatory response to antigenic stimulus   • defense response   • immune response   • negative regulation of response to stimulus   • negative regulation of immune response   • regulation of inflammatory response to antigenic stimulus   • response to external stimulus   • regulation of inflammatory response   • regulation of response to stimulus   • negative regulation of immune system process   • negative regulation of response to external stimulus   • negative regulation of defense response   • regulation of immune response   • inflammatory response   • positive regulation of adenylate cyclase activity   • positive regulation of molecular function   • regulation of molecular function   • positive regulation of cyclase activity   • activation of adenylate cyclase activity   • regulation of adenylate cyclase activity   • regulation of catalytic activity   • positive regulation of catalytic activity   • positive regulation of lyase activity   • response to dopamine   • cellular response to dopamine   • response to monoamine   • response to catecholamine   • adenylate cyclase-activating dopamine receptor signaling pathway   • cellular response to catecholamine stimulus   • G protein-coupled dopamine receptor signaling pathway   • cellular response to monoamine stimulus   • renal system process   • chemical homeostasis   • multicellular organismal-level water homeostasis   • multicellular organismal-level chemical homeostasis   • renal water homeostasis   • midbody   • cellular anatomical structure   • membrane-bounded organelle   • intracellular anatomical structure   • nucleus   • membrane-enclosed lumen   • intracellular membraneless organelle   • intracellular membrane-bounded organelle   • nucleolus   • intracellular organelle lumen   • intracellular organelle   • organelle lumen   • organelle   • membraneless organelle
Gene OntologyCellular Component• midbody   • cellular anatomical structure   • membrane-bounded organelle   • intracellular anatomical structure   • nucleus   • membrane-enclosed lumen   • intracellular membraneless organelle   • intracellular membrane-bounded organelle   • nucleolus   • intracellular organelle lumen   • intracellular organelle   • organelle lumen   • organelle   • membraneless organelle   • nuclear lumen   • cell periphery   • cell cortex   • cytoplasm   • protein-containing complex   • extrinsic component of plasma membrane   • catalytic complex   • plasma membrane protein complex   • cytoplasmic side of membrane   • membrane   • plasma membrane   • membrane protein complex   • heterotrimeric G-protein complex   • side of membrane   • cytoplasmic side of plasma membrane   • GTPase complex   • extrinsic component of membrane   • extrinsic component of cytoplasmic side of plasma membrane   • extracellular exosome   • extracellular vesicle   • extracellular organelle   • extracellular region   • extracellular space   • vesicle   • extracellular membrane-bounded organelle   • centrosome   • microtubule organizing center   • cytoskeleton   • microtubule cytoskeleton   • centriolar satellite   • cytosol   • nucleoplasm   • vacuolar membrane   • lytic vacuole   • vacuole   • lytic vacuole membrane   • bounding membrane of organelle   • lysosomal membrane   • organelle membrane   • lysosome   • Golgi apparatus   • endomembrane system   • cilium   • plasma membrane bounded cell projection   • ciliary basal body   • cell projection   • Golgi apparatus subcompartment   • organelle subcompartment   • trans-Golgi network membrane   • trans-Golgi network   • protein binding   • binding   • enzyme binding   • GTPase binding   • protein-containing complex binding   • pyrophosphatase activity   • GTPase activity   • ribonucleoside triphosphate phosphatase activity   • hydrolase activity, acting on acid anhydrides, in phosphorus-containing anhydrides   • hydrolase activity   • hydrolase activity, acting on acid anhydrides   • catalytic activity   • signaling receptor complex adaptor activity   • protein-macromolecule adaptor activity   • molecular adaptor activity   • signaling adaptor activity   • multicellular organismal process   • system process   • sensory perception of chemical stimulus   • sensory perception   • nervous system process   • sensory perception of taste   • developmental process   • sensory organ development   • eye development   • animal organ development   • retina development in camera-type eye   • visual system development   • multicellular organism development   • camera-type eye development   • anatomical structure development   • sensory system development   • system development   • cell population proliferation   • cellular process   • cellular response to stimulus   • regulation of biological process   • regulation of cellular process   • response to stimulus   • signaling   • biological regulation   • signal transduction   • cell communication   • response to ketone   • response to prostaglandin   • response to lipid   • response to endogenous stimulus   • response to alcohol   • cellular response to prostaglandin stimulus   • response to oxygen-containing compound   • cellular response to oxygen-containing compound   • cellular response to endogenous stimulus   • cellular response to prostaglandin E stimulus   • cellular response to chemical stimulus   • cellular response to alcohol   • response to hormone   • response to chemical   • cellular response to lipid   • response to prostaglandin E   • cellular response to ketone   • cellular response to hormone stimulus   • small GTPase-mediated signal transduction   • Ras protein signal transduction   • intracellular signal transduction   • intracellular signaling cassette   • phospholipase C-activating G protein-coupled receptor signaling pathway   • G protein-coupled receptor signaling pathway   • cellular response to nitrogen compound   • response to dopamine   • cellular response to dopamine   • response to monoamine   • response to catecholamine   • adenylate cyclase-activating dopamine receptor signaling pathway   • cellular response to catecholamine stimulus   • G protein-coupled dopamine receptor signaling pathway   • response to nitrogen compound   • adenylate cyclase-activating G protein-coupled receptor signaling pathway   • cellular response to monoamine stimulus   • adenylate cyclase-modulating G protein-coupled receptor signaling pathway   • synaptic signaling   • cellular response to acetylcholine   • cell-cell signaling   • acetylcholine receptor signaling pathway   • postsynaptic signal transduction   • G protein-coupled acetylcholine receptor signaling pathway   • response to acetylcholine   • non-motile cilium   • 9+0 non-motile cilium   • neuron projection   • photoreceptor disc membrane   • photoreceptor outer segment   • photoreceptor cell cilium   • synapse   • cell junction   • G protein-coupled amine receptor activity   • molecular transducer activity   • trace-amine receptor activity   • G protein-coupled receptor activity   • transmembrane signaling receptor activity   • signaling receptor activity   • adenylate cyclase-inhibiting G protein-coupled receptor signaling pathway   • endoplasmic reticulum subcompartment   • nuclear outer membrane-endoplasmic reticulum membrane network   • endoplasmic reticulum   • endoplasmic reticulum membrane   • G-protein beta-subunit binding   • fibroblast proliferation
SCOP2Domain Identifier• Transducin (heterotrimeric G protein), gamma chain
SCOP2Family Identifier• Transducin (heterotrimeric G protein), gamma chain
Membrane Protein Annotations-• Orientations of Proteins in Membranes database (OPM)   • Protein Data Bank of Transmembrane Proteins (PDBTM)   • MemProtMD


Details about the values in these tables can be found in the corresponding documentation page .
CodeHAI
PDB ResiduesL:L:?1
Environment DetailsOpen EMBL-EBI Page
CodeHAI
NameCyclohexylammonium Ion
SynonymsCyclohexylammonium Ion
Identifier
FormulaC6 H14 N
Molecular Weight100.182
SMILES
PubChem1549093
Formal Charge1
Total Atoms21
Total Chiral Atoms0
Total Bonds21
Total Aromatic Bonds0

PDBsumOpen PDBsum Page
ChainA
ProteinG Protein α Sub unit
UniProtP63092
Sequence
>8WCB_Chain_A
EDKAAVERS KMIEKQLQK DKQVYRRTL RLLLLGADN SGKSTIVKQ 
MRITSGIFE TKFQVDKVN FHMFDVGAQ DERRKWIQC FNDVTAIIF 
VVDSNRLQE ALNDFKSIW NNRWLRTIS VILFLNKQD LLAEKVLAK 
SKIEDYFPE FARYTTDAT PEPGEDPRV TRAKYFIRK EFVDISTAS 
GRHICYPHF TCAVDTENA RRIFNDCKD IILQMNLRE YNLV


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainB
ProteinG Protein β Sub unit
UniProtP62873
Sequence
>8WCB_Chain_B
LRQEAEQLK NQIRDARKA CADAPVGRI QMRTRRTLR GHLAKIYAM 
HWGTDSRLL VSASQDGKL IIWDSYTTN KVHAIPLRS SWVMTCAYA 
PSGNYVACG GLDNICSIY NLKTREGNV RVSRELAGH TGYLSCCRF 
LDDNQIVTS SGDTTCALW DIETGQQTT TFTGHTGDV MSLSLAPDT 
RLFVSGACD ASAKLWDVR EGMCRQTFT GHESDINAI CFFPNGNAF 
ATGSDDATC RLFDLRADQ ELMTYSHDN IICGITSVS FSKSGRLLL 
AGYDDFNCN VWDALKADR AGVLAHDNR VSCLGVTDD GMAVATGSW 
DSFLKIWN


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainG
ProteinG Protein γ Sub unit
UniProtP59768
Sequence
>8WCB_Chain_G
AQARKLVEQ LKMEANIDR IKVSKAAAD MAYCEAHAK EDPLLTPVP 
ASENPFR


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainR
ProteinReceptor
UniProtQ923Y8
Sequence
>8WCB_Chain_R
ASLYSLMSL IILATLVGN LIVIISISH FKQLHTPTN WLLHSMAIV 
DFLLCLIMP CSMVRTERC WYFGEILCK VHTSTDIML SSASIFHLA 
FISIDRYCA VCDPLRYKA KINISTILV MILVSWSLP AVYAFGMIF 
LNLVEELYS QVSDLGCSP FFSKVSGVL AFTSFIPGS VMLFVYYRI 
YFIAKGQAK AAKTLGIMV GVFLVCWCP FFLCTLDPF YVIPPSLND 
ALYGYLNSA LNPMVYAFF YPWFR


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  




This receptor, from the same or other species and bound to the same or other ligands, is also present in the following networks:
Show PDB Class SubFamily Type SubType Species Orthosteric Ligand Other Ligand(s) Protein Partners Resolution Date DOI
9JKQAAmineTrace Amine ReceptorsTA1Homo sapiensMETH-Gs/β1/γ22.662024-10-16doi.org/10.1021/acs.jmedchem.4c01961
9JKQ (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensMETH-2.662024-10-16doi.org/10.1021/acs.jmedchem.4c01961
8ZSVAAmineTrace Amine ReceptorsTA1Mus musculusRO5263397-chim(NtGi1-Gs)/β1/γ22.962024-07-2410.1016/j.celrep.2024.114505
8ZSV (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusRO5263397-2.962024-07-2410.1016/j.celrep.2024.114505
8ZSSAAmineTrace Amine ReceptorsTA1Homo sapiensRO5263397-chim(NtGi1-Gs)/β1/γ23.072024-07-2410.1016/j.celrep.2024.114505
8ZSS (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensRO5263397-3.072024-07-2410.1016/j.celrep.2024.114505
8ZSPAAmineTrace Amine ReceptorsTA1Homo sapiensLSD-chim(NtGi1L-Gs-CtGq)/β1/γ23.142024-07-2410.1016/j.celrep.2024.114505
8ZSP (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensLSD-3.142024-07-2410.1016/j.celrep.2024.114505
8ZSJAAmineTrace Amine ReceptorsTA1Homo sapiens--chim(NtGi1L-Gs-CtGq)/β1/γ22.82024-07-2410.1016/j.celrep.2024.114505
8ZSJ (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiens--2.82024-07-2410.1016/j.celrep.2024.114505
8UHBAAmineTrace Amine ReceptorsTA1Homo sapiensRO5256390-Gs/β1/γ23.352024-01-1010.1038/s41467-023-44601-4
8UHB (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensRO5256390-3.352024-01-1010.1038/s41467-023-44601-4
8WCCAAmineTrace Amine ReceptorsTA1Mus musculusCyclohexylammonium Ion--3.042023-12-2710.1016/j.cell.2023.10.014
8WCBAAmineTrace Amine ReceptorsTA1Mus musculusCyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ23.12023-12-2710.1016/j.cell.2023.10.014
8WCB (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusCyclohexylammonium Ion-3.12023-12-2710.1016/j.cell.2023.10.014
8WC9AAmineTrace Amine ReceptorsTA1Mus musculusZH8651-chim(NtGi1-Gs-CtGq)/β1/γ23.22023-12-2710.1016/j.cell.2023.10.014
8WC9 (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusZH8651-3.22023-12-2710.1016/j.cell.2023.10.014
8WCAAAmineTrace Amine ReceptorsTA1Homo sapiens2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ23.482023-12-2710.1016/j.cell.2023.10.014
8WCA (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiens2-Phenylethylamine-3.482023-12-2710.1016/j.cell.2023.10.014
8WC8AAmineTrace Amine ReceptorsTA1Homo sapiensZH8651-chim(NtGi1-Gs)/β1/γ22.92023-12-2710.1016/j.cell.2023.10.014
8WC8 (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensZH8651-2.92023-12-2710.1016/j.cell.2023.10.014
8WC7AAmineTrace Amine ReceptorsTA1Mus musculusZH8667-chim(NtGi1-Gs)/β1/γ23.12023-12-2710.1016/j.cell.2023.10.014
8WC7 (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusZH8667-3.12023-12-2710.1016/j.cell.2023.10.014
8WC6AAmineTrace Amine ReceptorsTA1Mus musculus2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ23.22023-12-2710.1016/j.cell.2023.10.014
8WC6 (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculus2-Phenylethylamine-3.22023-12-2710.1016/j.cell.2023.10.014
8WC5AAmineTrace Amine ReceptorsTA1Mus musculusTetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ23.32023-12-2710.1016/j.cell.2023.10.014
8WC5 (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusTetramethylammonium Ion-3.32023-12-2710.1016/j.cell.2023.10.014
8WC4AAmineTrace Amine ReceptorsTA1Mus musculusZH8651-chim(NtGi1-Gs)/β1/γ23.12023-12-2710.1016/j.cell.2023.10.014
8WC4 (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusZH8651-3.12023-12-2710.1016/j.cell.2023.10.014
8WC3AAmineTrace Amine ReceptorsTA1Mus musculusSEP-363856-chim(NtGi1-Gs)/β1/γ232023-12-2710.1016/j.cell.2023.10.014
8WC3 (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusSEP-363856-32023-12-2710.1016/j.cell.2023.10.014
8W8AAAmineTrace Amine ReceptorsTA1Homo sapiensRO5256390-chim(NtGi1L-Gs)/β1/γ22.82023-11-2210.1038/s41586-023-06775-1
8W8A (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensRO5256390-2.82023-11-2210.1038/s41586-023-06775-1
8W89AAmineTrace Amine ReceptorsTA1Homo sapiensPEA-chim(NtGi1L-Gs)/β1/γ232023-11-2210.1038/s41586-023-06775-1
8W89 (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensPEA-32023-11-2210.1038/s41586-023-06775-1
8W87AAmineTrace Amine ReceptorsTA1Homo sapiensMETH-chim(NtGi1L-Gs)/β1/γ22.82023-11-2210.1038/s41586-023-06775-1
8W87 (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensMETH-2.82023-11-2210.1038/s41586-023-06775-1
8W88AAmineTrace Amine ReceptorsTA1Homo sapiensSEP-363856-Gs/β1/γ22.62023-11-2210.1038/s41586-023-06775-1
8W88 (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensSEP-363856-2.62023-11-2210.1038/s41586-023-06775-1
8JSOAAmineTrace Amine ReceptorsTA1Homo sapiensAMPH-chim(NtGi1-Gs)/β1/γ23.42023-11-1510.1038/s41586-023-06804-z
8JSO (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensAMPH-3.42023-11-1510.1038/s41586-023-06804-z
8JLRAAmineTrace Amine ReceptorsTA1Homo sapiensA77636-chim(NtGi1-Gs)/β1/γ232023-11-1510.1038/s41586-023-06804-z
8JLR (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensA77636-32023-11-1510.1038/s41586-023-06804-z
8JLKAAmineTrace Amine ReceptorsTA1Mus musculusUlotaront-chim(NtGi1-Gs)/β1/γ23.222023-11-1510.1038/s41586-023-06804-z
8JLK (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusUlotaront-3.222023-11-1510.1038/s41586-023-06804-z
8JLJAAmineTrace Amine ReceptorsTA1Mus musculusT1AM-chim(NtGi1-Gs)/β1/γ23.12023-11-1510.1038/s41586-023-06804-z
8JLJ (No Gprot) AAmineTrace Amine ReceptorsTA1Mus musculusT1AM-3.12023-11-1510.1038/s41586-023-06804-z
8JLQAAmineTrace Amine ReceptorsTA1Homo sapiensFenoldopam-Gs/β1/γ22.842023-11-1510.1038/s41586-023-06804-z
8JLQ (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensFenoldopam-2.842023-11-1510.1038/s41586-023-06804-z
8JLPAAmineTrace Amine ReceptorsTA1Homo sapiensRalmitaront-Gs/β1/γ23.232023-11-1510.1038/s41586-023-06804-z
8JLP (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensRalmitaront-3.232023-11-1510.1038/s41586-023-06804-z
8JLOAAmineTrace Amine ReceptorsTA1Homo sapiensUlotaront-Gs/β1/γ23.522023-11-1510.1038/s41586-023-06804-z
8JLO (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensUlotaront-3.522023-11-1510.1038/s41586-023-06804-z
8JLNAAmineTrace Amine ReceptorsTA1Homo sapiensT1AM-Gs/β1/γ23.242023-11-1510.1038/s41586-023-06804-z
8JLN (No Gprot) AAmineTrace Amine ReceptorsTA1Homo sapiensT1AM-3.242023-11-1510.1038/s41586-023-06804-z




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