Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.29 1.81312402
2G.H1.01 4.9825229
3G.S2.03 7.051884219
4G.S2.06 4.7125409
5G.S2.08 3.645634106
6G.S3.01 3.7154105
7G.S3.03 5.7015508
8G.S3.06 11.67314217
9G.s3h2.03 4.23875409
10G.H2.01 4.0325419
11G.H2.06 5.921519
12G.H2.07 4.47917609
13G.h2s4.01 8.91625409
14G.h2s4.05 3.7975408
15G.S4.03 3.29688467
16G.S4.07 7.27754158
17G.s4h3.03 3.983754158
18G.s4h3.04 7.684374238
19G.H3.01 3.0515159
20G.H3.09 4.0965169
21G.H3.13 7.26256166
22G.H3.17 8.9245515
23G.S5.03 5.1125469
24G.S5.05 4.31458669
25G.hgh4.05 10.7194406
26G.hgh4.11 3.035836245
27G.hgh4.20 3.92812403
28G.H4.03 3.17188404
29G.H4.08 5.185403
30G.H4.10 8.18625407
31G.H4.12 6.446884114
32G.H4.14 4.23875405
33G.H4.15 6.83437408
34G.h4s6.12 4.3125402
35G.S6.02 5.914128
36G.s6h5.01 5.2575469
37G.s6h5.02 2.14313408
38G.s6h5.05 3.629569
39G.H5.08 5.2856108
40G.H5.13 3.861254128
41G.H5.17 6.90155125
42G.H5.19 3.136254178
43b.1x4 1.39188408
44b.lhb1x3 2.7975132
45b.lhb1x6 3.940624133
46b.b1x3 4.085457
47b.b1x6 7.58125409
48b.l1x3 7.99639
49b.l1x6 9.1195519
50b.b2x1 6.857518
51b.b2x3 3.96312436
52b.b2x5 5.12042637
53b.l2x5 9.79062455
54b.b3x1 3.35687455
55b.l3x1 7.60313419
56b.l3x2 5.19655209
57b.b4x2 3.44408
58b.b4x6 10.0521639
59b.b5x3 5.8165539
60b.b5x5 4.71688405
61b.l5x1 4.608754268
62b.l5x5 7.66792609
63b.b6x1 3.9075419
64b.b6x5 2.98187406
65b.l7x5 4.17688406
66b.b8x4 5.6825406
67b.l9x3 8.144519
68b.l9x6 5.4455518
69b.b10x5 3.643509
70b.b11x4 4.619519
71b.l11x2 8.93375419
72b.b12x6 8.1875718
73b.b13x7 6.889577
74b.l13x3 7.32679
75b.l13x6 5.2375519
76b.l13x7 4.2665579
77b.l15x1 4.90625417
78b.l15x2 4.52313409
79b.b16x4 10.4219476
80b.b16x6 7.36036778
81b.b16x7 5.486874279
82b.b17x7 7.8025448
83b.l17x3 9.44549
84b.l17x6 5.70125419
85b.b18x3 4.39312448
86b.l18x1 7.344586186
87b.l18x2 5.136884187
88b.l18x3 8.71813405
89b.b19x2 6.7995546
90b.b19x4 5.26875448
91b.b20x4 9.179548
92b.b20x6 6.223546
93b.b20x7 3.585409
94b.l20x2 5.394509
95b.b21x1 10.0556447
96b.b21x2 3.23125406
97b.b21x7 5.59167605
98b.l21x2 4.77562404
99b.b22x5 5.242926187
100b.l22x5 6.1925139
101b.b23x6 7.037086197
102b.l23x1 5.9925416
103b.b24x6 5.311254198
104b.b24x7 6.778754139
105b.l24x2 3.83055136
106b.l24x3 5.3425405
107b.l25x3 9.045634149
108b.l25x6 9.994518
109b.l26x1 6.84625437
110b.l27x1 10.505619
111b.l27x2 7.753754149
112b.b28x3 3.83125407
113b.b28x4 5.95555146
114b.b28x6 8.1865149
115b.b28x7 5.88937459
116g.l1x4 4.90375408
117g.ctx3 5.58333609
118g.ctx6 3.174176136
119g.ctx14 6.21375459
120g.ctx15 5.42062459
121g.ctx16 4.69938858
1221x35 9.4565526
1231x39 8.7145526
1241x50 6.394509
125I1x50 4.8698
1262x42 4.0735508
1272x46 5.1775489
1282x50 7.391589
1292x57 4.947526
1303x22 5.44875402
1313x26 4.72062426
1323x37 5.8235525
1333x43 5.105489
1343x50 4.27312489
135I2x51 4.413134106
136I2x53 5.8775176
1374x38 3.05312407
1384x56 3.9875424
1394x61 3.5525
140E2.W144 4.36063425
141E2x52 10.635524
1425x39 6.925626
1435x40 4.392524
1445x42 5.1775423
1455x43 4.06375425
1465x44 6.59875626
1475x58 5.72375409
1485x62 2.51125405
1495x69 3.968124254
1506x30 3.0655507
1516x44 6.1475409
1526x48 7.57875627
1536x52 8.85125427
154E3.Q263 1.78812402
1557x30 2.49403
1567x42 5.3075627
1577x49 8.09062489
1587x53 5.0315589
1597x55 3.2395506
1608x50 4.02214798
161Lig 7.820581320
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.l26x5 g.ctx4 97.63443.3525NoNo057
2g.ctx3 g.ctx4 97.68333.6225YesNo097
3g.ctx3 g.ctx5 99.64653.395YesNo099
4b.lhb1x11 g.ctx5 99.6913.1775NoNo049
5b.b25x7 b.lhb1x11 99.82416.005NoNo074
6b.b25x7 b.b28x6 10014.2375NoYes079
7b.b27x3 b.b28x6 49.85938.795NoYes089
8b.b27x3 b.l25x3 49.85446.845NoYes089
9b.l25x3 b.l27x2 99.63997.245YesYes1499
10b.l25x4 b.l27x2 99.91663.66NoYes059
11I1x49 b.l25x4 99.62517.59NoNo065
12I1x49 I1x50 99.56582.58NoYes068
132x40 I1x50 97.38295.15NoYes998
142x37 2x40 98.11058.0425NoNo089
152x37 2x39 97.98662.7475NoNo089
162x39 I2x53 33.2224.06NoYes1796
17G.H5.19 I2x53 35.85993.27YesYes1786
18G.H5.15 G.H5.19 35.61553.645NoYes088
19G.H5.15 G.h2s4.05 30.16173.04NoYes088
20b.b28x4 b.b28x6 50.17577.25YesYes1469
21b.b28x4 b.l25x3 49.95078.8425YesYes1469
22b.b2x3 b.b2x5 87.66493.7825YesYes367
23b.b26x2 b.b2x3 88.71225.67NoYes076
24b.b26x1 b.b26x2 88.65173.01NoNo097
25b.b26x1 b.l27x1 88.59175.8675NoYes099
26b.l3x1 b.l5x5 10.2686.2975YesYes099
27b.b2x1 b.l27x1 79.83156.5125YesYes189
28G.S1.04 G.h2s4.05 21.69452.95NoYes078
29G.S1.04 G.S4.03 21.55682.8525NoYes077
30b.l25x6 b.l27x1 11.440518.24YesYes189
31G.S4.03 G.S5.05 20.82944.08YesYes679
32G.S5.05 G.s6h5.01 19.31646.8125YesYes699
33G.S5.07 G.s6h5.01 18.21023.29NoYes099
34G.S5.07 G.s5hg.01 17.50555.2475NoNo099
35G.S4.07 G.s5hg.01 17.071911.0625YesNo089
36G.S4.07 G.s4h3.03 16.19734.3225YesYes1588
37b.b6x1 b.l9x6 80.26924.4875YesYes198
38b.b2x1 b.b6x1 78.42445.6875YesYes189
39G.H2.06 b.l9x6 78.78875.075YesYes198
40G.H2.06 b.l17x6 39.23156.57YesYes199
41G.s4h3.03 G.s4h3.15 15.61324.04YesNo1589
42G.hgh4.01 G.s4h3.15 15.4914.6525NoNo069
43G.hgh4.01 G.s4h3.04 15.34725.9575NoYes068
44G.HG.15 G.s4h3.04 14.915210.275NoYes078
45G.HG.15 G.hgh4.05 14.77110.0475NoYes076
46b.l23x1 b.l25x6 10.267713.1YesYes168
472x46 3x43 35.46863.805YesYes899
482x46 3x42 70.51875.63YesNo097
492x45 3x42 70.61014.075NoNo097
502x45 4x46 71.06577.3525NoNo097
512x42 4x46 71.15713.4525YesNo087
522x42 3x49 72.47038.06YesNo089
532x39 3x49 64.70248.3125NoNo1799
54b.l17x6 b.l19x1 39.86183.99YesNo099
55b.l17x5 b.l19x1 78.65973.68NoNo069
56b.l17x5 b.l19x2 78.42912.9425NoNo069
57b.b20x2 b.l19x2 77.96765.42NoNo069
58b.b20x2 b.b20x4 77.50575.495NoYes068
59b.b20x4 b.l17x3 21.267117.7725YesYes489
60b.b19x4 b.l17x3 20.04388.5575YesYes489
61b.b18x3 b.b19x4 39.58584.56YesYes488
62b.b14x2 b.b18x3 58.8873.485NoYes078
63b.b10x2 b.b14x2 58.14553.0125NoNo067
64b.b10x2 b.b14x3 44.74164.3625NoNo065
65b.b11x5 b.b14x3 43.99873.7525NoNo065
66b.b11x5 b.l13x7 42.5134.8475NoYes069
67b.l13x3 b.l13x7 23.12375.19YesYes799
68b.b16x4 b.l13x3 10.449218.6675YesYes769
69G.H2.06 b.b18x1 39.11214.1975YesNo199
70b.b18x1 b.l19x1 39.028610.4325NoNo099
71b.b20x4 b.b20x6 55.54864.01YesYes486
72b.b19x4 b.b20x6 20.0534.5375YesYes486
73b.b19x2 b.b20x6 20.52939.11YesYes466
74b.b18x3 b.b19x2 20.043.7675YesYes486
75b.b17x7 b.b20x6 14.79159.3775YesYes486
76b.l21x7 b.l23x1 10.03853.8875NoYes056
77b.b10x2 b.b10x4 12.6775.2225NoNo066
78b.l26x3 b.l26x5 92.83899.355NoNo075
79b.l26x1 b.l26x3 92.68396.8675YesNo377
80b.b2x5 b.l26x1 92.63059.3975YesYes377
81b.b10x4 b.b14x5 11.18753.6425NoNo065
82b.b14x5 b.l10x1 10.44284.8425NoNo053
83b.b13x4 b.b13x5 10.45623.925NoNo044
84b.b17x3 g.h1x10 11.2064.1975NoNo059
856x48 Lig 57.0193.51YesYes270
866x44 6x48 33.540412.025YesYes097
873x43 6x44 33.75363.3525YesYes099
886x48 7x45 32.29859.3225YesNo078
897x45 7x49 32.75211.2375NoYes089
902x46 7x49 32.57856.525YesYes899
913x30 4x61 11.62874.54NoYes265
923x30 4x60 30.89354.7075NoNo264
934x60 5x39 31.637213.5625NoYes246
943x33 5x39 23.15413.5175NoYes236
953x33 E2x52 11.78963.3525NoYes234
96E2x52 Lig 25.616931.85YesYes240
975x39 E2.V177 11.5442.84YesNo063
98E2.V177 E2x52 13.324910.8125NoYes034
993x33 5x40 11.87813.18NoYes234
1005x40 Lig 12.04068.0775YesYes240
1013x26 E2.V176 13.10794.47YesNo061
1023x26 3x30 18.49153.17YesNo266
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
1x351x3916.5552YesYes6622
1x352x645.7252YesNo6421
1x357x386.95252YesNo6521
1x392x577.1752YesYes6622
1x397x4210.77252YesYes6721
2x577x426.962YesYes6721
3x29E2x523.11750NoYes5421
3x33E2x523.35252NoYes3421
3x335x403.182NoYes3421
3x366x483.03252NoYes6711
3x36Lig8.3552NoYes6010
3x373x404.122YesNo5722
3x375x434.292YesYes5521
3x406x4812.33250NoYes7721
E2.V177E2x5210.81250NoYes0421
5x40E2x524.04252YesYes4411
E2x52Lig31.852YesYes4010
E2.E174Lig3.820NoYes0010
5x376x555.60750NoNo3521
5x406x553.5052YesNo4511
5x40Lig8.07752YesYes4010
5x436x523.512YesYes5711
5x445x474.5852YesNo6722
5x446x5217.822YesYes6721
5x476x528.99252NoYes7721
6x446x4812.0250YesYes9721
6x487x415.252YesNo7712
6x487x459.32252YesNo7812
6x48Lig3.512YesYes7010
6x517x413.63750NoNo5712
6x51Lig4.53250NoYes5010
6x52Lig5.08252YesYes7010
6x55Lig7.18252NoYes5010
7x387x424.64252NoYes5711
7x38Lig10.822NoYes5010
7x417x422.7850NoYes7721
7x42Lig4.85752YesYes7010
2x64Lig3.94750NoYes4010
5x405x433.1552YesYes4511
5x43Lig5.32YesYes5010
6x547x343.040NoNo4421
7x34Lig4.33250NoYes4010
6x517x372.5450NoNo5612
2x607x421.82750NoYes6721
E2.E174E2x511.32750NoNo0412

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusa2_onOrthosteric Liganda2b_on
100.00Consensusa2_on_gpOrthosteric Liganda2b_on_gp
100.00Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
100.00Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
100.00Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
78.57Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
73.33Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
71.43Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
70.59Single3NY9ICI118-5513NY9-β2-ICI118-551
70.59Single4UG2CGS216804UG2-A2A-CGS21680
69.23Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
69.23Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
66.67Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
66.67Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
66.67Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
64.29Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
64.29Single5IU7Q274563465IU7-A2A-Q27456346-Na
64.29Single5JTBZM-2413855JTB-A2A-ZM-241385
64.29Single6AQFZM-2413856AQF-A2A-ZM-241385
64.29Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
64.29Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
64.29Consensusa2_offOrthosteric Liganda2a_off
64.29Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
64.29Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
64.29Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
62.50Single2YDVNECA2YDV-A2A-NECA
62.50Single4UHRCGS216804UHR-A2A-CGS21680
62.50Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
62.50Single5G53NECA5G53-A2A-NECA-Gs
62.50Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
62.50Single6J21Aprepitant6J21-NK1-Aprepitant
62.50Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
62.50Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
62.50Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
62.50Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
61.11Single5WF6UK-4320975WF6-A2A-UK-432097
61.11Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
60.00Single3EMLZM-2413853EML-A2A-ZM-241385
60.00Single3NY8ICI118-5513NY8-β2-ICI118-551
60.00Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
60.00Single4GBRS-Carazolol4GBR-β2-S-Carazolol
60.00Single5IU8Q274563475IU8-A2A-Q27456347-Na
60.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
60.00Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
60.00Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
60.00Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
60.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
60.00Single6S0LZM-2413856S0L-A2A-ZM-241385
60.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
60.00Single7PYRPSB-21157PYR-A2A-PSB-2115
60.00Single8CU6LJ-45178CU6-A2A-LJ-4517
60.00Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
60.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
60.00Single9CHXS-Carazolol9CHX-β2-S-Carazolol
60.00Consensusa3_onOrthosteric Liganda3a_on
60.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
60.00Consensusdopamine_offOrthosteric Ligandd2_off d3_off
58.82Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
58.82Single7YITNalfurafine7YIT-κ-Nalfurafine
58.82Single8JWY2-1188JWY-A2A-2-118
58.82Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
58.82Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
58.82Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
57.89Single8WDTphotoNECA8WDT-A2A-photoNECA
57.14Single3PWHZM-2413853PWH-A2A-ZM-241385
57.14Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
57.14Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
57.14Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
57.14Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
56.25Single2RH1S-Carazolol2RH1-β2-S-Carazolol
56.25Single2YCWS-Carazolol2YCW-β1-S-Carazolol
56.25Single5D6LS-Carazolol5D6L-β2-S-Carazolol
56.25Single5IUAQ274563485IUA-A2A-Q27456348-Na
56.25Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
56.25Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
56.25Single6S0QZM-2413856S0Q-A2A-ZM-241385
56.25Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
56.25Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
56.25Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
56.25Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
56.25Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
56.25Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
56.25Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
56.25Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
56.25Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
56.25Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
56.25Single8GNEKW-63568GNE-A2A-KW-6356-Na
56.25Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
56.25Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
56.25Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
56.25Consensusa3_on_gpOrthosteric Liganda3a_on_gp
56.25Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
56.25Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
56.25Consensusadenosine_offOrthosteric Liganda1_off a2_off
56.25Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
56.25Consensusamine_offonOrthosteric Ligandamine_off amine_on
56.25Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
56.25Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
56.25Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
56.25Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
56.25Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
56.25Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
56.25Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
56.25Consensustrace-amine_onOrthosteric Ligandta1_on
55.56Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
55.56Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
55.56Single7EZCUKA7EZC-A2A-UKA
55.56Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
55.56Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
55.00Single3QAKUK-4320973QAK-A2A-UK-432097
53.85Single3UZAGTPL92363UZA-A2A-GTPL9236
53.33Single2YDOAdenosine2YDO-A2A-Adenosine
53.33Single3REYXAC3REY-A2A-XAC
53.33Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
53.33Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
53.33Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
53.33Single5IUBQ274563445IUB-A2A-Q27456344-Na
53.33Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
53.33Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
53.33Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
53.33Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
53.33Single5UVIZM-2413855UVI-A2A-ZM-241385
53.33Single6MH8ZM-2413856MH8-A2A-ZM-241385
53.33Single6PS0S-Carazolol6PS0-β2-S-Carazolol
53.33Single6PS4ICI118-5516PS4-β2-ICI118-551
53.33Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
53.33Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
53.33Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.33Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.33Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
53.33Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
53.33Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
53.33Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
53.33Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
53.33Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.33Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.33Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.33Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
53.33Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
53.33Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
53.33Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
53.33Single9BJKNaloxone9BJK-μ-Naloxone-NAM
53.33Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
53.33Consensusalpha1_onOrthosteric Ligandalpha1a_on
53.33Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
53.33Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
53.33Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
52.94Single5D5AS-Carazolol5D5A-β2-S-Carazolol
52.94Single5D5BS-Carazolol5D5B-β2-S-Carazolol
52.94Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
52.94Single7PX4PSB-21137PX4-A2A-PSB-2113
52.94Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
52.94Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
52.94Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
52.94Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
52.94Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
52.94Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
52.94Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
52.94Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
52.94Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
52.94Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
52.94Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
52.94Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
52.94Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
52.94Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
52.94Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
52.63Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
52.63Single6PT3DPI-2876PT3-δ-DPI-287
50.00Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
50.00Single3D4STimolol3D4S-β2-Timolol
50.00Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
50.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
50.00Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
50.00Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
50.00Single4AMIBucindolol4AMI-β1-Bucindolol
50.00Single4EJ4Naltrindole4EJ4-δ-Naltrindole
50.00Single4RWADIPP-NH24RWA-δ-DIPP-NH2
50.00Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
50.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
50.00Single5UIGCmpd-15UIG-A2A-Cmpd-1
50.00Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
50.00Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
50.00Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
50.00Single6PS1Timolol6PS1-β2-Timolol
50.00Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
50.00Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
50.00Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
50.00Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
50.00Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
50.00Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
50.00Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
50.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
50.00Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
50.00Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
50.00Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
50.00Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
50.00Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
50.00Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
50.00Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
50.00Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
50.00Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
50.00Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
50.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
50.00Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
50.00Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
50.00Single8JJ8Formoterol8JJ8-β2-Formoterol
50.00Single8JJOAlprenolol8JJO-β2-Alprenolol
50.00Single8JWZAB9288JWZ-A2A-AB928-Na
50.00Single8JXRLSD8JXR-D1-LSD
50.00Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
50.00Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
50.00Single8T1WCVN4248T1W-GPR6-CVN424
50.00Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
50.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
50.00Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
50.00Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
50.00Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
50.00Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
50.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
50.00Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
50.00Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
50.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
50.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
50.00Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
50.00Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
50.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
50.00Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
50.00Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
50.00Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
50.00Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
50.00Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
50.00Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
50.00Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
50.00Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
50.00Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
47.83Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
47.62Single6HLOAprepitant6HLO-NK1-Aprepitant
47.37Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
47.37Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
47.37Single7UM4AS26747237UM4-5-HT5A-AS2674723
47.37Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
47.37Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
47.37Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
47.37Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
47.06Single5C1MBU725C1M-μ-BU72
47.06Single5JQHS-Carazolol5JQH-β2-S-Carazolol
47.06Single5N2SPSB365N2S-A1-PSB36
47.06Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
47.06Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
47.06Single6PS6Timolol6PS6-β2-Timolol
47.06Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
47.06Single7C61Ergotamine7C61-5-HT1B-Ergotamine
47.06Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
47.06Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
47.06Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
47.06Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
47.06Single7WC6LSD7WC6-5-HT2A-LSD
47.06Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
47.06Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.06Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.06Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
47.06Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
47.06Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
47.06Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
47.06Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
47.06Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
47.06Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
47.06Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
47.06Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
47.06Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
47.06Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
47.06Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
47.06Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
47.06Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
47.06Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
47.06Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
47.06Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
46.67Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
46.67Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
46.67Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
46.67Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
46.67Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
46.67Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
46.67Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
46.67Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
46.67Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
46.67Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
46.67Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
46.67Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
46.67Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
46.67Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
46.67Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
46.67Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
46.67Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
46.67Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
46.67Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
46.67Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
46.67Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
46.67Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
46.67Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
46.67Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
46.67Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
46.67Consensusalpha2_offOrthosteric Ligandalpha2c_off
46.15Single3RFMCaffeine3RFM-A2A-Caffeine
46.15Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
46.15Single8A2OTheophylline8A2O-A2A-Theophylline-Na
45.45Single5WF5UK-4320975WF5-A2A-UK-432097
45.45Single6PT2KGCHM076PT2-δ-KGCHM07
45.45Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
45.45Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
45.45Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
45.45Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
45.45Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
45.00Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
45.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
45.00Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
44.44Single3P0GBI1671073P0G-β2-BI167107
44.44Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
44.44Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
44.44Single5V54Methiothepin5V54-5-HT1B-Methiothepin
44.44Single6H7JIsoprenaline6H7J-β1-Isoprenaline
44.44Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
44.44Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
44.44Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
44.44Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
44.44Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
44.44Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
44.44Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
44.44Single8E0GBU728E0G-μ-BU72
44.44Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
44.44Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
44.44Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
44.44Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
44.44Consensus5ht1_offOrthosteric Ligand5ht1b_off
44.44Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
44.44Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
44.44Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
44.44Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
44.44Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
44.44Consensustachykinin_offOrthosteric Ligandnk1_off
43.75Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
43.75Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
43.75Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
43.75Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
43.75Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
43.75Single6PS5S-Propranolol6PS5-β2-S-Propranolol
43.75Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
43.75Single6TPGEMPA6TPG-OX2-EMPA
43.75Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
43.75Single7AROLUF58337ARO-A2A-LUF5833-Na
43.75Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
43.75Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
43.75Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
43.75Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
43.75Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
43.75Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
43.75Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
43.75Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
43.75Single7T32ZM-2413857T32-A2A-ZM-241385
43.75Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
43.75Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
43.75Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
43.75Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
43.75Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
43.75Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
43.75Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
43.75Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
43.75Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
43.75Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
43.75Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
43.75Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
43.75Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
43.75Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
43.75Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
43.75Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
43.75Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
43.75Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
43.75Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
43.75Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
43.75Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
43.75Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
43.75Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
43.75Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
43.48Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
43.48Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
42.86Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
42.86Single4IARErgotamine4IAR-5-HT1B-Ergotamine
42.86Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
42.86Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
42.86Single7F8XNN90567F8X-CCKA-NN9056
42.86Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
42.86Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
42.86Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
42.86Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
42.86Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
42.86Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
42.11Single4LDEBI1671074LDE-β2-BI167107
42.11Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
42.11Single6MXTSalmeterol6MXT-β2-Salmeterol
42.11Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
42.11Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
42.11Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
42.11Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
42.11Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
42.11Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
42.11Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
42.11Single8JJLOlodaterol8JJL-β2-Olodaterol
42.11Single8XYIVUF106618XYI-CXCR3-VUF10661
42.11Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
42.11Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
42.11Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
42.11Consensusalpha1_offOrthosteric Ligandalpha1a_off
42.11Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
42.11Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
42.11Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
42.11Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
42.11Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
42.11Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
42.11Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
42.11Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
41.67Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
41.67Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
41.67Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
41.18Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
41.18Single2Y04Salbutamol2Y04-β1-Salbutamol
41.18Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
41.18Single5UENDU1725UEN-A1-DU172
41.18Single6H7MSalbutamol6H7M-β1-Salbutamol
41.18Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
41.18Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
41.18Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
41.18Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
41.18Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
41.18Single7UL4Alvimopan7UL4-μ-Alvimopan
41.18Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
41.18Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
41.18Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
41.18Single7WC7Lisuride7WC7-5-HT2A-Lisuride
41.18Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
41.18Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
41.18Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
41.18Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
41.18Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
41.18Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
41.18Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
41.18Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
41.18Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
41.18Single8RLNLUF58348RLN-A2A-LUF5834
41.18Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
41.18Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
41.18Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
41.18Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
41.18Single8X64Desloratadine8X64-H1-Desloratadine
41.18Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
41.18Consensus5ht5_onOrthosteric Ligand5ht5a_on
41.18Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
41.18Consensusalpha2_onOrthosteric Ligandalpha2b_on
41.18Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
41.18Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
41.18Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
40.91Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
40.91Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
40.91Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
40.91Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
40.91Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
40.91Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
40.91Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
40.91Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
40.00Single3PBLEticlopride3PBL-D3-Eticlopride
40.00Single5X93K-87945X93-ETB-K-8794
40.00Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
40.00Single6H7LDobutamine6H7L-β1-Dobutamine
40.00Single6IBLArformoterol6IBL-β1-Arformoterol
40.00Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
40.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
40.00Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
40.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
40.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
40.00Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
40.00Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
40.00Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
40.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
40.00Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
40.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
40.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
40.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
40.00Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
40.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
40.00Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
40.00Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
40.00Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
40.00Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
40.00Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
40.00Single8K5BNiacin8K5B-HCA2-Niacin
40.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
40.00Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
40.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
40.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
40.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
40.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
40.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
40.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
40.00Consensuscck_onOrthosteric Ligandccka_on cckb_on
40.00Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
40.00Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
40.00Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
40.00Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
40.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
40.00Consensusendothelin_offOrthosteric Ligandetb_off
40.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
40.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
40.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
40.00Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
39.13Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
39.13Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
38.89Single2Y03Isoprenaline2Y03-β1-Isoprenaline
38.89Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
38.89Single5N2RPSB-365N2R-A2A-PSB-36-Na
38.89Single5TVNLSD5TVN-5-HT2B-LSD
38.89Single5WQCEMPA5WQC-OX2-EMPA
38.89Single6E67BI1671076E67-β2-BI167107-Gs (fused)
38.89Single6HLPNetupitant6HLP-NK1-Netupitant
38.89Single6LUQHaloperidol6LUQ-D2-Haloperidol
38.89Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
38.89Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
38.89Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
38.89Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
38.89Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
38.89Single7SINNPS-21437SIN-CaS-NPS-2143
38.89Single7SINNPS-21437SIN-CaS-NPS-2143
38.89Single7W41PD1762527W41-BB2-PD176252
38.89Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.89Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.89Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
38.89Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
38.89Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
38.89Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
38.89Single8QOTNanobody-E8QOT-μ-Nanobody-E
38.89Single8TF5Oleic acid8TF5-GPR6-Oleic acid
38.89Single8ZMFA1L108ZMF-5-HT2C-A1L10
38.89Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
38.89Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
38.89Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
38.89Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
38.89Consensusbombesin_offOrthosteric Ligandbb2_off
38.89Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
38.89Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
38.89Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
38.89Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
38.46Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
38.46Single8PWNTheophylline8PWN-A2A-Theophylline
38.46Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
38.10Single5ZTYAM102575ZTY-CB2-AM10257
38.10Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
38.10Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
38.10Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
38.10Single7SK9CCX6627SK9-ACKR3-CCX662
38.10Single7XN9L-054,5227XN9-SST2-L-054,522
38.10Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
38.10Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
38.10Single8X5YAstemizole8X5Y-H1-Astemizole
38.10Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
38.10Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
38.10Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
38.10Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
37.50Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
37.50Single6JODAngiotensin II6JOD-AT2-Angiotensin II
37.50Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
37.50Single6ME2Ramelteon6ME2-MT1-Ramelteon
37.50Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
37.50Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
37.50Single6TODEMPA6TOD-OX1-EMPA-Na
37.50Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
37.50Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
37.50Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
37.50Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
37.50Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
37.50Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
37.50Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
37.50Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
37.50Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
37.50Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
37.50Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
37.50Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
37.50Single8GNGIstradefylline8GNG-A2A-Istradefylline
37.50Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
37.50Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
37.50Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
37.50Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
37.50Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.50Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
37.50Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
37.50Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
37.50Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
37.04Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
37.04Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
37.04Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
37.04Consensusbradykinin_onOrthosteric Ligandbk2_on
37.04Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
37.04Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
36.84Single4U15Tiotropium4U15-M3-Tiotropium
36.84Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
36.84Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
36.84Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
36.84Single6J20Aprepitant6J20-NK1-Aprepitant
36.84Single6OL9Tiotropium6OL9-M5-Tiotropium
36.84Single6TQ7SB-3348676TQ7-OX1-SB-334867
36.84Single6WGTLSD6WGT-5-HT2A-LSD
36.84Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
36.84Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
36.84Single7FEECP559407FEE-CB1-CP55940-ZCZ011
36.84Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
36.84Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
36.84Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
36.84Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
36.84Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
36.84Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.84Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
36.84Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
36.84Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
36.84Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
36.84Single8XVLZibotentan8XVL-ETA-Zibotentan
36.84Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
36.84Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
36.84Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.84Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
36.84Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
36.84Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
36.36Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
36.36Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
36.36Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
36.36Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
36.36Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
36.36Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
36.36Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
36.36Consensuslpl_onOrthosteric Ligands1p_on lpa_on
36.36Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
36.36Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.00Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
36.00Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
36.00Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
35.71Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
35.71Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
35.71Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
35.71Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
35.71Consensusbombesin_onOrthosteric Ligandbb2_on
35.71Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
35.71Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
35.71Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
35.71Consensussensory_onOrthosteric Ligandopsins_on
35.29Single4ZJCSB-6740424ZJC-OX1-SB-674042
35.29Single6A94Zotepine6A94-5-HT2A-Zotepine
35.29Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
35.29Single6KUXRS-799486KUX-α2a-RS-79948
35.29Single6TPNHTL66416TPN-OX2-HTL6641
35.29Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
35.29Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
35.29Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
35.29Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
35.29Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
35.29Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
35.29Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
35.29Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
35.29Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
35.29Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
35.29Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
35.29Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
35.29Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
35.29Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
35.29Single8K5CAcipimox8K5C-HCA2-Acipimox
35.29Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
35.29Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
35.29Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
35.29Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
35.29Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
35.29Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
35.29Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
35.29Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
35.29Consensushca_onOrthosteric Ligandhca2_on
35.29Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
35.00Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
35.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
35.00Single5CXVTiotropium5CXV-M1-Tiotropium
35.00Single6A93Risperidone6A93-5-HT2A-Risperidone
35.00Single6CM4Risperidone6CM4-D2-Risperidone
35.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
35.00Single6KQICP559406KQI-CB1-CP55940-Org27569
35.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
35.00Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
35.00Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.00Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
35.00Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
35.00Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
35.00Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
35.00Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.00Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
35.00Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
35.00Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
35.00Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
35.00Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
35.00Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
35.00Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
35.00Consensuslpa_offOrthosteric Ligandlpa1_off
35.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
35.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
35.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
34.78Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
34.78Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
34.78Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
34.78Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
34.62Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
34.62Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
34.62Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
33.33Single2Y01Dobutamine2Y01-β1-Dobutamine
33.33Single2Y02Carmoterol2Y02-β1-Carmoterol
33.33Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
33.33Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
33.33Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
33.33Single4QKX35V4QKX-β2-35V
33.33Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
33.33Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
33.33Single5DSGTiotropium5DSG-M4-Tiotropium
33.33Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
33.33Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
33.33Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
33.33Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
33.33Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
33.33Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
33.33Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
33.33Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
33.33Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
33.33Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
33.33Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
33.33Single6TOTLemborexant6TOT-OX1-Lemborexant
33.33Single7BU7BI1671077BU7-β1-BI167107
33.33Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
33.33Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
33.33Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
33.33Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
33.33Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
33.33Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
33.33Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
33.33Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
33.33Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
33.33Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
33.33Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
33.33Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
33.33Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
33.33Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
33.33Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
33.33Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
33.33Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
33.33Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
33.33Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
33.33Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
33.33Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
33.33Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
33.33Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
33.33Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
33.33Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
33.33Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
33.33Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
33.33Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
33.33Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
33.33Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
33.33Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
33.33Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
33.33Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
33.33Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
33.33Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
33.33Single8X63Mepyramine8X63-H1-Mepyramine
33.33Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
33.33Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
33.33Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
33.33Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
33.33Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
33.33Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
33.33Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
33.33Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
33.33Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
33.33Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
33.33Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusblt_onOrthosteric Ligandblt1_on
33.33Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
33.33Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
33.33Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
33.33Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
33.33Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
33.33Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
33.33Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
33.33Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
33.33Consensusgi_sensoryOrthosteric Ligandgi_opsins
33.33Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
33.33Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
33.33Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
33.33Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
33.33Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
33.33Consensushca_on_gpOrthosteric Ligandhca2_on_gp
33.33Consensushistamine_offOrthosteric Ligandh1_off
33.33Consensusleukotriene_onOrthosteric Ligandblt_on
33.33Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
33.33Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
33.33Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
33.33Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
33.33Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
33.33Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
33.33Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
33.33Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
33.33Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
33.33Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
33.33Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
33.33Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
33.33Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
32.14Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
32.00Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
32.00Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
32.00Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
32.00Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
31.82Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
31.82Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
31.82Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
31.82Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
31.82Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
31.82Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
31.82Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
31.82Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
31.82Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
31.82Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
31.82Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
31.58Single2Y00Dobutamine2Y00-β1-Dobutamine
31.58Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
31.58Single5WIUNemonapride5WIU-D4-Nemonapride
31.58Single5WIVNemonapride5WIV-D4-Nemonapride-Na
31.58Single5XPRBosentan5XPR-ETB-Bosentan
31.58Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
31.58Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
31.58Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
31.58Single6TP6Filorexant6TP6-OX1-Filorexant
31.58Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
31.58Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
31.58Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
31.58Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
31.58Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
31.58Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
31.58Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.58Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
31.58Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
31.58Single8JXSPF-61428JXS-D1-PF-6142
31.58Single8S4DCMF-0198S4D-Apelin-CMF-019
31.58Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
31.58Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
31.58Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
31.58Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
31.58Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
31.58Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
31.58Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
31.58Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
31.58Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
31.58Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
31.58Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.58Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.58Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
31.58Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
31.25Single6HLLCP999946HLL-NK1-CP99994
31.25Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
31.25Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
31.25Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
31.25Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
31.25Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
31.25Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
31.25Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
31.25Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
31.25Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
31.03Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
31.03Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
31.03Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
30.77Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
30.77Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
30.77Single5MZPCaffeine5MZP-A2A-Caffeine-Na
30.77Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
30.77Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.77Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
30.77Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
30.77Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
30.77Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.77Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
30.77Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
30.43Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
30.43Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
30.43Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
30.43Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
30.43Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
30.43Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.43Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.43Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
30.00Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
30.00Single4DJHJDTic4DJH-κ-JDTic
30.00Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
30.00Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
30.00Single5XR8AM8415XR8-CB1-AM841
30.00Single5XRAAM115425XRA-CB1-AM11542
30.00Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
30.00Single6E59L-7607356E59-NK1-L-760735
30.00Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
30.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
30.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
30.00Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
30.00Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
30.00Single7TUYGSK682753A7TUY-GPR183-GSK682753A
30.00Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
30.00Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
30.00Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
30.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
30.00Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
30.00Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
30.00Single8EA0Iperoxo8EA0-M3-Iperoxo
30.00Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
30.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
30.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
30.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
30.00Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
30.00Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
30.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
30.00Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
30.00Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
30.00Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
30.00Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
30.00Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
30.00Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
30.00Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
30.00Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
30.00Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
30.00Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
30.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
30.00Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
30.00Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
30.00Consensuslpa_onOrthosteric Ligandlpa1_on
30.00Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
30.00Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
30.00Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
30.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
30.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
30.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
29.63Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
29.63Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.63Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
29.41Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
29.41Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
29.41Single5WS3EMPA5WS3-OX2-EMPA
29.41Single6AKXA4R6AKX-CCR5-A4R
29.41Single6B73MP11046B73-κ-MP1104
29.41Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
29.41Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
29.41Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
29.41Single7F8ULintitript7F8U-CCKA-Lintitript
29.41Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
29.41Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
29.41Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
29.41Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
29.41Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
29.41Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
29.41Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
29.41Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
29.41Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
29.41Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
29.41Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
29.41Single8IWESpermidine8IWE-TA9-Spermidine
29.41Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
29.41Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
29.41Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
29.41Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.41Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
29.41Single8Y0HVUF114188Y0H-CXCR3-VUF11418
29.41Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
29.41Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
29.41Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
29.41Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
29.41Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
29.41Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
29.41Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
29.41Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
29.41Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
29.41Consensusorexin_offOrthosteric Ligandox2_off ox1_off
29.41Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
29.41Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
29.41Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
29.41Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
29.17Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
29.17Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
29.17Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
29.17Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
29.17Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
29.17Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
29.17Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
29.17Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
29.17Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
29.17Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
29.17Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
29.17Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
28.57Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
28.57Single4N4WSANT-14N4W-SMO-SANT-1
28.57Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
28.57Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
28.57Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
28.57Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
28.57Single7DFPSpiperone7DFP-D2-Spiperone
28.57Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
28.57Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
28.57Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
28.57Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
28.57Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
28.57Single7K15MKD0467K15-BLT1-MKD046-Na
28.57Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
28.57Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
28.57Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
28.57Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
28.57Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
28.57Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
28.57Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
28.57Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
28.57Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
28.57Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
28.57Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
28.57Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
28.57Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
28.57Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
28.57Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
28.57Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
28.57Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
28.57Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
28.57Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
28.57Consensuslpl_offOrthosteric Ligands1p_off lpa_off
28.57Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
28.57Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
28.57Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.00Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
28.00Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
28.00Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
28.00Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
28.00Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
28.00Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
28.00Consensusangiotensin_onOrthosteric Ligandat1_on
28.00Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
28.00Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
28.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
27.78Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
27.78Single3RZECidoxepin3RZE-H1-Cidoxepin
27.78Single4MBSMaraviroc4MBS-CCR5-Maraviroc
27.78Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
27.78Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
27.78Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
27.78Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
27.78Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
27.78Single6TPKRetosiban6TPK-OT-Retosiban
27.78Single6V9SGTPL114036V9S-OX1-GTPL11403
27.78Single6VI4JDTic6VI4-κ-JDTic
27.78Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
27.78Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.78Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
27.78Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
27.78Single7UL3Famotidine7UL3-H2-Famotidine
27.78Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
27.78Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
27.78Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
27.78Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
27.78Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
27.78Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
27.78Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
27.78Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.78Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
27.78Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
27.78Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
27.78Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
27.78Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
27.78Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
27.78Consensusopsins_offOrthosteric Ligandrhodopsin_off
27.78Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
27.78Consensussensory_offOrthosteric Ligandopsins_off
27.78Consensusvasop-oxy_offOrthosteric Ligandot_off
27.59Single6IGLIRL16206IGL-ETB-IRL1620
27.59Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
27.27Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
27.27Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
27.27Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
27.27Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
27.27Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
27.27Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
27.27Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single8XVJMacitentan8XVJ-ETA-Macitentan
27.27Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
27.27Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
27.27Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Consensusprostanoid_offOrthosteric Ligandep_off dp_off
26.92Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
26.92Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.92Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
26.92Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
26.92Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
26.92Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
26.92Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
26.92Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
26.92Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
26.92Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
26.92Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
26.92Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
26.92Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
26.92Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.92Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
26.92Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.92Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.92Consensusvasop-oxy_onOrthosteric Ligandv2_on
26.92Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
26.67Single5GLHEndothelin-15GLH-ETB-Endothelin-1
26.67Single6IGKEndothelin-36IGK-ETB-Endothelin-3
26.67Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
26.67Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
26.67Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.67Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
26.67Single9CHUNoradrenaline9CHU-β2-Noradrenaline
26.67Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
26.67Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
26.67Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
26.32Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
26.32Single4DAJTiotropium4DAJ-M3-Tiotropium
26.32Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
26.32Single4MQSIperoxo4MQS-M2-Iperoxo
26.32Single4U14Tiotropium4U14-M3-Tiotropium
26.32Single5DHHSB-6121115DHH-NOP-SB-612111
26.32Single5TGZAM65385TGZ-CB1-AM6538
26.32Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
26.32Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
26.32Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
26.32Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
26.32Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
26.32Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
26.32Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
26.32Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
26.32Single7V3ZCP559407V3Z-CB1-CP55940
26.32Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
26.32Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
26.32Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
26.32Single8K5DGSK2560738K5D-HCA2-GSK256073
26.32Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
26.32Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
26.32Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
26.32Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
26.32Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
26.32Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
26.32Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
26.32Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
26.09Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
26.09Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
26.09Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
26.09Single8QJ2pN1628QJ2-MC4-pN162-Gs
26.09Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
26.09Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
26.09Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
26.09Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
25.93Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
25.93Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.93Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
25.93Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
25.93Single8ZRTET-18ZRT-ETB-ET-1
25.81Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
25.81Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
25.81Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
25.00Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
25.00Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
25.00Single4NTJAZD12834NTJ-P2Y12-AZD1283
25.00Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
25.00Single5CGCHTL142425CGC-mGlu5-HTL14242
25.00Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
25.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
25.00Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
25.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
25.00Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
25.00Single6ME5Agomelatine6ME5-MT1-Agomelatine
25.00Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
25.00Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
25.00Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
25.00Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
25.00Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
25.00Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
25.00Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
25.00Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
25.00Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
25.00Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
25.00Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
25.00Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
25.00Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
25.00Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
25.00Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
25.00Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
25.00Single8WKYPG-9348WKY-MC4-PG-934
25.00Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
25.00Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
25.00Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
25.00Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
25.00Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
25.00Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
25.00Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
25.00Consensus5ht2_onOrthosteric Ligand5ht2b_on
25.00Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
25.00Consensusblt_offOrthosteric Ligandblt1_off
25.00Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
25.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
25.00Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
25.00Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
25.00Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
25.00Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
25.00Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
25.00Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
25.00Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
25.00Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
25.00Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
24.24Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
24.14Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
24.14Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
24.14Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
24.14Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
24.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
24.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
24.00Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
24.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
24.00Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
24.00Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
24.00Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
24.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
24.00Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
24.00Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
23.81Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
23.81Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
23.81Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
23.81Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
23.81Single7B6WCyclazosin7B6W-α1b-Cyclazosin
23.81Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
23.81Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
23.81Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
23.81Single7P2L4YI7P2L-mGlu5-4YI
23.81Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
23.81Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
23.81Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
23.81Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
23.81Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
23.81Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
23.81Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
23.81Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
23.81Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
23.81Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
23.81Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
23.81Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
23.81Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
23.81Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
23.81Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
23.81Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
23.81Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
23.81Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
23.81Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
23.53Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
23.53Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
23.53Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
23.53Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
23.53Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
23.53Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
23.53Single6TP4ACT-4622066TP4-OX1-ACT-462206
23.53Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
23.53Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
23.53Single7SRQLSD7SRQ-5-HT2B-LSD
23.53Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
23.53Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.53Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
23.53Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
23.53Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
23.53Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
23.53Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
23.53Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
23.53Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
23.53Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
23.53Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
23.53Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
23.33Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
23.33Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
23.33Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
23.33Consensusendothelin_onOrthosteric Ligandetb_on eta_on
23.33Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
23.08Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
23.08Single6W25SHU91196W25-MC4-SHU9119-Ca
23.08Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
23.08Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
23.08Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
23.08Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
23.08Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
22.73Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
22.73Single4XEENeurotensin4XEE-NTS1-Neurotensin
22.73Single4XESNeurotensin4XES-NTS1-Neurotensin
22.73Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
22.73Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
22.73Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
22.73Single6ZG4HTL00099366ZG4-M1-HTL0009936
22.73Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
22.73Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
22.73Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
22.73Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
22.73Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
22.73Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
22.73Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
22.73Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
22.73Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
22.73Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
22.73Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
22.73Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
22.73Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Consensusorexin_onOrthosteric Ligandox2_on
22.73Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
22.58Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
22.58Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
22.58Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
22.22Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
22.22Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
22.22Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
22.22Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
22.22Single4S0VSuvorexant4S0V-OX2-Suvorexant
22.22Single5ZKQABT-4915ZKQ-PAF-ABT-491
22.22Single6AKYMaraviroc6AKY-CCR5-Maraviroc
22.22Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
22.22Single6ME9Ramelteon6ME9-MT2-Ramelteon
22.22Single6TPJSuvorexant6TPJ-OX2-Suvorexant
22.22Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
22.22Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
22.22Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
22.22Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
22.22Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
22.22Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
22.22Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
22.22Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
22.22Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single7XRRLemborexant7XRR-OX2-Lemborexant
22.22Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
22.22Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
22.22Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
22.22Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
22.22Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
22.22Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.22Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
22.22Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
22.22Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.22Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.22Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
22.22Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.22Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
22.22Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
22.22Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
22.22Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
22.22Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
22.22Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
22.22Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.22Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
21.88Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
21.88Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
21.74Single4BUONeurotensin4BUO-NTS1-Neurotensin
21.74Single5CGDHTL142425CGD-mGlu5-HTL14242
21.74Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
21.74Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
21.74Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
21.74Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
21.74Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
21.74Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
21.74Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
21.74Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
21.74Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
21.74Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
21.74Consensuschemerin_onOrthosteric Ligandcml1_on
21.74Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
21.74Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
21.74Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
21.74Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
21.43Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
21.43Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
21.43Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
21.43Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
21.43Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
21.43Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
21.43Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
21.43Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
21.43Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
21.43Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
21.43Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
21.05Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
21.05Single6FFIMMPEP6FFI-mGlu5-MMPEP
21.05Single6IQLL7458706IQL-D4-L745870
21.05Single6TP3Nemorexant6TP3-OX1-Nemorexant
21.05Single6ZG9GSK10347026ZG9-M1-GSK1034702
21.05Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
21.05Single7VODCariprazine7VOD-5-HT2A-Cariprazine
21.05Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
21.05Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
21.05Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.05Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
21.05Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
21.05Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.05Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
21.05Single8IHKAcifran8IHK-HCA3-Acifran
21.05Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
21.05Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
21.05Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
21.05Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
21.05Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
21.05Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
21.05Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
20.83Single5EE7MK08935EE7-Glucagon-MK0893
20.83Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
20.83Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
20.83Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
20.83Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
20.83Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
20.83Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
20.83Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
20.83Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
20.83Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
20.83Single8IEIA1LYA8IEI-GPR156-A1LYA
20.83Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
20.83Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
20.83Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
20.83Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
20.83Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.83Consensuskisspeptin_onOrthosteric Ligandkiss1_on
20.69Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
20.69Single6FJ3PTH6FJ3-PTH1-PTH
20.69Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
20.69Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
20.69Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
20.69Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
20.69Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
20.69Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
20.69Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
20.69Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
20.00Single4QIMANTA XV4QIM-SMO-ANTA XV
20.00Single4XT1Fractalkine4XT1-US28-Fractalkine
20.00Single4YAYZD-71554YAY-AT1-ZD-7155
20.00Single5DHGC-355DHG-NOP-C-35
20.00Single6D27CAY104716D27-DP2-CAY10471
20.00Single6DRXLisuride6DRX-5-HT2B-Lisuride
20.00Single6FFHFenobam6FFH-mGlu5-Fenobam
20.00Single6IIVDaltroban6IIV-TP-Daltroban
20.00Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
20.00Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
20.00Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
20.00Single7QA8Peptide7QA8-STE2-Peptide
20.00Single7QA8Peptide7QA8-STE2-Peptide
20.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
20.00Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
20.00Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
20.00Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
20.00Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
20.00Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
20.00Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
20.00Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
20.00Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
20.00Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
20.00Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
20.00Single8IEBA1LYA8IEB-GPR156-A1LYA
20.00Single8IEPA1LYA8IEP-GPR156-A1LYA
20.00Single8IEPA1LYA8IEP-GPR156-A1LYA
20.00Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
20.00Single8KIGSHU91198KIG-MC3-SHU9119-Ca
20.00Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
20.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
20.00Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
20.00Single8XWNCXCL88XWN-CXCR2-CXCL8
20.00Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.00Single9IYAONO-97105319IYA-GPR55-ONO-9710531
20.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
20.00Consensuscck_offOrthosteric Ligandccka_off
20.00Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
20.00Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
20.00Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.00Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.00Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
20.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
19.44Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
19.44Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
19.35Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
19.35Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
19.35Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
19.35Single8IY6Endothelin-18IY6-ETB-Endothelin-1
19.23Single7XNACYN1548067XNA-SST2-CYN154806
19.23Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8IEBA1LYA8IEB-GPR156-A1LYA
19.23Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
19.23Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
19.23Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
19.23Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
19.23Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
19.23Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
19.23Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
19.23Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
19.05Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
19.05Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
19.05Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
19.05Single6D26Fevipiprant6D26-DP2-Fevipiprant
19.05Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
19.05Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
19.05Single7C4SS1P7C4S-S1P3-S1P
19.05Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
19.05Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
19.05Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
19.05Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
19.05Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
19.05Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
19.05Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
19.05Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
19.05Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
19.05Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
19.05Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
19.05Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
19.05Consensusdp_offOrthosteric Liganddp2_off
19.05Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
19.05Consensusep_offOrthosteric Ligandep4_off
19.05Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
18.92Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
18.75Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
18.52Single3OE0CVX153OE0-CXCR4-CVX15
18.52Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
18.52Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
18.52Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.52Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
18.52Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
18.52Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
18.18Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
18.18Single4BV0Neurotensin4BV0-NTS1-Neurotensin
18.18Single5TZRMK86665TZR-FFA1-MK8666
18.18Single5V56TC1145V56-SMO-TC114
18.18Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
18.18Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
18.18Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
18.18Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
18.18Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
18.18Single7R0CAVP7R0C-V2-AVP-Arrestin2
18.18Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
18.18Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
18.18Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
18.18Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
18.18Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
18.18Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
18.18Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
18.18Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
18.18Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
18.18Consensusneurotensin_onOrthosteric Ligandnts1_on
18.18Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.86Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
17.86Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
17.86Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
17.86Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
17.86Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
17.86Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
17.86Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
17.86Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
17.86Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
17.65Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
17.65Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
17.65Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
17.65Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
17.65Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
17.65Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
17.65Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
17.65Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.65Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
17.65Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
17.65Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
17.65Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
17.65Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
17.65Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
17.65Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
17.39Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
17.39Single4PY02MeSATP4PY0-P2Y12-2MeSATP
17.39Single5X33BIIL2605X33-BLT1-BIIL260
17.39Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
17.39Single6IIURamatroban6IIU-TP-Ramatroban
17.39Single6OS2TRV0266OS2-AT1-TRV026
17.39Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
17.39Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
17.39Single6YVRNTS8-136YVR-NTS1-NTS8-13
17.39Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
17.39Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
17.39Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
17.39Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
17.39Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
17.39Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
17.39Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
17.39Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
17.39Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
17.39Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.39Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
17.39Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.24Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
17.24Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
17.24Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
17.24Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
17.24Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
17.24Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
17.24Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
16.67Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
16.67Single3OE9IT1t3OE9-CXCR4-IT1t
16.67Single4XT3Fractalkine4XT3-US28-Fractalkine
16.67Single5L7IVismodegib5L7I-SMO-Vismodegib
16.67Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
16.67Single6K1QIRL25006K1Q-ETB-IRL2500
16.67Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
16.67Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
16.67Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
16.67Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
16.67Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
16.67Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
16.67Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
16.67Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
16.67Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
16.67Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
16.67Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
16.67Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
16.67Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
16.67Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
16.67Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
16.67Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
16.67Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
16.67Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
16.67Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
16.67Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
16.67Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
16.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8XVUCXCL28XVU-CXCR2-CXCL2
16.67Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
16.67Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
16.67Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single9B9Y7DY9B9Y-CB1-7DY
16.67Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
16.67Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
16.67Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
16.67Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
16.67Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Consensusgq_nucleotideOrthosteric Ligandgq_p2y
16.67Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
16.13Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
16.13Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
16.13Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
16.13Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
16.13Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
16.13Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
16.13Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
16.13Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
16.00Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
16.00Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
16.00Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single8XQJJN2418XQJ-Apelin-JN241
16.00Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
15.79Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
15.79Single4BWBNeurotensin4BWB-NTS1-Neurotensin
15.79Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
15.79Single6DS0Ly2660976DS0-5-HT2B-Ly266097
15.79Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
15.79Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
15.79Single7BR3Elagolix7BR3-GnRH1-Elagolix
15.79Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
15.79Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
15.79Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
15.79Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
15.79Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
15.79Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
15.79Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
15.79Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
15.79Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
15.79Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
15.79Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
15.79Consensusangiotensin_offOrthosteric Ligandat1_off
15.79Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
15.79Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
15.79Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.79Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
15.62Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
15.62Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
15.62Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
15.62Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
15.62Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
15.62Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
15.62Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
15.62Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
15.62Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
15.62Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
15.62Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
15.62Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
15.38Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
15.38Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
15.38Single8IEIA1LYA8IEI-GPR156-A1LYA
15.38Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.38Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
15.38Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
15.38Consensussomatostatin_offOrthosteric Ligandsst2_off
15.15Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
15.15Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
15.15Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
15.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
15.00Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
15.00Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
15.00Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
15.00Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
15.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
15.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
15.00Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
15.00Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
15.00Single7VV6C48/807VV6-MRGPRX2-C48/80
15.00Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
15.00Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
15.00Single8K2WAMG4878K2W-CXCR3-AMG487
15.00Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.00Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
15.00Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
15.00Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
15.00Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
15.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
15.00Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
15.00Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
15.00Consensusgrh_offOrthosteric Ligandgnrh1_off
14.81Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
14.81Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
14.81Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
14.81Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
14.81Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.71Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
14.71Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
14.71Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
14.71Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
14.29Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
14.29Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
14.29Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
14.29Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
14.29Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
14.29Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
14.29Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
14.29Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.29Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
14.29Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
14.29Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
14.29Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
14.29Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
14.29Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
14.29Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
14.29Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
14.29Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
14.29Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
14.29Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.29Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.29Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.29Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.29Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.29Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
13.89Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
13.89Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.89Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
13.89Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
13.89Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
13.89Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
13.89Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.79Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
13.79Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
13.79Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
13.64Single4JKVTaladegib4JKV-SMO-Taladegib
13.64Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
13.64Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
13.64Single6Z4SSR486926Z4S-NTS1-SR48692
13.64Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
13.64Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
13.64Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
13.64Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.64Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
13.64Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
13.64Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
13.51Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
13.33Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.33Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
13.33Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
13.33Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
13.33Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
13.33Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
13.04Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
13.04Single5V57TC1145V57-SMO-TC114
13.04Single7F1TMIP-1a7F1T-CCR5-MIP-1a
13.04Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
13.04Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.90Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
12.90Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
12.90Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
12.50Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
12.50Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
12.50Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
12.50Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
12.50Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
12.50Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.50Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.50Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
12.50Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
12.50Single8XQJJN2418XQJ-Apelin-JN241
12.50Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
12.50Single8XWACXCL18XWA-CXCR2-CXCL1
12.50Single8XWMCXCL68XWM-CXCR2-CXCL6
12.50Single8XWSCXCL58XWS-CXCR2-CXCL5
12.50Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
12.50Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.50Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.50Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
12.50Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.12Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
12.00Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
12.00Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
12.00Single8XWFCXCL38XWF-CXCR2-CXCL3
12.00Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
11.76Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
11.76Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
11.76Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
11.76Consensusp2y_offOrthosteric Ligandp2y1_off
11.54Single6KNMJN241-96KNM-Apelin-JN241-9
11.54Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single3OE6IT1t3OE6-CXCR4-IT1t
11.11Single4XNWMRS25004XNW-P2Y1-MRS2500
11.11Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
11.11Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
11.11Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Single7WC5Psilocin7WC5-5-HT2A-Psilocin
11.11Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
11.11Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
11.11Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
11.11Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
11.11Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
11.11Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
10.71Single7SK5CXCL127SK5-ACKR3-CXCL12
10.53Single6LI0C176LI0-GPR52-C17
10.53Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
10.53Single7UL2SR486927UL2-NTS1-SR48692-Na
10.53Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
10.53Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
10.53Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
10.53Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
10.53Consensusneurotensin_offOrthosteric Ligandnts1_off
10.53Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
10.00Single3ODUIT1t3ODU-CXCR4-IT1t
10.00Single5U09Taranabant5U09-CB1-Taranabant
10.00Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
10.00Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
10.00Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
10.00Single7F8YDevazepide7F8Y-CCKA-Devazepide
10.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
10.00Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
10.00Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
10.00Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
10.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
10.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
10.00Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
10.00Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
10.00Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
10.00Single9BA0A1AKN9BA0-CB1-A1AKN
10.00Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.00Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
9.52Single6ZINSR486926ZIN-NTS1-SR48692
9.52Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single7SK3CXCL127SK3-ACKR3-CXCL12
9.09Single5T04Neurotensin5T04-NTS1-Neurotensin
9.09Single6GPSMK08126GPS-CCR2-MK0812
9.09Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
9.09Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
9.09Single7F83PF-051904577F83-Ghrelin-PF-05190457
9.09Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
9.09Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
9.09Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
9.09Single7YXAONO-54306087YXA-S1P5-ONO-5430608
9.09Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
9.09Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
9.09Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
9.09Single9B9ZA1AKO9B9Z-CB1-A1AKO
9.09Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
9.09Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
8.82Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
8.70Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
8.70Single6GPXMK08126GPX-CCR2-MK0812
8.70Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
8.70Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
8.70Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
8.33Single6OS1TRV0266OS1-AT1-TRV026
8.33Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
8.33Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
8.33Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
8.33Single9BJKNAM9BJK-μ-Naloxone-NAM
8.00Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
8.00Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
7.69Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
7.69Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
7.69Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
7.41Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
7.41Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
7.41Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
7.14Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
7.14Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
7.14Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
6.90Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
6.67Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
6.25Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
6.25Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single7WC4Serotonin7WC4-5-HT2A-Serotonin
5.88Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.56Single3OE8IT1t3OE8-CXCR4-IT1t
5.56Single6TQ9SB-4081246TQ9-OX1-SB-408124
5.56Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
5.56Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
5.56Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
5.26Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
5.26Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
5.26Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
5.00Single4O9RCyclopamine4O9R-SMO-Cyclopamine
5.00Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
5.00Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
5.00Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
5.00Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.76Single4K5YCP-3763954K5Y-CRF1-CP-376395
4.76Single4QINSAG1.54QIN-SMO-SAG1.5
4.76Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
4.76Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
4.76Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
4.55Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
4.55Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
4.55Single8JD6N-(3-chlorophenyl)pyridine-2-carboxamide8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.35Single4Z9GCP-3763954Z9G-CRF1-CP-376395
4.35Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
4.35Single8GTIBMK-C2058GTI-CRF1-BMK-C205
4.35Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
4.17Single8GTGBMK-I1528GTG-CRF1-BMK-I152
4.17Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
4.00Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
4.00Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
3.85Single7SHEPI; PE7SHE-GPR158-PI; PE
3.85Single8GTMBMK-C2038GTM-CRF1-BMK-C203
3.70Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
3.33Single7SHEPI; PE7SHE-GPR158-PI; PE
3.33Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7

Consensus Members
Id Members
8HDP 8HDP-A2B-Adenosine-Gs/β1/γ2
7XY6 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
7XY7 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
8HDO 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
Net Summary
Imin 2.7825
Number of Linked Nodes 909
Number of Links 1069
Number of Hubs 161
Number of Links mediated by Hubs 609
Number of Communities 28
Number of Nodes involved in Communities 207
Number of Links involved in Communities 286
Path Summary
Number Of Nodes in MetaPath 103
Number Of Links MetaPath 102
Number of Shortest Paths 2709967
Length Of Smallest Path 3
Average Path Length 43.909
Length of Longest Path 80
Minimum Path Strength 0.36
Average Path Strength 5.80314
Maximum Path Strength 21.335
Minimum Path Correlation 0.7
Average Path Correlation 0.981342
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.33333
Average % Of Corr. Nodes 31.7047
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 46.0626
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
a2_on_gpa2b_on_gp



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