Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 1.58538503
2G.HN.37 2.20673402
3G.HN.52 1.74038404
4G.S1.02 5.04185544
5G.S1.05 5.37038409
6G.S1.06 3.74385548
7G.S2.03 5.54635418
8G.S2.05 6.06942413
9G.S2.08 7.25442445
10G.S3.01 4.65712444
11G.S3.03 7.51723547
12G.S3.04 6.96154516
13G.S3.06 8.254516
14G.S3.07 4.76981449
15G.s3h2.03 4.56831519
16G.H2.02 3.85192418
17G.H2.03 4.47173419
18G.H2.06 5.21407719
19G.H2.07 4.55856819
20G.H2.09 6.39288418
21G.h2s4.01 6.44138519
22G.S4.03 3.61558447
23G.S4.04 5.39969589
24G.s4h3.04 4.49103678
25G.H3.01 5.00731409
26G.H3.09 5.83923689
27G.H3.13 4.22635485
28G.H3.17 6.52295614
29G.H3.18 5.730774189
30G.S5.03 3.14385448
31G.S5.04 3.84508589
32G.S5.05 3.72165749
33G.S5.07 4.0375449
34G.HG.03 2.96365476
35G.HG.04 5.11846578
36G.HG.07 4.07481479
37G.HG.14 2.66231405
38G.hgh4.01 4.27577474
39G.hgh4.02 5.51407778
40G.hgh4.05 7.19885406
41G.H4.03 7.18865403
42G.H4.10 8.79519476
43G.H4.12 6.29077485
44G.H4.15 4.99596488
45G.h4s6.02 5.20808487
46G.h4s6.11 4.06212488
47G.h4s6.12 6.049044134
48G.S6.02 6.471085138
49G.s6h5.01 5.51135449
50G.s6h5.05 2.05831509
51G.H5.03 5.08192448
52G.H5.08 5.77423448
53G.H5.15 2.2775408
54G.H5.20 3.75673408
55G.H5.26 5.53615505
56b.1x4 1.58615708
57b.1x11 2.23865408
58b.h2x1 2.95808405
59b.lhb1x3 2.34431502
60b.b1x4 3.05138557
61b.b1x6 7.69788459
62b.l1x3 7.40253759
63b.b2x1 8.61431518
64b.b2x5 6.43641607
65b.b3x3 3.35288408
66b.l3x2 4.92415559
67b.b4x2 4.77135408
68b.b4x3 4.158654157
69b.b4x5 4.192884107
70b.b4x6 8.73571759
71b.l4x2 11.2527454
72b.b5x2 5.28962407
73b.b5x3 6.48718659
74b.b5x5 5.26754105
75b.b5x7 5.33827407
76b.l5x1 3.888315158
77b.l5x5 6.97571719
78b.b6x5 3.814187106
79b.l6x5 5.568084174
80b.b7x1 5.677085174
81b.b7x4 3.484424158
82b.l7x2 3.44218619
83b.l7x4 3.57442409
84b.b8x4 5.326465156
85b.l8x1 3.888654105
86b.l9x3 6.0056719
87b.l9x6 4.551461018
88b.b10x5 4.41218609
89b.l10x1 4.36827403
90b.b11x4 4.82138519
91b.l11x2 8.51385419
92b.b12x3 3.43212468
93b.b12x6 7.56824718
94b.b13x7 7.83723567
95b.l13x3 7.30487669
96b.l13x6 5.09862519
97b.l13x7 4.24808469
98b.b14x3 4.18038465
99b.b15x1 5.69242769
100b.b15x2 7.24673416
101b.b15x3 4.69519469
102b.l15x1 4.81415517
103b.l15x2 5.28954569
104b.b16x4 10.4254466
105b.b16x5 4.31215505
106b.b16x6 8.34128668
107b.b17x5 6.83904417
108b.b17x7 8.21231418
109b.l17x3 7.49637719
110b.l17x6 6.12519
111b.b18x3 5.125418
112b.l18x1 5.569528126
113b.l18x2 5.814127
114b.l18x3 6.988084125
115b.b19x2 7.75123516
116b.b19x4 5.96519418
117b.l19x2 5.63692519
118b.b20x2 5.13288416
119b.b20x4 10.3122518
120b.b20x6 7.61215516
121b.b20x7 4.32019409
122b.l20x2 4.95908509
123b.b21x1 6.45369517
124b.b21x2 2.79038406
125b.b21x5 4.90173404
126b.b21x7 6.08139505
127b.l21x5 3.68212494
128b.b22x5 4.576676127
129b.l22x5 5.210557149
130b.b23x1 3.47519405
131b.b23x6 6.70451797
132b.l23x1 7.81288406
133b.b24x4 8.06154496
134b.b24x6 7.20904498
135b.l24x2 4.145584146
136b.l24x3 4.47865405
137b.b25x3 7.49577495
138b.l25x3 8.818775119
139b.b26x3 4.04365406
140b.b27x1 2.76346406
141b.l27x1 10.6929719
142b.l27x2 7.451154119
143b.b28x3 3.91492557
144b.b28x4 8.133274116
145b.b28x6 9.938464119
146g.l1x4 3.492508
147g.h2x11 9.356544126
148g.ctx3 5.578086209
149g.ctx5 3.233854209
150g.ctx6 3.31185506
151g.ctx14 4.42431559
152g.ctx15 6.1325459
153g.ctx16 4.4475858
154Lig 32.4342320
155NT 12.9021623
1561x30 1.93354505
1571x35 4.38673405
1581x39 4.61756628
1591x50 5.67846409
1601x57 3.15519407
1612x38 4.886734166
1622x42 5.28916167
1632x44 2.19212406
1642x46 3.80058439
1652x50 6.01192439
1662x53 5.80558426
1672x60 6.70423426
1682x63 4.74365425
169E1x50 6.85923628
170E1x52 5.83215527
1713x32 5.7391627
1723x33 4.7525405
1733x36 4.46923437
1743x37 4.08231637
1753x42 6.17096437
1763x49 6.574234168
1773x50 6.555409
1783x51 7.127314228
1794x50 5.30019439
180E2 14.44141424
181E2x52 4.49192425
1825x35 5.16635422
1835x47 5.565408
1845x50 3.16269409
1855x58 5.8622739
186I3 4.459044134
1876x44 4.21092539
1886x47 3.05954507
1896x48 7.31169539
1906x49 3.42038406
1916x51 5.1168627
192E3 3.83338524
1937x42 5.65339527
1947x45 6.11323539
1957x49 4.64115639
1967x52 2.69712438
1977x53 4.98487639
1988x50 5.78138508
1998x54 2.01115406
200I2x57 5.260964160
201g.ntx4 0.344615400
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b2x3 b.b2x5 20.76874.29462NoYes067
2b.b26x2 b.b2x3 20.99335.35846NoNo076
3b.b26x1 b.b26x2 21.22253.04308NoNo097
4b.b26x1 b.l27x1 21.45315.13077NoYes099
5b.b2x1 b.l27x1 14.40238.45923YesYes189
6b.b2x1 b.l3x1 14.792415.6938YesNo189
7b.l3x1 b.l5x5 15.16375.39308NoYes199
8G.h2s4.01 b.l5x5 11.653811.4108YesYes199
9G.S1.05 G.h2s4.01 13.8029.93077YesYes099
10G.S1.05 G.S1.07 44.245.53692YesNo099
11G.S1.07 G.S4.04 44.36613.00077NoYes099
12G.S4.04 G.S5.04 89.84853.18462YesYes899
13G.S5.04 G.S5.06 91.37373.51385YesNo098
14G.S5.06 G.s4h3.01 91.94167.34615NoNo087
15G.HG.04 G.s4h3.01 93.21939.83615YesNo087
16G.H4.03 G.HG.04 96.70873.41385YesYes038
17G.H4.03 G.HG.01 97.73567.71538YesNo035
18G.HG.01 G.s6h5.02 97.78344.84923NoNo057
19G.s6h5.02 G.s6h5.05 97.83112.51308NoYes079
20G.s6h5.01 G.s6h5.05 98.11522.00154YesYes099
21G.S5.05 G.s6h5.01 985.98538YesYes499
22G.S4.03 G.S5.05 98.10223.28385YesYes479
23G.S1.04 G.S4.03 1005.27NoYes477
24G.S1.02 G.S1.04 49.94842.86538YesNo447
25G.H5.11 G.S1.02 49.87745.30308NoYes484
26G.H5.11 G.H5.15 99.82632.36231NoYes088
27G.H5.15 G.H5.19 99.58822.50615YesNo088
283x53 G.H5.19 99.52854.23692NoNo088
293x53 I2x57 99.46863.80769NoYes080
302x38 I2x57 49.85185.22923YesYes1660
312x38 2x42 49.24655.44077YesYes1667
32G.H3.17 b.l27x1 10.08932.95615YesYes149
33G.H3.15 G.H3.17 32.71784.79308NoYes084
34G.H3.15 G.H3.18 32.83123.90231NoYes089
35G.H3.18 G.S4.02 30.16658.11385YesNo1897
36G.S1.05 G.S4.02 30.36833.95077YesNo097
37G.S1.04 G.S3.03 50.09443.18615NoYes477
38G.H5.11 G.S3.03 50.0084.63538NoYes487
393x49 I2x57 49.43669.58385YesYes1680
402x42 3x49 49.276.38846YesYes1678
41b.b2x4 b.b6x5 11.57793.01846NoYes066
42b.b10x4 b.b2x4 11.676314.6677NoNo066
43b.b10x2 b.b10x4 11.19244.39308NoNo066
44b.b10x2 b.b14x3 11.31494.63923NoYes065
45b.b11x5 b.b14x3 14.6455.42769NoYes065
46b.b10x1 b.b11x5 19.47043.76154NoNo096
47b.b10x1 b.l9x6 19.59533.03154NoYes098
482x42 3x46 92.69944.26231YesNo079
493x46 7x53 92.50664.59846NoYes099
503x50 7x53 20.39615.46YesYes099
51G.H2.07 b.l9x6 50.14943.48692YesYes198
52G.H2.06 b.l9x6 31.1953.21308YesYes198
53G.H2.04 G.H2.07 49.28215NoYes099
54G.H2.04 G.H3.08 49.395.03231NoNo099
55G.H2.06 b.l17x6 30.40097.65923YesYes199
56G.H5.20 G.H5.25 13.14623.51231YesNo086
573x50 G.H5.25 14.05578.68923YesNo096
58G.H5.20 G.H5.26 12.15784.96462YesYes085
59b.l17x5 b.l17x6 30.88774.19NoYes169
60b.l17x5 b.l19x2 30.77513.05692NoYes169
61b.l17x3 b.l19x2 21.25493.97462YesYes199
62b.b19x4 b.l17x3 11.87297.79154YesYes189
63b.b17x7 b.b20x6 23.89349.47923YesYes186
64b.b17x7 b.b21x1 22.66463.94923YesYes187
65b.1x19 b.b21x1 19.28467.14692NoYes067
66b.1x15 b.1x19 17.15133.37154NoNo076
67b.1x15 g.h1x15 16.71571.87308NoNo078
68b.1x14 g.h1x15 15.84412NoNo048
69b.1x11 b.1x14 15.40821.43231YesNo084
70b.1x11 b.1x7 11.91721.83615YesNo088
71b.b20x4 b.b20x6 16.79265.09769YesYes186
72b.l23x1 b.l25x6 25.101619.3331YesNo068
73b.l21x7 b.l23x1 15.6255.02538NoYes056
74b.b23x6 b.l21x7 14.70432.89462YesNo975
75b.b23x6 b.b24x6 12.59847.34615YesYes978
76b.b21x7 b.b24x6 12.35688.53308YesYes058
777x49 7x53 66.30825.27769YesYes399
787x45 7x49 32.60525.29923YesYes399
796x48 7x45 26.333112.71YesYes399
806x48 7x41 24.13475.02154YesNo098
816x51 7x41 23.91282.84923YesNo078
826x51 Lig 19.96173.74154YesYes270
832x50 7x49 31.0025.80077YesYes399
842x50 7x46 29.17744.96385YesNo098
852x53 7x46 28.96233.65769YesNo068
862x53 3x32 24.35099.36231YesYes267
873x32 Lig 19.199.11692YesYes270
88E2 Lig 13.40641.0631YesYes240
89G.H3.08 G.S4.04 49.45155.70923NoYes099
90G.H3.17 b.l25x6 22.09983.69231YesNo148
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
7x34Lig4.569232NoYes5010
LigNT40.96082YesYes0301
1x28Lig3.617690NoYes4010
7x31Lig3.619232NoYes5010
E2Lig41.06312YesYes4010
E2x51Lig7.905382NoYes3010
E3Lig3.211542YesYes4010
5x32Lig5.419232NoYes2010
NTNT13.66622YesYes3311
7x24NT5.320NoYes7321
1x351x397.726920YesYes5821
1x357x353.993850YesNo5521
1x392x574.997692YesNo8812
1x392x613.398462YesNo8612
1x397x426.117692YesYes8712
2x533x329.362312YesYes6721
2x537x425.581542YesYes6722
2x603x324.774622YesYes6711
2x63E1x507.541542YesYes5812
E1x49E25.552312NoYes4421
E1x50E24.686922YesYes8421
3x22E25.695382NoYes4421
3x294x659.165382NoNo5512
3x327x423.22YesYes7712
3x334x618.613080YesNo5422
4x64E210.57152NoYes4421
4x645x356.244622NoYes4222
4x65E2x525.590NoYes5521
E2E247.40312YesYes4411
E2E2x519.654612YesNo4311
E2E2x525.167692YesYes4511
5x35E28.062YesYes2421
5x36E23.754622NoYes4411
5x39E24.025382NoYes5421
5x32E24.446922NoYes2411
6x516x522.886152YesNo7812
6x517x375.709232YesNo7612
6x517x386.913082YesNo7611
6x547x343.564620NoNo5521
6x547x374.750770NoNo5622
6x61E34.480NoYes4421
6x64E33.189230NoYes1421
7x387x426.263852NoYes6712
2x562x602.985382NoYes6621
2x577x427.103852NoYes8722
2x60Lig16.20082YesYes6010
2x63E24.694622YesYes5411
3x29Lig3.583852NoYes5010
3x323x335.072312YesYes7512
3x32Lig9.116922YesYes7010
4x61E2x524.271540NoYes4521
E2x52Lig2.938462YesYes5010
5x36Lig4.282NoYes4010
6x516x558.601542YesNo7612
6x51Lig3.741542YesYes7010
6x587x342.723080NoNo4521
6x617x272.880770NoNo4421
7x26E35.068460NoYes1421
7x27Lig6.583082NoYes4010
2x63Lig3.882312YesYes5010
1x39Lig2.732YesYes8010
7x38Lig7.595392NoYes6010
7x35Lig3.613852NoYes5010
2x563x322.908462NoYes6721
2x602x632.856152YesYes6511
6x517x412.849232YesNo7812
6x60E33.217690NoYes5421
1x397x392.734622YesNo8412
6x62Lig2.556150NoYes5010
7x28NT2.513082NoYes3321
5x335x362.389230NoNo1421
1x277x312.110NoNo3521
1x247x311.853850NoNo0521
1x32NT1.286152NoYes4321
2x67Lig0.5515380NoYes4010

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
90.91Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
80.95Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
75.00Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
73.91Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
66.67Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
66.67Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
66.67Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
62.50Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
61.54Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
60.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
59.26Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
59.26Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
59.26Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
58.62Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
57.69Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
57.69Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
56.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
55.56Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
53.57Single7SK3CXCL127SK3-ACKR3-CXCL12
53.57Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
53.33Single6IGKEndothelin-36IGK-ETB-Endothelin-3
52.17Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
52.17Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
51.61Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
50.00Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
50.00Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
50.00Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
50.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
50.00Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
50.00Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
50.00Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
50.00Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
48.39Single5GLHEndothelin-15GLH-ETB-Endothelin-1
48.28Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
48.28Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
48.28Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
48.28Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
48.15Single3OE0CVX153OE0-CXCR4-CVX15
48.15Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
48.15Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
48.15Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
48.00Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
48.00Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
48.00Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
48.00Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
48.00Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
47.83Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
46.88Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
46.67Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
46.67Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
46.43Single6JODAngiotensin II6JOD-AT2-Angiotensin II
46.43Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
46.43Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
46.43Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
46.43Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
46.43Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
46.43Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
46.43Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
46.43Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
46.15Single4XT1Fractalkine4XT1-US28-Fractalkine
46.15Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
46.15Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
46.15Single8XWNCXCL88XWN-CXCR2-CXCL8
46.15Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
46.15Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
45.83Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
45.83Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
45.83Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
45.45Single6D27CAY104716D27-DP2-CAY10471
45.45Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
45.16Single6IGLIRL16206IGL-ETB-IRL1620
45.16Single8IY6Endothelin-18IY6-ETB-Endothelin-1
45.16Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
45.16Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
45.16Consensusbradykinin_onOrthosteric Ligandbk2_on
45.16Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
45.16Consensusendothelin_onOrthosteric Ligandetb_on eta_on
45.16Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
44.83Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
44.83Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
44.83Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
44.83Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
44.44Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
44.44Single7SK5CXCL127SK5-ACKR3-CXCL12
44.44Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
44.00Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
44.00Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
44.00Single8XVUCXCL28XVU-CXCR2-CXCL2
44.00Single8XWFCXCL38XWF-CXCR2-CXCL3
44.00Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
43.75Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
43.75Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
43.75Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
43.75Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
43.48Single6D26Fevipiprant6D26-DP2-Fevipiprant
43.48Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
43.48Consensusdp_offOrthosteric Liganddp2_off
43.33Single4XT3Fractalkine4XT3-US28-Fractalkine
43.33Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
42.86Consensusangiotensin_onOrthosteric Ligandat1_on
42.86Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
42.86Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
42.86Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
42.86Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
42.86Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
42.86Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
42.31Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
42.31Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
42.31Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
41.94Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
41.94Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
41.67Single7F1TMIP-1a7F1T-CCR5-MIP-1a
41.67Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
41.67Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.67Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
41.38Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.38Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
41.38Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
41.38Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
41.18Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
40.91Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
40.91Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
40.91Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
40.91Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
40.91Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
40.91Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
40.74Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
40.74Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
40.74Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
40.62Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
40.62Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
40.00Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
40.00Single6OS2TRV0266OS2-AT1-TRV026
40.00Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
40.00Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
40.00Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
40.00Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
40.00Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
40.00Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
40.00Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
40.00Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
40.00Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
39.39Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
39.29Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
39.29Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
39.29Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
39.29Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
39.29Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
39.29Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
39.13Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
39.13Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
39.13Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
39.13Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
39.13Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
38.71Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
38.71Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
38.71Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
38.46Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
38.46Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
38.46Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
38.46Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
38.46Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
38.46Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.46Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.46Consensusprostanoid_offOrthosteric Ligandep_off dp_off
38.24Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
38.24Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
38.10Single3OE9IT1t3OE9-CXCR4-IT1t
37.93Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
37.93Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
37.93Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
37.93Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
37.84Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
37.84Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
37.50Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
37.50Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
37.50Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
37.04Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
37.04Single6KNMJN241-96KNM-Apelin-JN241-9
37.04Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.04Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
37.04Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
37.04Single8QJ2pN1628QJ2-MC4-pN162-Gs
37.04Single8XQJJN2418XQJ-Apelin-JN241
37.04Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.04Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.04Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
37.04Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
36.67Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
36.67Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
36.67Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
36.67Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
36.67Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
36.67Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
36.67Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
36.67Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
36.67Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
36.67Consensusvasop-oxy_onOrthosteric Ligandv2_on
36.67Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
36.36Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
36.36Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
36.36Single8GNGIstradefylline8GNG-A2A-Istradefylline
36.36Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
36.36Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
36.36Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
36.36Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
36.36Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
36.36Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
36.36Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
36.00Single6OS1TRV0266OS1-AT1-TRV026
36.00Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
36.00Single7PX4PSB-21137PX4-A2A-PSB-2113
36.00Single7TUYGSK682753A7TUY-GPR183-GSK682753A
36.00Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
36.00Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
36.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
36.00Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
36.00Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
36.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
36.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
36.00Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single7F8XNN90567F8X-CCKA-NN9056
35.71Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
35.71Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
35.71Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
35.71Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
35.71Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
35.71Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
35.71Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
35.48Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
35.48Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
35.48Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
35.48Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
35.48Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
35.48Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
35.48Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
35.48Single8ZRTET-18ZRT-ETB-ET-1
35.48Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
35.48Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
35.48Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
35.48Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
35.48Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.78Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
34.78Single7AROLUF58337ARO-A2A-LUF5833-Na
34.78Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
34.78Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
34.78Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
34.78Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
34.78Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
34.78Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
34.62Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
34.62Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
34.62Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
34.62Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
34.62Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.62Single8XWACXCL18XWA-CXCR2-CXCL1
34.62Single8XWMCXCL68XWM-CXCR2-CXCL6
34.62Single8XWSCXCL58XWS-CXCR2-CXCL5
34.62Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
34.62Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
34.62Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
34.62Consensuslpl_offOrthosteric Ligands1p_off lpa_off
34.62Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Consensusorexin_onOrthosteric Ligandox2_on
34.48Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
34.48Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
34.48Single7XNACYN1548067XNA-SST2-CYN154806
34.48Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
34.48Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
34.48Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
34.48Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
34.48Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
34.48Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
34.38Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
34.38Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
34.38Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
34.29Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
34.29Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
33.33Single3OE6IT1t3OE6-CXCR4-IT1t
33.33Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
33.33Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
33.33Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
33.33Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
33.33Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
33.33Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
33.33Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
33.33Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
33.33Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
33.33Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
33.33Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
33.33Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
33.33Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
33.33Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
33.33Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
33.33Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
33.33Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
33.33Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
33.33Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
33.33Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
33.33Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
33.33Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
33.33Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
33.33Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
33.33Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
33.33Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
33.33Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
32.56Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
32.35Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
32.26Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
32.26Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
32.26Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
32.26Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
32.26Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
32.26Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
32.26Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
32.14Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
32.14Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
32.14Single7XN9L-054,5227XN9-SST2-L-054,522
32.14Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
32.14Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
32.14Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
32.14Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
32.14Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
32.00Single5IUAQ274563485IUA-A2A-Q27456348-Na
32.00Single5N2RPSB-365N2R-A2A-PSB-36-Na
32.00Single5N2SPSB365N2S-A1-PSB36
32.00Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
32.00Single6S0QZM-2413856S0Q-A2A-ZM-241385
32.00Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
32.00Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
32.00Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
32.00Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
32.00Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
32.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
32.00Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
32.00Consensusadenosine_offOrthosteric Liganda1_off a2_off
31.82Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
31.82Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
31.82Consensusgq_nucleotideOrthosteric Ligandgq_p2y
31.82Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
31.25Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
31.25Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
31.25Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
31.25Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
31.25Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
31.03Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
31.03Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
31.03Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
31.03Single8WDTphotoNECA8WDT-A2A-photoNECA
31.03Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.03Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.03Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
31.03Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
31.03Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
31.03Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
31.03Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
31.03Consensussomatostatin_offOrthosteric Ligandsst2_off
30.77Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
30.77Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
30.77Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.77Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
30.77Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
30.77Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
30.77Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
30.77Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
30.77Consensusrelaxin_onOrthosteric Ligandrxfp4_on
30.77Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
30.43Single3ODUIT1t3ODU-CXCR4-IT1t
30.43Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
30.43Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
30.43Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
30.43Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
30.43Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
30.43Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
30.43Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
30.30Single6FJ3PTH6FJ3-PTH1-PTH
30.30Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.30Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
30.30Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single3QAKUK-4320973QAK-A2A-UK-432097
30.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
30.00Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
30.00Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
30.00Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
30.00Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
30.00Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
30.00Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
30.00Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
30.00Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
30.00Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
29.63Single4XEENeurotensin4XEE-NTS1-Neurotensin
29.63Single4XESNeurotensin4XES-NTS1-Neurotensin
29.63Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
29.63Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
29.63Single6YVRNTS8-136YVR-NTS1-NTS8-13
29.63Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
29.63Single7K15MKD0467K15-BLT1-MKD046-Na
29.63Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
29.63Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.63Single8JJLOlodaterol8JJL-β2-Olodaterol
29.63Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
29.63Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
29.63Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
29.63Single8XQJJN2418XQJ-Apelin-JN241
29.63Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
29.63Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
29.63Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
29.63Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
29.63Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
29.63Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
29.63Consensuslpa_offOrthosteric Ligandlpa1_off
29.63Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
29.63Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
29.41Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
29.41Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
29.17Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
29.17Single5IUBQ274563445IUB-A2A-Q27456344-Na
29.17Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
29.17Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
29.17Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
29.17Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
29.17Single6MH8ZM-2413856MH8-A2A-ZM-241385
29.17Single7T32ZM-2413857T32-A2A-ZM-241385
29.17Single8IHKAcifran8IHK-HCA3-Acifran
29.17Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
29.17Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
29.17Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
29.17Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
29.17Single8K5CAcipimox8K5C-HCA2-Acipimox
29.17Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
29.17Consensushca_onOrthosteric Ligandhca2_on
29.03Single5WF5UK-4320975WF5-A2A-UK-432097
29.03Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
29.03Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
29.03Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
29.03Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.03Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
29.03Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
29.03Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
29.03Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
29.03Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
29.03Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
29.03Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
29.03Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
29.03Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
29.03Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
28.57Single4BUONeurotensin4BUO-NTS1-Neurotensin
28.57Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
28.57Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
28.57Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
28.57Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
28.57Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
28.57Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
28.57Single7EZCUKA7EZC-A2A-UKA
28.57Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
28.57Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
28.57Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
28.57Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
28.57Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.57Consensuscck_onOrthosteric Ligandccka_on cckb_on
28.57Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
28.12Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
28.12Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
28.12Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
28.12Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.12Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single3EMLZM-2413853EML-A2A-ZM-241385
28.00Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
28.00Single5IU8Q274563475IU8-A2A-Q27456347-Na
28.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
28.00Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
28.00Single5UENDU1725UEN-A1-DU172
28.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
28.00Single6S0LZM-2413856S0L-A2A-ZM-241385
28.00Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
28.00Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
28.00Single7PYRPSB-21157PYR-A2A-PSB-2115
28.00Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
28.00Single8CU6LJ-45178CU6-A2A-LJ-4517
28.00Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
28.00Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
28.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
28.00Single8K5DGSK2560738K5D-HCA2-GSK256073
28.00Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
28.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
28.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
28.00Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
28.00Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
28.00Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
28.00Consensushca_on_gpOrthosteric Ligandhca2_on_gp
28.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
27.78Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
27.78Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
27.78Consensusbombesin_onOrthosteric Ligandbb2_on
27.78Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
27.78Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
27.59Single5WF6UK-4320975WF6-A2A-UK-432097
27.59Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.59Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
27.59Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
27.59Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
27.59Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
27.59Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
27.59Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
27.59Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single4XNWMRS25004XNW-P2Y1-MRS2500
27.27Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
27.27Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
27.27Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
27.27Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
27.27Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
26.92Single4JKVTaladegib4JKV-SMO-Taladegib
26.92Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
26.92Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
26.92Single7C61Ergotamine7C61-5-HT1B-Ergotamine
26.92Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
26.92Single7W41PD1762527W41-BB2-PD176252
26.92Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
26.92Single8GNEKW-63568GNE-A2A-KW-6356-Na
26.92Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
26.92Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
26.92Single8TF5Oleic acid8TF5-GPR6-Oleic acid
26.92Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
26.92Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
26.92Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
26.92Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
26.92Consensusbombesin_offOrthosteric Ligandbb2_off
26.92Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
26.92Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
26.92Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
26.92Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
26.67Single4IARErgotamine4IAR-5-HT1B-Ergotamine
26.67Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
26.67Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
26.67Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
26.67Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
26.67Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
26.67Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
26.67Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
26.67Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
26.67Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
26.67Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
26.67Consensuslpl_onOrthosteric Ligands1p_on lpa_on
26.67Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
26.67Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
26.47Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
26.47Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
26.09Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
26.09Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
26.09Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
26.09Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
26.09Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
26.09Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
26.09Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
25.93Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
25.93Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
25.93Single5V56TC1145V56-SMO-TC114
25.93Single5V57TC1145V57-SMO-TC114
25.93Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
25.93Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
25.93Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
25.93Single7B6WCyclazosin7B6W-α1b-Cyclazosin
25.93Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
25.93Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
25.93Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
25.93Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
25.93Single7R0CAVP7R0C-V2-AVP-Arrestin2
25.93Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
25.93Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
25.93Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
25.93Single8E0GBU728E0G-μ-BU72
25.93Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
25.93Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
25.93Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
25.93Single9BJKNAM9BJK-μ-Naloxone-NAM
25.93Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensusneurotensin_onOrthosteric Ligandnts1_on
25.93Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
25.93Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
25.93Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
25.81Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
25.81Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
25.81Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
25.81Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
25.71Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
25.71Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
25.71Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
25.64Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
25.64Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
25.00Single3PWHZM-2413853PWH-A2A-ZM-241385
25.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
25.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
25.00Single4BWBNeurotensin4BWB-NTS1-Neurotensin
25.00Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
25.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
25.00Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
25.00Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
25.00Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
25.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
25.00Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
25.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
25.00Single6A93Risperidone6A93-5-HT2A-Risperidone
25.00Single6AKYMaraviroc6AKY-CCR5-Maraviroc
25.00Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
25.00Single6MXTSalmeterol6MXT-β2-Salmeterol
25.00Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
25.00Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
25.00Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
25.00Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
25.00Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
25.00Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
25.00Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
25.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
25.00Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
25.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
25.00Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
25.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
25.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
25.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
25.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
25.00Single7XRRLemborexant7XRR-OX2-Lemborexant
25.00Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
25.00Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
25.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
25.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
25.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
25.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
25.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
25.00Single8XYIVUF106618XYI-CXCR3-VUF10661
25.00Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
25.00Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
25.00Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
25.00Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
25.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
25.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
25.00Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
25.00Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
25.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
25.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
25.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
25.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
25.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
25.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
25.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
25.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
25.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
24.32Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
24.32Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
24.24Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
24.24Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
24.24Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
24.24Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
24.24Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
24.24Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
24.24Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
24.24Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
24.24Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
24.24Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
24.14Single6IBLArformoterol6IBL-β1-Arformoterol
24.14Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
24.14Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
24.14Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
24.14Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
24.14Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.14Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
24.14Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
24.14Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
24.14Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
24.14Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
24.14Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
24.14Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
24.14Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
24.14Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
24.14Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
24.14Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
24.14Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
24.14Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
24.14Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
24.14Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
24.14Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
24.00Single3REYXAC3REY-A2A-XAC
24.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
24.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
24.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
24.00Single5JTBZM-2413855JTB-A2A-ZM-241385
24.00Single5UVIZM-2413855UVI-A2A-ZM-241385
24.00Single6AQFZM-2413856AQF-A2A-ZM-241385
24.00Single6V9SGTPL114036V9S-OX1-GTPL11403
24.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
24.00Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
24.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
24.00Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
24.00Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
24.00Single8K2WAMG4878K2W-CXCR3-AMG487
24.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
24.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
24.00Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
24.00Consensusa2_offOrthosteric Liganda2a_off
24.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
24.00Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
24.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
24.00Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
24.00Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
24.00Consensusgrh_offOrthosteric Ligandgnrh1_off
23.81Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
23.68Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
23.68Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
23.68Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
23.53Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
23.53Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
23.53Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
23.53Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
23.33Single4UG2CGS216804UG2-A2A-CGS21680
23.33Single5EE7MK08935EE7-Glucagon-MK0893
23.33Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
23.33Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
23.33Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
23.33Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
23.33Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
23.33Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
23.33Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
23.33Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
23.33Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
23.33Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
23.08Single4QIMANTA XV4QIM-SMO-ANTA XV
23.08Single4YAYZD-71554YAY-AT1-ZD-7155
23.08Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
23.08Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
23.08Single5TGZAM65385TGZ-CB1-AM6538
23.08Single5UIGCmpd-15UIG-A2A-Cmpd-1
23.08Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
23.08Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
23.08Single6TOTLemborexant6TOT-OX1-Lemborexant
23.08Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
23.08Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
23.08Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
23.08Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
23.08Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
23.08Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
23.08Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
23.08Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
23.08Single7UL4Alvimopan7UL4-μ-Alvimopan
23.08Single7V3ZCP559407V3Z-CB1-CP55940
23.08Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
23.08Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
23.08Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
23.08Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
23.08Single7YXAONO-54306087YXA-S1P5-ONO-5430608
23.08Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
23.08Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
23.08Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
23.08Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
23.08Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
23.08Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
23.08Single9B9ZA1AKO9B9Z-CB1-A1AKO
23.08Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
23.08Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
23.08Consensuscck_offOrthosteric Ligandccka_off
23.08Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
23.08Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
22.86Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
22.86Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
22.86Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
22.86Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
22.73Single3OE8IT1t3OE8-CXCR4-IT1t
22.73Single8A2OTheophylline8A2O-A2A-Theophylline-Na
22.73Consensusp2y_offOrthosteric Ligandp2y1_off
22.58Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
22.58Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
22.58Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
22.58Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
22.58Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
22.58Single8KIGSHU91198KIG-MC3-SHU9119-Ca
22.58Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
22.58Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
22.22Single2Y00Dobutamine2Y00-β1-Dobutamine
22.22Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
22.22Single5C1MBU725C1M-μ-BU72
22.22Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
22.22Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
22.22Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
22.22Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
22.22Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
22.22Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
22.22Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
22.22Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
22.22Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
22.22Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
22.22Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
22.22Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
22.22Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
22.22Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
22.22Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
22.22Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
22.22Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
22.22Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
22.22Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
22.22Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
22.22Single8JXSPF-61428JXS-D1-PF-6142
22.22Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
22.22Single8QOTNanobody-E8QOT-μ-Nanobody-E
22.22Single8S4DCMF-0198S4D-Apelin-CMF-019
22.22Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
22.22Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
22.22Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
22.22Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
22.22Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
22.22Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
22.22Consensusblt_offOrthosteric Ligandblt1_off
22.22Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
22.22Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
22.22Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
22.22Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
22.22Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
22.22Consensusep_offOrthosteric Ligandep4_off
22.22Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
22.22Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
22.22Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
21.88Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
21.88Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
21.88Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
21.88Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
21.88Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
21.88Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
21.88Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
21.88Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
21.74Single7V6A-7V6A-M4-PubChem 9864275-Gi1/β1/γ2
21.74Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
21.62Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
21.62Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
21.62Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
21.62Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
21.62Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
21.43Single3P0GBI1671073P0G-β2-BI167107
21.43Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
21.43Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
21.43Single4BV0Neurotensin4BV0-NTS1-Neurotensin
21.43Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
21.43Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
21.43Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
21.43Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
21.43Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
21.43Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
21.43Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
21.43Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
21.43Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
21.43Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
21.43Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
21.43Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
21.43Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
21.43Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
21.43Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
21.43Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
21.43Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
21.43Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
21.43Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
21.43Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
21.43Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
21.43Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
21.43Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
21.43Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
21.43Consensuslpa_onOrthosteric Ligandlpa1_on
21.43Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
21.43Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Single6PT2KGCHM076PT2-δ-KGCHM07
21.21Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
21.21Single6W25SHU91196W25-MC4-SHU9119-Ca
20.93Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
20.83Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
20.83Single4O9RCyclopamine4O9R-SMO-Cyclopamine
20.83Single5L7IVismodegib5L7I-SMO-Vismodegib
20.83Single6LI0C176LI0-GPR52-C17
20.83Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
20.83Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
20.83Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
20.83Single8K5BNiacin8K5B-HCA2-Niacin
20.83Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
20.83Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
20.83Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
20.83Single9B9Y7DY9B9Y-CB1-7DY
20.83Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
20.69Single4LDEBI1671074LDE-β2-BI167107
20.69Single4RWADIPP-NH24RWA-δ-DIPP-NH2
20.69Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
20.69Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
20.69Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
20.69Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
20.69Single6ZG4HTL00099366ZG4-M1-HTL0009936
20.69Single7DFPSpiperone7DFP-D2-Spiperone
20.69Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
20.69Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.69Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
20.69Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
20.69Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
20.69Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.69Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
20.69Single7YITNalfurafine7YIT-κ-Nalfurafine
20.69Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
20.69Single8JJ8Formoterol8JJ8-β2-Formoterol
20.69Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
20.69Single8JWY2-1188JWY-A2A-2-118
20.69Single8JWZAB9288JWZ-A2A-AB928-Na
20.69Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
20.69Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.69Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
20.69Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.69Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.69Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
20.69Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
20.69Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
20.69Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
20.69Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
20.69Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
20.69Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
20.69Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
20.69Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
20.69Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
20.69Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
20.69Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.69Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.59Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
20.59Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
20.59Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
20.51Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
20.51Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
20.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
20.00Single4QINSAG1.54QIN-SMO-SAG1.5
20.00Single4S0VSuvorexant4S0V-OX2-Suvorexant
20.00Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
20.00Single5U09Taranabant5U09-CB1-Taranabant
20.00Single5WS3EMPA5WS3-OX2-EMPA
20.00Single6AKXA4R6AKX-CCR5-A4R
20.00Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
20.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
20.00Single6H7LDobutamine6H7L-β1-Dobutamine
20.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
20.00Single6TPJSuvorexant6TPJ-OX2-Suvorexant
20.00Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
20.00Single7BR3Elagolix7BR3-GnRH1-Elagolix
20.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
20.00Single7F8ULintitript7F8U-CCKA-Lintitript
20.00Single7F8YDevazepide7F8Y-CCKA-Devazepide
20.00Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
20.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
20.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
20.00Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
20.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
20.00Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
20.00Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
20.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
20.00Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
20.00Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
20.00Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
20.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
20.00Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
20.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
20.00Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
20.00Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
20.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
20.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
20.00Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
20.00Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
20.00Single8Y0HVUF114188Y0H-CXCR3-VUF11418
20.00Single9BA0A1AKN9BA0-CB1-A1AKN
20.00Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
20.00Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
20.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
20.00Consensusangiotensin_offOrthosteric Ligandat1_off
20.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.00Consensuschemerin_onOrthosteric Ligandcml1_on
20.00Consensusendothelin_offOrthosteric Ligandetb_off
20.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
20.00Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
20.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
20.00Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusorexin_offOrthosteric Ligandox2_off ox1_off
20.00Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
20.00Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
19.51Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
19.51Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.44Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
19.44Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
19.44Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
19.44Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
19.44Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
19.44Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
19.35Single3NY9ICI118-5513NY9-β2-ICI118-551
19.35Single5ZTYAM102575ZTY-CB2-AM10257
19.35Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
19.35Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
19.35Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single7SK9CCX6627SK9-ACKR3-CCX662
19.35Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
19.35Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
19.35Single8X5YAstemizole8X5Y-H1-Astemizole
19.35Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
19.23Single2YDOAdenosine2YDO-A2A-Adenosine
19.23Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
19.23Single4ZJCSB-6740424ZJC-OX1-SB-674042
19.23Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
19.23Single6IQLL7458706IQL-D4-L745870
19.23Single6KUXRS-799486KUX-α2a-RS-79948
19.23Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
19.23Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
19.23Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
19.23Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
19.23Single6TP3Nemorexant6TP3-OX1-Nemorexant
19.23Single6TPGEMPA6TPG-OX2-EMPA
19.23Single6ZG9GSK10347026ZG9-M1-GSK1034702
19.23Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
19.23Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.23Single7UL3Famotidine7UL3-H2-Famotidine
19.23Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
19.23Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
19.23Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
19.23Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
19.23Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
19.23Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
19.23Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
19.23Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
19.23Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
19.23Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
19.23Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
19.23Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
19.23Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
19.23Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
19.23Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
19.05Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
18.92Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
18.92Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
18.92Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
18.92Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
18.75Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
18.75Single7QA8Peptide7QA8-STE2-Peptide
18.75Single7QA8Peptide7QA8-STE2-Peptide
18.75Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
18.75Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
18.75Single8IEBA1LYA8IEB-GPR156-A1LYA
18.75Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
18.75Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
18.75Single8WKYPG-9348WKY-MC4-PG-934
18.75Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.75Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.75Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.75Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
18.52Single2Y01Dobutamine2Y01-β1-Dobutamine
18.52Single2Y02Carmoterol2Y02-β1-Carmoterol
18.52Single2Y04Salbutamol2Y04-β1-Salbutamol
18.52Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
18.52Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
18.52Single4QKX35V4QKX-β2-35V
18.52Single5T04Neurotensin5T04-NTS1-Neurotensin
18.52Single6DRXLisuride6DRX-5-HT2B-Lisuride
18.52Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
18.52Single6GPSMK08126GPS-CCR2-MK0812
18.52Single6PS1Timolol6PS1-β2-Timolol
18.52Single7BU7BI1671077BU7-β1-BI167107
18.52Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
18.52Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
18.52Single7F83PF-051904577F83-Ghrelin-PF-05190457
18.52Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
18.52Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
18.52Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
18.52Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
18.52Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
18.52Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
18.52Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
18.52Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
18.52Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
18.52Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
18.52Single8RLNLUF58348RLN-A2A-LUF5834
18.52Single8T1WCVN4248T1W-GPR6-CVN424
18.52Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
18.52Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
18.52Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
18.52Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
18.52Single9CHXS-Carazolol9CHX-β2-S-Carazolol
18.52Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
18.52Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
18.52Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
18.52Consensusa3_onOrthosteric Liganda3a_on
18.52Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
18.52Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
18.52Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
18.42Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
18.42Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
18.42Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
18.42Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
18.42Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
18.42Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
18.18Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
18.18Single6HLOAprepitant6HLO-NK1-Aprepitant
18.18Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
18.18Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
18.18Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
18.18Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
18.18Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
18.18Single8PWNTheophylline8PWN-A2A-Theophylline
18.18Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
17.95Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
17.95Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
17.86Single2Y03Isoprenaline2Y03-β1-Isoprenaline
17.86Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
17.86Single5WIUNemonapride5WIU-D4-Nemonapride
17.86Single5WIVNemonapride5WIV-D4-Nemonapride-Na
17.86Single5WQCEMPA5WQC-OX2-EMPA
17.86Single6E67BI1671076E67-β2-BI167107-Gs (fused)
17.86Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
17.86Single6GPXMK08126GPX-CCR2-MK0812
17.86Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
17.86Single6LUQHaloperidol6LUQ-D2-Haloperidol
17.86Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
17.86Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
17.86Single6TP6Filorexant6TP6-OX1-Filorexant
17.86Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
17.86Single7C4SS1P7C4S-S1P3-S1P
17.86Single7SINNPS-21437SIN-CaS-NPS-2143
17.86Single7SINNPS-21437SIN-CaS-NPS-2143
17.86Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
17.86Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
17.86Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
17.86Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
17.86Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
17.86Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
17.86Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
17.86Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
17.86Consensusa3_on_gpOrthosteric Liganda3a_on_gp
17.86Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.86Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.86Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
17.86Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.86Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
17.86Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
17.86Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
17.86Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Consensustrace-amine_onOrthosteric Ligandta1_on
17.65Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
17.65Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.65Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.50Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
17.50Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.39Single3RFMCaffeine3RFM-A2A-Caffeine
17.39Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
17.39Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single2YDVNECA2YDV-A2A-NECA
17.24Single4UHRCGS216804UHR-A2A-CGS21680
17.24Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
17.24Single5G53NECA5G53-A2A-NECA-Gs
17.24Single5TZRMK86665TZR-FFA1-MK8666
17.24Single5XR8AM8415XR8-CB1-AM841
17.24Single5XRAAM115425XRA-CB1-AM11542
17.24Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
17.24Single6H7JIsoprenaline6H7J-β1-Isoprenaline
17.24Single6J20Aprepitant6J20-NK1-Aprepitant
17.24Single6J21Aprepitant6J21-NK1-Aprepitant
17.24Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
17.24Single6TQ7SB-3348676TQ7-OX1-SB-334867
17.24Single6WGTLSD6WGT-5-HT2A-LSD
17.24Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
17.24Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
17.24Single7FEECP559407FEE-CB1-CP55940-ZCZ011
17.24Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
17.24Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
17.24Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
17.24Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
17.24Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
17.24Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
17.24Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
17.24Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
17.24Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
17.24Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
17.24Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
17.24Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.24Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
17.24Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
17.24Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
17.24Single8XVLZibotentan8XVL-ETA-Zibotentan
17.24Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
17.24Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
17.24Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
17.24Consensusa2_onOrthosteric Liganda2b_on
17.24Consensusa2_on_gpOrthosteric Liganda2b_on_gp
17.24Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.24Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.24Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
17.24Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
17.24Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.24Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
17.24Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
17.24Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
17.24Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.24Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
17.14Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
17.14Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
17.14Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
17.07Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
16.67Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
16.67Single4AMIBucindolol4AMI-β1-Bucindolol
16.67Single4N4WSANT-14N4W-SMO-SANT-1
16.67Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
16.67Single4PY02MeSATP4PY0-P2Y12-2MeSATP
16.67Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
16.67Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
16.67Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
16.67Single5X33BIIL2605X33-BLT1-BIIL260
16.67Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
16.67Single6CM4Risperidone6CM4-D2-Risperidone
16.67Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
16.67Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
16.67Single6KQICP559406KQI-CB1-CP55940-Org27569
16.67Single6ME5Agomelatine6ME5-MT1-Agomelatine
16.67Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
16.67Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
16.67Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
16.67Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
16.67Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
16.67Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
16.67Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
16.67Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
16.67Single7WC5Psilocin7WC5-5-HT2A-Psilocin
16.67Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
16.67Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
16.67Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
16.67Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
16.67Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
16.67Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
16.67Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
16.67Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
16.67Single8JPSCCL78JPS-ACKR1-CCL7
16.67Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
16.67Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
16.67Consensusalpha1_offOrthosteric Ligandalpha1a_off
16.67Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
16.67Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
16.67Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.67Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
16.22Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
16.22Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
16.13Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
16.13Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
16.13Single5X93K-87945X93-ETB-K-8794
16.13Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
16.13Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
16.13Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
16.13Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
16.13Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
16.13Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
16.13Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
16.13Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
16.13Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
16.13Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
16.13Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
16.13Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
16.13Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
16.13Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
16.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
16.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
16.00Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
16.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
16.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
16.00Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
16.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
16.00Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
16.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
15.79Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
15.79Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
15.79Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
15.79Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
15.79Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
15.79Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
15.62Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
15.62Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
15.62Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
15.62Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
15.62Consensuskisspeptin_onOrthosteric Ligandkiss1_on
15.38Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
15.38Single6ME9Ramelteon6ME9-MT2-Ramelteon
15.38Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
15.38Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
15.38Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
15.38Single6TODEMPA6TOD-OX1-EMPA-Na
15.38Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
15.38Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
15.38Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
15.38Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
15.38Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
15.38Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
15.38Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
15.38Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
15.38Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
15.38Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
15.38Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
15.38Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
15.38Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
15.38Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
15.38Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
15.38Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
15.38Single8IWESpermidine8IWE-TA9-Spermidine
15.38Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
15.38Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
15.38Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
15.38Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
15.38Consensusalpha2_offOrthosteric Ligandalpha2c_off
15.38Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
15.22Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
15.15Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
15.15Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
15.15Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
15.15Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Single8IEIA1LYA8IEI-GPR156-A1LYA
15.15Single8IEPA1LYA8IEP-GPR156-A1LYA
15.15Single8IEPA1LYA8IEP-GPR156-A1LYA
15.15Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
15.15Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
15.15Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
15.00Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
14.81Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
14.81Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
14.81Single6PS0S-Carazolol6PS0-β2-S-Carazolol
14.81Single6PS4ICI118-5516PS4-β2-ICI118-551
14.81Single6PS5S-Propranolol6PS5-β2-S-Propranolol
14.81Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
14.81Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
14.81Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
14.81Single6ZINSR486926ZIN-NTS1-SR48692
14.81Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
14.81Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
14.81Single7VV6C48/807VV6-MRGPRX2-C48/80
14.81Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
14.81Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
14.81Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
14.81Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
14.81Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
14.81Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
14.81Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
14.81Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
14.81Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
14.81Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
14.81Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
14.81Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
14.81Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
14.81Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
14.81Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
14.81Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
14.81Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
14.81Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
14.71Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
14.71Single8IEBA1LYA8IEB-GPR156-A1LYA
14.29Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
14.29Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
14.29Single3NY8ICI118-5513NY8-β2-ICI118-551
14.29Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
14.29Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
14.29Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
14.29Single4GBRS-Carazolol4GBR-β2-S-Carazolol
14.29Single5DHGC-355DHG-NOP-C-35
14.29Single5DHHSB-6121115DHH-NOP-SB-612111
14.29Single6H7MSalbutamol6H7M-β1-Salbutamol
14.29Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
14.29Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
14.29Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
14.29Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
14.29Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
14.29Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
14.29Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
14.29Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
14.29Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
14.29Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
14.29Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
14.29Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
14.29Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
14.29Single7WC7Lisuride7WC7-5-HT2A-Lisuride
14.29Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
14.29Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
14.29Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
14.29Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
14.29Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
14.29Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
14.29Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
14.29Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
14.29Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
14.29Single8JJOAlprenolol8JJO-β2-Alprenolol
14.29Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
14.29Single8JXRLSD8JXR-D1-LSD
14.29Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
14.29Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
14.29Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
14.29Consensus5ht5_onOrthosteric Ligand5ht5a_on
14.29Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
14.29Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
14.29Consensusdopamine_offOrthosteric Ligandd2_off d3_off
14.29Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
14.29Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
14.29Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
13.95Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
13.89Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
13.89Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
13.89Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
13.79Single2RH1S-Carazolol2RH1-β2-S-Carazolol
13.79Single2YCWS-Carazolol2YCW-β1-S-Carazolol
13.79Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
13.79Single5D6LS-Carazolol5D6L-β2-S-Carazolol
13.79Single5JQHS-Carazolol5JQH-β2-S-Carazolol
13.79Single5TVNLSD5TVN-5-HT2B-LSD
13.79Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
13.79Single5XPRBosentan5XPR-ETB-Bosentan
13.79Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
13.79Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
13.79Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
13.79Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
13.79Single6PS6Timolol6PS6-β2-Timolol
13.79Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
13.79Single6Z4SSR486926Z4S-NTS1-SR48692
13.79Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
13.79Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
13.79Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
13.79Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.79Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
13.79Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
13.79Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
13.79Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
13.79Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
13.79Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.79Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
13.79Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
13.79Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
13.79Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
13.79Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
13.79Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
13.79Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
13.79Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
13.79Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
13.79Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
13.79Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
13.79Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
13.79Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
13.79Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
13.79Consensusamine_offonOrthosteric Ligandamine_off amine_on
13.79Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
13.79Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
13.79Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
13.79Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
13.79Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.64Single5MZPCaffeine5MZP-A2A-Caffeine-Na
13.64Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
13.64Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
13.51Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.33Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
13.33Single4DJHJDTic4DJH-κ-JDTic
13.33Single5D5AS-Carazolol5D5A-β2-S-Carazolol
13.33Single5D5BS-Carazolol5D5B-β2-S-Carazolol
13.33Single6E59L-7607356E59-NK1-L-760735
13.33Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
13.33Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
13.33Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
13.33Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
13.33Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
13.33Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
13.33Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
13.33Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
13.33Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
13.33Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
13.33Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
13.33Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
13.33Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
13.33Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
13.33Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
13.33Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
13.33Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
13.33Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
13.33Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
13.33Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
13.33Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
13.33Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
13.33Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
13.33Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.33Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
13.33Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
13.33Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
13.33Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
13.33Consensustachykinin_offOrthosteric Ligandnk1_off
13.04Single7WC4Serotonin7WC4-5-HT2A-Serotonin
13.04Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.04Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
13.04Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
13.04Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.90Single3D4STimolol3D4S-β2-Timolol
12.90Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
12.90Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
12.90Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
12.90Single6IIURamatroban6IIU-TP-Ramatroban
12.90Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
12.90Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
12.90Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.90Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
12.90Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.90Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
12.90Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
12.90Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.90Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
12.90Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
12.50Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
12.50Single6K1QIRL25006K1Q-ETB-IRL2500
12.50Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
12.50Single6TQ9SB-4081246TQ9-OX1-SB-408124
12.50Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
12.50Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.50Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
12.50Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
12.50Single7UM4AS26747237UM4-5-HT5A-AS2674723
12.50Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
12.50Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
12.50Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
12.50Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
12.50Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
12.50Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
12.50Single9CHUNoradrenaline9CHU-β2-Noradrenaline
12.50Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
12.50Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
12.50Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
12.50Consensussensory_onOrthosteric Ligandopsins_on
12.50Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single6PT3DPI-2876PT3-δ-DPI-287
12.12Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
12.12Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
12.12Single8IEIA1LYA8IEI-GPR156-A1LYA
12.12Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.00Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
12.00Single3UZAGTPL92363UZA-A2A-GTPL9236
12.00Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
12.00Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
12.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
12.00Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
12.00Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
12.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
12.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
12.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
12.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
12.00Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
12.00Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
12.00Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
12.00Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
12.00Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
12.00Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
12.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
12.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
12.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.00Consensus5ht2_onOrthosteric Ligand5ht2b_on
12.00Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.00Consensusgi_sensoryOrthosteric Ligandgi_opsins
12.00Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.00Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.00Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.00Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
12.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
11.76Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
11.76Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
11.54Single3PBLEticlopride3PBL-D3-Eticlopride
11.54Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
11.54Single6HLLCP999946HLL-NK1-CP99994
11.54Single6TP4ACT-4622066TP4-OX1-ACT-462206
11.54Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
11.54Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.54Single7SRQLSD7SRQ-5-HT2B-LSD
11.54Single7UL2SR486927UL2-NTS1-SR48692-Na
11.54Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
11.54Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
11.54Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.54Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
11.54Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
11.54Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
11.54Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
11.54Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
11.54Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
11.54Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
11.54Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
11.54Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
11.54Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
11.54Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
11.54Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.54Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.54Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
11.54Consensusneurotensin_offOrthosteric Ligandnts1_off
11.54Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
11.11Single6B73MP11046B73-κ-MP1104
11.11Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
11.11Single6ME2Ramelteon6ME2-MT1-Ramelteon
11.11Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
11.11Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
11.11Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
11.11Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
11.11Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
11.11Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
11.11Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
11.11Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
11.11Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
11.11Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
11.11Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
11.11Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
11.11Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
11.11Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
11.11Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
11.11Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
11.11Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
11.11Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
11.11Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
11.11Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
11.11Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
11.11Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
11.11Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
11.11Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
11.11Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.11Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
11.11Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.11Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
11.11Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
11.11Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
11.11Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
10.81Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
10.81Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
10.71Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
10.71Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
10.71Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
10.71Single6A94Zotepine6A94-5-HT2A-Zotepine
10.71Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
10.71Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
10.71Single6TPKRetosiban6TPK-OT-Retosiban
10.71Single6TPNHTL66416TPN-OX2-HTL6641
10.71Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
10.71Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
10.71Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
10.71Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
10.71Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
10.71Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
10.71Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
10.71Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
10.71Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
10.71Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
10.71Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
10.71Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
10.71Single7VODCariprazine7VOD-5-HT2A-Cariprazine
10.71Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
10.71Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
10.71Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.71Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
10.71Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
10.71Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.71Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
10.71Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
10.71Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
10.71Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
10.71Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
10.71Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
10.71Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
10.71Consensusalpha1_onOrthosteric Ligandalpha1a_on
10.71Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
10.71Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
10.71Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
10.71Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
10.71Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
10.71Consensusopsins_offOrthosteric Ligandrhodopsin_off
10.71Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
10.71Consensussensory_offOrthosteric Ligandopsins_off
10.71Consensusvasop-oxy_offOrthosteric Ligandot_off
10.34Single4DAJTiotropium4DAJ-M3-Tiotropium
10.34Single4EJ4Naltrindole4EJ4-δ-Naltrindole
10.34Single4MQSIperoxo4MQS-M2-Iperoxo
10.34Single4U14Tiotropium4U14-M3-Tiotropium
10.34Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
10.34Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
10.34Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
10.34Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
10.34Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
10.34Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
10.34Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
10.34Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
10.34Single6IIVDaltroban6IIV-TP-Daltroban
10.34Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.34Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
10.34Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.34Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
10.34Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
10.34Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
10.34Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
10.34Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
10.34Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
10.34Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
10.34Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
10.34Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
10.34Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
10.34Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
10.34Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
10.34Single8X63Mepyramine8X63-H1-Mepyramine
10.34Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
10.34Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
10.34Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
10.34Single9IYAONO-97105319IYA-GPR55-ONO-9710531
10.34Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.34Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.34Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
10.34Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
10.34Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
10.34Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
10.34Consensusalpha2_onOrthosteric Ligandalpha2b_on
10.34Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
10.34Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.34Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.34Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
10.34Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
10.34Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
10.34Consensusblt_onOrthosteric Ligandblt1_on
10.34Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
10.34Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
10.34Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
10.34Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
10.34Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
10.34Consensushistamine_offOrthosteric Ligandh1_off
10.34Consensusleukotriene_onOrthosteric Ligandblt_on
10.34Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
10.34Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
10.34Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
10.00Single5CGCHTL142425CGC-mGlu5-HTL14242
10.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
10.00Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
10.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
10.00Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
10.00Single7WC6LSD7WC6-5-HT2A-LSD
10.00Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8ZMFA1L108ZMF-5-HT2C-A1L10
10.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
10.00Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
10.00Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
10.00Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
10.00Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
10.00Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
10.00Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.00Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
10.00Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.00Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
10.00Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single4U15Tiotropium4U15-M3-Tiotropium
9.68Single5V54Methiothepin5V54-5-HT1B-Methiothepin
9.68Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
9.68Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
9.68Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
9.68Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
9.68Single6OL9Tiotropium6OL9-M5-Tiotropium
9.68Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
9.68Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
9.68Single8EA0Iperoxo8EA0-M3-Iperoxo
9.68Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
9.68Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
9.68Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
9.68Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
9.68Consensus5ht1_offOrthosteric Ligand5ht1b_off
9.68Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
9.68Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
9.68Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
9.68Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
9.68Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
9.68Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
9.38Single5CXVTiotropium5CXV-M1-Tiotropium
9.38Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
9.38Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
9.38Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
9.38Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
9.38Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
9.09Single5CGDHTL142425CGD-mGlu5-HTL14242
9.09Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
9.09Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
9.09Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
8.82Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
8.70Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
8.33Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
8.33Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
8.33Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.00Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
8.00Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
8.00Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
8.00Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
8.00Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
7.69Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
7.69Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
7.69Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
7.69Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
7.69Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
7.69Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
7.69Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
7.69Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
7.69Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
7.69Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
7.69Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
7.69Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
7.69Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
7.69Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
7.41Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
7.41Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
7.41Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
7.41Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
7.41Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
7.41Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
7.41Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
7.41Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
7.41Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
7.41Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.41Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
7.41Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
7.41Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
7.41Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
7.41Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
7.41Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
7.41Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
7.41Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.41Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
7.41Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.41Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
7.41Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
7.41Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.41Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.41Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
7.41Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.41Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
7.14Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
7.14Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
7.14Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
7.14Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
7.14Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
7.14Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
7.14Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
7.14Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.14Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
7.14Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
7.14Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
7.14Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
7.14Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
7.14Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
7.14Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
7.14Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
7.14Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
7.14Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
6.90Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
6.90Single3RZECidoxepin3RZE-H1-Cidoxepin
6.90Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
6.90Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
6.90Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
6.90Single6VI4JDTic6VI4-κ-JDTic
6.90Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
6.90Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
6.90Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
6.90Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
6.90Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
6.90Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
6.90Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
6.90Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
6.90Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
6.90Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
6.90Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
6.90Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
6.90Single9BJKNaloxone9BJK-μ-Naloxone-NAM
6.67Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
6.67Single5DSGTiotropium5DSG-M4-Tiotropium
6.67Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
6.67Single8X64Desloratadine8X64-H1-Desloratadine
6.67Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
6.67Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
6.45Single4NTJAZD12834NTJ-P2Y12-AZD1283
6.45Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
6.45Single6HLPNetupitant6HLP-NK1-Netupitant
6.45Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
6.45Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
6.45Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
6.45Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
6.45Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
6.45Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
6.45Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.45Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.45Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.45Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
6.25Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
6.25Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
6.25Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
6.06Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
6.06Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
5.88Single8XVJMacitentan8XVJ-ETA-Macitentan
4.76Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.76Single6D35Cholesterol6D35-SMO-Cholesterol
4.76Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.76Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.76Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.76Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.76Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
4.76Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
4.76Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
4.76Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
4.76Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.76Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
4.76Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.76Single7DTTCa7DTT-CaS-Ca-Ca
4.76Single7DTTCa7DTT-CaS-Ca-Ca
4.76Single7DTUTryptophan7DTU-CaS-Tryptophan
4.76Single7DTUTryptophan7DTU-CaS-Tryptophan
4.76Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.76Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.76Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.76Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.76Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.76Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.76Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.76Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.76Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.76Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.76Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.76Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.76Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.76Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.76Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.76Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.76Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.76Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.76Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.76Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.76Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.76Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.76Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.76Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.76Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.76Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.76Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.76Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.76Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.76Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.76Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
4.76Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.76Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.76Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.76Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.76Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.76Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.76Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.76Single7XW7K1-707XW7-TSH-K1-70
4.76Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.76Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.76Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.76Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.76Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.76Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.76Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.76Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.76Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.76Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.76Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.76Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.76Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.76Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.76Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.76Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.76Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.76Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
4.76Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
4.76Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.76Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.76Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
4.76Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
4.76Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.76Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.76Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
4.76Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
4.76Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
4.76Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
4.76Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
4.76Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
4.76Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.76Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.76Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.76Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.76Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.76Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.76Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.76Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.76Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.76Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.76Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.76Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.76Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.76Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.76Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.76Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.76Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.76Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
4.76Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
4.76Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.76Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
4.76Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
4.76Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.76Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.76Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8WVXNorrin8WVX-LGR4-Norrin
4.76Single8WVYNorrin8WVY-LGR4-Norrin
4.76Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.76Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.76Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.76Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.76Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.76Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.76Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.76Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.76Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.76Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.76Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.76Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.76Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.76Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.76Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.76Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.76Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
4.76Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.35Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.35Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.17Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
4.17Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
4.17Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.17Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.17Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
4.17Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.17Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.00Single5L7DCholesterol5L7D-SMO-Cholesterol
4.00Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.00Single8HS2Fab0468HS2-GPR20-Fab046
4.00Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.85Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
3.85Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
3.70Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
3.70Single7F61Cholesterol7F61-H3-PF-03654746-Cholesterol
3.57Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
3.45Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
3.33Single6FFIMMPEP6FFI-mGlu5-MMPEP
3.33Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.23Single6FFHFenobam6FFH-mGlu5-Fenobam
3.23Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
3.12Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.12Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.12Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.12Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
3.12Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
3.03Single7P2L4YI7P2L-mGlu5-4YI
3.03Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
3.03Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
3.03Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.03Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
2.70Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.70Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.56Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.56Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.50Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.33Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
6WWZ 6WWZ-CCR6-CCL20-Go/β1/γ2
8HNK 8HNK-CXCR3-CXCL11-Gi1/β1/γ2
8K3Z 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
8IC0 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
6LFM 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
8KFX 8KFX-CCR8-LMD-009-Gi1/β1/γ2
7F1Q 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
8HNL 8HNL-CXCR3-PS372424-Gi1/β1/γ2
8KFY 8KFY-CCR8-ZK-756326-Gi1/β1/γ2
7O7F 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
8U1U 8U1U-CCR8-CCL1-Gi1/β1/γ2
7VLA 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7XA3 7XA3-CCR2-CCL2-Gi1/β1/γ2
Net Summary
Imin 2.62538
Number of Linked Nodes 945
Number of Links 1173
Number of Hubs 201
Number of Links mediated by Hubs 764
Number of Communities 22
Number of Nodes involved in Communities 261
Number of Links involved in Communities 396
Path Summary
Number Of Nodes in MetaPath 91
Number Of Links MetaPath 90
Number of Shortest Paths 2712955
Length Of Smallest Path 3
Average Path Length 36.3372
Length of Longest Path 65
Minimum Path Strength 0.314231
Average Path Strength 5.17905
Maximum Path Strength 30.8651
Minimum Path Correlation 0.700769
Average Path Correlation 0.979506
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.85185
Average % Of Corr. Nodes 35.2273
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 56.61
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
gi_proteingi_chemokine
gi_chemerin



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