Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.30 2.90143404
2G.HN.41 1.16071404
3G.HN.51 4.93714404
4G.S3.03 5.88114508
5G.S3.04 7.79464417
6G.S3.06 8.11321417
7G.s3h2.03 4.99286419
8G.H2.01 6.26143409
9G.H2.06 6.42571519
10G.H2.07 7.47679419
11G.h2s4.01 8.75536419
12G.S4.04 4.13821409
13G.H3.08 4.045408
14G.H3.09 5.261676199
15G.H3.13 9.874575196
16G.H3.17 9.45095615
17G.S5.04 4.92429409
18G.S5.05 3.902146129
19G.HG.03 4.094206
20G.hgh4.05 7.88114506
21G.hgh4.20 3.4175403
22G.hgh4.21 4.93786404
23G.H4.03 3.235404
24G.H4.08 4.372553
25G.H4.10 10.4218407
26G.H4.12 6.04371554
27G.H4.15 7.03714408
28G.h4s6.20 6.69536474
29G.S6.02 7.58857578
30G.S6.05 7.38286555
31G.s6h5.01 5.35754129
32G.H5.03 5.153574129
33G.H5.05 3.876794115
34G.H5.08 5.342295118
35G.H5.13 4.985478
36G.H5.16 4.3825476
37G.H5.17 7.79286575
38g.l1x4 5.22536408
39g.h2x11 9.802144106
40g.ctx3 7.13536409
41g.ctx6 3.47857406
42g.ctx14 5.23943599
43g.ctx15 6.37821499
44g.ctx16 4.85321898
45g.ctx17 3.77643407
461x31 1.04607403
471x60 4.22964406
482x40 5.173145149
492x42 3.76592708
502x46 5.468574139
512x50 6.959435139
522x57 3.33714427
53E1x50 6.18214827
543x28 6.22743525
553x34 3.44754215
563x51 8.79071408
57I2x51 5.88107406
584x50 4.82409
594x58 4.201074214
60E2 16.11651123
615x37 2.78393402
625x39 6.38143426
635x47 8.742528
645x50 3.69393408
655x58 4.95429609
66I3 4.16939754
676x37 3.43408
686x44 5.56036429
696x48 7.70333628
706x49 3.8775406
716x51 8.31548626
726x52 8.96229527
73E3 5.33898722
747x34 4.35393425
757x39 4.685605
767x42 6.13286626
777x49 6.133934139
787x52 3.43893408
797x53 4.98457509
808x50 6.943576149
81Lig 8.038241320
82b.1x11 2.34714401
83b.1x13 2.84143407
84b.lhb1x3 3.11314502
85b.lhb1x6 3.54286403
86b.l1x3 8.93229569
87b.l1x6 9.48514519
88b.b2x1 6.852518
89b.b2x5 7.01629507
90b.b3x3 4.21408
91b.l3x1 8.91964419
92b.l3x2 5.974575189
93b.b4x3 4.284157
94b.b4x6 9.18405669
95b.l4x2 10.7782494
96b.b5x3 4.92551769
97b.b5x7 5.30607407
98b.l5x1 4.337435158
99b.l5x5 8.21314519
100b.b6x1 5.41036419
101b.b6x5 4.66607406
102b.l6x5 5.729294164
103b.b7x1 5.943934164
104b.b7x4 3.678574158
105b.b8x3 3.06786406
106b.b8x4 5.284295156
107b.l9x3 8.3375419
108b.l9x6 5.56667918
109b.b10x5 4.47143509
110b.b11x4 4.786519
111b.l11x2 8.02464419
112b.b12x5 3.86929446
113b.b12x6 8.03214618
114b.l12x1 3.34893406
115b.b13x7 7.26657547
116b.l13x3 7.05976649
117b.l13x6 6.48643419
118b.b15x1 6.98107449
119b.b15x2 5.97714436
120b.l15x2 6.26214449
121b.b16x4 10.3421446
122b.b16x5 3.93571505
123b.b16x6 7.69357648
124b.b17x5 7.08679437
125b.b17x7 7.42964438
126b.l17x3 8.34204739
127b.l17x6 9.33893419
128b.b18x3 5.13321438
129b.b18x5 5.25571405
130b.l18x1 6.427688106
131b.l18x2 6.22254107
132b.b19x2 6.70486536
133b.b19x4 5.96643438
134b.l19x2 8.15821439
135b.b20x4 10.4614538
136b.b20x6 6.36905636
137b.b20x7 4.57571409
138b.l20x2 7.78714409
139b.b21x1 8.89786437
140b.b21x2 3.24607406
141b.b21x7 5.38388705
142b.l21x2 4.62643404
143b.b22x5 5.124575107
144b.l22x5 7.32643409
145b.b23x6 7.3456177
146b.l23x1 6.69357416
147b.b24x4 8.579644176
148b.b24x6 7.050714178
149b.l24x3 3.97571505
150b.l25x3 8.09086589
151b.l25x6 13.78518
152b.l27x1 10.2945719
153b.l27x2 8.59393489
154b.b28x2 5.70286484
155b.b28x3 3.71929407
156b.b28x4 6.45686586
157b.b28x6 10.2311489
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b2x3 b.b2x5 21.64824.65143NoYes067
2b.b26x2 b.b2x3 21.96135.32286NoNo076
3b.b26x1 b.b26x2 22.11933.19429NoNo097
4b.b26x1 b.l27x1 22.2785.11714NoYes099
5b.b2x1 b.l27x1 45.02025.92571YesYes189
6b.l25x6 b.l27x1 67.525524.7043YesYes189
7b.b22x1 b.l25x6 67.71745.17143NoYes188
8b.b22x1 b.b22x2 83.52893.88571NoNo088
9b.b22x2 b.b26x3 83.65996.43714NoNo086
10b.b23x3 b.b26x3 83.76083.95429NoNo076
11b.b23x3 b.b27x1 98.19874.68286NoNo076
12b.b27x1 g.ctx5 98.6183.19286NoNo069
13b.lhb1x11 g.ctx5 98.7465.85714NoNo049
14b.b25x7 b.lhb1x11 98.87395.65428NoNo074
15b.b25x7 b.b28x6 99.129515.1314NoYes079
16b.b27x3 b.b28x6 49.5548.83571NoYes089
17b.b27x3 b.l25x3 49.60847.04143NoYes089
18b.l25x3 b.l27x2 99.5048.46143YesYes899
19b.l25x4 b.l27x2 99.97367.22429NoYes059
20I1x49 b.l25x4 10011.3986NoNo065
211x60 I1x49 50.22893.03571YesNo066
221x60 I1x50 50.21465.71286YesNo068
238x50 I1x50 50.02087.13286YesNo1498
247x54 8x50 99.605211.75NoYes079
251x53 7x54 99.56435.82857NoNo097
261x53 7x50 99.42.52429NoNo099
271x50 7x50 99.27628.38NoNo099
281x50 2x50 99.027110NoYes099
292x46 2x50 46.97455.23571YesYes1399
302x46 3x42 21.86094.63286YesNo098
312x45 3x42 21.78476.62286NoNo098
322x45 4x46 21.1585.39429NoNo098
332x42 4x46 21.08523.82857YesNo088
342x42 3x49 61.44016.99429YesNo088
353x49 I2x53 60.97297.71857NoNo087
363x53 I2x53 60.27178.57857NoNo087
373x53 G.H5.19 60.03794.81NoNo088
38G.H5.15 G.H5.19 59.57013.78571NoNo088
39G.H5.15 I2x50 59.33614.35714NoNo088
40G.H5.12 I2x50 15.20217NoNo778
41G.H5.12 I2x51 14.98463.74286NoYes076
42b.b28x4 b.b28x6 49.68468.12YesYes869
43b.b28x4 b.l25x3 49.82778.04714YesYes869
448x49 I1x49 49.80953.91429NoNo076
458x47 8x49 49.80753.36429NoNo087
468x47 8x50 49.80385.85143NoYes089
472x46 3x43 25.09574.55YesNo1398
483x43 7x53 50.42096.53NoYes089
493x46 7x53 42.18064.90286NoYes099
502x42 3x46 42.02173.88714YesNo089
512x50 7x49 51.54856.73143YesYes1399
523x43 7x49 25.47614.51NoYes1389
53G.H2.07 b.l9x6 18.49065.65YesYes198
54b.b6x1 b.l9x6 41.09656.5YesYes198
55b.b2x1 b.b6x1 41.38737.69714YesYes189
56G.H2.04 G.H2.07 18.19057NoYes099
57G.H5.16 I2x50 43.89994.06286YesNo768
585x68 G.H5.16 42.97427.49714NoYes776
595x68 G.H5.13 21.1277.08714NoYes778
60G.H5.13 G.S6.02 20.64963.94143YesYes788
61G.H5.10 G.S6.02 39.868111.6571NoYes078
62G.H5.10 G.S5.03 18.97046.4NoNo079
635x68 G.H5.17 21.61049.01143NoYes775
64G.H5.17 G.S6.02 20.64959.40714YesYes758
65G.H2.04 G.H3.08 18.02866.42NoYes098
66G.H3.08 G.S4.04 17.40686.26429YesYes089
67G.S4.04 G.S5.04 11.89723.65286YesYes099
68G.S5.03 G.S5.05 18.0093.23NoYes099
69G.S5.05 G.s6h5.01 18.995.18857YesYes1299
70G.H5.10 G.S6.04 20.418510.0829NoNo079
71G.S5.05 G.S6.04 18.0154.04YesNo099
72G.s6h5.01 G.s6h5.05 13.36264.33714YesNo1299
73G.s6h5.02 G.s6h5.05 24.7352.89NoNo089
74G.HG.02 G.s6h5.02 22.85853.33286NoNo098
75G.HG.02 G.HG.03 20.92583.88NoYes096
76G.HG.03 G.s5hg.01 15.12725.84143YesNo2069
77G.S4.07 G.s5hg.01 13.19456.60857NoNo089
78G.H5.03 G.S5.05 15.18085.87YesYes1299
79G.H5.03 G.s6h5.05 13.3054.61714YesNo1299
80b.l21x7 b.l23x1 17.01673.77857NoYes056
81b.l21x7 b.l23x2 16.67996.22429NoNo058
82b.b23x6 b.l23x2 16.00364.92857YesNo078
83b.b23x6 b.b24x6 13.95736.20143YesYes1778
84b.b21x7 b.b24x6 13.66668.40714YesYes058
85b.b20x5 b.b21x7 11.80964.85571NoYes075
86b.b20x5 b.b21x4 11.63573.16429NoNo075
87b.b21x4 g.h2x1 10.75122.34143NoNo058
88b.b21x2 g.h2x1 10.57613.68429YesNo068
89b.1x19 b.b21x2 10.05085.17286NoYes036
90b.b2x5 b.l4x1 12.09024.94YesNo075
916x48 7x45 26.60638.07143YesNo089
927x45 7x49 26.83475.83857NoYes099
93b.b10x1 b.l9x6 11.70663.08571NoYes098
94b.b10x1 b.b11x5 11.54293.72571NoNo096
95b.b24x7 b.l22x5 10.773514.4614NoYes099
96b.b24x7 b.lhb1x6 13.59156.88286NoYes093
97b.lhb1x6 b.lhb1x9 14.0163.73YesNo033
98b.b23x1 b.lhb1x9 14.15813.46429NoNo053
99b.b23x3 b.b24x5 14.60163.83143NoNo075
100b.b23x1 b.b24x5 14.30265.10857NoNo055
101G.S4.07 G.s1h1.04 11.26144.42429NoNo089
102b.b22x1 b.l23x1 15.68093.92571NoYes186
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
2x563x283.327142NoYes7521
2x563x327.512NoNo7721
2x567x424.512NoYes7621
2x577x423.788572YesYes7621
2x593x288.112862NoYes5521
2x603x283.617140NoYes7521
3x28E1x5010.44432YesYes5712
3x28Lig5.635712YesYes5010
3x327x429.032NoYes7611
3x32Lig16.68862NoYes7010
3x334x574.614290NoNo5712
3x33Lig8.878570NoYes5010
3x366x489.284290NoYes6812
3x36Lig7.158570NoYes6010
3x375x4619.361430NoNo6521
E2E264.99712YesYes3322
5x39E27.142862YesYes6322
E2E2x525.661432YesNo3421
E2x52Lig17.98572NoYes4010
5x395x439.265712YesNo6521
5x43Lig5.932860NoYes5010
5x446x525.470NoYes5721
5x446x553.405710NoNo5522
5x461Lig4.301430NoYes5010
5x476x5219.292YesYes8721
6x486x515.298572YesYes8621
6x486x526.32YesYes8721
6x516x528.421432YesYes6711
6x516x557.077142YesNo6512
6x517x345.172862YesYes6512
6x517x3816.57142YesNo6511
6x51Lig7.351432YesYes6010
6x52Lig5.332YesYes7010
6x557x345.021432NoYes5522
7x387x4211.29712NoYes5611
7x38Lig14.88712NoYes5010
7x397x423.445710YesYes5621
7x42Lig4.725712YesYes6010
2x59E1x503.305712NoYes5722
7x35Lig3.585710NoYes3010
3x29E2x522.221430NoNo4421
7x31Lig2.035710NoYes2010

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
92.86Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
92.86Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
92.86Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
92.86Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
86.67Single6IBLArformoterol6IBL-β1-Arformoterol
86.67Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
85.71Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
84.62Single6H7MSalbutamol6H7M-β1-Salbutamol
80.00Single4LDEBI1671074LDE-β2-BI167107
80.00Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
80.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
80.00Single8JJ8Formoterol8JJ8-β2-Formoterol
78.57Single2Y03Isoprenaline2Y03-β1-Isoprenaline
78.57Single6E67BI1671076E67-β2-BI167107-Gs (fused)
78.57Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
78.57Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
78.57Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
78.57Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
78.57Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
78.57Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
78.57Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
78.57Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
76.92Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
76.92Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
76.92Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
76.92Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
76.92Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
76.92Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
76.92Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
76.92Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
75.00Single6H7LDobutamine6H7L-β1-Dobutamine
75.00Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
75.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
75.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
73.33Single3P0GBI1671073P0G-β2-BI167107
73.33Single6H7JIsoprenaline6H7J-β1-Isoprenaline
73.33Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
73.33Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
73.33Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
73.33Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
73.33Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
73.33Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
71.43Single2Y01Dobutamine2Y01-β1-Dobutamine
71.43Single2Y04Salbutamol2Y04-β1-Salbutamol
71.43Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
71.43Single4QKX35V4QKX-β2-35V
71.43Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
71.43Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
71.43Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
71.43Single7BU7BI1671077BU7-β1-BI167107
71.43Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
71.43Single7WC7Lisuride7WC7-5-HT2A-Lisuride
71.43Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
71.43Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
71.43Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
71.43Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
71.43Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
71.43Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
71.43Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
71.43Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
71.43Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
71.43Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
71.43Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
71.43Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
71.43Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
71.43Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
71.43Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
71.43Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
69.23Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
69.23Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
69.23Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
69.23Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
69.23Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
69.23Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
68.75Single4AMIBucindolol4AMI-β1-Bucindolol
68.75Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
68.75Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
68.75Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
68.75Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
68.75Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
66.67Single2RH1S-Carazolol2RH1-β2-S-Carazolol
66.67Single2Y00Dobutamine2Y00-β1-Dobutamine
66.67Single4IARErgotamine4IAR-5-HT1B-Ergotamine
66.67Single5JQHS-Carazolol5JQH-β2-S-Carazolol
66.67Single5WIUNemonapride5WIU-D4-Nemonapride
66.67Single5WIVNemonapride5WIV-D4-Nemonapride-Na
66.67Single7WC6LSD7WC6-5-HT2A-LSD
66.67Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
66.67Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
66.67Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
66.67Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
66.67Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
66.67Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
66.67Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
66.67Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
66.67Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
66.67Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
66.67Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
66.67Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
66.67Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
66.67Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
66.67Consensusamine_offonOrthosteric Ligandamine_off amine_on
66.67Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
66.67Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
66.67Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
66.67Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
66.67Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
66.67Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
66.67Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
66.67Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
66.67Consensustrace-amine_onOrthosteric Ligandta1_on
64.71Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
64.71Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
64.29Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
64.29Single6KUXRS-799486KUX-α2a-RS-79948
64.29Single6PS0S-Carazolol6PS0-β2-S-Carazolol
64.29Single6PS4ICI118-5516PS4-β2-ICI118-551
64.29Single6PS5S-Propranolol6PS5-β2-S-Propranolol
64.29Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
64.29Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
64.29Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
64.29Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
64.29Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
64.29Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
64.29Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
64.29Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
64.29Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
64.29Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
64.29Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
64.29Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
64.29Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
64.29Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
64.29Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
64.29Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
64.29Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
64.29Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
64.29Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
62.50Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
62.50Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
62.50Single5D5AS-Carazolol5D5A-β2-S-Carazolol
62.50Single5D5BS-Carazolol5D5B-β2-S-Carazolol
62.50Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
62.50Single6WGTLSD6WGT-5-HT2A-LSD
62.50Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
62.50Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
62.50Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
62.50Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
62.50Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
62.50Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
62.50Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
62.50Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
62.50Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
62.50Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
62.50Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
62.50Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
62.50Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
62.50Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
62.50Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
61.54Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
61.54Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
61.54Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
61.11Single8X5YAstemizole8X5Y-H1-Astemizole
60.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
60.00Single2Y02Carmoterol2Y02-β1-Carmoterol
60.00Single3NY8ICI118-5513NY8-β2-ICI118-551
60.00Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
60.00Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
60.00Single4GBRS-Carazolol4GBR-β2-S-Carazolol
60.00Single6PS1Timolol6PS1-β2-Timolol
60.00Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
60.00Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
60.00Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
60.00Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
60.00Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
60.00Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
60.00Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
60.00Single8JJOAlprenolol8JJO-β2-Alprenolol
60.00Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
60.00Single8JXRLSD8JXR-D1-LSD
60.00Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
60.00Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
60.00Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
60.00Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
60.00Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
60.00Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
60.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
60.00Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
60.00Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
60.00Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
60.00Consensus5ht5_onOrthosteric Ligand5ht5a_on
60.00Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
60.00Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
60.00Consensusdopamine_offOrthosteric Ligandd2_off d3_off
60.00Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
58.82Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
58.82Single3D4STimolol3D4S-β2-Timolol
58.82Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
58.82Single6MXTSalmeterol6MXT-β2-Salmeterol
58.82Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
58.82Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
58.82Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
58.82Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
58.82Single8JJLOlodaterol8JJL-β2-Olodaterol
58.82Consensusalpha1_offOrthosteric Ligandalpha1a_off
58.82Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
58.82Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
57.89Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
57.89Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
57.89Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
57.89Single8WDTphotoNECA8WDT-A2A-photoNECA
57.14Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
57.14Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
57.14Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
57.14Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
57.14Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
57.14Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
57.14Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
57.14Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
57.14Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
57.14Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
57.14Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
57.14Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
57.14Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
57.14Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
57.14Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
57.14Consensusalpha2_offOrthosteric Ligandalpha2c_off
57.14Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
57.14Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
57.14Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
56.25Single2YCWS-Carazolol2YCW-β1-S-Carazolol
56.25Single5D6LS-Carazolol5D6L-β2-S-Carazolol
56.25Single5TVNLSD5TVN-5-HT2B-LSD
56.25Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
56.25Single7C61Ergotamine7C61-5-HT1B-Ergotamine
56.25Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
56.25Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
56.25Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
56.25Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
56.25Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
56.25Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
56.25Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
55.56Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
55.56Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
55.56Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
53.85Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
53.85Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
53.33Single6A94Zotepine6A94-5-HT2A-Zotepine
53.33Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
53.33Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
53.33Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
53.33Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
53.33Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
53.33Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
53.33Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
53.33Single7UL3Famotidine7UL3-H2-Famotidine
53.33Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
53.33Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
53.33Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
53.33Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
53.33Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
53.33Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
53.33Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
53.33Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
53.33Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
53.33Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
53.33Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
53.33Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
53.33Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
53.33Consensusalpha1_onOrthosteric Ligandalpha1a_on
53.33Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
53.33Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
53.33Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
52.94Single2YDVNECA2YDV-A2A-NECA
52.94Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
52.94Single4U15Tiotropium4U15-M3-Tiotropium
52.94Single4UHRCGS216804UHR-A2A-CGS21680
52.94Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
52.94Single5G53NECA5G53-A2A-NECA-Gs
52.94Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
52.94Single6OL9Tiotropium6OL9-M5-Tiotropium
52.94Single7B6WCyclazosin7B6W-α1b-Cyclazosin
52.94Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
52.94Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
52.94Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
52.94Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
52.94Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
52.94Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
52.94Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
52.63Single3NY9ICI118-5513NY9-β2-ICI118-551
52.63Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
50.00Single3PBLEticlopride3PBL-D3-Eticlopride
50.00Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
50.00Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
50.00Single5CXVTiotropium5CXV-M1-Tiotropium
50.00Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
50.00Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
50.00Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
50.00Single6CM4Risperidone6CM4-D2-Risperidone
50.00Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
50.00Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
50.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
50.00Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
50.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
50.00Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
50.00Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
50.00Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
50.00Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
50.00Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
50.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
50.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
50.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
50.00Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
50.00Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
50.00Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
50.00Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
50.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
50.00Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
50.00Single8X64Desloratadine8X64-H1-Desloratadine
50.00Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
50.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
50.00Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
50.00Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
50.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Single9CHXS-Carazolol9CHX-β2-S-Carazolol
50.00Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
50.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
50.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
50.00Consensusalpha2_onOrthosteric Ligandalpha2b_on
50.00Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
50.00Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
50.00Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
50.00Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
50.00Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
50.00Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
50.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
50.00Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
47.37Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
47.37Single5X93K-87945X93-ETB-K-8794
47.37Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
47.37Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
47.37Single7UM4AS26747237UM4-5-HT5A-AS2674723
47.37Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
47.37Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
47.37Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
47.37Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
47.37Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
47.37Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
47.37Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
47.37Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
47.06Single5C1MBU725C1M-μ-BU72
47.06Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
47.06Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
47.06Single6PS6Timolol6PS6-β2-Timolol
47.06Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
47.06Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
47.06Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
47.06Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
47.06Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
47.06Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
47.06Single8JXSPF-61428JXS-D1-PF-6142
47.06Single8ZMFA1L108ZMF-5-HT2C-A1L10
47.06Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
47.06Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
47.06Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
47.06Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
47.06Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
47.06Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
46.67Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
46.67Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
46.67Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
46.67Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
46.67Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
46.67Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
46.67Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
46.67Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
46.67Single8IWESpermidine8IWE-TA9-Spermidine
46.67Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
46.67Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
46.67Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
46.67Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
46.67Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
46.67Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
46.67Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
46.67Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
46.67Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
46.15Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
46.15Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
46.15Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
46.15Single9CHUNoradrenaline9CHU-β2-Noradrenaline
46.15Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
46.15Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
45.00Single4UG2CGS216804UG2-A2A-CGS21680
45.00Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
45.00Single7SK9CCX6627SK9-ACKR3-CCX662
44.44Single5V54Methiothepin5V54-5-HT1B-Methiothepin
44.44Single6J21Aprepitant6J21-NK1-Aprepitant
44.44Single6TQ7SB-3348676TQ7-OX1-SB-334867
44.44Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
44.44Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
44.44Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
44.44Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
44.44Single8E0GBU728E0G-μ-BU72
44.44Single8EA0Iperoxo8EA0-M3-Iperoxo
44.44Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
44.44Consensus5ht1_offOrthosteric Ligand5ht1b_off
44.44Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
44.44Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
44.44Consensustachykinin_offOrthosteric Ligandnk1_off
43.75Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
43.75Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
43.75Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
43.75Single6TPGEMPA6TPG-OX2-EMPA
43.75Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
43.75Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
43.75Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
43.75Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
43.75Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
43.75Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
43.75Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
43.75Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
43.75Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
43.75Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
43.75Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
43.75Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
43.75Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
43.75Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
43.75Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
42.86Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
42.86Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.86Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.86Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
42.86Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
42.86Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
42.86Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
42.86Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
42.86Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
42.86Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
42.86Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
42.86Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
42.86Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
42.11Single4RWADIPP-NH24RWA-δ-DIPP-NH2
42.11Single6A93Risperidone6A93-5-HT2A-Risperidone
42.11Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
42.11Single7YITNalfurafine7YIT-κ-Nalfurafine
42.11Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
42.11Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
42.11Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
42.11Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
42.11Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
42.11Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
42.11Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
42.11Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
42.11Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
42.11Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
42.11Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
42.11Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
41.18Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
41.18Single4DAJTiotropium4DAJ-M3-Tiotropium
41.18Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
41.18Single4EJ4Naltrindole4EJ4-δ-Naltrindole
41.18Single4MQSIperoxo4MQS-M2-Iperoxo
41.18Single4U14Tiotropium4U14-M3-Tiotropium
41.18Single5DSGTiotropium5DSG-M4-Tiotropium
41.18Single6DRXLisuride6DRX-5-HT2B-Lisuride
41.18Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
41.18Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
41.18Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
41.18Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
41.18Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
41.18Single7UL4Alvimopan7UL4-μ-Alvimopan
41.18Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
41.18Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
41.18Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
41.18Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
41.18Single8T1WCVN4248T1W-GPR6-CVN424
41.18Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
41.18Single8X63Mepyramine8X63-H1-Mepyramine
41.18Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
41.18Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
41.18Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
41.18Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
41.18Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
41.18Consensushistamine_offOrthosteric Ligandh1_off
41.18Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
41.18Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
41.18Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
40.91Single3QAKUK-4320973QAK-A2A-UK-432097
40.91Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
40.91Single6HLOAprepitant6HLO-NK1-Aprepitant
40.91Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
40.00Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
40.00Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
40.00Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
40.00Single7EZCUKA7EZC-A2A-UKA
40.00Single7SRQLSD7SRQ-5-HT2B-LSD
40.00Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
40.00Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
40.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
40.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
40.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
40.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
40.00Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
40.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
40.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
40.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
40.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
40.00Consensusendothelin_offOrthosteric Ligandetb_off
40.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
40.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
40.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
40.00Consensusprostanoid_offOrthosteric Ligandep_off dp_off
39.13Single5WF5UK-4320975WF5-A2A-UK-432097
39.13Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
39.13Consensusangiotensin_onOrthosteric Ligandat1_on
39.13Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
38.89Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
38.89Single5WQCEMPA5WQC-OX2-EMPA
38.89Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
38.89Single6D26Fevipiprant6D26-DP2-Fevipiprant
38.89Single6LUQHaloperidol6LUQ-D2-Haloperidol
38.89Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
38.89Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
38.89Single6TP6Filorexant6TP6-OX1-Filorexant
38.89Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
38.89Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
38.89Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.89Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
38.89Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
38.89Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
38.89Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
38.89Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
38.89Consensusdp_offOrthosteric Liganddp2_off
38.46Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
38.10Single5WF6UK-4320975WF6-A2A-UK-432097
38.10Single6PT3DPI-2876PT3-δ-DPI-287
38.10Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
38.10Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
38.10Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
37.50Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
37.50Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
37.50Single6AKXA4R6AKX-CCR5-A4R
37.50Single6AKYMaraviroc6AKY-CCR5-Maraviroc
37.50Single6DS0Ly2660976DS0-5-HT2B-Ly266097
37.50Single6ME2Ramelteon6ME2-MT1-Ramelteon
37.50Single6TODEMPA6TOD-OX1-EMPA-Na
37.50Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
37.50Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
37.50Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
37.50Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
37.50Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
37.50Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
37.50Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
37.50Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
37.50Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
37.50Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
37.50Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
37.50Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
37.50Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
37.50Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
37.50Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
37.50Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
37.50Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
37.50Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
37.50Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
37.50Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
37.50Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
37.50Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
37.50Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
37.50Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
37.50Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
36.84Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
36.84Single4DJHJDTic4DJH-κ-JDTic
36.84Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
36.84Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
36.84Single6J20Aprepitant6J20-NK1-Aprepitant
36.84Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
36.84Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
36.84Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
36.84Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
36.84Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
36.84Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
36.84Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
36.84Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
36.84Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
36.84Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
36.84Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
36.84Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
36.84Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
36.84Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
36.84Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
36.84Single8XVLZibotentan8XVL-ETA-Zibotentan
36.84Consensusa2_onOrthosteric Liganda2b_on
36.84Consensusa2_on_gpOrthosteric Liganda2b_on_gp
36.84Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
36.84Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
36.84Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
36.84Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
36.84Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
36.84Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
36.84Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
36.36Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
36.36Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
36.36Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
36.36Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
36.36Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
36.36Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
36.36Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
36.36Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
36.00Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
36.00Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
36.00Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
35.71Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
35.71Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
35.71Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
35.71Consensussensory_onOrthosteric Ligandopsins_on
35.29Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
35.29Single2YDOAdenosine2YDO-A2A-Adenosine
35.29Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
35.29Single3REYXAC3REY-A2A-XAC
35.29Single3RZECidoxepin3RZE-H1-Cidoxepin
35.29Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
35.29Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
35.29Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
35.29Single4MBSMaraviroc4MBS-CCR5-Maraviroc
35.29Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
35.29Single4ZJCSB-6740424ZJC-OX1-SB-674042
35.29Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
35.29Single6TPNHTL66416TPN-OX2-HTL6641
35.29Single6VI4JDTic6VI4-κ-JDTic
35.29Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
35.29Single7AROLUF58337ARO-A2A-LUF5833-Na
35.29Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
35.29Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
35.29Single7T32ZM-2413857T32-A2A-ZM-241385
35.29Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
35.29Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
35.29Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
35.29Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
35.29Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
35.29Single8K5CAcipimox8K5C-HCA2-Acipimox
35.29Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
35.29Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
35.29Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
35.29Single9BJKNaloxone9BJK-μ-Naloxone-NAM
35.29Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
35.29Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
35.29Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
35.29Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
35.29Consensusopsins_offOrthosteric Ligandrhodopsin_off
35.29Consensussensory_offOrthosteric Ligandopsins_off
35.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
35.00Single6ZG4HTL00099366ZG4-M1-HTL0009936
35.00Single7DFPSpiperone7DFP-D2-Spiperone
35.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
35.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
35.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
35.00Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
35.00Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
35.00Single8JWY2-1188JWY-A2A-2-118
35.00Single8JWZAB9288JWZ-A2A-AB928-Na
35.00Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
35.00Single8XYIVUF106618XYI-CXCR3-VUF10661
35.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
35.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
35.00Consensusorexin_onOrthosteric Ligandox2_on
34.78Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
34.78Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
34.78Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
34.78Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
34.78Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
34.78Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
34.78Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
34.62Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
34.62Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
33.33Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
33.33Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
33.33Single3UZAGTPL92363UZA-A2A-GTPL9236
33.33Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
33.33Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
33.33Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
33.33Single5DHGC-355DHG-NOP-C-35
33.33Single5DHHSB-6121115DHH-NOP-SB-612111
33.33Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
33.33Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
33.33Single5UIGCmpd-15UIG-A2A-Cmpd-1
33.33Single6D27CAY104716D27-DP2-CAY10471
33.33Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
33.33Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
33.33Single6PT2KGCHM076PT2-δ-KGCHM07
33.33Single6TOTLemborexant6TOT-OX1-Lemborexant
33.33Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
33.33Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
33.33Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
33.33Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
33.33Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
33.33Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
33.33Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Single7WC5Psilocin7WC5-5-HT2A-Psilocin
33.33Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
33.33Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
33.33Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
33.33Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
33.33Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
33.33Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
33.33Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
33.33Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
33.33Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
33.33Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
33.33Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
33.33Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
33.33Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
33.33Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
33.33Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
33.33Single8RLNLUF58348RLN-A2A-LUF5834
33.33Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
33.33Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
33.33Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
33.33Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
33.33Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
33.33Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
33.33Consensus5ht2_onOrthosteric Ligand5ht2b_on
33.33Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Consensusa3_onOrthosteric Liganda3a_on
33.33Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
33.33Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusblt_onOrthosteric Ligandblt1_on
33.33Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
33.33Consensuschemerin_onOrthosteric Ligandcml1_on
33.33Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
33.33Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
33.33Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
33.33Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
33.33Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
33.33Consensusleukotriene_onOrthosteric Ligandblt_on
33.33Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
33.33Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
33.33Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
33.33Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
33.33Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
33.33Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
33.33Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
32.14Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
32.14Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
32.14Consensusbradykinin_onOrthosteric Ligandbk2_on
32.14Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
32.14Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
32.00Single6JODAngiotensin II6JOD-AT2-Angiotensin II
32.00Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
32.00Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
32.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
32.00Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
32.00Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
32.00Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Consensusvasop-oxy_onOrthosteric Ligandv2_on
32.00Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
31.82Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
31.82Single7XN9L-054,5227XN9-SST2-L-054,522
31.82Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
31.82Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
31.82Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
31.82Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
31.82Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
31.58Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
31.58Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
31.58Single5IUAQ274563485IUA-A2A-Q27456348-Na
31.58Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
31.58Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
31.58Single5XPRBosentan5XPR-ETB-Bosentan
31.58Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
31.58Single6HLPNetupitant6HLP-NK1-Netupitant
31.58Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
31.58Single6S0QZM-2413856S0Q-A2A-ZM-241385
31.58Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
31.58Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
31.58Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
31.58Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
31.58Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
31.58Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
31.58Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
31.58Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
31.58Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
31.58Single8TF5Oleic acid8TF5-GPR6-Oleic acid
31.58Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
31.58Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
31.58Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
31.58Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
31.58Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
31.58Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
31.58Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
31.58Consensusa3_on_gpOrthosteric Liganda3a_on_gp
31.58Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
31.58Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
31.58Consensusadenosine_offOrthosteric Liganda1_off a2_off
31.58Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
31.58Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
31.58Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
31.25Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
31.25Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
31.25Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
31.25Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
31.25Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
31.25Single6HLLCP999946HLL-NK1-CP99994
31.25Single6TP4ACT-4622066TP4-OX1-ACT-462206
31.25Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
31.25Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
31.25Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
31.25Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
31.25Single8K5BNiacin8K5B-HCA2-Niacin
31.25Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
31.25Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
31.25Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
31.25Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
31.03Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
31.03Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
31.03Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
31.03Consensusbombesin_onOrthosteric Ligandbb2_on
31.03Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
31.03Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
30.77Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
30.77Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
30.77Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.43Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
30.43Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
30.43Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
30.43Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
30.43Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
30.43Consensuslpl_onOrthosteric Ligands1p_on lpa_on
30.43Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
30.43Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
30.43Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
30.00Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
30.00Single6E59L-7607356E59-NK1-L-760735
30.00Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
30.00Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
30.00Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
30.00Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
30.00Single7TUYGSK682753A7TUY-GPR183-GSK682753A
30.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
30.00Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
30.00Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
30.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
30.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
30.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
30.00Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
30.00Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
30.00Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
30.00Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
30.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
30.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
30.00Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
30.00Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
29.63Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
29.63Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
29.63Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
29.63Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
29.63Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
29.41Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
29.41Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
29.41Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
29.41Single5WS3EMPA5WS3-OX2-EMPA
29.41Single6B73MP11046B73-κ-MP1104
29.41Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
29.41Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
29.41Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
29.41Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
29.41Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
29.41Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
29.41Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
29.41Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
29.41Single8GNGIstradefylline8GNG-A2A-Istradefylline
29.41Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
29.41Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
29.41Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
29.41Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
29.41Single8Y0HVUF114188Y0H-CXCR3-VUF11418
29.41Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
29.41Consensusangiotensin_offOrthosteric Ligandat1_off
29.41Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
29.41Consensusorexin_offOrthosteric Ligandox2_off ox1_off
29.41Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
29.41Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
29.41Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
29.41Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
29.41Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
29.41Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
29.17Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
29.17Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
29.17Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
29.17Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
29.17Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
29.17Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
29.17Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
29.03Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
28.57Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
28.57Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
28.57Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
28.57Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
28.57Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
28.57Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
28.57Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
28.57Single7K15MKD0467K15-BLT1-MKD046-Na
28.57Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
28.57Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
28.57Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
28.57Single7WC4Serotonin7WC4-5-HT2A-Serotonin
28.57Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
28.57Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
28.57Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
28.57Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
28.57Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
28.57Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
28.57Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
28.57Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
28.57Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
28.57Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
28.57Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
28.57Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
28.57Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
28.57Consensuslpa_offOrthosteric Ligandlpa1_off
28.57Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
28.57Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
28.57Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
28.57Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.00Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
28.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
28.00Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.78Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
27.78Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
27.78Single5IUBQ274563445IUB-A2A-Q27456344-Na
27.78Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
27.78Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
27.78Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
27.78Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
27.78Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
27.78Single6AQFZM-2413856AQF-A2A-ZM-241385
27.78Single6IQLL7458706IQL-D4-L745870
27.78Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
27.78Single6TP3Nemorexant6TP3-OX1-Nemorexant
27.78Single6V9SGTPL114036V9S-OX1-GTPL11403
27.78Single7VODCariprazine7VOD-5-HT2A-Cariprazine
27.78Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
27.78Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
27.78Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
27.78Single8IHKAcifran8IHK-HCA3-Acifran
27.78Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
27.78Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
27.78Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
27.78Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
27.78Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
27.78Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
27.78Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
27.78Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
27.78Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
27.78Consensushca_onOrthosteric Ligandhca2_on
27.59Single6IGLIRL16206IGL-ETB-IRL1620
27.59Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
27.59Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
27.27Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
27.27Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
27.27Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
27.27Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
27.27Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
27.27Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
27.27Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
27.27Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
27.27Single8XVJMacitentan8XVJ-ETA-Macitentan
27.27Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
27.27Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
27.27Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
27.27Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
26.92Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
26.92Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.92Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
26.92Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
26.92Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
26.67Single5GLHEndothelin-15GLH-ETB-Endothelin-1
26.67Single6IGKEndothelin-36IGK-ETB-Endothelin-3
26.67Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
26.67Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
26.32Single3EMLZM-2413853EML-A2A-ZM-241385
26.32Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
26.32Single4YAYZD-71554YAY-AT1-ZD-7155
26.32Single5IU8Q274563475IU8-A2A-Q27456347-Na
26.32Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
26.32Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
26.32Single5UENDU1725UEN-A1-DU172
26.32Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
26.32Single6GPSMK08126GPS-CCR2-MK0812
26.32Single6S0LZM-2413856S0L-A2A-ZM-241385
26.32Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
26.32Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
26.32Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
26.32Single7PYRPSB-21157PYR-A2A-PSB-2115
26.32Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
26.32Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
26.32Single7YXAONO-54306087YXA-S1P5-ONO-5430608
26.32Single8CU6LJ-45178CU6-A2A-LJ-4517
26.32Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
26.32Single8K5DGSK2560738K5D-HCA2-GSK256073
26.32Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
26.32Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
26.32Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
26.32Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
26.32Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
26.32Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
26.32Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
26.32Consensushca_on_gpOrthosteric Ligandhca2_on_gp
26.32Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
26.32Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
26.09Single5ZTYAM102575ZTY-CB2-AM10257
26.09Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
26.09Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
26.09Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
26.09Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
26.09Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
26.09Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
26.09Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
26.09Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
26.09Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
26.09Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
26.09Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
26.09Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
26.09Consensuskisspeptin_onOrthosteric Ligandkiss1_on
26.09Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
26.09Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
25.93Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
25.93Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
25.93Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.93Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
25.93Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
25.93Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
25.93Single8ZRTET-18ZRT-ETB-ET-1
25.81Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
25.81Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
25.00Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
25.00Single5CGCHTL142425CGC-mGlu5-HTL14242
25.00Single5N2RPSB-365N2R-A2A-PSB-36-Na
25.00Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
25.00Single6GPXMK08126GPX-CCR2-MK0812
25.00Single6ME5Agomelatine6ME5-MT1-Agomelatine
25.00Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
25.00Single7C4SS1P7C4S-S1P3-S1P
25.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
25.00Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
25.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
25.00Single7F8XNN90567F8X-CCKA-NN9056
25.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
25.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7SINNPS-21437SIN-CaS-NPS-2143
25.00Single7SINNPS-21437SIN-CaS-NPS-2143
25.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
25.00Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
25.00Single7W41PD1762527W41-BB2-PD176252
25.00Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
25.00Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
25.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
25.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
25.00Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
25.00Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
25.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
25.00Single8S4DCMF-0198S4D-Apelin-CMF-019
25.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
25.00Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
25.00Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
25.00Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
25.00Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
25.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
25.00Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
25.00Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
25.00Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
25.00Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
25.00Consensusblt_offOrthosteric Ligandblt1_off
25.00Consensusbombesin_offOrthosteric Ligandbb2_off
25.00Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
25.00Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
25.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.00Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.00Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
25.00Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
25.00Consensusgi_sensoryOrthosteric Ligandgi_opsins
25.00Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
25.00Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
25.00Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
25.00Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
25.00Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
25.00Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
25.00Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
25.00Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
25.00Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
25.00Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
25.00Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
25.00Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
25.00Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.24Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
24.14Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
24.14Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
24.14Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
24.00Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
24.00Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
24.00Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
24.00Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
24.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
24.00Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
24.00Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
24.00Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
24.00Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
24.00Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
24.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
23.81Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
23.81Single5XR8AM8415XR8-CB1-AM841
23.81Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
23.81Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
23.81Single7PX4PSB-21137PX4-A2A-PSB-2113
23.81Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
23.81Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
23.81Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
23.81Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
23.81Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
23.81Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
23.81Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
23.81Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
23.81Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.81Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
23.81Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
23.81Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
23.81Single9BJKNAM9BJK-μ-Naloxone-NAM
23.81Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
23.81Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.81Consensuslpa_onOrthosteric Ligandlpa1_on
23.81Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
23.81Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
23.53Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
23.53Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
23.53Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
23.53Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
23.53Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
23.53Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
23.53Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
23.53Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
23.53Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
23.53Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
23.53Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
23.53Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
23.53Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
23.53Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
23.53Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
23.53Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
23.53Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
23.53Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
23.33Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
23.33Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
23.33Consensusendothelin_onOrthosteric Ligandetb_on eta_on
23.33Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
23.08Single3OE0CVX153OE0-CXCR4-CVX15
23.08Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
23.08Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
23.08Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
23.08Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
22.73Single4N4WSANT-14N4W-SMO-SANT-1
22.73Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
22.73Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
22.73Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
22.73Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
22.73Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
22.73Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
22.73Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
22.73Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
22.73Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
22.73Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
22.73Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
22.73Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
22.73Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.73Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
22.73Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
22.73Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
22.73Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
22.73Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
22.73Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
22.73Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
22.73Consensuslpl_offOrthosteric Ligands1p_off lpa_off
22.73Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
22.73Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
22.58Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
22.58Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
22.58Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
22.58Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
22.58Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
22.22Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
22.22Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
22.22Single3PWHZM-2413853PWH-A2A-ZM-241385
22.22Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
22.22Single4S0VSuvorexant4S0V-OX2-Suvorexant
22.22Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
22.22Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
22.22Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
22.22Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
22.22Single6ME9Ramelteon6ME9-MT2-Ramelteon
22.22Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
22.22Single6TPJSuvorexant6TPJ-OX2-Suvorexant
22.22Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
22.22Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
22.22Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
22.22Single7F8ULintitript7F8U-CCKA-Lintitript
22.22Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
22.22Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
22.22Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
22.22Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
22.22Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
22.22Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
22.22Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
22.22Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
22.22Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
22.22Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
22.22Single7XRRLemborexant7XRR-OX2-Lemborexant
22.22Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
22.22Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
22.22Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
22.22Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
22.22Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
22.22Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
22.22Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
22.22Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
22.22Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
22.22Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.22Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
22.22Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
22.22Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.22Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.22Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
21.88Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
21.74Single5CGDHTL142425CGD-mGlu5-HTL14242
21.74Single6K1QIRL25006K1Q-ETB-IRL2500
21.74Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.74Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
21.74Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
21.74Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
21.74Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
21.74Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
21.74Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
21.74Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
21.74Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
21.74Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
21.74Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
21.74Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
21.74Consensuscck_onOrthosteric Ligandccka_on cckb_on
21.74Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
21.74Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
21.43Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
21.43Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
21.43Single5MZPCaffeine5MZP-A2A-Caffeine-Na
21.43Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
21.43Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.43Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
21.43Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
21.43Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
21.43Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
21.43Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
21.43Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
21.43Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
21.43Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
21.43Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
21.05Single5IU7Q274563465IU7-A2A-Q27456346-Na
21.05Single5JTBZM-2413855JTB-A2A-ZM-241385
21.05Single5UVIZM-2413855UVI-A2A-ZM-241385
21.05Single6MH8ZM-2413856MH8-A2A-ZM-241385
21.05Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
21.05Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
21.05Single6ZG9GSK10347026ZG9-M1-GSK1034702
21.05Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
21.05Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
21.05Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.05Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
21.05Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
21.05Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
21.05Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
21.05Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
21.05Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.05Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
21.05Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
21.05Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
21.05Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Consensusa2_offOrthosteric Liganda2a_off
21.05Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
21.05Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
20.83Single5EE7MK08935EE7-Glucagon-MK0893
20.83Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
20.83Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
20.83Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
20.83Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
20.83Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
20.83Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
20.69Single4XT3Fractalkine4XT3-US28-Fractalkine
20.69Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
20.69Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
20.69Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
20.00Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
20.00Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
20.00Single5TGZAM65385TGZ-CB1-AM6538
20.00Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
20.00Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
20.00Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
20.00Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
20.00Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
20.00Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
20.00Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.00Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
20.00Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
20.00Single7QA8Peptide7QA8-STE2-Peptide
20.00Single7QA8Peptide7QA8-STE2-Peptide
20.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
20.00Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
20.00Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
20.00Single7V3ZCP559407V3Z-CB1-CP55940
20.00Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
20.00Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
20.00Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
20.00Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.00Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
20.00Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
20.00Single8PWNTheophylline8PWN-A2A-Theophylline
20.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
20.00Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
20.00Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
20.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
20.00Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
20.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
20.00Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
20.00Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.00Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.00Consensussomatostatin_offOrthosteric Ligandsst2_off
19.44Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
19.44Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
19.35Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
19.35Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
19.35Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
19.35Single8IY6Endothelin-18IY6-ETB-Endothelin-1
19.35Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
19.23Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
19.23Single7XNACYN1548067XNA-SST2-CYN154806
19.23Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
19.23Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
19.23Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
19.23Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
19.23Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
19.23Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
19.05Single5N2SPSB365N2S-A1-PSB36
19.05Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
19.05Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
19.05Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
19.05Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
19.05Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
19.05Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
19.05Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
19.05Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
19.05Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.05Single8GNEKW-63568GNE-A2A-KW-6356-Na
19.05Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
19.05Single8QOTNanobody-E8QOT-μ-Nanobody-E
19.05Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
19.05Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
19.05Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
19.05Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
19.05Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
19.05Consensusep_offOrthosteric Ligandep4_off
19.05Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
19.05Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
18.75Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
18.75Single3RFMCaffeine3RFM-A2A-Caffeine
18.75Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
18.75Single6TQ9SB-4081246TQ9-OX1-SB-408124
18.75Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
18.75Single8A2OTheophylline8A2O-A2A-Theophylline-Na
18.52Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
18.52Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
18.52Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
18.52Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
18.52Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
18.52Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
18.52Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
18.52Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
18.52Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.52Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
18.52Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
18.52Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
18.52Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
18.52Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
18.52Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
18.52Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
18.52Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
18.52Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
18.18Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
18.18Single5XRAAM115425XRA-CB1-AM11542
18.18Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
18.18Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
18.18Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
18.18Single7F1TMIP-1a7F1T-CCR5-MIP-1a
18.18Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
18.18Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
18.18Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
18.18Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
18.18Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
18.18Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
18.18Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
18.18Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
18.18Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
18.18Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
18.18Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
18.18Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
18.18Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
18.18Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
18.18Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
18.18Consensusrelaxin_onOrthosteric Ligandrxfp4_on
18.18Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
17.86Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
17.86Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
17.86Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
17.86Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
17.86Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
17.86Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
17.86Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
17.86Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
17.65Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
17.65Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.65Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
17.65Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
17.65Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
17.65Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
17.65Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
17.65Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
17.39Single5X33BIIL2605X33-BLT1-BIIL260
17.39Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
17.39Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
17.39Single6OS2TRV0266OS2-AT1-TRV026
17.39Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
17.39Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
17.39Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
17.39Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
17.39Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
17.39Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
17.39Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
17.24Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
17.24Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
17.24Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
17.24Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
17.24Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
17.24Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
17.24Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
17.24Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
17.24Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
17.24Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
16.67Single3OE9IT1t3OE9-CXCR4-IT1t
16.67Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
16.67Single5L7IVismodegib5L7I-SMO-Vismodegib
16.67Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
16.67Single6LI0C176LI0-GPR52-C17
16.67Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
16.67Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
16.67Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
16.67Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.67Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
16.67Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
16.67Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
16.67Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
16.67Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
16.67Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
16.67Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
16.67Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
16.67Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
16.67Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
16.67Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
16.67Single9B9Y7DY9B9Y-CB1-7DY
16.67Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.67Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.67Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
16.67Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
16.67Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
16.67Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
16.13Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
16.13Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
16.13Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
16.00Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
16.00Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
16.00Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
16.00Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
16.00Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
16.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
16.00Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
16.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
16.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
16.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
16.00Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
16.00Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
16.00Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
15.79Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
15.79Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
15.79Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
15.79Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
15.79Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
15.79Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
15.79Single9BA0A1AKN9BA0-CB1-A1AKN
15.79Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
15.62Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
15.62Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
15.62Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
15.62Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
15.62Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
15.38Single4XT1Fractalkine4XT1-US28-Fractalkine
15.38Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
15.38Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8IEBA1LYA8IEB-GPR156-A1LYA
15.38Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
15.38Single8WKYPG-9348WKY-MC4-PG-934
15.38Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
15.38Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
15.38Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
15.38Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
15.15Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
15.00Single6FFIMMPEP6FFI-mGlu5-MMPEP
15.00Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
15.00Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
15.00Single6TPKRetosiban6TPK-OT-Retosiban
15.00Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
15.00Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
15.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
15.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
15.00Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
15.00Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.00Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
15.00Single8K2WAMG4878K2W-CXCR3-AMG487
15.00Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
15.00Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
15.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
15.00Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
15.00Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
15.00Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
15.00Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.00Consensusvasop-oxy_offOrthosteric Ligandot_off
14.81Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
14.81Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
14.81Single7SK5CXCL127SK5-ACKR3-CXCL12
14.81Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
14.81Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
14.81Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
14.81Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
14.81Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
14.71Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
14.71Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
14.71Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
14.71Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
14.29Single6FFHFenobam6FFH-mGlu5-Fenobam
14.29Single6IIVDaltroban6IIV-TP-Daltroban
14.29Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
14.29Single6W25SHU91196W25-MC4-SHU9119-Ca
14.29Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
14.29Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
14.29Single7F83PF-051904577F83-Ghrelin-PF-05190457
14.29Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
14.29Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
14.29Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
14.29Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
14.29Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
14.29Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
14.29Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
14.29Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
14.29Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
14.29Single9B9ZA1AKO9B9Z-CB1-A1AKO
14.29Single9IYAONO-97105319IYA-GPR55-ONO-9710531
14.29Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
14.29Consensuscck_offOrthosteric Ligandccka_off
14.29Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
14.29Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
14.29Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
13.89Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
13.89Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
13.79Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
13.79Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
13.79Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
13.79Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
13.79Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
13.79Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
13.79Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
13.79Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
13.79Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
13.79Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
13.79Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
13.79Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
13.64Single4NTJAZD12834NTJ-P2Y12-AZD1283
13.64Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
13.64Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
13.64Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
13.64Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
13.64Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
13.64Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
13.64Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
13.64Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
13.51Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
13.33Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
13.33Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
13.33Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
13.33Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
13.33Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
13.04Single6OS1TRV0266OS1-AT1-TRV026
13.04Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
13.04Single7FEECP559407FEE-CB1-CP55940-ZCZ011
13.04Single7P2L4YI7P2L-mGlu5-4YI
13.04Single7R0CAVP7R0C-V2-AVP-Arrestin2
13.04Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
13.04Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
13.04Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
13.04Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
13.04Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
13.04Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
13.04Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
13.04Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
13.04Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
13.04Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
13.04Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.04Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
13.04Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
13.04Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.04Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single6FJ3PTH6FJ3-PTH1-PTH
12.90Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
12.90Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
12.90Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
12.90Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
12.90Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
12.90Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
12.90Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
12.90Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
12.50Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
12.50Single6IIURamatroban6IIU-TP-Ramatroban
12.50Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
12.50Single6KQICP559406KQI-CB1-CP55940-Org27569
12.50Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
12.50Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
12.50Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
12.50Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
12.50Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
12.50Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
12.50Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
12.50Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
12.50Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
12.50Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
12.50Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
12.50Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
12.50Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
12.50Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
12.50Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
12.50Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
12.50Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
12.50Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
12.50Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
12.20Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
12.12Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
12.12Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
12.12Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
12.12Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
12.12Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
12.12Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
12.12Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
12.12Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
12.00Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
12.00Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
12.00Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
12.00Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
12.00Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
12.00Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
12.00Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single3OE8IT1t3OE8-CXCR4-IT1t
11.76Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
11.76Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
11.76Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
11.54Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
11.54Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
11.54Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
11.54Single8IEIA1LYA8IEI-GPR156-A1LYA
11.54Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
11.54Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
11.11Single3OE6IT1t3OE6-CXCR4-IT1t
11.11Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
11.11Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
11.11Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
11.11Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
11.11Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
11.11Single7V6A-7V6A-M4-PubChem 9864275-Gi1/β1/γ2
11.11Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
11.11Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.11Single8IEIA1LYA8IEI-GPR156-A1LYA
11.11Single8IEPA1LYA8IEP-GPR156-A1LYA
11.11Single8IEPA1LYA8IEP-GPR156-A1LYA
11.11Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.11Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
11.11Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
11.11Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
11.11Single8KIGSHU91198KIG-MC3-SHU9119-Ca
11.11Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
11.11Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
11.11Single8XWNCXCL88XWN-CXCR2-CXCL8
11.11Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
11.11Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
11.11Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
10.81Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
10.81Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.71Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
10.71Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
10.71Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
10.71Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single8IEBA1LYA8IEB-GPR156-A1LYA
10.71Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
10.71Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
10.53Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
10.53Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
10.53Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
10.53Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
10.53Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
10.53Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
10.53Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
10.53Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
10.53Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.53Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
10.53Consensusgq_nucleotideOrthosteric Ligandgq_p2y
10.53Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.34Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
10.34Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.34Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
10.00Single3ODUIT1t3ODU-CXCR4-IT1t
10.00Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
10.00Single5U09Taranabant5U09-CB1-Taranabant
10.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
10.00Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
10.00Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
10.00Single7BR3Elagolix7BR3-GnRH1-Elagolix
10.00Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
10.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
10.00Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
10.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
10.00Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
10.00Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
10.00Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
10.00Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
10.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
9.68Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
9.68Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
9.68Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
9.68Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
9.52Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
9.52Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
9.52Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
9.52Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
9.52Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.52Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
9.52Consensusgrh_offOrthosteric Ligandgnrh1_off
9.38Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
9.38Single7SK3CXCL127SK3-ACKR3-CXCL12
9.38Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
9.38Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
9.09Single4QIMANTA XV4QIM-SMO-ANTA XV
9.09Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
9.09Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
9.09Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
9.09Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
9.09Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
9.09Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.09Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
9.09Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
9.09Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
9.09Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
9.09Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
9.09Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
9.09Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
8.82Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
8.82Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
8.70Single4JKVTaladegib4JKV-SMO-Taladegib
8.70Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
8.70Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.70Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
8.70Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
8.70Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
8.70Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
8.70Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
8.70Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
8.57Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
8.33Single5TZRMK86665TZR-FFA1-MK8666
8.33Single5V56TC1145V56-SMO-TC114
8.33Single5V57TC1145V57-SMO-TC114
8.33Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
8.33Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
8.33Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
8.33Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
8.33Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
8.33Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
8.00Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
8.00Single4PY02MeSATP4PY0-P2Y12-2MeSATP
8.00Single4XEENeurotensin4XEE-NTS1-Neurotensin
8.00Single4XESNeurotensin4XES-NTS1-Neurotensin
8.00Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
8.00Single6YVRNTS8-136YVR-NTS1-NTS8-13
8.00Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
8.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
8.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
8.00Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
8.00Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
8.00Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
8.00Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
8.00Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
8.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.89Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
7.69Single4BUONeurotensin4BUO-NTS1-Neurotensin
7.69Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
7.69Single8XVUCXCL28XVU-CXCR2-CXCL2
7.69Single8XWFCXCL38XWF-CXCR2-CXCL3
7.69Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
7.69Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single6KNMJN241-96KNM-Apelin-JN241-9
7.41Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
7.41Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
7.41Single8XQJJN2418XQJ-Apelin-JN241
7.41Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
7.41Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
7.41Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
7.14Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.14Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
7.14Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.14Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
6.90Single7SHEPI; PE7SHE-GPR158-PI; PE
6.90Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
6.90Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
6.67Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
6.67Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
6.67Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
6.45Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
6.25Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
6.25Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
5.88Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
5.88Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
5.88Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
5.88Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.56Consensusp2y_offOrthosteric Ligandp2y1_off
5.26Single4XNWMRS25004XNW-P2Y1-MRS2500
5.26Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.26Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
5.26Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
5.26Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
5.26Single7F61Cholesterol7F61-H3-PF-03654746-Cholesterol
5.26Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
5.26Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
5.13Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
5.00Single4O9RCyclopamine4O9R-SMO-Cyclopamine
5.00Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
4.76Single4BWBNeurotensin4BWB-NTS1-Neurotensin
4.76Single4QINSAG1.54QIN-SMO-SAG1.5
4.76Single4XNVBPTU4XNV-P2Y1-BPTU
4.76Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
4.76Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
4.76Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
4.76Single7F8YDevazepide7F8Y-CCKA-Devazepide
4.76Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
4.76Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
4.76Single7WV9ZCZ0117WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
4.76Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
4.76Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
4.76Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
4.76Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
4.55Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
4.55Single6ZINSR486926ZIN-NTS1-SR48692
4.55Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
4.55Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
4.55Single8IYXYL-3658IYX-GPR34-YL-365
4.55Single8JD6N-(3-chlorophenyl)pyridine-2-carboxamide8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
4.35Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.35Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
4.35Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
4.35Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
4.35Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
4.35Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
4.17Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
4.17Single6Z4SSR486926Z4S-NTS1-SR48692
4.17Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
4.17Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
4.17Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
4.00Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
4.00Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
4.00Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
4.00Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
4.00Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
4.00Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
4.00Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.00Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
4.00Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
4.00Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
4.00Consensusneurotensin_onOrthosteric Ligandnts1_on
4.00Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
4.00Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
3.85Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
3.85Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
3.85Single7SHEPI; PE7SHE-GPR158-PI; PE
3.85Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
3.85Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.85Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
3.85Single8XQJJN2418XQJ-Apelin-JN241
3.85Single8XWACXCL18XWA-CXCR2-CXCL1
3.85Single8XWMCXCL68XWM-CXCR2-CXCL6
3.85Single8XWSCXCL58XWS-CXCR2-CXCL5
3.85Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
3.85Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
3.85Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
3.85Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
3.85Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
3.70Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
3.70Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
3.70Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
3.70Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
3.70Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
3.57Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
3.57Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
3.45Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
3.33Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7

Consensus Members
Id Members
7DHI 7DHI-β2-Salbutamol-Gs/β1/γ2
7XJI 7XJI-β3-Solabegron-Gs/β1/γ2
7JJO 7JJO-β1-Isoprenaline-Gs/β1/γ2
6NI3 6NI3-β2-BI167107-Gs/β1/γ2
8DCR 8DCR-β1-Dobutamine-Gs/β1/γ2
7XJH 7XJH-β3-Isoproterenol-Gs/β1/γ2
7DH5 7DH5-β3-Mirabegron-Gs/β1/γ2
Net Summary
Imin 3.02857
Number of Linked Nodes 888
Number of Links 1046
Number of Hubs 157
Number of Links mediated by Hubs 608
Number of Communities 23
Number of Nodes involved in Communities 200
Number of Links involved in Communities 282
Path Summary
Number Of Nodes in MetaPath 103
Number Of Links MetaPath 102
Number of Shortest Paths 4106044
Length Of Smallest Path 3
Average Path Length 44.6701
Length of Longest Path 73
Minimum Path Strength 0.357857
Average Path Strength 6.46469
Maximum Path Strength 20.8057
Minimum Path Correlation 0.7
Average Path Correlation 0.979802
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.51515
Average % Of Corr. Nodes 28.7087
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 38.1518
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
gs_aminegs_5ht
gs_adrenergic
gs_dopamine
gs_histamine
gs_trace-amine



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Download gs_adrenergic.zip



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