Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
11x50 6.8654189
21x52 4.39254146
31x57 4.93407
4I1x49 8.615476
52x46 4.618519
62x50 6.185189
72x64 4.67403
8E1x50 7.5285108
9E1x52 5.4854107
103x29 7.5075406
113x34 4.6454215
123x37 4.628517
133x50 7.0275409
14I2x51 4.9225405
15I2x57 7.04254197
16E2.M165 2.6954203
17E2x51 4.44113
18E2.Y172 12.6454114
195x39 6.6954115
205x46 4.4125415
215x47 5.172518
225x50 4.295419
235x51 4.2516
245x58 5.25228
255x64 5.8954235
266x44 4.2925419
276x48 4.635619
286x51 7.8925406
296x52 4.142508
306x58 2.8825243
316x61 6.825402
327x42 3.2575416
337x53 5.244519
347x55 3.71754147
357x58 2.6075404
367x62 5.235146
37G.HN.43 3.5625409
38G.S1.02 5.0325405
39G.H1.01 2.98333609
40G.H1.10 4.255408
41G.S3.02 5.7375444
42G.S3.04 9.935446
43G.S3.05 3.61507
44G.S3.06 8.1525445
45G.S3.08 5.5175409
46G.h2s4.01 4.326549
47G.S4.04 5.7325489
48G.S4.05 3.524267
49G.s4h3.03 6.185438
50G.s4h3.04 6.8875438
51G.s4h3.05 5.986539
52G.H3.09 5.432589
53G.H3.13 4.026585
54G.H3.17 8.62405
55G.H3.18 5.334289
56G.S5.04 3.6225489
57G.S5.05 3.54667609
58G.HG.04 4.12167639
59G.HG.15 4.73437
60G.hgh4.01 4.21436
61G.hgh4.02 4.28667637
62G.H4.03 5.2275404
63G.H4.11 3.0375437
64G.H4.15 3.165408
65G.h4s6.02 4.345488
66G.S6.02 6.695257
67G.S6.04 6.99409
68G.H5.08 4.0954278
69G.H5.23 4.09754194
70b.lhb1x6 3.9185123
71b.b1x6 6.1409
72b.l1x3 8.0945169
73b.b2x5 7.228507
74b.b3x6 6.54754169
75b.l3x2 4.795169
76b.b4x6 9.64409
77b.l4x2 9.92754154
78b.b5x3 6.818509
79b.b5x5 3.9025405
80b.l5x1 4.1725498
81b.l5x5 6.31286749
82b.b6x5 3.5325406
83b.l6x5 5.5054174
84b.b7x1 5.85254174
85b.l7x2 4.6875449
86b.b8x4 4.782596
87b.b9x4 5.5475409
88b.l9x3 5.30571769
89b.l9x6 4.584548
90b.b10x5 4.005669
91b.l10x1 3.945403
92b.l11x2 6.918569
93b.b12x6 8.02667668
94b.l12x1 3.4075466
95b.b13x3 6.0875464
96b.b13x7 5.694557
97b.l13x3 6.47429759
98b.l13x6 4.292549
99b.b14x3 3.5975455
100b.b15x1 5.054559
101b.b15x3 3.985459
102b.l15x2 5.055459
103b.b16x4 9.215456
104b.b16x5 3.4725405
105b.b16x6 7.082558
106b.b17x7 6.76428
107b.l17x3 8.48529
108b.l17x6 5.406529
109b.b18x3 4.015428
110b.b18x5 4.2875405
111b.l18x1 5.551437136
112b.b19x2 5.41526
113b.b19x4 4.4428
114b.l19x2 7.136529
115b.b20x3 2.616508
116b.b20x4 8.688528
117b.b20x6 5.67167626
118b.b20x7 2.8175409
119b.l20x2 5.7475409
120b.b21x7 4.224505
121b.b22x5 3.4925137
122b.l22x5 6.474129
123b.b23x6 4.888507
124b.b24x5 3.0675405
125b.b24x7 5.82254129
126b.b25x3 4.165405
127b.b25x7 5.775477
128b.l25x3 9.1075479
129b.l26x3 6.26254307
130b.b27x3 3.9275408
131b.l27x1 12.3465299
132b.l27x2 7.206579
133b.b28x4 4.9275476
134b.b28x6 6.548579
135g.h1x13 3.485409
136g.l1x6 4.7925408
137g.h2x13 4.66754136
138g.ctx5 4.865609
139g.ctx8 3.2885126
140g.ctx17 5.6354159
141g.ctx18 5.1356158
142Lig 6.591821110
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
16x48 Lig 43.46913.54YesYes190
26x44 6x48 51.76535.01YesYes199
33x43 6x44 63.09672.51NoYes189
43x43 7x53 63.37036.04NoYes189
53x50 7x53 41.378.23YesYes099
63x50 5x58 42.65937.2YesYes098
73x47 5x58 85.44933.82NoYes2298
83x47 5x57 85.77123.26NoNo096
93x51 5x57 85.92646.52NoNo086
103x51 5x61 86.08153.1NoNo088
115x61 5x65 86.39172.85NoNo088
125x65 I3.R215 87.47612.43NoNo085
13I3.F213 I3.R215 87.78554.28NoNo045
145x68 I3.F213 90.25446.41NoNo054
155x68 G.H5.13 93.81479.53NoNo058
16G.H5.13 G.S6.02 93.95383.45NoYes2587
17G.H5.10 G.S6.02 95.03158.01NoYes067
18G.H5.10 G.S5.03 95.18373.25NoNo068
19G.S5.03 G.S5.05 47.76432.51NoYes089
20G.S5.05 G.S6.04 51.17485.66YesYes099
21G.S6.04 G.s6h5.05 99.03825.04YesNo099
22G.s6h5.02 G.s6h5.05 99.20453.11NoNo079
23G.HG.01 G.s6h5.02 99.37053.23NoNo057
24G.H4.03 G.HG.01 99.5367.17YesNo045
25G.H4.03 G.HG.04 66.70484.13YesYes049
26G.HG.04 G.s4h3.01 33.49353.65YesNo397
27G.S5.06 G.s4h3.01 33.49825.54NoNo087
28G.S5.04 G.S5.06 66.33532.77YesNo098
29G.S4.04 G.S5.04 65.83613.65YesYes899
30G.H3.08 G.S4.04 1004.87NoYes099
31G.H2.04 G.H3.08 99.94373.64NoNo099
32G.H2.04 G.H2.07 99.83254NoNo099
33G.H2.07 G.S3.08 99.77627.36NoYes099
34G.S2.01 G.S3.08 47.45899.22NoYes099
35G.S2.01 b.l5x5 36.78453.52NoYes499
36b.l3x1 b.l5x5 72.16359.86NoYes099
37b.b2x1 b.l3x1 72.002410.15NoNo089
38b.b2x1 b.l27x1 71.50153.86NoYes2989
39b.l25x6 b.l27x1 70.663916.99NoYes089
40b.l23x1 b.l25x6 70.503717.87NoNo068
41b.l21x7 b.l23x1 70.18356.22NoNo056
42b.b23x6 b.l21x7 69.8642.69YesNo075
43b.b23x6 b.b24x6 64.86233.86YesNo078
44b.b21x7 b.b24x6 64.70243.86YesNo058
45b.b21x5 b.b21x7 62.59398.38NoYes045
46b.b21x5 b.h2x1 62.4311.31NoNo045
47b.h2x1 b.h2x5 61.28082.95NoNo055
48b.h2x5 b.lhb1x3 61.11653.04NoNo052
49b.l22x5 b.lhb1x3 60.45873.76YesNo092
506x40 7x53 41.33814.84NoYes079
515x58 6x40 42.49273.63YesNo087
52G.H5.06 G.S5.03 47.57342.51NoNo038
53G.H5.06 G.S6.04 47.642614.71NoYes039
54G.H4.03 G.H4.07 33.11224YesNo045
55G.H4.07 G.S6.05 33.11142.77NoNo054
56G.S5.06 G.S6.05 32.87086.09NoNo084
57G.H4.11 G.HG.04 33.61892.51YesYes379
58G.H4.11 G.H4.15 33.56622.51YesYes078
59G.H4.15 G.S4.06 33.80923.93YesNo087
60G.S4.04 G.S4.06 33.80552.62YesNo097
61G.S3.08 G.h2s4.01 38.1982.62YesYes099
62G.h2s4.01 b.l5x5 36.83746.01YesYes499
632x50 7x49 16.38436.73YesNo099
642x46 7x49 16.71776.87YesNo099
652x60 Lig 10.446218.93NoYes060
662x60 3x29 10.10956.79NoYes066
674x61 Lig 10.44622.78NoYes040
683x29 4x61 10.10954.15YesNo064
693x29 4x65 10.105814.67YesNo065
706x51 6x52 12.03445.44YesYes068
71b.l22x5 g.ctx8 51.70254.86YesYes1296
72g.ctx5 g.ctx8 51.27994.07YesYes096
73g.ctx5 g.ctx6 50.87464.83YesNo097
74b.l26x5 g.ctx6 48.26435.03NoNo057
75b.l26x5 g.ctx17 46.72583.35NoYes059
76g.ctx17 g.ctx18 42.55244.33YesYes1598
77b.b1x4 g.ctx18 41.60988.55NoYes078
78b.b1x4 b.b5x1 20.71982.59NoNo075
79b.b1x6 b.b5x1 20.54692.95YesNo095
80b.b1x6 b.b4x6 40.396610.25YesYes099
81b.b4x6 b.b5x3 31.63389.28YesYes099
82G.HN.43 b.b5x3 30.6077.27YesYes099
83G.HN.39 G.HN.43 28.87362.51NoYes059
84b.b1x4 b.b28x5 20.71983.76NoNo075
85b.b1x6 b.b28x5 20.54694.28YesNo095
86G.HN.39 b.b5x5 28.52323.39NoYes055
87G.S3.08 G.s3h2.03 14.09582.87YesNo099
88G.S2.01 b.l7x2 10.60515.71NoYes499
89G.s3h2.03 b.l7x2 11.01952.66NoYes099
90b.l7x2 b.l9x6 22.00334.69YesYes498
91G.H2.06 b.l9x6 12.30773.58NoYes098
92G.H2.06 b.l17x6 11.95766.91NoYes099
93b.l17x5 b.l17x6 11.52535.89NoYes269
94b.l17x5 b.l19x2 11.37835.89NoYes269
95b.b4x5 b.b5x5 13.73525.3NoYes075
96b.b3x3 b.b4x5 13.03253.07NoNo087
97b.b3x3 b.b4x3 12.68114.47NoNo087
98b.b4x3 b.l5x1 24.65892.77NoYes078
99b.b5x5 b.l8x8 14.08742.77YesNo054
100b.b5x7 b.l8x8 13.38473.07NoNo074
101b.b4x3 b.b5x7 12.68182.85NoNo077
102b.b8x4 b.l5x1 20.43494.69YesYes968
103b.b7x2 b.b8x4 16.91693.79NoYes086
104b.b6x5 b.b7x2 16.21252.52YesNo068
105b.b6x5 b.l6x4 13.39464.35YesNo065
106b.l6x3 b.l6x4 12.693.71NoNo065
1072x46 7x53 18.34863.52YesYes199
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
1x352x643.150NoYes5321
1x362x642.850NoYes5321
1x397x424.870NoYes7621
2x537x422.620NoYes6621
2x603x296.790NoYes6612
2x60Lig18.930NoYes6010
2x64Lig11.180YesYes3010
3x294x614.150YesNo6421
3x366x483.491NoYes7911
3x36Lig5.271NoYes7010
3x374x532.541YesNo7812
3x374x5610.551YesNo7412
3x375x463.751YesYes7512
3x37Lig4.371YesYes7010
4x565x462.951NoYes4522
4x61Lig2.780NoYes4010
5x395x437.3911YesNo5521
5x436x552.630NoNo5612
5x43Lig8.240NoYes5010
6x446x485.011YesYes9921
6x486x523.171YesYes9812
6x487x415.191YesNo9812
6x487x457.411YesNo9912
6x48Lig3.541YesYes9010
6x516x525.440YesYes6822
6x516x5515.120YesNo6622
6x517x384.840YesNo6521
7x35Lig6.830NoYes4010
7x387x422.511NoYes5611
7x38Lig6.211NoYes5010
7x42Lig3.031YesYes6010
3x33Lig2.130NoYes4010
3x323x331.960NoNo6421
3x373x411.931YesNo7512
1x322x641.50NoYes4321

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
100.00Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
100.00Consensusblt_onOrthosteric Ligandblt1_on
100.00Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
100.00Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
100.00Consensusleukotriene_onOrthosteric Ligandblt_on
100.00Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
58.82Single7SK9CCX6627SK9-ACKR3-CCX662
47.37Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
47.06Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
47.06Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
46.67Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
44.44Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
44.44Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
44.44Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
44.44Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
44.44Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
44.44Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
43.75Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
43.75Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
43.75Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
43.75Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
43.75Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
43.75Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
42.86Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
42.86Single6B73MP11046B73-κ-MP1104
42.86Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
42.86Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
42.86Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
42.86Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
42.11Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
42.11Single8X5YAstemizole8X5Y-H1-Astemizole
42.11Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
42.11Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
41.18Single4DJHJDTic4DJH-κ-JDTic
41.18Single4U15Tiotropium4U15-M3-Tiotropium
41.18Single6OL9Tiotropium6OL9-M5-Tiotropium
41.18Single6TQ7SB-3348676TQ7-OX1-SB-334867
41.18Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
41.18Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
41.18Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
41.18Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
41.18Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
41.18Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
41.18Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
41.18Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
41.18Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
41.18Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
41.18Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
41.18Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
41.18Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
41.18Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
41.18Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
40.91Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
40.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
40.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
40.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
40.00Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
40.00Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
40.00Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
40.00Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
40.00Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
40.00Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
40.00Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
40.00Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
40.00Single8K5CAcipimox8K5C-HCA2-Acipimox
40.00Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
40.00Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.00Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
40.00Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
40.00Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
40.00Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
40.00Consensusalpha1_onOrthosteric Ligandalpha1a_on
40.00Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
40.00Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
40.00Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
40.00Consensuslpl_onOrthosteric Ligands1p_on lpa_on
40.00Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
38.89Single3D4STimolol3D4S-β2-Timolol
38.89Single5CXVTiotropium5CXV-M1-Tiotropium
38.89Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
38.89Single6A93Risperidone6A93-5-HT2A-Risperidone
38.89Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
38.89Single6ZG4HTL00099366ZG4-M1-HTL0009936
38.89Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
38.89Single7YITNalfurafine7YIT-κ-Nalfurafine
38.89Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
38.89Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
38.89Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
38.89Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
38.89Single8JWZAB9288JWZ-A2A-AB928-Na
38.89Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
38.89Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
38.89Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
38.89Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
38.89Consensusalpha1_offOrthosteric Ligandalpha1a_off
38.89Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
38.89Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
38.89Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
38.89Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
38.89Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
38.89Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
38.89Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
38.89Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
38.89Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
38.46Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
38.10Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
38.10Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
38.10Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
37.50Single3NY8ICI118-5513NY8-β2-ICI118-551
37.50Single4EJ4Naltrindole4EJ4-δ-Naltrindole
37.50Single4GBRS-Carazolol4GBR-β2-S-Carazolol
37.50Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
37.50Single4YAYZD-71554YAY-AT1-ZD-7155
37.50Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
37.50Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
37.50Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
37.50Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
37.50Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
37.50Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
37.50Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
37.50Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
37.50Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
37.50Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
37.50Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
37.50Single8JXRLSD8JXR-D1-LSD
37.50Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
37.50Single8T1WCVN4248T1W-GPR6-CVN424
37.50Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
37.50Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
37.50Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
37.50Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
37.50Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
37.50Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
37.50Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
37.50Consensusalpha2_onOrthosteric Ligandalpha2b_on
37.50Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
37.50Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
37.50Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
37.50Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
37.50Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
37.50Consensusdopamine_offOrthosteric Ligandd2_off d3_off
37.50Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
37.50Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
37.50Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
37.50Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
37.50Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
37.50Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
36.84Single5X93K-87945X93-ETB-K-8794
36.84Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
36.84Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
36.84Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
36.84Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
36.84Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
36.84Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.84Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
36.84Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
36.84Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
36.84Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
36.84Consensusendothelin_offOrthosteric Ligandetb_off
36.84Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
36.84Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
36.36Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
35.71Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
35.71Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
35.71Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
35.71Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
35.71Single8K5BNiacin8K5B-HCA2-Niacin
35.71Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
35.71Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
35.71Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
35.29Single2RH1S-Carazolol2RH1-β2-S-Carazolol
35.29Single2YCWS-Carazolol2YCW-β1-S-Carazolol
35.29Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
35.29Single5C1MBU725C1M-μ-BU72
35.29Single5D6LS-Carazolol5D6L-β2-S-Carazolol
35.29Single5WQCEMPA5WQC-OX2-EMPA
35.29Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
35.29Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
35.29Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
35.29Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
35.29Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
35.29Single6TP6Filorexant6TP6-OX1-Filorexant
35.29Single7C4SS1P7C4S-S1P3-S1P
35.29Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
35.29Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
35.29Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
35.29Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
35.29Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
35.29Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.29Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.29Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
35.29Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
35.29Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
35.29Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
35.29Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
35.29Single8ZMFA1L108ZMF-5-HT2C-A1L10
35.29Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
35.29Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
35.29Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
35.29Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
35.29Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
35.29Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
35.29Consensusamine_offonOrthosteric Ligandamine_off amine_on
35.29Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
35.29Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
35.29Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
35.29Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
35.29Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
35.29Consensusblt_offOrthosteric Ligandblt1_off
35.29Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
35.29Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
35.29Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
35.29Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
35.29Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
35.29Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
35.29Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.29Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.29Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
35.29Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
35.29Consensustrace-amine_onOrthosteric Ligandta1_on
35.00Single4UG2CGS216804UG2-A2A-CGS21680
35.00Single5ZTYAM102575ZTY-CB2-AM10257
35.00Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
35.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
35.00Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
34.78Single6JODAngiotensin II6JOD-AT2-Angiotensin II
34.78Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
33.33Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
33.33Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
33.33Single2YDVNECA2YDV-A2A-NECA
33.33Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
33.33Single4IARErgotamine4IAR-5-HT1B-Ergotamine
33.33Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
33.33Single4UHRCGS216804UHR-A2A-CGS21680
33.33Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
33.33Single5D5AS-Carazolol5D5A-β2-S-Carazolol
33.33Single5D5BS-Carazolol5D5B-β2-S-Carazolol
33.33Single5G53NECA5G53-A2A-NECA-Gs
33.33Single5V54Methiothepin5V54-5-HT1B-Methiothepin
33.33Single5WS3EMPA5WS3-OX2-EMPA
33.33Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
33.33Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
33.33Single6AKXA4R6AKX-CCR5-A4R
33.33Single6AKYMaraviroc6AKY-CCR5-Maraviroc
33.33Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
33.33Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
33.33Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
33.33Single6TODEMPA6TOD-OX1-EMPA-Na
33.33Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
33.33Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
33.33Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
33.33Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
33.33Single7FEECP559407FEE-CB1-CP55940-ZCZ011
33.33Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
33.33Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
33.33Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
33.33Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
33.33Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
33.33Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
33.33Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
33.33Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
33.33Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
33.33Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
33.33Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
33.33Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
33.33Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
33.33Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
33.33Single8E0GBU728E0G-μ-BU72
33.33Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
33.33Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
33.33Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
33.33Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
33.33Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
33.33Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
33.33Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
33.33Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
33.33Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
33.33Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
33.33Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
33.33Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
33.33Single8IWESpermidine8IWE-TA9-Spermidine
33.33Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
33.33Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
33.33Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
33.33Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
33.33Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
33.33Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
33.33Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
33.33Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
33.33Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
33.33Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
33.33Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
33.33Single8WDTphotoNECA8WDT-A2A-photoNECA
33.33Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
33.33Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
33.33Single8Y0HVUF114188Y0H-CXCR3-VUF11418
33.33Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
33.33Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
33.33Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
33.33Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
33.33Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
33.33Consensus5ht1_offOrthosteric Ligand5ht1b_off
33.33Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
33.33Consensusa2_onOrthosteric Liganda2b_on
33.33Consensusa2_on_gpOrthosteric Liganda2b_on_gp
33.33Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
33.33Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
33.33Consensusangiotensin_offOrthosteric Ligandat1_off
33.33Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
33.33Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
33.33Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
33.33Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
33.33Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
33.33Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
33.33Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
33.33Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
33.33Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
33.33Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
33.33Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
33.33Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
33.33Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
33.33Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
33.33Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
33.33Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
33.33Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
33.33Consensusorexin_offOrthosteric Ligandox2_off ox1_off
33.33Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
33.33Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
33.33Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
33.33Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
33.33Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
33.33Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
33.33Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
31.82Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
31.82Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
31.58Single4AMIBucindolol4AMI-β1-Bucindolol
31.58Single4LDEBI1671074LDE-β2-BI167107
31.58Single5X33BIIL2605X33-BLT1-BIIL260
31.58Single6CM4Risperidone6CM4-D2-Risperidone
31.58Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
31.58Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
31.58Single6KQICP559406KQI-CB1-CP55940-Org27569
31.58Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
31.58Single7DFPSpiperone7DFP-D2-Spiperone
31.58Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
31.58Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
31.58Single7K15MKD0467K15-BLT1-MKD046-Na
31.58Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
31.58Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
31.58Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
31.58Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.58Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
31.58Single8JJ8Formoterol8JJ8-β2-Formoterol
31.58Single8JWY2-1188JWY-A2A-2-118
31.58Single8XYIVUF106618XYI-CXCR3-VUF10661
31.58Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
31.58Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
31.58Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
31.58Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
31.58Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
31.58Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
31.58Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
31.58Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
31.58Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
31.58Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
31.58Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
31.58Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
31.58Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
31.58Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
31.58Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
31.58Consensusorexin_onOrthosteric Ligandox2_on
31.58Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
31.25Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
31.25Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
31.25Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
31.25Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
31.25Single4MBSMaraviroc4MBS-CCR5-Maraviroc
31.25Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
31.25Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
31.25Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
31.25Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
31.25Single6PS0S-Carazolol6PS0-β2-S-Carazolol
31.25Single6PS4ICI118-5516PS4-β2-ICI118-551
31.25Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
31.25Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
31.25Single6TPGEMPA6TPG-OX2-EMPA
31.25Single6TPNHTL66416TPN-OX2-HTL6641
31.25Single6VI4JDTic6VI4-κ-JDTic
31.25Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
31.25Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
31.25Single6ZG9GSK10347026ZG9-M1-GSK1034702
31.25Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
31.25Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
31.25Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
31.25Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
31.25Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
31.25Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
31.25Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
31.25Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
31.25Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
31.25Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.25Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
31.25Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
31.25Single7UL3Famotidine7UL3-H2-Famotidine
31.25Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
31.25Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
31.25Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
31.25Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
31.25Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
31.25Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
31.25Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
31.25Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
31.25Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
31.25Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
31.25Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
31.25Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.25Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
31.25Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
31.25Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
31.25Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
31.25Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
31.25Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
31.25Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
31.25Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
31.25Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
31.25Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
31.25Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
31.25Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
31.25Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
31.25Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
31.25Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.25Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
31.25Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
31.25Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
31.25Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
31.25Single9BJKNaloxone9BJK-μ-Naloxone-NAM
31.25Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
31.25Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
31.25Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
31.25Consensushca_onOrthosteric Ligandhca2_on
30.77Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
30.77Single6TQ9SB-4081246TQ9-OX1-SB-408124
30.77Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
30.77Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
30.77Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
30.77Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.77Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
30.77Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
30.77Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
30.43Single5WF5UK-4320975WF5-A2A-UK-432097
30.43Single6PT2KGCHM076PT2-δ-KGCHM07
30.43Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
30.43Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
30.43Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
30.43Consensusangiotensin_onOrthosteric Ligandat1_on
30.43Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
30.43Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
30.00Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
30.00Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
30.00Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
30.00Single6H7LDobutamine6H7L-β1-Dobutamine
30.00Single6IBLArformoterol6IBL-β1-Arformoterol
30.00Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
30.00Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
30.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
30.00Single7EZCUKA7EZC-A2A-UKA
30.00Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
30.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
30.00Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
30.00Single7UM4AS26747237UM4-5-HT5A-AS2674723
30.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
30.00Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
30.00Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
30.00Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
30.00Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.00Single8XVJMacitentan8XVJ-ETA-Macitentan
30.00Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
30.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
30.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
30.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
30.00Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
30.00Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
30.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
30.00Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
30.00Consensusprostanoid_offOrthosteric Ligandep_off dp_off
29.41Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
29.41Single2Y01Dobutamine2Y01-β1-Dobutamine
29.41Single2Y04Salbutamol2Y04-β1-Salbutamol
29.41Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
29.41Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
29.41Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
29.41Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
29.41Single4MQSIperoxo4MQS-M2-Iperoxo
29.41Single4QKX35V4QKX-β2-35V
29.41Single4U14Tiotropium4U14-M3-Tiotropium
29.41Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
29.41Single5DHHSB-6121115DHH-NOP-SB-612111
29.41Single5DSGTiotropium5DSG-M4-Tiotropium
29.41Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
29.41Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
29.41Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
29.41Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
29.41Single6GPSMK08126GPS-CCR2-MK0812
29.41Single6H7MSalbutamol6H7M-β1-Salbutamol
29.41Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
29.41Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
29.41Single6TOTLemborexant6TOT-OX1-Lemborexant
29.41Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.41Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
29.41Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
29.41Single7BU7BI1671077BU7-β1-BI167107
29.41Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
29.41Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
29.41Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
29.41Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
29.41Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
29.41Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
29.41Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
29.41Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
29.41Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
29.41Single7UL4Alvimopan7UL4-μ-Alvimopan
29.41Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
29.41Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
29.41Single7V3ZCP559407V3Z-CB1-CP55940
29.41Single7WC7Lisuride7WC7-5-HT2A-Lisuride
29.41Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
29.41Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
29.41Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
29.41Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
29.41Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
29.41Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
29.41Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
29.41Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
29.41Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
29.41Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
29.41Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
29.41Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
29.41Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
29.41Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
29.41Single8JJOAlprenolol8JJO-β2-Alprenolol
29.41Single8K5DGSK2560738K5D-HCA2-GSK256073
29.41Single8RLNLUF58348RLN-A2A-LUF5834
29.41Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
29.41Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
29.41Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
29.41Single8X64Desloratadine8X64-H1-Desloratadine
29.41Single9CHXS-Carazolol9CHX-β2-S-Carazolol
29.41Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
29.41Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
29.41Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
29.41Consensus5ht5_onOrthosteric Ligand5ht5a_on
29.41Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
29.41Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
29.41Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
29.41Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
29.41Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
29.41Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
29.41Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
29.41Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
29.41Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
29.41Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
29.41Consensushca_on_gpOrthosteric Ligandhca2_on_gp
29.41Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
29.17Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
29.17Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
29.17Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
29.17Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
29.17Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
29.17Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
29.17Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
29.17Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
29.17Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
28.57Single3NY9ICI118-5513NY9-β2-ICI118-551
28.57Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
28.57Single5WF6UK-4320975WF6-A2A-UK-432097
28.57Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
28.57Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
28.57Single6PT3DPI-2876PT3-δ-DPI-287
28.57Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
28.57Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
28.57Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
28.57Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
28.57Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
28.57Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
28.57Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
28.57Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
28.57Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
28.57Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
28.57Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
28.57Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
28.57Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
28.57Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
28.57Consensusbombesin_onOrthosteric Ligandbb2_on
28.57Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
28.57Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
28.57Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
28.57Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
28.57Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
28.57Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
28.57Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
28.57Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
28.00Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
28.00Single8ZRTET-18ZRT-ETB-ET-1
27.78Single2Y00Dobutamine2Y00-β1-Dobutamine
27.78Single2Y03Isoprenaline2Y03-β1-Isoprenaline
27.78Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
27.78Single5JQHS-Carazolol5JQH-β2-S-Carazolol
27.78Single5WIUNemonapride5WIU-D4-Nemonapride
27.78Single5WIVNemonapride5WIV-D4-Nemonapride-Na
27.78Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
27.78Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
27.78Single6E67BI1671076E67-β2-BI167107-Gs (fused)
27.78Single6GPXMK08126GPX-CCR2-MK0812
27.78Single6HLPNetupitant6HLP-NK1-Netupitant
27.78Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
27.78Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
27.78Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
27.78Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
27.78Single6PS6Timolol6PS6-β2-Timolol
27.78Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
27.78Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
27.78Single7C61Ergotamine7C61-5-HT1B-Ergotamine
27.78Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
27.78Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
27.78Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
27.78Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
27.78Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
27.78Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
27.78Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
27.78Single7WC6LSD7WC6-5-HT2A-LSD
27.78Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.78Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
27.78Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
27.78Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
27.78Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
27.78Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.78Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
27.78Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
27.78Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
27.78Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.78Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
27.78Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
27.78Single8TF5Oleic acid8TF5-GPR6-Oleic acid
27.78Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.78Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.78Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
27.78Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
27.78Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
27.78Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
27.78Consensusa3_on_gpOrthosteric Liganda3a_on_gp
27.78Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
27.78Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
27.78Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
27.78Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
27.78Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
27.78Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
27.78Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
27.78Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
27.78Consensusep_offOrthosteric Ligandep4_off
27.78Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
27.78Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
27.78Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
27.27Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
27.27Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
27.27Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
27.27Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
27.27Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
26.92Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
26.92Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
26.67Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
26.67Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
26.67Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
26.67Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
26.67Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
26.67Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
26.67Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
26.67Single7SRQLSD7SRQ-5-HT2B-LSD
26.67Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
26.67Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
26.67Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
26.67Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
26.67Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
26.67Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
26.67Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
26.67Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.67Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
26.67Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
26.67Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
26.67Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
26.67Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
26.67Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
26.67Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
26.67Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
26.67Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
26.32Single3P0GBI1671073P0G-β2-BI167107
26.32Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
26.32Single5XR8AM8415XR8-CB1-AM841
26.32Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
26.32Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
26.32Single6H7JIsoprenaline6H7J-β1-Isoprenaline
26.32Single6J21Aprepitant6J21-NK1-Aprepitant
26.32Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
26.32Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
26.32Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
26.32Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
26.32Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
26.32Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
26.32Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
26.32Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
26.32Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
26.32Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
26.32Single8EA0Iperoxo8EA0-M3-Iperoxo
26.32Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
26.32Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
26.32Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
26.32Single8XVLZibotentan8XVL-ETA-Zibotentan
26.32Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
26.32Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
26.32Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
26.32Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
26.32Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
26.32Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
26.32Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
26.32Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
26.32Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
26.32Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
26.32Consensustachykinin_offOrthosteric Ligandnk1_off
26.09Single3QAKUK-4320973QAK-A2A-UK-432097
26.09Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
26.09Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
26.09Single6HLOAprepitant6HLO-NK1-Aprepitant
26.09Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
26.09Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
26.09Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
26.09Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
26.09Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
26.09Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
26.09Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
26.09Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
26.09Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
25.93Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
25.93Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
25.93Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
25.93Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
25.00Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
25.00Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
25.00Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
25.00Single4RWADIPP-NH24RWA-δ-DIPP-NH2
25.00Single4S0VSuvorexant4S0V-OX2-Suvorexant
25.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
25.00Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
25.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
25.00Single6IGLIRL16206IGL-ETB-IRL1620
25.00Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
25.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
25.00Single6ME9Ramelteon6ME9-MT2-Ramelteon
25.00Single6MXTSalmeterol6MXT-β2-Salmeterol
25.00Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
25.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
25.00Single6TPJSuvorexant6TPJ-OX2-Suvorexant
25.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
25.00Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
25.00Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
25.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
25.00Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
25.00Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
25.00Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
25.00Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
25.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
25.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
25.00Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
25.00Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
25.00Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
25.00Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
25.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
25.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
25.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
25.00Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
25.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
25.00Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
25.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
25.00Single7XRRLemborexant7XRR-OX2-Lemborexant
25.00Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
25.00Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
25.00Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
25.00Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
25.00Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
25.00Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
25.00Single8JJLOlodaterol8JJL-β2-Olodaterol
25.00Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
25.00Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
25.00Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
25.00Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
25.00Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
25.00Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
25.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
25.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
25.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
25.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
25.00Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
25.00Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
25.00Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
25.00Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
25.00Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
25.00Consensuslpa_offOrthosteric Ligandlpa1_off
25.00Consensuslpl_offOrthosteric Ligands1p_off lpa_off
25.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
25.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
25.00Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
25.00Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
25.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
24.00Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
24.00Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.00Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
24.00Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
24.00Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
24.00Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
24.00Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
24.00Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
24.00Consensusvasop-oxy_onOrthosteric Ligandv2_on
24.00Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
23.81Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
23.81Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
23.81Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
23.81Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
23.81Single6K1QIRL25006K1Q-ETB-IRL2500
23.81Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
23.81Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
23.81Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
23.81Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
23.81Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
23.81Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
23.81Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
23.53Single2YDOAdenosine2YDO-A2A-Adenosine
23.53Single3RZECidoxepin3RZE-H1-Cidoxepin
23.53Single6A94Zotepine6A94-5-HT2A-Zotepine
23.53Single6KUXRS-799486KUX-α2a-RS-79948
23.53Single6PS5S-Propranolol6PS5-β2-S-Propranolol
23.53Single6TP3Nemorexant6TP3-OX1-Nemorexant
23.53Single6V9SGTPL114036V9S-OX1-GTPL11403
23.53Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
23.53Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
23.53Single7T32ZM-2413857T32-A2A-ZM-241385
23.53Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
23.53Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
23.53Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
23.53Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.53Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.53Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
23.53Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
23.53Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
23.53Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
23.53Single8IHKAcifran8IHK-HCA3-Acifran
23.53Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
23.53Single8K2WAMG4878K2W-CXCR3-AMG487
23.53Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
23.53Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
23.53Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.53Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.53Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.53Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.53Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
23.53Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
23.53Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
23.53Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
23.53Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
23.53Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
23.53Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
23.53Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
23.53Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
23.53Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
23.53Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
23.53Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
23.53Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
23.53Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.53Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
23.53Consensusopsins_offOrthosteric Ligandrhodopsin_off
23.53Consensussensory_offOrthosteric Ligandopsins_off
23.33Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
23.33Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
23.08Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
23.08Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
23.08Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
23.08Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
23.08Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
23.08Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
23.08Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
23.08Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
23.08Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
23.08Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
23.08Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
23.08Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.73Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
22.73Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
22.73Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
22.73Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
22.73Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
22.73Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
22.73Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
22.73Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
22.73Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
22.22Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
22.22Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
22.22Single4DAJTiotropium4DAJ-M3-Tiotropium
22.22Single5DHGC-355DHG-NOP-C-35
22.22Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
22.22Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
22.22Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
22.22Single5UIGCmpd-15UIG-A2A-Cmpd-1
22.22Single6DRXLisuride6DRX-5-HT2B-Lisuride
22.22Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
22.22Single6PS1Timolol6PS1-β2-Timolol
22.22Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
22.22Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
22.22Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
22.22Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
22.22Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
22.22Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
22.22Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
22.22Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
22.22Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
22.22Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
22.22Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
22.22Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
22.22Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
22.22Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
22.22Single7YXAONO-54306087YXA-S1P5-ONO-5430608
22.22Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
22.22Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
22.22Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.22Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
22.22Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
22.22Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
22.22Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
22.22Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
22.22Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
22.22Single8X63Mepyramine8X63-H1-Mepyramine
22.22Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
22.22Single9IYAONO-97105319IYA-GPR55-ONO-9710531
22.22Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
22.22Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
22.22Consensusa3_onOrthosteric Liganda3a_on
22.22Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
22.22Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
22.22Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
22.22Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
22.22Consensushistamine_offOrthosteric Ligandh1_off
22.22Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
22.22Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
22.22Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
22.22Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
22.22Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
22.22Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
21.74Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
21.74Single7QA8Peptide7QA8-STE2-Peptide
21.74Single7QA8Peptide7QA8-STE2-Peptide
21.74Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
21.74Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
21.74Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
21.74Single8WKYPG-9348WKY-MC4-PG-934
21.74Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
21.74Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
21.74Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
21.74Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
21.74Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
21.74Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
21.74Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
21.74Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.43Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
21.43Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.43Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
21.43Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
21.43Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
21.43Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
21.43Single9CHUNoradrenaline9CHU-β2-Noradrenaline
21.43Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
21.43Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
21.43Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.43Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.43Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
21.43Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
21.43Consensussensory_onOrthosteric Ligandopsins_on
21.05Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
21.05Single5CGCHTL142425CGC-mGlu5-HTL14242
21.05Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
21.05Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
21.05Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
21.05Single5TVNLSD5TVN-5-HT2B-LSD
21.05Single5XPRBosentan5XPR-ETB-Bosentan
21.05Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
21.05Single6D26Fevipiprant6D26-DP2-Fevipiprant
21.05Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
21.05Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
21.05Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
21.05Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
21.05Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
21.05Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
21.05Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.05Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
21.05Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
21.05Single8JXSPF-61428JXS-D1-PF-6142
21.05Single8S4DCMF-0198S4D-Apelin-CMF-019
21.05Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
21.05Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
21.05Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
21.05Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
21.05Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
21.05Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
21.05Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
21.05Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
21.05Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
21.05Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
21.05Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
21.05Consensusdp_offOrthosteric Liganddp2_off
21.05Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
21.05Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
21.05Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.05Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.05Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
21.05Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.05Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.05Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
20.83Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
20.83Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
20.83Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
20.83Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
20.83Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
20.83Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
20.83Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
20.83Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
20.83Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
20.83Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
20.83Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
20.83Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
20.83Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
20.83Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
20.69Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
20.69Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
20.69Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
20.69Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
20.69Consensusbradykinin_onOrthosteric Ligandbk2_on
20.69Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
20.69Consensusendothelin_onOrthosteric Ligandetb_on eta_on
20.69Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
20.69Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
20.59Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.59Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.00Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
20.00Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
20.00Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
20.00Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
20.00Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
20.00Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
20.00Single5GLHEndothelin-15GLH-ETB-Endothelin-1
20.00Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
20.00Single5XRAAM115425XRA-CB1-AM11542
20.00Single6E59L-7607356E59-NK1-L-760735
20.00Single6IGKEndothelin-36IGK-ETB-Endothelin-3
20.00Single6J20Aprepitant6J20-NK1-Aprepitant
20.00Single6ME5Agomelatine6ME5-MT1-Agomelatine
20.00Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
20.00Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
20.00Single6W25SHU91196W25-MC4-SHU9119-Ca
20.00Single6WGTLSD6WGT-5-HT2A-LSD
20.00Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
20.00Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
20.00Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
20.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
20.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
20.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
20.00Single7P2L4YI7P2L-mGlu5-4YI
20.00Single7TUYGSK682753A7TUY-GPR183-GSK682753A
20.00Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
20.00Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
20.00Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
20.00Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
20.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
20.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
20.00Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
20.00Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
20.00Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
20.00Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
20.00Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
20.00Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
20.00Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
20.00Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.00Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
20.00Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
20.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
20.00Single9BJKNAM9BJK-μ-Naloxone-NAM
20.00Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
20.00Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
20.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
20.00Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
20.00Consensus5ht2_onOrthosteric Ligand5ht2b_on
20.00Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
20.00Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
20.00Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
20.00Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
20.00Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
20.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
20.00Consensuslpa_onOrthosteric Ligandlpa1_on
20.00Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
20.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
20.00Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
20.00Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
20.00Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
20.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
20.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
20.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
20.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
19.35Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
19.35Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
19.23Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
19.23Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
19.23Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
19.23Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
19.23Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
19.23Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
19.23Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
19.23Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
19.23Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
19.23Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
19.23Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
19.05Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
19.05Single4N4WSANT-14N4W-SMO-SANT-1
19.05Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
19.05Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
19.05Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
19.05Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
19.05Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
19.05Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
19.05Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
19.05Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
19.05Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.05Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
19.05Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
18.75Single3PBLEticlopride3PBL-D3-Eticlopride
18.75Single5L7IVismodegib5L7I-SMO-Vismodegib
18.75Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
18.75Single6HLLCP999946HLL-NK1-CP99994
18.75Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
18.75Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
18.75Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
18.75Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
18.75Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
18.75Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
18.75Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
18.75Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
18.75Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
18.75Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
18.75Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
18.75Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
18.75Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
18.75Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.75Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
18.75Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
18.75Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
18.75Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
18.75Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
18.75Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
18.52Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
18.52Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
18.52Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
18.52Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
18.52Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
18.52Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
18.52Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
18.52Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
18.52Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.18Single5CGDHTL142425CGD-mGlu5-HTL14242
18.18Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
18.18Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
18.18Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
18.18Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
18.18Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
18.18Consensuscck_onOrthosteric Ligandccka_on cckb_on
18.18Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
18.18Consensuschemerin_onOrthosteric Ligandcml1_on
18.18Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
18.18Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
18.18Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single4XT3Fractalkine4XT3-US28-Fractalkine
17.86Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
17.86Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
17.86Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
17.86Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
17.86Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
17.65Single3PWHZM-2413853PWH-A2A-ZM-241385
17.65Single5ZKQABT-4915ZKQ-PAF-ABT-491
17.65Single6DS0Ly2660976DS0-5-HT2B-Ly266097
17.65Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
17.65Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
17.65Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
17.65Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
17.65Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
17.65Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.65Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
17.65Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
17.65Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
17.65Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
17.65Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
17.65Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
17.65Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
17.65Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.65Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.65Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
17.65Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
17.65Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.65Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
17.65Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
17.65Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
17.50Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
17.39Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
17.39Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
17.39Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
17.39Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
17.39Single7XN9L-054,5227XN9-SST2-L-054,522
17.39Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
17.39Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
17.39Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
17.39Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
17.39Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
17.39Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
17.39Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
17.24Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
17.24Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
16.67Single3REYXAC3REY-A2A-XAC
16.67Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
16.67Single4XT1Fractalkine4XT1-US28-Fractalkine
16.67Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
16.67Single6AQFZM-2413856AQF-A2A-ZM-241385
16.67Single6FFIMMPEP6FFI-mGlu5-MMPEP
16.67Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
16.67Single6IQLL7458706IQL-D4-L745870
16.67Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
16.67Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
16.67Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
16.67Single6TPKRetosiban6TPK-OT-Retosiban
16.67Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
16.67Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
16.67Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
16.67Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
16.67Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
16.67Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
16.67Single7F8XNN90567F8X-CCKA-NN9056
16.67Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
16.67Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
16.67Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
16.67Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
16.67Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
16.67Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
16.67Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
16.67Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
16.67Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
16.67Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
16.67Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
16.67Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
16.67Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
16.67Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8IY6Endothelin-18IY6-ETB-Endothelin-1
16.67Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
16.67Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
16.67Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single8KIGSHU91198KIG-MC3-SHU9119-Ca
16.67Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
16.67Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
16.67Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
16.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
16.67Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
16.67Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
16.67Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
16.67Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
16.67Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
16.67Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
16.67Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
16.67Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
16.67Consensusvasop-oxy_offOrthosteric Ligandot_off
16.13Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
16.13Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
16.13Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
16.00Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
16.00Single7SK5CXCL127SK5-ACKR3-CXCL12
16.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
16.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
16.00Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
16.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
15.79Single2Y02Carmoterol2Y02-β1-Carmoterol
15.79Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
15.79Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
15.79Single5IU8Q274563475IU8-A2A-Q27456347-Na
15.79Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
15.79Single5TGZAM65385TGZ-CB1-AM6538
15.79Single6FFHFenobam6FFH-mGlu5-Fenobam
15.79Single6IIVDaltroban6IIV-TP-Daltroban
15.79Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
15.79Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
15.79Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
15.79Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
15.79Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
15.79Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
15.79Single7PYRPSB-21157PYR-A2A-PSB-2115
15.79Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
15.79Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
15.79Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
15.79Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
15.79Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
15.79Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
15.79Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
15.79Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
15.79Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
15.79Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
15.79Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
15.79Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
15.79Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
15.62Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
15.62Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
15.62Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
15.62Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
15.38Single3OE0CVX153OE0-CXCR4-CVX15
15.38Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
15.38Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
15.38Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
15.38Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
15.38Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.38Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
15.38Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
15.38Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.38Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
15.38Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.00Single4NTJAZD12834NTJ-P2Y12-AZD1283
15.00Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
15.00Single5IUAQ274563485IUA-A2A-Q27456348-Na
15.00Single5N2RPSB-365N2R-A2A-PSB-36-Na
15.00Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
15.00Single6LUQHaloperidol6LUQ-D2-Haloperidol
15.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
15.00Single6S0QZM-2413856S0Q-A2A-ZM-241385
15.00Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
15.00Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
15.00Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
15.00Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
15.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
15.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
15.00Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
15.00Single7SINNPS-21437SIN-CaS-NPS-2143
15.00Single7SINNPS-21437SIN-CaS-NPS-2143
15.00Single7W41PD1762527W41-BB2-PD176252
15.00Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
15.00Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.00Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
15.00Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
15.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
15.00Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
15.00Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
15.00Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
15.00Consensusadenosine_offOrthosteric Liganda1_off a2_off
15.00Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
15.00Consensusbombesin_offOrthosteric Ligandbb2_off
14.81Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
14.81Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
14.81Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
14.81Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
14.81Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
14.81Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
14.81Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
14.81Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
14.81Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.81Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
14.81Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
14.81Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
14.81Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
14.81Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
14.71Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
14.71Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
14.29Single5TZRMK86665TZR-FFA1-MK8666
14.29Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
14.29Single6OS1TRV0266OS1-AT1-TRV026
14.29Single7B6WCyclazosin7B6W-α1b-Cyclazosin
14.29Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
14.29Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
14.29Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
14.29Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
14.29Single7PX4PSB-21137PX4-A2A-PSB-2113
14.29Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
14.29Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
14.29Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
14.29Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
14.29Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
14.29Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
14.29Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
14.29Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
14.29Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
14.29Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
14.29Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
14.29Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
14.29Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
14.29Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
14.29Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
14.29Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
14.29Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
14.29Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
14.29Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
14.29Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
14.29Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
14.29Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
13.79Single6FJ3PTH6FJ3-PTH1-PTH
13.79Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
13.79Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
13.79Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
13.79Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
13.79Single7SK3CXCL127SK3-ACKR3-CXCL12
13.79Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
13.79Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
13.79Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
13.79Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
13.64Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
13.64Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
13.64Single6IIURamatroban6IIU-TP-Ramatroban
13.64Single6OS2TRV0266OS2-AT1-TRV026
13.64Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
13.64Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.64Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
13.64Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
13.64Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
13.64Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
13.64Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
13.64Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
13.64Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
13.64Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
13.64Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
13.64Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.64Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.64Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.33Single3OE8IT1t3OE8-CXCR4-IT1t
13.33Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
13.33Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
13.33Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
13.33Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
13.33Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
13.33Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
13.33Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
13.33Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
13.33Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
13.33Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
13.33Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
13.33Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
13.33Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
13.33Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
13.16Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
13.04Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
13.04Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
13.04Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
13.04Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
13.04Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
13.04Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
13.04Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
13.04Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
13.04Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
13.04Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
13.04Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
13.04Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
13.04Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
13.04Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
13.04Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
12.90Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
12.90Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
12.90Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
12.90Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
12.82Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
12.50Single3OE6IT1t3OE6-CXCR4-IT1t
12.50Single3UZAGTPL92363UZA-A2A-GTPL9236
12.50Single5EE7MK08935EE7-Glucagon-MK0893
12.50Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
12.50Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
12.50Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
12.50Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
12.50Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
12.50Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
12.50Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
12.50Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
12.50Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
12.50Single7WC5Psilocin7WC5-5-HT2A-Psilocin
12.50Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
12.50Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
12.50Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
12.50Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
12.50Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
12.50Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8QJ2pN1628QJ2-MC4-pN162-Gs
12.50Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
12.50Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
12.50Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
12.50Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
12.50Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
12.50Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
12.50Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
12.50Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Consensusgi_sensoryOrthosteric Ligandgi_opsins
12.50Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
12.50Consensuskisspeptin_onOrthosteric Ligandkiss1_on
12.50Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.12Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
12.12Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
12.12Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
12.12Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
12.12Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
12.00Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
12.00Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
12.00Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
12.00Single8XWNCXCL88XWN-CXCR2-CXCL8
12.00Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
12.00Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
12.00Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
12.00Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
12.00Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
12.00Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Consensussomatostatin_offOrthosteric Ligandsst2_off
11.76Single3OE9IT1t3OE9-CXCR4-IT1t
11.76Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
11.76Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
11.76Single6LI0C176LI0-GPR52-C17
11.76Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
11.76Single6TP4ACT-4622066TP4-OX1-ACT-462206
11.76Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
11.76Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
11.76Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
11.76Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
11.76Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
11.76Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
11.76Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.76Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
11.76Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
11.76Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
11.76Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
11.76Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
11.76Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
11.76Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
11.54Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
11.54Single7XNACYN1548067XNA-SST2-CYN154806
11.54Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
11.54Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
11.54Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
11.54Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
11.54Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
11.54Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
11.54Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
11.43Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
11.43Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
11.43Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
11.11Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
11.11Single3ODUIT1t3ODU-CXCR4-IT1t
11.11Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
11.11Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
11.11Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
11.11Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
11.11Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
11.11Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
11.11Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
11.11Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
11.11Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
11.11Single7F8ULintitript7F8U-CCKA-Lintitript
11.11Single7F8YDevazepide7F8Y-CCKA-Devazepide
11.11Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
11.11Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
11.11Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
11.11Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
11.11Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
11.11Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
11.11Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
11.11Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
11.11Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
11.11Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
11.11Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
11.11Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
11.11Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
11.11Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
11.11Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
11.11Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
11.11Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
11.11Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
11.11Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
11.11Single9BA0A1AKN9BA0-CB1-A1AKN
11.11Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
11.11Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
11.11Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
11.11Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
11.11Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
11.11Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
11.11Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.11Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.11Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.71Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
10.71Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
10.71Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
10.71Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
10.71Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
10.71Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
10.53Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
10.53Single5IU7Q274563465IU7-A2A-Q27456346-Na
10.53Single5IUBQ274563445IUB-A2A-Q27456344-Na
10.53Single5JTBZM-2413855JTB-A2A-ZM-241385
10.53Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
10.53Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
10.53Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
10.53Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
10.53Single6MH8ZM-2413856MH8-A2A-ZM-241385
10.53Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
10.53Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
10.53Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
10.53Single7AROLUF58337ARO-A2A-LUF5833-Na
10.53Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
10.53Single7VODCariprazine7VOD-5-HT2A-Cariprazine
10.53Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.53Single8IYXYL-3658IYX-GPR34-YL-365
10.53Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
10.53Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
10.53Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
10.53Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
10.53Consensusa2_offOrthosteric Liganda2a_off
10.53Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
10.53Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.34Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
10.34Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
10.34Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
10.34Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
10.34Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
10.00Single3EMLZM-2413853EML-A2A-ZM-241385
10.00Single4QIMANTA XV4QIM-SMO-ANTA XV
10.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
10.00Single5UENDU1725UEN-A1-DU172
10.00Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
10.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
10.00Single6D27CAY104716D27-DP2-CAY10471
10.00Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
10.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
10.00Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
10.00Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
10.00Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
10.00Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
10.00Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
10.00Single6S0LZM-2413856S0L-A2A-ZM-241385
10.00Single7F83PF-051904577F83-Ghrelin-PF-05190457
10.00Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
10.00Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
10.00Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
10.00Single8CU6LJ-45178CU6-A2A-LJ-4517
10.00Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.00Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
10.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
10.00Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
10.00Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
10.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
10.00Single9B9ZA1AKO9B9Z-CB1-A1AKO
10.00Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
10.00Consensuscck_offOrthosteric Ligandccka_off
10.00Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
10.00Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
10.00Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.00Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
10.00Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
10.00Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
10.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
10.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
9.68Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
9.68Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
9.68Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
9.52Single4JKVTaladegib4JKV-SMO-Taladegib
9.52Single5N2SPSB365N2S-A1-PSB36
9.52Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
9.52Single8GNEKW-63568GNE-A2A-KW-6356-Na
9.52Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
9.52Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
9.52Single8QOTNanobody-E8QOT-μ-Nanobody-E
9.52Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
9.52Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
9.38Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
9.38Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
9.38Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
9.38Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
9.09Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
9.09Single5V56TC1145V56-SMO-TC114
9.09Single5V57TC1145V57-SMO-TC114
9.09Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
9.09Single7F1TMIP-1a7F1T-CCR5-MIP-1a
9.09Single7R0CAVP7R0C-V2-AVP-Arrestin2
9.09Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
9.09Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
9.09Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
9.09Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
9.09Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
9.09Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
9.09Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
9.09Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
9.09Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
9.09Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
9.09Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
9.09Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
9.09Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
8.70Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
8.70Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
8.70Single4PY02MeSATP4PY0-P2Y12-2MeSATP
8.70Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
8.70Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.70Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
8.70Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
8.70Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
8.70Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
8.70Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
8.70Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
8.70Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
8.70Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
8.70Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
8.70Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
8.33Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
8.33Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
8.33Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
8.33Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
8.33Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
8.33Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
8.33Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
8.33Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.11Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
8.00Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
8.00Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
8.00Single8IEIA1LYA8IEI-GPR156-A1LYA
8.00Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
8.00Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
7.69Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
7.69Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
7.69Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
7.69Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.69Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
7.69Single8IEBA1LYA8IEB-GPR156-A1LYA
7.69Single8IEIA1LYA8IEI-GPR156-A1LYA
7.69Single8IEPA1LYA8IEP-GPR156-A1LYA
7.69Single8IEPA1LYA8IEP-GPR156-A1LYA
7.69Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
7.69Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
7.69Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
7.69Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
7.69Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.69Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.41Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
7.41Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
7.41Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
7.41Single7SHEPI; PE7SHE-GPR158-PI; PE
7.41Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8IEBA1LYA8IEB-GPR156-A1LYA
7.41Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
7.14Single5MZPCaffeine5MZP-A2A-Caffeine-Na
7.14Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
7.14Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
7.14Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
7.14Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
6.90Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
6.90Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
6.90Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
6.67Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
6.67Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
6.67Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
6.67Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
6.67Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
6.67Single7WC4Serotonin7WC4-5-HT2A-Serotonin
6.67Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
6.67Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
6.67Single8PWNTheophylline8PWN-A2A-Theophylline
6.67Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
6.67Single9GE2Cholesterol9GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
6.45Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
6.45Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
6.45Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
6.25Single3RFMCaffeine3RFM-A2A-Caffeine
6.25Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
6.25Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
6.25Single8A2OTheophylline8A2O-A2A-Theophylline-Na
6.25Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
6.06Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
5.88Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.88Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
5.88Single7F61Cholesterol7F61-H3-PF-03654746-Cholesterol
5.88Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
5.88Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
5.88Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
5.88Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.88Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single4O9RCyclopamine4O9R-SMO-Cyclopamine
5.56Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
5.56Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
5.56Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
5.56Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
5.56Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.56Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
5.56Single9B9Y7DY9B9Y-CB1-7DY
5.56Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
5.56Consensusgq_nucleotideOrthosteric Ligandgq_p2y
5.56Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
5.41Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
5.26Single4BWBNeurotensin4BWB-NTS1-Neurotensin
5.26Single4K5YCP-3763954K5Y-CRF1-CP-376395
5.26Single4QINSAG1.54QIN-SMO-SAG1.5
5.26Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
5.26Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
5.26Single5U09Taranabant5U09-CB1-Taranabant
5.26Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
5.26Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
5.26Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
5.26Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
5.26Single7BR3Elagolix7BR3-GnRH1-Elagolix
5.26Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
5.26Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.26Single8G94CD698G94-S1P1-CD69-Gi1/β1/γ2
5.26Single8GNGIstradefylline8GNG-A2A-Istradefylline
5.26Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
5.26Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
5.26Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
5.26Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
5.26Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
5.26Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
5.00Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
5.00Single5UVIZM-2413855UVI-A2A-ZM-241385
5.00Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
5.00Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
5.00Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
5.00Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
5.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
5.00Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
5.00Consensusgrh_offOrthosteric Ligandgnrh1_off
5.00Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
4.76Single4Z9GCP-3763954Z9G-CRF1-CP-376395
4.76Single5T04Neurotensin5T04-NTS1-Neurotensin
4.76Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
4.76Single8GTIBMK-C2058GTI-CRF1-BMK-C205
4.76Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
4.76Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
4.55Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
4.55Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
4.55Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
4.55Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8GTGBMK-I1528GTG-CRF1-BMK-I152
4.55Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
4.55Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
4.55Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
4.55Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
4.35Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
4.35Single4BV0Neurotensin4BV0-NTS1-Neurotensin
4.35Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
4.35Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
4.35Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
4.35Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
4.35Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
4.35Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
4.35Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Consensusneurotensin_onOrthosteric Ligandnts1_on
4.35Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
4.17Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
4.17Single4XEENeurotensin4XEE-NTS1-Neurotensin
4.17Single4XESNeurotensin4XES-NTS1-Neurotensin
4.17Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
4.17Single6YVRNTS8-136YVR-NTS1-NTS8-13
4.17Single7SHEPI; PE7SHE-GPR158-PI; PE
4.17Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
4.17Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.17Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.17Single8GTMBMK-C2038GTM-CRF1-BMK-C203
4.17Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
4.17Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
4.17Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
4.17Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
4.17Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
4.17Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
4.17Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
4.00Single4BUONeurotensin4BUO-NTS1-Neurotensin
4.00Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
4.00Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
4.00Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
4.00Single8XVUCXCL28XVU-CXCR2-CXCL2
4.00Single8XWFCXCL38XWF-CXCR2-CXCL3
4.00Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
3.85Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
3.85Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
3.85Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
3.85Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
3.85Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
3.70Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
3.70Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.57Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
3.57Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
2.94Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2

Consensus Members
Id Members
7VKT 7VKT-BLT1-LTB4-Gi1/β1/γ2
Net Summary
Imin 2.51
Number of Linked Nodes 835
Number of Links 967
Number of Hubs 142
Number of Links mediated by Hubs 543
Number of Communities 30
Number of Nodes involved in Communities 194
Number of Links involved in Communities 252
Path Summary
Number Of Nodes in MetaPath 108
Number Of Links MetaPath 107
Number of Shortest Paths 4975221
Length Of Smallest Path 3
Average Path Length 54.2437
Length of Longest Path 88
Minimum Path Strength 1.16
Average Path Strength 5.36919
Maximum Path Strength 21.84
Minimum Path Correlation 0.7
Average Path Correlation 0.99411
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.63934
Average % Of Corr. Nodes 28.3448
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 39.4003
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following differences:
Id1st Network2nd Network
blt1_off_on_gpblt1_on_gpblt1_off
This network is also present in following consensuses:
IdComponents
blt_on_gpblt1_on_gp



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