Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.hns1.01 7.205404
2G.H1.01 5.15409
3G.S2.08 4.115476
4G.S3.03 6.9854178
5G.S3.06 12.465427
6G.H2.06 6.315629
7G.H2.07 4.5975409
8G.h2s4.01 11.3409
9G.S4.06 4.9675407
10G.H3.09 4.34143739
11G.H3.13 8.13167636
12G.H3.17 11.9967625
13G.S5.03 5.63754149
14G.S5.05 5.3625149
15G.hgh4.02 4.2725408
16G.hgh4.08 8.3275436
17G.hgh4.11 3.4625435
18G.hgh4.20 10.0825403
19G.H4.07 10.2625435
20G.H4.08 8.7225433
21G.H4.10 9.712507
22G.H4.12 5.76714734
23G.H4.15 8.715408
24G.H4.16 4.256534
25G.h4s6.02 4.226537
26G.h4s6.12 6.6275432
27G.h4s6.20 6.655474
28G.S6.02 7.864578
29G.S6.03 4.7525435
30G.S6.05 9.6525435
31G.s6h5.01 5.86754149
32G.H5.05 5.6675475
33G.H5.08 6.62578
34G.H5.12 6.085477
35G.H5.17 8.15675
36G.H5.23 7.382594
37b.1x3 3.4625408
38b.1x10 4.2075408
39b.h2x1 4.2825115
40b.lhb1x3 3.616502
41b.lhb1x6 5.2745113
42b.lhb1x11 4.7125484
43b.l1x3 8.73714749
44b.l1x6 9.914529
45b.b2x1 8.516528
46b.b2x5 6.76547
47b.b3x4 5.6725449
48b.b4x3 3.5685107
49b.b4x5 5.364107
50b.b4x6 11.4467649
51b.l4x1 5.1075445
52b.b5x3 6.962509
53b.l5x1 4.3665108
54b.l5x5 8.67714729
55b.b6x1 4.4825429
56b.b6x2 4.1125408
57b.b7x1 5.5275404
58b.b7x4 4.1254108
59b.l7x2 4.165429
60b.b8x3 3.055406
61b.b8x4 6.2865106
62b.l8x3 4.7425403
63b.l9x3 6.9745159
64b.l9x6 6.03333628
65b.l9x7 3.49407
66b.b10x2 3.5425466
67b.b10x5 4.582509
68b.l10x3 5.6406
69b.b11x4 5.35754159
70b.b11x5 4.0125466
71b.b12x6 10.11336158
72b.b12x7 3.7375409
73b.b13x3 9.58754154
74b.b13x7 10.625467
75b.l13x3 8.544569
76b.l13x6 7.29409
77b.b14x3 4.5575465
78b.b15x1 9.055469
79b.b15x2 9.5925456
80b.l15x1 5.5225427
81b.b16x4 9.83566
82b.b16x5 7.2775455
83b.b16x6 8.85833668
84b.b17x5 7.474557
85b.b17x7 10.3325458
86b.l17x3 9.91667659
87b.b18x3 5.4825458
88b.l18x1 6.268336166
89b.l18x2 6.034167
90b.b19x2 9.8925456
91b.l19x2 7.06167659
92b.b20x2 6.9225456
93b.b20x4 9.72833658
94b.b20x6 7.826556
95b.l20x2 9.795409
96b.b21x1 10.3875457
97b.b21x6 5.6825451
98b.b21x7 5.991676125
99b.l21x9 5.68406
100b.b22x5 4.846167
101b.l22x5 7.865119
102b.b23x6 8.281676127
103b.l23x1 8.755426
104b.b24x3 3.752585
105b.b24x4 10.54126
106b.b24x5 3.81505
107b.l24x2 5.86254116
108b.l25x3 7.47833689
109b.l25x6 12.88528
110b.l25x7 3.9175487
111b.b26x3 3.844586
112b.l26x1 6.325447
113b.b27x1 4.5825486
114b.b27x3 4.534588
115b.l27x1 9.955629
116b.l27x2 7.3125489
117b.b28x4 6.6486
118b.b28x6 8.41333689
119g.l1x4 5.216508
120g.h2x11 9.4854166
121g.h2x15 6.3775406
122g.ctx3 5.05833609
123g.ctx6 3.7454116
124g.ctx15 9.47449
125g.ctx16 7.04857748
126Lig 12.54093410
127NT.W67 9.63406
128NT.T71 7.884135
129NT.W73 6.775139
130NT.T76 5.564137
131NT.F90 5.09415
132NT.R103 7.4385138
133NT.W110 14.62754139
134NT.Y118 7.1525417
135NT.K127 4.285403
1361x40 2.8925415
1371x43 6.12833618
1381x47 6.934518
1391x54 4.325409
1401x64 5.99254256
1412x50 7.9975499
1422x54 4.085408
1432x56 4.775419
1442x57 7.35571718
1452x60 8.842518
1462x67 10.455417
1472x71 4.4725407
1483x36 7.554517
1493x41 5.416515
1503x44 7.8375418
1513x45 7.14415
1523x46 9.958519
1533x50 9.14409
1543x53 7.76833698
1553x54 7.0525499
1563x55 5.26408
1573x58 6.325498
158I2.F248 7.965476
1594x53 6.745419
1604x60 7.9525418
1614x64 11.075418
162E2x50 3.86419
163E2x51 11.77519
1645x37 9.974517
1655x39 6.87417
1665x54 7.33254189
1675x64 9.295479
168I3.D327 5.155436
169I3.I328 4.865436
1706x49 5.374509
1716x52 7.626518
1726x53 9.858518
1736x56 7.4125406
1747x49 6.35333619
1757x58 3.97409
1768x53 7.8954257
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.l1x4 b.l3x2 15.71112.21NoNo069
2G.hns1.01 b.l1x4 16.03063.52YesNo046
3G.S1.03 G.hns1.01 16.819917.49NoYes094
4G.S1.03 G.S3.06 17.02035.34NoYes097
5G.S3.06 b.l5x5 18.616924.05YesYes279
6G.h2s4.01 b.l5x5 94.120812.03YesYes099
7G.H2.07 G.h2s4.01 94.37796.01YesYes099
8G.H2.07 G.S3.08 1003.68YesNo099
9G.S3.07 G.S3.08 99.87972.92NoNo099
10G.H1.01 G.S3.07 99.83915.53YesNo099
11G.H1.01 G.s1h1.05 99.63234.59YesNo099
12G.S4.05 G.s1h1.05 99.50524.85NoNo079
13G.H1.04 G.S4.05 98.37523.07NoNo2277
14G.H1.04 G.H1.08 99.06492.92NoNo079
15G.H1.08 G.H5.04 98.78865.83NoNo098
16G.H5.04 G.S2.08 98.74163.07NoYes086
17G.H5.08 G.S2.08 98.28036.55YesYes786
18b.l5x5 b.l7x2 29.6715.69YesYes299
19b.l7x2 b.l9x6 29.28893.52YesYes298
20b.l13x6 b.l9x6 18.70111.49YesYes098
21G.H2.06 b.l9x6 21.1323.58YesYes298
22G.H2.04 G.H2.07 14.75374NoYes099
23G.H2.04 G.H3.08 14.55189.72NoNo098
24G.H2.06 b.l19x1 21.88275.53YesNo299
25b.b22x1 b.l25x6 36.28573.88NoYes288
26b.b22x1 b.b22x2 38.70443.2NoNo088
27b.b22x2 b.b26x3 38.46044.5NoYes086
28b.b26x3 b.b27x1 15.4682.98YesYes866
29G.H3.17 b.l23x1 17.98546.7YesYes256
30G.H3.17 b.l27x1 16.296210.31YesYes259
31b.l1x6 b.l27x1 28.544213.92YesYes299
32b.l1x6 b.l3x1 28.773812.2YesNo299
33b.l3x1 b.l5x5 57.62874.38NoYes299
34b.b2x1 b.l27x1 37.57284.82YesYes289
35b.b2x1 b.l3x1 28.807318.04YesNo289
36G.H5.08 G.H5.12 97.11767.48YesYes787
37G.H5.12 G.H5.16 16.65354.67YesNo776
385x64 G.H5.16 16.606913.56YesNo796
39G.H5.10 G.S6.02 13.990913.79NoYes078
405x64 G.H5.17 11.40549.9YesYes795
41G.H3.08 G.S4.04 14.16567.31NoNo089
42G.H3.09 G.S4.04 12.93114.29YesNo099
43G.H4.12 G.H4.16 11.91883.64YesYes344
44G.H4.16 G.h4s6.02 14.06633YesYes347
45G.H3.09 G.h4s6.02 10.49673.96YesYes397
46G.H5.12 I2.S247 81.30247.91YesNo777
47G.H5.15 I2.S247 81.3746.19NoNo087
48G.H5.15 G.H5.19 81.29923.98NoNo088
493x57 G.H5.19 80.99886.43NoNo078
50G.H5.20 G.H5.26 11.59144.15NoNo088
513x53 3x57 80.084817.58YesNo987
52b.b27x3 b.l25x3 11.3856.85YesYes889
53b.b26x3 b.b27x3 15.93714.42YesYes868
54b.l17x5 b.l19x1 21.72494.42NoNo069
55b.l17x5 b.l19x2 21.54862.94NoYes069
56b.b20x4 b.l19x2 15.2833.57YesYes589
57b.b20x4 b.b20x6 14.80226.41YesYes586
58b.b17x7 b.b20x6 11.423911.79YesYes586
59b.b27x1 g.ctx5 13.48664.47YesNo069
60g.ctx3 g.ctx5 13.21715.43YesNo099
61b.b21x5 b.h2x1 10.19824.24NoYes045
62b.l11x1 b.l13x6 19.43755.03NoYes099
63b.b11x6 b.l11x1 19.25573.71NoNo099
64b.b11x6 b.l9x3 19.073615.34NoYes099
65b.b11x4 b.l9x3 17.75745.48YesYes1599
66b.b11x4 b.l9x7 11.30074.42YesYes097
67b.b6x2 b.l9x7 10.72142.95YesYes087
68b.b10x2 b.b6x2 10.14293.38YesYes068
69b.l21x7 b.l23x1 30.55844.67NoYes056
70b.b23x6 b.l21x7 29.55474.03YesNo075
71b.b23x6 b.b24x6 20.434410.61YesNo1278
72b.b21x7 b.b24x6 19.99646.75YesNo1258
73b.b21x5 b.b21x7 10.663610.78NoYes045
742x49 3x53 76.02583.63NoYes098
752x49 3x50 73.80426.83NoYes099
762x53 3x50 80.971411.93NoYes099
772x53 2x56 35.67953NoYes199
782x56 3x43 35.27125.96YesNo198
792x60 3x43 70.68314.46YesNo188
802x60 Lig 61.04015.96YesYes180
812x53 2x57 45.19866.09NoYes198
822x57 3x43 35.709720.54YesNo188
83Lig NT.N69 15.483913.83YesNo104
84NT.L70 NT.N69 15.13734.12NoNo064
85NT.L70 NT.T71 14.79062.95NoYes065
86b.l25x6 b.l27x1 49.31715.99YesYes289
87b.l23x1 b.l25x6 14.821217.87YesYes268
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x36Lig5.911YesYes7010
3x37Lig10.171NoYes7010
3x40Lig13.911NoYes5010
5x37Lig9.181YesYes7010
7x38Lig11.241NoYes6010
7x41Lig4.311NoYes7010
7x42Lig17.951NoYes7010
1x47Lig5.751YesYes8010
2x60Lig5.961YesYes8010
E2.I289Lig11.691NoYes8010
E3.K365Lig3.041NoYes2010
1x36Lig16.071NoYes4010
1x40Lig3.671YesYes5010
1x43Lig11.351YesYes8010
2x67Lig12.011YesYes7010
E1.F200Lig28.791NoYes4010
E2x52Lig11.571NoYes5010
E2.T288Lig6.621NoYes4010
1x33Lig2.951NoYes2010
E1.E204Lig17.160NoYes4010
LigNT.E367.721YesNo0601
LigNT.C378.081YesNo0601
LigNT.F937.231YesNo0401
1x29Lig10.850NoYes1010
LigNT.D1268.161YesNo0101
LigNT.V405.051YesNo0301
LigNT.F906.091YesYes0501
LigNT.N6913.831YesNo0401
LigNT.Y1183.51YesYes0701
NT.E36NT.L9215.91NoNo6412
E1.C208NT.C377.280NoNo4621
NT.Q41NT.V404.30NoNo4321
NT.L70NT.N694.120NoNo6421
NT.C122NT.F906.980NoYes9521
NT.D125NT.F904.780NoYes2521
NT.P119NT.Y11812.520NoYes5721
NT.I120NT.Y1187.250NoYes6721
NT.A121NT.Y1185.340NoYes5721
NT.A121NT.D1254.630NoNo5222
1x301x334.230NoNo2221
1x321x369.020NoNo3421
1x367x383.591NoNo4611
1x401x434.781YesYes5811
1x431x443.751YesNo8712
1x431x472.981YesYes8811
1x432x688.051YesNo8712
1x437x425.861YesNo8711
1x472x608.231YesYes8811
1x472x6412.621YesNo8712
1x477x465.091YesNo8912
2x603x409.151YesNo8511
2x603x4314.461YesNo8812
2x603x446.411YesYes8812
2x643x365.240NoYes7721
2x672x684.151YesNo7712
2x672x717.051YesYes7712
2x673x3618.611YesYes7711
2x71E1.F2006.090YesNo7421
3x363x405.241YesNo7511
3x375x373.291NoYes7711
3x375x395.491NoYes7712
3x446x5312.381YesYes8822
4x64E2.T2883.881YesNo8421
E2x50E2x524.671YesNo9521
5x33E2.T2888.770NoNo3421
5x37E2.I28915.271YesNo7811
5x375x397.051YesYes7712
5x375x4015.081YesNo7712
6x537x418.981YesNo8721
E3.D362E3.K3654.150NoNo4221
7x37E3.K3658.620NoNo8221
7x377x418.10NoNo8721
2x633x362.770NoYes6721
1x39Lig2.620NoYes5010
NT.F90NT.I892.511YesNo5512
NT.F93NT.K1272.481NoYes4312
1x371x401.740NoYes3521
E1.S205Lig1.530NoYes1010
3x33Lig1.510NoYes5010
1x40E1.D2011.381YesNo5412

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
95.45Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
76.00Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
75.00Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
73.08Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
71.43Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
69.23Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
69.23Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
67.86Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
67.86Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
66.67Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
66.67Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
64.29Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
64.29Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
58.06Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
51.52Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
51.43Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
50.00Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
48.57Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
48.39Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
48.39Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
46.67Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
45.16Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
44.83Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
44.83Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
43.75Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
43.33Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
42.42Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
41.94Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
41.94Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
41.94Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
41.94Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
41.94Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
41.94Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
41.94Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
41.18Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
40.62Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
40.62Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
40.62Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
40.62Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
40.00Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
40.00Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
40.00Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
39.39Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
39.39Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
39.39Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
39.39Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
39.39Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
39.39Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
38.71Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
38.71Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
38.71Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
38.46Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
38.24Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
38.24Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
37.93Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
37.50Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
37.50Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
37.50Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
37.50Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
37.50Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
37.50Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
37.14Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
37.14Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
36.36Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
36.36Consensusglp_onOrthosteric Ligandglp1_on glp2_on
36.36Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
36.11Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
36.11Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
36.11Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
35.48Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
35.48Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
35.48Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
35.29Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
35.14Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
35.14Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
34.38Consensuscalcitonin_onOrthosteric Ligandctlike_on
34.38Consensuspac_onOrthosteric Ligandpac1_on
34.38Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
34.29Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
34.21Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
33.33Single6FJ3PTH6FJ3-PTH1-PTH
33.33Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
33.33Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
33.33Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
33.33Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
33.33Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
33.33Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
33.33Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
33.33Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
33.33Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
32.56Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
32.43Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
32.43Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
32.35Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
32.35Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
32.35Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
32.35Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
32.35Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
32.26Single5WF5UK-4320975WF5-A2A-UK-432097
32.26Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
32.14Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
32.14Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
32.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
32.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
31.58Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
31.58Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
31.58Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
31.58Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
31.43Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
31.43Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
31.43Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
31.43Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
31.43Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
31.43Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
31.25Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
31.25Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
31.25Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
31.25Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
31.25Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
31.25Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
31.25Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
31.25Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
31.25Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
31.03Single7SK9CCX6627SK9-ACKR3-CCX662
31.03Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
30.77Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
30.77Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
30.30Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
30.30Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
30.00Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
30.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
30.00Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
29.73Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
29.73Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
29.73Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
29.63Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
29.41Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
29.41Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
29.27Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
29.27Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
29.17Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
29.17Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
29.03Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
29.03Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
29.03Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
28.95Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
28.57Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
28.57Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
28.57Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
28.57Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
28.21Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
28.21Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.21Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
28.12Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
28.12Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
28.12Consensusangiotensin_onOrthosteric Ligandat1_on
28.12Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
28.00Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
27.91Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
27.78Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
27.78Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
27.78Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
27.59Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
27.59Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
27.59Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
27.59Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
27.27Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
27.27Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
27.27Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
27.27Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
27.27Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
27.27Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.03Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
27.03Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
26.92Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
26.92Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
26.92Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
26.92Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
26.92Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
26.92Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
26.92Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
26.92Consensushca_on_gpOrthosteric Ligandhca2_on_gp
26.67Single4UG2CGS216804UG2-A2A-CGS21680
26.67Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
26.67Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
26.67Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
26.47Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
26.47Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
26.47Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
26.47Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
25.93Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
25.93Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
25.93Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
25.93Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
25.93Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
25.93Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
25.93Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
25.93Consensusa3_on_gpOrthosteric Liganda3a_on_gp
25.93Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
25.93Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
25.93Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
25.93Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
25.81Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
25.81Single7QA8Peptide7QA8-STE2-Peptide
25.81Single7QA8Peptide7QA8-STE2-Peptide
25.81Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
25.81Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
25.81Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
25.81Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
25.81Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
25.81Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
25.81Consensuslpl_onOrthosteric Ligands1p_on lpa_on
25.81Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
25.81Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
25.71Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
25.71Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
25.71Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
25.71Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
25.71Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
25.00Single2YDVNECA2YDV-A2A-NECA
25.00Single3QAKUK-4320973QAK-A2A-UK-432097
25.00Single4UHRCGS216804UHR-A2A-CGS21680
25.00Single5G53NECA5G53-A2A-NECA-Gs
25.00Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
25.00Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
25.00Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
25.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
25.00Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
25.00Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
25.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
25.00Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
25.00Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
25.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
25.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
25.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
25.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
25.00Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
25.00Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
25.00Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
25.00Single8K5BNiacin8K5B-HCA2-Niacin
25.00Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
25.00Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
25.00Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
25.00Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
25.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
25.00Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
25.00Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.00Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
25.00Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
25.00Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
25.00Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
25.00Consensusrelaxin_onOrthosteric Ligandrxfp4_on
25.00Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
25.00Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
25.00Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
25.00Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
25.00Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
25.00Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
24.39Consensuspth_onOrthosteric Ligandpth1_on pth2_on
24.32Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
24.32Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
24.32Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
24.24Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
24.24Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
24.24Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
24.24Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.24Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
24.24Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
24.24Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
24.24Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
24.14Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
24.14Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
24.14Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
24.14Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
24.14Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
24.14Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
24.14Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
24.14Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
24.14Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
24.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
24.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
24.00Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
24.00Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
24.00Single8IWESpermidine8IWE-TA9-Spermidine
24.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
24.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
24.00Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
24.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
24.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
24.00Consensusangiotensin_offOrthosteric Ligandat1_off
24.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
24.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
24.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
23.68Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
23.68Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
23.68Consensusbombesin_onOrthosteric Ligandbb2_on
23.68Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
23.68Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
23.53Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
23.53Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
23.53Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
23.53Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.53Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
23.53Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
23.53Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
23.53Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
23.33Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
23.33Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
23.33Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
23.33Single7EZCUKA7EZC-A2A-UKA
23.33Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
23.33Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
23.33Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
23.33Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
23.33Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
23.33Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
23.33Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
23.33Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
23.33Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
23.08Single2YDOAdenosine2YDO-A2A-Adenosine
23.08Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
23.08Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
23.08Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
23.08Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
23.08Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
23.08Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
23.08Single8K5CAcipimox8K5C-HCA2-Acipimox
23.08Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
23.08Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
23.08Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
23.08Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
23.08Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
23.08Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.08Consensushca_onOrthosteric Ligandhca2_on
22.86Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
22.86Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
22.86Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
22.86Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
22.86Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
22.86Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
22.86Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.86Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
22.86Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
22.86Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
22.86Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.58Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
22.58Single5WF6UK-4320975WF6-A2A-UK-432097
22.58Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
22.58Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
22.58Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
22.58Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
22.58Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
22.58Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
22.58Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
22.50Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.50Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
22.22Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
22.22Single4XT3Fractalkine4XT3-US28-Fractalkine
22.22Single4YAYZD-71554YAY-AT1-ZD-7155
22.22Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
22.22Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
22.22Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
22.22Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
22.22Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
22.22Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
22.22Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
22.22Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
22.22Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
22.22Single8K5DGSK2560738K5D-HCA2-GSK256073
22.22Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
22.22Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
22.22Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
22.22Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
22.22Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
22.22Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
22.22Single9JEAAtropine9JEA-M1-Atropine
22.22Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
22.22Consensusa3_onOrthosteric Liganda3a_on
22.22Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
22.22Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Consensusblt_onOrthosteric Ligandblt1_on
22.22Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
22.22Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
22.22Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
22.22Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
22.22Consensusleukotriene_onOrthosteric Ligandblt_on
22.22Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
22.22Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
22.22Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
22.22Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
21.88Single4XT1Fractalkine4XT1-US28-Fractalkine
21.88Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
21.88Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
21.88Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
21.88Single8WDTphotoNECA8WDT-A2A-photoNECA
21.88Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.88Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
21.88Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
21.88Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
21.88Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
21.88Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
21.88Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.62Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
21.62Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
21.62Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
21.62Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
21.62Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.62Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
21.62Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
21.62Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.62Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.43Single5C1MBU725C1M-μ-BU72
21.43Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
21.43Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
21.43Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
21.43Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
21.43Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
21.43Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
21.43Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
21.43Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
21.43Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
21.43Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
21.43Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.43Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.43Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
21.43Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
21.43Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
21.43Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
21.43Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
21.43Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
21.43Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
21.43Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
21.43Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
21.43Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
21.43Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
21.43Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
21.43Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.43Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.43Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
21.43Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.43Consensustrace-amine_onOrthosteric Ligandta1_on
21.21Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
21.21Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
21.21Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
21.21Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
21.21Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
21.21Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
21.21Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
21.21Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
21.05Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
21.05Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
21.05Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
21.05Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
21.05Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
21.05Consensusbradykinin_onOrthosteric Ligandbk2_on
21.05Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
21.05Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
20.93Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.93Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
20.83Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
20.83Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
20.83Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
20.83Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
20.83Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
20.83Single9LRCHistamine9LRC-H4-Histamine
20.83Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
20.83Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
20.83Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
20.69Single4U15Tiotropium4U15-M3-Tiotropium
20.69Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
20.69Single5V54Methiothepin5V54-5-HT1B-Methiothepin
20.69Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
20.69Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
20.69Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
20.69Single6OL9Tiotropium6OL9-M5-Tiotropium
20.69Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
20.69Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
20.69Single7TUYGSK682753A7TUY-GPR183-GSK682753A
20.69Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
20.69Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
20.69Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
20.69Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
20.69Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
20.69Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
20.69Single8E0GBU728E0G-μ-BU72
20.69Single8EA0Iperoxo8EA0-M3-Iperoxo
20.69Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
20.69Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
20.69Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
20.69Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.69Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
20.69Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
20.69Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
20.69Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
20.69Consensus5ht1_offOrthosteric Ligand5ht1b_off
20.69Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
20.69Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
20.69Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
20.69Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
20.69Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
20.69Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
20.69Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.69Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
20.59Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
20.59Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
20.59Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
20.59Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
20.59Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
20.59Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
20.59Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
20.59Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
20.59Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
20.59Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
20.59Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
20.59Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
20.59Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
20.59Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
20.59Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
20.59Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
20.59Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
20.51Single5GLHEndothelin-15GLH-ETB-Endothelin-1
20.51Single6IGKEndothelin-36IGK-ETB-Endothelin-3
20.51Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.51Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
20.51Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
20.00Single3D4STimolol3D4S-β2-Timolol
20.00Single5CXVTiotropium5CXV-M1-Tiotropium
20.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
20.00Single6A93Risperidone6A93-5-HT2A-Risperidone
20.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
20.00Single6JODAngiotensin II6JOD-AT2-Angiotensin II
20.00Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
20.00Single6OS2TRV0266OS2-AT1-TRV026
20.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
20.00Single6ZG4HTL00099366ZG4-M1-HTL0009936
20.00Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
20.00Single7DFPSpiperone7DFP-D2-Spiperone
20.00Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
20.00Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.00Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
20.00Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
20.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
20.00Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
20.00Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
20.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
20.00Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
20.00Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
20.00Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
20.00Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
20.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
20.00Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
20.00Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
20.00Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
20.00Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
20.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
20.00Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
20.00Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
20.00Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.00Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8XYIVUF106618XYI-CXCR3-VUF10661
20.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
20.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
20.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
20.00Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
20.00Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
20.00Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
20.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
20.00Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
20.00Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
20.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.00Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.00Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.00Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
20.00Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
20.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
20.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
20.00Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
20.00Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
20.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
20.00Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
20.00Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
20.00Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
20.00Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
20.00Consensuslpl_offOrthosteric Ligands1p_off lpa_off
20.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
20.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
20.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
20.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
20.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
20.00Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
20.00Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
20.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.00Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
20.00Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
20.00Consensusvasop-oxy_onOrthosteric Ligandv2_on
20.00Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
19.51Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
19.44Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
19.44Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
19.44Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
19.44Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
19.44Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
19.44Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
19.44Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
19.44Single8ZRTET-18ZRT-ETB-ET-1
19.44Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
19.44Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
19.44Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
19.44Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
19.44Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
19.44Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
19.44Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
19.35Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
19.35Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
19.35Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
19.35Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
19.35Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
19.35Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.35Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
19.35Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
19.35Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
19.35Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
19.35Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
19.35Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
19.35Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
19.35Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
19.35Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.35Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
19.35Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
19.35Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
19.35Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
19.35Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
19.35Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
19.35Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
19.35Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
19.35Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Consensusprostanoid_offOrthosteric Ligandep_off dp_off
19.35Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
19.35Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
19.35Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
19.23Single5U09Taranabant5U09-CB1-Taranabant
19.23Single6AKXA4R6AKX-CCR5-A4R
19.23Single6AKYMaraviroc6AKY-CCR5-Maraviroc
19.23Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
19.23Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.23Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.23Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
19.23Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
19.23Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
19.23Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
19.23Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
19.23Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
19.23Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
19.23Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
19.23Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
19.23Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
19.23Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
19.23Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
19.23Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
19.23Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
19.23Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
19.23Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
19.23Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
19.23Single8Y0HVUF114188Y0H-CXCR3-VUF11418
19.23Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
19.23Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
19.23Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
19.23Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
19.23Consensusalpha2_offOrthosteric Ligandalpha2c_off
19.23Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
19.23Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
19.23Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
19.23Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
19.23Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.23Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
19.23Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
19.05Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
18.92Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
18.92Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
18.92Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
18.75Single3NY9ICI118-5513NY9-β2-ICI118-551
18.75Single5ZTYAM102575ZTY-CB2-AM10257
18.75Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
18.75Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
18.75Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
18.75Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
18.75Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
18.75Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
18.75Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8QJ2pN1628QJ2-MC4-pN162-Gs
18.75Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
18.75Single8X5YAstemizole8X5Y-H1-Astemizole
18.75Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
18.75Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
18.75Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
18.75Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
18.75Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
18.75Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
18.52Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
18.52Single4MBSMaraviroc4MBS-CCR5-Maraviroc
18.52Single6PS0S-Carazolol6PS0-β2-S-Carazolol
18.52Single6PS4ICI118-5516PS4-β2-ICI118-551
18.52Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
18.52Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
18.52Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
18.52Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
18.52Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
18.52Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
18.52Single7F61PF-036547467F61-H3-PF-03654746
18.52Single7T32ZM-2413857T32-A2A-ZM-241385
18.52Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
18.52Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
18.52Single7UL3Famotidine7UL3-H2-Famotidine
18.52Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
18.52Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
18.52Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
18.52Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
18.52Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
18.52Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
18.52Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
18.52Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
18.52Single8IHKAcifran8IHK-HCA3-Acifran
18.52Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
18.52Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
18.52Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
18.52Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
18.52Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
18.52Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
18.52Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
18.52Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
18.52Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
18.52Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
18.52Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
18.52Single9AS5Mescaline9AS5-5-HT2A-Mescaline
18.52Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
18.52Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
18.52Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
18.52Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
18.52Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
18.42Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
18.42Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
18.42Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
18.42Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
18.42Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
18.42Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
18.37Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
18.18Single4IARErgotamine4IAR-5-HT1B-Ergotamine
18.18Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
18.18Single7F8XNN90567F8X-CCKA-NN9056
18.18Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
18.18Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
18.18Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
18.18Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
18.18Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
18.18Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
18.18Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
18.18Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
18.18Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
18.18Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
18.18Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
18.18Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
18.18Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
18.18Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
18.18Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
17.95Single6IGLIRL16206IGL-ETB-IRL1620
17.95Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
17.95Consensusendothelin_onOrthosteric Ligandetb_on eta_on
17.86Single2Y04Salbutamol2Y04-β1-Salbutamol
17.86Single3NY8ICI118-5513NY8-β2-ICI118-551
17.86Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
17.86Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
17.86Single4GBRS-Carazolol4GBR-β2-S-Carazolol
17.86Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
17.86Single4MQSIperoxo4MQS-M2-Iperoxo
17.86Single4QKX35V4QKX-β2-35V
17.86Single4U14Tiotropium4U14-M3-Tiotropium
17.86Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
17.86Single5DHHSB-6121115DHH-NOP-SB-612111
17.86Single5DSGTiotropium5DSG-M4-Tiotropium
17.86Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
17.86Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
17.86Single5TGZAM65385TGZ-CB1-AM6538
17.86Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
17.86Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
17.86Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
17.86Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
17.86Single6H7MSalbutamol6H7M-β1-Salbutamol
17.86Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
17.86Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
17.86Single6PS1Timolol6PS1-β2-Timolol
17.86Single6TOTLemborexant6TOT-OX1-Lemborexant
17.86Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
17.86Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
17.86Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
17.86Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
17.86Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
17.86Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
17.86Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
17.86Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
17.86Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
17.86Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
17.86Single7UL4Alvimopan7UL4-μ-Alvimopan
17.86Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
17.86Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
17.86Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
17.86Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
17.86Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
17.86Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
17.86Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
17.86Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
17.86Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
17.86Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
17.86Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
17.86Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
17.86Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
17.86Single8JJOAlprenolol8JJO-β2-Alprenolol
17.86Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
17.86Single8T1WCVN4248T1W-GPR6-CVN424
17.86Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
17.86Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
17.86Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
17.86Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
17.86Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
17.86Single9AS1DMT9AS1-5-HT2A-DMT
17.86Single9CHXS-Carazolol9CHX-β2-S-Carazolol
17.86Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
17.86Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
17.86Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
17.86Consensus5ht5_onOrthosteric Ligand5ht5a_on
17.86Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
17.86Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
17.86Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
17.86Consensusalpha2_onOrthosteric Ligandalpha2b_on
17.86Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
17.86Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
17.86Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
17.86Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
17.86Consensusdopamine_offOrthosteric Ligandd2_off d3_off
17.86Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
17.86Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
17.86Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
17.86Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
17.86Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
17.86Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
17.86Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
17.86Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
17.86Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
17.65Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
17.65Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
17.65Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
17.65Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
17.65Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
17.65Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
17.65Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
17.65Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.65Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
17.65Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
17.65Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.50Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
17.24Single2RH1S-Carazolol2RH1-β2-S-Carazolol
17.24Single2Y03Isoprenaline2Y03-β1-Isoprenaline
17.24Single2YCWS-Carazolol2YCW-β1-S-Carazolol
17.24Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
17.24Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
17.24Single5D6LS-Carazolol5D6L-β2-S-Carazolol
17.24Single5JQHS-Carazolol5JQH-β2-S-Carazolol
17.24Single5N2RPSB-365N2R-A2A-PSB-36-Na
17.24Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
17.24Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
17.24Single5WIUNemonapride5WIU-D4-Nemonapride
17.24Single5WIVNemonapride5WIV-D4-Nemonapride-Na
17.24Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
17.24Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
17.24Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
17.24Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
17.24Single6D26Fevipiprant6D26-DP2-Fevipiprant
17.24Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
17.24Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
17.24Single6PS6Timolol6PS6-β2-Timolol
17.24Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
17.24Single6TP6Filorexant6TP6-OX1-Filorexant
17.24Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
17.24Single7C4SS1P7C4S-S1P3-S1P
17.24Single7C61Ergotamine7C61-5-HT1B-Ergotamine
17.24Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
17.24Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
17.24Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
17.24Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
17.24Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
17.24Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
17.24Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.24Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
17.24Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
17.24Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8S4DCMF-0198S4D-Apelin-CMF-019
17.24Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
17.24Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
17.24Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
17.24Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
17.24Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
17.24Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
17.24Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
17.24Single8ZMFA1L108ZMF-5-HT2C-A1L10
17.24Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
17.24Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
17.24Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
17.24Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
17.24Single9B9ZA1AKO9B9Z-CB1-A1AKO
17.24Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
17.24Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
17.24Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
17.24Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
17.24Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
17.24Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
17.24Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
17.24Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
17.24Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
17.24Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
17.24Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
17.24Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
17.24Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
17.24Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
17.24Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
17.24Consensusamine_offonOrthosteric Ligandamine_off amine_on
17.24Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
17.24Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
17.24Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
17.24Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
17.24Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
17.24Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
17.24Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
17.24Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
17.24Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.24Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
17.24Consensusdp_offOrthosteric Liganddp2_off
17.24Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
17.24Consensusep_offOrthosteric Ligandep4_off
17.24Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
17.24Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
17.24Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
17.24Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
17.24Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
17.14Single6PT2KGCHM076PT2-δ-KGCHM07
17.14Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.14Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
17.14Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
17.14Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.14Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
17.14Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.14Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
17.07Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
17.07Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
17.07Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
16.67Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
16.67Single4DJHJDTic4DJH-κ-JDTic
16.67Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
16.67Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
16.67Single5D5AS-Carazolol5D5A-β2-S-Carazolol
16.67Single5D5BS-Carazolol5D5B-β2-S-Carazolol
16.67Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
16.67Single6H7JIsoprenaline6H7J-β1-Isoprenaline
16.67Single6J21Aprepitant6J21-NK1-Aprepitant
16.67Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
16.67Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
16.67Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
16.67Single6OS1TRV0266OS1-AT1-TRV026
16.67Single6TQ7SB-3348676TQ7-OX1-SB-334867
16.67Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
16.67Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
16.67Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
16.67Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
16.67Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
16.67Single7P2L4YI7P2L-mGlu5-4YI
16.67Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
16.67Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
16.67Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
16.67Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
16.67Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
16.67Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
16.67Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
16.67Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
16.67Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
16.67Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
16.67Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
16.67Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
16.67Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
16.67Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
16.67Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
16.67Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
16.67Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
16.67Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
16.67Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
16.67Single9AS9RS130-1809AS9-5-HT2A-RS130-180
16.67Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
16.67Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
16.67Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
16.67Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
16.67Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
16.67Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
16.67Consensusa2_onOrthosteric Liganda2b_on
16.67Consensusa2_on_gpOrthosteric Liganda2b_on_gp
16.67Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
16.67Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
16.67Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
16.67Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
16.67Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
16.67Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
16.67Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
16.67Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
16.67Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
16.67Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
16.67Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
16.67Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
16.67Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
16.67Consensuslpa_onOrthosteric Ligandlpa1_on
16.67Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
16.67Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
16.67Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
16.67Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
16.67Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
16.67Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
16.67Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
16.22Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
16.22Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
16.22Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
16.22Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
16.22Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
16.22Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
16.13Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
16.13Single4AMIBucindolol4AMI-β1-Bucindolol
16.13Single4LDEBI1671074LDE-β2-BI167107
16.13Single4N4WSANT-14N4W-SMO-SANT-1
16.13Single4XEENeurotensin4XEE-NTS1-Neurotensin
16.13Single4XESNeurotensin4XES-NTS1-Neurotensin
16.13Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
16.13Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
16.13Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
16.13Single6IIURamatroban6IIU-TXA2-Ramatroban
16.13Single6YVRNTS8-136YVR-NTS1-NTS8-13
16.13Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
16.13Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
16.13Single7K15MKD0467K15-BLT1-MKD046-Na
16.13Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
16.13Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
16.13Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
16.13Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
16.13Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
16.13Single7YITNalfurafine7YIT-κ-Nalfurafine
16.13Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
16.13Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
16.13Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
16.13Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
16.13Single8JJ8Formoterol8JJ8-β2-Formoterol
16.13Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
16.13Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
16.13Single8JWY2-1188JWY-A2A-2-118
16.13Single8JWZAB9288JWZ-A2A-AB928-Na
16.13Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.13Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
16.13Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
16.13Single9DGIZ85267113509DGI-CB1-Z8526711350
16.13Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
16.13Consensusalpha1_offOrthosteric Ligandalpha1a_off
16.13Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
16.13Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
16.13Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
16.13Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
16.13Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
16.13Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
16.13Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
16.13Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
16.13Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
16.13Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
16.13Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
16.13Consensuslpa_offOrthosteric Ligandlpa1_off
16.13Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensusorexin_onOrthosteric Ligandox2_on
16.00Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
16.00Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
16.00Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
16.00Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
16.00Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
16.00Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
16.00Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
16.00Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
16.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
16.00Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
15.79Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
15.79Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
15.79Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
15.79Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
15.62Single4BUONeurotensin4BUO-NTS1-Neurotensin
15.62Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
15.62Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
15.62Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
15.62Single5X93K-87945X93-ETB-K-8794
15.62Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
15.62Single6H7LDobutamine6H7L-β1-Dobutamine
15.62Single6IBLArformoterol6IBL-β1-Arformoterol
15.62Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
15.62Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
15.62Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
15.62Single7UM4AS26747237UM4-5-HT5A-AS2674723
15.62Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
15.62Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
15.62Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
15.62Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
15.62Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
15.62Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
15.62Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
15.62Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
15.62Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
15.62Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
15.62Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
15.62Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
15.62Consensuscck_onOrthosteric Ligandccka_on cckb_on
15.62Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
15.62Consensuschemerin_onOrthosteric Ligandcml1_on
15.62Consensusendothelin_offOrthosteric Ligandetb_off
15.62Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
15.62Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
15.62Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
15.62Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
15.38Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
15.38Single3OE9IT1t3OE9-CXCR4-IT1t
15.38Single4O9RCyclopamine4O9R-SMO-Cyclopamine
15.38Single5L7IVismodegib5L7I-SMO-Vismodegib
15.38Single6LI0C176LI0-GPR52-C17
15.38Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
15.38Single7SRQLSD7SRQ-5-HT2B-LSD
15.38Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
15.38Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
15.38Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
15.38Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
15.38Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
15.38Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
15.38Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
15.38Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
15.38Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
15.38Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
15.15Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
15.15Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
15.15Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
15.15Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
15.15Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
15.15Single7XN9L-054,5227XN9-SST2-L-054,522
15.15Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
15.15Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
15.15Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
15.15Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
15.15Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
15.15Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
15.15Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
15.15Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
15.15Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
15.15Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
15.00Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
15.00Single8IY6Endothelin-18IY6-ETB-Endothelin-1
15.00Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
14.81Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
14.81Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
14.81Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
14.81Single4BWBNeurotensin4BWB-NTS1-Neurotensin
14.81Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
14.81Single4QINSAG1.54QIN-SMO-SAG1.5
14.81Single4S0VSuvorexant4S0V-OX2-Suvorexant
14.81Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
14.81Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
14.81Single5ZKQABT-4915ZKQ-PAF-ABT-491
14.81Single6B73MP11046B73-κ-MP1104
14.81Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
14.81Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
14.81Single6ME2Ramelteon6ME2-MT1-Ramelteon
14.81Single6ME9Ramelteon6ME9-MT2-Ramelteon
14.81Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
14.81Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
14.81Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
14.81Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
14.81Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
14.81Single6TPJSuvorexant6TPJ-OX2-Suvorexant
14.81Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
14.81Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
14.81Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
14.81Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
14.81Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
14.81Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
14.81Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
14.81Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
14.81Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
14.81Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
14.81Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
14.81Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
14.81Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
14.81Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
14.81Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
14.81Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
14.81Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
14.81Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
14.81Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
14.81Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
14.81Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
14.81Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
14.71Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
14.71Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
14.71Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
14.71Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
14.71Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
14.71Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
14.71Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
14.71Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
14.71Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
14.71Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.71Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
14.71Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
14.71Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
14.71Single9M4TSilodosin9M4T-Alpha1A-Silodosin
14.71Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
14.63Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
14.63Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
14.29Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
14.29Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
14.29Single4ZJCSB-6740424ZJC-OX1-SB-674042
14.29Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
14.29Single5IU7Q274563465IU7-A2A-Q27456346-Na
14.29Single5IUBQ274563445IUB-A2A-Q27456344-Na
14.29Single5JTBZM-2413855JTB-A2A-ZM-241385
14.29Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
14.29Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
14.29Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
14.29Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
14.29Single6FFIMMPEP6FFI-mGlu5-MMPEP
14.29Single6HLOAprepitant6HLO-NK1-Aprepitant
14.29Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
14.29Single6KUXRS-799486KUX-α2a-RS-79948
14.29Single6PS5S-Propranolol6PS5-β2-S-Propranolol
14.29Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
14.29Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
14.29Single6TP3Nemorexant6TP3-OX1-Nemorexant
14.29Single6TPGEMPA6TPG-OX2-EMPA
14.29Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
14.29Single6V9SGTPL114036V9S-OX1-GTPL11403
14.29Single6VI4JDTic6VI4-κ-JDTic
14.29Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
14.29Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
14.29Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
14.29Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
14.29Single6ZG9GSK10347026ZG9-M1-GSK1034702
14.29Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
14.29Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
14.29Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
14.29Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
14.29Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
14.29Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
14.29Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
14.29Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
14.29Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7SK5CXCL127SK5-ACKR3-CXCL12
14.29Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
14.29Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
14.29Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
14.29Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
14.29Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
14.29Single7XNACYN1548067XNA-SST2-CYN154806
14.29Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
14.29Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.29Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
14.29Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
14.29Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
14.29Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
14.29Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
14.29Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
14.29Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
14.29Single8K2WAMG4878K2W-CXCR3-AMG487
14.29Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
14.29Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
14.29Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
14.29Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
14.29Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
14.29Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
14.29Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
14.29Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
14.29Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
14.29Single8ZPMAMD0708ZPM-CXCR4-AMD070
14.29Single9AS3LSD9AS3-5-HT2A-LSD
14.29Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
14.29Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
14.29Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
14.29Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
14.29Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
14.29Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
14.29Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
14.29Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
14.29Consensusa2_offOrthosteric Liganda2a_off
14.29Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
14.29Consensusalpha1_onOrthosteric Ligandalpha1a_on
14.29Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
14.29Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
14.29Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
14.29Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
14.29Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
14.29Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
14.29Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
14.29Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
14.29Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
14.29Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
14.29Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
14.29Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
14.29Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
14.29Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
14.29Consensusopsins_offOrthosteric Ligandrhodopsin_off
14.29Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.29Consensussensory_offOrthosteric Ligandopsins_off
14.29Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
13.89Single3OE0CVX153OE0-CXCR4-CVX15
13.89Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
13.89Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
13.89Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.89Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
13.89Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
13.89Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
13.89Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
13.79Single2Y01Dobutamine2Y01-β1-Dobutamine
13.79Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
13.79Single3EMLZM-2413853EML-A2A-ZM-241385
13.79Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
13.79Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
13.79Single4DAJTiotropium4DAJ-M3-Tiotropium
13.79Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
13.79Single4EJ4Naltrindole4EJ4-δ-Naltrindole
13.79Single5DHGC-355DHG-NOP-C-35
13.79Single5IU8Q274563475IU8-A2A-Q27456347-Na
13.79Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
13.79Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
13.79Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
13.79Single5T04Neurotensin5T04-NTS1-Neurotensin
13.79Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
13.79Single6DRXLisuride6DRX-5-HT2B-Lisuride
13.79Single6FFHFenobam6FFH-mGlu5-Fenobam
13.79Single6GPSMK08126GPS-CCR2-MK0812
13.79Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
13.79Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
13.79Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
13.79Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
13.79Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
13.79Single6S0LZM-2413856S0L-A2A-ZM-241385
13.79Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
13.79Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
13.79Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
13.79Single7BU7BI1671077BU7-β1-BI167107
13.79Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
13.79Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
13.79Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
13.79Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
13.79Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
13.79Single7PYRPSB-21157PYR-A2A-PSB-2115
13.79Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
13.79Single7V3ZCP559407V3Z-CB1-CP55940
13.79Single7WC7Lisuride7WC7-5-HT2A-Lisuride
13.79Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
13.79Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
13.79Single7YXAONO-54306087YXA-S1P5-ONO-5430608
13.79Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
13.79Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
13.79Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
13.79Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
13.79Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
13.79Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
13.79Single8JXRLSD8JXR-D1-LSD
13.79Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
13.79Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
13.79Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
13.79Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
13.79Single8X63Mepyramine8X63-H1-Mepyramine
13.79Single8X64Desloratadine8X64-H1-Desloratadine
13.79Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
13.79Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
13.79Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
13.79Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
13.79Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
13.79Single9H37A1IR09H37-A2A-A1IR0-Na
13.79Single9IYAONO-97105319IYA-GPR55-ONO-9710531
13.79Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
13.79Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
13.79Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
13.79Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
13.79Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
13.79Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
13.79Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
13.79Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
13.79Consensushistamine_offOrthosteric Ligandh1_off
13.51Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
13.51Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
13.51Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
13.33Single2Y00Dobutamine2Y00-β1-Dobutamine
13.33Single4JKVTaladegib4JKV-SMO-Taladegib
13.33Single5IUAQ274563485IUA-A2A-Q27456348-Na
13.33Single5N2SPSB365N2S-A1-PSB36
13.33Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
13.33Single5TVNLSD5TVN-5-HT2B-LSD
13.33Single5WQCEMPA5WQC-OX2-EMPA
13.33Single6E67BI1671076E67-β2-BI167107-Gs(CT)
13.33Single6GPXMK08126GPX-CCR2-MK0812
13.33Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
13.33Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
13.33Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
13.33Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
13.33Single6S0QZM-2413856S0Q-A2A-ZM-241385
13.33Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
13.33Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
13.33Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
13.33Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
13.33Single7SINNPS-21437SIN-CaS-NPS-2143
13.33Single7SINNPS-21437SIN-CaS-NPS-2143
13.33Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
13.33Single7WC6LSD7WC6-5-HT2A-LSD
13.33Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
13.33Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
13.33Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
13.33Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
13.33Single8GNEKW-63568GNE-A2A-KW-6356-Na
13.33Single8JXSPF-61428JXS-D1-PF-6142
13.33Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
13.33Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
13.33Single8QOTNanobody-E8QOT-μ-Nanobody-E
13.33Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
13.33Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
13.33Single8TF5Oleic acid8TF5-GPR6-Oleic acid
13.33Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9EHSLUF76029EHS-A3A-LUF7602
13.33Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
13.33Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
13.33Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
13.33Single9HC04YI9HC0-mGlu5-4YI
13.33Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
13.33Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
13.33Consensusadenosine_offOrthosteric Liganda1_off a2_off
13.33Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
13.33Consensusblt_offOrthosteric Ligandblt1_off
13.33Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
13.33Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
13.33Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
13.33Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
13.33Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
13.33Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
13.16Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
13.04Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
12.90Single3P0GBI1671073P0G-β2-BI167107
12.90Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
12.90Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
12.90Single4BV0Neurotensin4BV0-NTS1-Neurotensin
12.90Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
12.90Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
12.90Single5V56TC1145V56-SMO-TC114
12.90Single5V57TC1145V57-SMO-TC114
12.90Single5XR8AM8415XR8-CB1-AM841
12.90Single5XRAAM115425XRA-CB1-AM11542
12.90Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
12.90Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
12.90Single6WGTLSD6WGT-5-HT2A-LSD
12.90Single7B6WCyclazosin7B6W-α1b-Cyclazosin
12.90Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
12.90Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
12.90Single7F1TMIP-1a7F1T-CCR5-MIP-1a
12.90Single7FEECP559407FEE-CB1-CP55940-ZCZ011
12.90Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
12.90Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
12.90Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
12.90Single7PX4PSB-21137PX4-A2A-PSB-2113
12.90Single7R0CAVP7R0C-V2-AVP-Arrestin2
12.90Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
12.90Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
12.90Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
12.90Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
12.90Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
12.90Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
12.90Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
12.90Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
12.90Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
12.90Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
12.90Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
12.90Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
12.90Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
12.90Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
12.90Single8ZWFJR14a8ZWF-C3aB-JR14a
12.90Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
12.90Single9BJKNaloxone9BJK-μ-Naloxone-NAM
12.90Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
12.90Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
12.90Consensusneurotensin_onOrthosteric Ligandnts1_on
12.90Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.82Single7SK3CXCL127SK3-ACKR3-CXCL12
12.82Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
12.82Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
12.50Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
12.50Single4RWADIPP-NH24RWA-δ-DIPP-NH2
12.50Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
12.50Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
12.50Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
12.50Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
12.50Single6CM4Risperidone6CM4-D2-Risperidone
12.50Single6KQICP559406KQI-CB1-CP55940-Org27569
12.50Single6MXTSalmeterol6MXT-β2-Salmeterol
12.50Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
12.50Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
12.50Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.50Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
12.50Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
12.50Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
12.50Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
12.50Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
12.50Single8HS2Fab0468HS2-GPR20-Fab046
12.50Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
12.50Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
12.50Single8JJLOlodaterol8JJL-β2-Olodaterol
12.50Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
12.50Single8PWNTheophylline8PWN-A2A-Theophylline
12.50Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
12.50Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
12.50Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
12.50Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.50Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.50Single9BJKNAM9BJK-μ-Naloxone-NAM
12.50Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.50Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
12.50Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
12.50Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
12.50Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
12.50Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
12.50Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.50Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
12.50Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
12.50Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.50Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
12.50Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.20Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
12.20Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
12.12Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
12.12Single5CGDHTL142425CGD-mGlu5-HTL14242
12.12Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
12.12Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
12.12Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
12.12Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
12.12Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
12.12Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
12.12Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
12.12Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
12.12Single8XVJMacitentan8XVJ-ETA-Macitentan
12.12Single8XVUCXCL28XVU-CXCR2-CXCL2
12.12Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
12.12Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
12.12Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
12.12Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
12.12Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
12.00Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
12.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
12.00Single8A2OTheophylline8A2O-A2A-Theophylline-Na
12.00Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
12.00Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
12.00Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
12.00Single9CHUNoradrenaline9CHU-β2-Noradrenaline
11.90Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
11.76Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
11.76Single6PT3DPI-2876PT3-δ-DPI-287
11.76Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
11.76Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
11.76Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
11.76Single8XQJJN2418XQJ-Apelin-JN241
11.76Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
11.76Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
11.76Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
11.76Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
11.76Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
11.76Single9IPYJR14a9IPY-C3aB-JR14a
11.76Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
11.76Consensuskisspeptin_onOrthosteric Ligandkiss1_on
11.76Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.63Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
11.54Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
11.54Single3OE6IT1t3OE6-CXCR4-IT1t
11.54Single3UZAGTPL92363UZA-A2A-GTPL9236
11.54Single4XNWMRS25004XNW-P2Y1-MRS2500
11.54Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
11.54Single6ME5Agomelatine6ME5-MT1-Agomelatine
11.54Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
11.54Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
11.54Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
11.54Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.54Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
11.54Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
11.54Consensus5ht2_onOrthosteric Ligand5ht2b_on
11.54Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
11.54Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
11.54Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
11.54Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
11.43Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
11.43Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Single8XWNCXCL88XWN-CXCR2-CXCL8
11.43Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
11.43Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
11.43Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
11.43Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
11.43Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
11.43Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Consensussomatostatin_offOrthosteric Ligandsst2_off
11.11Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
11.11Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
11.11Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
11.11Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
11.11Single3PBLEticlopride3PBL-D3-Eticlopride
11.11Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
11.11Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
11.11Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
11.11Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
11.11Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
11.11Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
11.11Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
11.11Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.11Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.11Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
11.11Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
11.11Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
11.11Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
11.11Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
11.11Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
11.11Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
11.11Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9B9Y7DY9B9Y-CB1-7DY
11.11Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
11.11Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
11.11Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
11.11Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
11.11Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
11.11Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
11.11Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.11Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.11Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
11.11Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
11.11Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
11.11Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
11.11Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
10.81Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
10.81Single6W25SHU91196W25-MC4-SHU9119-Ca
10.81Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.81Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.71Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
10.71Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
10.71Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
10.71Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
10.71Single3ODUIT1t3ODU-CXCR4-IT1t
10.71Single3PWHZM-2413853PWH-A2A-ZM-241385
10.71Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
10.71Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
10.71Single5WS3EMPA5WS3-OX2-EMPA
10.71Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
10.71Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
10.71Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
10.71Single6TODEMPA6TOD-OX1-EMPA-Na
10.71Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
10.71Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
10.71Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
10.71Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
10.71Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
10.71Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
10.71Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
10.71Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
10.71Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
10.71Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
10.71Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
10.71Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8GNGIstradefylline8GNG-A2A-Istradefylline
10.71Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
10.71Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
10.71Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
10.71Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
10.71Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
10.71Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
10.71Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
10.71Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
10.71Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
10.71Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
10.71Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
10.71Single9H2XA1IR19H2X-A2A-A1IR1-Na
10.71Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
10.71Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
10.71Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
10.71Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.71Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.71Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.71Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
10.71Consensusorexin_offOrthosteric Ligandox2_off ox1_off
10.71Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
10.71Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
10.71Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.71Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
10.53Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
10.53Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
10.53Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
10.53Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
10.34Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
10.34Single3RZECidoxepin3RZE-H1-Cidoxepin
10.34Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
10.34Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
10.34Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
10.34Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
10.34Single5UVIZM-2413855UVI-A2A-ZM-241385
10.34Single6A94Zotepine6A94-5-HT2A-Zotepine
10.34Single6AQFZM-2413856AQF-A2A-ZM-241385
10.34Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
10.34Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
10.34Single6IQLL7458706IQL-D4-L745870
10.34Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
10.34Single6MH8ZM-2413856MH8-A2A-ZM-241385
10.34Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
10.34Single7AROLUF58337ARO-A2A-LUF5833-Na
10.34Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
10.34Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
10.34Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
10.34Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
10.34Single7VV6C48/807VV6-MRGPRX2-C48/80
10.34Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
10.34Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
10.34Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
10.34Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
10.34Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
10.34Single8RLNLUF58348RLN-A2A-LUF5834
10.34Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
10.34Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
10.34Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
10.34Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
10.34Single8ZPNAMD31008ZPN-CXCR4-AMD3100
10.34Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9BA0A1AKN9BA0-CB1-A1AKN
10.34Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
10.34Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
10.34Consensusgrh_offOrthosteric Ligandgnrh1_off
10.26Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
10.26Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
10.00Single2Y02Carmoterol2Y02-β1-Carmoterol
10.00Single4QIMANTA XV4QIM-SMO-ANTA XV
10.00Single5UENDU1725UEN-A1-DU172
10.00Single5UIGCmpd-15UIG-A2A-Cmpd-1
10.00Single6D27CAY104716D27-DP2-CAY10471
10.00Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
10.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
10.00Single6IIVDaltroban6IIV-TXA2-Daltroban
10.00Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
10.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
10.00Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
10.00Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
10.00Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
10.00Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
10.00Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
10.00Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
10.00Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
10.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
10.00Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
10.00Single8CU6LJ-45178CU6-A2A-LJ-4517
10.00Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
10.00Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.00Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.00Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
10.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
10.00Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
10.00Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
10.00Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
10.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
10.00Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
10.00Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
10.00Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
10.00Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
10.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
10.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
10.00Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.00Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
10.00Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
10.00Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
10.00Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
9.76Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
9.76Single9KDFRES-701-39KDF-ETB-RES-701-3
9.68Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
9.68Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
9.68Single5CGCHTL142425CGC-mGlu5-HTL14242
9.68Single6LUQHaloperidol6LUQ-D2-Haloperidol
9.68Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
9.68Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
9.68Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
9.68Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
9.68Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
9.68Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
9.68Single7W41PD1762527W41-BB2-PD176252
9.68Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
9.68Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.68Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
9.68Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
9.68Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
9.68Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
9.68Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
9.68Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
9.68Single9HAPTolvaptan9HAP-V2-Tolvaptan
9.68Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
9.68Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
9.68Consensusbombesin_offOrthosteric Ligandbb2_off
9.68Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
9.38Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
9.38Single5TZRMK86665TZR-FFA1-MK8666
9.38Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
9.38Single6J20Aprepitant6J20-NK1-Aprepitant
9.38Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
9.38Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
9.38Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
9.38Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
9.38Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
9.38Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
9.38Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
9.38Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
9.38Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
9.38Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single8XVLZibotentan8XVL-ETA-Zibotentan
9.38Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
9.38Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
9.38Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
9.38Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
9.38Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
9.38Consensustachykinin_offOrthosteric Ligandnk1_off
9.09Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
9.09Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
9.09Single5X33BIIL2605X33-BLT1-BIIL260
9.09Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
9.09Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
9.09Single8XQJJN2418XQJ-Apelin-JN241
9.09Single8XWACXCL18XWA-CXCR2-CXCL1
9.09Single8XWMCXCL68XWM-CXCR2-CXCL6
9.09Single8XWSCXCL58XWS-CXCR2-CXCL5
9.09Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
9.09Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
9.09Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
8.82Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
8.82Single6K1QIRL25006K1Q-ETB-IRL2500
8.82Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
8.82Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
8.82Single8XWFCXCL38XWF-CXCR2-CXCL3
8.82Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
8.82Single8ZPLHF511168ZPL-CXCR4-HF51116
8.82Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
8.57Single6KNMJN241-96KNM-Apelin-JN241-9
8.57Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
8.57Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
8.57Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
8.57Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
8.57Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
8.57Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
8.57Single9JF4PD1683689JF4-BB1-PD168368
8.57Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single5MZPCaffeine5MZP-A2A-Caffeine-Na
8.33Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
8.33Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
8.33Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.33Single8IEBA1LYA8IEB-GPR156-A1LYA
8.33Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
8.33Single8KIGSHU91198KIG-MC3-SHU9119-Ca
8.33Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
8.33Single8WKYPG-9348WKY-MC4-PG-934
8.33Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
8.33Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
8.33Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.33Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
8.11Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
8.11Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
8.11Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
8.11Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
8.00Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
8.00Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
8.00Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.00Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
7.89Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
7.89Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
7.89Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
7.89Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
7.69Single3OE8IT1t3OE8-CXCR4-IT1t
7.69Single3RFMCaffeine3RFM-A2A-Caffeine
7.69Single6TQ9SB-4081246TQ9-OX1-SB-408124
7.69Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
7.69Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
7.69Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
7.69Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
7.69Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
7.69Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
7.69Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
7.69Consensusp2y_offOrthosteric Ligandp2y1_off
7.69Consensussensory_onOrthosteric Ligandopsins_on
7.50Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
7.41Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
7.41Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
7.41Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
7.41Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
7.41Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
7.41Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
7.41Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
7.41Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
7.41Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
7.41Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.41Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.41Single8JPSCCL78JPS-ACKR1-CCL7
7.41Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
7.41Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
7.41Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.41Consensusgi_sensoryOrthosteric Ligandgi_opsins
7.41Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
7.41Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.41Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
7.14Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
7.14Single6HLLCP999946HLL-NK1-CP99994
7.14Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
7.14Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
7.14Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
7.14Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
7.14Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.14Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
7.14Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
7.14Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
7.14Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
7.14Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
7.14Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
7.14Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
7.14Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
7.14Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
7.14Single9AS7Psilocin9AS7-5-HT2A-Psilocin
7.14Consensusgq_nucleotideOrthosteric Ligandgq_p2y
7.14Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
6.90Single4XNVBPTU4XNV-P2Y1-BPTU
6.90Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
6.90Single6DS0Ly2660976DS0-5-HT2B-Ly266097
6.90Single7BR3Elagolix7BR3-GnRH1-Elagolix
6.90Single7F8ULintitript7F8U-CCKA-Lintitript
6.90Single7F8YDevazepide7F8Y-CCKA-Devazepide
6.90Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
6.90Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
6.90Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
6.90Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
6.90Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
6.90Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
6.90Single7XRRLemborexant7XRR-OX2-Lemborexant
6.90Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
6.90Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
6.90Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
6.90Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
6.90Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
6.67Single3REYXAC3REY-A2A-XAC
6.67Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
6.67Single6TPNHTL66416TPN-OX2-HTL6641
6.67Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
6.67Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8IYXYL-3658IYX-GPR34-YL-365
6.67Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
6.67Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
6.67Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
6.67Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
6.67Single9ARXSerotonin9ARX-5-HT2A-Serotonin
6.67Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
6.67Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.45Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
6.45Single7F83PF-051904577F83-Ghrelin-PF-05190457
6.45Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
6.45Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
6.45Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
6.45Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
6.45Consensuscck_offOrthosteric Ligandccka_off
6.45Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
6.25Single4NTJAZD12834NTJ-P2Y12-AZD1283
6.25Single5XPRBosentan5XPR-ETB-Bosentan
6.25Single6HLPNetupitant6HLP-NK1-Netupitant
6.25Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
6.25Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
6.25Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
6.25Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Single6E59L-7607356E59-NK1-L-760735
6.06Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
6.06Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
6.06Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
6.06Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
6.06Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
6.06Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
6.06Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.88Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
5.88Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
5.88Single4PY02MeSATP4PY0-P2Y12-2MeSATP
5.88Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
5.88Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.88Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.88Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
5.88Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
5.88Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
5.88Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.88Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.71Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
5.71Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.71Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
5.71Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.41Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.41Single8IEIA1LYA8IEI-GPR156-A1LYA
5.41Single8IEIA1LYA8IEI-GPR156-A1LYA
5.41Single8IEPA1LYA8IEP-GPR156-A1LYA
5.41Single8IEPA1LYA8IEP-GPR156-A1LYA
5.41Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
5.26Single8IEBA1LYA8IEB-GPR156-A1LYA
5.26Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
5.00Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
4.55Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.55Single6D35Cholesterol6D35-SMO-Cholesterol
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.55Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.55Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.55Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
4.55Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.55Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.55Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.55Single7XW7K1-707XW7-TSH-K1-70
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.55Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.55Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.55Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WVXNorrin8WVX-LGR4-Norrin
4.55Single8WVYNorrin8WVY-LGR4-Norrin
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.55Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9KHHNorrin9KHH-LGR4-Norrin
4.55Single9S37NB219S37-LGR4-NB21
4.55Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.17Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.17Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.17Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.17Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.00Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
4.00Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
4.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.00Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.00Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.00Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.00Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.00Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
3.85Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
3.85Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
3.85Single5L7DCholesterol5L7D-SMO-Cholesterol
3.85Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.85Single7WC4Serotonin7WC4-5-HT2A-Serotonin
3.85Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.70Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
3.70Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.70Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
3.70Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.57Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
3.57Single7WC5Psilocin7WC5-5-HT2A-Psilocin
3.57Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
3.57Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
3.57Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
3.57Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
3.57Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
3.45Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
3.45Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.45Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
3.45Single7UL2SR486927UL2-NTS1-SR48692-Na
3.45Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.45Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
3.45Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.45Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.45Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.45Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
3.45Consensusneurotensin_offOrthosteric Ligandnts1_off
3.45Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
3.33Single4K5YCP-3763954K5Y-CRF1-CP-376395
3.33Single6C1QNDT95137276C1Q-C5a1-PMX53-NDT9513727
3.33Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
3.33Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.33Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.33Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.33Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.33Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.33Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.33Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.33Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.33Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.33Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.33Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.23Single6TPKRetosiban6TPK-OT-Retosiban
3.23Single7VODCariprazine7VOD-5-HT2A-Cariprazine
3.23Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.23Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.23Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.23Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
3.23Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
3.23Consensusvasop-oxy_offOrthosteric Ligandot_off
3.12Single4Z9GCP-3763954Z9G-CRF1-CP-376395
3.12Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
3.12Single8GTIBMK-C2058GTI-CRF1-BMK-C205
3.12Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
3.03Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
3.03Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
3.03Single8GTGBMK-I1528GTG-CRF1-BMK-I152
3.03Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
3.03Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
2.94Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
2.94Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
2.94Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
2.86Single8GTMBMK-C2038GTM-CRF1-BMK-C203
2.86Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
2.78Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
2.70Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
2.70Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
2.63Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.63Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.50Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.50Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.44Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.27Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
8E3Z 8E3Z-VPAC1-VIP-Gs/β1/γ2
Net Summary
Imin 2.92
Number of Linked Nodes 936
Number of Links 1138
Number of Hubs 176
Number of Links mediated by Hubs 653
Number of Communities 25
Number of Nodes involved in Communities 275
Number of Links involved in Communities 402
Path Summary
Number Of Nodes in MetaPath 88
Number Of Links MetaPath 87
Number of Shortest Paths 1252118
Length Of Smallest Path 3
Average Path Length 30.8881
Length of Longest Path 58
Minimum Path Strength 1.335
Average Path Strength 6.78775
Maximum Path Strength 21.31
Minimum Path Correlation 0.7
Average Path Correlation 0.989228
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.7027
Average % Of Corr. Nodes 53.4636
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 49.0849
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
vpac_on_gpvpac1_on_gp
vpac2_on_gp



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