Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 2.43182502
2G.HN.45 1.3175404
3G.S1.01 4.68023436
4G.S1.02 4.92527545
5G.H1.01 3.94909549
6G.S2.05 4.7325433
7G.S2.08 6.97659445
8G.S3.03 8.33409447
9G.S3.04 6.37418536
10G.S3.05 3.07848647
11G.S3.06 7.06076635
12G.S3.07 3.58523449
13G.s3h2.03 4.16545539
14G.H2.02 3.8225438
15G.H2.04 3.36818409
16G.H2.06 4.91151639
17G.H2.07 4.63758639
18G.s4h3.04 6.40961728
19G.s4h3.05 8.82796429
20G.H3.01 6.19773429
21G.H3.09 4.76831729
22G.H3.13 3.67477425
23G.H3.17 7.39073505
24G.H3.18 5.848184179
25G.S5.03 3.24327548
26G.S5.04 3.19568429
27G.S5.05 3.50136649
28G.S5.07 3.66068449
29G.HG.04 5.68055529
30G.HG.07 4.29527529
31G.HG.15 4.24159427
32G.hgh4.01 4.64523406
33G.hgh4.02 6.10318627
34G.hgh4.05 8.3375427
35G.H4.03 5.19273624
36G.H4.05 4.34841424
37G.H4.10 10.1902426
38G.H4.15 4.09073528
39G.h4s6.02 4.93591428
40G.h4s6.11 4.73409427
41G.S6.02 5.66288647
42G.S6.05 4.11364424
43G.H5.03 4.51382548
44G.H5.08 5.51655548
45G.H5.13 4.91545548
46G.H5.17 4.264554185
47G.H5.23 3.180914114
48G.H5.25 4.339094117
49G.H5.26 2.819095185
50b.1x1 2.40709504
51b.1x11 3.21023408
52b.lhb1x3 3.3425152
53b.lhb1x11 3.24795474
54b.b1x3 4.61682467
55b.b1x4 3.37068467
56b.b1x6 6.01618569
57b.l1x3 8.23569
58b.b2x1 7.130735148
59b.b2x5 5.90697667
60b.b3x2 5.04091465
61b.b3x3 3.361364108
62b.l3x2 4.4625409
63b.b4x3 3.331144107
64b.b4x6 8.27987769
65b.b5x2 5.33591407
66b.b5x3 5.88242669
67b.b5x5 4.20045405
68b.b5x7 5.26341407
69b.l5x1 4.108184108
70b.l5x5 7.07167639
71b.b6x5 4.03182406
72b.l6x5 5.579094164
73b.b7x1 5.777095164
74b.b7x4 2.691095108
75b.l7x2 3.16659439
76b.b8x4 4.855106
77b.l8x5 2.8925193
78b.l9x3 6.82561639
79b.l9x6 4.031641038
80b.b10x5 3.63833609
81b.l10x1 3.46841403
82b.b11x4 5.50045439
83b.l11x2 6.49764539
84b.b12x6 8.18727738
85b.b13x7 7.38564587
86b.l13x3 7.31712689
87b.l13x6 3.68709539
88b.b15x2 6.27114456
89b.l15x2 4.47673589
90b.b16x4 9.78273486
91b.b16x5 4.16709555
92b.b16x6 8.29985688
93b.b17x4 4.52795455
94b.b17x5 5.90045457
95b.b17x7 6.78864458
96b.l17x3 7.54167659
97b.l17x6 5.83673539
98b.b18x3 4.25886458
99b.l18x1 5.971437126
100b.l18x2 6.051594127
101b.b19x2 5.75015656
102b.b19x4 5.74545458
103b.l19x2 6.38704459
104b.b20x4 9.188558
105b.b20x6 6.08255556
106b.b20x7 3.58614409
107b.l20x2 7.06409
108b.b21x1 7.03673557
109b.b21x2 4.21841406
110b.b21x5 5.165494
111b.b21x7 4.88258695
112b.b22x5 5.376735127
113b.l22x5 6.680234159
114b.b23x6 6.85864697
115b.l23x1 7.23454406
116b.b24x4 7.60068496
117b.b24x6 5.66727498
118b.l24x2 4.712054156
119b.l24x3 4.37527505
120b.b25x3 5.35432495
121b.l25x3 7.74836579
122b.l27x1 9.432736149
123b.l27x2 7.05932479
124b.b28x3 4.18773467
125b.b28x4 5.96341476
126b.b28x6 6.82679
127g.h1x1 2.33764502
128g.h1x11 2.81955409
129g.l1x2 3.92432452
130g.l1x4 6.115458
131g.h2x11 7.395914126
132g.ctx3 6.13212679
133g.ctx6 3.54955406
134g.ctx16 4.48104768
135g.ctx17 2.62591407
136Lig 6.414481510
137NT 16.33991016
1381x39 3.735616
1391x40 1.8675403
1401x50 5.205409
141I1x50 7.30754138
1422x38 2.94227
1432x39 3.87841408
1442x40 6.788186139
1452x42 5.49127508
1462x46 4.06159409
1472x50 5.42109509
1482x57 5.08364716
1492x60 5.99568415
1502x61 4.12205415
1512x64 3.06864414
1523x25 9.54891519
1533x28 5.43303616
1543x29 9.22114415
1553x33 6.01545515
1563x43 3.57477409
1573x44 4.09864407
1583x46 4.255684118
1593x49 5.134555229
1603x50 4.874096119
1613x51 4.95773408
162I2x50 3.14341408
1634x41 4.792954225
1644x42 4.6875407
1654x50 3.851144239
166E2 14.41381914
1675x39 7.11121617
1685x48 1.21136404
1695x58 3.359747119
1705x62 6.233184246
1716x44 4.4175419
1726x48 5.94883718
1736x52 5.77955406
1746x55 3.79227416
175E3 5.84327512
1767x31 5.27818413
1777x45 7.24727419
1787x53 4.048915119
179I3 3.47985640
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.l4x2 g.ctx15 16.055411.2545NoNo049
2b.l26x5 g.ctx15 16.40235.03182NoNo059
3b.l26x5 g.ctx4 31.34963.65727NoNo057
4g.ctx3 g.ctx4 31.69254.09818YesNo097
5g.ctx3 g.ctx5 37.99963.57727YesNo799
6b.lhb1x11 g.ctx5 38.50332.82636YesNo749
7b.b28x6 b.lhb1x11 39.4412.74727YesYes794
8b.b27x3 b.b28x6 23.75918.38091NoYes089
9b.b26x3 b.b27x3 72.31493.35091NoNo068
10b.b22x2 b.b26x3 72.2174.09455NoNo086
11b.b22x1 b.b22x2 72.16523.63636NoNo088
12b.b22x1 b.l23x1 72.11532.63091NoYes086
13b.l23x1 b.l25x6 53.993816.2409YesNo068
14b.l25x6 b.l27x1 52.056316.9009NoYes089
15b.b2x1 b.l27x1 51.28095.78818YesYes1489
16b.b2x1 b.l3x1 51.766812.0918YesNo089
17b.l3x1 b.l5x5 51.69625.97545NoYes099
18b.b27x3 b.l25x3 82.717.59273NoYes089
19b.l25x3 b.l27x2 99.68275.38364YesYes799
20b.l25x4 b.l27x2 1004.83727NoYes059
21I1x48 b.l25x4 99.97725.27909NoNo065
22I1x48 I1x51 99.95952.97727NoNo067
232x41 I1x51 99.93952.97091NoNo047
242x41 4x42 99.91924.17545NoYes047
252x42 4x42 76.18276.97182YesYes087
262x42 3x46 72.05393.60273YesYes088
273x46 3x50 24.04094.78364YesYes1189
283x50 G.H5.25 24.04457.06727YesYes1197
29G.H5.20 G.H5.25 22.26663.01909NoYes097
30G.H5.20 G.H5.26 22.48893.65455NoYes095
31G.H5.17 G.H5.26 21.48873.49727YesYes1855
32G.H5.09 I3 10.32243.29273NoYes440
33b.b28x4 b.b28x6 17.57246.01091YesYes769
34b.b28x4 b.l25x3 17.65366.78818YesYes769
35G.H5.17 G.h4s6.12 14.78694.66364YesNo054
36G.S6.02 G.h4s6.12 14.281912.0382YesNo074
37G.H2.04 G.H2.07 28.24014.54545YesYes099
38G.H2.07 b.l7x2 20.91112.79727YesYes399
39b.l5x5 b.l7x2 49.53093.72818YesYes399
40b.l7x2 b.l9x6 27.76712.87636YesYes398
41G.H2.04 G.H3.08 27.66912.76091YesNo099
42G.H3.08 G.S4.04 27.48023.43455NoNo099
43G.H3.09 G.S4.04 27.283114.0318YesNo099
44G.H3.09 G.H4.15 12.09243.21455YesYes298
45g.ctx3 g.ctx6 17.28347.77273YesYes096
46b.l22x5 g.ctx6 16.34033.97545YesYes096
47b.h2x1 b.h2x5 12.25524.15455NoNo055
48b.b21x5 b.h2x1 11.01336.16818YesNo045
49b.b20x5 b.b21x7 24.1635.11364NoYes075
50b.b20x5 b.b21x4 23.9774.65455NoNo075
51b.b20x7 b.b21x4 23.81014.56545YesNo095
52b.b20x7 b.l20x2 23.31673.46364YesYes099
53b.l20x2 g.l1x5 22.53545.69636YesNo094
54g.l1x3 g.l1x5 22.45470.381818NoNo014
55g.l1x2 g.l1x3 22.38210.381818YesNo021
56b.b21x1 g.l1x2 12.06823.18182YesYes572
57b.1x19 b.b21x1 11.27527.58NoYes067
58b.1x15 b.1x19 10.25534.78364NoNo076
59b.b2x5 b.b3x2 10.39288.28273YesYes675
60b.b10x1 b.l9x6 22.57372.54273NoYes098
61b.b10x1 b.b11x5 22.4354.00091NoNo096
62b.b11x5 b.b14x3 11.24074.22818NoNo065
63b.b10x2 b.b14x3 11.79025.19364NoNo065
64b.b10x2 b.b10x4 10.32634.81091NoNo066
65b.b10x4 b.b2x4 10.11838.92636NoNo066
66b.l26x3 b.l26x5 14.64665.54364NoNo075
67b.l26x1 b.l26x3 13.21165.65182NoNo677
68b.b2x5 b.l26x1 12.888810.6982YesNo677
69b.l11x1 b.l9x6 12.49244.87364NoYes398
70b.b11x6 b.l11x1 12.35682.86909NoNo399
71b.b11x6 b.l9x3 10.606814.5818NoYes399
72b.b11x5 b.l13x7 11.58034.70182NoNo069
73b.l13x3 b.l13x7 10.17635.53818YesNo099
74b.b21x7 b.b24x6 24.63874.20818YesYes958
75b.b23x6 b.b24x6 24.31347.63YesYes978
76b.l21x7 b.l23x1 27.37095.79909NoYes056
77b.l21x7 b.l23x2 27.066.50636NoNo058
78b.b23x6 b.l23x2 26.33054.70455YesNo078
792x46 3x46 26.38982.59273YesYes098
802x46 3x43 20.6133.52273YesYes099
813x43 6x44 44.19213.21273YesYes099
826x44 6x48 42.72547.28909YesYes198
836x48 Lig 38.3044.08YesYes180
843x46 7x53 24.19026.04364YesYes1189
853x43 7x53 25.09013.94364YesYes099
864x42 4x46 18.66073.16182YesNo077
872x45 4x46 18.37394.76273NoNo097
882x45 4x50 18.44576.48182NoYes099
893x38 4x50 17.78114.00727NoYes2379
903x38 4x53 17.64922.81273NoNo078
913x37 4x53 17.06052.72NoNo068
923x37 Lig 16.98084.79182NoYes060
933x32 Lig 10.59524.19091NoYes160
94E2 Lig 13.33535.79727YesYes140
957x38 Lig 10.59727.31909NoYes050
962x57 3x32 10.16365.22364YesNo166
972x57 7x38 10.13725.35818YesNo065
981x39 2x57 11.05733.26455YesYes166
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
LigNT7.053641YesYes0601
2x60Lig7.414551YesYes5010
2x64Lig4.657271YesYes4010
3x29Lig7.652731YesYes5010
3x32Lig4.190911NoYes6010
3x33Lig16.19451YesYes5010
3x36Lig8.840911NoYes6010
3x37Lig4.791820NoYes6010
E2Lig5.797271YesYes4010
5x47Lig5.410911NoYes7010
6x48Lig4.081YesYes8010
6x51Lig5.121821NoYes6010
6x55Lig5.051821YesYes6010
7x38Lig7.319090NoYes5010
NTNT29.38821YesYes6611
3x22NT5.344551NoYes3621
3x25NT4.991YesYes9621
E2NT61.46641YesYes4611
E1x50NT3.325451NoYes5621
E1x501NT14.01091NoYes5621
E3NT6.177271YesYes2621
2x573x325.223641YesNo6621
2x577x385.358181YesNo6521
2x602x642.573641YesYes5411
2x603x288.767271YesYes5612
2x603x325.227271YesNo5611
2x643x283.355451YesYes4612
E1x50E1x5014.825451NoNo5522
3x28E1x504.114551YesNo6522
3x253x287.272731YesYes9622
3x253x2913.87821YesYes9521
3x25E217.86821YesYes9421
3x26E219.20271NoYes6421
3x283x294.548181YesYes6521
3x29E210.80551YesYes5411
3x33E23.624551YesYes5411
3x335x396.377271YesYes5712
3x335x432.921YesNo5611
3x366x484.761821NoYes6811
3x374x532.720NoNo6812
3x406x484.108180NoYes7821
4x594x602.984551NoNo5522
4x59E24.761821NoYes5421
4x595x393.941821NoYes5722
4x60E29.754551NoYes5421
4x605x3914.03641NoYes5722
5x36E210.27641NoYes4421
5x38E25.611821NoYes4421
5x39E29.401821YesYes7421
E2E242.82731YesYes4411
5x37E22.586361NoYes3421
5x40E22.780911NoYes6421
6x58E213.18551NoYes4421
7x31E27.625451YesYes3421
5x365x389.624551NoNo4422
5x395x436.353641YesNo7621
5x406x553.431NoYes6621
5x446x523.857270NoYes5622
5x446x552.695450NoYes5621
5x476x489.110911NoYes7811
5x476x5212.56821NoYes7612
6x446x487.289091YesYes9821
6x447x453.515451YesYes9922
6x487x4510.171YesYes8912
6x516x553.991821NoYes6611
6x587x316.908181NoYes4322
E3E34.937271YesYes2222
7x31E33.683641YesYes3222
3x253x263.735451YesNo9622
5x43Lig2.641NoYes6010
7x32NT2.254551NoYes1621
6x487x412.121821YesNo8712
7x34E21.967270NoYes4421
2x64E1x471.688181YesNo4412
4x63E21.490910NoYes5421
2x533x361.292730NoNo8621
3x303x330.9609090NoYes6521

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
93.75Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
93.75Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
93.33Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
93.33Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
83.33Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
76.47Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
76.47Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
75.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
73.33Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
70.59Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
70.59Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
68.75Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
68.42Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
64.71Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
64.71Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
64.71Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
64.71Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
63.16Single5ZTYAM102575ZTY-CB2-AM10257
63.16Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
62.50Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
62.50Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
61.11Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
61.11Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
61.11Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
61.11Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
61.11Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
61.11Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
61.11Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
60.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
60.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
60.00Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
60.00Consensuslpl_onOrthosteric Ligands1p_on lpa_on
60.00Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
58.82Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
57.89Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
57.89Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
57.89Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
57.14Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
56.25Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
55.56Single8E0GBU728E0G-μ-BU72
55.56Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
55.56Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
54.55Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
52.94Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
52.94Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
52.94Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
52.94Single9CHXS-Carazolol9CHX-β2-S-Carazolol
52.94Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
52.63Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
52.63Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
52.63Single7YITNalfurafine7YIT-κ-Nalfurafine
52.63Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
52.63Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
52.63Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
52.63Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
52.63Consensuslpa_offOrthosteric Ligandlpa1_off
52.63Consensuslpl_offOrthosteric Ligands1p_off lpa_off
52.17Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
50.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
50.00Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
50.00Single5C1MBU725C1M-μ-BU72
50.00Single5X93K-87945X93-ETB-K-8794
50.00Single6AKXA4R6AKX-CCR5-A4R
50.00Single6B73MP11046B73-κ-MP1104
50.00Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
50.00Single7C4SS1P7C4S-S1P3-S1P
50.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
50.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
50.00Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
50.00Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
50.00Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
50.00Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
50.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
50.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
50.00Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
50.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
50.00Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
50.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
50.00Single8TF5Oleic acid8TF5-GPR6-Oleic acid
50.00Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
50.00Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
50.00Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
50.00Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
50.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
50.00Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
50.00Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
50.00Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
50.00Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
50.00Consensusendothelin_offOrthosteric Ligandetb_off
50.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
50.00Consensusorexin_offOrthosteric Ligandox2_off ox1_off
50.00Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
50.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
48.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
47.83Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
47.83Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
47.62Single4UG2CGS216804UG2-A2A-CGS21680
47.62Single7SK9CCX6627SK9-ACKR3-CCX662
47.62Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
47.62Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
47.62Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
47.62Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
47.62Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
47.62Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
47.37Single2YDVNECA2YDV-A2A-NECA
47.37Single4DJHJDTic4DJH-κ-JDTic
47.37Single4UHRCGS216804UHR-A2A-CGS21680
47.37Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
47.37Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
47.37Single5G53NECA5G53-A2A-NECA-Gs
47.37Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
47.37Single6TQ7SB-3348676TQ7-OX1-SB-334867
47.37Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
47.37Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
47.37Single7FEECP559407FEE-CB1-CP55940-ZCZ011
47.37Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
47.37Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
47.37Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
47.37Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
47.37Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
47.37Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
47.37Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
47.37Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
47.37Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
47.37Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
47.37Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
47.37Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
47.37Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
47.37Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
47.37Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
47.37Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
47.37Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
47.37Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
47.37Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
47.06Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
47.06Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
47.06Single4MBSMaraviroc4MBS-CCR5-Maraviroc
47.06Single4ZJCSB-6740424ZJC-OX1-SB-674042
47.06Single6TPGEMPA6TPG-OX2-EMPA
47.06Single6TPNHTL66416TPN-OX2-HTL6641
47.06Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
47.06Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
47.06Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
47.06Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
47.06Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
47.06Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
47.06Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
47.06Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
47.06Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
47.06Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
47.06Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
47.06Consensusalpha1_onOrthosteric Ligandalpha1a_on
47.06Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
47.06Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
47.06Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
46.15Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
46.15Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
46.15Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
46.15Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
45.83Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
45.45Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
45.45Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
45.45Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
45.45Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
45.45Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
45.45Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
45.00Single3D4STimolol3D4S-β2-Timolol
45.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
45.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
45.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
45.00Single6KQICP559406KQI-CB1-CP55940-Org27569
45.00Single6ZG4HTL00099366ZG4-M1-HTL0009936
45.00Single7DFPSpiperone7DFP-D2-Spiperone
45.00Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
45.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
45.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
45.00Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
45.00Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
45.00Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
45.00Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
45.00Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
45.00Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
45.00Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
45.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
45.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
45.00Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
45.00Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
45.00Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
45.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
45.00Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
45.00Consensusorexin_onOrthosteric Ligandox2_on
44.44Single3NY8ICI118-5513NY8-β2-ICI118-551
44.44Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
44.44Single4EJ4Naltrindole4EJ4-δ-Naltrindole
44.44Single4GBRS-Carazolol4GBR-β2-S-Carazolol
44.44Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
44.44Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
44.44Single6TOTLemborexant6TOT-OX1-Lemborexant
44.44Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
44.44Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
44.44Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
44.44Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
44.44Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
44.44Single7UL4Alvimopan7UL4-μ-Alvimopan
44.44Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
44.44Single7V3ZCP559407V3Z-CB1-CP55940
44.44Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
44.44Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
44.44Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
44.44Single8T1WCVN4248T1W-GPR6-CVN424
44.44Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
44.44Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
44.44Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
44.44Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
44.44Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
44.44Consensus5ht5_onOrthosteric Ligand5ht5a_on
44.44Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
44.44Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
44.44Consensusalpha2_onOrthosteric Ligandalpha2b_on
44.44Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
44.44Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
44.44Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
44.44Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
44.44Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
44.44Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
44.44Consensusblt_onOrthosteric Ligandblt1_on
44.44Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
44.44Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
44.44Consensusdopamine_offOrthosteric Ligandd2_off d3_off
44.44Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
44.44Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
44.44Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
44.44Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
44.44Consensusleukotriene_onOrthosteric Ligandblt_on
44.44Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
44.00Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
44.00Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
43.75Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
43.75Single7SRQLSD7SRQ-5-HT2B-LSD
43.75Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
43.75Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
43.75Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
43.75Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
43.75Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
43.75Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
42.86Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
42.86Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
42.86Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
42.86Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
42.86Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
42.86Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
42.86Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
42.86Single7UM4AS26747237UM4-5-HT5A-AS2674723
42.86Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
42.86Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
42.86Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
42.86Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
42.86Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.86Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
42.86Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
42.86Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
42.86Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
42.86Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.86Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
42.86Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
42.86Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
42.86Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
42.86Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
42.31Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
42.11Single2RH1S-Carazolol2RH1-β2-S-Carazolol
42.11Single2YCWS-Carazolol2YCW-β1-S-Carazolol
42.11Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
42.11Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
42.11Single5D6LS-Carazolol5D6L-β2-S-Carazolol
42.11Single5WQCEMPA5WQC-OX2-EMPA
42.11Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
42.11Single5XPRBosentan5XPR-ETB-Bosentan
42.11Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
42.11Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
42.11Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
42.11Single6TP6Filorexant6TP6-OX1-Filorexant
42.11Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
42.11Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
42.11Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
42.11Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
42.11Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
42.11Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
42.11Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.11Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
42.11Single8JXSPF-61428JXS-D1-PF-6142
42.11Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
42.11Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
42.11Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
42.11Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
42.11Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
42.11Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
42.11Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
42.11Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
42.11Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
42.11Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
42.11Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
42.11Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
42.11Consensusamine_offonOrthosteric Ligandamine_off amine_on
42.11Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
42.11Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
42.11Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
42.11Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
42.11Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
42.11Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
42.11Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
42.11Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
42.11Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
42.11Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
42.11Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
42.11Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
42.11Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
42.11Consensustrace-amine_onOrthosteric Ligandta1_on
41.67Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
41.67Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.67Consensusangiotensin_onOrthosteric Ligandat1_on
41.67Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
41.67Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
41.67Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
41.18Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
41.18Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
41.18Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
41.18Single5WS3EMPA5WS3-OX2-EMPA
41.18Single6AKYMaraviroc6AKY-CCR5-Maraviroc
41.18Single6TODEMPA6TOD-OX1-EMPA-Na
41.18Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
41.18Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
41.18Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
41.18Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
41.18Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
41.18Single7XRRLemborexant7XRR-OX2-Lemborexant
41.18Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
41.18Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
41.18Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
41.18Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
41.18Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
41.18Single8Y0HVUF114188Y0H-CXCR3-VUF11418
41.18Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
41.18Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
41.18Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
41.18Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
41.18Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
41.18Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
41.18Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
41.18Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
40.91Single3NY9ICI118-5513NY9-β2-ICI118-551
40.91Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
40.91Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
40.91Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
40.91Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
40.91Single8QJ2pN1628QJ2-MC4-pN162-Gs
40.91Single8X5YAstemizole8X5Y-H1-Astemizole
40.91Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
40.74Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
40.74Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
40.00Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
40.00Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
40.00Single4U15Tiotropium4U15-M3-Tiotropium
40.00Single5D5AS-Carazolol5D5A-β2-S-Carazolol
40.00Single5D5BS-Carazolol5D5B-β2-S-Carazolol
40.00Single5XR8AM8415XR8-CB1-AM841
40.00Single5XRAAM115425XRA-CB1-AM11542
40.00Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
40.00Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
40.00Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
40.00Single6H7JIsoprenaline6H7J-β1-Isoprenaline
40.00Single6J21Aprepitant6J21-NK1-Aprepitant
40.00Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
40.00Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
40.00Single6OL9Tiotropium6OL9-M5-Tiotropium
40.00Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
40.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
40.00Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
40.00Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
40.00Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
40.00Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
40.00Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
40.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
40.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
40.00Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
40.00Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
40.00Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
40.00Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
40.00Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
40.00Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
40.00Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
40.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
40.00Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
40.00Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
40.00Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
40.00Single8XVLZibotentan8XVL-ETA-Zibotentan
40.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
40.00Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
40.00Consensusa2_onOrthosteric Liganda2b_on
40.00Consensusa2_on_gpOrthosteric Liganda2b_on_gp
40.00Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
40.00Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
40.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
40.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
40.00Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
40.00Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
40.00Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
40.00Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
40.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
40.00Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
40.00Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
40.00Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
40.00Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
40.00Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
40.00Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
40.00Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
39.29Single6IGLIRL16206IGL-ETB-IRL1620
39.13Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
39.13Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
39.13Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
39.13Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
39.13Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
39.13Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
39.13Single8WDTphotoNECA8WDT-A2A-photoNECA
39.13Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
39.13Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
38.89Single2YDOAdenosine2YDO-A2A-Adenosine
38.89Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
38.89Single3RZECidoxepin3RZE-H1-Cidoxepin
38.89Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
38.89Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
38.89Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
38.89Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
38.89Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
38.89Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
38.89Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
38.89Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
38.89Single6PS0S-Carazolol6PS0-β2-S-Carazolol
38.89Single6PS4ICI118-5516PS4-β2-ICI118-551
38.89Single6PS5S-Propranolol6PS5-β2-S-Propranolol
38.89Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
38.89Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
38.89Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
38.89Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
38.89Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
38.89Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
38.89Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
38.89Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
38.89Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
38.89Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
38.89Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
38.89Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.89Single7UL3Famotidine7UL3-H2-Famotidine
38.89Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
38.89Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
38.89Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
38.89Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
38.89Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
38.89Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
38.89Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.89Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
38.89Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
38.89Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
38.89Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
38.89Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
38.89Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
38.89Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
38.89Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
38.89Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
38.89Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
38.89Single8K5CAcipimox8K5C-HCA2-Acipimox
38.89Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
38.89Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.89Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
38.89Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.89Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.89Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.89Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
38.89Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
38.89Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
38.89Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.89Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
38.89Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
38.89Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
38.89Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
38.89Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
38.89Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
38.89Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
38.89Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
38.89Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
38.89Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
38.89Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
38.89Consensushca_onOrthosteric Ligandhca2_on
38.89Consensusopsins_offOrthosteric Ligandrhodopsin_off
38.89Consensussensory_offOrthosteric Ligandopsins_off
38.46Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
38.46Single8ZRTET-18ZRT-ETB-ET-1
38.46Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
38.46Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
38.10Single4AMIBucindolol4AMI-β1-Bucindolol
38.10Single4LDEBI1671074LDE-β2-BI167107
38.10Single4RWADIPP-NH24RWA-δ-DIPP-NH2
38.10Single5CXVTiotropium5CXV-M1-Tiotropium
38.10Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
38.10Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
38.10Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
38.10Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
38.10Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
38.10Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
38.10Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
38.10Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
38.10Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
38.10Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
38.10Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.10Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
38.10Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
38.10Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
38.10Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
38.10Single8JWY2-1188JWY-A2A-2-118
38.10Single8JWZAB9288JWZ-A2A-AB928-Na
38.10Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
38.10Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.10Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
38.10Single8XYIVUF106618XYI-CXCR3-VUF10661
38.10Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
38.10Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
38.10Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
38.10Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
38.10Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
38.10Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
37.93Single5GLHEndothelin-15GLH-ETB-Endothelin-1
37.93Single6IGKEndothelin-36IGK-ETB-Endothelin-3
37.93Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
37.93Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
37.93Consensusbombesin_onOrthosteric Ligandbb2_on
37.93Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
37.93Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
37.50Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
37.50Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
37.50Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
37.50Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
37.50Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
37.50Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
37.50Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
37.50Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
37.50Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
37.50Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
37.50Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
37.50Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
37.50Consensus5ht2_onOrthosteric Ligand5ht2b_on
37.50Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.50Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
37.50Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
37.50Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
37.50Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
37.50Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
37.04Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
36.84Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
36.84Single2Y04Salbutamol2Y04-β1-Salbutamol
36.84Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
36.84Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
36.84Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
36.84Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
36.84Single4MQSIperoxo4MQS-M2-Iperoxo
36.84Single4U14Tiotropium4U14-M3-Tiotropium
36.84Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
36.84Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
36.84Single5TGZAM65385TGZ-CB1-AM6538
36.84Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
36.84Single6DRXLisuride6DRX-5-HT2B-Lisuride
36.84Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
36.84Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
36.84Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
36.84Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
36.84Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
36.84Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
36.84Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
36.84Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
36.84Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
36.84Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
36.84Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
36.84Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
36.84Single7WC7Lisuride7WC7-5-HT2A-Lisuride
36.84Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
36.84Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
36.84Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
36.84Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
36.84Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
36.84Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
36.84Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
36.84Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
36.84Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
36.84Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
36.84Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
36.84Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
36.84Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
36.84Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
36.84Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
36.84Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
36.84Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
36.84Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
36.84Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
36.84Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
36.84Single8JJOAlprenolol8JJO-β2-Alprenolol
36.84Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
36.84Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
36.84Single8JXRLSD8JXR-D1-LSD
36.84Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
36.84Single8RLNLUF58348RLN-A2A-LUF5834
36.84Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.84Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
36.84Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
36.84Single8X63Mepyramine8X63-H1-Mepyramine
36.84Single8X64Desloratadine8X64-H1-Desloratadine
36.84Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
36.84Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
36.84Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
36.84Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
36.84Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
36.84Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
36.84Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
36.84Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
36.84Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
36.84Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
36.84Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
36.84Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
36.84Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
36.84Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
36.84Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
36.84Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
36.84Consensushca_on_gpOrthosteric Ligandhca2_on_gp
36.84Consensushistamine_offOrthosteric Ligandh1_off
36.84Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
36.84Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
36.67Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
36.67Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
36.36Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
36.36Single6K1QIRL25006K1Q-ETB-IRL2500
36.36Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
36.36Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
36.36Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
36.36Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
36.36Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
36.36Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
36.00Single5WF5UK-4320975WF5-A2A-UK-432097
36.00Single6PT2KGCHM076PT2-δ-KGCHM07
36.00Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
36.00Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
36.00Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.00Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
36.00Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
36.00Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
35.71Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
35.71Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
35.48Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
35.48Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
35.29Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
35.29Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
35.29Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
35.29Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
35.29Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
35.29Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
35.29Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
35.29Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
35.29Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
35.29Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
35.29Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
35.29Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
35.29Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
35.29Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
35.29Single8K5BNiacin8K5B-HCA2-Niacin
35.29Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
35.29Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
35.29Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.29Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
35.29Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
35.29Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
35.29Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
35.00Single2Y03Isoprenaline2Y03-β1-Isoprenaline
35.00Single5JQHS-Carazolol5JQH-β2-S-Carazolol
35.00Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
35.00Single5TVNLSD5TVN-5-HT2B-LSD
35.00Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
35.00Single6E67BI1671076E67-β2-BI167107-Gs (fused)
35.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
35.00Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
35.00Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
35.00Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
35.00Single6PS6Timolol6PS6-β2-Timolol
35.00Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
35.00Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
35.00Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
35.00Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
35.00Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
35.00Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
35.00Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
35.00Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
35.00Single7W41PD1762527W41-BB2-PD176252
35.00Single7WC6LSD7WC6-5-HT2A-LSD
35.00Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.00Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
35.00Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
35.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
35.00Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.00Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
35.00Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
35.00Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
35.00Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.00Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
35.00Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
35.00Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
35.00Single8S4DCMF-0198S4D-Apelin-CMF-019
35.00Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.00Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
35.00Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
35.00Consensusa3_on_gpOrthosteric Liganda3a_on_gp
35.00Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
35.00Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
35.00Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
35.00Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
35.00Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
35.00Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
35.00Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
35.00Consensusbombesin_offOrthosteric Ligandbb2_off
35.00Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.00Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.00Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
34.78Single6PT3DPI-2876PT3-δ-DPI-287
34.78Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
34.78Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
34.78Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
34.78Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
34.78Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
34.78Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
34.62Single6JODAngiotensin II6JOD-AT2-Angiotensin II
34.62Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
34.62Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
34.62Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
34.62Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
34.62Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
34.62Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
34.62Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
34.62Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
34.62Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
34.62Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
34.62Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
34.62Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
34.62Consensusvasop-oxy_onOrthosteric Ligandv2_on
34.62Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
34.48Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
34.48Consensusendothelin_onOrthosteric Ligandetb_on eta_on
34.48Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
33.33Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
33.33Single3P0GBI1671073P0G-β2-BI167107
33.33Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
33.33Single4IARErgotamine4IAR-5-HT1B-Ergotamine
33.33Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
33.33Single4S0VSuvorexant4S0V-OX2-Suvorexant
33.33Single4XT1Fractalkine4XT1-US28-Fractalkine
33.33Single5V54Methiothepin5V54-5-HT1B-Methiothepin
33.33Single6E59L-7607356E59-NK1-L-760735
33.33Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
33.33Single6J20Aprepitant6J20-NK1-Aprepitant
33.33Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
33.33Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
33.33Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
33.33Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
33.33Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
33.33Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
33.33Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
33.33Single6TPJSuvorexant6TPJ-OX2-Suvorexant
33.33Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
33.33Single6WGTLSD6WGT-5-HT2A-LSD
33.33Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
33.33Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
33.33Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
33.33Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
33.33Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
33.33Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
33.33Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
33.33Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
33.33Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
33.33Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
33.33Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
33.33Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
33.33Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
33.33Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
33.33Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
33.33Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
33.33Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
33.33Single7TUYGSK682753A7TUY-GPR183-GSK682753A
33.33Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
33.33Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
33.33Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
33.33Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
33.33Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
33.33Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
33.33Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
33.33Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
33.33Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
33.33Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
33.33Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
33.33Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
33.33Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
33.33Single8EA0Iperoxo8EA0-M3-Iperoxo
33.33Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
33.33Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
33.33Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
33.33Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
33.33Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
33.33Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
33.33Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
33.33Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
33.33Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
33.33Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
33.33Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
33.33Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
33.33Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
33.33Single8IEBA1LYA8IEB-GPR156-A1LYA
33.33Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
33.33Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
33.33Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
33.33Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
33.33Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
33.33Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
33.33Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
33.33Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
33.33Single8WKYPG-9348WKY-MC4-PG-934
33.33Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
33.33Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
33.33Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
33.33Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
33.33Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
33.33Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
33.33Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
33.33Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
33.33Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
33.33Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
33.33Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
33.33Consensus5ht1_offOrthosteric Ligand5ht1b_off
33.33Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
33.33Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
33.33Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
33.33Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
33.33Consensusalpha2_offOrthosteric Ligandalpha2c_off
33.33Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
33.33Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
33.33Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
33.33Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
33.33Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
33.33Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
33.33Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
33.33Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
33.33Consensuslpa_onOrthosteric Ligandlpa1_on
33.33Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
33.33Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
33.33Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
33.33Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
33.33Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
33.33Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
33.33Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
33.33Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
33.33Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
33.33Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
33.33Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
32.35Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
32.35Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
32.26Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
32.14Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
32.14Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
32.14Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
32.14Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
32.00Single3QAKUK-4320973QAK-A2A-UK-432097
32.00Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
32.00Single6HLOAprepitant6HLO-NK1-Aprepitant
32.00Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
32.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
32.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
32.00Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
32.00Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
32.00Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
32.00Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
32.00Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
32.00Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
32.00Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
32.00Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
32.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
32.00Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
32.00Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
31.82Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
31.82Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
31.82Single6A93Risperidone6A93-5-HT2A-Risperidone
31.82Single6CM4Risperidone6CM4-D2-Risperidone
31.82Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
31.82Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
31.82Single6MXTSalmeterol6MXT-β2-Salmeterol
31.82Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
31.82Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
31.82Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
31.82Single7K15MKD0467K15-BLT1-MKD046-Na
31.82Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
31.82Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
31.82Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
31.82Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
31.82Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
31.82Single8JJ8Formoterol8JJ8-β2-Formoterol
31.82Single8JJLOlodaterol8JJL-β2-Olodaterol
31.82Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
31.82Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
31.82Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
31.82Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
31.82Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
31.82Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
31.82Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
31.82Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
31.82Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
31.82Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
31.82Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
31.82Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
31.82Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
31.58Single6A94Zotepine6A94-5-HT2A-Zotepine
31.58Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
31.58Single6IQLL7458706IQL-D4-L745870
31.58Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
31.58Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
31.58Single6TP3Nemorexant6TP3-OX1-Nemorexant
31.58Single6TPKRetosiban6TPK-OT-Retosiban
31.58Single6V9SGTPL114036V9S-OX1-GTPL11403
31.58Single6VI4JDTic6VI4-κ-JDTic
31.58Single6ZG9GSK10347026ZG9-M1-GSK1034702
31.58Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
31.58Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
31.58Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
31.58Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
31.58Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
31.58Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.58Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
31.58Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.58Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
31.58Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
31.58Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
31.58Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single8IHKAcifran8IHK-HCA3-Acifran
31.58Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
31.58Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
31.58Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
31.58Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
31.58Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
31.58Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
31.58Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
31.58Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.58Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
31.58Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
31.58Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
31.58Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
31.58Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
31.58Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
31.58Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
31.58Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
31.58Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
31.58Single9BJKNaloxone9BJK-μ-Naloxone-NAM
31.58Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
31.58Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
31.58Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
31.58Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
31.58Consensusvasop-oxy_offOrthosteric Ligandot_off
31.43Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
31.25Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
31.25Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
31.25Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
31.25Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
31.25Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
31.25Single9CHUNoradrenaline9CHU-β2-Noradrenaline
31.25Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
31.25Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
31.03Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
31.03Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
31.03Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
31.03Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
31.03Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
31.03Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
30.77Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
30.77Single6W25SHU91196W25-MC4-SHU9119-Ca
30.77Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
30.77Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
30.77Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
30.77Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
30.77Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
30.77Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
30.77Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
30.43Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
30.43Single6H7LDobutamine6H7L-β1-Dobutamine
30.43Single6IBLArformoterol6IBL-β1-Arformoterol
30.43Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
30.43Single7EZCUKA7EZC-A2A-UKA
30.43Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
30.43Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.43Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
30.43Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
30.43Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
30.43Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
30.43Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.43Single8XVJMacitentan8XVJ-ETA-Macitentan
30.43Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
30.43Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
30.43Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
30.43Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
30.43Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
30.43Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Consensusprostanoid_offOrthosteric Ligandep_off dp_off
30.30Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
30.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
30.00Single2Y02Carmoterol2Y02-β1-Carmoterol
30.00Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
30.00Single4DAJTiotropium4DAJ-M3-Tiotropium
30.00Single4QKX35V4QKX-β2-35V
30.00Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
30.00Single4YAYZD-71554YAY-AT1-ZD-7155
30.00Single5DHGC-355DHG-NOP-C-35
30.00Single5DHHSB-6121115DHH-NOP-SB-612111
30.00Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
30.00Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
30.00Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
30.00Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
30.00Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
30.00Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
30.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
30.00Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
30.00Single6H7MSalbutamol6H7M-β1-Salbutamol
30.00Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
30.00Single6PS1Timolol6PS1-β2-Timolol
30.00Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.00Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
30.00Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
30.00Single7BU7BI1671077BU7-β1-BI167107
30.00Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
30.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
30.00Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
30.00Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
30.00Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
30.00Single8CU6LJ-45178CU6-A2A-LJ-4517
30.00Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
30.00Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
30.00Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
30.00Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
30.00Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
30.00Single8IY6Endothelin-18IY6-ETB-Endothelin-1
30.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
30.00Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
30.00Single8K5DGSK2560738K5D-HCA2-GSK256073
30.00Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
30.00Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
30.00Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
30.00Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.00Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
30.00Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
30.00Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
30.00Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
30.00Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
30.00Single9IYAONO-97105319IYA-GPR55-ONO-9710531
30.00Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
30.00Consensusa3_onOrthosteric Liganda3a_on
30.00Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
30.00Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
30.00Consensusbradykinin_onOrthosteric Ligandbk2_on
30.00Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
30.00Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
30.00Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
30.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
30.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
29.63Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
29.63Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
29.63Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
29.63Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
29.63Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
29.63Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
29.63Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
29.63Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
29.63Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
29.63Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
29.41Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
29.41Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
29.41Single3OE6IT1t3OE6-CXCR4-IT1t
29.41Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
29.41Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
29.41Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
29.41Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
29.41Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
29.41Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
29.41Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
29.41Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
29.41Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
29.41Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
29.41Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
29.41Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
29.41Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
29.41Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
29.41Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
29.41Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
29.41Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
29.41Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
29.17Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
29.17Single5WF6UK-4320975WF6-A2A-UK-432097
29.17Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
29.17Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
29.17Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
29.17Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
29.17Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
29.17Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
29.17Single8IEIA1LYA8IEI-GPR156-A1LYA
29.17Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
29.17Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
29.17Consensuskisspeptin_onOrthosteric Ligandkiss1_on
29.03Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
29.03Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
29.03Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
29.03Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
29.03Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
29.03Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
28.57Single5N2RPSB-365N2R-A2A-PSB-36-Na
28.57Single5N2SPSB365N2S-A1-PSB36
28.57Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
28.57Single5WIUNemonapride5WIU-D4-Nemonapride
28.57Single5WIVNemonapride5WIV-D4-Nemonapride-Na
28.57Single6D26Fevipiprant6D26-DP2-Fevipiprant
28.57Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
28.57Single6HLPNetupitant6HLP-NK1-Netupitant
28.57Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
28.57Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
28.57Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
28.57Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
28.57Single7C61Ergotamine7C61-5-HT1B-Ergotamine
28.57Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
28.57Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
28.57Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
28.57Single7SINNPS-21437SIN-CaS-NPS-2143
28.57Single7SINNPS-21437SIN-CaS-NPS-2143
28.57Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
28.57Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
28.57Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
28.57Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
28.57Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
28.57Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
28.57Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
28.57Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
28.57Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
28.57Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
28.57Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
28.57Single8ZMFA1L108ZMF-5-HT2C-A1L10
28.57Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
28.57Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
28.57Consensusadenosine_offOrthosteric Liganda1_off a2_off
28.57Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
28.57Consensusblt_offOrthosteric Ligandblt1_off
28.57Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
28.57Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
28.57Consensusdp_offOrthosteric Liganddp2_off
28.57Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
28.57Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
28.57Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
28.57Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
28.57Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
28.57Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
28.12Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
28.12Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
28.12Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
28.00Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
28.00Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
28.00Single7QA8Peptide7QA8-STE2-Peptide
28.00Single7QA8Peptide7QA8-STE2-Peptide
28.00Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
28.00Single8IEIA1LYA8IEI-GPR156-A1LYA
28.00Single8IEPA1LYA8IEP-GPR156-A1LYA
28.00Single8IEPA1LYA8IEP-GPR156-A1LYA
28.00Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
28.00Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
28.00Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
28.00Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
28.00Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
28.00Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.00Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.00Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
28.00Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
28.00Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
28.00Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
27.78Single3OE9IT1t3OE9-CXCR4-IT1t
27.78Single3PBLEticlopride3PBL-D3-Eticlopride
27.78Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
27.78Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
27.78Single6HLLCP999946HLL-NK1-CP99994
27.78Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
27.78Single6TP4ACT-4622066TP4-OX1-ACT-462206
27.78Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
27.78Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
27.78Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
27.78Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
27.78Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
27.78Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
27.78Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
27.78Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.78Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
27.78Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
27.78Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
27.78Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
27.78Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
27.78Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
27.78Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
27.78Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
27.78Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.78Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
27.78Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
27.78Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
27.78Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
27.78Single9B9Y7DY9B9Y-CB1-7DY
27.78Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
27.78Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
27.78Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
27.78Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
27.78Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
27.78Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
27.59Single4XT3Fractalkine4XT3-US28-Fractalkine
27.59Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
27.59Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
27.59Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
27.59Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
27.59Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
27.59Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
27.59Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
27.59Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
27.59Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
27.59Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
27.50Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
27.27Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
27.27Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
27.27Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
27.27Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
27.27Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
27.27Single7B6WCyclazosin7B6W-α1b-Cyclazosin
27.27Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
27.27Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
27.27Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
27.27Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
27.27Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
27.27Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
27.27Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
27.27Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
27.27Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
27.27Consensustachykinin_offOrthosteric Ligandnk1_off
26.92Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
26.92Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
26.92Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
26.92Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
26.92Single8IEBA1LYA8IEB-GPR156-A1LYA
26.92Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
26.92Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
26.92Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
26.92Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
26.92Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
26.67Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
26.67Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
26.67Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
26.67Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
26.67Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
26.67Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
26.67Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
26.47Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
26.47Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
26.32Single3ODUIT1t3ODU-CXCR4-IT1t
26.32Single3PWHZM-2413853PWH-A2A-ZM-241385
26.32Single5ZKQABT-4915ZKQ-PAF-ABT-491
26.32Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
26.32Single6DS0Ly2660976DS0-5-HT2B-Ly266097
26.32Single6ME2Ramelteon6ME2-MT1-Ramelteon
26.32Single6ME9Ramelteon6ME9-MT2-Ramelteon
26.32Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
26.32Single7BR3Elagolix7BR3-GnRH1-Elagolix
26.32Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
26.32Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
26.32Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
26.32Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.32Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
26.32Single8GNGIstradefylline8GNG-A2A-Istradefylline
26.32Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
26.32Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
26.32Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
26.32Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
26.32Single8IWESpermidine8IWE-TA9-Spermidine
26.32Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
26.32Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
26.32Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
26.32Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
26.32Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
26.32Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
26.32Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
26.32Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
26.09Single4N4WSANT-14N4W-SMO-SANT-1
26.09Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
26.09Single5X33BIIL2605X33-BLT1-BIIL260
26.09Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
26.09Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
26.09Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
26.09Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
26.09Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.09Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
26.09Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
26.09Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
26.09Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
26.09Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.09Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.93Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
25.93Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
25.93Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
25.93Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
25.93Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
25.81Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
25.81Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
25.81Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
25.81Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
25.81Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
25.81Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
25.81Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
25.00Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
25.00Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
25.00Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
25.00Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
25.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
25.00Single5JTBZM-2413855JTB-A2A-ZM-241385
25.00Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
25.00Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
25.00Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
25.00Single6AQFZM-2413856AQF-A2A-ZM-241385
25.00Single6KUXRS-799486KUX-α2a-RS-79948
25.00Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
25.00Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
25.00Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
25.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
25.00Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
25.00Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
25.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
25.00Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
25.00Single7AROLUF58337ARO-A2A-LUF5833-Na
25.00Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
25.00Single7T32ZM-2413857T32-A2A-ZM-241385
25.00Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
25.00Single7VODCariprazine7VOD-5-HT2A-Cariprazine
25.00Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
25.00Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
25.00Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
25.00Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
25.00Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8PWNTheophylline8PWN-A2A-Theophylline
25.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
25.00Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
25.00Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
25.00Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
25.00Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
25.00Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
25.00Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
25.00Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
25.00Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
25.00Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
25.00Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
25.00Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
25.00Consensusa2_offOrthosteric Liganda2a_off
25.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
25.00Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
25.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
25.00Consensuscck_onOrthosteric Ligandccka_on cckb_on
25.00Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
25.00Consensuschemerin_onOrthosteric Ligandcml1_on
25.00Consensusgrh_offOrthosteric Ligandgnrh1_off
25.00Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
25.00Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
25.00Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
25.00Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
25.00Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
25.00Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
24.24Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
24.24Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
24.24Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
24.14Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
24.14Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
24.14Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
24.14Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
24.14Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
24.14Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
24.14Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
24.14Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.14Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
24.14Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
24.14Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
24.14Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
24.14Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
24.14Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
24.00Single5EE7MK08935EE7-Glucagon-MK0893
24.00Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
24.00Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
24.00Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
24.00Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.00Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
24.00Single7XN9L-054,5227XN9-SST2-L-054,522
24.00Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
24.00Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
24.00Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
24.00Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
23.81Single2Y01Dobutamine2Y01-β1-Dobutamine
23.81Single3EMLZM-2413853EML-A2A-ZM-241385
23.81Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
23.81Single5DSGTiotropium5DSG-M4-Tiotropium
23.81Single5IU8Q274563475IU8-A2A-Q27456347-Na
23.81Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
23.81Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
23.81Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
23.81Single5UENDU1725UEN-A1-DU172
23.81Single5UIGCmpd-15UIG-A2A-Cmpd-1
23.81Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
23.81Single6GPSMK08126GPS-CCR2-MK0812
23.81Single6S0LZM-2413856S0L-A2A-ZM-241385
23.81Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
23.81Single7F83PF-051904577F83-Ghrelin-PF-05190457
23.81Single7PYRPSB-21157PYR-A2A-PSB-2115
23.81Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
23.81Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
23.81Single7YXAONO-54306087YXA-S1P5-ONO-5430608
23.81Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.81Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
23.81Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
23.81Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
23.81Consensuscck_offOrthosteric Ligandccka_off
23.81Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
23.81Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
23.81Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
23.81Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
23.53Single3OE8IT1t3OE8-CXCR4-IT1t
23.53Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
23.53Single6TQ9SB-4081246TQ9-OX1-SB-408124
23.53Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
23.53Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
23.53Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
23.53Single8A2OTheophylline8A2O-A2A-Theophylline-Na
23.53Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
23.53Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
23.53Consensussensory_onOrthosteric Ligandopsins_on
23.33Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
23.33Single6FJ3PTH6FJ3-PTH1-PTH
23.33Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
23.33Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
23.33Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
23.33Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
23.33Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
23.33Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
23.08Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
23.08Single7F8XNN90567F8X-CCKA-NN9056
23.08Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
23.08Single8KIGSHU91198KIG-MC3-SHU9119-Ca
23.08Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
23.08Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
23.08Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
22.86Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
22.73Single2Y00Dobutamine2Y00-β1-Dobutamine
22.73Single4NTJAZD12834NTJ-P2Y12-AZD1283
22.73Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
22.73Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
22.73Single5CGCHTL142425CGC-mGlu5-HTL14242
22.73Single5IUAQ274563485IUA-A2A-Q27456348-Na
22.73Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
22.73Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
22.73Single6GPXMK08126GPX-CCR2-MK0812
22.73Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
22.73Single6LUQHaloperidol6LUQ-D2-Haloperidol
22.73Single6S0QZM-2413856S0Q-A2A-ZM-241385
22.73Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
22.73Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
22.73Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
22.73Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
22.73Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
22.73Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.73Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
22.73Single8GNEKW-63568GNE-A2A-KW-6356-Na
22.73Single8QOTNanobody-E8QOT-μ-Nanobody-E
22.73Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
22.73Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
22.73Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
22.73Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
22.73Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
22.73Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
22.73Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
22.73Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
22.73Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
22.73Consensusep_offOrthosteric Ligandep4_off
22.73Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
22.73Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
22.58Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
22.58Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
22.58Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
22.58Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
22.58Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.58Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
22.58Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
22.58Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
22.58Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
22.22Single6ME5Agomelatine6ME5-MT1-Agomelatine
22.22Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
22.22Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
22.22Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
22.22Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
22.22Single7WC5Psilocin7WC5-5-HT2A-Psilocin
22.22Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.22Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
22.22Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
22.22Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
22.22Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
22.22Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
22.22Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
22.22Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
22.22Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
22.22Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
22.22Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
22.22Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
22.22Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
22.22Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
22.22Consensusgi_sensoryOrthosteric Ligandgi_opsins
22.22Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
22.22Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
21.88Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
21.88Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
21.88Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
21.88Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
21.88Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
21.88Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
21.88Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
21.88Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
21.88Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
21.74Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
21.74Single4BV0Neurotensin4BV0-NTS1-Neurotensin
21.74Single5TZRMK86665TZR-FFA1-MK8666
21.74Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
21.74Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
21.74Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
21.74Single7PX4PSB-21137PX4-A2A-PSB-2113
21.74Single7R0CAVP7R0C-V2-AVP-Arrestin2
21.74Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
21.74Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
21.74Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
21.74Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
21.74Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
21.74Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
21.74Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
21.74Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.74Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
21.74Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
21.74Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
21.74Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
21.74Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.74Consensusneurotensin_onOrthosteric Ligandnts1_on
21.74Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
21.74Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
21.74Consensusrelaxin_onOrthosteric Ligandrxfp4_on
21.74Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
21.43Single3OE0CVX153OE0-CXCR4-CVX15
21.43Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
21.43Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
21.43Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
21.43Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
21.43Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
21.43Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
21.43Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
21.43Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
21.43Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
21.43Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
21.43Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
21.05Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
21.05Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
21.05Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
21.05Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
21.05Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
21.05Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
21.05Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
20.83Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
20.83Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
20.83Single4XEENeurotensin4XEE-NTS1-Neurotensin
20.83Single4XESNeurotensin4XES-NTS1-Neurotensin
20.83Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
20.83Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
20.83Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
20.83Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
20.83Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
20.83Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
20.83Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
20.83Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.83Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
20.83Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.69Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
20.69Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
20.69Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.69Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
20.69Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
20.69Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
20.69Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
20.59Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
20.59Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
20.59Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
20.51Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
20.00Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
20.00Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
20.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
20.00Single4BUONeurotensin4BUO-NTS1-Neurotensin
20.00Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
20.00Single5CGDHTL142425CGD-mGlu5-HTL14242
20.00Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
20.00Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
20.00Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
20.00Single5U09Taranabant5U09-CB1-Taranabant
20.00Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
20.00Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
20.00Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
20.00Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
20.00Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
20.00Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
20.00Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
20.00Single7F8ULintitript7F8U-CCKA-Lintitript
20.00Single7F8YDevazepide7F8Y-CCKA-Devazepide
20.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
20.00Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
20.00Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
20.00Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
20.00Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
20.00Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
20.00Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
20.00Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
20.00Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
20.00Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
20.00Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
20.00Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
20.00Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
20.00Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
20.00Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9BA0A1AKN9BA0-CB1-A1AKN
20.00Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
20.00Consensusangiotensin_offOrthosteric Ligandat1_off
20.00Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
20.00Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
20.00Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
20.00Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
20.00Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
20.00Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
20.00Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
20.00Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
20.00Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
20.00Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
19.35Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
19.35Single7SK3CXCL127SK3-ACKR3-CXCL12
19.35Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
19.35Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
19.23Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
19.23Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
19.23Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
19.23Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
19.23Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
19.05Single3REYXAC3REY-A2A-XAC
19.05Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
19.05Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
19.05Single5IUBQ274563445IUB-A2A-Q27456344-Na
19.05Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
19.05Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
19.05Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
19.05Single5UVIZM-2413855UVI-A2A-ZM-241385
19.05Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
19.05Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
19.05Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
19.05Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
19.05Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
19.05Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
18.92Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
18.75Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
18.75Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
18.75Single5MZPCaffeine5MZP-A2A-Caffeine-Na
18.75Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
18.75Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
18.75Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
18.75Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
18.75Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
18.75Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
18.52Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
18.52Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
18.52Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
18.52Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
18.52Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
18.52Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
18.52Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
18.52Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single4QIMANTA XV4QIM-SMO-ANTA XV
18.18Single5T04Neurotensin5T04-NTS1-Neurotensin
18.18Single6D27CAY104716D27-DP2-CAY10471
18.18Single6IIVDaltroban6IIV-TP-Daltroban
18.18Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
18.18Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
18.18Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
18.18Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
18.18Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
18.18Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
18.18Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
18.18Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
18.18Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
18.18Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
18.18Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
18.18Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
18.18Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
18.18Single9B9ZA1AKO9B9Z-CB1-A1AKO
18.18Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
18.18Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
18.18Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
17.86Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
17.86Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
17.86Single7XNACYN1548067XNA-SST2-CYN154806
17.86Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.86Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
17.86Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
17.65Single7WC4Serotonin7WC4-5-HT2A-Serotonin
17.39Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
17.39Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
17.39Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
17.39Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
17.39Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
17.39Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
17.39Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
17.39Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
17.39Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
17.24Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
17.24Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
17.24Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
17.24Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
17.14Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
16.67Single3RFMCaffeine3RFM-A2A-Caffeine
16.67Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
16.67Single5V56TC1145V56-SMO-TC114
16.67Single6OS1TRV0266OS1-AT1-TRV026
16.67Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
16.67Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
16.67Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
16.67Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
16.67Single7P2L4YI7P2L-mGlu5-4YI
16.67Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
16.67Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
16.67Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
16.67Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
16.67Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
16.67Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
16.67Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
16.67Single9BJKNAM9BJK-μ-Naloxone-NAM
16.67Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
16.67Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.22Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
16.22Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
16.13Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
16.13Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
16.13Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
16.00Single4PY02MeSATP4PY0-P2Y12-2MeSATP
16.00Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
16.00Single6IIURamatroban6IIU-TP-Ramatroban
16.00Single6OS2TRV0266OS2-AT1-TRV026
16.00Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
16.00Single6YVRNTS8-136YVR-NTS1-NTS8-13
16.00Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
16.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
16.00Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.00Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
16.00Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
16.00Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
16.00Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
16.00Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
16.00Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
16.00Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
16.00Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
16.00Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.00Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
15.79Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
15.79Single3UZAGTPL92363UZA-A2A-GTPL9236
15.79Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
15.79Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
15.62Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
15.62Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
15.38Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
15.38Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
15.38Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
15.38Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
15.38Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
15.38Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
15.00Single6LI0C176LI0-GPR52-C17
15.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
15.00Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
15.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
15.00Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
15.00Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
15.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
15.00Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Consensusgq_nucleotideOrthosteric Ligandgq_p2y
15.00Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.81Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
14.81Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
14.81Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
14.81Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
14.81Single8XQJJN2418XQJ-Apelin-JN241
14.81Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
14.81Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
14.81Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
14.81Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
14.81Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
14.81Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
14.71Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
14.29Single4BWBNeurotensin4BWB-NTS1-Neurotensin
14.29Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
14.29Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
14.29Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
14.29Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
14.29Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
14.29Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
14.29Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
14.29Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
14.29Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
14.29Single8XWNCXCL88XWN-CXCR2-CXCL8
14.29Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
14.29Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
14.29Consensussomatostatin_offOrthosteric Ligandsst2_off
13.79Single7SK5CXCL127SK5-ACKR3-CXCL12
13.79Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
13.79Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
13.64Single6FFIMMPEP6FFI-mGlu5-MMPEP
13.64Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
13.64Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
13.64Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
13.64Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
13.64Single7VV6C48/807VV6-MRGPRX2-C48/80
13.64Single8K2WAMG4878K2W-CXCR3-AMG487
13.64Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
13.64Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
13.64Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
13.64Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
13.16Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
13.16Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
13.04Single6FFHFenobam6FFH-mGlu5-Fenobam
13.04Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
13.04Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
13.04Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
13.04Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
13.04Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
13.04Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
13.04Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
12.90Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
12.50Single4JKVTaladegib4JKV-SMO-Taladegib
12.50Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
12.50Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
12.50Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
12.50Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
12.50Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
12.12Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
12.00Single5V57TC1145V57-SMO-TC114
12.00Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
12.00Single7F1TMIP-1a7F1T-CCR5-MIP-1a
12.00Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
12.00Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
11.76Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
11.54Single8XQJJN2418XQJ-Apelin-JN241
11.11Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
11.11Single8XVUCXCL28XVU-CXCR2-CXCL2
11.11Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
10.71Single6KNMJN241-96KNM-Apelin-JN241-9
10.53Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
10.53Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
10.53Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
10.53Consensusp2y_offOrthosteric Ligandp2y1_off
10.34Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
10.34Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
10.34Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
10.00Single4XNWMRS25004XNW-P2Y1-MRS2500
10.00Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
10.00Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
10.00Single7SHEPI; PE7SHE-GPR158-PI; PE
10.00Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
10.00Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
10.00Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
10.00Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
10.00Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
9.52Single4O9RCyclopamine4O9R-SMO-Cyclopamine
9.52Single5L7IVismodegib5L7I-SMO-Vismodegib
9.52Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.52Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
9.52Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
9.52Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
9.38Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
9.09Single4QINSAG1.54QIN-SMO-SAG1.5
9.09Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
9.09Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
9.09Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
9.09Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
9.09Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
9.09Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
9.09Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
9.09Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
9.09Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.70Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
8.70Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
8.70Single6ZINSR486926ZIN-NTS1-SR48692
8.70Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
8.70Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single8IYXYL-3658IYX-GPR34-YL-365
8.70Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
8.33Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
8.00Single6Z4SSR486926Z4S-NTS1-SR48692
8.00Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
8.00Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
7.69Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
7.69Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
7.69Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
7.69Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
7.41Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
7.41Single8XWACXCL18XWA-CXCR2-CXCL1
7.41Single8XWMCXCL68XWM-CXCR2-CXCL6
7.41Single8XWSCXCL58XWS-CXCR2-CXCL5
7.41Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
7.14Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
7.14Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
7.14Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
7.14Single8XWFCXCL38XWF-CXCR2-CXCL3
7.14Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
6.90Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
6.67Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
6.67Single6D35Cholesterol6D35-SMO-Cholesterol
6.67Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
6.67Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
6.67Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
6.67Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
6.67Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
6.67Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
6.67Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
6.67Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
6.67Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
6.67Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
6.67Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
6.67Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
6.67Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
6.67Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
6.67Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
6.67Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
6.67Single7DTTCa7DTT-CaS-Ca-Ca
6.67Single7DTTCa7DTT-CaS-Ca-Ca
6.67Single7DTUTryptophan7DTU-CaS-Tryptophan
6.67Single7DTUTryptophan7DTU-CaS-Tryptophan
6.67Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
6.67Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
6.67Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
6.67Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
6.67Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.67Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.67Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.67Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.67Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
6.67Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
6.67Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
6.67Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
6.67Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
6.67Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
6.67Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
6.67Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
6.67Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
6.67Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
6.67Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
6.67Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
6.67Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
6.67Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
6.67Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
6.67Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
6.67Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
6.67Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.67Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.67Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.67Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.67Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
6.67Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
6.67Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
6.67Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
6.67Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
6.67Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
6.67Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.67Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.67Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.67Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
6.67Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.67Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.67Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.67Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
6.67Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
6.67Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
6.67Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
6.67Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
6.67Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
6.67Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
6.67Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
6.67Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
6.67Single7XW7K1-707XW7-TSH-K1-70
6.67Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
6.67Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
6.67Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
6.67Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
6.67Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
6.67Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
6.67Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
6.67Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
6.67Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
6.67Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
6.67Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
6.67Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
6.67Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
6.67Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
6.67Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
6.67Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
6.67Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
6.67Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
6.67Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
6.67Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
6.67Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
6.67Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
6.67Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
6.67Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
6.67Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
6.67Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
6.67Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
6.67Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
6.67Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
6.67Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
6.67Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
6.67Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
6.67Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
6.67Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
6.67Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
6.67Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
6.67Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
6.67Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
6.67Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.67Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
6.67Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
6.67Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
6.67Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
6.67Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
6.67Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
6.67Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
6.67Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
6.67Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
6.67Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
6.67Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
6.67Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
6.67Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
6.67Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
6.67Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
6.67Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
6.67Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
6.67Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
6.67Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
6.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.67Single8WVXNorrin8WVX-LGR4-Norrin
6.67Single8WVYNorrin8WVY-LGR4-Norrin
6.67Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
6.67Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
6.67Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
6.67Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
6.67Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
6.67Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
6.67Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
6.67Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.67Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.67Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.67Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.67Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.67Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
6.67Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
6.67Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
6.67Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.67Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.67Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.67Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
6.67Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
6.67Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
6.67Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
6.67Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
6.67Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
6.67Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
6.67Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
6.67Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
6.45Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
6.25Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
6.25Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
6.25Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
6.25Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
6.25Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
6.25Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
6.25Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
6.25Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
6.25Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
6.25Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.25Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
6.25Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
6.25Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.88Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
5.88Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
5.88Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
5.56Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
5.56Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
5.56Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
5.56Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
5.56Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
5.56Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
5.26Single5L7DCholesterol5L7D-SMO-Cholesterol
5.26Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
5.26Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
5.26Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
5.26Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
5.26Single8HS2Fab0468HS2-GPR20-Fab046
5.26Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
5.26Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
5.26Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
5.00Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
4.76Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
4.76Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
4.76Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
4.76Single8JPSCCL78JPS-ACKR1-CCL7
4.76Single8ZPLCholesterol8ZPL-CXCR4-HF51116-Cholesterol
4.76Single8ZPMCholesterol8ZPM-CXCR4-AMD070-Cholesterol
4.55Single8HNNSCH5467388HNN-CXCR3-SCH546738
4.55Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.55Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
4.55Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.35Single4K5YCP-3763954K5Y-CRF1-CP-376395
4.00Single4Z9GCP-3763954Z9G-CRF1-CP-376395
4.00Single8GTIBMK-C2058GTI-CRF1-BMK-C205
4.00Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
4.00Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
4.00Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
3.85Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
3.85Single8GTGBMK-I1528GTG-CRF1-BMK-I152
3.85Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
3.85Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
3.85Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
3.85Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
3.57Single7SHEPI; PE7SHE-GPR158-PI; PE
3.57Single8GTMBMK-C2038GTM-CRF1-BMK-C203
3.23Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
3.23Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
3.03Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
3.03Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.94Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.70Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
7VIE 7VIE-S1P1-S1P-Gi1/β1/γ2
7EW3 7EW3-S1P3-S1P-Gi1/β1/γ2
7EVY 7EVY-S1P1-Siponimod-Gi1/β1/γ2
7EW1 7EW1-S1P5-Siponimod-Gi1/β1/γ2
7VIF 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
7VIG 7VIG-S1P1-CBP-307-Gi1/β1/γ2
7EVZ 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
7EW4 7EW4-S1P3-CYM5541-Gi1/β1/γ2
7EW2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
7EW0 7EW0-S1P1-Ozanimod-Gi1/β1/γ2
7EW7 7EW7-S1P1-SEW2871-Gi1/β1/γ2
Net Summary
Imin 2.52
Number of Linked Nodes 884
Number of Links 1103
Number of Hubs 179
Number of Links mediated by Hubs 693
Number of Communities 24
Number of Nodes involved in Communities 264
Number of Links involved in Communities 389
Path Summary
Number Of Nodes in MetaPath 99
Number Of Links MetaPath 98
Number of Shortest Paths 1038115
Length Of Smallest Path 3
Average Path Length 27.7681
Length of Longest Path 61
Minimum Path Strength 0.274091
Average Path Strength 5.12717
Maximum Path Strength 40.3345
Minimum Path Correlation 0.700909
Average Path Correlation 0.976254
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2
Average % Of Corr. Nodes 46.0214
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 50.33
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
gi_lipidgi_cannabinoid
gi_ffa
gi_leukotriene
gi_lpa
gi_s1p



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