Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.51 8.13404
2G.s1h1.04 6.04254169
3G.H1.01 4.7485209
4G.S2.01 5.845429
5G.S2.03 9.335429
6G.S3.03 6.345608
7G.S3.04 12.485427
8G.S3.06 12.368527
9G.H2.04 8.124199
10G.H2.06 5.525649
11G.H2.07 6.17409
12G.h2s4.01 8.878529
13G.S4.04 5.65509
14G.s4h3.04 9.125218
15G.H3.01 10.6854169
16G.H3.09 6.8425409
17G.H3.13 11.075406
18G.H3.17 9.092525
19G.S5.05 6.8575409
20G.S5.07 6.43409
21G.hgh4.02 5.51254178
22G.hgh4.04 5.354176
23G.hgh4.05 10.9075406
24G.hgh4.08 5.25406
25G.hgh4.20 7.43254123
26G.hgh4.21 6.3575404
27G.H4.10 9.3085177
28G.H4.15 7.2025408
29G.S6.02 10.3067698
30G.S6.05 7.8754125
31G.s6h5.01 7.1375409
32G.s6h5.05 7.18409
33G.H5.08 6.0665158
34G.H5.23 5.23833614
35b.ntx3 3.8225185
36b.1x4 3.7485188
37b.lhb1x3 4.5185102
38b.lhb1x11 5.145474
39b.b1x3 6.05254137
40b.l1x3 9.1685119
41b.l1x6 13.3375429
42b.b2x1 11.885428
43b.b2x5 6.95167607
44b.l3x2 6.935119
45b.b4x2 5.915408
46b.b4x3 6.24467
47b.b4x6 10.22176119
48b.b5x3 6.55409
49b.b5x5 5.605405
50b.b5x7 7.845467
51b.l5x1 4.225468
52b.l5x5 9.00571729
53b.b6x5 4.55286766
54b.l6x5 6.5425484
55b.b7x1 7.294584
56b.b7x2 4.9025468
57b.b8x4 5.16667666
58b.l8x1 4.5575465
59b.l8x3 3.9025483
60b.l8x5 3.495483
61b.l8x8 6.1375464
62b.l9x3 7.816549
63b.l9x6 6.03333648
64b.b10x5 5.34833609
65b.l10x1 4.21403
66b.b11x4 6.0875449
67b.b11x6 7.1075449
68b.l11x2 8.1275449
69b.b12x3 4.585458
70b.b12x6 10.415648
71b.b13x3 7.62444
72b.b13x7 9.136557
73b.l13x3 9.195659
74b.l13x7 5.07459
75b.b14x3 5.12455
76b.b15x1 7.874559
77b.b15x2 9.48436
78b.l15x2 5.992559
79b.b16x4 11.8225456
80b.b16x5 6.2675405
81b.b16x6 9.04333658
82b.b17x5 7.7175437
83b.b17x7 8.0725438
84b.l17x3 8.18639
85b.l17x6 7.43449
86b.b18x3 5.095438
87b.b18x5 5.4275405
88b.l18x1 8.27254236
89b.l18x2 6.0154237
90b.b19x2 8.61667636
91b.b19x4 6.6575438
92b.l19x2 7.84539
93b.b20x4 12.422538
94b.b20x6 7.632536
95b.b21x1 9.236537
96b.b21x3 9.5075436
97b.b21x5 7.0575404
98b.b21x7 6.66505
99b.l21x2 7.2775404
100b.l22x5 7.881676109
101b.b23x2 5.705406
102b.b23x6 7.47571727
103b.l23x1 5.925426
104b.b24x4 8.515426
105b.b24x6 6.955428
106b.l24x2 6.4954106
107b.l24x3 5.2625405
108b.b25x7 9.355477
109b.l25x3 7.774579
110b.l25x6 11.958528
111b.l27x1 10.8375829
112b.l27x2 6.5925479
113b.b28x3 5.3245117
114b.b28x4 8.2475476
115b.b28x6 8.27667679
116g.h1x11 3.1475409
117g.ctx3 7.35409
118g.ctx6 3.4406
119g.ctx14 5.2825139
120g.ctx16 6.305717138
121I1.H58 6.8475405
122I1.R60 5.155406
1232x39 7.5025418
1242x42 4.71333617
1252x43 5.312518
1262x46 6.28419
1272x50 7.42519
1282x51 5.1675407
129E1x50 8.295406
130E1.D99 3.22405
1313x33 4.605407
1323x34 8.495417
1333x46 6.245419
1343x49 8.425419
1353x50 8.615419
1363x51 6.682507
137I2x51 6.108505
138E2.Y174 10.255406
139E2.Y178 11.58254143
140E2.W182 7.998517
141E2x51 6.9875408
1425x39 6.735407
1435x57 3.8025407
1445x69 6.805406
1456x26 9.5675497
1466x34 5.08518
1476x38 4.765418
1486x48 9.054518
1496x54 7.024504
1506x55 2.25407
1517x31 6.17754143
1527x45 7.262519
1537x46 6.48333619
1547x49 7.7775419
1557x52 3.3975408
1567x53 8.08519
157Lig 6.979381610
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b3x1 b.b4x7 17.08564.07NoNo058
2b.b3x1 b.b6x5 16.05163.52NoYes056
3b.b4x7 b.l2x5 22.77315.48NoNo085
4b.l2x5 b.l4x2 23.290229.84NoNo054
5b.l4x2 g.ctx16 24.2747.22NoYes048
6b.l4x1 g.ctx16 16.52695.28NoYes058
7b.b2x5 b.l4x1 16.78524.94YesNo075
8b.b2x5 b.b3x2 23.553610.25YesNo075
9b.b3x2 b.b4x6 23.29456.83NoYes059
10b.b28x5 g.ctx16 16.52697.54NoYes1358
11b.b28x5 b.b2x5 17.30263.52NoYes057
12b.b5x7 b.b5x8 11.37413.39YesNo075
13b.b4x2 b.b5x8 11.88998.36YesNo085
14b.b4x2 b.l3x2 14.48278.3YesYes089
15b.b2x3 b.b2x5 80.00546.98NoYes067
16b.b26x2 b.b2x3 80.26194.86NoNo076
17b.b26x1 b.b26x2 80.51853.44NoNo097
18b.b26x1 b.l27x1 80.77514.94NoYes099
19b.b2x1 b.l27x1 10012.54YesYes289
20b.b2x1 b.l3x1 10021.42YesNo289
21b.l3x1 b.l5x5 1009.86NoYes299
22G.h2s4.01 b.l5x5 10013.03YesYes299
23G.S1.05 G.h2s4.01 42.869414.61NoYes099
24G.S1.05 G.S1.07 43.42059.69NoNo098
25G.H3.12 G.S1.07 43.50225.71NoNo1988
26G.H3.12 G.S4.04 1005.02NoYes089
27G.S4.04 G.S5.04 1004.87YesNo099
28G.S5.04 G.S5.06 1004.15NoNo098
29G.S5.06 G.S6.05 1004.87NoYes085
30G.H4.12 G.S6.05 1007.48NoYes045
31G.H4.12 G.S6.03 10011.53NoNo045
326x25 G.S6.03 1006.32NoNo045
336x25 G.S6.02 10016.91NoYes048
34G.H5.10 G.S6.02 10011.49NoYes078
35G.H5.10 G.S6.04 10012.61NoNo079
36G.S5.05 G.S6.04 1006.79YesNo099
37G.H5.07 G.S5.05 1005.02NoYes099
38G.H5.07 G.S4.03 1004.42NoNo097
39G.S1.04 G.S4.03 1005.71NoNo077
40G.S1.04 G.S3.03 1004.87NoYes078
41G.S1.02 G.S3.03 1007.31NoYes068
42G.H2.07 G.h2s4.01 87.22234.01YesYes099
43G.H2.04 G.H2.07 1007YesYes099
44G.H2.04 G.H3.12 87.00317.52YesNo1998
45G.H2.04 G.H3.08 87.003113.1YesNo098
46G.H3.08 G.S4.04 87.08184.78NoYes089
47G.S1.02 I2x51 1003.65NoYes065
48G.S3.01 G.S3.03 1003.93NoYes058
49G.S3.01 I2x51 10010.49NoYes055
50G.H2.06 b.l9x6 65.06963.58YesYes498
51G.H2.07 b.l9x6 88.7653.86YesYes098
52G.H2.06 b.l17x6 32.27675.53YesYes499
53G.H2.06 b.b18x1 32.27715.6YesNo099
54G.H3.17 b.l27x1 20.92663.75YesYes259
55b.l25x6 b.l27x1 20.926621.99YesYes289
56G.H3.17 b.l23x1 20.4094.47YesYes256
57b.l23x1 b.l25x6 20.4099.53YesYes268
58G.H5.12 I2x51 1006.2NoYes075
59G.H5.12 I2x50 1005.02NoNo078
60G.H5.15 I2x51 1003.77NoYes085
61G.H5.15 I2x50 1003.39NoNo088
62G.H5.16 I2x50 1003.28NoNo068
63G.H5.16 G.H5.20 1005.54NoNo068
646x34 G.H5.23 95.18044.79YesYes184
656x34 G.H5.20 1004.24YesNo088
662x39 G.H5.23 92.32558.25YesYes184
672x39 3x50 92.307310.69YesYes189
683x50 6x34 92.60673.72YesYes198
69b.l13x6 b.l9x6 13.82046.9NoYes498
70b.l13x5 b.l13x6 13.6591.68NoNo059
71b.l13x5 b.l15x2 13.30941.68NoYes059
72b.l13x3 b.l15x2 11.20977.56YesYes599
73b.l17x6 b.l19x1 32.10695.32YesNo099
74b.l17x5 b.l19x1 63.86564.42NoNo069
75b.b19x6 b.l17x5 26.37974.89NoNo396
76b.b19x6 b.l17x3 26.033112.55NoYes399
77b.b19x4 b.l17x3 29.85218.21YesYes389
78b.b19x4 b.b20x6 15.9687.78YesYes386
79b.b17x7 b.b20x6 32.977710.72YesYes386
80b.b17x7 b.b21x1 27.77175.97YesYes387
81b.1x19 b.b21x1 20.830210.72NoYes067
82b.b18x1 b.l19x1 32.104712.12NoNo099
83b.l17x5 b.l19x2 37.13997.36NoYes369
84b.l17x3 b.l19x2 26.03366.3YesYes399
85b.b20x4 b.l17x3 19.438711.28YesYes389
86b.b20x4 b.b20x6 23.95234.28YesYes386
87b.b20x2 b.l19x2 10.413514.45NoYes069
88b.1x19 b.b21x2 12.15125.84NoNo066
89b.l26x5 g.ctx4 20.73376.71NoNo057
90g.ctx3 g.ctx4 19.96174.83YesNo097
91b.b21x5 b.h2x1 13.48699.9YesNo045
92b.l21x7 b.l23x1 39.78234.67NoYes256
93b.b23x6 b.l21x7 37.71034.03YesNo275
94b.l22x1 g.ctx3 17.38188.83NoYes099
95b.b23x1 b.l22x1 17.12274.5NoNo059
96b.b3x4 b.b4x6 10.35154.94NoYes1199
97b.b3x4 b.l1x3 10.09328.37NoYes1199
98b.b4x4 b.b4x6 10.351512.92NoYes089
99b.b4x4 b.l1x3 10.092211.93NoYes089
100b.l1x3 b.l3x2 19.1495.04YesYes1199
101b.l26x3 b.l26x5 21.18274.16NoNo075
102b.l26x1 b.l26x3 21.43848.67NoNo2277
103b.b2x5 b.l26x1 21.955112.13YesNo077
104b.b18x3 b.b19x4 13.19094.56YesYes388
105b.b21x5 b.b21x7 16.056611.97YesYes045
106b.b21x7 b.b23x2 10.36624.69YesYes056
107b.b21x7 b.b24x6 27.89156.75YesYes058
108b.b23x6 b.b24x6 28.91328.68YesYes278
1093x25 E2x50 13.56697.28NoNo099
1103x28 E2x50 27.13373.24NoNo069
1113x28 3x32 31.20335.78NoNo068
1123x32 Lig 62.39045.99NoYes080
1136x48 Lig 50.84574.82YesYes180
1146x48 7x45 54.563612.43YesYes189
1157x45 7x49 1009.42YesYes199
1167x49 7x53 1006.9YesYes199
1172x43 7x53 91.48193.52YesYes189
1182x39 2x43 92.92916.09YesYes188
1197x46 Lig 1004.7YesYes190
1207x45 7x46 51.51516.6YesYes199
1212x50 7x46 1009.14YesYes199
1222x50 7x49 57.61226.65YesYes199
1232x46 2x50 57.62268.14YesYes199
1242x46 7x53 63.37214.69YesYes199
1253x46 7x53 91.560110.78YesYes199
1262x39 3x46 91.57394.98YesYes189
1276x41 7x53 45.707314.51NoYes089
1285x58 6x41 46.21444.25NoNo098
1295x58 6x38 46.27815.49NoYes098
1306x34 6x38 46.40544.24YesYes188
131E2.S181 Lig 40.69775.3NoYes180
132E2.P179 E2.S181 39.3433.56NoNo088
133E2.P179 E2.Y178 36.6311.13NoYes083
1347x31 E2.Y178 21.70710.1YesYes1433
1357x28 E2.Y178 10.853515.43NoYes1413
1362x65 Lig 13.56599.07NoYes170
1371x36 2x65 12.2114.58NoNo067
138E2.V176 E2x50 12.21023.42NoNo049
1393x24 E1x50 13.567110.25NoYes066
1403x24 E1.D99 10.85376.79NoYes065
1414x61 E2.Y174 10.85142.34NoYes056
1423x33 E2.Y174 21.70174.84YesYes076
1433x33 E2x51 29.83953.77YesYes078
1443x32 E2x51 29.84434.98NoYes088
145E2.W182 E2x51 29.84447.02YesYes078
146E2.W182 Lig 58.321412.86YesYes170
147E2x51 E2x52 27.131312.18YesNo085
1485x39 E2x52 21.70658.53YesNo075
1494x59 5x39 13.56424.87NoYes087
150E3.L282 E3.M276 10.85427.07NoNo041
1517x31 E3.L282 12.2115.3YesNo034
152E2.Q177 E2.W182 25.77779.86NoYes077
1536x54 6x58 12.2117.78YesNo046
1546x54 7x34 23.06457.31YesNo046
1557x34 E2.Q177 24.42112.66NoNo067
1564x59 E2.V171 10.85141.49NoNo084
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
1x362x654.580NoNo6721
1x381x424.290NoNo5822
1x387x3923.520NoNo5821
1x39Lig6.670NoYes7010
1x427x425.190NoNo8821
1x43Lig5.60NoYes6010
2x503x396.441YesNo9822
2x507x469.141YesYes9921
2x547x463.991NoYes8911
2x54Lig5.861NoYes8010
2x57Lig10.40NoYes7010
2x61Lig9.460NoYes8010
2x65E2.S1818.371NoNo7811
2x65Lig9.071NoYes7010
3x283x325.780NoNo6821
3x32E2x514.980NoYes8812
3x32Lig5.990NoYes8010
3x36Lig6.030NoYes7010
3x397x467.91NoYes8921
3x406x4813.670NoYes8821
E2.Q177E2.W1829.860NoYes7721
E2.P179E2.S1813.560NoNo8821
E2.S181Lig5.31NoYes8010
E2.W182E2x517.021YesYes7812
7x35E2.W1823.420NoYes7721
7x38E2.W1826.831NoYes7711
E2.W182Lig12.861YesYes7010
6x487x417.781YesNo8812
6x487x4512.431YesYes8912
6x487x466.571YesYes8911
6x48Lig4.821YesYes8010
7x357x3912.150NoNo7821
7x38Lig7.811NoYes7010
7x39Lig4.290NoYes8010
7x42Lig10.40NoYes8010
7x457x466.61YesYes9921
7x46Lig4.71YesYes9010
2x573x313.170NoNo7512
2x58Lig2.410NoYes8010

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
100.00Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
100.00Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
100.00Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
93.33Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
87.50Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
81.25Single6IIURamatroban6IIU-TXA2-Ramatroban
81.25Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
81.25Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
76.47Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
76.47Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
75.00Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
73.33Single6IIVDaltroban6IIV-TXA2-Daltroban
72.22Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
72.22Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
70.59Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
70.59Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
70.59Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
68.75Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
66.67Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
66.67Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
64.71Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
64.71Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
64.71Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
62.50Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
60.00Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
58.82Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
58.82Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
58.82Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
57.89Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
57.89Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
56.25Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
55.56Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
55.00Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
55.00Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
42.86Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
36.84Single5TGZAM65385TGZ-CB1-AM6538
36.84Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
35.29Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
35.00Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
35.00Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
33.33Single5U09Taranabant5U09-CB1-Taranabant
33.33Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
33.33Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
31.82Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
31.82Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
31.82Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
31.58Single2YDOAdenosine2YDO-A2A-Adenosine
31.58Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
31.58Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
31.58Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
31.58Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
31.58Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
31.58Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
31.25Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
30.43Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
30.00Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
30.00Single7YXAONO-54306087YXA-S1P5-ONO-5430608
30.00Single8T1WCVN4248T1W-GPR6-CVN424
30.00Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
30.00Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
30.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
30.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
30.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
30.00Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
29.63Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
29.41Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
29.17Single5ZTYAM102575ZTY-CB2-AM10257
29.17Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
28.57Single5CGCHTL142425CGC-mGlu5-HTL14242
28.57Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
28.57Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
28.57Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
28.57Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
28.57Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
28.57Single9B9ZA1AKO9B9Z-CB1-A1AKO
28.57Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
28.57Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
28.57Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
28.57Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
28.57Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
28.57Consensusep_offOrthosteric Ligandep4_off
28.57Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
28.57Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Consensustrace-amine_onOrthosteric Ligandta1_on
27.78Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
27.78Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
27.78Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
27.78Single8K5BNiacin8K5B-HCA2-Niacin
27.78Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
27.78Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
27.78Single9B9Y7DY9B9Y-CB1-7DY
27.78Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
27.27Single2YDVNECA2YDV-A2A-NECA
27.27Single4UHRCGS216804UHR-A2A-CGS21680
27.27Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
27.27Single5G53NECA5G53-A2A-NECA-Gs
27.27Single5XR8AM8415XR8-CB1-AM841
27.27Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
27.27Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
27.27Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
27.27Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
27.27Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
27.27Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
27.27Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
26.32Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
26.32Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
26.32Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.32Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.32Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
26.32Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
26.32Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
26.32Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
26.32Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
26.32Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
26.32Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
26.32Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
26.32Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
26.32Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
26.32Single8Y0HVUF114188Y0H-CXCR3-VUF11418
26.32Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
26.32Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
26.32Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
26.32Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
26.32Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
26.32Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
26.32Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.32Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
26.09Single4N4WSANT-14N4W-SMO-SANT-1
26.09Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
26.09Single6KQICP559406KQI-CB1-CP55940-Org27569
26.09Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
26.09Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
26.09Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
26.09Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
26.09Single9DGIZ85267113509DGI-CB1-Z8526711350
26.09Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
26.09Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
26.09Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
26.09Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
25.81Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
25.00Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
25.00Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
25.00Single5CGDHTL142425CGD-mGlu5-HTL14242
25.00Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
25.00Single6ZG9GSK10347026ZG9-M1-GSK1034702
25.00Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
25.00Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
25.00Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
25.00Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
25.00Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
25.00Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
25.00Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
25.00Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
25.00Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
25.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
25.00Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
25.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
25.00Single8IHKAcifran8IHK-HCA3-Acifran
25.00Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
25.00Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
25.00Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
25.00Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
25.00Single8K5CAcipimox8K5C-HCA2-Acipimox
25.00Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
25.00Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
25.00Single8XVJMacitentan8XVJ-ETA-Macitentan
25.00Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
25.00Single9BA0A1AKN9BA0-CB1-A1AKN
25.00Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
25.00Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
25.00Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
25.00Consensusalpha1_onOrthosteric Ligandalpha1a_on
25.00Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
25.00Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
25.00Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
25.00Consensushca_onOrthosteric Ligandhca2_on
24.14Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
24.00Single3NY9ICI118-5513NY9-β2-ICI118-551
24.00Single4UG2CGS216804UG2-A2A-CGS21680
24.00Single6PT3DPI-2876PT3-δ-DPI-287
24.00Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
24.00Single7SK9CCX6627SK9-ACKR3-CCX662
24.00Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
24.00Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
24.00Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
24.00Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
23.81Single3NY8ICI118-5513NY8-β2-ICI118-551
23.81Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
23.81Single4EJ4Naltrindole4EJ4-δ-Naltrindole
23.81Single4GBRS-Carazolol4GBR-β2-S-Carazolol
23.81Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
23.81Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
23.81Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
23.81Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
23.81Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
23.81Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
23.81Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
23.81Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.81Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
23.81Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
23.81Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
23.81Single7V3ZCP559407V3Z-CB1-CP55940
23.81Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
23.81Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
23.81Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
23.81Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
23.81Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
23.81Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
23.81Single8JJOAlprenolol8JJO-β2-Alprenolol
23.81Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
23.81Single8JXRLSD8JXR-D1-LSD
23.81Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
23.81Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
23.81Single9CHXS-Carazolol9CHX-β2-S-Carazolol
23.81Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
23.81Single9JEAAtropine9JEA-M1-Atropine
23.81Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
23.81Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
23.81Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
23.81Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
23.81Consensusalpha2_onOrthosteric Ligandalpha2b_on
23.81Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
23.81Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
23.81Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
23.81Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
23.81Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
23.81Consensusdopamine_offOrthosteric Ligandd2_off d3_off
23.81Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
23.81Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
23.81Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
23.81Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
23.81Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
23.81Consensushca_on_gpOrthosteric Ligandhca2_on_gp
23.81Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
23.81Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
23.53Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.53Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
23.33Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
23.33Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
23.33Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
23.08Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
23.08Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
23.08Single7QA8Peptide7QA8-STE2-Peptide
23.08Single7QA8Peptide7QA8-STE2-Peptide
23.08Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
23.08Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
23.08Single8WDTphotoNECA8WDT-A2A-photoNECA
23.08Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Single9M4TSilodosin9M4T-Alpha1A-Silodosin
23.08Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
23.08Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
22.86Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
22.73Single2RH1S-Carazolol2RH1-β2-S-Carazolol
22.73Single2YCWS-Carazolol2YCW-β1-S-Carazolol
22.73Single5D6LS-Carazolol5D6L-β2-S-Carazolol
22.73Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
22.73Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
22.73Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
22.73Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
22.73Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
22.73Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
22.73Single6PS6Timolol6PS6-β2-Timolol
22.73Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
22.73Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
22.73Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
22.73Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
22.73Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
22.73Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
22.73Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
22.73Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
22.73Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
22.73Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
22.73Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
22.73Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
22.73Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
22.73Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
22.73Single9HC04YI9HC0-mGlu5-4YI
22.73Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
22.73Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
22.73Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
22.73Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
22.73Consensusamine_offonOrthosteric Ligandamine_off amine_on
22.73Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
22.73Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
22.73Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
22.73Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
22.73Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
22.73Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
22.73Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
22.73Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
22.73Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
22.73Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.73Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.58Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
22.58Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
22.58Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
22.58Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
22.58Consensusglp_onOrthosteric Ligandglp1_on glp2_on
22.58Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
22.22Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
22.22Single3QAKUK-4320973QAK-A2A-UK-432097
22.22Single6HLOAprepitant6HLO-NK1-Aprepitant
22.22Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
22.22Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
22.22Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
22.22Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
22.22Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
22.22Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
22.22Single9LRCHistamine9LRC-H4-Histamine
22.22Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
22.22Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
22.22Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
22.22Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
22.22Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
21.88Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
21.88Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
21.88Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
21.74Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
21.74Single4DJHJDTic4DJH-κ-JDTic
21.74Single4U15Tiotropium4U15-M3-Tiotropium
21.74Single5D5AS-Carazolol5D5A-β2-S-Carazolol
21.74Single5D5BS-Carazolol5D5B-β2-S-Carazolol
21.74Single5XRAAM115425XRA-CB1-AM11542
21.74Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
21.74Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
21.74Single6J21Aprepitant6J21-NK1-Aprepitant
21.74Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
21.74Single6OL9Tiotropium6OL9-M5-Tiotropium
21.74Single6TQ7SB-3348676TQ7-OX1-SB-334867
21.74Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
21.74Single7FEECP559407FEE-CB1-CP55940-ZCZ011
21.74Single7P2L4YI7P2L-mGlu5-4YI
21.74Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
21.74Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
21.74Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
21.74Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
21.74Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
21.74Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
21.74Single8EA0Iperoxo8EA0-M3-Iperoxo
21.74Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
21.74Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
21.74Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
21.74Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
21.74Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
21.74Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
21.74Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
21.74Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
21.74Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
21.74Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
21.74Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
21.74Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
21.74Single9BJKNaloxone9BJK-μ-Naloxone-NAM
21.74Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
21.74Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
21.74Consensusa2_onOrthosteric Liganda2b_on
21.74Consensusa2_on_gpOrthosteric Liganda2b_on_gp
21.74Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
21.74Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
21.74Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
21.74Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
21.74Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
21.74Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
21.74Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
21.74Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
21.74Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
21.74Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
21.74Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
21.74Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
21.74Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
21.74Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
21.43Single5WF5UK-4320975WF5-A2A-UK-432097
21.43Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
21.43Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
21.21Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
21.21Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
21.05Single5L7IVismodegib5L7I-SMO-Vismodegib
21.05Single6LI0C176LI0-GPR52-C17
21.05Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
21.05Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
21.05Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
21.05Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
21.05Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
21.05Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
21.05Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
21.05Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
21.05Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
20.83Single3D4STimolol3D4S-β2-Timolol
20.83Single4AMIBucindolol4AMI-β1-Bucindolol
20.83Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
20.83Single5CXVTiotropium5CXV-M1-Tiotropium
20.83Single5X33BIIL2605X33-BLT1-BIIL260
20.83Single6A93Risperidone6A93-5-HT2A-Risperidone
20.83Single6CM4Risperidone6CM4-D2-Risperidone
20.83Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
20.83Single6ZG4HTL00099366ZG4-M1-HTL0009936
20.83Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
20.83Single7DFPSpiperone7DFP-D2-Spiperone
20.83Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
20.83Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.83Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
20.83Single7YITNalfurafine7YIT-κ-Nalfurafine
20.83Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
20.83Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
20.83Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
20.83Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
20.83Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
20.83Single8XYIVUF106618XYI-CXCR3-VUF10661
20.83Single9BJKNAM9BJK-μ-Naloxone-NAM
20.83Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.83Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.83Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
20.83Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
20.83Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
20.83Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
20.83Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
20.83Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
20.83Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
20.83Consensuslpl_offOrthosteric Ligands1p_off lpa_off
20.83Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
20.83Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
20.83Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
20.83Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
20.83Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
20.69Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
20.69Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
20.69Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
20.69Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
20.69Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
20.69Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
20.59Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
20.59Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
20.59Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
20.51Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
20.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
20.00Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
20.00Single5X93K-87945X93-ETB-K-8794
20.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
20.00Single6AKXA4R6AKX-CCR5-A4R
20.00Single6AKYMaraviroc6AKY-CCR5-Maraviroc
20.00Single6B73MP11046B73-κ-MP1104
20.00Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
20.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
20.00Single6H7LDobutamine6H7L-β1-Dobutamine
20.00Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.00Single6TODEMPA6TOD-OX1-EMPA-Na
20.00Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
20.00Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
20.00Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
20.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
20.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
20.00Single7EZCUKA7EZC-A2A-UKA
20.00Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
20.00Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
20.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
20.00Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
20.00Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
20.00Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
20.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
20.00Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
20.00Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
20.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
20.00Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
20.00Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
20.00Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
20.00Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
20.00Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
20.00Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
20.00Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
20.00Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
20.00Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
20.00Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
20.00Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
20.00Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
20.00Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
20.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
20.00Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
20.00Single8IWESpermidine8IWE-TA9-Spermidine
20.00Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
20.00Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
20.00Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
20.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
20.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
20.00Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
20.00Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
20.00Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
20.00Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
20.00Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.00Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
20.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
20.00Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
20.00Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
20.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
20.00Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
20.00Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
20.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
20.00Consensusangiotensin_offOrthosteric Ligandat1_off
20.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
20.00Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
20.00Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
20.00Consensusendothelin_offOrthosteric Ligandetb_off
20.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
20.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
20.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
20.00Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
20.00Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
20.00Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
20.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
20.00Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.00Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
20.00Consensusprostanoid_offOrthosteric Ligandep_off dp_off
20.00Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
20.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
19.44Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
19.44Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
19.44Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
19.44Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
19.44Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
19.44Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.35Single6FJ3PTH6FJ3-PTH1-PTH
19.35Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
19.35Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
19.35Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
19.35Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
19.35Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
19.35Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
19.35Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
19.35Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
19.35Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
19.35Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
19.35Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
19.35Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
19.35Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
19.35Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
19.23Single5WF6UK-4320975WF6-A2A-UK-432097
19.23Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
19.23Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
19.23Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
19.23Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
19.23Single8X5YAstemizole8X5Y-H1-Astemizole
19.23Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
19.23Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
19.23Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
19.23Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
19.05Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
19.05Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
19.05Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
19.05Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
19.05Single4MBSMaraviroc4MBS-CCR5-Maraviroc
19.05Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
19.05Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
19.05Single4ZJCSB-6740424ZJC-OX1-SB-674042
19.05Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
19.05Single6FFIMMPEP6FFI-mGlu5-MMPEP
19.05Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
19.05Single6PS0S-Carazolol6PS0-β2-S-Carazolol
19.05Single6PS4ICI118-5516PS4-β2-ICI118-551
19.05Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
19.05Single6TPGEMPA6TPG-OX2-EMPA
19.05Single6VI4JDTic6VI4-κ-JDTic
19.05Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
19.05Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
19.05Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
19.05Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
19.05Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
19.05Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
19.05Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
19.05Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
19.05Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
19.05Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
19.05Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
19.05Single7F61PF-036547467F61-H3-PF-03654746
19.05Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.05Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
19.05Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
19.05Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
19.05Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
19.05Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
19.05Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
19.05Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
19.05Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
19.05Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
19.05Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
19.05Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
19.05Single8K2WAMG4878K2W-CXCR3-AMG487
19.05Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
19.05Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
19.05Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
19.05Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
19.05Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
19.05Single8ZPMAMD0708ZPM-CXCR4-AMD070
19.05Single9AS5Mescaline9AS5-5-HT2A-Mescaline
19.05Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
19.05Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
19.05Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
19.05Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
19.05Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
19.05Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
19.05Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
19.05Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
19.05Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
19.05Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
19.05Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
19.05Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
19.05Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
19.05Consensusopsins_offOrthosteric Ligandrhodopsin_off
19.05Consensussensory_offOrthosteric Ligandopsins_off
18.75Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
18.75Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
18.75Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
18.75Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
18.75Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
18.75Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
18.75Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
18.75Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
18.75Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
18.75Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
18.75Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
18.52Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
18.52Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
18.52Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
18.52Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
18.52Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
18.52Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
18.52Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
18.52Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
18.52Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
18.52Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
18.52Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
18.52Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.18Single2Y01Dobutamine2Y01-β1-Dobutamine
18.18Single2Y04Salbutamol2Y04-β1-Salbutamol
18.18Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
18.18Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
18.18Single4DAJTiotropium4DAJ-M3-Tiotropium
18.18Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
18.18Single4MQSIperoxo4MQS-M2-Iperoxo
18.18Single4QKX35V4QKX-β2-35V
18.18Single4U14Tiotropium4U14-M3-Tiotropium
18.18Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
18.18Single4YAYZD-71554YAY-AT1-ZD-7155
18.18Single5DHHSB-6121115DHH-NOP-SB-612111
18.18Single5DSGTiotropium5DSG-M4-Tiotropium
18.18Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
18.18Single6FFHFenobam6FFH-mGlu5-Fenobam
18.18Single6H7MSalbutamol6H7M-β1-Salbutamol
18.18Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
18.18Single6PS1Timolol6PS1-β2-Timolol
18.18Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
18.18Single6TOTLemborexant6TOT-OX1-Lemborexant
18.18Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
18.18Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
18.18Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
18.18Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
18.18Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.18Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
18.18Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
18.18Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
18.18Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
18.18Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
18.18Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
18.18Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
18.18Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
18.18Single7UL4Alvimopan7UL4-μ-Alvimopan
18.18Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
18.18Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
18.18Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
18.18Single7WC7Lisuride7WC7-5-HT2A-Lisuride
18.18Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
18.18Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
18.18Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
18.18Single8CU6LJ-45178CU6-A2A-LJ-4517
18.18Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
18.18Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
18.18Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
18.18Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
18.18Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
18.18Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
18.18Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
18.18Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
18.18Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
18.18Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
18.18Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
18.18Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
18.18Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
18.18Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
18.18Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
18.18Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
18.18Single8K5DGSK2560738K5D-HCA2-GSK256073
18.18Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
18.18Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
18.18Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
18.18Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
18.18Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
18.18Single8X63Mepyramine8X63-H1-Mepyramine
18.18Single8X64Desloratadine8X64-H1-Desloratadine
18.18Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
18.18Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
18.18Single9AS1DMT9AS1-5-HT2A-DMT
18.18Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
18.18Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
18.18Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
18.18Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
18.18Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
18.18Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.18Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.18Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
18.18Consensusa3_onOrthosteric Liganda3a_on
18.18Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
18.18Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
18.18Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
18.18Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
18.18Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
18.18Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
18.18Consensusblt_onOrthosteric Ligandblt1_on
18.18Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
18.18Consensusbradykinin_onOrthosteric Ligandbk2_on
18.18Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
18.18Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
18.18Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
18.18Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
18.18Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
18.18Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
18.18Consensushistamine_offOrthosteric Ligandh1_off
18.18Consensusleukotriene_onOrthosteric Ligandblt_on
18.18Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
18.18Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
18.18Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
18.18Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
18.18Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
18.18Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
17.95Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
17.86Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
17.86Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
17.86Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
17.86Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
17.86Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
17.86Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
17.86Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
17.86Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
17.86Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
17.86Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
17.86Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
17.86Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
17.65Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
17.65Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
17.65Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
17.65Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.65Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.65Consensusbombesin_onOrthosteric Ligandbb2_on
17.65Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
17.65Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.39Single2Y00Dobutamine2Y00-β1-Dobutamine
17.39Single2Y03Isoprenaline2Y03-β1-Isoprenaline
17.39Single4JKVTaladegib4JKV-SMO-Taladegib
17.39Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
17.39Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
17.39Single5C1MBU725C1M-μ-BU72
17.39Single5JQHS-Carazolol5JQH-β2-S-Carazolol
17.39Single5N2RPSB-365N2R-A2A-PSB-36-Na
17.39Single5N2SPSB365N2S-A1-PSB36
17.39Single5WQCEMPA5WQC-OX2-EMPA
17.39Single6GPXMK08126GPX-CCR2-MK0812
17.39Single6HLPNetupitant6HLP-NK1-Netupitant
17.39Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
17.39Single6LUQHaloperidol6LUQ-D2-Haloperidol
17.39Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
17.39Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
17.39Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
17.39Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
17.39Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
17.39Single6TP6Filorexant6TP6-OX1-Filorexant
17.39Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
17.39Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
17.39Single7C4SS1P7C4S-S1P3-S1P
17.39Single7C61Ergotamine7C61-5-HT1B-Ergotamine
17.39Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
17.39Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
17.39Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
17.39Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
17.39Single7SINNPS-21437SIN-CaS-NPS-2143
17.39Single7SINNPS-21437SIN-CaS-NPS-2143
17.39Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
17.39Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
17.39Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
17.39Single7W41PD1762527W41-BB2-PD176252
17.39Single7WC6LSD7WC6-5-HT2A-LSD
17.39Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
17.39Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
17.39Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
17.39Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
17.39Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
17.39Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
17.39Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
17.39Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
17.39Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
17.39Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
17.39Single8S4DCMF-0198S4D-Apelin-CMF-019
17.39Single8TF5Oleic acid8TF5-GPR6-Oleic acid
17.39Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
17.39Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
17.39Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
17.39Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
17.39Single8ZMFA1L108ZMF-5-HT2C-A1L10
17.39Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
17.39Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
17.39Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
17.39Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
17.39Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
17.39Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
17.39Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
17.39Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
17.39Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
17.39Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
17.39Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
17.39Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
17.39Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
17.39Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
17.39Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
17.39Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
17.39Consensusa3_on_gpOrthosteric Liganda3a_on_gp
17.39Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.39Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.39Consensusadenosine_offOrthosteric Liganda1_off a2_off
17.39Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
17.39Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
17.39Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
17.39Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
17.39Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
17.39Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
17.39Consensusblt_offOrthosteric Ligandblt1_off
17.39Consensusbombesin_offOrthosteric Ligandbb2_off
17.39Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
17.39Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
17.39Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.39Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
17.39Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
17.39Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
17.24Single6PT2KGCHM076PT2-δ-KGCHM07
17.24Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
17.24Single6W25SHU91196W25-MC4-SHU9119-Ca
17.24Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
17.24Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
17.24Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
17.24Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.24Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
17.24Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
17.24Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
17.24Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
17.24Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
17.24Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
17.14Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
17.14Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
17.14Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.07Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
16.67Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
16.67Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
16.67Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
16.67Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
16.67Single5V54Methiothepin5V54-5-HT1B-Methiothepin
16.67Single5V56TC1145V56-SMO-TC114
16.67Single5V57TC1145V57-SMO-TC114
16.67Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
16.67Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
16.67Single6H7JIsoprenaline6H7J-β1-Isoprenaline
16.67Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
16.67Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
16.67Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
16.67Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
16.67Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
16.67Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
16.67Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
16.67Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
16.67Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
16.67Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
16.67Single7TUYGSK682753A7TUY-GPR183-GSK682753A
16.67Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
16.67Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
16.67Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
16.67Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
16.67Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
16.67Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
16.67Single8E0GBU728E0G-μ-BU72
16.67Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
16.67Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
16.67Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
16.67Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
16.67Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
16.67Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
16.67Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
16.67Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
16.67Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
16.67Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
16.67Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
16.67Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8XVLZibotentan8XVL-ETA-Zibotentan
16.67Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
16.67Single9AS9RS130-1809AS9-5-HT2A-RS130-180
16.67Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
16.67Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
16.67Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
16.67Single9CHUNoradrenaline9CHU-β2-Noradrenaline
16.67Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
16.67Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
16.67Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
16.67Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
16.67Consensus5ht1_offOrthosteric Ligand5ht1b_off
16.67Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
16.67Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
16.67Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
16.67Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
16.67Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
16.67Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
16.67Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
16.67Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
16.67Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
16.67Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
16.67Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
16.67Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
16.67Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
16.67Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
16.67Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
16.67Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
16.67Consensussensory_onOrthosteric Ligandopsins_on
16.22Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
16.13Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
16.13Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
16.13Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
16.13Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
16.13Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
16.13Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
16.13Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
16.13Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
16.13Single8ZRTET-18ZRT-ETB-ET-1
16.13Consensuscalcitonin_onOrthosteric Ligandctlike_on
16.13Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
16.13Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
16.13Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
16.13Consensuspac_onOrthosteric Ligandpac1_on
16.13Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.13Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
16.00Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
16.00Single4LDEBI1671074LDE-β2-BI167107
16.00Single4RWADIPP-NH24RWA-δ-DIPP-NH2
16.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
16.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
16.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
16.00Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
16.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
16.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
16.00Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
16.00Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
16.00Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
16.00Single7K15MKD0467K15-BLT1-MKD046-Na
16.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
16.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
16.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
16.00Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
16.00Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
16.00Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
16.00Single8JJ8Formoterol8JJ8-β2-Formoterol
16.00Single8JWY2-1188JWY-A2A-2-118
16.00Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
16.00Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.00Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
16.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
16.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
16.00Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
16.00Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
16.00Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
16.00Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
16.00Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
16.00Consensuslpa_offOrthosteric Ligandlpa1_off
16.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.00Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
15.79Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
15.79Single3OE6IT1t3OE6-CXCR4-IT1t
15.79Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
15.79Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
15.79Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
15.79Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
15.79Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
15.79Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.79Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
15.79Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
15.79Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.79Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
15.79Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
15.79Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
15.79Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
15.79Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
15.79Consensus5ht2_onOrthosteric Ligand5ht2b_on
15.79Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.79Consensusgi_sensoryOrthosteric Ligandgi_opsins
15.79Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
15.79Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
15.79Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.79Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
15.79Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
15.79Consensuspth_onOrthosteric Ligandpth1_on pth2_on
15.79Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
15.79Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
15.62Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.62Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
15.62Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
15.62Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
15.62Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
15.62Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
15.62Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
15.62Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
15.62Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
15.62Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
15.38Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
15.38Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
15.38Single6IBLArformoterol6IBL-β1-Arformoterol
15.38Single6K1QIRL25006K1Q-ETB-IRL2500
15.38Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
15.38Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
15.38Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
15.38Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
15.38Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
15.38Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
15.38Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
15.38Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
15.38Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
15.38Consensuscck_onOrthosteric Ligandccka_on cckb_on
15.38Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
15.38Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
15.38Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.38Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.38Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
15.38Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
15.15Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
15.15Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
15.15Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
15.15Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
15.15Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
15.15Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
15.15Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
15.15Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
15.15Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
15.15Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
15.15Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
15.15Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
15.15Single9KDFRES-701-39KDF-ETB-RES-701-3
15.15Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
15.15Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
15.15Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
15.00Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
15.00Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
15.00Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
15.00Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
15.00Single3OE9IT1t3OE9-CXCR4-IT1t
15.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
15.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
15.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
15.00Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
15.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
15.00Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
15.00Single7SRQLSD7SRQ-5-HT2B-LSD
15.00Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
15.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
15.00Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
15.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
15.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
15.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
15.00Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
15.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
15.00Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
15.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.00Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
15.00Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.00Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
15.00Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
15.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
15.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
15.00Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
15.00Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
15.00Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
15.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
15.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
15.00Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
15.00Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
15.00Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
14.81Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
14.81Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
14.81Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
14.81Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
14.81Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
14.81Single7XN9L-054,5227XN9-SST2-L-054,522
14.81Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
14.81Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
14.81Single9JF4PD1683689JF4-BB1-PD168368
14.81Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
14.81Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
14.81Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
14.81Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single6IGLIRL16206IGL-ETB-IRL1620
14.71Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
14.71Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
14.71Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
14.71Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
14.71Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
14.71Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
14.71Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
14.71Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
14.71Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
14.71Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
14.71Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
14.29Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
14.29Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
14.29Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
14.29Single3ODUIT1t3ODU-CXCR4-IT1t
14.29Single4IARErgotamine4IAR-5-HT1B-Ergotamine
14.29Single4S0VSuvorexant4S0V-OX2-Suvorexant
14.29Single4XT1Fractalkine4XT1-US28-Fractalkine
14.29Single5WS3EMPA5WS3-OX2-EMPA
14.29Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
14.29Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
14.29Single6TPJSuvorexant6TPJ-OX2-Suvorexant
14.29Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
14.29Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
14.29Single7F8XNN90567F8X-CCKA-NN9056
14.29Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
14.29Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
14.29Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
14.29Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
14.29Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
14.29Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
14.29Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
14.29Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
14.29Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
14.29Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
14.29Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
14.29Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
14.29Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
14.29Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
14.29Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
14.29Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
14.29Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
14.29Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
14.29Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
14.29Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
14.29Single8GNGIstradefylline8GNG-A2A-Istradefylline
14.29Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
14.29Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
14.29Single8KIGSHU91198KIG-MC3-SHU9119-Ca
14.29Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
14.29Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
14.29Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
14.29Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
14.29Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
14.29Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
14.29Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
14.29Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
14.29Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
14.29Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
14.29Single9H2XA1IR19H2X-A2A-A1IR1-Na
14.29Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
14.29Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
14.29Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
14.29Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
14.29Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
14.29Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
14.29Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
14.29Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
14.29Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
14.29Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
14.29Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
14.29Consensusorexin_offOrthosteric Ligandox2_off ox1_off
14.29Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
14.29Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
14.29Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
14.29Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
14.29Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
13.89Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
13.89Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
13.89Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
13.89Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
13.79Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
13.79Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
13.79Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
13.79Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
13.79Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
13.79Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
13.79Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
13.79Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
13.79Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
13.79Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
13.79Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
13.79Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
13.64Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
13.64Single3RZECidoxepin3RZE-H1-Cidoxepin
13.64Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
13.64Single5IU7Q274563465IU7-A2A-Q27456346-Na
13.64Single5JTBZM-2413855JTB-A2A-ZM-241385
13.64Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
13.64Single6A94Zotepine6A94-5-HT2A-Zotepine
13.64Single6AQFZM-2413856AQF-A2A-ZM-241385
13.64Single6KUXRS-799486KUX-α2a-RS-79948
13.64Single6MH8ZM-2413856MH8-A2A-ZM-241385
13.64Single6PS5S-Propranolol6PS5-β2-S-Propranolol
13.64Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
13.64Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
13.64Single6TP3Nemorexant6TP3-OX1-Nemorexant
13.64Single6TPKRetosiban6TPK-OT-Retosiban
13.64Single6TPNHTL66416TPN-OX2-HTL6641
13.64Single6V9SGTPL114036V9S-OX1-GTPL11403
13.64Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
13.64Single7AROLUF58337ARO-A2A-LUF5833-Na
13.64Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
13.64Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
13.64Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
13.64Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.64Single7T32ZM-2413857T32-A2A-ZM-241385
13.64Single7UL3Famotidine7UL3-H2-Famotidine
13.64Single7VODCariprazine7VOD-5-HT2A-Cariprazine
13.64Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
13.64Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
13.64Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
13.64Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
13.64Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.64Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.64Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
13.64Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
13.64Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
13.64Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
13.64Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
13.64Single8RLNLUF58348RLN-A2A-LUF5834
13.64Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
13.64Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
13.64Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
13.64Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
13.64Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.64Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.64Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
13.64Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
13.64Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
13.64Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
13.64Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
13.64Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
13.64Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
13.64Single8ZPNAMD31008ZPN-CXCR4-AMD3100
13.64Single9AS3LSD9AS3-5-HT2A-LSD
13.64Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
13.64Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
13.64Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
13.64Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
13.64Consensusa2_offOrthosteric Liganda2a_off
13.64Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
13.64Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
13.64Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
13.64Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
13.64Consensusvasop-oxy_offOrthosteric Ligandot_off
13.51Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
13.51Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
13.33Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
13.33Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
13.33Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
13.33Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
13.33Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
13.33Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
13.33Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
13.33Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.33Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
13.33Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
13.33Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
13.33Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
13.33Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
13.33Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.33Consensusangiotensin_onOrthosteric Ligandat1_on
13.33Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
13.33Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
13.33Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
13.33Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
13.33Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
13.33Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
13.04Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
13.04Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
13.04Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
13.04Single3EMLZM-2413853EML-A2A-ZM-241385
13.04Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
13.04Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
13.04Single4QIMANTA XV4QIM-SMO-ANTA XV
13.04Single5DHGC-355DHG-NOP-C-35
13.04Single5IU8Q274563475IU8-A2A-Q27456347-Na
13.04Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
13.04Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
13.04Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
13.04Single5UENDU1725UEN-A1-DU172
13.04Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
13.04Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
13.04Single6DRXLisuride6DRX-5-HT2B-Lisuride
13.04Single6GPSMK08126GPS-CCR2-MK0812
13.04Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
13.04Single6S0LZM-2413856S0L-A2A-ZM-241385
13.04Single7BU7BI1671077BU7-β1-BI167107
13.04Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
13.04Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
13.04Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
13.04Single7PYRPSB-21157PYR-A2A-PSB-2115
13.04Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
13.04Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
13.04Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
13.04Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
13.04Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
13.04Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
13.04Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
13.04Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
13.04Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
13.04Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
13.04Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
13.04Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
13.04Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
13.04Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
13.04Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
13.04Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
13.04Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
13.04Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
13.04Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
13.04Single9H37A1IR09H37-A2A-A1IR0-Na
13.04Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
13.04Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
13.04Consensus5ht5_onOrthosteric Ligand5ht5a_on
13.04Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
13.04Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
13.04Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
13.04Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
13.04Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
13.04Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
13.04Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
12.90Single6JODAngiotensin II6JOD-AT2-Angiotensin II
12.90Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
12.90Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
12.90Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
12.90Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
12.90Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
12.90Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
12.90Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
12.90Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
12.90Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
12.90Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
12.50Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
12.50Single5IUAQ274563485IUA-A2A-Q27456348-Na
12.50Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
12.50Single5TVNLSD5TVN-5-HT2B-LSD
12.50Single5WIUNemonapride5WIU-D4-Nemonapride
12.50Single5WIVNemonapride5WIV-D4-Nemonapride-Na
12.50Single5XPRBosentan5XPR-ETB-Bosentan
12.50Single6D26Fevipiprant6D26-DP2-Fevipiprant
12.50Single6E67BI1671076E67-β2-BI167107-Gs(CT)
12.50Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
12.50Single6S0QZM-2413856S0Q-A2A-ZM-241385
12.50Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
12.50Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
12.50Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
12.50Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
12.50Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
12.50Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
12.50Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
12.50Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
12.50Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
12.50Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
12.50Single8GNEKW-63568GNE-A2A-KW-6356-Na
12.50Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
12.50Single8JXSPF-61428JXS-D1-PF-6142
12.50Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
12.50Single8QOTNanobody-E8QOT-μ-Nanobody-E
12.50Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
12.50Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
12.50Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
12.50Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
12.50Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
12.50Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9EHSLUF76029EHS-A3A-LUF7602
12.50Single9HAPTolvaptan9HAP-V2-Tolvaptan
12.50Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
12.50Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.50Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.50Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
12.50Consensusdp_offOrthosteric Liganddp2_off
12.50Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
12.50Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
12.50Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
12.50Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
12.50Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
12.12Single4XT3Fractalkine4XT3-US28-Fractalkine
12.12Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
12.12Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
12.12Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
12.12Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
12.12Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
12.12Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
12.12Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
12.12Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
12.12Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
12.12Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
12.12Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
12.00Single3P0GBI1671073P0G-β2-BI167107
12.00Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
12.00Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
12.00Single6E59L-7607356E59-NK1-L-760735
12.00Single6J20Aprepitant6J20-NK1-Aprepitant
12.00Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
12.00Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
12.00Single6WGTLSD6WGT-5-HT2A-LSD
12.00Single7B6WCyclazosin7B6W-α1b-Cyclazosin
12.00Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
12.00Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.00Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
12.00Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
12.00Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
12.00Single7PX4PSB-21137PX4-A2A-PSB-2113
12.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
12.00Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
12.00Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
12.00Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
12.00Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
12.00Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
12.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
12.00Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
12.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
12.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
12.00Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
12.00Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.00Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
12.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
12.00Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
12.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
12.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
12.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
12.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
12.00Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.00Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
12.00Consensustachykinin_offOrthosteric Ligandnk1_off
11.76Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
11.76Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
11.76Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
11.76Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
11.76Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
11.76Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
11.76Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
11.76Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
11.76Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
11.76Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
11.76Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
11.76Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
11.76Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
11.54Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
11.54Single6MXTSalmeterol6MXT-β2-Salmeterol
11.54Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
11.54Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
11.54Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
11.54Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
11.54Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
11.54Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
11.54Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.54Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
11.54Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
11.54Single8JJLOlodaterol8JJL-β2-Olodaterol
11.54Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
11.54Single8JWZAB9288JWZ-A2A-AB928-Na
11.54Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
11.54Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
11.54Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
11.54Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
11.54Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
11.54Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
11.54Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
11.54Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
11.54Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
11.54Consensusorexin_onOrthosteric Ligandox2_on
11.54Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
11.54Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.54Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.43Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
11.43Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
11.43Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
11.43Consensusendothelin_onOrthosteric Ligandetb_on eta_on
11.43Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
11.11Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
11.11Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
11.11Single5GLHEndothelin-15GLH-ETB-Endothelin-1
11.11Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
11.11Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
11.11Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
11.11Single6IGKEndothelin-36IGK-ETB-Endothelin-3
11.11Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
11.11Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
11.11Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
11.11Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
11.11Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
11.11Single7UM4AS26747237UM4-5-HT5A-AS2674723
11.11Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
11.11Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
11.11Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.11Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
11.11Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
11.11Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
11.11Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
11.11Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
11.11Single8PWNTheophylline8PWN-A2A-Theophylline
11.11Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
11.11Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
11.11Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
11.11Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
11.11Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
11.11Consensuschemerin_onOrthosteric Ligandcml1_on
11.11Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
11.11Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
11.11Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
11.11Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
11.11Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
11.11Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
10.81Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
10.81Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
10.71Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
10.71Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
10.71Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
10.71Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
10.71Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
10.71Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
10.71Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
10.71Single8QJ2pN1628QJ2-MC4-pN162-Gs
10.71Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
10.71Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
10.71Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
10.71Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
10.71Single9IPYJR14a9IPY-C3aB-JR14a
10.71Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
10.71Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
10.71Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
10.71Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
10.71Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
10.53Single3OE8IT1t3OE8-CXCR4-IT1t
10.53Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
10.53Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.53Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
10.53Single8A2OTheophylline8A2O-A2A-Theophylline-Na
10.53Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
10.53Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
10.53Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
10.53Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
10.53Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
10.34Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
10.34Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
10.34Single8IEBA1LYA8IEB-GPR156-A1LYA
10.34Single8IEIA1LYA8IEI-GPR156-A1LYA
10.34Single8IEIA1LYA8IEI-GPR156-A1LYA
10.34Single8IEPA1LYA8IEP-GPR156-A1LYA
10.34Single8IEPA1LYA8IEP-GPR156-A1LYA
10.34Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
10.34Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
10.34Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
10.34Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
10.34Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
10.34Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
10.34Consensuslpl_onOrthosteric Ligands1p_on lpa_on
10.34Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
10.34Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
10.34Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
10.26Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
10.00Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
10.00Single3UZAGTPL92363UZA-A2A-GTPL9236
10.00Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
10.00Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
10.00Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
10.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
10.00Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
10.00Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
10.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
10.00Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
10.00Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
10.00Single7XNACYN1548067XNA-SST2-CYN154806
10.00Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
10.00Single8IEBA1LYA8IEB-GPR156-A1LYA
10.00Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.00Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
10.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
10.00Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
10.00Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
10.00Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
10.00Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
10.00Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
10.00Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
10.00Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
10.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
10.00Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
10.00Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
9.68Single3OE0CVX153OE0-CXCR4-CVX15
9.68Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
9.68Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
9.68Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
9.68Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
9.68Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
9.68Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
9.68Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
9.68Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
9.52Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
9.52Single3PBLEticlopride3PBL-D3-Eticlopride
9.52Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
9.52Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
9.52Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
9.52Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
9.52Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
9.52Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
9.52Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
9.52Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
9.52Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
9.52Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
9.52Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
9.52Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
9.52Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
9.52Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.52Single9AS7Psilocin9AS7-5-HT2A-Psilocin
9.52Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
9.52Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
9.52Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
9.38Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
9.38Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
9.38Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
9.38Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
9.38Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
9.38Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
9.38Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
9.38Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
9.38Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
9.38Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
9.38Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
9.38Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
9.38Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
9.38Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
9.38Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
9.38Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
9.38Consensusvasop-oxy_onOrthosteric Ligandv2_on
9.38Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
9.09Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
9.09Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
9.09Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
9.09Single3PWHZM-2413853PWH-A2A-ZM-241385
9.09Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
9.09Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
9.09Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
9.09Single4XNVBPTU4XNV-P2Y1-BPTU
9.09Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
9.09Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
9.09Single6DS0Ly2660976DS0-5-HT2B-Ly266097
9.09Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
9.09Single6ME2Ramelteon6ME2-MT1-Ramelteon
9.09Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
9.09Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
9.09Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
9.09Single7F8ULintitript7F8U-CCKA-Lintitript
9.09Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
9.09Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
9.09Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
9.09Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
9.09Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
9.09Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
9.09Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
9.09Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
9.09Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
9.09Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
9.09Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
9.09Single7XRRLemborexant7XRR-OX2-Lemborexant
9.09Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
9.09Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
9.09Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
9.09Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
9.09Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
9.09Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
9.09Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
9.09Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
9.09Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
9.09Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
9.09Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
9.09Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
9.09Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
9.09Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
9.09Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
9.09Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
8.82Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
8.82Single7SK3CXCL127SK3-ACKR3-CXCL12
8.82Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
8.82Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
8.82Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
8.82Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
8.82Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
8.70Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
8.70Single5IUBQ274563445IUB-A2A-Q27456344-Na
8.70Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
8.70Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
8.70Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
8.70Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
8.70Single5UVIZM-2413855UVI-A2A-ZM-241385
8.70Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
8.70Single6IQLL7458706IQL-D4-L745870
8.70Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
8.70Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
8.70Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
8.70Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
8.70Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
8.70Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
8.70Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
8.70Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
8.70Single9ARXSerotonin9ARX-5-HT2A-Serotonin
8.70Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
8.70Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
8.70Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
8.70Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
8.70Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
8.57Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
8.33Single2Y02Carmoterol2Y02-β1-Carmoterol
8.33Single6D27CAY104716D27-DP2-CAY10471
8.33Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
8.33Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
8.33Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
8.33Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
8.33Single7F83PF-051904577F83-Ghrelin-PF-05190457
8.33Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
8.33Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
8.33Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
8.33Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
8.33Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
8.33Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
8.33Single8IY6Endothelin-18IY6-ETB-Endothelin-1
8.33Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
8.33Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
8.33Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
8.33Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
8.33Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
8.33Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
8.33Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
8.11Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
8.11Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
8.00Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
8.00Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
8.00Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
8.00Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
8.00Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
8.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
8.00Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
8.00Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
8.00Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
8.00Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
8.00Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
7.89Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
7.69Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
7.69Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
7.69Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
7.69Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
7.69Single7R0CAVP7R0C-V2-AVP-Arrestin2
7.69Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
7.69Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
7.69Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
7.69Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
7.69Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
7.69Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
7.69Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
7.69Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
7.69Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
7.69Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
7.69Single8ZWFJR14a8ZWF-C3aB-JR14a
7.69Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
7.69Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
7.69Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
7.69Consensuslpa_onOrthosteric Ligandlpa1_on
7.69Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
7.69Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
7.50Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
7.41Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
7.41Single6OS2TRV0266OS2-AT1-TRV026
7.41Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
7.41Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
7.41Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
7.41Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
7.41Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
7.41Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
7.41Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
7.14Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
7.14Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
7.14Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8XVUCXCL28XVU-CXCR2-CXCL2
7.14Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
7.14Single8ZPLHF511168ZPL-CXCR4-HF51116
7.14Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
7.14Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
7.14Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
7.14Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
6.90Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
6.90Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
6.90Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
6.90Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
6.90Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
6.90Consensuskisspeptin_onOrthosteric Ligandkiss1_on
6.67Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
6.67Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
6.67Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
6.67Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
6.67Single8W8SAA-148W8S-GPR101-AA-14
6.67Single8WKYPG-9348WKY-MC4-PG-934
6.67Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
6.67Single8XWNCXCL88XWN-CXCR2-CXCL8
6.67Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
6.67Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
6.67Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
6.67Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
6.67Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
6.67Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
6.67Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
6.67Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
6.67Consensussomatostatin_offOrthosteric Ligandsst2_off
6.45Single7SK5CXCL127SK5-ACKR3-CXCL12
6.45Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
6.45Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
6.45Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
6.45Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
6.45Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
6.45Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
6.45Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
6.45Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
6.45Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
6.25Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
6.25Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
6.25Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
6.25Single8W8RAA-148W8R-GPR101-AA-14-chim(NtGi1-Gs)/β1/γ2
6.25Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
6.25Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
6.25Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
6.25Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
6.25Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
6.25Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
6.25Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
6.06Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
6.06Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
6.06Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
5.88Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
5.88Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
5.88Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
5.88Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
5.71Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
5.56Single5MZPCaffeine5MZP-A2A-Caffeine-Na
5.26Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
5.26Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
5.26Single7WC4Serotonin7WC4-5-HT2A-Serotonin
5.26Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
5.26Single8HS2Fab0468HS2-GPR20-Fab046
5.26Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
5.26Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
5.26Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
5.13Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
5.00Single3RFMCaffeine3RFM-A2A-Caffeine
5.00Single6TQ9SB-4081246TQ9-OX1-SB-408124
5.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
5.00Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
5.00Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
5.00Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
5.00Consensusp2y_offOrthosteric Ligandp2y1_off
4.76Single4XNWMRS25004XNW-P2Y1-MRS2500
4.76Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.76Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
4.76Single6ME5Agomelatine6ME5-MT1-Agomelatine
4.76Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
4.76Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
4.76Single7WC5Psilocin7WC5-5-HT2A-Psilocin
4.76Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
4.76Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
4.76Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
4.76Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
4.76Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
4.76Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
4.55Single4O9RCyclopamine4O9R-SMO-Cyclopamine
4.55Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
4.55Single6HLLCP999946HLL-NK1-CP99994
4.55Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
4.55Single6TP4ACT-4622066TP4-OX1-ACT-462206
4.55Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
4.55Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
4.55Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
4.55Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
4.55Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
4.55Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
4.55Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.55Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
4.55Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.55Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
4.55Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.55Consensusgq_nucleotideOrthosteric Ligandgq_p2y
4.55Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
4.35Single4BWBNeurotensin4BWB-NTS1-Neurotensin
4.35Single4K5YCP-3763954K5Y-CRF1-CP-376395
4.35Single4QINSAG1.54QIN-SMO-SAG1.5
4.35Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
4.35Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
4.35Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
4.35Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
4.35Single6ME9Ramelteon6ME9-MT2-Ramelteon
4.35Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
4.35Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
4.35Single7BR3Elagolix7BR3-GnRH1-Elagolix
4.35Single7F8YDevazepide7F8Y-CCKA-Devazepide
4.35Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
4.35Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
4.35Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
4.35Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
4.35Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
4.35Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
4.35Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
4.35Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
4.35Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
4.35Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
4.35Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
4.35Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
4.35Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
4.17Single3REYXAC3REY-A2A-XAC
4.17Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
4.17Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
4.17Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
4.17Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
4.17Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.17Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.17Single7VV6C48/807VV6-MRGPRX2-C48/80
4.17Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
4.17Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
4.17Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
4.17Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
4.17Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Consensusgrh_offOrthosteric Ligandgnrh1_off
4.00Single4Z9GCP-3763954Z9G-CRF1-CP-376395
4.00Single5T04Neurotensin5T04-NTS1-Neurotensin
4.00Single5UIGCmpd-15UIG-A2A-Cmpd-1
4.00Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
4.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
4.00Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
4.00Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.00Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
4.00Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
4.00Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
4.00Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
4.00Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
4.00Single8GTIBMK-C2058GTI-CRF1-BMK-C205
4.00Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
4.00Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
4.00Single9IYAONO-97105319IYA-GPR55-ONO-9710531
4.00Consensuscck_offOrthosteric Ligandccka_off
4.00Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
4.00Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
4.00Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
4.00Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
3.85Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
3.85Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
3.85Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.85Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
3.85Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.85Single8GTGBMK-I1528GTG-CRF1-BMK-I152
3.85Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
3.85Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
3.85Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
3.85Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
3.85Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
3.85Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
3.85Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
3.85Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
3.85Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
3.85Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
3.85Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
3.70Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
3.70Single4BV0Neurotensin4BV0-NTS1-Neurotensin
3.70Single5TZRMK86665TZR-FFA1-MK8666
3.70Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
3.70Single6OS1TRV0266OS1-AT1-TRV026
3.70Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
3.70Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
3.70Single7F1TMIP-1a7F1T-CCR5-MIP-1a
3.70Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
3.70Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
3.70Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
3.70Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
3.70Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.70Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
3.70Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
3.70Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
3.70Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
3.70Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
3.70Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
3.70Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
3.70Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
3.70Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
3.70Consensusneurotensin_onOrthosteric Ligandnts1_on
3.70Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
3.57Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
3.57Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
3.57Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
3.57Single4PY02MeSATP4PY0-P2Y12-2MeSATP
3.57Single4XEENeurotensin4XEE-NTS1-Neurotensin
3.57Single4XESNeurotensin4XES-NTS1-Neurotensin
3.57Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
3.57Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
3.57Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
3.57Single6YVRNTS8-136YVR-NTS1-NTS8-13
3.57Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
3.57Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.57Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
3.57Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
3.57Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.57Single8GTMBMK-C2038GTM-CRF1-BMK-C203
3.57Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
3.57Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
3.57Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
3.57Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
3.57Single8XQJJN2418XQJ-Apelin-JN241
3.57Single8XWACXCL18XWA-CXCR2-CXCL1
3.57Single8XWMCXCL68XWM-CXCR2-CXCL6
3.57Single8XWSCXCL58XWS-CXCR2-CXCL5
3.57Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
3.57Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
3.57Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
3.57Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
3.57Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
3.57Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
3.57Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
3.57Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
3.45Single4BUONeurotensin4BUO-NTS1-Neurotensin
3.45Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
3.45Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
3.45Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.45Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
3.45Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
3.45Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
3.45Single8XWFCXCL38XWF-CXCR2-CXCL3
3.45Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
3.45Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
3.45Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.45Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.33Single6KNMJN241-96KNM-Apelin-JN241-9
3.33Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
3.33Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
3.33Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
3.33Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
3.33Single8XQJJN2418XQJ-Apelin-JN241
3.33Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
3.33Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
3.33Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
3.23Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
3.23Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
3.23Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
3.23Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.23Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
3.23Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
3.23Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
3.23Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
3.12Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
3.12Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
2.86Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2

Consensus Members
Id Members
8XJO 8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
Net Summary
Imin 3.28
Number of Linked Nodes 876
Number of Links 1037
Number of Hubs 157
Number of Links mediated by Hubs 584
Number of Communities 25
Number of Nodes involved in Communities 205
Number of Links involved in Communities 294
Path Summary
Number Of Nodes in MetaPath 157
Number Of Links MetaPath 156
Number of Shortest Paths 40836824
Length Of Smallest Path 3
Average Path Length 64.5072
Length of Longest Path 67
Minimum Path Strength 1.3
Average Path Strength 8.53769
Maximum Path Strength 23.18
Minimum Path Correlation 0.7
Average Path Correlation 1
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.17391
Average % Of Corr. Nodes 55.6455
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 64.4905
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
prostanoid_on_gptp_on_gp
fp-alpha_on_gp



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Download tp_on_gp.zip



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