Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg Int. Strength Num Of Links Community ConSurf
1A:A:?17 4.745403
2A:A:?34 4.71415
3A:A:?37 9.38571713
4A:A:H41 5.672536
5A:A:L44 10.1975419
6A:A:N50 5.8725229
7A:A:?53 6.79409
8A:A:?63 5.8075409
9A:A:F212 8.838509
10A:A:Q227 8.4325419
11A:A:R228 8.0725419
12A:A:R232 8.425418
13A:A:?233 5.0125419
14A:A:W234 8.5325409
15A:A:?237 8.716518
16A:A:?253 7.166199
17A:A:F273 7.4425439
18A:A:W277 9.65833636
19A:A:W281 8.038515
20A:A:F290 7.2275489
21A:A:N292 5.424589
22A:A:Q294 7.9425436
23A:A:?300 4.4525409
24A:A:?311 13.78336195
25A:A:?318 11.6714737
26A:A:E330 5.798503
27A:A:D331 8.8475404
28A:A:?338 8.396535
29A:A:?339 10.62633
30A:A:F340 8.2575406
31A:A:R342 7.83333635
32A:A:F345 7.3025438
33A:A:?358 10.5962834
34A:A:?359 18.5325436
35A:A:?360 14.8788838
36A:A:F363 7.91435
37A:A:T364 9.062589
38A:A:?365 9.30833687
39A:A:R373 6.5275436
40A:A:?379 5.3925439
41A:A:I382 5.658537
42A:A:?391 8.96333664
43B:B:L7 5.8408
44B:B:N16 8.31401
45B:B:I18 4.4825407
46B:B:?25 4.352503
47B:B:V40 6.2025473
48B:B:R49 5.1525407
49B:B:L51 9.5409
50B:B:H54 7.65286719
51B:B:I58 6.9325419
52B:B:?59 10.4414718
53B:B:M61 5.79416
54B:B:W63 8.47167617
55B:B:Q75 13.3825419
56B:B:D76 7.98667619
57B:B:?77 8.265418
58B:B:L79 4.715407
59B:B:W82 8.59571719
60B:B:?85 14.27836204
61B:B:N88 7.3925407
62B:B:I93 4.84457
63B:B:L95 6.2475408
64B:B:W99 10.9067619
65B:B:M101 5.2975419
66B:B:?103 6.442508
67B:B:?105 9.07444956
68B:B:?109 6.6525455
69B:B:N110 7.8675454
70B:B:?111 7.532731154
71B:B:V112 5.854558
72B:B:?114 7.825658
73B:B:L117 5.8175419
74B:B:?121 6.97458
75B:B:I123 5.1456
76B:B:?124 7.835856
77B:B:L139 4.4725409
78B:B:H142 7.644519
79B:B:?144 11.466518
80B:B:?145 9.794551118
81B:B:L146 6.6575457
82B:B:?148 12.3017656
83B:B:?149 13.62558
84B:B:F151 7.978559
85B:B:D154 6.408556
86B:B:S161 8.916519
87B:B:?162 9.658519
88B:B:D163 8.915619
89B:B:T165 7.84417
90B:B:W169 7.555408
91B:B:D170 3.915409
92B:B:F180 10.756517
93B:B:H183 7.142519
94B:B:?185 7.9375415
95B:B:D186 8.306519
96B:B:V200 8.6675416
97B:B:?204 9.15833617
98B:B:D205 6.2875419
99B:B:?209 8.9925416
100B:B:W211 10.0514718
101B:B:H225 11.3417619
102B:B:I232 7.17418
103B:B:?233 7.905403
104B:B:F234 8.605405
105B:B:F235 9.02833676
106B:B:P236 7.04477
107B:B:N237 12.92475
108B:B:?238 5.3025477
109B:B:N239 11.525472
110B:B:F241 9.292516
111B:B:T243 7.6675418
112B:B:D247 10.305419
113B:B:?250 13.5175418
114B:B:R251 14.58518
115B:B:F253 9.17516
116B:B:D254 6.4425409
117B:B:D258 10.21417
118B:B:?264 15.0283605
119B:B:I269 4.135414
120B:B:?271 9.81515
121B:B:I273 7.735416
122B:B:F278 7.26333677
123B:B:?282 5.18667679
124B:B:R283 8.9579
125B:B:?289 10.7791017
126B:B:D290 8.648516
127B:B:N293 6.39415
128B:B:?294 7.46415
129B:B:N295 11.69416
130B:B:W297 10.5375418
131B:B:R304 8.326515
132B:B:H311 8.5565109
133B:B:R314 10.928518
134B:B:?317 7.64833617
135B:B:T321 8.35417
136B:B:D323 6.88417
137B:B:?324 7.1025419
138B:B:W332 9.33619
139B:B:D333 7.01409
140B:B:?337 5.981437106
141B:B:W339 9.081676109
142G:G:?20 4.2625406
143G:G:?40 13.5486776
144G:G:?41 9.182577
145G:G:D48 7.35409
146G:G:N59 6.874509
147G:G:F61 6.6125408
148H:H:?2 17.28754150
149L:L:?31 14.614520
150L:L:?34 9.08520
151L:L:N39 6.3525260
152L:L:I49 4.4375400
153L:L:?52 8.49667620
154L:L:?55 17.73520
155L:L:?56 19.94420
156L:L:?61 10.3556990
157L:L:T63 5.8025420
158L:L:?68 6.954520
159L:L:?69 5.315400
160L:L:M71 6.108520
161L:L:V77 4.4725490
162L:L:?83 13.805620
163L:L:?84 10.845620
164L:L:V85 4.695420
165L:L:S88 4.4454120
166L:L:?89 8.3654120
167L:L:F98 5.3425280
168L:L:H103 8.7425400
169L:L:?108 11.6283620
170L:L:?111 14.635620
171L:L:?112 13.7256920
172L:L:?113 15.172520
173L:L:H114 11.02620
174L:L:?115 6.18833620
175N:N:?43 13.585160
176N:N:?46 11.095400
177N:N:?54 10.654500
178N:N:?57 17.1675820
179N:N:?58 14.76620
180N:N:Q74 9.13420
181N:N:?77 8.2775400
182N:N:?79 10.2543790
183N:N:R80 8.6675420
184N:N:L89 6.84160
185N:N:?92 16.38254160
186N:N:?102 9.475400
187N:N:?108 7.76520
188N:N:Q109 6.845420
189N:N:?110 9.155420
190N:N:R115 9.8525420
191N:N:?120 8.765620
192N:N:?124 6.44400
193N:N:?130 9.8125400
194R:R:?58 12.59405
195R:R:?62 5.415404
196R:R:I64 5.78407
197R:R:Q82 10.9675406
198R:R:F94 7.3075409
199R:R:D95 8.054136
200R:R:L100 5.7375409
201R:R:N107 11.0575427
202R:R:?113 10.3025401
203R:R:I114 5.3925408
204R:R:I120 6.54254135
205R:R:?126 8.36405
206R:R:?127 10.9083626
207R:R:L128 5.7725408
208R:R:?131 11.124527
209R:R:N132 5.378528
210R:R:T133 7.9925428
211R:R:?134 6.63405
212R:R:I135 5.5425407
213R:R:F138 6.35254305
214R:R:D140 5.61754133
215R:R:?143 8.2685134
216R:R:F151 8.005405
217R:R:I152 5.3025424
218R:R:E154 8.862527
219R:R:I155 5.6875428
220R:R:?156 16.1867627
221R:R:N158 7.67833629
222R:R:?166 6.255404
223R:R:Q170 11.25254153
224R:R:N173 5.19404
225R:R:L181 4.7975408
226R:R:?182 12.1675826
227R:R:?183 8.7325427
228R:R:N184 9.62714729
229R:R:F186 10.436528
230R:R:H192 6.4425405
231R:R:F194 8.635409
232R:R:N195 14.1245155
233R:R:L202 6.56407
234R:R:H209 6.7425401
235R:R:F218 10.085408
236R:R:?223 7.14254177
237R:R:P224 8.9925408
238R:R:L227 4.57254148
239R:R:I229 4.38407
240R:R:?240 14.3745172
241R:R:?241 11.7425177
242R:R:?254 9.295312
243R:R:L256 3.895408
244R:R:P260 5.5275406
245R:R:F265 7.63754147
246R:R:?275 14.17336318
247R:R:F282 7.615148
248R:R:?333 12.38254181
249R:R:?336 10.19254186
250R:R:E354 8.555407
251R:R:D355 7.845447
252R:R:?359 13.685446
253R:R:R363 9.558549
254R:R:I366 5.36549
255R:R:?376 4.4975467
256R:R:N377 8.6375469
257R:R:?389 14.20297113
258R:R:N400 8.90254217
259R:R:L401 6.26668
260R:R:D405 8.096569
261R:R:?407 6.9025447
262R:R:?411 7.4051047
263R:R:D419 9.955449
264R:R:?426 12.25329
265R:R:?427 14.2754327
266R:R:W433 14.39449
267R:R:?438 11.48448
268R:R:?439 16.014549
269R:R:?455 8.994508
270R:R:R464 9.8175468
271R:R:?470 7.45403
272R:R:I472 6.884535
273R:R:M487 8.124217
274R:R:?490 8.7625408
275R:R:W491 7.1445215
276R:R:?508 10.7244948
277R:R:?514 10.3367649
278R:R:F515 6.65649
279R:R:?527 8.60143707
280R:R:L532 3.32409
281R:R:?543 7.44667667
282R:R:?545 10.0583666
283R:R:?546 10.7711069
284R:R:?550 5.66167669
285R:R:N555 7.7625437
286R:R:?581 6.115649
287R:R:?612 8.61833647
288R:R:?617 6.02509
289R:R:N619 7.845469
290R:R:L622 4.5575409
291R:R:?623 7.05333669
292R:R:F630 6.215408
293R:R:D633 9.65254118
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Int. Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.

Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1B:B:?59 B:B:I58 10.15065.55YesYes189
2A:A:?237 B:B:?59 1007.21YesYes188
3A:A:?237 B:B:W99 1007.32YesYes189
4A:A:F222 B:B:W99 10023.05NoYes069
5B:B:?59 B:B:Q75 10019.42YesYes189
6B:B:Q75 B:B:W99 1009.86YesYes199
7A:A:E209 A:A:F222 1008.16NoNo096
8A:A:?211 A:A:E209 1007.11NoNo049
9A:A:?211 A:A:F212 1004.36NoYes049
10A:A:F212 A:A:F219 10017.15YesNo098
11A:A:F219 A:A:H41 1005.66NoYes386
12A:A:?379 A:A:F219 1005.22YesNo398
13A:A:H41 R:R:I472 1007.95YesYes365
14A:A:?379 R:R:I472 1006.11YesYes395
15A:A:?225 A:A:Q227 10.48724.64NoYes099
16A:A:?225 A:A:F208 10.58954.25NoNo096
17A:A:D223 A:A:F208 10.64145.97NoNo096
18A:A:D223 A:A:L45 12.27095.43NoNo098
19A:A:F212 A:A:M221 12.90424.98YesNo098
20B:B:?59 B:B:W332 1007.75YesYes189
21A:A:W281 B:B:W332 72.33887.5YesYes159
22B:B:R314 B:B:W332 10020.99YesYes189
23A:A:?237 B:B:L117 11.0057.41YesYes189
24A:A:W281 B:B:D290 71.7938.93YesYes156
25B:B:D290 B:B:R314 71.78568.34YesYes168
26A:A:R380 R:R:I472 1007.52NoYes075
27A:A:Q384 A:A:R380 1008.18NoNo067
28A:A:Q384 R:R:I468 1004.12NoNo067
29A:A:L388 R:R:I468 1005.71NoNo087
30A:A:L388 A:A:L393 1005.54NoNo089
31A:A:?391 A:A:L393 1009.42YesNo049
32A:A:?391 R:R:R464 10016.54YesYes648
33B:B:?233 B:B:I232 17.25366.11YesYes038
34B:B:F241 B:B:I232 15.69178.79YesYes168
35B:B:F222 B:B:F241 15.434712.86NoYes186
36B:B:F222 B:B:Q220 1008.2NoNo187
37B:B:D258 B:B:Q220 10010.44YesNo177
38B:B:D258 B:B:R22 10015.48YesNo076
39B:B:I18 B:B:R22 68.10126.26YesNo076
40B:B:I18 G:G:A23 1003.25YesNo078
41G:G:?20 G:G:A23 1002.82YesNo068
42G:G:?20 G:G:V16 84.53823.55YesNo067
43B:B:L7 G:G:V16 70.44862.98YesNo087
44B:B:L7 G:G:A12 35.22453.15YesNo085
45B:B:L4 G:G:A12 28.17961.58NoNo045
46B:B:D258 G:G:R27 70.446510.72YesNo178
47B:B:I18 G:G:R27 1005.01YesNo078
48B:B:Q220 G:G:I25 72.79454.12NoNo172
49G:G:I25 G:G:R27 70.44646.26NoNo128
50B:B:L14 G:G:?20 28.17964.95NoYes086
51B:B:?15 B:B:I18 49.31423.41NoYes067
52B:B:?15 B:B:N16 42.26934.1NoYes061
53B:B:E12 B:B:N16 14.089815.77NoYes041
54B:B:L14 G:G:L19 14.08984.15NoNo089
55B:B:N16 B:B:R19 14.089812.05YesNo014
56B:B:Q17 G:G:A23 14.08981.52NoNo048
57B:B:Q259 B:B:R22 37.57467.01NoNo066
58B:B:A26 B:B:Q259 35.22624.55NoNo036
59B:B:?25 B:B:A26 32.87793.37YesNo033
60B:B:?25 B:B:D27 23.48455.81YesNo038
61B:B:D27 G:G:S31 11.74248.83NoNo089
62B:B:?317 B:B:M61 39.26294.54YesYes176
63B:B:?317 B:B:V315 71.30914.79YesNo077
64B:B:?288 B:B:V315 71.17235.2NoNo077
65B:B:?288 B:B:?289 71.035727NoYes177
66B:B:?289 B:B:W297 76.21785.54YesYes178
67B:B:?264 B:B:W297 66.303222.15YesYes058
68B:B:?317 B:B:?59 1007.21YesYes178
69B:B:?289 B:B:D290 1006.6YesYes176
70B:B:R314 B:B:T274 71.228611.64YesNo188
71B:B:?289 B:B:T274 71.0938.6YesNo178
72B:B:?289 B:B:N295 12.200218.7YesYes176
73B:B:?319 B:B:W63 29.84528.94NoYes057
74B:B:L284 B:B:V296 14.93844.47NoNo055
75B:B:I43 B:B:L284 13.69415.71NoNo035
76B:B:F253 B:B:T243 61.27439.08YesYes168
77B:B:?224 B:B:F253 61.27084.25NoYes066
78B:B:?289 B:B:I273 10012.49YesYes176
79B:B:?250 B:B:I273 1006.11YesYes186
80B:B:?250 B:B:R251 1006.5YesYes188
81B:B:H225 B:B:T243 61.846810.95YesYes198
82B:B:?244 B:B:I273 65.71657.47NoYes056
83B:B:?319 B:B:V320 27.47575.2NoNo057
84B:B:S277 B:B:V320 27.33694.85NoNo057
85B:B:E260 B:B:F253 1004.66NoYes066
86B:B:?264 B:B:T263 62.4078.6YesNo051
87B:B:?306 B:B:R304 15.482612.71NoYes045
88B:B:L4 G:G:S8 14.08983NoNo044
89B:B:L7 G:G:R13 21.13472.43YesNo086
90G:G:I9 G:G:R13 14.089810.02NoNo026
91R:R:?623 R:R:R464 1008.27YesYes698
92R:R:?623 R:R:L401 1005.38YesYes698
93R:R:D405 R:R:L401 1006.79YesYes698
94R:R:D405 R:R:S616 1008.83YesNo099
95R:R:M408 R:R:S616 1009.2NoNo089
96R:R:?612 R:R:M408 1008.25YesNo078
97R:R:?612 R:R:F515 10011.85YesYes479
98R:R:?411 R:R:F515 1004.74YesYes479
99R:R:?411 R:R:L412 1009.42YesNo478
100R:R:I366 R:R:L412 1005.71YesNo498
101R:R:I366 R:R:M357 1005.83YesNo497
102R:R:D419 R:R:M357 1009.7YesNo497
103R:R:D419 R:R:I356 1005.6YesNo098
104R:R:I356 R:R:S512 1004.64NoNo089
105R:R:E354 R:R:S512 1004.31YesNo079
106R:R:?353 R:R:E354 1008.51NoYes097
107R:R:?280 R:R:?353 1009.52NoNo099
108R:R:?279 R:R:?280 10025.4NoNo099
109R:R:?279 R:R:F282 1007.83NoYes098
110R:R:F265 R:R:F282 1007.5YesYes1478
111R:R:F265 R:R:L248 1006.09YesNo1479
112R:R:L227 R:R:L248 1004.15YesNo1489
113R:R:L202 R:R:L227 1004.15YesYes078
114R:R:L202 R:R:L204 10011.07YesNo079
115R:R:L181 R:R:L204 1004.15YesNo089
116R:R:I155 R:R:L181 84.28254.28YesYes088
117R:R:I155 R:R:L153 22.3688.56YesNo089
118R:R:L128 R:R:L153 21.12754.15YesNo089
119R:R:L401 R:R:N619 1008.24YesYes689
120R:R:N615 R:R:N619 1005.45NoYes099
121R:R:?581 R:R:N615 10013.23YesNo099
122R:R:?581 R:R:?612 1004.32YesYes497
123R:R:?623 R:R:L457 1005.38YesNo699
124R:R:L457 R:R:N619 1009.61NoYes699
125R:R:?426 R:R:S512 1004.38YesNo099
126R:R:?426 R:R:?427 10028.81YesYes3297
127R:R:?427 R:R:A281 1006.13YesNo078
128R:R:A281 R:R:R262 1004.15NoNo085
129R:R:F282 R:R:R262 10011.76YesNo085
130R:R:I245 R:R:L248 20.6154.28NoNo1489
131R:R:I245 R:R:L242 20.20744.28NoNo089
132R:R:?241 R:R:L242 39.58854.83YesNo079
133R:R:?240 R:R:?241 35.465723.48YesYes1727
134R:R:?240 R:R:R219 33.140923.63YesNo021
135R:R:H192 R:R:R219 30.60829.03YesNo051
136H:H:?2 R:R:H192 23.93128.08YesYes005
137R:R:F265 R:R:P260 29.29257.22YesYes076
138R:R:L237 R:R:P260 21.4618.21NoYes076
139R:R:L237 R:R:L242 20.21025.54NoNo079
140H:H:?2 R:R:Q170 19.06716.72YesYes1503
141R:R:?279 R:R:?343 96.262115.87NoNo099
142R:R:?343 R:R:R342 95.85737.81NoNo094
143R:R:E270 R:R:R342 95.655311.63NoNo064
144R:R:E270 R:R:R247 95.45355.82NoNo065
145R:R:R247 R:R:T226 90.83665.17NoNo054
146R:R:S201 R:R:T226 90.03466.4NoNo054
147R:R:E203 R:R:S201 89.83424.31NoNo055
148R:R:?182 R:R:E203 89.63416.75YesNo065
149L:L:?115 R:R:?182 73.27155.62YesYes206
150L:L:?115 N:N:?120 30.06566.19YesYes200
151N:N:?120 N:N:T118 15.60244.74YesNo000
152L:L:V77 N:N:T118 15.38914.76YesNo000
153R:R:?180 R:R:L181 91.2576.61NoYes058
154R:R:?180 R:R:E154 90.68538.7NoYes057
155R:R:?127 R:R:E154 89.96814.18YesYes267
156L:L:?111 R:R:?127 46.07234.32YesYes206
157L:L:?111 L:L:?83 67.16517.46YesYes200
158L:L:?83 L:L:?84 52.235323.81YesYes200
159L:L:?52 L:L:?84 85.8746.35YesYes200
160L:L:?52 L:L:Q51 58.52337.13YesNo000
161L:L:N39 L:L:Q51 38.60125.28YesNo000
162L:L:I49 L:L:N39 17.43434.25YesYes000
163L:L:I49 L:L:N102 41.09234.25YesNo000
164H:H:?4 L:L:N102 29.885523.41NoNo000
165L:L:?115 L:L:H114 42.54748.44YesYes200
166L:L:?111 L:L:H114 23.028222.03YesYes200
167L:L:?112 R:R:?127 37.765318.33YesYes206
168L:L:?112 L:L:V85 53.48264.35YesYes200
169L:L:?84 L:L:V85 52.23874.79YesYes200
170L:L:?112 L:L:H114 18.89887.5YesYes200
171L:L:Q51 N:N:V64 18.67817.16NoNo000
172L:L:I49 N:N:V64 34.86564.61YesNo000
173L:L:?52 L:L:H103 22.413412.39YesYes000
174L:L:H103 N:N:V64 18.67859.69YesNo000
175H:H:?4 L:L:P48 18.67857.37NoNo000
176L:L:?108 L:L:?83 13.69120.63YesYes200
177L:L:?108 L:L:?56 11.22499.52YesYes200
178L:L:F42 L:L:N39 14.9448.46NoYes2600
179L:L:F42 N:N:L65 13.6994.87NoNo000
180L:L:?46 L:L:P48 14.94282.86NoNo000
181L:L:?46 L:L:A47 11.20712.75NoNo000
182N:N:?120 N:N:D119 10.88354.36YesNo000
183R:R:I155 R:R:N158 58.68534.25YesYes289
184R:R:?131 R:R:N158 24.01365.88YesYes279
185R:R:?131 R:R:N132 35.43035.88YesYes278
186L:L:M71 R:R:N132 22.3937.01YesYes208
187L:L:?68 L:L:M71 28.19235.9YesYes200
188R:R:?156 R:R:?182 12.444415.86YesYes276
189R:R:?131 R:R:?156 12.069630.16YesYes277
190R:R:N107 R:R:N132 11.18265.45YesYes278
191L:L:?68 L:L:?69 25.73838.87YesYes000
192L:L:?69 L:L:L65 23.2484.13YesNo000
193L:L:L65 N:N:E39 22.41793.98NoNo000
194R:R:N158 R:R:T133 18.26388.77YesYes298
195N:N:?46 N:N:E39 19.927311.35YesNo000
196N:N:?46 N:N:I47 14.94629.17YesNo000
197N:N:I47 N:N:P90 13.28576.77NoNo000
198R:R:I135 R:R:T133 15.87197.6YesYes078
199R:R:I114 R:R:I135 30.00315.89YesYes087
200R:R:?113 R:R:I114 15.85745.55YesYes018
201R:R:?62 R:R:E87 10.015511.86YesNo045
202R:R:I161 R:R:N158 16.19235.66NoYes079
203R:R:I135 R:R:I161 15.80064.42YesNo077
204R:R:?171 R:R:Q170 15.84516.96NoYes043
205R:R:?171 R:R:F145 15.01124.25NoNo043
206R:R:?143 R:R:F145 14.177416.71YesNo043
207B:B:M61 B:B:W63 38.84268.14YesYes167
208A:A:L45 A:A:M221 12.32377.07NoNo088
209B:B:?233 B:B:S277 27.19834.82YesNo035
210B:B:?41 B:B:I43 12.454.98NoNo013
211B:B:?306 B:B:V296 14.37527.79NoNo045
212B:B:?224 B:B:R251 62.372812.71NoYes068
213B:B:?244 B:B:H225 64.60565.61NoYes059
214B:B:E260 B:B:R251 61.817820.93NoYes068
215B:B:E260 B:B:T263 61.85129.88NoNo061
216B:B:F222 B:B:F253 10015NoYes186
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1 Node2 LinkStrength Comm IsNode1Hub? IsNode2Hub? Node1Cons Node2Cons Node1Shell Node2Shell
H:H:?3 L:L:N76 25.87 0 No No 0 0 1 0
H:H:?3 N:N:A103 4.24 0 No No 0 0 1 0
H:H:?4 L:L:P48 7.37 0 No No 0 0 1 0
H:H:?4 L:L:L50 7.45 0 No No 0 0 1 0
H:H:?4 L:L:N102 23.41 0 No No 0 0 1 0
H:H:?5 N:N:N33 27.11 0 No No 0 0 1 0
L:L:F41 R:R:?328 4.25 26 No No 0 1 0 1
L:L:M71 R:R:N107 8.41 2 Yes Yes 0 7 0 1
L:L:M71 R:R:N132 7.01 2 Yes Yes 0 8 0 1
L:L:L72 R:R:N132 4.12 0 No Yes 0 8 0 1
L:L:L72 R:R:H160 7.71 0 No No 0 3 0 1
L:L:V73 R:R:N132 4.43 0 No Yes 0 8 0 1
L:L:?89 R:R:E148 9.02 12 Yes No 0 5 0 1
L:L:R91 R:R:S149 7.91 12 No No 0 3 0 1
L:L:E101 R:R:S149 8.62 12 No No 0 3 0 1
L:L:T110 R:R:E102 8.47 2 No No 0 7 0 1
L:L:?111 R:R:?127 4.32 2 Yes Yes 0 6 0 1
L:L:?112 R:R:E102 10.31 2 Yes No 0 7 0 1
L:L:?112 R:R:?127 18.33 2 Yes Yes 0 6 0 1
L:L:?112 R:R:I152 4.16 2 Yes Yes 0 4 0 1
L:L:?113 R:R:I152 6.94 2 Yes Yes 0 4 0 1
L:L:?115 R:R:E154 7.11 2 Yes Yes 0 7 0 1
L:L:?115 R:R:?182 5.62 2 Yes Yes 0 6 0 1
N:N:Q66 R:R:N150 11.88 0 No No 0 5 0 1
N:N:L69 R:R:D330 5.43 0 No No 0 4 0 1
N:N:P70 R:R:R247 7.21 0 No No 0 5 0 1
N:N:R115 R:R:D157 10.72 2 Yes No 0 6 0 1
N:N:R115 R:R:?182 8.27 2 Yes Yes 0 6 0 1
N:N:R115 R:R:?183 5.3 2 Yes Yes 0 7 0 1
N:N:R115 R:R:E206 15.12 2 Yes No 0 4 0 1
N:N:?124 R:R:Q82 7.94 0 Yes Yes 0 6 0 1
N:N:H126 R:R:?58 16.26 0 No Yes 0 5 0 1
R:R:?58 R:R:A57 9.19 0 Yes No 5 4 1 2
R:R:?58 R:R:L59 8.08 0 Yes No 5 7 1 2
R:R:?58 R:R:Q82 16.83 0 Yes Yes 5 6 1 1
R:R:Q82 R:R:S81 7.22 0 Yes No 6 6 1 2
R:R:Q106 R:R:S81 4.33 0 No No 7 6 2 2
R:R:N107 R:R:Q82 11.88 2 Yes Yes 7 6 1 1
R:R:N107 R:R:Q106 18.49 2 Yes No 7 7 1 2
R:R:N107 R:R:N132 5.45 2 Yes Yes 7 8 1 1
R:R:?126 R:R:?127 12.85 0 Yes Yes 5 6 2 1
R:R:?126 R:R:E148 6.32 0 Yes No 5 5 2 1
R:R:?127 R:R:S129 10.22 2 Yes No 6 7 1 2
R:R:?127 R:R:I152 5.55 2 Yes Yes 6 4 1 1
R:R:?127 R:R:E154 14.18 2 Yes Yes 6 7 1 1
R:R:E154 R:R:S129 10.06 2 Yes No 7 7 1 2
R:R:?131 R:R:N132 5.88 2 Yes Yes 7 8 2 1
R:R:?131 R:R:?156 30.16 2 Yes Yes 7 7 2 2
R:R:?131 R:R:D157 5.81 2 Yes No 7 6 2 1
R:R:?134 R:R:H160 6.73 0 Yes No 5 3 2 1
R:R:I152 R:R:T178 4.56 2 Yes No 4 6 1 2
R:R:?156 R:R:E154 4.26 2 Yes Yes 7 7 2 1
R:R:?180 R:R:E154 8.7 0 No Yes 5 7 2 1
R:R:?156 R:R:D157 17.44 2 Yes No 7 6 2 1
R:R:?156 R:R:?182 15.86 2 Yes Yes 7 6 2 1
R:R:?156 R:R:N184 14.7 2 Yes Yes 7 9 2 2
R:R:?180 R:R:?182 16.87 0 No Yes 5 6 2 1
R:R:?182 R:R:?183 15.26 2 Yes Yes 6 7 1 1
R:R:?182 R:R:N184 10.68 2 Yes Yes 6 9 1 2
R:R:?182 R:R:E203 16.75 2 Yes No 6 5 1 2
R:R:?182 R:R:?205 8.03 2 Yes No 6 7 1 2
R:R:?183 R:R:N184 8.38 2 Yes Yes 7 9 1 2
R:R:?183 R:R:N207 5.99 2 Yes No 7 9 1 2
R:R:N184 R:R:N207 5.45 2 Yes No 9 9 2 2
R:R:?205 R:R:E206 9.49 0 No No 7 4 2 1
R:R:R247 R:R:T226 5.17 0 No No 5 4 1 2
R:R:E270 R:R:R247 5.82 0 No No 6 5 2 1
R:R:?328 R:R:W329 5.96 0 No No 1 3 1 2
R:R:?331 R:R:D330 18.48 18 No No 1 4 2 1
R:R:?126 R:R:N150 4.1 0 Yes No 5 5 2 1
R:R:?77 R:R:E102 3.95 0 No No 5 7 2 1
L:L:H107 R:R:R53 2.26 0 No No 0 2 0 1
H:H:?5 N:N:N50 1.23 0 No No 0 0 1 0

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
50.00Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
33.33Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
33.33Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
25.00Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
25.00Single6D35Cholesterol6D35-SMO-Cholesterol
25.00Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
25.00Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
25.00Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
25.00Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
25.00Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
25.00Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
25.00Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
25.00Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
25.00Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
25.00Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
25.00Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
25.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
25.00Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
25.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
25.00Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
25.00Single7DTTCa7DTT-CaS-Ca-Ca
25.00Single7DTTCa7DTT-CaS-Ca-Ca
25.00Single7DTUTryptophan7DTU-CaS-Tryptophan
25.00Single7DTUTryptophan7DTU-CaS-Tryptophan
25.00Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
25.00Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
25.00Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
25.00Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
25.00Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
25.00Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
25.00Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
25.00Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
25.00Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
25.00Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
25.00Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
25.00Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
25.00Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
25.00Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
25.00Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
25.00Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
25.00Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
25.00Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
25.00Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
25.00Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
25.00Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
25.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
25.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
25.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
25.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
25.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
25.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
25.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
25.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
25.00Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
25.00Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
25.00Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
25.00Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
25.00Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
25.00Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
25.00Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
25.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
25.00Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
25.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
25.00Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
25.00Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
25.00Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
25.00Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
25.00Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
25.00Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
25.00Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
25.00Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
25.00Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
25.00Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
25.00Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
25.00Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
25.00Single7XW7K1-707XW7-TSH-K1-70
25.00Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
25.00Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
25.00Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
25.00Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
25.00Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
25.00Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
25.00Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
25.00Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
25.00Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
25.00Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
25.00Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
25.00Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
25.00Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
25.00Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
25.00Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
25.00Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
25.00Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
25.00Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
25.00Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
25.00Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
25.00Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
25.00Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
25.00Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
25.00Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
25.00Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
25.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
25.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
25.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
25.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
25.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
25.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
25.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
25.00Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
25.00Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
25.00Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
25.00Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
25.00Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
25.00Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
25.00Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
25.00Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
25.00Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
25.00Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
25.00Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
25.00Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
25.00Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
25.00Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
25.00Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
25.00Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
25.00Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
25.00Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
25.00Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
25.00Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
25.00Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
25.00Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
25.00Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
25.00Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
25.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
25.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
25.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8WVXNorrin8WVX-LGR4-Norrin
25.00Single8WVYNorrin8WVY-LGR4-Norrin
25.00Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
25.00Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
25.00Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
25.00Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
25.00Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
25.00Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
25.00Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
25.00Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
25.00Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
25.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
25.00Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
25.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
25.00Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
25.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
25.00Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
25.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
25.00Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
25.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
25.00Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
25.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
25.00Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
25.00Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
25.00Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
25.00Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
25.00Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
25.00Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
25.00Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
25.00Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
20.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
20.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
20.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
20.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
20.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
20.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
20.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
20.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
20.00Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
20.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
20.00Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
20.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
16.67Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
16.67Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
14.29Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
14.29Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
12.50Single5L7DCholesterol5L7D-SMO-Cholesterol
12.50Single8HS2Fab0468HS2-GPR20-Fab046
12.50Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
12.50Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.50Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
11.11Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
11.11Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
11.11Consensusp2y_offOrthosteric Ligandp2y1_off
10.00Single4XNWMRS25004XNW-P2Y1-MRS2500
10.00Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
10.00Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
10.00Single8JPSCCL78JPS-ACKR1-CCL7
10.00Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
10.00Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
9.09Single4O9RCyclopamine4O9R-SMO-Cyclopamine
9.09Single6LI0C176LI0-GPR52-C17
9.09Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
9.09Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
9.09Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
9.09Single9B9Y7DY9B9Y-CB1-7DY
8.33Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
8.33Single4BWBNeurotensin4BWB-NTS1-Neurotensin
8.33Single4QINSAG1.54QIN-SMO-SAG1.5
8.33Single5U09Taranabant5U09-CB1-Taranabant
8.33Single6FJ3PTH6FJ3-PTH1-PTH
8.33Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
8.33Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
8.33Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
8.33Single7BR3Elagolix7BR3-GnRH1-Elagolix
8.33Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
8.33Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
8.33Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
8.33Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
8.33Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
8.33Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
8.33Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
8.33Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
8.33Single9BA0A1AKN9BA0-CB1-A1AKN
8.33Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.33Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.33Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
8.33Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
8.33Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
8.33Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
7.69Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
7.69Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
7.69Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
7.69Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
7.69Single7VV6C48/807VV6-MRGPRX2-C48/80
7.69Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
7.69Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
7.69Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
7.69Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
7.69Consensusgrh_offOrthosteric Ligandgnrh1_off
7.69Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
7.69Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
7.14Single4QIMANTA XV4QIM-SMO-ANTA XV
7.14Single5T04Neurotensin5T04-NTS1-Neurotensin
7.14Single5TGZAM65385TGZ-CB1-AM6538
7.14Single6D27CAY104716D27-DP2-CAY10471
7.14Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
7.14Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
7.14Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
7.14Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
7.14Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
7.14Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
7.14Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
7.14Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
7.14Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
7.14Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
7.14Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
7.14Single7YXAONO-54306087YXA-S1P5-ONO-5430608
7.14Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
7.14Single9B9ZA1AKO9B9Z-CB1-A1AKO
7.14Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
7.14Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
7.14Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
7.14Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
7.14Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
6.67Single4JKVTaladegib4JKV-SMO-Taladegib
6.67Single5C1MBU725C1M-μ-BU72
6.67Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
6.67Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
6.67Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
6.67Single7C4SS1P7C4S-S1P3-S1P
6.67Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
6.67Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
6.67Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
6.67Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
6.67Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
6.67Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
6.67Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
6.67Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
6.67Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
6.67Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
6.25Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
6.25Single4BV0Neurotensin4BV0-NTS1-Neurotensin
6.25Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
6.25Single5V56TC1145V56-SMO-TC114
6.25Single5V57TC1145V57-SMO-TC114
6.25Single6OS1TRV0266OS1-AT1-TRV026
6.25Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
6.25Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
6.25Single7F1TMIP-1a7F1T-CCR5-MIP-1a
6.25Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
6.25Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
6.25Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
6.25Single7R0CAVP7R0C-V2-AVP-Arrestin2
6.25Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
6.25Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
6.25Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
6.25Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
6.25Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
6.25Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
6.25Single8E0GBU728E0G-μ-BU72
6.25Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.25Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
6.25Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
6.25Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
6.25Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
6.25Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
6.25Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
6.25Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
6.25Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
6.25Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
6.25Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
6.25Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
6.25Consensuslpa_onOrthosteric Ligandlpa1_on
6.25Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
6.25Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Consensusneurotensin_onOrthosteric Ligandnts1_on
6.25Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
6.25Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
6.25Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
6.25Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
5.88Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
5.88Single4XEENeurotensin4XEE-NTS1-Neurotensin
5.88Single4XESNeurotensin4XES-NTS1-Neurotensin
5.88Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
5.88Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
5.88Single6OS2TRV0266OS2-AT1-TRV026
5.88Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
5.88Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
5.88Single6YVRNTS8-136YVR-NTS1-NTS8-13
5.88Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
5.88Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
5.88Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
5.88Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
5.88Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
5.88Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
5.88Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
5.88Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
5.88Single8XQJJN2418XQJ-Apelin-JN241
5.88Single8XWACXCL18XWA-CXCR2-CXCL1
5.88Single8XWMCXCL68XWM-CXCR2-CXCL6
5.88Single8XWSCXCL58XWS-CXCR2-CXCL5
5.88Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
5.88Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
5.88Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
5.88Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
5.88Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
5.88Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
5.88Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
5.88Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
5.88Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
5.88Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
5.88Consensuslpa_offOrthosteric Ligandlpa1_off
5.88Consensuslpl_offOrthosteric Ligands1p_off lpa_off
5.88Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
5.88Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
5.88Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
5.88Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
5.88Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
5.88Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
5.88Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
5.88Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
5.56Single4BUONeurotensin4BUO-NTS1-Neurotensin
5.56Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
5.56Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
5.56Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
5.56Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
5.56Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
5.56Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
5.56Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
5.56Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
5.56Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
5.56Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
5.56Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
5.56Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
5.56Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
5.56Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
5.56Single8XVUCXCL28XVU-CXCR2-CXCL2
5.56Single8XWFCXCL38XWF-CXCR2-CXCL3
5.56Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
5.56Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
5.56Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
5.56Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
5.56Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
5.56Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
5.56Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
5.56Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
5.26Single6KNMJN241-96KNM-Apelin-JN241-9
5.26Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
5.26Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
5.26Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
5.26Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
5.26Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
5.26Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
5.26Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
5.26Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
5.26Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
5.26Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single8QJ2pN1628QJ2-MC4-pN162-Gs
5.26Single8XQJJN2418XQJ-Apelin-JN241
5.26Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
5.26Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
5.26Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
5.26Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
5.26Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
5.26Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
5.26Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
5.00Single4XT1Fractalkine4XT1-US28-Fractalkine
5.00Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
5.00Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
5.00Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
5.00Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
5.00Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
5.00Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
5.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
5.00Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
5.00Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
5.00Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
5.00Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
5.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.00Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
5.00Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
5.00Single8XWNCXCL88XWN-CXCR2-CXCL8
5.00Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
5.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
5.00Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
5.00Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
5.00Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
5.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
5.00Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
5.00Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
5.00Consensuslpl_onOrthosteric Ligands1p_on lpa_on
5.00Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
5.00Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
5.00Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
4.76Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
4.76Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
4.76Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
4.76Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
4.76Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
4.76Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
4.76Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
4.76Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
4.76Single7SK5CXCL127SK5-ACKR3-CXCL12
4.76Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
4.76Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
4.76Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
4.76Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
4.76Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
4.76Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
4.76Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
4.76Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
4.76Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
4.76Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
4.76Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
4.55Single3OE0CVX153OE0-CXCR4-CVX15
4.55Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
4.55Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
4.55Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
4.55Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
4.55Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
4.55Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
4.55Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
4.55Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
4.55Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
4.55Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
4.55Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
4.55Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
4.55Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
4.55Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
4.55Consensusangiotensin_onOrthosteric Ligandat1_on
4.55Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
4.55Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
4.55Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
4.55Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
4.55Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
4.55Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
4.55Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
4.55Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
4.55Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
4.35Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
4.35Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
4.35Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
4.35Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
4.35Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
4.35Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
4.35Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
4.35Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
4.35Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
4.35Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
4.35Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
4.35Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
4.35Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
4.35Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
4.35Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
4.35Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
4.35Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
4.35Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
4.35Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
4.35Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
4.35Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
4.35Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
4.35Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
4.35Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
4.35Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
4.35Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
4.35Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
4.35Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
4.35Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
4.35Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
4.35Consensusvasop-oxy_onOrthosteric Ligandv2_on
4.35Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
4.17Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
4.17Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
4.17Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
4.17Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
4.17Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
4.17Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
4.17Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
4.17Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
4.17Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
4.17Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
4.17Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
4.17Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
4.17Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
4.17Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
4.17Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
4.17Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
4.17Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
4.17Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
4.17Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
4.17Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
4.17Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
4.17Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
4.17Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
4.17Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
4.17Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
4.17Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
4.17Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
4.17Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
4.17Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
4.00Single4XT3Fractalkine4XT3-US28-Fractalkine
4.00Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
4.00Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
4.00Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
4.00Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
4.00Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
4.00Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
4.00Single7SK3CXCL127SK3-ACKR3-CXCL12
4.00Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
4.00Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
4.00Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
4.00Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
4.00Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
4.00Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
4.00Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
4.00Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
4.00Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
4.00Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
4.00Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
4.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
4.00Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
4.00Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
4.00Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
3.85Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
3.85Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
3.85Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
3.85Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
3.85Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
3.85Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
3.85Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
3.85Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
3.85Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
3.85Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
3.85Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
3.85Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
3.85Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
3.85Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
3.85Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
3.85Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3
3.85Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
3.85Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
3.85Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
3.85Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
3.85Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
3.85Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
3.85Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
3.85Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
3.70Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
3.70Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
3.70Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
3.70Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
3.70Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
3.70Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
3.70Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
3.70Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
3.70Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
3.70Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
3.70Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
3.70Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
3.70Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
3.70Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
3.70Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
3.70Single8IY6Endothelin-18IY6-ETB-Endothelin-1
3.70Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
3.70Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
3.70Consensusbradykinin_onOrthosteric Ligandbk2_on
3.70Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
3.70Consensusendothelin_onOrthosteric Ligandetb_on eta_on
3.70Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
3.70Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
3.57Single5GLHEndothelin-15GLH-ETB-Endothelin-1
3.57Single6IGKEndothelin-36IGK-ETB-Endothelin-3
3.57Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
3.57Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
3.57Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
3.57Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
3.57Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
3.57Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
3.57Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
3.57Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
3.45Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
3.45Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
3.45Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
3.45Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
3.45Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
3.45Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
3.45Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
3.45Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
3.45Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
3.45Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
3.45Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
3.33Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
3.33Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
3.33Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
3.33Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
3.33Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
3.33Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
3.33Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.23Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
3.23Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
3.23Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
3.23Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
3.23Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
3.23Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
3.23Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
3.23Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.12Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
3.03Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
3.03Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
2.94Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
2.86Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
2.78Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
2.56Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1

PDB Summary
PDB 7FIG
Class A
SubFamily Protein
Type Glycoprotein Hormone
SubType LH
Species Homo Sapiens
Ligand hCG
Other Ligand(s) -
Protein Partners chim(NtGi1L-Gs)/Beta1/Gamma2
PDB Resolution 3.9
Date 2021-09-29
D.O.I. 10.1038/s41586-021-03924-2
Net Summary
Imin 4.11
Number of Linked Nodes 1365
Number of Links 1738
Number of Hubs 293
Number of Links mediated by Hubs 1115
Number of Communities 34
Number of Nodes involved in Communities 392
Number of Links involved in Communities 594
Path Summary
Number Of Nodes in MetaPath 217
Number Of Links MetaPath 216
Number of Shortest Paths 67121727
Length Of Smallest Path 3
Average Path Length 128
Length of Longest Path 82
Minimum Path Strength 1.225
Average Path Strength 16.0014
Maximum Path Strength 34.055
Minimum Path Correlation 0.74
Average Path Correlation 1
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.08333
Average % Of Corr. Nodes 99.2046
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 66.1618
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .
CodeCMS
PDB ResiduesA:A:?10 A:A:?237 A:A:?359 A:A:?365 A:A:?379 B:B:?25 B:B:?103 B:B:?114 B:B:?121 B:B:?148 B:B:?149 B:B:?166 B:B:?204 B:B:?218 B:B:?233 B:B:?250 B:B:?271 B:B:?294 B:B:?317 G:G:?41 L:L:?31 L:L:?34 L:L:?52 L:L:?55 L:L:?56 L:L:?83 L:L:?84 L:L:?106 L:L:?108 L:L:?111 N:N:?29 N:N:?43 N:N:?46 N:N:?54 N:N:?58 N:N:?77 N:N:?92 N:N:?108 N:N:?110 N:N:?113 N:N:?120 N:N:?130 R:R:?131 R:R:?156 R:R:?279 R:R:?280 R:R:?336 R:R:?343 R:R:?353 R:R:?399 R:R:?407 R:R:?439 R:R:?514 R:R:?543 R:R:?545 R:R:?581 R:R:?617 R:R:?643 R:R:?644
Environment DetailsOpen EMBL-EBI Page
CodeCMS
NameCARBAMOYL SARCOSINE
Synonyms
Identifier
FormulaC4 H8 N2 O3
Molecular Weight132.118
SMILES
PubChem439375
Formal Charge0
Total Atoms17
Total Chiral Atoms0
Total Bonds16
Total Aromatic Bonds0

CodeLMS
PDB ResiduesA:A:?17 A:A:?24 A:A:?28 A:A:?32 A:A:?34 A:A:?53 A:A:?58 A:A:?211 A:A:?216 A:A:?233 A:A:?274 A:A:?293 A:A:?300 A:A:?305 A:A:?307 A:A:?338 B:B:?15 B:B:?23 B:B:?57 B:B:?78 B:B:?89 B:B:?127 B:B:?209 B:B:?280 B:B:?301 B:B:?337 G:G:?14 G:G:?20 G:G:?29 G:G:?32 G:G:?46 L:L:?68 L:L:?69 L:L:?75 L:L:?87 L:L:?99 L:L:?115 N:N:?22 N:N:?40 N:N:?124 R:R:?62 R:R:?77 R:R:?109 R:R:?126 R:R:?137 R:R:?143 R:R:?180 R:R:?205 R:R:?212 R:R:?225 R:R:?233 R:R:?257 R:R:?258 R:R:?339 R:R:?390 R:R:?423 R:R:?477 R:R:?510 R:R:?548 R:R:?563 R:R:?566 R:R:?569 R:R:?570 R:R:?595 R:R:?605 R:R:?628 R:R:?640
Environment DetailsOpen EMBL-EBI Page
CodeLMS
Name[(2r,3s,4r,5r)-5-(6-Amino-9h-Purin-9-Yl)-3,4-Dihydroxytetrahydro-2-Furanyl]Methyl Sulfamate
Synonyms[(2r,3s,4r,5r)-5-(6-Amino-9h-Purin-9-Yl)-3,4-Dihydroxytetrahydro-2-Furanyl]Methyl Sulfamate
Identifier
FormulaC10 H14 N6 O6 S
Molecular Weight346.32
SMILES
PubChem97576
Formal Charge0
Total Atoms37
Total Chiral Atoms4
Total Bonds39
Total Aromatic Bonds10

CodeTMR
PDB ResiduesA:A:?37 A:A:?63 A:A:?253 A:A:?311 A:A:?318 A:A:?339 A:A:?358 A:A:?360 A:A:?391 B:B:?59 B:B:?85 B:B:?105 B:B:?111 B:B:?124 B:B:?145 B:B:?264 B:B:?289 G:G:?40 L:L:?61 L:L:?89 L:L:?112 L:L:?113 N:N:?57 N:N:?79 N:N:?102 R:R:?58 R:R:?113 R:R:?127 R:R:?182 R:R:?240 R:R:?254 R:R:?275 R:R:?331 R:R:?333 R:R:?359 R:R:?389 R:R:?411 R:R:?426 R:R:?427 R:R:?455 R:R:?470 R:R:?508 R:R:?527 R:R:?546 R:R:?550 R:R:?612 R:R:?623
Environment DetailsOpen EMBL-EBI Page
CodeTMR
Name2,6-dideoxy-4-S-methyl-4-thio-beta-D-ribo-hexopyranose
Synonyms2,6-DIDEOXY-4-THIOMETHYL-BETA-D-RIBOHEXOPYRANOSIDE; 2,6-dideoxy-4-S-methyl-4-thio-beta-D-ribo-hexose; 2,6-dideoxy-4-S-methyl-4-thio-D-ribo-hexose; 2,6-dideoxy-4-S-methyl-4-thio-ribo-hexose
Identifier
FormulaC7 H14 O3 S
Molecular Weight178.249
SMILES
PubChem447846
Formal Charge0
Total Atoms25
Total Chiral Atoms4
Total Bonds25
Total Aromatic Bonds0

CodeGLM
PDB ResiduesA:A:?47 A:A:?52 A:A:?225 A:A:?304 A:A:?329 A:A:?353 A:A:?355 B:B:?41 B:B:?53 B:B:?64 B:B:?77 B:B:?109 B:B:?115 B:B:?116 B:B:?131 B:B:?141 B:B:?144 B:B:?162 B:B:?174 B:B:?182 B:B:?185 B:B:?202 B:B:?216 B:B:?224 B:B:?238 B:B:?244 B:B:?272 B:B:?282 B:B:?288 B:B:?306 B:B:?310 B:B:?319 B:B:?324 B:B:?330 L:L:?46 L:L:?54 L:L:?96 L:L:?97 N:N:?42 N:N:?56 N:N:?67 N:N:?91 N:N:?95 N:N:?121 N:N:?122 R:R:?71 R:R:?117 R:R:?134 R:R:?166 R:R:?171 R:R:?183 R:R:?185 R:R:?196 R:R:?216 R:R:?220 R:R:?223 R:R:?241 R:R:?328 R:R:?334 R:R:?358 R:R:?376 R:R:?409 R:R:?424 R:R:?436 R:R:?438 R:R:?443 R:R:?489 R:R:?490 R:R:?504 R:R:?642
Environment DetailsOpen EMBL-EBI Page
CodeGLM
Name
Synonyms
Identifier
Formula
Molecular Weight
SMILES
PubChem
Formal Charge
Total Atoms
Total Chiral Atoms
Total Bonds
Total Aromatic Bonds

CodeNAG
PDB ResiduesH:H:?1 H:H:?2 H:H:?3 H:H:?4 H:H:?5
Environment DetailsOpen EMBL-EBI Page
CodeNAG
NameN-Acetylglucosamine
SynonymsN-Acetyl-D-glucosamine
Identifier
FormulaC8 H15 N O6
Molecular Weight221.208
SMILES
PubChem24139
Formal Charge0
Total Atoms30
Total Chiral Atoms5
Total Bonds30
Total Aromatic Bonds0

PDBsumOpen PDBsum Page
ChainA
ProteinG Protein α Sub unit
UniProtP04896
Sequence
>7FIG_Chain_A
?TLSAED?A AVERS?MIE ?QLQ?D?QV ?RATHRLLL L?ADNS??S 
TIV?QMRI? HVNIFET?F QVD?VNFHM FDV?AQRDE RR?WIQ?FN 
DVTAIIFVV DSSD?NRLQ EALNDF?SI WNNRWLRTI SVILFLN?Q 
DLLAE?VLA ??S?IED?F PEFAR?TTP EDATPEP?E DPRVTRA?? 
FIRDEFLRI STAS?D?RH ???PHFT?S VDTENARRI FND?RDIIQ 
RMHLRQ?EL L


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainB
ProteinG Protein β Sub unit
UniProtP54311
Sequence
>7FIG_Chain_B
ELDQLRQEA EQL?NQIRD AR?A?ADAT LSQITNNID PV?RIQMRT 
RRTLR?HLA ?I?AMHW?T DSRLLVSAS QD??LIIWD S?TTN?VHA 
IPLRSSWVM T?A?APS?N ?VA???LDN I?SI?NL?T RE?NVRVSR 
ELA?HT??L S??RFLDDN QIVTSS?DT T?ALWDIET ?QQTTTFT? 
HT?DVMSLS LAPDTRLFV S?A?DASA? LWDVRE?M? RQTFT?HES 
DINAI?FFP N?NAFAT?S DDAT?RLFD LRADQELMT ?SHDNII?? 
ITSVSFS?S ?RLLLA??D DFN?NVWDA L?ADRA?VL A?HDNRVS? 
L?VTDD?MA VAT?SWDSF L?IWN


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainG
ProteinG Protein γ Sub unit
UniProtP63212
Sequence
>7FIG_Chain_G
TASIAQAR? LVEQL?MEA NIDRI?VS? AAADLMA?? EAHA?EDPL 
LTPVPASEN PFR


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainR
ProteinReceptor
UniProtP22888
Sequence
>7FIG_Chain_R
TRLSLA?LP V?VIPSQAF R?LNEVI?I EISQIDSLE RIEANAFDN 
LLNLSEILI QNT?NLR?I EP?AFINLP RL??LSI?N T?IR?FPDV 
T?VFSSESN FILEI?DNL HITTIP?NA FQ?MNNESV TL?L??N?F 
EEVQSHAFN ?TTLTSLEL ?ENVHLE?M HN?AFR?AT ?P?TLDISS 
T?LQALPS? ?LESIQRLI ATSS?SL?? LPSRETFVN LLEATLT?P 
IH??AFRNL P?WD?E??F ?LP?TPR?A PEPDAFNP? EDIM??DFL 
RVLIWLINI LAIM?NMTV LFVLLTSR? ?LTVPRFLM ?NLSFADF? 
M?L?LLLIA SVDSQT??Q ??NHAIDWQ T?S??STA? FFTVFASEL 
SV?TLTVIT LERWHTIT? AIHLDQ?LR LRHAILIML ??WLFSSLI 
AMLPLV?VS N?M?VSI?F PMDVETTLS QV?ILTILI LNVVAFFII 
?A??I?I?F AVRNPELMA TN?DT?IA? ?MAILIFTD FT?MAPISF 
FAISAAF?V PLITVTNS? VLLVLF?PI NS?ANPFL? AIFT?TFQR 
DFFLLLS?F ???


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  




This receptor, from the same or other species and bound to the same or other ligands, is also present in the following networks:
Show PDB Class SubFamily Type SubType Species Orthosteric Ligand Other Ligand(s) Protein Partners Resolution Date DOI
6ZFZAAmineAcetylcholine (muscarinic)M1Homo sapiens77-LH-28-1--2.172021-10-0610.1016/j.cell.2021.11.001
7FIJAProteinGlycoprotein HormoneLHHomo sapiens---3.82021-09-2910.1038/s41586-021-03924-2
7FIIAProteinGlycoprotein HormoneLHHomo sapienshCG-chim(NtGi1-Gs)/β1/γ24.32021-09-2910.1038/s41586-021-03924-2
7FII (No Gprot) AProteinGlycoprotein HormoneLHHomo sapienshCG-4.32021-09-2910.1038/s41586-021-03924-2
7FIHAProteinGlycoprotein HormoneLHHomo sapienshCGOrg43553chim(NtGi1-Gs)/β1/γ23.22021-09-2910.1038/s41586-021-03924-2
7FIH (No Gprot) AProteinGlycoprotein HormoneLHHomo sapienshCGOrg435533.22021-09-2910.1038/s41586-021-03924-2
7FIGAProteinGlycoprotein HormoneLHHomo sapienshCG-chim(NtGi1L-Gs)/β1/γ23.92021-09-2910.1038/s41586-021-03924-2
7FIG (No Gprot) AProteinGlycoprotein HormoneLHHomo sapienshCG-3.92021-09-2910.1038/s41586-021-03924-2
5OLHANucleotideAdenosineA2AHomo sapiensVipadenantNa-2.62018-01-1710.1038/s41598-017-18570-w
5GLHAPeptideEndothelinETBHomo sapiensEndothelin-1--2.82016-09-0710.1038/nature19319




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