Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1g.h1x1 3.53542402
2g.l1x4 4.48892548
3g.h2x11 8.139484126
4g.ctx3 5.76403699
5g.ctx6 3.039596
6g.ctx14 5.487294109
7g.ctx15 5.903654109
8g.ctx16 4.565218108
91x32 2.55625404
101x35 7.04025525
111x39 6.47975526
121x43 3.12719425
131x50 5.46656439
141x57 3.42094408
151x60 1.93177406
162x42 4.68333408
172x46 4.18687439
182x50 4.96333639
192x57 4.00656426
202x64 3.47375503
213x34 3.68635405
223x35 3.03896407
233x37 3.64167406
243x42 4.90583438
253x49 5.009694179
263x50 5.47375539
273x53 5.750424178
28I2x51 4.08177476
29I2x53 4.959584177
304x42 2.75646407
314x50 3.93458539
32E2 10.84421823
335x39 5.77781426
345x40 3.96073425
355x51 2.7126406
365x58 3.45406839
376x48 5.45875738
386x51 3.67967526
396x55 3.88229425
406x59 2.95933524
41E3 3.14012723
427x38 4.47292525
437x39 3.99427425
447x42 4.27302427
457x49 5.85698439
468x48 2.89188404
478x50 3.62633509
488x54 2.29219407
49Lig 5.823081520
50G.S1.06 5.08656469
51G.S1.07 4.6499419
52G.S2.02 1.97094406
53G.S2.03 4.33292519
54G.S2.05 4.83281413
55G.S2.06 4.94817508
56G.S2.08 4.99475575
57G.s2s3.01 5.76323475
58G.S3.03 5.1069777
59G.S3.04 8.73458417
60G.S3.06 7.04115416
61G.H2.06 5.0299419
62G.H2.07 4.27232719
63G.h2s4.01 6.37275519
64G.S4.02 4.31094417
65G.S4.03 3.56802468
66G.S4.04 5.24692519
67G.s4h3.02 3.738444119
68G.s4h3.04 5.756046118
69G.s4h3.05 4.675424119
70G.H3.01 4.87885409
71G.H3.09 6.385419
72G.H3.13 4.57479416
73G.H3.17 6.41903615
74G.H3.18 5.49875419
75G.S5.02 3.11708416
76G.S5.03 4.06792468
77G.S5.05 3.44833869
78G.HG.14 2.53104405
79G.hgh4.02 4.39583408
80G.hgh4.05 7.066506
81G.H4.03 3.55729404
82G.H4.08 2.44802403
83G.H4.10 7.57042406
84G.H4.15 5.38135408
85G.S6.02 5.88933508
86G.S6.05 3.91813605
87G.s6h5.02 2.47875407
88G.H5.03 4.47692568
89G.H5.08 4.72653678
90G.H5.13 4.1795507
91G.H5.20 3.7675408
92G.H5.23 4.06417404
93G.H5.26 3.70725507
94b.1x1 2.71792404
95b.1x7 2.81708408
96b.1x11 2.98938408
97b.1x15 3.49531447
98b.1x19 5.2475446
99b.h2x1 3.75469405
100b.lhb1x3 2.29192502
101b.lhb1x6 3.54183593
102b.b1x4 4.213754107
103b.l1x3 7.98659
104b.l1x6 8.34948419
105b.b2x1 7.31967518
106b.b2x5 6.22076657
107b.b3x3 3.33854408
108b.l3x2 5.35983559
109b.b4x3 4.003754147
110b.b4x5 4.085944187
111b.b4x6 8.2878759
112b.b5x2 5.27417407
113b.b5x3 5.64185759
114b.b5x7 5.07052407
115b.l5x1 4.029335148
116b.l5x5 6.50137719
117b.b6x5 3.84217506
118b.l6x5 5.433334154
119b.b7x1 5.123335154
120b.b8x4 5.33854406
121b.b9x3 3.90948406
122b.l9x3 7.20174619
123b.l9x6 4.73906818
124b.b10x5 4.86927409
125b.l10x1 3.60342503
126b.b11x4 5.30135419
127b.l11x2 7.69396419
128b.b12x6 9.06708618
129b.b13x7 7.434587
130b.l13x3 7.63375689
131b.l13x7 4.16975589
132b.b15x2 6.3001446
133b.l15x2 5.33392589
134b.b16x4 10.3795486
135b.b16x5 4.11448405
136b.b16x6 7.46244788
137b.b17x7 8.38771448
138b.l17x3 8.57264649
139b.l17x6 5.68775519
140b.b18x3 4.45698448
141b.l18x1 6.338517126
142b.l18x2 5.990944127
143b.b19x2 6.38785646
144b.b19x4 6.01396448
145b.l19x2 6.92125409
146b.b20x2 5.26698446
147b.b20x4 9.92683548
148b.b20x6 6.84028646
149b.b20x7 4.04688409
150b.l20x2 6.9425409
151b.b21x1 9.16865447
152b.b21x2 3.67406
153b.b21x5 3.8475404
154b.b21x7 5.67438605
155b.b22x5 5.592085127
156b.l22x5 7.00283599
157b.b23x6 6.715076167
158b.l23x1 7.42427416
159b.b24x4 6.344584166
160b.b24x6 7.161874168
161b.l24x3 4.02677405
162b.l25x3 10.84764139
163b.l25x6 10.5462418
164b.b26x3 3.38677406
165b.l27x1 8.99863719
166b.l27x2 8.197084139
167b.b28x2 5.84375404
168b.b28x4 8.109484136
169b.b28x6 8.39555139
170G.HN.29 0.302188400
171E1 1.975420
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1g.h1x10 g.h1x13 10.10732.15333NoNo091
2b.b17x3 g.h1x10 10.92325.02208NoNo059
3b.l13x3 b.l13x7 11.27745.3625YesYes899
4b.b11x5 b.l13x7 19.4775.38458NoYes069
5b.b11x5 b.b14x3 19.99555.88042NoNo065
6b.b10x2 b.b14x3 20.2565.61958NoNo065
7b.b10x2 b.b10x4 20.51663.77125NoNo066
8b.b10x4 b.b2x4 26.96068.88833NoNo066
9b.b2x4 b.b6x5 27.21753.04292NoYes066
10b.b3x1 b.b6x5 30.2023.90667NoYes056
11b.b3x1 b.l2x3 30.43314.80542NoNo058
12b.l2x3 b.l2x5 30.66572.975NoNo085
13b.l2x5 b.l4x2 31.086420.6208NoNo054
14b.l4x2 g.ctx16 27.246.0175NoYes1048
15b.l4x1 g.ctx16 31.11234.78792NoYes058
16b.b2x5 b.l4x1 31.3085.35333YesNo075
17b.b2x3 b.b2x5 38.7944.41292NoYes567
18b.b26x2 b.b2x3 59.77315.265NoNo076
19b.b26x1 b.b26x2 60.15443.36833NoNo097
20b.b26x1 b.l27x1 60.34534.88958NoYes099
21b.b2x1 b.l27x1 27.0468.23875YesYes189
22b.b2x1 b.l3x1 27.849713.0121YesNo189
23b.l3x1 b.l5x5 28.21874.70042NoYes199
24G.h2s4.01 b.l5x5 17.001511.2342YesYes199
25G.H2.07 G.h2s4.01 13.99373.50833YesYes199
26G.H2.05 G.H2.07 43.3173.28833NoYes079
27G.H2.05 b.l17x6 42.80693.965NoYes079
28b.l17x5 b.l17x6 44.10132.88458NoYes069
29b.l17x5 b.l19x2 43.83714.04958NoYes069
30b.b20x2 b.l19x2 36.70068.97333YesYes069
31b.b20x2 b.b20x4 29.83624.14833YesYes468
32b.b20x4 b.b20x6 29.03774.76667YesYes486
33b.b17x7 b.b20x6 21.654912.6379YesYes486
34b.b17x7 b.b21x1 19.49344.18208YesYes487
35b.1x14 b.1x15 14.12633.14417NoYes047
36b.1x11 b.1x14 13.5382.88167YesNo084
37b.l5x5 b.l7x2 13.66425.17167YesNo199
38G.H2.07 b.l7x2 13.95733.51167YesNo199
39b.1x19 b.b21x1 10.57288.18833YesYes467
40b.l26x5 g.ctx4 11.01595.45042NoNo057
41g.ctx3 g.ctx4 10.78894.22625YesNo097
42b.b21x5 b.b21x7 10.14576.83458YesYes045
433x36 Lig 47.51545.36667NoYes060
443x36 6x48 47.36823.13875NoYes068
456x48 7x45 56.89727.36208YesNo389
467x45 7x49 57.6898.23625NoYes399
473x43 7x49 61.9884.95542NoYes389
483x43 7x53 71.61734.73917NoNo389
493x50 7x53 71.81586.98792YesNo399
503x50 G.H5.25 69.95657.99583YesNo097
51G.H5.20 G.H5.25 70.15364.4975YesNo087
52G.H5.20 G.H5.26 71.3574.26YesYes087
53G.H5.17 G.H5.26 77.89744.72833NoYes057
54G.H5.13 G.H5.17 78.70893.89208YesNo075
55G.H5.13 G.S6.02 82.86828.2375YesYes078
56G.H5.10 G.S6.02 84.24768.87708NoYes078
57G.H5.10 G.S5.03 42.97196.0125NoYes078
58G.S5.03 G.S5.05 41.61983.40042YesYes689
59G.S5.05 G.s6h5.01 98.8355.35042YesNo699
60G.S5.07 G.s6h5.01 1004.32583NoNo099
61G.S5.07 G.s5hg.01 99.97152.97292NoNo099
62G.s4h3.02 G.s5hg.01 99.09023.9525YesNo1199
63G.HG.07 G.s4h3.02 99.87183.1875NoYes1199
64G.HG.07 G.s4h3.04 98.74229.94125NoYes1198
65G.HG.04 G.s4h3.04 98.9254.85333NoYes088
66G.HG.04 G.s4h3.01 98.84857.52792NoNo086
67G.S5.06 G.s4h3.01 98.82246.89083NoNo096
68G.S5.04 G.S5.06 97.89383.57542NoNo099
69G.H4.15 G.S5.04 97.90124.97417YesNo089
70G.H3.09 G.H4.15 97.47194.95625YesYes098
71G.H3.09 G.S4.04 96.995211.1629YesYes199
72G.S1.07 G.S4.04 64.41674.67125YesYes199
73G.S1.07 G.S4.02 60.5253.32917YesYes197
74G.H3.18 G.S4.02 60.53347.59208YesYes197
75G.H3.15 G.H3.18 60.35875.58583NoYes089
76G.H3.15 G.H3.17 60.24485.25375NoYes085
77G.H3.17 b.l27x1 39.95153.3575YesYes159
78G.H5.10 G.S6.04 41.48692.94083NoNo079
79G.S5.05 G.S6.04 41.51542.9225YesNo699
803x53 G.H5.19 12.82513.985YesNo087
81G.H5.15 G.H5.19 13.02813.08583NoNo087
82G.H5.15 I2x51 13.24423.61875NoYes086
83G.S1.04 G.S3.03 16.15183.51333NoYes077
84G.S1.04 G.S4.03 15.64623.09208NoYes078
85G.S4.03 G.S5.05 16.27563.58YesYes689
86b.b22x1 b.b22x2 10.24613.33333NoNo088
87b.b22x1 b.l25x6 10.1862.80208NoYes188
88E2 Lig 15.52228.52583YesYes230
89b.b4x2 b.b5x8 10.53193.62417NoNo085
90b.b5x7 b.b5x8 10.29633.10667YesNo075
91b.b4x2 b.l3x2 12.17876.34NoYes089
92G.H2.07 b.l9x6 14.33045.42625YesYes198
93G.H2.04 G.H2.07 32.51863.5NoYes099
94G.H2.04 G.H3.08 32.47874.08375NoNo099
95G.H3.08 G.S4.04 32.634.94958NoYes099
96b.l1x3 b.l3x2 13.09153.2025YesYes599
97b.b4x6 b.l1x3 13.55113.96792YesYes599
98b.l11x1 b.l9x6 13.01245.61333NoYes198
99b.b11x6 b.l11x1 13.73652.93917NoNo199
100b.b11x6 b.l9x3 12.144915.1687NoYes199
101b.b19x4 b.l17x3 10.39078.95458YesYes489
102b.l23x1 b.l25x6 19.234619.0558YesYes168
103b.l21x7 b.l23x1 19.06264.01708NoYes056
104b.l21x7 b.l23x2 18.82166.09458NoNo058
105b.b23x6 b.l23x2 18.09983.7375YesNo078
106b.b21x7 b.b24x6 14.401711.6979YesYes058
107b.b23x6 b.b24x6 15.18547.19625YesYes1678
108b.b3x2 b.b4x6 21.14994.88917NoYes559
109b.b2x3 b.b3x2 20.79542.885NoNo565
110G.H3.17 b.l25x6 19.68075.45792YesYes158
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
1x322x643.663330YesYes4321
1x351x3911.342YesYes5622
1x352x644.724172YesYes5321
1x357x3511.992YesNo5322
1x357x384.257082YesYes5521
1x392x575.276672YesYes6622
1x397x428.428752YesYes6721
2x577x423.1752YesYes6721
3x22E215.73422NoYes3321
3x25E22.963332NoYes9321
3x26E24.919582NoYes5321
3x29E2x523.597082NoNo4411
3x33Lig8.423330NoYes4010
3x366x483.138750NoYes6812
3x36Lig5.366670NoYes6010
3x373x413.137080YesNo6412
3x375x433.77250YesNo6512
3x375x4614.196670YesNo6812
4x605x398.190420NoYes4612
5x39E25.0952YesYes6321
E2E254.70332YesYes3311
5x36E29.082NoYes5321
E2E2x5110.50542YesNo3412
E2E2x528.783332YesNo3411
E2x52Lig18.65082NoYes4010
E2Lig8.525832YesYes3010
5x406x554.824172YesYes5511
5x40Lig3.922082YesYes5010
6x487x413.276673YesNo8722
6x517x373.41252YesNo6512
6x517x383.084172YesYes6511
6x517x415.042082YesNo6712
6x51Lig3.698752YesYes6010
6x55Lig5.133752YesYes5010
7x38Lig7.710832YesYes5010
7x42Lig3.172922YesYes7010
6x516x523.160832YesNo6712
7x347x384.343332NoYes4511
2x64Lig2.894580YesYes3010
7x34Lig5.317922NoYes4010
7x357x382.969172NoYes3521
3x37Lig3.460420YesYes6010
2x533x362.896670NoNo8621
2x602x642.783330NoYes7321
2x632x643.303330NoYes3321
E1x49E23.448330NoYes0321
3x29Lig2.782NoYes4010
4x64E25.9650NoYes0321
5x365x403.42NoYes5521
5x406x593.696672YesYes5412
6x556x592.883332YesYes5412
6x586x625.2652NoNo4021
6x587x3411.2152NoNo4421
6x62Lig4.240NoYes0010
4x60Lig4.048330NoYes4010
5x376x552.687920NoYes3521
5x33E22.363330NoYes0321
1x427x422.315420NoYes7721
E1E22.118332YesYes0321
3x21E22.104170NoYes6321
4x63E22.07252NoYes5321
6x63E21.870NoYes0321
5x30E20.240NoYes0321

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
80.00Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
77.78Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
68.75Consensusa3_on_gpOrthosteric Liganda3a_on_gp
68.75Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
68.75Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
66.67Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
66.67Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
62.50Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
62.50Consensusa3_onOrthosteric Liganda3a_on
62.50Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
58.82Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
58.82Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
56.25Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
55.56Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
55.56Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
55.56Consensusa2_onOrthosteric Liganda2b_on
55.56Consensusa2_on_gpOrthosteric Liganda2b_on_gp
55.56Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
55.56Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
55.56Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
55.56Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
54.55Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
53.33Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
52.63Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
52.38Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
52.38Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
52.38Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
52.17Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
50.00Single3PWHZM-2413853PWH-A2A-ZM-241385
50.00Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
50.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
50.00Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
50.00Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
50.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
50.00Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
50.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
50.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
50.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
50.00Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
47.62Single3NY9ICI118-5513NY9-β2-ICI118-551
47.62Single4UG2CGS216804UG2-A2A-CGS21680
47.37Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
47.37Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
47.37Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
47.37Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
47.37Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
47.37Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
47.37Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
47.37Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
47.37Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
47.06Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
47.06Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
45.83Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
45.83Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
45.45Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
45.45Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
45.45Consensuslpl_onOrthosteric Ligands1p_on lpa_on
45.45Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
45.45Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
45.00Single4RWADIPP-NH24RWA-δ-DIPP-NH2
45.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
45.00Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
45.00Single7YITNalfurafine7YIT-κ-Nalfurafine
45.00Single8JWY2-1188JWY-A2A-2-118
45.00Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
45.00Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
45.00Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
45.00Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
45.00Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
45.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
45.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
44.44Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
44.44Single5UIGCmpd-15UIG-A2A-Cmpd-1
44.44Single6PS1Timolol6PS1-β2-Timolol
44.44Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
44.44Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
44.44Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
44.44Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
44.44Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
44.44Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
44.44Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
44.44Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
44.44Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
44.44Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
44.44Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
44.44Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
44.44Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
44.00Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
43.75Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
43.75Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
43.75Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
43.48Single3QAKUK-4320973QAK-A2A-UK-432097
43.48Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
43.48Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
43.48Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
42.86Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
42.86Single7EZCUKA7EZC-A2A-UKA
42.86Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
42.86Single7UM4AS26747237UM4-5-HT5A-AS2674723
42.86Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.86Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
42.31Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
42.11Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
42.11Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
42.11Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
42.11Single7C61Ergotamine7C61-5-HT1B-Ergotamine
42.11Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
42.11Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
42.11Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
42.11Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.11Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
42.11Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
42.11Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
42.11Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
42.11Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
42.11Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
42.11Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
42.11Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
42.11Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
42.11Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
42.11Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
41.67Single5WF5UK-4320975WF5-A2A-UK-432097
41.67Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
41.18Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
41.18Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
41.18Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
41.18Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
41.18Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
41.18Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
41.18Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
41.18Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
41.18Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
41.18Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
41.18Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
41.18Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
41.18Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
41.18Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
41.18Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
41.18Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
41.18Consensusalpha2_offOrthosteric Ligandalpha2c_off
40.91Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
40.91Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
40.91Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
40.91Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
40.91Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
40.91Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
40.91Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
40.91Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
40.91Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
40.91Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
40.74Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
40.00Single2YDVNECA2YDV-A2A-NECA
40.00Single3RFMCaffeine3RFM-A2A-Caffeine
40.00Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
40.00Single4UHRCGS216804UHR-A2A-CGS21680
40.00Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
40.00Single5G53NECA5G53-A2A-NECA-Gs
40.00Single6H7JIsoprenaline6H7J-β1-Isoprenaline
40.00Single6J21Aprepitant6J21-NK1-Aprepitant
40.00Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
40.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
40.00Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
40.00Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
40.00Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
40.00Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
40.00Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
40.00Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
40.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
40.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
40.00Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
40.00Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
40.00Single8E0GBU728E0G-μ-BU72
40.00Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
40.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
40.00Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
40.00Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
40.00Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
40.00Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
40.00Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
40.00Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
40.00Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
40.00Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
40.00Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
40.00Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
40.00Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
40.00Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
40.00Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
40.00Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
40.00Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
39.13Single4IARErgotamine4IAR-5-HT1B-Ergotamine
39.13Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
39.13Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
39.13Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
39.13Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
39.13Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
39.13Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
39.13Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
39.13Single8WDTphotoNECA8WDT-A2A-photoNECA
39.13Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
39.13Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
38.89Single2YDOAdenosine2YDO-A2A-Adenosine
38.89Single3REYXAC3REY-A2A-XAC
38.89Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
38.89Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
38.89Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
38.89Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
38.89Single5IU7Q274563465IU7-A2A-Q27456346-Na
38.89Single5IUBQ274563445IUB-A2A-Q27456344-Na
38.89Single5JTBZM-2413855JTB-A2A-ZM-241385
38.89Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
38.89Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
38.89Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
38.89Single6AQFZM-2413856AQF-A2A-ZM-241385
38.89Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
38.89Single6MH8ZM-2413856MH8-A2A-ZM-241385
38.89Single6PS0S-Carazolol6PS0-β2-S-Carazolol
38.89Single6PS4ICI118-5516PS4-β2-ICI118-551
38.89Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
38.89Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
38.89Single7AROLUF58337ARO-A2A-LUF5833-Na
38.89Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
38.89Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
38.89Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.89Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
38.89Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
38.89Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
38.89Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
38.89Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
38.89Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
38.89Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
38.89Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
38.89Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
38.89Single8K5CAcipimox8K5C-HCA2-Acipimox
38.89Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
38.89Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
38.89Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
38.89Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
38.89Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
38.89Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
38.89Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
38.89Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
38.89Consensusa2_offOrthosteric Liganda2a_off
38.89Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
38.89Consensushca_onOrthosteric Ligandhca2_on
38.89Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
38.46Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
38.46Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
38.46Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
38.46Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
38.46Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
38.46Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
38.46Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
38.46Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
38.46Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
38.10Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
38.10Single3D4STimolol3D4S-β2-Timolol
38.10Single4LDEBI1671074LDE-β2-BI167107
38.10Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
38.10Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
38.10Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
38.10Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
38.10Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
38.10Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
38.10Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
38.10Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
38.10Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
38.10Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
38.10Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
38.10Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
38.10Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
38.10Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
38.10Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
38.10Single8JJ8Formoterol8JJ8-β2-Formoterol
38.10Single8JWZAB9288JWZ-A2A-AB928-Na
38.10Single8XYIVUF106618XYI-CXCR3-VUF10661
38.10Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
38.10Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
38.10Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
38.10Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
38.10Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
38.10Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
38.10Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
38.10Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.50Single3UZAGTPL92363UZA-A2A-GTPL9236
37.50Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
37.50Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
37.50Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
37.50Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
37.50Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
37.50Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
37.50Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
37.50Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
37.50Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
37.04Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
37.04Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
36.84Single2Y04Salbutamol2Y04-β1-Salbutamol
36.84Single3EMLZM-2413853EML-A2A-ZM-241385
36.84Single3NY8ICI118-5513NY8-β2-ICI118-551
36.84Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
36.84Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
36.84Single4EJ4Naltrindole4EJ4-δ-Naltrindole
36.84Single4GBRS-Carazolol4GBR-β2-S-Carazolol
36.84Single5IU8Q274563475IU8-A2A-Q27456347-Na
36.84Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
36.84Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
36.84Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
36.84Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
36.84Single5UENDU1725UEN-A1-DU172
36.84Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
36.84Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
36.84Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
36.84Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
36.84Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
36.84Single6S0LZM-2413856S0L-A2A-ZM-241385
36.84Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
36.84Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
36.84Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
36.84Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
36.84Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
36.84Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
36.84Single7PYRPSB-21157PYR-A2A-PSB-2115
36.84Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
36.84Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
36.84Single7UL4Alvimopan7UL4-μ-Alvimopan
36.84Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
36.84Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
36.84Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
36.84Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
36.84Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
36.84Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
36.84Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
36.84Single8CU6LJ-45178CU6-A2A-LJ-4517
36.84Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
36.84Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
36.84Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
36.84Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
36.84Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
36.84Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
36.84Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
36.84Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
36.84Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
36.84Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
36.84Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
36.84Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
36.84Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
36.84Single8JJOAlprenolol8JJO-β2-Alprenolol
36.84Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
36.84Single8RLNLUF58348RLN-A2A-LUF5834
36.84Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
36.84Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
36.84Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
36.84Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
36.84Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
36.84Single9CHXS-Carazolol9CHX-β2-S-Carazolol
36.84Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
36.84Single9IYAONO-97105319IYA-GPR55-ONO-9710531
36.84Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
36.84Consensus5ht5_onOrthosteric Ligand5ht5a_on
36.84Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
36.84Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
36.84Consensusalpha2_onOrthosteric Ligandalpha2b_on
36.84Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
36.84Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
36.84Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
36.84Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
36.84Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
36.84Consensusdopamine_offOrthosteric Ligandd2_off d3_off
36.84Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
36.84Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
36.84Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
36.84Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
36.84Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
36.84Consensushca_on_gpOrthosteric Ligandhca2_on_gp
36.36Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
36.36Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
36.36Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
36.36Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
36.36Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
36.36Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
36.36Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
36.36Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
36.36Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
36.36Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
36.36Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
36.36Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.36Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
36.36Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
36.36Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
36.36Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
36.36Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.36Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
36.36Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
36.36Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
36.36Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
36.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
36.00Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
36.00Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
36.00Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
36.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
36.00Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
36.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
36.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
35.71Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
35.71Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
35.71Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
35.71Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
35.71Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
35.71Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
35.71Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
35.48Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
35.29Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
35.29Single7SRQLSD7SRQ-5-HT2B-LSD
35.29Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
35.29Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
35.29Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
35.29Single8K5BNiacin8K5B-HCA2-Niacin
35.29Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
35.00Single2RH1S-Carazolol2RH1-β2-S-Carazolol
35.00Single2Y03Isoprenaline2Y03-β1-Isoprenaline
35.00Single2YCWS-Carazolol2YCW-β1-S-Carazolol
35.00Single4NTJAZD12834NTJ-P2Y12-AZD1283
35.00Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
35.00Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
35.00Single5C1MBU725C1M-μ-BU72
35.00Single5D6LS-Carazolol5D6L-β2-S-Carazolol
35.00Single5IUAQ274563485IUA-A2A-Q27456348-Na
35.00Single5JQHS-Carazolol5JQH-β2-S-Carazolol
35.00Single5N2SPSB365N2S-A1-PSB36
35.00Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
35.00Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
35.00Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
35.00Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
35.00Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
35.00Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
35.00Single6PS6Timolol6PS6-β2-Timolol
35.00Single6S0QZM-2413856S0Q-A2A-ZM-241385
35.00Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
35.00Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
35.00Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
35.00Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
35.00Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
35.00Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
35.00Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
35.00Single7SINNPS-21437SIN-CaS-NPS-2143
35.00Single7SINNPS-21437SIN-CaS-NPS-2143
35.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
35.00Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
35.00Single7WC6LSD7WC6-5-HT2A-LSD
35.00Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
35.00Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
35.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
35.00Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
35.00Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
35.00Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
35.00Single8GNEKW-63568GNE-A2A-KW-6356-Na
35.00Single8S4DCMF-0198S4D-Apelin-CMF-019
35.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
35.00Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
35.00Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
35.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
35.00Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
35.00Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
35.00Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
35.00Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
35.00Consensusadenosine_offOrthosteric Liganda1_off a2_off
35.00Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
35.00Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
35.00Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
35.00Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
35.00Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
35.00Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
35.00Consensusamine_offonOrthosteric Ligandamine_off amine_on
35.00Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
35.00Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
35.00Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
35.00Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
35.00Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
35.00Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
35.00Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
35.00Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
35.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
35.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
35.00Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
35.00Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
35.00Consensustrace-amine_onOrthosteric Ligandta1_on
34.78Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
34.78Single5WF6UK-4320975WF6-A2A-UK-432097
34.78Single5ZTYAM102575ZTY-CB2-AM10257
34.78Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
34.78Single6PT3DPI-2876PT3-δ-DPI-287
34.78Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
34.78Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
34.78Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
34.78Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
34.78Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
34.78Single8QJ2pN1628QJ2-MC4-pN162-Gs
34.78Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
34.78Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
34.78Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
34.78Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
34.62Single6JODAngiotensin II6JOD-AT2-Angiotensin II
34.62Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
34.62Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
34.62Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
34.62Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.62Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.62Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
34.48Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
34.48Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
34.48Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
34.48Consensusbradykinin_onOrthosteric Ligandbk2_on
34.48Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
34.48Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
33.33Single3P0GBI1671073P0G-β2-BI167107
33.33Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
33.33Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
33.33Single5D5AS-Carazolol5D5A-β2-S-Carazolol
33.33Single5D5BS-Carazolol5D5B-β2-S-Carazolol
33.33Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
33.33Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
33.33Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
33.33Single5TZRMK86665TZR-FFA1-MK8666
33.33Single5V54Methiothepin5V54-5-HT1B-Methiothepin
33.33Single5XR8AM8415XR8-CB1-AM841
33.33Single5XRAAM115425XRA-CB1-AM11542
33.33Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
33.33Single6J20Aprepitant6J20-NK1-Aprepitant
33.33Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
33.33Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
33.33Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
33.33Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
33.33Single6TODEMPA6TOD-OX1-EMPA-Na
33.33Single6TQ7SB-3348676TQ7-OX1-SB-334867
33.33Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
33.33Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
33.33Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
33.33Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
33.33Single7F8XNN90567F8X-CCKA-NN9056
33.33Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single7FEECP559407FEE-CB1-CP55940-ZCZ011
33.33Single7PX4PSB-21137PX4-A2A-PSB-2113
33.33Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
33.33Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
33.33Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
33.33Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
33.33Single7TUYGSK682753A7TUY-GPR183-GSK682753A
33.33Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
33.33Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
33.33Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
33.33Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
33.33Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
33.33Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
33.33Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
33.33Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
33.33Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
33.33Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
33.33Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
33.33Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
33.33Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
33.33Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
33.33Single8GNGIstradefylline8GNG-A2A-Istradefylline
33.33Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
33.33Single8IEBA1LYA8IEB-GPR156-A1LYA
33.33Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
33.33Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
33.33Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
33.33Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
33.33Single8IWESpermidine8IWE-TA9-Spermidine
33.33Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
33.33Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
33.33Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
33.33Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
33.33Single8PWNTheophylline8PWN-A2A-Theophylline
33.33Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
33.33Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
33.33Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
33.33Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
33.33Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
33.33Single8WKYPG-9348WKY-MC4-PG-934
33.33Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
33.33Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
33.33Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
33.33Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
33.33Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
33.33Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
33.33Consensus5ht1_offOrthosteric Ligand5ht1b_off
33.33Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
33.33Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
33.33Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
33.33Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
33.33Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
33.33Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
33.33Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
33.33Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
33.33Consensusbombesin_onOrthosteric Ligandbb2_on
33.33Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
33.33Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
33.33Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
33.33Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
33.33Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
33.33Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
33.33Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
33.33Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
33.33Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
33.33Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
33.33Consensuslpa_onOrthosteric Ligandlpa1_on
33.33Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
33.33Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
33.33Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
33.33Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
32.14Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
32.00Single6HLOAprepitant6HLO-NK1-Aprepitant
32.00Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
32.00Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
32.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
32.00Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
32.00Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
32.00Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
32.00Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
32.00Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
31.82Single4AMIBucindolol4AMI-β1-Bucindolol
31.82Single4PY02MeSATP4PY0-P2Y12-2MeSATP
31.82Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
31.82Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
31.82Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
31.82Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
31.82Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
31.82Single6KQICP559406KQI-CB1-CP55940-Org27569
31.82Single6MXTSalmeterol6MXT-β2-Salmeterol
31.82Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
31.82Single6ZG4HTL00099366ZG4-M1-HTL0009936
31.82Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
31.82Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
31.82Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
31.82Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
31.82Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
31.82Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
31.82Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.82Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
31.82Single8JJLOlodaterol8JJL-β2-Olodaterol
31.82Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.82Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
31.82Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
31.82Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.82Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
31.82Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
31.82Consensusalpha1_offOrthosteric Ligandalpha1a_off
31.82Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
31.82Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
31.82Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
31.82Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
31.82Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
31.82Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
31.82Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
31.82Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
31.82Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
31.82Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
31.82Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
31.82Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
31.82Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
31.82Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
31.82Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
31.82Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
31.82Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
31.82Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
31.82Consensuslpa_offOrthosteric Ligandlpa1_off
31.82Consensuslpl_offOrthosteric Ligands1p_off lpa_off
31.82Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
31.82Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
31.82Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
31.82Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
31.58Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
31.58Single4ZJCSB-6740424ZJC-OX1-SB-674042
31.58Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
31.58Single5UVIZM-2413855UVI-A2A-ZM-241385
31.58Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
31.58Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
31.58Single6PS5S-Propranolol6PS5-β2-S-Propranolol
31.58Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
31.58Single6TPGEMPA6TPG-OX2-EMPA
31.58Single6V9SGTPL114036V9S-OX1-GTPL11403
31.58Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
31.58Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
31.58Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
31.58Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
31.58Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
31.58Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
31.58Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
31.58Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.58Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.58Single7T32ZM-2413857T32-A2A-ZM-241385
31.58Single7UL3Famotidine7UL3-H2-Famotidine
31.58Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
31.58Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
31.58Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
31.58Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.58Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.58Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
31.58Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
31.58Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
31.58Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
31.58Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
31.58Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
31.58Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
31.58Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
31.58Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
31.58Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
31.58Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.58Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
31.58Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.58Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.58Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.58Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.58Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
31.58Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
31.58Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
31.58Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
31.58Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
31.58Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single9BJKNaloxone9BJK-μ-Naloxone-NAM
31.58Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
31.58Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
31.58Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
31.58Consensusalpha1_onOrthosteric Ligandalpha1a_on
31.58Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
31.58Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
31.58Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
31.58Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
31.58Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
31.58Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
31.25Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
31.25Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
31.03Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
31.03Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
31.03Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
31.03Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
30.77Single3OE0CVX153OE0-CXCR4-CVX15
30.77Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
30.77Single6PT2KGCHM076PT2-δ-KGCHM07
30.77Single6W25SHU91196W25-MC4-SHU9119-Ca
30.77Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
30.77Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
30.77Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
30.77Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
30.77Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
30.77Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.77Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
30.77Consensusangiotensin_onOrthosteric Ligandat1_on
30.77Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
30.77Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
30.43Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
30.43Single5X93K-87945X93-ETB-K-8794
30.43Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
30.43Single6H7LDobutamine6H7L-β1-Dobutamine
30.43Single6IBLArformoterol6IBL-β1-Arformoterol
30.43Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
30.43Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
30.43Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
30.43Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
30.43Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
30.43Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
30.43Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
30.43Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
30.43Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
30.43Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
30.43Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
30.43Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
30.43Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
30.43Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
30.43Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
30.43Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
30.43Consensuscck_onOrthosteric Ligandccka_on cckb_on
30.43Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
30.43Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
30.43Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
30.43Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
30.43Consensusendothelin_offOrthosteric Ligandetb_off
30.43Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
30.43Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
30.43Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Consensusprostanoid_offOrthosteric Ligandep_off dp_off
30.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
30.00Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
30.00Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
30.00Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
30.00Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
30.00Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
30.00Single4QKX35V4QKX-β2-35V
30.00Single4YAYZD-71554YAY-AT1-ZD-7155
30.00Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
30.00Single6DRXLisuride6DRX-5-HT2B-Lisuride
30.00Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
30.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
30.00Single6H7MSalbutamol6H7M-β1-Salbutamol
30.00Single6IGLIRL16206IGL-ETB-IRL1620
30.00Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
30.00Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
30.00Single6TOTLemborexant6TOT-OX1-Lemborexant
30.00Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single7BU7BI1671077BU7-β1-BI167107
30.00Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
30.00Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
30.00Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
30.00Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
30.00Single7V3ZCP559407V3Z-CB1-CP55940
30.00Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
30.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
30.00Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
30.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
30.00Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
30.00Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
30.00Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
30.00Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
30.00Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
30.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
30.00Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
30.00Single8JXRLSD8JXR-D1-LSD
30.00Single8K5DGSK2560738K5D-HCA2-GSK256073
30.00Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
30.00Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
30.00Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
30.00Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
30.00Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
30.00Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
30.00Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
30.00Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
30.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
30.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
30.00Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
30.00Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
30.00Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
30.00Consensusblt_onOrthosteric Ligandblt1_on
30.00Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
30.00Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
30.00Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
30.00Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
30.00Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
30.00Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
30.00Consensusleukotriene_onOrthosteric Ligandblt_on
30.00Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
30.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
30.00Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
30.00Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
29.63Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
29.63Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
29.63Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
29.63Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
29.63Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
29.63Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
29.63Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
29.63Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
29.63Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
29.63Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
29.63Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
29.63Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
29.41Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
29.41Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
29.41Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.41Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
29.41Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
29.41Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
29.41Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
29.41Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
29.41Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
29.41Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
29.41Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
29.41Consensus5ht2_onOrthosteric Ligand5ht2b_on
29.41Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.41Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
29.41Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
29.17Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
29.17Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
29.17Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
29.17Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
29.17Single7SK9CCX6627SK9-ACKR3-CCX662
29.17Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
29.17Single7XN9L-054,5227XN9-SST2-L-054,522
29.17Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
29.17Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
29.17Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
29.17Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
29.17Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
29.17Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
29.03Single5GLHEndothelin-15GLH-ETB-Endothelin-1
29.03Single6IGKEndothelin-36IGK-ETB-Endothelin-3
29.03Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
28.57Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
28.57Single5N2RPSB-365N2R-A2A-PSB-36-Na
28.57Single5TVNLSD5TVN-5-HT2B-LSD
28.57Single5WQCEMPA5WQC-OX2-EMPA
28.57Single6E67BI1671076E67-β2-BI167107-Gs (fused)
28.57Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
28.57Single6TP6Filorexant6TP6-OX1-Filorexant
28.57Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
28.57Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
28.57Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
28.57Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
28.57Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
28.57Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
28.57Single7W41PD1762527W41-BB2-PD176252
28.57Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
28.57Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
28.57Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
28.57Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
28.57Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
28.57Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
28.57Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
28.57Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
28.57Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
28.57Single8JXSPF-61428JXS-D1-PF-6142
28.57Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
28.57Single8QOTNanobody-E8QOT-μ-Nanobody-E
28.57Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
28.57Single8TF5Oleic acid8TF5-GPR6-Oleic acid
28.57Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
28.57Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
28.57Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
28.57Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
28.57Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
28.57Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
28.57Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
28.57Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
28.57Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
28.57Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
28.57Consensusbombesin_offOrthosteric Ligandbb2_off
28.57Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.57Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
28.57Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
28.57Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
28.57Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
28.57Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
28.57Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
28.57Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
28.57Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
28.12Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
28.12Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
28.00Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
28.00Single4XT1Fractalkine4XT1-US28-Fractalkine
28.00Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
28.00Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
28.00Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
28.00Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
28.00Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.00Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
28.00Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
28.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.00Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
28.00Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
28.00Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
28.00Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.00Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.00Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
28.00Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single3PBLEticlopride3PBL-D3-Eticlopride
27.78Single6HLLCP999946HLL-NK1-CP99994
27.78Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
27.78Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
27.78Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
27.78Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
27.78Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
27.78Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
27.78Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
27.78Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
27.78Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
27.78Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
27.78Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
27.78Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
27.78Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
27.78Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
27.78Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
27.78Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.78Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
27.78Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
27.78Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
27.78Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
27.78Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
27.78Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
27.78Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
27.78Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
27.78Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
27.78Consensusgq_nucleotideOrthosteric Ligandgq_p2y
27.78Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
27.78Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
27.59Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
27.59Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
27.59Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
27.59Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
27.59Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
27.59Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
27.59Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
27.27Single4DJHJDTic4DJH-κ-JDTic
27.27Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
27.27Single4U15Tiotropium4U15-M3-Tiotropium
27.27Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
27.27Single6E59L-7607356E59-NK1-L-760735
27.27Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
27.27Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
27.27Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
27.27Single6OL9Tiotropium6OL9-M5-Tiotropium
27.27Single6WGTLSD6WGT-5-HT2A-LSD
27.27Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
27.27Single7B6WCyclazosin7B6W-α1b-Cyclazosin
27.27Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
27.27Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
27.27Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
27.27Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
27.27Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
27.27Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
27.27Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
27.27Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
27.27Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
27.27Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
27.27Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
27.27Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
27.27Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
27.27Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
27.27Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
27.27Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
27.27Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
27.27Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
27.27Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
27.27Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
27.27Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
27.27Single8XVLZibotentan8XVL-ETA-Zibotentan
27.27Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
27.27Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
27.27Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
27.27Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
27.27Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
27.27Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
27.27Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
27.27Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
27.27Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
27.27Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Consensusrelaxin_onOrthosteric Ligandrxfp4_on
27.27Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
27.27Consensustachykinin_offOrthosteric Ligandnk1_off
26.92Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
26.92Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
26.92Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
26.92Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
26.92Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
26.92Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
26.92Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
26.92Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
26.92Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
26.92Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
26.92Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
26.92Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
26.92Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
26.92Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
26.92Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
26.92Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
26.92Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
26.67Single5MZPCaffeine5MZP-A2A-Caffeine-Na
26.67Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
26.67Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
26.67Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
26.32Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
26.32Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
26.32Single4S0VSuvorexant4S0V-OX2-Suvorexant
26.32Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
26.32Single5WS3EMPA5WS3-OX2-EMPA
26.32Single5ZKQABT-4915ZKQ-PAF-ABT-491
26.32Single6AKXA4R6AKX-CCR5-A4R
26.32Single6B73MP11046B73-κ-MP1104
26.32Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
26.32Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
26.32Single6ME2Ramelteon6ME2-MT1-Ramelteon
26.32Single6ME9Ramelteon6ME9-MT2-Ramelteon
26.32Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
26.32Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
26.32Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
26.32Single6TPJSuvorexant6TPJ-OX2-Suvorexant
26.32Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
26.32Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
26.32Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.32Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
26.32Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.32Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.32Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
26.32Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
26.32Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
26.32Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
26.32Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
26.32Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
26.32Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
26.32Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
26.32Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
26.32Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
26.32Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
26.32Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.32Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.32Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
26.32Single8Y0HVUF114188Y0H-CXCR3-VUF11418
26.32Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
26.32Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
26.32Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
26.32Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
26.32Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.32Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
26.32Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
26.32Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
26.32Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
26.32Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.32Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.32Consensusorexin_offOrthosteric Ligandox2_off ox1_off
26.32Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
26.32Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
26.32Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
26.32Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
26.32Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
26.32Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
26.32Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
26.09Single4N4WSANT-14N4W-SMO-SANT-1
26.09Single4XEENeurotensin4XEE-NTS1-Neurotensin
26.09Single4XESNeurotensin4XES-NTS1-Neurotensin
26.09Single5CXVTiotropium5CXV-M1-Tiotropium
26.09Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
26.09Single6A93Risperidone6A93-5-HT2A-Risperidone
26.09Single6CM4Risperidone6CM4-D2-Risperidone
26.09Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
26.09Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
26.09Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
26.09Single7DFPSpiperone7DFP-D2-Spiperone
26.09Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
26.09Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
26.09Single7K15MKD0467K15-BLT1-MKD046-Na
26.09Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
26.09Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
26.09Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
26.09Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
26.09Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
26.09Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
26.09Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
26.09Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
26.09Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
26.09Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
26.09Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
26.09Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
26.09Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
26.09Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
26.09Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
26.09Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Consensusorexin_onOrthosteric Ligandox2_on
25.93Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
25.93Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
25.93Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
25.93Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
25.93Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.93Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
25.93Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
25.93Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
25.81Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
25.81Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
25.81Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
25.00Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
25.00Single3RZECidoxepin3RZE-H1-Cidoxepin
25.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
25.00Single4BUONeurotensin4BUO-NTS1-Neurotensin
25.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
25.00Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
25.00Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
25.00Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
25.00Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
25.00Single6IQLL7458706IQL-D4-L745870
25.00Single6KUXRS-799486KUX-α2a-RS-79948
25.00Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
25.00Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
25.00Single6TP3Nemorexant6TP3-OX1-Nemorexant
25.00Single6TPKRetosiban6TPK-OT-Retosiban
25.00Single6TPNHTL66416TPN-OX2-HTL6641
25.00Single6VI4JDTic6VI4-κ-JDTic
25.00Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
25.00Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
25.00Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
25.00Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
25.00Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
25.00Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
25.00Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
25.00Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
25.00Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
25.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
25.00Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
25.00Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
25.00Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
25.00Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
25.00Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
25.00Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
25.00Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
25.00Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
25.00Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
25.00Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.00Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
25.00Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
25.00Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
25.00Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
25.00Single8IHKAcifran8IHK-HCA3-Acifran
25.00Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
25.00Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
25.00Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
25.00Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
25.00Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
25.00Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
25.00Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
25.00Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
25.00Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
25.00Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
25.00Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
25.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
25.00Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
25.00Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
25.00Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
25.00Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
25.00Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
25.00Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
25.00Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
25.00Consensusopsins_offOrthosteric Ligandrhodopsin_off
25.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
25.00Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
25.00Consensussensory_offOrthosteric Ligandopsins_off
25.00Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
25.00Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
25.00Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
25.00Consensusvasop-oxy_offOrthosteric Ligandot_off
25.00Consensusvasop-oxy_onOrthosteric Ligandv2_on
25.00Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
24.32Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
24.14Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
24.14Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
24.14Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
24.14Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
24.14Single8ZRTET-18ZRT-ETB-ET-1
24.14Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
24.14Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
24.14Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
24.14Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
24.00Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
24.00Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
24.00Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
24.00Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
24.00Single8IEIA1LYA8IEI-GPR156-A1LYA
24.00Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
24.00Single8X5YAstemizole8X5Y-H1-Astemizole
24.00Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
24.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
24.00Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
24.00Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
24.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
24.00Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
24.00Consensuskisspeptin_onOrthosteric Ligandkiss1_on
24.00Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
24.00Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
23.81Single2Y01Dobutamine2Y01-β1-Dobutamine
23.81Single2Y02Carmoterol2Y02-β1-Carmoterol
23.81Single4MQSIperoxo4MQS-M2-Iperoxo
23.81Single4QIMANTA XV4QIM-SMO-ANTA XV
23.81Single4U14Tiotropium4U14-M3-Tiotropium
23.81Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
23.81Single5DHGC-355DHG-NOP-C-35
23.81Single5DHHSB-6121115DHH-NOP-SB-612111
23.81Single5DSGTiotropium5DSG-M4-Tiotropium
23.81Single5TGZAM65385TGZ-CB1-AM6538
23.81Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
23.81Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
23.81Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
23.81Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
23.81Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
23.81Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
23.81Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
23.81Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
23.81Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
23.81Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
23.81Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
23.81Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
23.81Single7WC7Lisuride7WC7-5-HT2A-Lisuride
23.81Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
23.81Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.81Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
23.81Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
23.81Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
23.81Single8T1WCVN4248T1W-GPR6-CVN424
23.81Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
23.81Single8X63Mepyramine8X63-H1-Mepyramine
23.81Single8X64Desloratadine8X64-H1-Desloratadine
23.81Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
23.81Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
23.81Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
23.81Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
23.81Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
23.81Consensushistamine_offOrthosteric Ligandh1_off
23.81Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
23.53Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
23.53Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
23.53Single9CHUNoradrenaline9CHU-β2-Noradrenaline
23.33Single4XT3Fractalkine4XT3-US28-Fractalkine
23.33Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
23.33Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
23.33Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
23.33Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
23.33Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
23.33Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
23.33Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
23.33Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
23.08Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
23.08Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
23.08Single7QA8Peptide7QA8-STE2-Peptide
23.08Single7QA8Peptide7QA8-STE2-Peptide
23.08Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
23.08Single8IEPA1LYA8IEP-GPR156-A1LYA
23.08Single8IEPA1LYA8IEP-GPR156-A1LYA
23.08Single8KIGSHU91198KIG-MC3-SHU9119-Ca
23.08Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
23.08Single8XWNCXCL88XWN-CXCR2-CXCL8
23.08Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
23.08Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
23.08Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
23.08Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
23.08Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
23.08Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
22.73Single2Y00Dobutamine2Y00-β1-Dobutamine
22.73Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
22.73Single5WIUNemonapride5WIU-D4-Nemonapride
22.73Single5WIVNemonapride5WIV-D4-Nemonapride-Na
22.73Single5XPRBosentan5XPR-ETB-Bosentan
22.73Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
22.73Single6D26Fevipiprant6D26-DP2-Fevipiprant
22.73Single6HLPNetupitant6HLP-NK1-Netupitant
22.73Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
22.73Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
22.73Single6LUQHaloperidol6LUQ-D2-Haloperidol
22.73Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
22.73Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
22.73Single7C4SS1P7C4S-S1P3-S1P
22.73Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
22.73Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
22.73Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
22.73Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
22.73Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
22.73Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
22.73Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
22.73Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
22.73Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
22.73Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
22.73Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
22.73Single8ZMFA1L108ZMF-5-HT2C-A1L10
22.73Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
22.73Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
22.73Consensusblt_offOrthosteric Ligandblt1_off
22.73Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
22.73Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
22.73Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
22.73Consensusdp_offOrthosteric Liganddp2_off
22.73Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
22.73Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
22.73Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
22.58Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
22.58Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
22.58Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
22.58Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
22.22Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
22.22Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
22.22Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
22.22Single6ME5Agomelatine6ME5-MT1-Agomelatine
22.22Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
22.22Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
22.22Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
22.22Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
22.22Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
22.22Single7XNACYN1548067XNA-SST2-CYN154806
22.22Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8IEBA1LYA8IEB-GPR156-A1LYA
22.22Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
22.22Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
22.22Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
22.22Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
22.22Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
22.22Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
22.22Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
22.22Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
22.22Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
22.22Consensusgi_sensoryOrthosteric Ligandgi_opsins
22.22Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
22.22Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
22.22Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
22.22Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
22.22Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
22.22Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
22.22Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
21.88Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
21.88Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
21.88Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
21.88Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
21.88Consensusendothelin_onOrthosteric Ligandetb_on eta_on
21.74Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
21.74Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
21.74Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
21.74Single4BV0Neurotensin4BV0-NTS1-Neurotensin
21.74Single5V56TC1145V56-SMO-TC114
21.74Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
21.74Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
21.74Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
21.74Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
21.74Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
21.74Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
21.74Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
21.74Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8EA0Iperoxo8EA0-M3-Iperoxo
21.74Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
21.74Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
21.74Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
21.74Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
21.74Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
21.74Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
21.74Consensusneurotensin_onOrthosteric Ligandnts1_on
21.74Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
21.74Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
21.74Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
21.74Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
21.62Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
21.62Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
21.43Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
21.43Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
21.43Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
21.43Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
21.43Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
21.21Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
21.21Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
21.21Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
21.05Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
21.05Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
21.05Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
21.05Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
21.05Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
21.05Single3OE9IT1t3OE9-CXCR4-IT1t
21.05Single5L7IVismodegib5L7I-SMO-Vismodegib
21.05Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
21.05Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
21.05Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
21.05Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
21.05Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.05Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
21.05Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
21.05Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
21.05Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.05Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
21.05Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
21.05Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
21.05Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
21.05Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.05Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
21.05Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
21.05Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.83Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
20.83Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
20.83Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
20.83Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
20.83Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
20.83Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
20.83Single6YVRNTS8-136YVR-NTS1-NTS8-13
20.83Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
20.83Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
20.83Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
20.83Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
20.83Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
20.83Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
20.83Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
20.83Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
20.83Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
20.83Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
20.83Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.83Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
20.83Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.69Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
20.69Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
20.69Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
20.69Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
20.69Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
20.69Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
20.69Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
20.69Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
20.59Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
20.59Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
20.59Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
20.59Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
20.59Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
20.00Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
20.00Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
20.00Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
20.00Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
20.00Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
20.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
20.00Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
20.00Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
20.00Single6AKYMaraviroc6AKY-CCR5-Maraviroc
20.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
20.00Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
20.00Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
20.00Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
20.00Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
20.00Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
20.00Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
20.00Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
20.00Single7F8ULintitript7F8U-CCKA-Lintitript
20.00Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
20.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
20.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
20.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
20.00Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
20.00Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
20.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
20.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
20.00Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
20.00Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
20.00Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
20.00Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
20.00Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
20.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
20.00Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
20.00Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
20.00Single7XRRLemborexant7XRR-OX2-Lemborexant
20.00Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
20.00Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
20.00Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
20.00Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
20.00Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
20.00Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
20.00Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
20.00Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
20.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
20.00Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
20.00Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8XVJMacitentan8XVJ-ETA-Macitentan
20.00Single8XVUCXCL28XVU-CXCR2-CXCL2
20.00Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
20.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
20.00Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
20.00Consensusangiotensin_offOrthosteric Ligandat1_off
20.00Consensuschemerin_onOrthosteric Ligandcml1_on
20.00Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
20.00Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
20.00Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
20.00Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
20.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
19.44Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
19.44Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
19.44Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
19.44Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.35Single6FJ3PTH6FJ3-PTH1-PTH
19.35Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
19.35Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
19.35Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
19.35Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
19.35Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
19.35Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
19.35Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
19.35Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
19.23Single5EE7MK08935EE7-Glucagon-MK0893
19.23Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
19.23Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
19.23Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
19.23Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
19.23Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
19.05Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
19.05Single6A94Zotepine6A94-5-HT2A-Zotepine
19.05Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
19.05Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
19.05Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
19.05Single6ZG9GSK10347026ZG9-M1-GSK1034702
19.05Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
19.05Single7VV6C48/807VV6-MRGPRX2-C48/80
19.05Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
19.05Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
19.05Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
19.05Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single8K2WAMG4878K2W-CXCR3-AMG487
19.05Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
19.05Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
19.05Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
19.05Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
19.05Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
18.75Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
18.75Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
18.75Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
18.75Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
18.75Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
18.75Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
18.75Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
18.75Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
18.75Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
18.60Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
18.52Single8IEIA1LYA8IEI-GPR156-A1LYA
18.52Consensussomatostatin_offOrthosteric Ligandsst2_off
18.18Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
18.18Single4DAJTiotropium4DAJ-M3-Tiotropium
18.18Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
18.18Single6D27CAY104716D27-DP2-CAY10471
18.18Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
18.18Single6GPSMK08126GPS-CCR2-MK0812
18.18Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
18.18Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
18.18Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
18.18Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
18.18Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
18.18Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
18.18Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
18.18Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
18.18Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
18.18Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
18.18Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
18.18Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
18.18Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
18.18Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
18.18Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
18.18Single8IY6Endothelin-18IY6-ETB-Endothelin-1
18.18Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
18.18Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
18.18Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
18.18Consensuscck_offOrthosteric Ligandccka_off
18.18Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
18.18Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
18.18Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
18.18Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
18.18Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
18.18Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
18.18Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
17.86Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
17.86Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
17.86Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.86Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
17.65Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
17.65Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
17.65Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
17.39Single4JKVTaladegib4JKV-SMO-Taladegib
17.39Single5CGCHTL142425CGC-mGlu5-HTL14242
17.39Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
17.39Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
17.39Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
17.39Single6GPXMK08126GPX-CCR2-MK0812
17.39Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
17.39Single6Z4SSR486926Z4S-NTS1-SR48692
17.39Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
17.39Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
17.39Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
17.39Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
17.39Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
17.39Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
17.39Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
17.39Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
17.39Consensusep_offOrthosteric Ligandep4_off
17.39Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
17.24Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
17.24Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
17.24Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
17.24Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
17.24Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
17.24Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
17.24Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
17.14Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
17.14Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
16.67Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
16.67Single5V57TC1145V57-SMO-TC114
16.67Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
16.67Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
16.67Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
16.67Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
16.67Single7F1TMIP-1a7F1T-CCR5-MIP-1a
16.67Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
16.67Single7P2L4YI7P2L-mGlu5-4YI
16.67Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
16.67Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
16.67Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
16.67Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
16.67Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
16.67Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
16.67Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
16.67Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
16.67Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
16.67Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
16.67Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
16.67Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
16.67Consensusp2y_offOrthosteric Ligandp2y1_off
16.67Consensussensory_onOrthosteric Ligandopsins_on
16.22Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
16.13Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
16.13Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
16.13Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
16.13Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single5X33BIIL2605X33-BLT1-BIIL260
16.00Single6OS2TRV0266OS2-AT1-TRV026
16.00Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
16.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
16.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
16.00Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single8XWACXCL18XWA-CXCR2-CXCL1
16.00Single8XWMCXCL68XWM-CXCR2-CXCL6
16.00Single8XWSCXCL58XWS-CXCR2-CXCL5
16.00Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
15.79Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
15.79Single3OE6IT1t3OE6-CXCR4-IT1t
15.79Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
15.79Single4XNWMRS25004XNW-P2Y1-MRS2500
15.79Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
15.79Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
15.79Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
15.79Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
15.79Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
15.79Single7WC5Psilocin7WC5-5-HT2A-Psilocin
15.79Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
15.79Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
15.79Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
15.79Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
15.79Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
15.79Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
15.62Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
15.62Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
15.62Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
15.62Single7SK3CXCL127SK3-ACKR3-CXCL12
15.62Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
15.38Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
15.38Single5CGDHTL142425CGD-mGlu5-HTL14242
15.38Single6K1QIRL25006K1Q-ETB-IRL2500
15.38Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
15.38Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8XWFCXCL38XWF-CXCR2-CXCL3
15.38Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
15.38Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
15.38Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
15.38Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
15.15Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
15.15Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
15.15Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
15.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
15.00Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
15.00Single6TP4ACT-4622066TP4-OX1-ACT-462206
15.00Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
15.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
15.00Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
15.00Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
15.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
15.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
15.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.00Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single9B9Y7DY9B9Y-CB1-7DY
15.00Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
15.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
14.81Single6KNMJN241-96KNM-Apelin-JN241-9
14.81Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
14.81Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single8XQJJN2418XQJ-Apelin-JN241
14.71Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
14.71Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
14.71Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
14.71Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
14.71Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
14.71Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
14.29Single3ODUIT1t3ODU-CXCR4-IT1t
14.29Single4BWBNeurotensin4BWB-NTS1-Neurotensin
14.29Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
14.29Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
14.29Single7BR3Elagolix7BR3-GnRH1-Elagolix
14.29Single7F8YDevazepide7F8Y-CCKA-Devazepide
14.29Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
14.29Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
14.29Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
14.29Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
14.29Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
14.29Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
14.29Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
14.29Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
14.29Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
14.29Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
14.29Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.29Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
14.29Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
14.29Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
14.29Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
14.29Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
14.29Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
14.29Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
14.29Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
14.29Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
14.29Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
14.29Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
13.89Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
13.79Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
13.79Single7SK5CXCL127SK5-ACKR3-CXCL12
13.64Single6FFIMMPEP6FFI-mGlu5-MMPEP
13.64Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
13.64Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
13.64Single6ZINSR486926ZIN-NTS1-SR48692
13.64Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
13.64Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
13.64Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
13.64Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8IYXYL-3658IYX-GPR34-YL-365
13.64Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
13.64Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
13.64Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
13.64Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
13.64Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
13.64Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
13.64Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
13.64Consensusgrh_offOrthosteric Ligandgnrh1_off
13.33Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.33Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.33Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.16Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
13.04Single5T04Neurotensin5T04-NTS1-Neurotensin
13.04Single6FFHFenobam6FFH-mGlu5-Fenobam
13.04Single6IIVDaltroban6IIV-TP-Daltroban
13.04Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
13.04Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
13.04Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
13.04Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
13.04Single7YXAONO-54306087YXA-S1P5-ONO-5430608
13.04Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
13.04Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
13.04Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
12.90Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
12.90Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
12.90Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
12.50Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
12.50Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
12.50Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
12.50Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
12.50Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
12.50Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
12.00Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
12.00Single6OS1TRV0266OS1-AT1-TRV026
12.00Single7R0CAVP7R0C-V2-AVP-Arrestin2
12.00Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
12.00Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
12.00Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
12.00Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
12.00Single9BJKNAM9BJK-μ-Naloxone-NAM
11.90Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
11.76Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
11.76Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
11.76Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
11.76Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
11.76Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
11.76Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
11.63Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
11.54Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
11.54Single6IIURamatroban6IIU-TP-Ramatroban
11.54Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
11.54Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
11.54Single8XQJJN2418XQJ-Apelin-JN241
11.54Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
11.43Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
11.11Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
11.11Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
11.11Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
11.11Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
11.11Single7WC4Serotonin7WC4-5-HT2A-Serotonin
11.11Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.11Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
11.11Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
11.11Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
10.81Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
10.71Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
10.53Single3OE8IT1t3OE8-CXCR4-IT1t
10.53Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
10.34Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
10.26Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
10.26Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
10.00Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
10.00Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
10.00Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
10.00Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
10.00Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
10.00Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
10.00Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
10.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
10.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
9.52Single4O9RCyclopamine4O9R-SMO-Cyclopamine
9.52Single6LI0C176LI0-GPR52-C17
9.52Single7UL2SR486927UL2-NTS1-SR48692-Na
9.52Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
9.52Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
9.52Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
9.52Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
9.52Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
9.52Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
9.52Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
9.52Consensusneurotensin_offOrthosteric Ligandnts1_off
9.52Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
9.38Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
9.09Single4QINSAG1.54QIN-SMO-SAG1.5
9.09Single5U09Taranabant5U09-CB1-Taranabant
9.09Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
9.09Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
9.09Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
9.09Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
9.09Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
9.09Single9BA0A1AKN9BA0-CB1-A1AKN
9.09Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
9.09Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.70Single7VODCariprazine7VOD-5-HT2A-Cariprazine
8.70Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
8.33Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
8.33Single7F83PF-051904577F83-Ghrelin-PF-05190457
8.33Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
8.33Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
8.33Single9B9ZA1AKO9B9Z-CB1-A1AKO
8.33Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
8.00Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
8.00Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
7.89Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
7.69Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
7.69Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
7.41Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
7.14Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
7.14Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
7.14Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
7.14Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
6.90Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
6.90Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
6.67Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
6.67Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
6.45Single7SHEPI; PE7SHE-GPR158-PI; PE
5.88Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
5.88Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
5.56Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
5.56Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.00Single6TQ9SB-4081246TQ9-OX1-SB-408124
5.00Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
5.00Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
5.00Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
4.76Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
4.76Single8JPSCCL78JPS-ACKR1-CCL7
4.76Single8WG8Peptide8WG8-Glucagon-Peptide-chim(NtGi1-Gs)/β1/γ2
4.55Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
4.55Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
4.35Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
4.35Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
4.35Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
4.17Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
4.00Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
3.85Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
3.57Single7SHEPI; PE7SHE-GPR158-PI; PE
3.12Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7

Consensus Members
Id Members
adenosine_on_gp a1_on_gp
a2_on_gp
a3_on_gp
p2y_on_gp p2y1_on_gp
p2y10_on_gp
p2y12_on_gp
Net Summary
Imin 2.77792
Number of Linked Nodes 942
Number of Links 1098
Number of Hubs 171
Number of Links mediated by Hubs 668
Number of Communities 20
Number of Nodes involved in Communities 218
Number of Links involved in Communities 313
Path Summary
Number Of Nodes in MetaPath 111
Number Of Links MetaPath 110
Number of Shortest Paths 1199796
Length Of Smallest Path 3
Average Path Length 33.152
Length of Longest Path 72
Minimum Path Strength 0.410139
Average Path Strength 5.37302
Maximum Path Strength 17.4646
Minimum Path Correlation 0.70125
Average Path Correlation 0.967786
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.51515
Average % Of Corr. Nodes 35.8083
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 48.4679
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following differences:
Id1st Network2nd Network
nucleotide_off_on_gpnucleotide_on_gpnucleotide_off
This network is also present in following consensuses:
IdComponents
nucleotide_offon_gpnucleotide_on_gp
nucleotide_off
class-a_on_gpsensory_on_gp
alicarboxylic_on_gp
amine_on_gp
lipid_on_gp
nucleotide_on_gp
peptide_on_gp
protein_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download nucleotide_on_gp.zip



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