Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.36 4.779274134
2G.hns1.01 6.87014154
3G.S1.01 2.90354407
4G.s1h1.04 3.45698409
5G.H1.01 2.90367509
6G.S2.02 2.70656405
7G.S3.03 5.26132608
8G.S3.04 7.22094427
9G.S3.06 8.31906427
10G.H2.06 5.35979439
11G.H2.07 5.51052409
12G.s4h3.04 1.55865408
13G.H3.01 4.15167409
14G.H3.08 4.29948408
15G.H3.09 4.482996179
16G.H3.13 8.586464176
17G.H3.17 7.65639625
18G.S5.07 4.10687409
19G.hgh4.04 2.988335116
20G.hgh4.05 6.88617506
21G.hgh4.11 3.65427405
22G.hgh4.20 5.15771403
23G.hgh4.21 3.91865404
24G.H4.03 3.37979404
25G.H4.08 6.17323463
26G.H4.10 8.588835117
27G.H4.12 5.85948464
28G.H4.14 5.883964115
29G.H4.15 6.79448408
30G.h4s6.12 4.37708402
31G.h4s6.20 6.12448404
32G.S6.02 7.01135408
33G.S6.05 5.99808565
34G.H5.03 4.10055129
35G.H5.06 4.88764124
36G.H5.08 4.721326168
37G.H5.17 4.729255185
38G.H5.19 5.69427448
39b.1x4 2.51646408
40b.1x6 3.856564193
41b.1x9 4.362194194
42b.1x19 6.67177456
43b.l1x3 7.33325509
44b.l1x6 8.73467529
45b.b2x1 7.54117528
46b.b2x5 5.93492507
47b.l3x2 5.547835159
48b.b4x3 4.2275497
49b.b4x6 8.81625679
50b.b5x3 4.45806679
51b.b5x7 4.95896407
52b.l5x1 3.75058598
53b.l5x5 7.82535629
54b.b6x5 3.67742596
55b.b7x1 4.91975504
56b.l7x4 4.03479409
57b.b8x4 5.61219406
58b.b9x4 5.84125409
59b.l9x3 7.37927439
60b.l9x6 6.15762738
61b.b10x5 5.05625509
62b.l11x2 7.33833439
63b.b12x6 8.03525538
64b.b13x7 7.364584257
65b.l13x3 7.988335269
66b.l13x6 6.59062439
67b.b15x1 6.131675259
68b.l15x2 5.244675269
69b.b16x4 7.56052406
70b.b16x5 4.19385405
71b.b16x6 8.217755258
72b.b17x7 6.46033558
73b.l17x3 7.909246279
74b.l17x6 7.49031439
75b.b18x3 4.30667458
76b.l18x1 6.059958106
77b.l18x2 5.893854107
78b.l18x3 6.769584105
79b.b19x2 7.30062456
80b.l19x2 7.405634279
81b.b20x4 10.3675408
82b.b20x6 7.17948456
83b.b21x1 5.62146457
84b.b21x5 4.94042404
85b.b21x7 5.83583505
86b.l21x2 5.86917404
87b.l22x5 4.774755219
88b.b23x1 4.04698405
89b.b23x2 4.06104406
90b.b23x6 6.562926147
91b.l23x1 5.97448426
92b.b24x4 6.962924146
93b.b24x6 6.648854148
94b.l24x3 4.07708405
95b.l25x3 8.18225589
96b.l25x6 11.0965528
97b.l27x1 9.29202729
98b.l27x2 7.60802489
99b.b28x4 7.95687486
100b.b28x6 8.82948489
101g.ntx8 1.56844404
102g.l1x4 5.8285558
103g.h2x11 7.879484106
104g.ctx3 5.25283509
105g.ctx6 3.68198406
106g.ctx14 6.22208409
107g.ctx15 6.180424229
108g.ctx16 4.956317228
109Lig 15.11892510
110NT 135.918515
1111x36 5.43083515
1121x39 6.06475517
1131x43 6.65944617
1141x47 4.284287
1151x50 4.34146409
1161x60 5.311984297
1172x39 4.79732749
1182x47 3.86802408
1192x50 7.77382608
1202x53 6.39883508
1212x60 5.49042516
122E1 20.48781113
1233x33 7.40975517
1243x34 4.20042509
1253x35 4.93937405
1263x40 6.20844408
1273x41 4.34156406
1283x42 9.769516309
1293x46 8.45031409
1303x49 5.63583648
131I2 5.54393747
1324x50 6.881585309
1334x60 6.71433518
1344x64 6.98438418
135E2 7.43281115
136E2x51 9.74075518
1375x40 4.52094414
1385x41 9.56008516
1395x44 9.26135416
1405x58 5.25292409
1415x68 6.579584189
1426x29 2.89917405
1436x44 3.79562409
1446x51 4.60167407
145E3 5.964421014
1467x31 4.53115404
1477x35 4.67219406
1488x53 8.423134298
1498x56 4.16687407
1508x60 2.87823407
151H.hahb.04 0.708542400
152H.HB.05 1.38925500
153H.hbhc.04 1.61604600
154H.HC.06 1.58198400
155H.hchd.01 0.769833500
156H.hdhe.01 0.899167500
157H.HE.04 1.97354400
158H.HE.05 1.02658500
159G.hfs2.03 0.968854400
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1G.HN.40 b.b5x2 13.99357.41083NoNo077
2G.HN.40 b.b5x3 14.24644.735NoYes079
3b.b4x4 b.b5x3 14.87763.93708NoYes789
4b.b4x4 b.l1x3 46.490710.1633NoYes089
5b.b3x6 b.l1x3 78.732610.6329NoYes099
6b.b3x6 b.l3x2 78.85247.11583NoYes099
7G.hns1.01 b.l3x2 79.49063.30625YesYes1549
8G.S1.03 G.hns1.01 81.097512.4754NoYes094
9G.S1.03 G.S3.06 81.78334.00708NoYes097
10G.S3.06 b.l5x5 82.921316.1608YesYes279
11b.l3x1 b.l5x5 84.10414.93125NoYes299
12b.l1x6 b.l3x1 39.73127.00583YesNo299
13b.l1x6 b.l27x1 39.812916.8267YesYes299
14b.l25x6 b.l27x1 99.204721.6162YesYes289
15b.b22x1 b.l25x6 99.41175.17208NoYes288
16b.b22x1 b.b22x2 99.79883.8NoNo088
17b.b22x2 b.b26x3 99.82413.56458NoNo086
18b.b23x3 b.b26x3 99.84943.40333NoNo076
19b.b23x3 b.b27x1 99.87463.725NoNo076
20b.b27x1 g.ctx5 99.953.3525NoNo069
21b.lhb1x11 g.ctx5 99.9753.71042NoNo049
22b.b25x7 b.lhb1x11 1004.7675NoNo074
23b.b24x3 b.b25x7 33.2944.5625NoNo057
24b.b24x3 b.l25x7 33.27784.48NoNo057
25b.l25x3 b.l25x7 33.24563.57375YesNo097
26b.l25x3 b.l27x2 99.53368.29542YesYes899
27b.l25x4 b.l27x2 99.47486.65042NoYes059
28I1x49 b.l25x4 49.086110.4408NoNo075
298x53 I1x49 48.996715.6562YesNo087
308x53 I1x50 96.55444.14458YesNo2989
318x49 I1x50 96.40129.055NoNo099
322x39 8x49 95.33792.76167YesNo099
332x39 3x49 26.13553.77167YesYes498
343x49 3x53 25.53599.23042YesNo488
353x53 G.H5.19 23.975612.4808NoYes488
36G.H5.15 G.H5.19 23.30713.37167NoYes088
37G.H5.15 G.S1.02 23.07954.4175NoNo086
38b.b2x1 b.l3x1 44.49114.8879YesNo289
39b.b2x1 b.l27x1 59.42148.9225YesYes289
40b.b25x7 b.b28x6 66.731412.6233NoYes079
41b.b27x3 b.b28x6 33.24086.06208NoYes089
42b.b27x3 b.l25x3 33.22465.53542NoYes089
43b.b28x4 b.b28x6 33.45838.7YesYes869
44b.b28x4 b.l25x3 33.265912.1175YesYes869
458x56 b.l25x4 50.29534.32208YesNo075
468x53 8x56 49.10396.3YesYes087
47G.S1.02 G.S3.03 22.62427.82375NoYes068
48G.H5.08 G.S3.03 21.48523.3025YesYes088
49G.H5.08 G.H5.12 20.34515.745YesNo087
50G.H5.12 G.H5.16 19.88873.79542NoNo076
515x68 G.H5.16 19.66057.12125YesNo096
525x68 G.H5.13 11.98388.23958YesNo1898
53G.H5.13 G.S6.02 11.75736.80083NoYes088
54G.H5.10 G.S6.02 11.076412.4021NoYes078
55G.H5.10 G.S6.04 10.38619.19042NoNo079
56G.H5.06 G.S6.04 10.15597.23875YesNo049
57G.S5.06 G.S6.05 13.91824.51667NoYes085
58G.S5.04 G.S5.06 13.9945.13208NoNo098
59G.H4.15 G.S5.04 14.06976.64958YesNo089
60G.H3.09 G.H4.15 14.82416.20667YesYes098
61G.H3.09 G.S4.04 16.08744.42167YesNo099
62G.H3.08 G.S4.04 16.15275.68375YesNo089
63G.H2.04 G.H3.08 16.36517.28292NoYes098
64G.H2.04 G.H2.07 16.44236.5NoYes099
65G.H2.07 b.l9x6 16.65414.37917YesYes098
66b.b6x1 b.l9x6 24.27867.48375NoYes098
67b.b2x1 b.b6x1 24.42023.79042YesNo089
682x43 3x46 59.76611.8488NoYes099
692x39 2x43 63.76244.4175YesNo099
70b.b4x7 b.l2x5 11.358414.6429NoNo085
71b.l26x5 g.ctx4 51.76274.12208NoNo057
72g.ctx3 g.ctx4 51.23294.22625YesNo097
73g.ctx3 g.ctx6 48.82625.54208YesYes096
74b.l22x5 g.ctx6 46.70693.6925YesYes096
75b.l22x5 b.l24x2 43.25024.3025YesNo096
76b.l24x2 g.h2x12 40.85263.70167NoNo067
77b.l18x1 g.h2x12 40.5862.9675YesNo067
78b.l18x1 b.l18x3 28.03968.66083YesYes1065
79b.l18x3 b.l18x4 25.63281.62833YesNo057
80b.l14x2 b.l18x4 25.36363.38333NoNo047
81b.l14x1 b.l14x2 25.09441.63625NoNo044
82b.b18x5 b.l14x1 24.0173.29208NoNo054
83b.b15x2 b.b18x5 23.47818.74167NoNo065
84b.b15x2 b.b19x2 19.13616.5575NoYes566
85b.b17x7 b.b19x2 16.96849.15625YesYes586
86b.b17x7 b.b21x1 13.45714.97833YesYes587
87b.b21x1 g.l1x4 10.2043.67208YesYes578
88b.b22x5 b.l18x1 10.03747.94708NoYes1076
89b.b3x4 b.b4x6 31.49115.61208NoYes799
90b.b3x2 b.b4x6 62.50134.41417NoYes059
91b.b2x5 b.b3x2 62.24037.16292YesNo075
92b.l26x3 b.l26x5 51.62066.17917NoNo075
93b.l26x1 b.l26x3 51.86226.085NoNo2377
94b.b2x5 b.l26x1 52.926610.1592YesNo077
95b.l2x3 b.l2x5 11.17893.27375NoNo085
96b.b3x1 b.l2x3 10.90726.33208NoNo058
97b.b3x1 b.b6x5 10.63544.24792NoYes056
982x46 3x46 57.24376.18458NoYes099
992x46 2x50 56.80475.37875NoYes098
1002x50 3x39 55.149616.1117YesNo089
1012x53 3x39 47.16078.83833YesNo089
1021x43 2x53 24.22767.20083YesYes078
1031x43 Lig 19.94785.49708YesYes170
1042x53 3x36 20.04957.40792YesNo086
1053x36 Lig 19.82311.5754NoYes160
106b.b3x4 b.l1x3 31.8826.21625NoYes099
107b.b4x4 b.b4x6 31.487613.0671NoYes789
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x33Lig10.03291YesYes7010
3x36Lig11.57541NoYes6010
5x41Lig7.517921YesYes6010
7x34Lig5.176671NoYes5010
7x37Lig4.664171NoYes8010
1x43Lig5.497081YesYes7010
2x57Lig5.31751NoYes7010
3x32Lig3.570421NoYes6010
7x38Lig7.626251NoYes7010
E2Lig13.35831YesYes5010
7x30Lig8.38251NoYes5010
1x32Lig9.503750NoYes5010
1x35Lig4.781NoYes6010
1x36Lig8.2851YesYes5010
1x39Lig10.29871YesYes7010
2x60Lig8.549171YesYes6010
2x64Lig9.82751NoYes7010
E2x52Lig11.71421NoYes5010
2x68Lig13.420NoYes3010
1x29Lig11.00581NoYes2010
LigNT35.69461YesYes0501
E1Lig52.52131YesYes3010
NTNT311.1081YesYes5511
E1NT18.14171YesYes3511
1x357x357.865421NoYes6612
1x357x383.751NoNo6711
1x361x395.398751YesYes5711
1x361x403.9351YesNo5712
1x362x618.627921YesNo5712
1x391x434.676251YesYes7711
1x392x615.893751YesNo7712
1x397x384.056251YesNo7711
1x432x537.200831YesYes7812
1x432x546.483751YesNo7712
1x432x578.095831YesNo7711
1x437x428.002921YesNo7912
2x533x367.407920YesNo8621
2x602x617.606251YesNo6712
2x603x325.6551YesNo6611
2x66E13.376671NoYes3321
2x67E17.3650NoYes3321
E1E166.05121YesYes3311
3x25E14.257081NoYes9321
E1E2x503.322921YesNo3912
3x25E2x507.281NoNo9922
3x26E211.58871NoYes8521
3x26E2x5123.40711NoYes8822
3x293x323.177920NoNo5621
3x29E2x524.224580NoNo5521
3x334x609.506251YesYes7812
3x335x415.165831YesYes7611
3x335x435.363331YesNo7712
4x604x646.558751YesYes8822
4x605x4311.79291YesNo8722
4x644x685.19251YesNo8622
4x64E2x5112.75041YesYes8822
4x68E27.060421NoYes6521
E2E2x516.042081YesYes5812
E2E27.468751YesYes5511
5x41E215.67751YesYes6511
5x415x433.863751YesNo6712
5x415x4415.57541YesYes6612
5x44E310.18631YesYes6422
6x517x377.163750YesNo7821
E3E314.45711YesYes4422
7x30E34.282921NoYes5412
7x33E34.556671NoYes7422
7x307x343.781251NoNo5511
7x337x375.37251NoNo7821
E2NT3.536671YesYes5511
2x602x643.8051YesNo6711
3x293x336.980420NoYes5721
4x64E23.435831YesYes8521
5x40E23.323751YesYes4521
1x25Lig4.771NoYes0010
5x39E22.80NoYes3521
1x292x651.9851NoNo2412
1x241x251.980NoNo0021
3x24E11.919580NoYes3321
2x603x281.836671YesNo6712
2x69E11.496250NoYes4321
1x361x370.90751YesNo5412
3x23E10.86251NoYes3321

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusglp_onOrthosteric Ligandglp1_on glp2_on
88.00Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
84.00Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
80.77Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
80.00Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
79.31Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
79.17Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
79.17Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
78.57Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
77.78Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
76.00Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
76.00Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
75.86Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
74.07Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
74.07Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
74.07Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
73.08Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
73.08Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
73.08Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
73.08Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
72.00Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
72.00Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
70.37Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
70.37Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
69.23Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
69.23Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
69.23Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
68.97Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
67.86Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
67.86Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
66.67Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
66.67Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
66.67Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
66.67Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
66.67Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
66.67Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
65.52Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
65.38Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
65.38Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
65.38Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
65.38Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
65.38Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
64.29Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
64.29Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
64.29Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
64.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
62.96Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
62.96Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
62.07Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
61.54Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
61.29Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
60.71Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
60.71Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
58.82Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
58.82Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
58.62Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
58.33Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
58.06Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
57.14Consensuspac_onOrthosteric Ligandpac1_on
56.76Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
55.56Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
55.17Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
54.55Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
54.55Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
54.55Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
53.85Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
53.33Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
53.12Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
53.12Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
52.94Consensuspth_onOrthosteric Ligandpth1_on pth2_on
51.85Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
51.61Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
51.61Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
51.52Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
51.52Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
51.35Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
50.00Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
50.00Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
50.00Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
50.00Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
50.00Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
48.39Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
48.28Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
46.88Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
46.15Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
45.71Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
45.16Single6FJ3PTH6FJ3-PTH1-PTH
45.16Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
44.83Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
44.83Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
44.44Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
42.86Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
42.42Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
42.42Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
41.94Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
41.67Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
41.38Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
40.74Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
40.62Single4XT3Fractalkine4XT3-US28-Fractalkine
40.00Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
40.00Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
39.39Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
39.39Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
39.39Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
39.39Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
39.39Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
39.39Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
39.29Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
38.89Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
38.71Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
38.71Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
38.71Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
38.71Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
38.24Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
38.24Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
38.24Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
38.24Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
38.24Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
38.24Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
37.93Single4XT1Fractalkine4XT1-US28-Fractalkine
37.93Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
37.84Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
37.50Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
37.50Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
37.50Consensuscalcitonin_onOrthosteric Ligandctlike_on
37.50Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
37.04Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
37.04Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
36.67Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
36.36Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
36.36Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
36.36Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
36.36Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
36.36Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
36.36Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
36.36Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
36.36Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
36.36Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
36.11Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
36.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
36.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
35.71Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
35.71Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
35.29Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
35.29Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
35.29Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
35.29Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
35.00Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
34.62Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
34.62Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
34.62Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
34.48Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
34.48Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
34.38Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
34.38Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
34.38Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
34.38Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
34.38Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
34.38Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
34.29Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
34.29Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
34.21Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
34.15Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
33.33Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
33.33Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
33.33Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
33.33Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
33.33Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
33.33Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
33.33Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
33.33Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
32.43Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
32.43Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
32.35Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
32.35Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
32.35Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
32.35Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
32.26Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
32.26Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
32.26Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
32.14Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
32.14Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
32.14Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
32.14Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
32.14Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
32.14Consensuslpl_offOrthosteric Ligands1p_off lpa_off
32.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
31.58Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
31.58Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
31.43Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
31.43Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
31.43Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
31.43Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
31.43Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
31.25Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
31.25Consensusangiotensin_onOrthosteric Ligandat1_on
31.25Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
31.25Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
31.03Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
31.03Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
30.77Single7V3ZCP559407V3Z-CB1-CP55940
30.77Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
30.77Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
30.77Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
30.77Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
30.77Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
30.77Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
30.77Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
30.77Consensushca_on_gpOrthosteric Ligandhca2_on_gp
30.56Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
30.56Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
30.56Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
30.43Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
30.30Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
30.30Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
30.30Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
30.30Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
30.00Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
30.00Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
30.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
30.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
30.00Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
29.73Single6IGKEndothelin-36IGK-ETB-Endothelin-3
29.73Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
29.73Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
29.63Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
29.63Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
29.63Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
29.63Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
29.63Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
29.63Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
29.63Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
29.63Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
29.63Single9EHSLUF76029EHS-A3A-LUF7602
29.63Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
29.63Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
29.63Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
29.41Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
29.41Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
29.41Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
29.41Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
29.41Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
29.41Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.41Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
29.41Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
29.41Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
29.27Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
29.17Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
29.17Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
29.17Single8K5BNiacin8K5B-HCA2-Niacin
29.17Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
29.03Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
29.03Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
29.03Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.03Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.03Consensuslpl_onOrthosteric Ligands1p_on lpa_on
29.03Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
29.03Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.95Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
28.57Single5XR8AM8415XR8-CB1-AM841
28.57Single7TUYGSK682753A7TUY-GPR183-GSK682753A
28.57Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
28.57Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
28.57Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
28.57Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
28.57Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
28.57Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
28.21Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
28.12Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
28.12Single7XNACYN1548067XNA-SST2-CYN154806
28.12Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
28.12Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
28.12Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
28.12Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
28.12Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
28.12Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
28.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
28.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
28.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
28.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
28.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
28.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
28.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
27.78Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
27.78Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
27.78Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
27.78Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
27.78Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
27.59Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
27.59Single6OS2TRV0266OS2-AT1-TRV026
27.59Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
27.59Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
27.59Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
27.59Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
27.59Single8XYIVUF106618XYI-CXCR3-VUF10661
27.59Single9DGIZ85267113509DGI-CB1-Z8526711350
27.59Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
27.59Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
27.59Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
27.59Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
27.59Consensuslpa_offOrthosteric Ligandlpa1_off
27.59Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
27.59Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
27.27Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
27.27Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
27.27Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
27.27Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
27.03Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
26.92Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
26.92Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
26.92Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
26.92Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
26.92Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
26.92Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
26.92Single8K5CAcipimox8K5C-HCA2-Acipimox
26.92Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
26.92Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
26.92Consensushca_onOrthosteric Ligandhca2_on
26.83Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
26.67Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
26.67Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
26.67Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
26.67Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
26.67Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
26.67Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
26.67Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
26.67Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
26.67Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
26.47Single6JODAngiotensin II6JOD-AT2-Angiotensin II
26.47Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
26.47Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
26.47Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.47Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
26.47Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
26.47Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
26.47Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
26.32Single5GLHEndothelin-15GLH-ETB-Endothelin-1
26.32Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
26.32Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
26.32Consensusbombesin_onOrthosteric Ligandbb2_on
26.32Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
26.32Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.32Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
26.32Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
26.32Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
26.19Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
26.19Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
25.93Single4YAYZD-71554YAY-AT1-ZD-7155
25.93Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
25.93Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
25.93Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
25.93Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
25.93Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
25.93Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
25.93Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
25.93Single8K5DGSK2560738K5D-HCA2-GSK256073
25.93Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
25.93Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
25.93Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
25.93Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
25.93Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
25.93Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
25.81Single4UG2CGS216804UG2-A2A-CGS21680
25.81Single5ZTYAM102575ZTY-CB2-AM10257
25.81Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
25.81Single7SK9CCX6627SK9-ACKR3-CCX662
25.81Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
25.81Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
25.81Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
25.81Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
25.81Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
25.81Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
25.81Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
25.71Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
25.71Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
25.71Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
25.71Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
25.71Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
25.71Single8ZRTET-18ZRT-ETB-ET-1
25.71Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
25.71Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
25.71Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
25.71Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
25.00Single5C1MBU725C1M-μ-BU72
25.00Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
25.00Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
25.00Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
25.00Single7C4SS1P7C4S-S1P3-S1P
25.00Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
25.00Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
25.00Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
25.00Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
25.00Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
25.00Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
25.00Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
25.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
25.00Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
25.00Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
25.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
25.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
25.00Single9B9ZA1AKO9B9Z-CB1-A1AKO
25.00Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
25.00Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
25.00Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.00Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
25.00Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
25.00Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
25.00Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
25.00Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
25.00Consensussomatostatin_offOrthosteric Ligandsst2_off
24.32Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
24.32Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
24.32Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
24.32Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
24.24Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
24.24Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
24.24Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
24.24Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
24.24Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
24.24Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
24.24Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
24.24Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
24.24Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
24.14Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
24.14Single5XRAAM115425XRA-CB1-AM11542
24.14Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
24.14Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
24.14Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
24.14Single7FEECP559407FEE-CB1-CP55940-ZCZ011
24.14Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
24.14Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
24.14Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
24.14Single8E0GBU728E0G-μ-BU72
24.14Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
24.14Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
24.14Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
24.14Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
24.14Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
24.14Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
24.14Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
24.14Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
24.14Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
24.14Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
24.00Single6LI0C176LI0-GPR52-C17
24.00Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
24.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
24.00Single9B9Y7DY9B9Y-CB1-7DY
23.68Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
23.68Single8IY6Endothelin-18IY6-ETB-Endothelin-1
23.68Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
23.68Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
23.68Consensusbradykinin_onOrthosteric Ligandbk2_on
23.68Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
23.68Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
23.68Consensusendothelin_onOrthosteric Ligandetb_on eta_on
23.68Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
23.53Single6W25SHU91196W25-MC4-SHU9119-Ca
23.53Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
23.53Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
23.53Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
23.53Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
23.53Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
23.53Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
23.53Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
23.53Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
23.53Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
23.53Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
23.53Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
23.53Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
23.53Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
23.53Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
23.33Single4XEENeurotensin4XEE-NTS1-Neurotensin
23.33Single4XESNeurotensin4XES-NTS1-Neurotensin
23.33Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
23.33Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
23.33Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
23.33Single6KQICP559406KQI-CB1-CP55940-Org27569
23.33Single6YVRNTS8-136YVR-NTS1-NTS8-13
23.33Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
23.33Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
23.33Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
23.33Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
23.33Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
23.33Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
23.33Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
23.33Single8JWY2-1188JWY-A2A-2-118
23.33Single8JWZAB9288JWZ-A2A-AB928-Na
23.33Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
23.33Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
23.33Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
23.33Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
23.33Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
23.33Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
23.33Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
23.33Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
23.08Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
23.08Single4BWBNeurotensin4BWB-NTS1-Neurotensin
23.08Single5U09Taranabant5U09-CB1-Taranabant
23.08Single5ZKQABT-4915ZKQ-PAF-ABT-491
23.08Single6AKXA4R6AKX-CCR5-A4R
23.08Single6AKYMaraviroc6AKY-CCR5-Maraviroc
23.08Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
23.08Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
23.08Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
23.08Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
23.08Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
23.08Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
23.08Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
23.08Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
23.08Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
23.08Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
23.08Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
23.08Consensusangiotensin_offOrthosteric Ligandat1_off
23.08Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
23.08Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
23.08Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
22.92Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
22.86Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
22.86Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
22.86Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
22.86Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
22.86Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
22.86Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
22.86Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
22.86Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.86Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
22.86Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
22.86Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.86Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.86Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
22.86Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
22.86Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
22.86Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
22.86Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
22.86Consensusvasop-oxy_onOrthosteric Ligandv2_on
22.86Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
22.58Single4BUONeurotensin4BUO-NTS1-Neurotensin
22.58Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
22.58Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
22.58Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
22.58Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
22.58Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
22.58Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
22.58Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
22.58Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
22.58Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
22.58Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
22.58Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
22.58Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
22.58Consensuscck_onOrthosteric Ligandccka_on cckb_on
22.58Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
22.58Consensuschemerin_onOrthosteric Ligandcml1_on
22.58Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
22.58Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.58Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.58Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
22.58Consensusprostanoid_offOrthosteric Ligandep_off dp_off
22.58Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
22.58Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
22.58Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
22.50Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
22.50Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
22.50Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
22.22Single4MBSMaraviroc4MBS-CCR5-Maraviroc
22.22Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
22.22Single7F61PF-036547467F61-H3-PF-03654746
22.22Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
22.22Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
22.22Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
22.22Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
22.22Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
22.22Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
22.22Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
22.22Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
22.22Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
22.22Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
22.22Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
22.22Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
22.22Single8RLNLUF58348RLN-A2A-LUF5834
22.22Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
22.22Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.22Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
22.22Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
22.22Single9BA0A1AKN9BA0-CB1-A1AKN
22.22Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
22.22Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
22.22Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
22.22Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
22.22Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
22.22Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
22.22Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
22.22Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
22.22Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
21.88Single3NY9ICI118-5513NY9-β2-ICI118-551
21.88Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
21.88Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
21.88Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
21.88Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.88Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
21.88Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
21.88Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
21.88Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
21.88Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
21.88Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.88Single8QJ2pN1628QJ2-MC4-pN162-Gs
21.88Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
21.88Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
21.88Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
21.88Single9IPYJR14a9IPY-C3aB-JR14a
21.88Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
21.88Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
21.74Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
21.74Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
21.62Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
21.62Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
21.62Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
21.62Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
21.62Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
21.62Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
21.43Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
21.43Single5UENDU1725UEN-A1-DU172
21.43Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
21.43Single6PS1Timolol6PS1-β2-Timolol
21.43Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
21.43Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
21.43Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
21.43Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
21.43Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
21.43Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
21.43Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
21.43Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
21.43Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
21.43Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
21.43Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
21.43Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
21.43Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
21.43Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
21.43Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.43Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.43Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.43Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
21.43Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
21.43Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
21.43Single9CHXS-Carazolol9CHX-β2-S-Carazolol
21.43Consensusa3_onOrthosteric Liganda3a_on
21.43Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
21.43Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
21.43Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
21.21Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
21.21Single7QA8Peptide7QA8-STE2-Peptide
21.21Single7QA8Peptide7QA8-STE2-Peptide
21.21Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
21.21Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
21.21Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
21.21Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
21.21Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
21.21Single8WDTphotoNECA8WDT-A2A-photoNECA
21.21Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.21Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
21.21Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
21.21Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
21.21Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
21.05Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
21.05Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
20.69Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
20.69Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
20.69Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
20.69Single6D26Fevipiprant6D26-DP2-Fevipiprant
20.69Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
20.69Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
20.69Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
20.69Single7C61Ergotamine7C61-5-HT1B-Ergotamine
20.69Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
20.69Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
20.69Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
20.69Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
20.69Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
20.69Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
20.69Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
20.69Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
20.69Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
20.69Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.69Single8JXSPF-61428JXS-D1-PF-6142
20.69Single8S4DCMF-0198S4D-Apelin-CMF-019
20.69Single8TF5Oleic acid8TF5-GPR6-Oleic acid
20.69Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
20.69Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.69Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.69Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
20.69Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
20.69Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
20.69Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
20.69Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
20.69Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
20.69Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
20.69Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
20.69Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
20.69Consensusa3_on_gpOrthosteric Liganda3a_on_gp
20.69Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
20.69Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
20.69Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
20.69Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
20.69Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
20.69Consensusdp_offOrthosteric Liganddp2_off
20.69Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
20.69Consensusep_offOrthosteric Ligandep4_off
20.69Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
20.69Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
20.69Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
20.69Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.69Consensustrace-amine_onOrthosteric Ligandta1_on
20.59Single3QAKUK-4320973QAK-A2A-UK-432097
20.59Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
20.59Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
20.59Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
20.59Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
20.59Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
20.59Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
20.59Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
20.59Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
20.59Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
20.59Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
20.59Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
20.59Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
20.59Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
20.59Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
20.59Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
20.59Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
20.59Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
20.59Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
20.51Single6IGLIRL16206IGL-ETB-IRL1620
20.51Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
20.51Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
20.51Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
20.51Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
20.00Single2YDVNECA2YDV-A2A-NECA
20.00Single3OE0CVX153OE0-CXCR4-CVX15
20.00Single3P0GBI1671073P0G-β2-BI167107
20.00Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
20.00Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
20.00Single4BV0Neurotensin4BV0-NTS1-Neurotensin
20.00Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
20.00Single4UHRCGS216804UHR-A2A-CGS21680
20.00Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
20.00Single5G53NECA5G53-A2A-NECA-Gs
20.00Single5WF5UK-4320975WF5-A2A-UK-432097
20.00Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
20.00Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
20.00Single6OS1TRV0266OS1-AT1-TRV026
20.00Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
20.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
20.00Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
20.00Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
20.00Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
20.00Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
20.00Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
20.00Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
20.00Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
20.00Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
20.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
20.00Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
20.00Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
20.00Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
20.00Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
20.00Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
20.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
20.00Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
20.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
20.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
20.00Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
20.00Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
20.00Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
20.00Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
20.00Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
20.00Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
20.00Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
20.00Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
20.00Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
20.00Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.00Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
20.00Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
20.00Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
20.00Single8ZWFJR14a8ZWF-C3aB-JR14a
20.00Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
20.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
20.00Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
20.00Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusa2_onOrthosteric Liganda2b_on
20.00Consensusa2_on_gpOrthosteric Liganda2b_on_gp
20.00Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
20.00Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
20.00Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
20.00Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
20.00Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
20.00Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
20.00Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
20.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
20.00Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
20.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
20.00Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
20.00Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
20.00Consensuslpa_onOrthosteric Ligandlpa1_on
20.00Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
20.00Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusneurotensin_onOrthosteric Ligandnts1_on
20.00Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.00Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
20.00Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
19.51Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
19.44Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
19.44Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
19.35Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
19.35Single6A93Risperidone6A93-5-HT2A-Risperidone
19.35Single6IIURamatroban6IIU-TXA2-Ramatroban
19.35Single6MXTSalmeterol6MXT-β2-Salmeterol
19.35Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
19.35Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
19.35Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
19.35Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
19.35Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
19.35Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
19.35Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
19.35Single7YITNalfurafine7YIT-κ-Nalfurafine
19.35Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
19.35Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
19.35Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single8JJ8Formoterol8JJ8-β2-Formoterol
19.35Single8JJLOlodaterol8JJL-β2-Olodaterol
19.35Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
19.35Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
19.35Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
19.35Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
19.35Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
19.35Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
19.35Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
19.35Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
19.35Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
19.35Consensusalpha1_offOrthosteric Ligandalpha1a_off
19.35Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
19.35Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
19.35Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
19.35Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
19.35Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
19.35Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
19.35Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
19.35Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
19.35Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
19.35Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
19.35Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
19.35Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
19.35Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
19.35Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
19.35Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
19.23Single3OE9IT1t3OE9-CXCR4-IT1t
19.23Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
19.23Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
19.23Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
19.23Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
19.23Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
19.23Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
19.23Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
18.92Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
18.92Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
18.92Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
18.92Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
18.92Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
18.92Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
18.75Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
18.75Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
18.75Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
18.75Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
18.75Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
18.75Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
18.75Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
18.75Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
18.75Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
18.75Single7EZCUKA7EZC-A2A-UKA
18.75Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
18.75Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
18.75Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
18.75Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
18.75Single7UM4AS26747237UM4-5-HT5A-AS2674723
18.75Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
18.75Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
18.75Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
18.75Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
18.75Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
18.75Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
18.75Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.75Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
18.75Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
18.75Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
18.75Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
18.75Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
18.75Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
18.75Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
18.75Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
18.52Single3PWHZM-2413853PWH-A2A-ZM-241385
18.52Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
18.52Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
18.52Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
18.52Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
18.52Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
18.52Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
18.52Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
18.52Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
18.52Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
18.52Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
18.52Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
18.52Single8GNGIstradefylline8GNG-A2A-Istradefylline
18.52Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
18.52Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
18.52Single8IWESpermidine8IWE-TA9-Spermidine
18.52Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
18.52Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
18.52Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
18.52Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
18.52Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
18.52Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
18.52Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
18.52Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
18.52Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
18.52Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
18.52Consensusalpha2_offOrthosteric Ligandalpha2c_off
18.42Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
18.42Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
18.42Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
18.42Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
18.42Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
18.42Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
18.42Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
18.42Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
18.18Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
18.18Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
18.18Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
18.18Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
18.18Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
18.18Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
18.18Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
18.18Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
18.18Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
18.18Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
18.18Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
18.18Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.95Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
17.95Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
17.86Single2YDOAdenosine2YDO-A2A-Adenosine
17.86Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
17.86Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
17.86Single6PS0S-Carazolol6PS0-β2-S-Carazolol
17.86Single6PS4ICI118-5516PS4-β2-ICI118-551
17.86Single6PS5S-Propranolol6PS5-β2-S-Propranolol
17.86Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
17.86Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
17.86Single7AROLUF58337ARO-A2A-LUF5833-Na
17.86Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
17.86Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
17.86Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Single7T32ZM-2413857T32-A2A-ZM-241385
17.86Single7UL3Famotidine7UL3-H2-Famotidine
17.86Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
17.86Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
17.86Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
17.86Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
17.86Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
17.86Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
17.86Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
17.86Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
17.86Single8IHKAcifran8IHK-HCA3-Acifran
17.86Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
17.86Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
17.86Single8K2WAMG4878K2W-CXCR3-AMG487
17.86Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
17.86Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
17.86Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
17.86Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
17.86Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
17.86Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
17.86Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
17.86Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
17.86Single8ZPMAMD0708ZPM-CXCR4-AMD070
17.86Single9AS5Mescaline9AS5-5-HT2A-Mescaline
17.86Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
17.86Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
17.86Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
17.86Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
17.86Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
17.86Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
17.86Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
17.86Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
17.65Single4IARErgotamine4IAR-5-HT1B-Ergotamine
17.65Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
17.65Single7F8XNN90567F8X-CCKA-NN9056
17.65Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
17.65Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
17.65Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
17.65Single8KIGSHU91198KIG-MC3-SHU9119-Ca
17.65Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
17.65Single8WKYPG-9348WKY-MC4-PG-934
17.65Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.65Single9M4TSilodosin9M4T-Alpha1A-Silodosin
17.65Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
17.65Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
17.50Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
17.50Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
17.39Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single2Y04Salbutamol2Y04-β1-Salbutamol
17.24Single3NY8ICI118-5513NY8-β2-ICI118-551
17.24Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
17.24Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
17.24Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
17.24Single4GBRS-Carazolol4GBR-β2-S-Carazolol
17.24Single4QKX35V4QKX-β2-35V
17.24Single5DHHSB-6121115DHH-NOP-SB-612111
17.24Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
17.24Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
17.24Single5T04Neurotensin5T04-NTS1-Neurotensin
17.24Single5TGZAM65385TGZ-CB1-AM6538
17.24Single5UIGCmpd-15UIG-A2A-Cmpd-1
17.24Single6D27CAY104716D27-DP2-CAY10471
17.24Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
17.24Single6GPSMK08126GPS-CCR2-MK0812
17.24Single6H7MSalbutamol6H7M-β1-Salbutamol
17.24Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
17.24Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
17.24Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
17.24Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
17.24Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
17.24Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
17.24Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
17.24Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
17.24Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
17.24Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
17.24Single7UL4Alvimopan7UL4-μ-Alvimopan
17.24Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
17.24Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
17.24Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
17.24Single7WC7Lisuride7WC7-5-HT2A-Lisuride
17.24Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
17.24Single7YXAONO-54306087YXA-S1P5-ONO-5430608
17.24Single8CU6LJ-45178CU6-A2A-LJ-4517
17.24Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
17.24Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
17.24Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
17.24Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
17.24Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
17.24Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
17.24Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
17.24Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
17.24Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
17.24Single8JJOAlprenolol8JJO-β2-Alprenolol
17.24Single8JXRLSD8JXR-D1-LSD
17.24Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
17.24Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
17.24Single8T1WCVN4248T1W-GPR6-CVN424
17.24Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
17.24Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
17.24Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
17.24Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
17.24Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
17.24Single9AS1DMT9AS1-5-HT2A-DMT
17.24Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
17.24Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
17.24Single9H37A1IR09H37-A2A-A1IR0-Na
17.24Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
17.24Consensus5ht5_onOrthosteric Ligand5ht5a_on
17.24Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
17.24Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
17.24Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
17.24Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
17.24Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
17.24Consensusblt_onOrthosteric Ligandblt1_on
17.24Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
17.24Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
17.24Consensusdopamine_offOrthosteric Ligandd2_off d3_off
17.24Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
17.24Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
17.24Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
17.24Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
17.24Consensusleukotriene_onOrthosteric Ligandblt_on
17.24Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
17.24Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
17.14Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
17.14Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
17.14Single7SK5CXCL127SK5-ACKR3-CXCL12
17.14Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
17.14Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
17.07Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
16.67Single2RH1S-Carazolol2RH1-β2-S-Carazolol
16.67Single2Y03Isoprenaline2Y03-β1-Isoprenaline
16.67Single2YCWS-Carazolol2YCW-β1-S-Carazolol
16.67Single4JKVTaladegib4JKV-SMO-Taladegib
16.67Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
16.67Single5D6LS-Carazolol5D6L-β2-S-Carazolol
16.67Single5JQHS-Carazolol5JQH-β2-S-Carazolol
16.67Single5N2RPSB-365N2R-A2A-PSB-36-Na
16.67Single5N2SPSB365N2S-A1-PSB36
16.67Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
16.67Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
16.67Single5TVNLSD5TVN-5-HT2B-LSD
16.67Single5WIUNemonapride5WIU-D4-Nemonapride
16.67Single5WIVNemonapride5WIV-D4-Nemonapride-Na
16.67Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
16.67Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
16.67Single6E67BI1671076E67-β2-BI167107-Gs(CT)
16.67Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
16.67Single6GPXMK08126GPX-CCR2-MK0812
16.67Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
16.67Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
16.67Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
16.67Single6PS6Timolol6PS6-β2-Timolol
16.67Single6PT2KGCHM076PT2-δ-KGCHM07
16.67Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
16.67Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
16.67Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
16.67Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
16.67Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
16.67Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
16.67Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
16.67Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
16.67Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
16.67Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
16.67Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
16.67Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
16.67Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
16.67Single8HS2Fab0468HS2-GPR20-Fab046
16.67Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
16.67Single8QOTNanobody-E8QOT-μ-Nanobody-E
16.67Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
16.67Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
16.67Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
16.67Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
16.67Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
16.67Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
16.67Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
16.67Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
16.67Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
16.67Consensusadenosine_offOrthosteric Liganda1_off a2_off
16.67Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
16.67Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
16.67Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
16.67Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
16.67Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
16.67Consensusamine_offonOrthosteric Ligandamine_off amine_on
16.67Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
16.67Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
16.67Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
16.67Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
16.67Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
16.67Consensusblt_offOrthosteric Ligandblt1_off
16.67Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
16.67Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
16.67Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
16.67Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
16.67Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.67Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.67Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
16.67Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
16.22Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
16.22Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
16.22Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
16.22Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
16.13Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
16.13Single4DJHJDTic4DJH-κ-JDTic
16.13Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
16.13Single5D5AS-Carazolol5D5A-β2-S-Carazolol
16.13Single5D5BS-Carazolol5D5B-β2-S-Carazolol
16.13Single5V56TC1145V56-SMO-TC114
16.13Single5V57TC1145V57-SMO-TC114
16.13Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
16.13Single6H7JIsoprenaline6H7J-β1-Isoprenaline
16.13Single6J21Aprepitant6J21-NK1-Aprepitant
16.13Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
16.13Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
16.13Single6TQ7SB-3348676TQ7-OX1-SB-334867
16.13Single6WGTLSD6WGT-5-HT2A-LSD
16.13Single7B6WCyclazosin7B6W-α1b-Cyclazosin
16.13Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
16.13Single7F1TMIP-1a7F1T-CCR5-MIP-1a
16.13Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
16.13Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
16.13Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
16.13Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
16.13Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
16.13Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
16.13Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
16.13Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
16.13Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
16.13Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
16.13Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
16.13Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
16.13Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
16.13Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
16.13Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
16.13Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
16.13Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.13Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
16.13Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
16.13Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
16.13Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
16.13Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
16.13Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.13Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
16.13Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
16.13Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
16.13Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
16.13Single9BJKNaloxone9BJK-μ-Naloxone-NAM
16.13Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
16.13Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
16.13Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
16.13Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
16.13Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
16.13Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
16.13Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.13Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
16.13Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
16.13Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
16.13Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
16.13Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
16.13Consensusrelaxin_onOrthosteric Ligandrxfp4_on
16.13Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
16.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
16.00Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
16.00Single9CHUNoradrenaline9CHU-β2-Noradrenaline
16.00Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
15.79Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
15.79Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
15.79Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
15.79Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
15.62Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
15.62Single3D4STimolol3D4S-β2-Timolol
15.62Single4AMIBucindolol4AMI-β1-Bucindolol
15.62Single4LDEBI1671074LDE-β2-BI167107
15.62Single4N4WSANT-14N4W-SMO-SANT-1
15.62Single4RWADIPP-NH24RWA-δ-DIPP-NH2
15.62Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
15.62Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
15.62Single6CM4Risperidone6CM4-D2-Risperidone
15.62Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
15.62Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
15.62Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
15.62Single6ZG4HTL00099366ZG4-M1-HTL0009936
15.62Single7DFPSpiperone7DFP-D2-Spiperone
15.62Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
15.62Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
15.62Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
15.62Single7K15MKD0467K15-BLT1-MKD046-Na
15.62Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
15.62Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
15.62Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
15.62Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
15.62Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
15.62Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.62Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
15.62Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
15.62Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
15.62Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
15.62Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
15.62Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
15.62Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
15.62Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
15.62Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
15.62Single9BJKNAM9BJK-μ-Naloxone-NAM
15.62Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
15.62Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
15.62Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
15.62Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
15.62Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
15.62Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
15.62Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
15.62Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
15.62Consensusorexin_onOrthosteric Ligandox2_on
15.62Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.62Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Single3OE6IT1t3OE6-CXCR4-IT1t
15.38Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
15.38Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
15.38Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
15.38Single7SK3CXCL127SK3-ACKR3-CXCL12
15.38Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
15.38Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
15.38Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
15.38Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
15.38Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
15.38Single9LRCHistamine9LRC-H4-Histamine
15.38Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
15.38Consensus5ht2_onOrthosteric Ligand5ht2b_on
15.38Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
15.38Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
15.15Single5X93K-87945X93-ETB-K-8794
15.15Single6H7LDobutamine6H7L-β1-Dobutamine
15.15Single6IBLArformoterol6IBL-β1-Arformoterol
15.15Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
15.15Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.15Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
15.15Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
15.15Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
15.15Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
15.15Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
15.15Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
15.15Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
15.15Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
15.15Single8XVUCXCL28XVU-CXCR2-CXCL2
15.15Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
15.15Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
15.15Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
15.15Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
15.15Consensusendothelin_offOrthosteric Ligandetb_off
15.15Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
15.15Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
15.00Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
15.00Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
15.00Single9KDFRES-701-39KDF-ETB-RES-701-3
14.81Single7SRQLSD7SRQ-5-HT2B-LSD
14.81Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
14.81Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
14.81Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
14.81Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
14.81Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
14.81Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
14.81Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
14.81Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
14.81Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
14.81Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
14.81Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
14.81Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
14.81Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
14.81Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
14.81Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
14.81Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
14.81Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
14.81Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
14.81Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
14.81Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
14.81Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
14.81Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
14.81Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
14.81Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
14.81Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
14.81Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
14.81Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
14.81Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
14.81Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
14.71Single5WF6UK-4320975WF6-A2A-UK-432097
14.71Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
14.71Single6PT3DPI-2876PT3-δ-DPI-287
14.71Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
14.71Single7XN9L-054,5227XN9-SST2-L-054,522
14.71Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
14.71Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
14.71Single8X5YAstemizole8X5Y-H1-Astemizole
14.71Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
14.71Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
14.71Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
14.71Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
14.71Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
14.29Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
14.29Single3ODUIT1t3ODU-CXCR4-IT1t
14.29Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
14.29Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
14.29Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
14.29Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
14.29Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
14.29Single6B73MP11046B73-κ-MP1104
14.29Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
14.29Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
14.29Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
14.29Single6ME2Ramelteon6ME2-MT1-Ramelteon
14.29Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
14.29Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
14.29Single7BR3Elagolix7BR3-GnRH1-Elagolix
14.29Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
14.29Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
14.29Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
14.29Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
14.29Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
14.29Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.29Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.29Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
14.29Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
14.29Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
14.29Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
14.29Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
14.29Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
14.29Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
14.29Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
14.29Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
14.29Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
14.29Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
14.29Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
14.29Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
14.29Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
14.29Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
14.29Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
14.29Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
14.29Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.29Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
14.29Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
14.29Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
14.29Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
14.29Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
14.29Single8XWNCXCL88XWN-CXCR2-CXCL8
14.29Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
14.29Single8Y0HVUF114188Y0H-CXCR3-VUF11418
14.29Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
14.29Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
14.29Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
14.29Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
14.29Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
14.29Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
14.29Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
14.29Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
14.29Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
14.29Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
14.29Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
14.29Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
14.29Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
14.29Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
14.29Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
14.29Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
14.29Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
14.29Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
14.29Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
14.29Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
14.29Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
14.29Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.29Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
14.29Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusorexin_offOrthosteric Ligandox2_off ox1_off
14.29Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
14.29Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
13.89Single6HLOAprepitant6HLO-NK1-Aprepitant
13.89Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
13.89Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
13.89Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
13.89Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
13.89Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
13.89Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
13.89Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
13.79Single3REYXAC3REY-A2A-XAC
13.79Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
13.79Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
13.79Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
13.79Single4ZJCSB-6740424ZJC-OX1-SB-674042
13.79Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
13.79Single5IU7Q274563465IU7-A2A-Q27456346-Na
13.79Single5IUBQ274563445IUB-A2A-Q27456344-Na
13.79Single5JTBZM-2413855JTB-A2A-ZM-241385
13.79Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
13.79Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
13.79Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
13.79Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
13.79Single6A94Zotepine6A94-5-HT2A-Zotepine
13.79Single6AQFZM-2413856AQF-A2A-ZM-241385
13.79Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
13.79Single6KUXRS-799486KUX-α2a-RS-79948
13.79Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
13.79Single6MH8ZM-2413856MH8-A2A-ZM-241385
13.79Single6TPGEMPA6TPG-OX2-EMPA
13.79Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
13.79Single6V9SGTPL114036V9S-OX1-GTPL11403
13.79Single6VI4JDTic6VI4-κ-JDTic
13.79Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
13.79Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
13.79Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
13.79Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
13.79Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
13.79Single6ZG9GSK10347026ZG9-M1-GSK1034702
13.79Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
13.79Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
13.79Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
13.79Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
13.79Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
13.79Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
13.79Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
13.79Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
13.79Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
13.79Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
13.79Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
13.79Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
13.79Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
13.79Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
13.79Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
13.79Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
13.79Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
13.79Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
13.79Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
13.79Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8ZPNAMD31008ZPN-CXCR4-AMD3100
13.79Single9AS3LSD9AS3-5-HT2A-LSD
13.79Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
13.79Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
13.79Consensusa2_offOrthosteric Liganda2a_off
13.79Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
13.79Consensusalpha1_onOrthosteric Ligandalpha1a_on
13.79Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
13.79Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
13.79Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
13.79Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
13.79Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
13.79Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
13.79Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
13.79Consensusgrh_offOrthosteric Ligandgnrh1_off
13.79Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
13.51Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.51Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
13.51Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
13.51Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.51Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.51Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.33Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
13.33Single2Y01Dobutamine2Y01-β1-Dobutamine
13.33Single2Y02Carmoterol2Y02-β1-Carmoterol
13.33Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
13.33Single3EMLZM-2413853EML-A2A-ZM-241385
13.33Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
13.33Single4DAJTiotropium4DAJ-M3-Tiotropium
13.33Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
13.33Single4EJ4Naltrindole4EJ4-δ-Naltrindole
13.33Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
13.33Single4MQSIperoxo4MQS-M2-Iperoxo
13.33Single4QIMANTA XV4QIM-SMO-ANTA XV
13.33Single4U14Tiotropium4U14-M3-Tiotropium
13.33Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
13.33Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
13.33Single5DHGC-355DHG-NOP-C-35
13.33Single5IU8Q274563475IU8-A2A-Q27456347-Na
13.33Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
13.33Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
13.33Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
13.33Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
13.33Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
13.33Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
13.33Single6DRXLisuride6DRX-5-HT2B-Lisuride
13.33Single6IIVDaltroban6IIV-TXA2-Daltroban
13.33Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
13.33Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
13.33Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
13.33Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
13.33Single6S0LZM-2413856S0L-A2A-ZM-241385
13.33Single6TOTLemborexant6TOT-OX1-Lemborexant
13.33Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
13.33Single7BU7BI1671077BU7-β1-BI167107
13.33Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
13.33Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
13.33Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
13.33Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
13.33Single7PYRPSB-21157PYR-A2A-PSB-2115
13.33Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
13.33Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
13.33Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
13.33Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
13.33Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
13.33Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
13.33Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
13.33Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
13.33Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
13.33Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
13.33Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
13.33Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
13.33Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
13.33Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
13.33Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
13.33Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
13.33Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
13.33Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
13.33Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
13.33Single8X63Mepyramine8X63-H1-Mepyramine
13.33Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
13.33Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
13.33Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
13.33Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
13.33Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
13.33Single9JEAAtropine9JEA-M1-Atropine
13.33Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
13.33Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
13.33Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
13.33Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
13.33Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
13.33Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
13.33Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
13.33Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
13.33Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
13.33Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
13.33Consensusalpha2_onOrthosteric Ligandalpha2b_on
13.33Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
13.33Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
13.33Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
13.33Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
13.33Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
13.33Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
13.33Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
13.33Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
13.33Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
13.33Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
13.33Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
13.33Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
13.33Consensushistamine_offOrthosteric Ligandh1_off
13.33Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
13.33Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
13.16Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
13.16Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
13.16Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
13.16Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
12.90Single2Y00Dobutamine2Y00-β1-Dobutamine
12.90Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
12.90Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
12.90Single5IUAQ274563485IUA-A2A-Q27456348-Na
12.90Single5WQCEMPA5WQC-OX2-EMPA
12.90Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
12.90Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
12.90Single6LUQHaloperidol6LUQ-D2-Haloperidol
12.90Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
12.90Single6S0QZM-2413856S0Q-A2A-ZM-241385
12.90Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
12.90Single6TP6Filorexant6TP6-OX1-Filorexant
12.90Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
12.90Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
12.90Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
12.90Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
12.90Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
12.90Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
12.90Single7W41PD1762527W41-BB2-PD176252
12.90Single7WC6LSD7WC6-5-HT2A-LSD
12.90Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
12.90Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
12.90Single8GNEKW-63568GNE-A2A-KW-6356-Na
12.90Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
12.90Single8ZMFA1L108ZMF-5-HT2C-A1L10
12.90Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
12.90Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
12.90Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
12.90Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
12.90Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
12.90Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
12.90Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
12.90Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.90Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.90Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
12.90Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
12.90Consensusbombesin_offOrthosteric Ligandbb2_off
12.90Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
12.90Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
12.90Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
12.90Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
12.90Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
12.90Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
12.90Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
12.90Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.82Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
12.50Single4U15Tiotropium4U15-M3-Tiotropium
12.50Single5V54Methiothepin5V54-5-HT1B-Methiothepin
12.50Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
12.50Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
12.50Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
12.50Single6J20Aprepitant6J20-NK1-Aprepitant
12.50Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
12.50Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
12.50Single6OL9Tiotropium6OL9-M5-Tiotropium
12.50Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
12.50Single7PX4PSB-21137PX4-A2A-PSB-2113
12.50Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
12.50Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
12.50Single8EA0Iperoxo8EA0-M3-Iperoxo
12.50Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
12.50Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
12.50Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
12.50Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
12.50Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
12.50Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
12.50Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
12.50Consensus5ht1_offOrthosteric Ligand5ht1b_off
12.50Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
12.50Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
12.50Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.50Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
12.50Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
12.50Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
12.50Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
12.50Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
12.50Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
12.12Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
12.12Single5CXVTiotropium5CXV-M1-Tiotropium
12.12Single5X33BIIL2605X33-BLT1-BIIL260
12.12Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
12.12Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
12.12Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single8XQJJN2418XQJ-Apelin-JN241
12.12Single8XWMCXCL68XWM-CXCR2-CXCL6
12.12Single8XWSCXCL58XWS-CXCR2-CXCL5
12.12Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
12.12Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.12Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
12.12Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
12.12Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
12.00Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
12.00Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
12.00Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
12.00Single8PWNTheophylline8PWN-A2A-Theophylline
12.00Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.00Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.76Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
11.76Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
11.76Single6K1QIRL25006K1Q-ETB-IRL2500
11.76Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
11.76Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
11.76Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
11.76Single8XVJMacitentan8XVJ-ETA-Macitentan
11.76Single8XWFCXCL38XWF-CXCR2-CXCL3
11.76Single8ZPLHF511168ZPL-CXCR4-HF51116
11.76Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
11.76Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
11.54Single3OE8IT1t3OE8-CXCR4-IT1t
11.54Single3RFMCaffeine3RFM-A2A-Caffeine
11.54Single6TQ9SB-4081246TQ9-OX1-SB-408124
11.54Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
11.54Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
11.54Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
11.54Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
11.54Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
11.54Consensusp2y_offOrthosteric Ligandp2y1_off
11.43Single6KNMJN241-96KNM-Apelin-JN241-9
11.43Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
11.43Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
11.43Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
11.43Single8XQJJN2418XQJ-Apelin-JN241
11.43Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
11.43Single9JF4PD1683689JF4-BB1-PD168368
11.11Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
11.11Single4XNWMRS25004XNW-P2Y1-MRS2500
11.11Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
11.11Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
11.11Single6ME5Agomelatine6ME5-MT1-Agomelatine
11.11Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
11.11Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
11.11Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.11Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.11Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
11.11Single8IEBA1LYA8IEB-GPR156-A1LYA
11.11Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
11.11Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
11.11Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
11.11Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
11.11Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
11.11Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
11.11Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
11.11Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
11.11Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.11Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
11.11Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
11.11Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
11.11Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
10.81Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
10.71Single3PBLEticlopride3PBL-D3-Eticlopride
10.71Single4O9RCyclopamine4O9R-SMO-Cyclopamine
10.71Single5L7IVismodegib5L7I-SMO-Vismodegib
10.71Single6HLLCP999946HLL-NK1-CP99994
10.71Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
10.71Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
10.71Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.71Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
10.71Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
10.71Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
10.71Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
10.71Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.71Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.71Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
10.71Single9AS7Psilocin9AS7-5-HT2A-Psilocin
10.71Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
10.71Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
10.71Consensusgq_nucleotideOrthosteric Ligandgq_p2y
10.71Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.71Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
10.34Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
10.34Single4QINSAG1.54QIN-SMO-SAG1.5
10.34Single4S0VSuvorexant4S0V-OX2-Suvorexant
10.34Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
10.34Single5WS3EMPA5WS3-OX2-EMPA
10.34Single6DS0Ly2660976DS0-5-HT2B-Ly266097
10.34Single6ME9Ramelteon6ME9-MT2-Ramelteon
10.34Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
10.34Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
10.34Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.34Single6TODEMPA6TOD-OX1-EMPA-Na
10.34Single6TPJSuvorexant6TPJ-OX2-Suvorexant
10.34Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
10.34Single7F8ULintitript7F8U-CCKA-Lintitript
10.34Single7F8YDevazepide7F8Y-CCKA-Devazepide
10.34Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
10.34Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
10.34Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
10.34Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
10.34Single7XRRLemborexant7XRR-OX2-Lemborexant
10.34Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
10.34Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
10.34Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
10.34Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
10.34Single9H2XA1IR19H2X-A2A-A1IR1-Na
10.34Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
10.34Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.34Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.34Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
10.34Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.34Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
10.34Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
10.26Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
10.00Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
10.00Single3RZECidoxepin3RZE-H1-Cidoxepin
10.00Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
10.00Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
10.00Single5UVIZM-2413855UVI-A2A-ZM-241385
10.00Single6IQLL7458706IQL-D4-L745870
10.00Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
10.00Single6TP3Nemorexant6TP3-OX1-Nemorexant
10.00Single6TPNHTL66416TPN-OX2-HTL6641
10.00Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
10.00Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
10.00Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
10.00Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
10.00Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
10.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
10.00Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
10.00Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
10.00Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
10.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.00Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
10.00Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
10.00Single9ARXSerotonin9ARX-5-HT2A-Serotonin
10.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
10.00Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
10.00Consensusopsins_offOrthosteric Ligandrhodopsin_off
10.00Consensussensory_offOrthosteric Ligandopsins_off
9.68Single5DSGTiotropium5DSG-M4-Tiotropium
9.68Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single7F83PF-051904577F83-Ghrelin-PF-05190457
9.68Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
9.68Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
9.68Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
9.68Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
9.68Single8X64Desloratadine8X64-H1-Desloratadine
9.68Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
9.68Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
9.68Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
9.68Single9IYAONO-97105319IYA-GPR55-ONO-9710531
9.68Consensuscck_offOrthosteric Ligandccka_off
9.68Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
9.68Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
9.38Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
9.38Single5CGCHTL142425CGC-mGlu5-HTL14242
9.38Single5XPRBosentan5XPR-ETB-Bosentan
9.38Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
9.38Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
9.38Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
9.38Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
9.38Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
9.38Single7SINNPS-21437SIN-CaS-NPS-2143
9.38Single7SINNPS-21437SIN-CaS-NPS-2143
9.38Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
9.38Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
9.38Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
9.38Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
9.38Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
9.38Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
9.38Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
9.38Single9HAPTolvaptan9HAP-V2-Tolvaptan
9.38Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
9.09Single5TZRMK86665TZR-FFA1-MK8666
9.09Single6E59L-7607356E59-NK1-L-760735
9.09Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
9.09Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
9.09Single7R0CAVP7R0C-V2-AVP-Arrestin2
9.09Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
9.09Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
9.09Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
9.09Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
9.09Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
9.09Single8XVLZibotentan8XVL-ETA-Zibotentan
9.09Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
9.09Single9AS9RS130-1809AS9-5-HT2A-RS130-180
9.09Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
9.09Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
9.09Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
9.09Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
9.09Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
9.09Consensustachykinin_offOrthosteric Ligandnk1_off
8.82Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
8.82Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
8.82Single4PY02MeSATP4PY0-P2Y12-2MeSATP
8.82Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
8.82Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
8.82Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
8.82Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.82Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
8.82Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
8.82Single8XWACXCL18XWA-CXCR2-CXCL1
8.82Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
8.57Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
8.57Single5CGDHTL142425CGD-mGlu5-HTL14242
8.57Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.57Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
8.57Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
8.33Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
8.33Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
8.33Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.33Consensuskisspeptin_onOrthosteric Ligandkiss1_on
8.11Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.11Single8IEIA1LYA8IEI-GPR156-A1LYA
8.11Single8IEIA1LYA8IEI-GPR156-A1LYA
8.11Single8IEPA1LYA8IEP-GPR156-A1LYA
8.11Single8IEPA1LYA8IEP-GPR156-A1LYA
8.11Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.11Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.11Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
8.11Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
8.00Single5MZPCaffeine5MZP-A2A-Caffeine-Na
8.00Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
7.89Single8IEBA1LYA8IEB-GPR156-A1LYA
7.69Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
7.69Single7WC4Serotonin7WC4-5-HT2A-Serotonin
7.50Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
7.41Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
7.41Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
7.41Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.41Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
7.41Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
7.41Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
7.41Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
7.41Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
7.41Consensussensory_onOrthosteric Ligandopsins_on
7.14Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
7.14Single3UZAGTPL92363UZA-A2A-GTPL9236
7.14Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
7.14Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
7.14Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
7.14Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
7.14Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
7.14Single7WC5Psilocin7WC5-5-HT2A-Psilocin
7.14Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.14Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
7.14Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
7.14Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
7.14Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
7.14Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
7.14Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.14Consensusgi_sensoryOrthosteric Ligandgi_opsins
7.14Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.14Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.14Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
7.14Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
7.14Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
6.90Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
6.90Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
6.90Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
6.90Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
6.90Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
6.90Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
6.90Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
6.90Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
6.90Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
6.90Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
6.90Single7UL2SR486927UL2-NTS1-SR48692-Na
6.90Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
6.90Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
6.90Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
6.90Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
6.90Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.90Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.90Consensusneurotensin_offOrthosteric Ligandnts1_off
6.90Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
6.67Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
6.67Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
6.67Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
6.67Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
6.67Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
6.67Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
6.67Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
6.67Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
6.67Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
6.67Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.67Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.67Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
6.67Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
6.67Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
6.67Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
6.67Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
6.67Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
6.67Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
6.67Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.67Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.67Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
6.67Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
6.45Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
6.45Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
6.45Single6TPKRetosiban6TPK-OT-Retosiban
6.45Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
6.45Single7VODCariprazine7VOD-5-HT2A-Cariprazine
6.45Single7VV6C48/807VV6-MRGPRX2-C48/80
6.45Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
6.45Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
6.45Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
6.45Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
6.45Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
6.45Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.45Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.45Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
6.45Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.45Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.45Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.45Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.45Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
6.45Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
6.45Consensusvasop-oxy_offOrthosteric Ligandot_off
6.25Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
6.25Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
6.25Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
6.25Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
6.25Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
6.25Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
6.25Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.25Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
6.25Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
6.25Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
6.06Single4NTJAZD12834NTJ-P2Y12-AZD1283
6.06Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
6.06Single6HLPNetupitant6HLP-NK1-Netupitant
6.06Single6Z4SSR486926Z4S-NTS1-SR48692
6.06Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.06Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
6.06Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.06Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
6.06Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
6.06Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.06Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.06Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.06Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.06Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.06Single9HC04YI9HC0-mGlu5-4YI
5.88Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
5.88Single7P2L4YI7P2L-mGlu5-4YI
5.88Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.88Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.88Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.71Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
5.71Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.71Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.71Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.71Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.56Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
5.56Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
5.41Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
5.41Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
5.26Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
4.35Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.35Single6D35Cholesterol6D35-SMO-Cholesterol
4.35Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.35Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.35Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.35Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.35Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
4.35Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.35Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.35Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
4.35Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.35Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
4.35Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.35Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.35Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.35Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.35Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.35Single7DTTCa7DTT-CaS-Ca-Ca
4.35Single7DTTCa7DTT-CaS-Ca-Ca
4.35Single7DTUTryptophan7DTU-CaS-Tryptophan
4.35Single7DTUTryptophan7DTU-CaS-Tryptophan
4.35Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.35Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.35Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.35Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.35Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.35Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.35Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.35Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.35Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.35Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.35Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.35Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.35Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.35Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.35Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.35Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.35Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.35Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.35Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.35Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.35Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.35Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.35Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.35Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.35Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.35Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.35Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.35Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.35Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.35Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.35Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.35Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.35Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.35Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.35Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.35Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.35Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
4.35Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.35Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.35Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.35Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.35Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.35Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.35Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.35Single7XW7K1-707XW7-TSH-K1-70
4.35Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.35Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.35Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.35Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.35Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.35Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.35Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.35Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.35Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.35Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.35Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.35Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.35Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.35Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.35Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.35Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.35Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.35Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.35Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.35Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.35Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.35Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.35Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.35Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.35Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.35Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.35Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.35Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.35Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.35Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.35Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.35Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.35Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.35Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.35Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.35Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.35Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.35Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.35Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.35Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.35Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.35Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.35Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.35Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.35Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.35Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.35Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.35Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.35Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.35Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.35Single8WVXNorrin8WVX-LGR4-Norrin
4.35Single8WVYNorrin8WVY-LGR4-Norrin
4.35Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.35Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.35Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.35Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.35Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.35Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.35Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.35Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.35Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.35Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.35Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.35Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.35Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.35Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.35Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.35Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.35Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.35Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.35Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.35Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.35Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.35Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.35Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.35Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.35Single9KHHNorrin9KHH-LGR4-Norrin
4.35Single9S37NB219S37-LGR4-NB21
4.35Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.17Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.17Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.17Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.17Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.17Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.17Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.17Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.17Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.17Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.17Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.17Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.17Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.17Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.17Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.17Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.17Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.00Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.00Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.00Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
3.85Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
3.85Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
3.85Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
3.85Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
3.85Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.70Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
3.70Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
3.70Single5L7DCholesterol5L7D-SMO-Cholesterol
3.70Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
3.70Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.70Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.57Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
3.57Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
3.45Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
3.45Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
3.45Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
3.45Single8JPSCCL78JPS-ACKR1-CCL7
3.45Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.33Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
3.33Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
3.33Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
3.33Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
3.33Single6TP4ACT-4622066TP4-OX1-ACT-462206
3.33Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.33Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
3.33Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.33Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
3.33Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
3.23Single4XNVBPTU4XNV-P2Y1-BPTU
3.23Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
3.23Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
3.23Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
3.12Single6FFIMMPEP6FFI-mGlu5-MMPEP
3.12Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
3.12Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
3.12Single6ZINSR486926ZIN-NTS1-SR48692
3.12Single8IYXYL-3658IYX-GPR34-YL-365
3.12Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.12Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
3.03Single6FFHFenobam6FFH-mGlu5-Fenobam
2.94Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
2.94Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
2.86Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
2.86Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
2.56Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.56Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.44Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.44Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.38Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.22Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
glp1_on_gp 7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
7X8R-GLP-1-BOC5-Gs/β1/γ2
6X19-GLP-1-CHU-128-Gs/β1/γ2
6X1A-GLP-1-Danuglipron-Gs/β1/γ2
6X18-GLP-1-GLP-1-Gs/β1/γ2
8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
7KI0-GLP-1-Semaglutide-Gs/β1/γ2
7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
7X8S-GLP-1-WB4-24-Gs/β1/γ2
8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
glp2_on_gp 7D68-GLP-2-GLP-2-Gs/β1/γ2
Net Summary
Imin 3.11667
Number of Linked Nodes 1019
Number of Links 1151
Number of Hubs 159
Number of Links mediated by Hubs 647
Number of Communities 30
Number of Nodes involved in Communities 181
Number of Links involved in Communities 241
Path Summary
Number Of Nodes in MetaPath 108
Number Of Links MetaPath 107
Number of Shortest Paths 4958851
Length Of Smallest Path 3
Average Path Length 51.0583
Length of Longest Path 98
Minimum Path Strength 0.09625
Average Path Strength 6.62635
Maximum Path Strength 29.9431
Minimum Path Correlation 0.7
Average Path Correlation 0.922971
Maximum Path Correlation 0.995417
Minimum % Of Corr. Nodes 1.11111
Average % Of Corr. Nodes 24.779
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 43.6978
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
glucagon_on_gpglp_on_gp
gluc_on_gp
secretin_on_gp
gip_on_gp



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