Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg Int. Strength Num Of Links Community ConSurf
1A:A:Y37 9.78254164
2A:A:H41 8.9425406
3A:A:N50 8.124579
4A:A:K53 5.12579
5A:A:Y63 5.44254179
6A:A:F219 6.835688
7A:A:F222 10.8325417
8A:A:K233 5.965619
9A:A:W234 5.616509
10A:A:C237 5.9925418
11A:A:F238 11.91419
12A:A:I245 4.594157
13A:A:V247 3.8475477
14A:A:D249 9.305478
15A:A:D252 9.6525478
16A:A:Y253 4.756508
17A:A:R265 10.7725479
18A:A:F273 5.63254189
19A:A:N278 6.14754118
20A:A:W281 8.65833615
21A:A:R283 7.14113
22A:A:I288 5.4125159
23A:A:F290 5.6865159
24A:A:N292 5.816579
25A:A:K293 7.02479
26A:A:Q294 6.248556
27A:A:E314 4.52254196
28A:A:F315 8.506506
29A:A:Y318 10.7975456
30A:A:P321 5.734555
31A:A:E330 7.216553
32A:A:D331 9.7375454
33A:A:V334 4.878554
34A:A:T335 7.01454
35A:A:K338 9.452555
36A:A:Y339 6.06833653
37A:A:F340 12.4625407
38A:A:R342 7.43554
39A:A:F345 8.045408
40A:A:R356 5.81254112
41A:A:H357 10.72254117
42A:A:C359 3.9854185
43A:A:Y360 8.2475408
44A:A:F363 8.96455
45A:A:R374 5.274204
46A:A:F376 7.72167688
47A:A:R380 9.265487
48A:A:R385 8.68685
49A:A:Y391 6.272564
50B:B:I18 4.3407
51B:B:V40 3.4325403
52B:B:R48 7.6875427
53B:B:L51 7.9375429
54B:B:H54 10.712529
55B:B:K57 10.698519
56B:B:Y59 9.53418
57B:B:M61 4.0175406
58B:B:W63 6.976527
59B:B:R68 9.87425
60B:B:L69 4.9775425
61B:B:L70 5.2025425
62B:B:V71 4.4275428
63B:B:S72 4.8075429
64B:B:Q75 10.2625419
65B:B:D76 6.6385169
66B:B:K78 4.92408
67B:B:L79 3.866527
68B:B:I80 9.3125428
69B:B:I81 5.035427
70B:B:W82 13.172529
71B:B:S84 4.08425
72B:B:K89 7.736529
73B:B:H91 5.185425
74B:B:L95 3.916528
75B:B:W99 8.92167619
76B:B:M101 5.98419
77B:B:Y105 3.905826
78B:B:Y111 5.83404
79B:B:N119 4.68419
80B:B:I123 3.6325416
81B:B:Y124 6.25526
82B:B:L126 4.0325425
83B:B:H142 9.5275419
84B:B:Y145 6.4818
85B:B:R150 5.474226
86B:B:F151 4.675619
87B:B:L152 3.615403
88B:B:I157 3.744517
89B:B:T159 4.202519
90B:B:D163 7.462519
91B:B:W169 9.77667618
92B:B:Q176 7.175414
93B:B:F180 7.786597
94B:B:H183 7.88333699
95B:B:M188 4.9575418
96B:B:L190 4.744225
97B:B:V200 6.394536
98B:B:D205 6.196599
99B:B:K209 11.8625496
100B:B:L210 4.08535
101B:B:W211 8.93833698
102B:B:Q220 7.0275437
103B:B:H225 8.67857739
104B:B:D228 8.855419
105B:B:I232 5.65438
106B:B:F234 7.07435
107B:B:F235 7.7345126
108B:B:P236 5.6554127
109B:B:N237 7.274505
110B:B:F241 7.052536
111B:B:T243 6.6775438
112B:B:D247 7.08439
113B:B:T249 6.2025436
114B:B:R251 7.4975838
115B:B:F253 6.62571736
116B:B:D254 6.8125129
117B:B:R256 11.12409
118B:B:Q259 3.85406
119B:B:Y264 6.34505
120B:B:H266 6.1175414
121B:B:I269 3.93514
122B:B:F278 7.7865127
123B:B:R283 9.0975409
124B:B:Y289 6.38286717
125B:B:D290 6.025416
126B:B:N295 7.51416
127B:B:W297 6.7475418
128B:B:R304 6.87515
129B:B:H311 9.0375419
130B:B:N313 5.08417
131B:B:R314 11.965618
132B:B:L318 3.735406
133B:B:T321 8.1475427
134B:B:M325 4.8325425
135B:B:V327 4.1825406
136B:B:T329 5.1925408
137B:B:W332 13.06619
138B:B:D333 7.454519
139B:B:K337 7.0725416
140B:B:W339 8.034519
141B:B:N340 7.515429
142G:G:L19 5.6409
143G:G:R27 8.445438
144G:G:D48 7.2625239
145G:G:L51 3.44606
146G:G:N59 6.542529
147G:G:P60 7.81429
148G:G:F61 5.46928
149L:L:R1 9.11254130
150L:L:E4 4.73440
151L:L:H9 5.554130
152L:L:W14 6.944500
153R:R:L187 3.8405
154R:R:Y191 5.05547
155R:R:Y195 5.79333647
156R:R:L202 3.995409
157R:R:F212 8.35407
158R:R:T218 5.64467
159R:R:R219 7.116569
160R:R:F230 8.866548
161R:R:R233 6.86571748
162R:R:I237 4.905447
163R:R:L244 4.7175405
164R:R:F288 6.492507
165R:R:Y290 6.1954109
166R:R:Y296 8.056547
167R:R:Y297 7.5654106
168R:R:W298 12.5865109
169R:R:L300 3.7675408
170R:R:V301 5.5775408
171R:R:E302 10.4625409
172R:R:Y305 8.81468
173R:R:L306 5.105469
174R:R:L309 10.125468
175R:R:F311 10.495466
176R:R:F315 10.765486
177R:R:W329 9.73754109
178R:R:P332 5.514109
179R:R:W339 6.172508
180R:R:R343 12.04754148
181R:R:D353 6.5675405
182R:R:K359 4.4265143
183R:R:K360 7.17754137
184R:R:W361 7.555138
185R:R:Q364 8.3354137
186R:R:I367 4.7325447
187R:R:F378 7.624569
188R:R:K388 7.67489
189R:R:F417 6.91833669
190R:R:H420 9.08167648
191R:R:Y421 11.0617648
192R:R:F424 7.196547
193R:R:M425 4.0225406
194R:R:Y429 7.5954136
195R:R:W437 7.0575405
196R:R:Y443 9.5875444
197R:R:N448 6.382546
198R:R:F450 5.57447
199R:R:Q451 8.16449
200R:R:I458 4.93408
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Int. Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.

Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1B:B:L69 B:B:R68 18.70453.64YesYes255
2B:B:S84 G:G:F61 17.98095.28YesYes258
3B:B:Y85 G:G:F61 17.95817.22NoYes248
4B:B:R68 B:B:Y85 20.088714.4YesNo254
5B:B:S84 B:B:W63 17.20684.94YesYes257
6B:B:M61 B:B:W63 20.00224.65YesYes067
7B:B:C317 B:B:M61 24.59874.86NoYes076
8B:B:C317 B:B:S316 24.9363.44NoNo079
9B:B:S316 B:B:W332 25.11334.94NoYes099
10B:B:N313 B:B:W332 79.19899.04YesYes179
11B:B:D333 B:B:N313 91.83424.04YesYes197
12B:B:D312 B:B:D333 99.898210.65NoYes059
13B:B:D312 R:R:R214 99.904919.06NoNo057
14R:R:E469 R:R:R214 99.91396.98NoNo097
15R:R:E469 R:R:F212 99.920916.32NoYes097
16R:R:F212 R:R:L215 99.94014.87YesNo079
17R:R:L215 R:R:V466 99.94595.96NoNo099
18R:R:I470 R:R:V466 99.96673.07NoNo059
19R:R:I208 R:R:I470 99.97122.94NoNo085
20R:R:I208 R:R:V204 99.98673.07NoNo085
21R:R:F461 R:R:V204 99.98993.93NoNo085
22R:R:F461 R:R:I457 99.99283.77NoNo086
23R:R:I457 R:R:I458 1002.94NoYes068
24R:R:I458 R:R:Y459 98.49987.25YesNo088
25R:R:L416 R:R:Y459 98.497414.07NoNo098
26R:R:E302 R:R:L416 80.09379.28YesNo099
27R:R:E302 R:R:H223 29.002211.08YesNo099
28A:A:Y391 R:R:H223 27.53733.27YesNo649
29R:R:F417 R:R:L416 23.02763.65YesNo099
30R:R:F417 R:R:L306 19.24373.65YesYes699
31A:A:Y391 R:R:L306 18.26868.21YesYes649
32A:A:L388 R:R:K388 33.13055.64NoYes089
33A:A:L388 R:R:L385 35.92394.15NoNo088
34A:A:L393 R:R:L385 38.88125.54NoNo088
35A:A:L393 A:A:Y391 39.17553.52NoYes084
36A:A:D378 A:A:Y360 20.197510.34NoYes078
37A:A:D381 A:A:Y360 21.030612.64NoYes088
38A:A:D381 R:R:K388 21.27885.53NoYes889
39B:B:K57 B:B:W332 67.001617.4YesYes199
40B:B:K57 B:B:Q75 20.634212.2YesYes199
41B:B:Q75 B:B:W99 20.22156.57YesYes199
42A:A:F238 B:B:W99 19.382914.03YesYes199
43A:A:F238 A:A:L44 23.695824.36YesNo099
44A:A:L44 A:A:L46 22.828311.07NoNo098
45A:A:F246 A:A:L46 22.61083.65NoNo098
46A:A:N292 A:A:T364 15.90045.85YesNo099
47A:A:F290 A:A:T364 16.52189.08YesNo099
48A:A:D378 A:A:H362 10.099111.35NoNo079
49B:B:L69 B:B:Y105 18.15023.52YesYes256
50B:B:C148 B:B:T102 13.76273.38NoNo068
51B:B:C149 B:B:T102 14.08963.38NoNo088
52B:B:C149 B:B:T159 14.25893.38NoYes089
53B:B:H142 B:B:T159 19.00984.11YesYes199
54B:B:K57 B:B:Y59 46.22367.17YesYes198
55B:B:H142 B:B:S161 25.644413.95YesNo199
56B:B:G162 B:B:S161 26.88563.71NoNo099
57B:B:G162 B:B:Y145 27.07210.14NoYes098
58A:A:W234 B:B:Y145 10.23915.79YesYes098
59B:B:M101 B:B:Y59 45.85329.58YesYes198
60B:B:M101 B:B:Y145 45.92955.99YesYes198
61A:A:K233 B:B:Y145 38.70253.58YesYes198
62A:A:K233 B:B:D228 19.00789.68YesYes199
63A:A:K233 B:B:D246 19.21235.53YesNo099
64A:A:F246 A:A:F273 22.3933.22NoYes099
65A:A:F273 A:A:F345 18.19158.57YesYes098
66A:A:F345 A:A:L270 17.45798.53YesNo086
67A:A:E344 A:A:L270 17.23176.63NoNo056
68A:A:E314 A:A:E344 16.7697.61YesNo1965
69A:A:E314 A:A:F340 16.32423.5YesYes067
70A:A:F340 A:A:Y318 10.454520.63YesYes076
71B:B:D290 B:B:R314 15.35827.15YesYes168
72B:B:D228 B:B:S227 18.9912.94YesNo096
73B:B:S227 B:B:S245 37.46613.26NoNo069
74B:B:H225 B:B:S245 33.72768.37YesNo399
75B:B:F253 B:B:H225 24.22053.39YesYes369
76B:B:F222 B:B:F253 16.548215NoYes386
77B:B:F222 B:B:Q220 16.20367.03NoYes387
78B:B:D258 B:B:Q220 12.836210.44NoYes377
79B:B:D258 G:G:R27 12.06248.34NoYes378
80B:B:I18 G:G:R27 11.29576.26YesYes078
81B:B:D246 B:B:S227 18.84895.89NoNo096
82B:B:W297 B:B:Y264 10.13238.68YesYes085
83B:B:C271 B:B:D290 18.42224.67NoYes156
84B:B:C271 B:B:Y289 15.90654.03NoYes157
85B:B:W297 B:B:Y289 10.96845.79YesYes187
86R:R:E302 R:R:L226 65.076511.93YesNo099
87R:R:F230 R:R:L226 35.19356.09YesNo089
88R:R:L226 R:R:S229 29.9054.5NoNo099
89R:R:N295 R:R:S229 28.5455.96NoNo089
90R:R:N295 R:R:R233 56.787813.26NoYes088
91R:R:F230 R:R:N295 28.59219.33YesNo088
92L:L:E4 R:R:R233 14.7353.49YesYes408
93R:R:R233 R:R:Y195 16.207812.35YesYes487
94L:L:E4 R:R:M445 14.81528.12YesNo006
95L:L:L7 R:R:M445 14.49945.65NoNo006
96L:L:L7 R:R:M441 14.18574.24NoNo006
97R:R:I237 R:R:R233 25.75533.76YesYes478
98R:R:F288 R:R:I237 13.02123.77YesYes077
99R:R:M441 R:R:W437 11.715515.12NoYes065
100R:R:F184 R:R:W437 10.59213.01NoYes065
101L:L:W14 R:R:F184 30.524410.02YesNo006
102L:L:W14 R:R:E180 19.782211.99YesNo003
103R:R:Y191 R:R:Y195 12.70183.97YesYes477
104R:R:D241 R:R:Y191 22.9446.9NoYes087
105R:R:D241 R:R:Y245 22.34888.05NoNo084
106L:L:R11 R:R:Y245 22.214531.9NoNo004
107L:L:R11 R:R:F184 21.01818.17NoNo006
108R:R:I237 R:R:Y191 12.65324.84YesYes477
109L:L:R21 R:R:E180 13.49812.33NoNo003
110L:L:D17 L:L:R21 12.610815.48NoNo000
111L:L:D17 L:L:R20 11.711810.72NoNo000
112L:L:R20 R:R:E35 10.81242.33NoNo005
113B:B:N313 B:B:R314 12.5924.82YesYes178
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1 Node2 LinkStrength Comm IsNode1Hub? IsNode2Hub? Node1Cons Node2Cons Node1Shell Node2Shell
L:L:R1 R:R:W361 7 13 Yes Yes 0 8 0 1
L:L:R1 R:R:Q364 4.67 13 Yes Yes 0 7 0 1
L:L:R1 R:R:Y429 15.43 13 Yes Yes 0 6 0 1
L:L:V2 R:R:I367 3.07 0 No Yes 0 7 0 1
L:L:A3 R:R:E444 6.03 0 No No 0 7 0 1
L:L:E4 R:R:Y195 3.37 4 Yes Yes 0 7 0 1
L:L:E4 R:R:R233 3.49 4 Yes Yes 0 8 0 1
L:L:E4 R:R:M445 8.12 4 Yes No 0 6 0 1
L:L:E4 R:R:N448 3.94 4 Yes Yes 0 6 0 1
L:L:I5 R:R:Q364 8.23 0 No Yes 0 7 0 1
L:L:Q6 R:R:Y429 4.51 13 No Yes 0 6 0 1
L:L:L7 R:R:M441 4.24 0 No No 0 6 0 1
L:L:L7 R:R:M445 5.65 0 No No 0 6 0 1
L:L:M8 R:R:V285 3.04 0 No No 0 6 0 1
L:L:M8 R:R:F288 3.73 0 No Yes 0 7 0 1
L:L:M8 R:R:D353 4.16 0 No Yes 0 5 0 1
L:L:H9 R:R:S355 8.37 13 Yes No 0 7 0 1
L:L:H9 R:R:K360 3.93 13 Yes Yes 0 7 0 1
L:L:H9 R:R:Y429 3.27 13 Yes Yes 0 6 0 1
L:L:R11 R:R:F184 18.17 0 No No 0 6 0 1
L:L:R11 R:R:Y245 31.9 0 No No 0 4 0 1
L:L:A12 R:R:D353 4.63 0 No Yes 0 5 0 1
L:L:A12 R:R:L354 3.15 0 No No 0 5 0 1
L:L:W14 R:R:E180 11.99 0 Yes No 0 3 0 1
L:L:W14 R:R:R181 4 0 Yes No 0 3 0 1
L:L:W14 R:R:F184 10.02 0 Yes No 0 6 0 1
L:L:R19 R:R:T33 6.47 0 No No 0 7 0 1
L:L:F23 R:R:E36 7 0 No No 0 6 0 1
L:L:L27 R:R:F39 7.31 0 No No 0 7 0 1
L:L:I31 R:R:R43 3.76 0 No No 0 4 0 1
R:R:K34 R:R:M32 11.52 0 No No 4 6 2 1
R:R:F39 R:R:L40 3.65 0 No No 7 5 1 2
R:R:Q47 R:R:R43 5.84 0 No No 6 4 2 1
R:R:R181 R:R:T178 9.06 0 No No 3 3 1 2
R:R:E180 R:R:V432 4.28 0 No No 3 5 1 1
R:R:F184 R:R:W437 3.01 0 No Yes 6 5 1 2
R:R:L187 R:R:M441 5.65 0 Yes No 5 6 2 1
R:R:Y191 R:R:Y195 3.97 4 Yes Yes 7 7 2 1
R:R:I237 R:R:Y191 4.84 4 Yes Yes 7 7 2 2
R:R:D241 R:R:Y191 6.9 0 No Yes 8 7 2 2
R:R:R233 R:R:Y195 12.35 4 Yes Yes 8 7 1 1
R:R:A234 R:R:Y195 4 0 No Yes 8 7 2 1
R:R:I237 R:R:Y195 7.25 4 Yes Yes 7 7 2 1
R:R:S449 R:R:Y195 3.82 4 No Yes 9 7 2 1
R:R:I237 R:R:R233 3.76 4 Yes Yes 7 8 2 1
R:R:L292 R:R:R233 7.29 0 No Yes 6 8 2 1
R:R:N295 R:R:R233 13.26 0 No Yes 8 8 2 1
R:R:R233 R:R:Y421 3.09 4 Yes Yes 8 8 1 2
R:R:N448 R:R:R233 4.82 4 Yes Yes 6 8 1 1
R:R:F288 R:R:S236 3.96 0 Yes No 7 7 1 2
R:R:F288 R:R:I237 3.77 0 Yes Yes 7 7 1 2
R:R:K240 R:R:L244 4.23 0 No Yes 7 5 2 2
R:R:F288 R:R:K240 16.13 0 Yes No 7 7 1 2
R:R:D241 R:R:Y245 8.05 0 No No 8 4 2 1
R:R:L244 R:R:Y245 3.52 0 Yes No 5 4 2 1
R:R:L244 R:R:V285 2.98 0 Yes No 5 6 2 1
R:R:D353 R:R:L244 8.14 0 Yes Yes 5 5 1 2
R:R:L289 R:R:V285 2.98 0 No No 7 6 2 1
R:R:F288 R:R:L289 4.87 0 Yes No 7 7 1 2
R:R:L292 R:R:Y296 5.86 0 No Yes 6 7 2 2
R:R:A293 R:R:I367 3.25 0 No Yes 6 7 2 1
R:R:I367 R:R:Y296 9.67 4 Yes Yes 7 7 1 2
R:R:I371 R:R:Y296 6.04 4 No Yes 7 7 2 2
R:R:Y296 R:R:Y421 14.89 4 Yes Yes 7 8 2 2
R:R:C351 R:R:D353 9.34 0 No Yes 9 5 2 1
R:R:N358 R:R:W361 6.78 0 No Yes 4 8 2 1
R:R:K360 R:R:W361 8.12 13 Yes Yes 7 8 1 1
R:R:K360 R:R:Q364 9.49 13 Yes Yes 7 7 1 1
R:R:K360 R:R:Y429 7.17 13 Yes Yes 7 6 1 1
R:R:Q364 R:R:W361 10.95 13 Yes Yes 7 8 1 1
R:R:V365 R:R:W361 4.9 0 No Yes 5 8 2 1
R:R:I367 R:R:I371 2.94 4 Yes No 7 7 1 2
R:R:I371 R:R:Y421 4.84 4 No Yes 7 8 2 2
R:R:H420 R:R:Y421 22.87 4 Yes Yes 8 8 2 2
R:R:H420 R:R:N448 5.1 4 Yes Yes 8 6 2 1
R:R:N448 R:R:Y421 12.79 4 Yes Yes 6 8 1 2
R:R:E444 R:R:F424 8.16 0 No Yes 7 7 1 2
R:R:E431 R:R:V432 7.13 0 No No 3 5 2 1
R:R:M441 R:R:W437 15.12 0 No Yes 6 5 1 2
R:R:E444 R:R:N448 5.26 0 No Yes 7 6 1 1
L:L:Q10 R:R:V432 2.87 0 No No 0 5 0 1
L:L:R20 R:R:E35 2.33 0 No No 0 5 0 1
L:L:R21 R:R:E180 2.33 0 No No 0 3 0 1
R:R:E35 R:R:F39 2.33 0 No No 5 7 1 1
R:R:M32 R:R:T33 1.51 0 No No 6 7 1 1
L:L:Q16 R:R:M32 1.36 0 No No 0 6 0 1
L:L:R11 R:R:D185 1.19 0 No No 0 2 0 1

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
70.83Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
66.67Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
66.67Single8YFOAc-LA-PTH Analog8YFO-PTH1-Ac-LA-PTH Analog-chim(NtGi1-Gs)/β1/γ2
63.33Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
62.96Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
62.07Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
60.71Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
60.71Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
60.00Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
59.26Single6FJ3PTH6FJ3-PTH1-PTH
58.06Single7Y36PTH7Y36-PTH1-PTH-Gs/β1/γ2
56.67Single8FLULA-PTH Analog8FLU-PTH1-LA-PTH Analog-Gs/β1/γ2
56.25Consensuspth_onOrthosteric Ligandpth1_on pth2_on
55.17Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
54.29Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
53.85Single9B5YLA-PTH Analog9B5Y-PTH1-LA-PTH Analog-chim(NtGi1-Gq)/β1/γ2
53.85Single9LXRLA-PTH Analog9LXR-PTH1-LA-PTH Analog-Arrestin2
53.57Single6NBFLA-PTH Analog6NBF-PTH1-LA-PTH Analog-Gs/β1/γ2
53.57Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
53.57Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
53.12Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
51.72Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
51.72Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
51.52Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
50.00Single6NBHLA-PTH Analog6NBH-PTH1-LA-PTH Analog-Gs/β1/γ2
50.00Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
50.00Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
50.00Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
50.00Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
50.00Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Single9P93VIP9P93-PAC1-VIP-Gs/β1/γ2
50.00Consensuscalcitonin_onOrthosteric Ligandctlike_on
48.57Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
48.28Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
48.28Single9P92VIP9P92-PAC1-VIP-Gs/β1/γ2
46.67Single9P94PACAP279P94-PAC1-PACAP27-Gs/β1/γ2
46.43Single6M1IPACAP276M1I-PAC1-PACAP27-Gs/β1/γ2
46.43Single6NIYCalcitonin-16NIY-CT-Calcitonin-1-Gs/β1/γ2
45.16Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
45.16Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
45.16Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
44.83Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
44.83Single9E2AGLP-19E2A-GLP-1-GLP-1-Gs/β1/γ2
44.12Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
44.12Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
43.75Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
43.75Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
43.59Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
43.33Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
43.33Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
43.33Single9BLBCagrilintide (non-acylated)9BLB-CT-Cagrilintide (non-acylated)-Gs/β1/γ2
43.33Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
42.86Single6VN7PACAP276VN7-VPAC1-PACAP27-Gs/β1/γ2
42.42Single6LPBPACAP276LPB-PAC1-PACAP27-Gs/β1/γ1
41.94Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
41.94Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
41.94Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
41.94Single7S1MExendin-4-D-Ala7S1M-GLP-1-Exendin-4-D-Ala-Gs/β1/γ2
41.38Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
41.38Single9BLCCagrilintide (non-acylated)9BLC-CT-Cagrilintide (non-acylated)-Gs/β1/γ2
41.38Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
40.74Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
40.62Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
40.62Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
40.62Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
40.62Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
40.62Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
40.62Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
40.00Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
40.00Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
40.00Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
40.00Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
40.00Consensuspac_onOrthosteric Ligandpac1_on
40.00Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
39.39Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
39.39Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
38.89Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
38.71Single6NBILA-PTH Analog6NBI-PTH1-LA-PTH Analog-Gs/β1/γ2
38.71Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
38.71Single7VABTirzepatide (non-acylated)7VAB-GIP-Tirzepatide (non-acylated)-chim(NtGi1-Gs)/β1/γ2
38.71Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
38.71Single9BLWCagrilintide (non-acylated)9BLW-CT (AMY1)-Cagrilintide (non-acylated)-Gs/β1/γ2; RAMP1
38.71Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
38.71Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
38.71Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
38.71Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
38.24Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
38.24Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
38.24Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
37.93Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
37.93Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
37.93Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
37.50Single6P9XCorticoliberin-16P9X-CRF1-Corticoliberin-1-Gs/β1/γ2
37.50Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
37.50Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
37.50Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
37.50Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
37.14Single6WPWZP37806WPW-Glucagon-ZP3780-Gs/β1/γ2
37.14Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
36.84Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
36.67Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
36.67Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
36.67Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
36.67Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
36.67Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
36.67Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
36.67Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
36.36Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
36.36Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
36.36Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
36.11Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
35.71Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
35.71Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
35.71Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
35.48Single5YQZNNC17025YQZ-Glucagon-NNC1702
35.48Single7TYHCalcitonin7TYH-CT (AMY2)-Calcitonin-Gs/β1/γ2; RAMP2
35.29Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
34.48Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
34.48Single7VBITirzepatide (non-acylated)7VBI-GLP-1-Tirzepatide (non-acylated)-Gs/β1/γ2
34.38Single6P9YPACAP276P9Y-PAC1-PACAP27-Gs/β1/γ2
34.38Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
34.38Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
34.29Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
33.33Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
33.33Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
33.33Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
33.33Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
33.33Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
33.33Single8FU6ZP37808FU6-Glucagon-ZP3780-Gs/β1/γ2
33.33Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
33.33Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
33.33Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
33.33Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
33.33Consensusglp_onOrthosteric Ligandglp1_on glp2_on
33.33Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
32.50Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
32.43Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
32.35Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
32.35Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
32.35Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
32.35Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
32.35Consensuspth1_onOrthosteric Ligand6NBF-PTH1-LA-PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-PTH-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
32.35Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
32.35Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
32.26Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
32.14Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
31.71Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
31.25Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
30.30Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
30.30Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
30.00Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
29.73Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
29.73Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-LA-PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-PTH-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
29.63Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
29.41Single7AD3Alpha-factor mating pheromone7AD3-STE2; STE2-α-factor mating pheromone-Gi1/STE4/γ2
29.03Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
29.03Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
29.03Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
29.03Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
27.78Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-CCL3-Gi1/β1/γ2
27.59Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
27.50Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
27.27Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
27.27Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
27.27Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
27.27Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-CXCL8-Gi1/β1/γ2 6LFM-CXCR2-CXCL8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-CCL3-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
26.92Single8ZRKGSK12922638ZRK-GPR119-GSK1292263-Gs/β1/γ2
26.92Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
26.92Single9KO4CCL219KO4-CCR7-CCL21-Gi1/β1/γ2
26.67Single4XT1CX3CL14XT1-US28-CX3CL1
26.67Single9L3YChemerin9L3Y-CML2-Chemerin-Gi1/β1/γ2
26.47Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
26.47Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
26.47Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-CCL3-Gi1/β1/γ2
26.47Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
26.47Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
25.93Single9L16CCL219L16-CCR7-CCL21
25.93Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
25.81Single7RKMCX3CL17RKM-US28-CX3CL1-Gi1/β1/γ2
25.81Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
25.71Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
25.71Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
25.71Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
25.71Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
25.00Single5U09Taranabant5U09-CB1-Taranabant
25.00Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
25.00Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
25.00Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
25.00Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
25.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
25.00Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
25.00Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
25.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
24.32Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
24.32Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
24.24Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
24.24Single8WSTMCH8WST-MCH2-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.14Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
24.14Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
24.14Single7Y27Somatostatin-147Y27-SST2-Somatostatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.14Single7Y65C5a (C-terminal peptide)7Y65-C5a1-C5a (C-terminal peptide)-Gi1/β1/γ2
24.14Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
24.14Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
24.00Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
24.00Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
24.00Single9ASBCa; Ca; Cyclomethyltryptophan; R-568; PO49ASB-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; R-568; PO49AXF-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
23.81Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
23.68Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Exendin-4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Tirzepatide (non-acylated)-Gs/β1/γ2
23.53Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
23.53Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
23.53Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
23.33Single4UG2CGS216804UG2-A2A-CGS21680
23.33Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
23.33Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
23.33Single8QJ2pN1628QJ2-MC4-pN162-Gs/β1/γ2
23.33Single9KZ2EP679KZ2-C3aB-EP67-Go/β1/γ2
23.33Single9UMJEP549UMJ-C3aB-EP54-Go/β1/γ2
23.08Single5TGZAM65385TGZ-CB1-AM6538
23.08Single9AVGCa; Ca; Cyclomethyltryptophan; R-568; PO49AVG-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs)/β1/γ2
23.08Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Exendin-4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Tirzepatide (non-acylated)-Gs/β1/γ2
22.86Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
22.86Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-C5a-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a-Gi1/β1/γ2 7Y64-C5a1-C5a-Gi1/β1/γ2
22.86Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
22.86Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
22.73Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS; CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
22.58Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
22.58Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
22.58Single7QA8Antagonist Peptide7QA8-STE2; STE2-Antagonist Peptide
22.58Single7QA8Antagonist Peptide7QA8-STE2; STE2-Antagonist Peptide
22.58Single9KWGC5a9KWG-C5a1-C5a-Go/β1/γ2
22.58Single9UYJChemerin-99UYJ-CML2-Chemerin-9-Arrestin2
22.58Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
22.58Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
22.50Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
22.22Single5N2RPSB365N2R-A2A-PSB36-Na
22.22Single5N2SPSB365N2S-A1-PSB36
22.22Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
22.22Single7EPFNAM5977EPF-mGlu2-NAM597
22.22Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
22.22Single8TF5Oleic acid8TF5-GPR6-Oleic acid
22.22Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
22.22Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9AVLCa; Ca; Cyclomethyltryptophan; R-568; PO49AVL-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-Gi3/β2/γ2
22.22Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; R-568; PO49AXF-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9B9ZMRI-18679B9Z-CB1-MRI-1867
22.22Single9KPFSalicin9KPF-TAS2R16-Salicin-Gi1/β1/γ2
22.22Consensusadenosine_offOrthosteric Liganda1_off a2_off
22.22Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
22.22Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
22.22Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
21.88Single3QAKUK-4320973QAK-A2A-UK-432097
21.88Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
21.88Single7F1QCCL37F1Q-CCR5-CCL3-Gi1/β1/γ2
21.88Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
21.88Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
21.88Single7XNACYN1548067XNA-SST2-CYN154806
21.88Single8JZZC5a-des-Arg8JZZ-C5a1-C5a-des-Arg-Go/β1/γ2
21.88Single8WSSMCH8WSS-MCH1-MCH-Gi1/β1/γ1
21.88Single8Z7JJN241-98Z7J-Apelin-JN241-9-Gi1/β1/γ2
21.88Single9JFK(Pen5)-Urotensin II9JFK-UT-(Pen5)-Urotensin II-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.88Single9KV6TLQP219KV6-C3aB-TLQP21-Go/β1/γ2
21.88Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
21.88Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
21.74Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-PubChem 25101223-Gi1/β1/γ2
21.43Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
21.43Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
21.43Single5XRAAM115425XRA-CB1-AM11542
21.43Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
21.43Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
21.43Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
21.43Single7PX4PSB-21137PX4-A2A-PSB-2113
21.43Single8FN1Neurotensin-(8-13)8FN1-NTS1-Neurotensin-(8-13)-chim(NtGi1-Go)/β1/γ2
21.43Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
21.43Single8I9LC3a8I9L-C3aB-C3a-Go/β1/γ2
21.43Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
21.43Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
21.43Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; R-568; PO49AYF-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4-Gi1/β1/γ2
21.43Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
21.43Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
21.43Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
21.43Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
21.21Single3OE0CVX153OE0-CXCR4-CVX15
21.21Single5WF5UK-4320975WF5-A2A-UK-432097
21.21Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
21.21Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
21.21Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.21Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
21.21Single9MEUCXCL129MEU-CXCR4-CXCL12
21.21Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
21.21Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
21.05Single5GLHEndothelin-15GLH-ETB-Endothelin-1
21.05Single6IGKEndothelin-36IGK-ETB-Endothelin-3
20.83Single3OE9IT1t3OE9-CXCR4-IT1t
20.83Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS; CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS; CaS-Ca-Ca; Tryptophan; '6218; PO4
20.69Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
20.69Single4XEENeurotensin-(8-13)4XEE-NTS1-Neurotensin-(8-13)
20.69Single4XESNeurotensin-(8-13)4XES-NTS1-Neurotensin-(8-13)
20.69Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
20.69Single6YVRNeurotensin-(6-13)6YVR-NTS1-Neurotensin-(6-13)
20.69Single7EPENAM5637EPE-mGlu2-NAM563
20.69Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
20.69Single7K15MKD0467K15-BLT1-MKD046-Na
20.69Single7L0SNeurotensin-(8-13)7L0S-NTS1-Neurotensin-(8-13)-Gi1/β1/γ1
20.69Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
20.69Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
20.69Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
20.69Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
20.69Single8ID9Icosapent8ID9-FFA4-Icosapent-Gi1/β1/γ2
20.69Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
20.69Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
20.69Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
20.69Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
20.69Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
20.69Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
20.69Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
20.69Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
20.69Consensuslpa_offOrthosteric Ligandlpa1_off
20.69Consensuslpl_offOrthosteric Ligands1p_off lpa_off
20.69Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
20.69Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
20.59Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
20.59Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
20.59Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
20.59Single8X8LCortistatin-148X8L-SST5-Cortistatin-14-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.59Single8XZJWN3538XZJ-Apelin; Apelin-WN353-Gi1/β1/γ2
20.59Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
20.59Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
20.59Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
20.59Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
20.59Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
20.59Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
20.59Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
20.00Single4BUONeurotensin-(8-13)4BUO-NTS1-Neurotensin-(8-13)
20.00Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
20.00Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
20.00Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
20.00Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
20.00Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
20.00Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
20.00Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
20.00Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
20.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
20.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
20.00Single7M3FCa; Ca; Tryptophan; Cinacalcet7M3F-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet
20.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; R-568; PO47SIL-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4
20.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; R-568; PO47SIL-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4
20.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
20.00Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
20.00Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
20.00Single7Y64C5a7Y64-C5a1-C5a-Gi1/β1/γ2
20.00Single8E0GBU728E0G-μ-BU72
20.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
20.00Single8HK5C5a8HK5-C5a1-C5a-Gi1/β1/γ2
20.00Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
20.00Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
20.00Single8IA2C5a8IA2-C5a1-C5a-Go/β1/γ2
20.00Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
20.00Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
20.00Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
20.00Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
20.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS; CaS-Tryptophan; Cinacalcet; PO4; Ca
20.00Single8WRZAM8418WRZ-CB1-AM841-Arrestin2
20.00Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
20.00Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
20.00Single8XVUCXCL28XVU-CXCR2-CXCL2
20.00Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
20.00Single9AVLCa; Ca; Cyclomethyltryptophan; R-568; PO49AVL-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-Gi3/β2/γ2
20.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS; CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
20.00Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
20.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
20.00Single9JFYNeuropeptide-SF9JFY-NPFF2-Neuropeptide-SF-Gi1/β1/γ2
20.00Single9JKXAcifran9JKX-HCA3-Acifran-Gi1/β1/γ2
20.00Single9KUGEP679KUG-C5a1-EP67-Go/β1/γ2
20.00Single9KWXC5a-des-Arg9KWX-C5a1-C5a-des-Arg-Go/β1/γ2
20.00Single9UYMChemerin-99UYM-CML2-Chemerin-9-chim(Arrestin3-CtArrestin2)
20.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.00Consensuscck_onOrthosteric Ligandccka_on cckb_on
20.00Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
20.00Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
20.00Consensusgi_apelinOrthosteric Ligand8XZH-Apelin; Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin; Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin; Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin; Apelin-Apelin-13-Gi1/β1/γ2
20.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM-5541-Gi1/β1/γ2 7EW2-S1P3-FTY720-P-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
20.00Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
20.00Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-14-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.44Single4XT3CX3CL14XT3-US28-CX3CL1
19.44Single7SK3CXCL127SK3-ACKR3-CXCL12
19.44Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
19.44Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
19.44Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
19.44Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
19.35Single3NY9PubChem 9131033NY9-β2-PubChem 913103
19.35Single5WF6UK-4320975WF6-A2A-UK-432097
19.35Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
19.35Single7RKFCX3CL17RKF-US28-CX3CL1-GDP-chim(NtGi1-G11)/β1/γ2
19.35Single7RKNCX3CL17RKN-US28-CX3CL1-Gi1/β1/γ2
19.35Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
19.35Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
19.35Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
19.35Single9KZ8EP679KZ8-C3aB-EP67-Go/β1/γ2
19.35Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
19.35Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
19.35Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Sulfated Gastrin-(10-17)-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
19.35Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
19.35Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
19.23Single2YDOAdenosine2YDO-A2A-Adenosine
19.23Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
19.23Single5IU7Q274563465IU7-A2A-Q27456346-Na
19.23Single5IUBQ274563445IUB-A2A-Q27456344-Na
19.23Single5JTBZM-2413855JTB-A2A-ZM-241385
19.23Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
19.23Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
19.23Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
19.23Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
19.23Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
19.23Single7AROLUF58337ARO-A2A-LUF5833-Na
19.23Single7T32ZM-2413857T32-A2A-ZM-241385
19.23Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
19.23Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
19.23Single8GURCP559408GUR-CB2-CP55940-Gi1/β1/γ2
19.23Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
19.23Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
19.23Single8JIMMonomethyl fumarate8JIM-HCA2-Monomethyl fumarate-Gi1/β1/γ2
19.23Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
19.23Single8K5CAcipimox8K5C-HCA2-Acipimox
19.23Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
19.23Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
19.23Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS; CaS-Tryptophan; Cinacalcet; PO4; Ca
19.23Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS; CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single9ASBCa; Ca; Cyclomethyltryptophan; R-568; PO49ASB-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single9AVGCa; Ca; Cyclomethyltryptophan; R-568; PO49AVG-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs)/β1/γ2
19.23Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
19.23Single9KPDSalicin9KPD-TAS2R16-Salicin-chim(Gs-CtGt3)/β1/γ2
19.23Single9KXSEP679KXS-C5a1-EP67-Go/β1/γ2
19.23Single9M2FNeuropeptide-FF9M2F-NPFF1-Neuropeptide-FF-Gi1/β1/γ2
19.23Single9P1TZM-2413859P1T-A2A-ZM-241385
19.23Consensusa2_offOrthosteric Liganda2a_off
19.23Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA47070-Na 5N2R-A2A-PSB36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-Etrumadenant-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-PubChem 984073-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
19.23Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-CXCL8-Gi1/β1/γ2
19.23Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
19.23Consensusgrh_offOrthosteric Ligandgnrh1_off
19.23Consensushca_onOrthosteric Ligandhca2_on
19.23Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
19.23Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
18.92Single7EIBKallidin-des-Arg107EIB-BK1-Kallidin-des-Arg10-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Single7QBCAlpha-factor mating pheromone7QBC-STE2; STE2-α-factor mating pheromone
18.92Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
18.92Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
18.92Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
18.92Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
18.92Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
18.92Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
18.75Single7F8XNN90567F8X-CCKA-NN9056
18.75Single7L0RNeurotensin-(8-13)7L0R-NTS1-Neurotensin-(8-13)-Gi1/β1/γ1
18.75Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
18.75Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
18.75Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
18.75Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
18.75Single8IEIPubChem 1347468948IEI-GPR156; GPR156-PubChem 134746894
18.75Single8IEPPubChem 1347468948IEP-GPR156; GPR156-PubChem 134746894
18.75Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
18.75Single8WDTphotoNECA8WDT-A2A-photoNECA
18.75Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
18.75Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
18.75Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs)/β1/γ2
18.75Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
18.75Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-C5-guano-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-DAMGO-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
18.75Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
18.75Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
18.75Consensussomatostatin_offOrthosteric Ligandsst2_off
18.52Single3EMLZM-2413853EML-A2A-ZM-241385
18.52Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
18.52Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
18.52Single5IU8Q274563475IU8-A2A-Q27456347-Na
18.52Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
18.52Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
18.52Single5UENDU1725UEN-A1-DU172
18.52Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
18.52Single6D27CAY104716D27-DP2-CAY10471
18.52Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
18.52Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
18.52Single6S0LZM-2413856S0L-A2A-ZM-241385
18.52Single6Z4VNeurotensin-(9-13)6Z4V-NTS1-Neurotensin-(9-13)
18.52Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
18.52Single7M3JNPS-2143; PO47M3J-CaS; CaS-NPS-2143; PO4
18.52Single7PYRPSB-21157PYR-A2A-PSB-2115
18.52Single7V3ZCP559407V3Z-CB1-CP55940
18.52Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
18.52Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
18.52Single8CU6LJ-45178CU6-A2A-LJ-4517
18.52Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
18.52Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
18.52Single8J6PNiacin8J6P-HCA2-Niacin-PubChem 25101223-Gi1/β1/γ2
18.52Single8JIINiacin8JII-HCA2-Niacin-PubChem 25101223-Gi1/β1/γ2
18.52Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
18.52Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
18.52Single9JQZGrapiprant 9JQZ-EP4-Grapiprant
18.52Single9KUXCMPD6449KUX-Apelin; Apelin-CMPD644-Arrestin2
18.52Single9P1SZM-2413859P1S-A2A-ZM-241385
18.52Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
18.52Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
18.52Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
18.52Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-Monomethyl fumarate-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
18.52Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-Monomethyl fumarate-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
18.52Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-Monomethyl fumarate-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
18.52Consensushca_on_gpOrthosteric Ligandhca2_on_gp
18.52Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
18.52Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
18.52Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
18.42Single7QBCAlpha-factor mating pheromone7QBC-STE2; STE2-α-factor mating pheromone
18.42Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
18.42Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
18.18Single6DO1(Sar1,Ile8)-Angiotensin II6DO1-AT1-(Sar1,Ile8)-Angiotensin II
18.18Single6HLOAprepitant6HLO-NK1-Aprepitant
18.18Single7SK5CXCL127SK5-ACKR3-CXCL12
18.18Single7XKEDehydroepiandrosterone7XKE-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
18.18Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
18.18Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
18.18Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
18.18Single9ME1CXCL129ME1-CXCR4-CXCL12
18.18Single9UMXEP549UMX-C5a1-EP54-Go/β1/γ2
18.18Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Sulfated Gastrin-(10-17)-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.18Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.18Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-Gi1/β1/γ2 7NA8-Ghrelin-Ibutamoren-Gi1/β1/γ2
18.18Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM-5541-Gi1/β1/γ2 7EW2-S1P3-FTY720-P-Gi1/β1/γ2
18.18Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
18.18Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
17.95Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.95Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.95Consensusbombesin_onOrthosteric Ligandbb2_on
17.95Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
17.95Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-1-Gs/β1/γ2
17.95Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
17.95Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
17.95Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
17.95Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
17.86Single5IUAQ274563485IUA-A2A-Q27456348-Na
17.86Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
17.86Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
17.86Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
17.86Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
17.86Single6KPCAM120336KPC-CB2-AM12033
17.86Single6LFMCXCL86LFM-CXCR2-CXCL8-Gi1/β1/γ2
17.86Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
17.86Single6S0QZM-2413856S0Q-A2A-ZM-241385
17.86Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
17.86Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
17.86Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
17.86Single7M3JNPS-2143; PO47M3J-CaS; CaS-NPS-2143; PO4
17.86Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
17.86Single7SINNPS-21437SIN-CaS; CaS-NPS-2143
17.86Single7SINNPS-21437SIN-CaS; CaS-NPS-2143
17.86Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
17.86Single7W41PD1762527W41-BB2-PD176252
17.86Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
17.86Single8GNEKW-63568GNE-A2A-KW-6356-Na
17.86Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
17.86Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
17.86Single8QOTNanobody-E8QOT-μ-Nanobody-E
17.86Single8S4DCMF-0198S4D-Apelin-CMF-019
17.86Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
17.86Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
17.86Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutamate-VU0155041-Gi3/β1/γ2
17.86Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
17.86Single8ZYTNeurotensin-(8-13)8ZYT-NTS1-Neurotensin-(8-13)-SBI-553-Arrestin2
17.86Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; R-568; PO49AYF-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4-Gi1/β1/γ2
17.86Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
17.86Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
17.86Single9EHSLUF76029EHS-A3A-LUF7602
17.86Single9JKSPubChem 442501769JKS-HCA3-PubChem 44250176-Gi1/β1/γ2
17.86Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
17.86Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
17.86Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
17.86Consensusblt_offOrthosteric Ligandblt1_off
17.86Consensusbombesin_offOrthosteric Ligandbb2_off
17.86Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-AM12033-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
17.86Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-AM12033-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
17.86Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-CXCL8-Gi1/β1/γ2
17.86Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
17.86Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
17.86Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
17.65Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
17.65Single6MEOGp160; CD46MEO-CCR5-Gp160; CD4
17.65Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.65Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
17.65Single8K6NNeuropeptide-Y8K6N-Y2-Neuropeptide-Y-Gi2/β1/γ1
17.65Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.65Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.65Single9UYIChemerin-99UYI-CML2-Chemerin-9-Arrestin2
17.65Consensusangiotensin_onOrthosteric Ligandat1_on
17.65Consensusat1_onOrthosteric Ligand7F6G-AT1-(Sar1)-Angiotensin II-Gq/β1/γ2
17.65Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Sulfated Gastrin-(10-17)-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.65Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
17.65Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-14-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
17.65Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
17.65Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
17.65Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
17.50Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
17.50Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
17.39Single8A2OTheophylline8A2O-A2A-Theophylline-Na
17.39Single8Y02All-trans-Retinal8Y02-OPN1SW-All-trans-Retinal-Gi1/β1/γ2
17.24Single2YDVNECA2YDV-A2A-NECA
17.24Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
17.24Single3ZEVNeurotensin-(7-13)3ZEV-NTS1-Neurotensin-(7-13)
17.24Single4BV0Neurotensin-(7-13)4BV0-NTS1-Neurotensin-(7-13)
17.24Single4UHRCGS216804UHR-A2A-CGS21680
17.24Single5G53NECA5G53-A2A-NECA-Gs
17.24Single5XR8AM120335XR8-CB1-AM12033
17.24Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
17.24Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
17.24Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
17.24Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
17.24Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
17.24Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
17.24Single7F1TCCL37F1T-CCR5-CCL3
17.24Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
17.24Single7L0PNeurotensin-(8-13)7L0P-NTS1-Neurotensin-(8-13)-Gi1/β1/γ1
17.24Single7L0QNeurotensin-(8-13)7L0Q-NTS1-Neurotensin-(8-13)-Gi1/β1/γ1
17.24Single7M8W15r-Methyl-PGD27M8W-DP2-15r-Methyl-PGD2-Na
17.24Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
17.24Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
17.24Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
17.24Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single7XOWSulfated Gastrin-(10-17)7XOW-CCKB-Sulfated Gastrin-(10-17)-chim(NtGi1-Gq)/β1/γ2
17.24Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
17.24Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
17.24Single8FMZNeurotensin-(8-13)8FMZ-NTS1-Neurotensin-(8-13)-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single8HQCC5a8HQC-C5a1-C5a-Go/β1/γ2
17.24Single8I2GPubChem 675302408I2G-FSH-FSH-PubChem 67530240-Gs/β1/γ2
17.24Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
17.24Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
17.24Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
17.24Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8UGWCGS216808UGW-A2A-CGS21680
17.24Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
17.24Single8WU1MDMB-Fubinaca8WU1-CB1-MDMB-Fubinaca-Arrestin2
17.24Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
17.24Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.24Single8XZICMF-0198XZI-Apelin; Apelin-CMF-019-Gi1/β1/γ2
17.24Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
17.24Single9IZGLPA9IZG-LPA1-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single9JCLADP9JCL-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
17.24Single9KVPSB2901579KVP-C3aB-SB290157-Go/β1/γ2
17.24Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
17.24Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-AM12033-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
17.24Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.24Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
17.24Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
17.24Consensuslpa_onOrthosteric Ligandlpa1_on
17.24Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
17.24Consensusneurotensin_onOrthosteric Ligandnts1_on
17.24Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-(8-13)-Gi1/β1/γ1
17.24Consensusrelaxin_onOrthosteric Ligandrxfp4_on
17.24Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
17.14Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
17.14Single6METGp160; CD46MET-CCR5-Gp160; CD4
17.14Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.14Single7F6G(Sar1)-Angiotensin II7F6G-AT1-(Sar1)-Angiotensin II-Gq/β1/γ2
17.14Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
17.14Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
17.14Single8IEDPubChem 1347468948IED-GPR156; GPR156-PubChem 134746894-Go/β1/γ2
17.14Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
17.14Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
17.14Consensusapelin_onOrthosteric Ligand8XZH-Apelin; Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin; Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin; Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin; Apelin-Apelin-13-Gi1/β1/γ2
17.14Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin; Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin; Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin; Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin; Apelin-Apelin-13-Gi1/β1/γ2
17.14Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-(Sar1)-Angiotensin II-Gq/β1/γ2
17.14Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-C5a-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a-Gi1/β1/γ2
17.14Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
17.14Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-(Sar1)-Angiotensin II-Gq/β1/γ2
17.14Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.14Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
17.14Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
17.14Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.14Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.14Consensusvasop-oxy_onOrthosteric Ligandv2_on
17.14Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
17.07Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-1-Gs/β1/γ2
17.07Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
16.67Single3OE6IT1t3OE6-CXCR4-IT1t
16.67Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
16.67Single4XNWMRS25004XNW-P2Y1-MRS2500
16.67Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
16.67Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
16.67Single6IIURamatroban6IIU-TXA2-Ramatroban
16.67Single6KQICP559406KQI-CB1-CP55940-Org27569
16.67Single6OS0Angiotensin II6OS0-AT1-Angiotensin II
16.67Single6OS2TRV0266OS2-AT1-TRV026
16.67Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
16.67Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
16.67Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
16.67Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS; CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
16.67Single7EO4Siponimod7EO4-S1P1-Siponimod-Gi1/β1/γ2
16.67Single7EW2FTY720-P7EW2-S1P3-FTY720-P-Gi1/β1/γ2
16.67Single7F9YGhrelin7F9Y-Ghrelin-Ghrelin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
16.67Single7QBIAlpha-factor mating pheromone7QBI-STE2; STE2-α-factor mating pheromone
16.67Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
16.67Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
16.67Single7W0LPubChem 1227019087W0L-Apelin; Apelin-PubChem 122701908-Gi1/β1/γ2
16.67Single7W0LPubChem 1227019087W0L-Apelin; Apelin-PubChem 122701908-Gi1/β1/γ2
16.67Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
16.67Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
16.67Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
16.67Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
16.67Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8HK2C3a8HK2-C3aB-C3a-Gi1/β1/γ2
16.67Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
16.67Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
16.67Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
16.67Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
16.67Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
16.67Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
16.67Single8U26Substance-P8U26-NK1-Substance-P-Gs/β1/γ2
16.67Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8XQEApelin-138XQE-Apelin; Apelin-Apelin-13-Gi1/β1/γ2
16.67Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
16.67Single8XWMCXCL68XWM-CXCR2-CXCL6
16.67Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.67Single8ZRTEndothelin-18ZRT-ETB-Endothelin-1
16.67Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
16.67Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
16.67Single9IJRC179IJR-GPR52-C17-Arrestin2
16.67Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
16.67Single9KT93,5-DHBA9KT9-HCA1-3,5-DHBA-Gi1/β1/γ2
16.67Single9KZKC3a (fragment)9KZK-C3aB-C3a (fragment)-Go/β1/γ2
16.67Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
16.67Single9M8POleic monoethanolamide9M8P-GPR3 ; GPR3-Oleic monoethanolamide-AF64394
16.67Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
16.67Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
16.67Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
16.67Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
16.67Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
16.67Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
16.67Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
16.67Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-(8-13)-Gi1/β1/γ1
16.67Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
16.67Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.67Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
16.67Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
16.67Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
16.67Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
16.67Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
16.67Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-(8-13)-Gi1/β1/γ1
16.67Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
16.67Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM-5541-Gi1/β1/γ2 7EW2-S1P3-FTY720-P-Gi1/β1/γ2
16.22Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
16.22Single7QBIAlpha-factor mating pheromone7QBI-STE2; STE2-α-factor mating pheromone
16.22Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
16.22Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
16.22Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
16.22Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
16.13Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
16.13Single7EZCUK-4320977EZC-A2A-UK-432097
16.13Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.13Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
16.13Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
16.13Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
16.13Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
16.13Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
16.13Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
16.13Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
16.13Single8FN0Neurotensin-(8-13)8FN0-NTS1-Neurotensin-(8-13)-SBI-553-chim(NtGi1-Go)/β1/γ2
16.13Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
16.13Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
16.13Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
16.13Single8JPFNeurotensin-(8-13)8JPF-NTS1-Neurotensin-(8-13)-SBI-553
16.13Single8XGSKisspeptin-18XGS-Kiss1-Kisspeptin-1-chim(NtGi1-Gq)/β1/γ2
16.13Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8XWFCXCL38XWF-CXCR2-CXCL3
16.13Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
16.13Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
16.13Single9IZFLPA9IZF-LPA1-LPA-Gi1/β1/γ2
16.13Single9KT8Acifran9KT8-HCA2-Acifran-Gi1/β1/γ2
16.13Single9KV8TLQP219KV8-C3aB-TLQP21-Go/β1/γ2
16.13Single9L79AR2314539L79-GPR119-AR231453-chim(NtGi1-Gs)/β1/γ2
16.13Single9M1HPGE29M1H-EP1-PGE2-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single9UYHChemerin-99UYH-CML2-Chemerin-9-Arrestin2
16.13Single9WP9S1P9WP9-S1P3-S1P-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.13Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.13Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
16.13Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
16.13Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
16.13Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
16.13Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
16.13Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single6LI0C176LI0-GPR52-C17
16.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
16.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS; CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
16.00Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
16.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
16.00Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
16.00Single8K5BNiacin8K5B-HCA2-Niacin
16.00Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
16.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
16.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
16.00Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
16.00Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
16.00Single9B9YTaranabant9B9Y-CB1-Taranabant
16.00Single9EPRAll-trans-Retinal9EPR-Rhodopsin-All-trans-Retinal-Gi1/β1/γ2
16.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
16.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
15.91Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.91Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
15.79Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
15.79Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
15.79Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
15.79Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
15.79Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
15.79Single8ZH8QRFP268ZH8-QRFP-QRFP26-Gq/β1/γ1
15.79Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
15.62Single5ZTYAM102575ZTY-CB2-AM10257
15.62Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
15.62Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
15.62Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
15.62Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
15.62Single7XN9L-0545227XN9-SST2-L-054522
15.62Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
15.62Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
15.62Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
15.62Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
15.62Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
15.62Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
15.62Single8XZFWN5618XZF-Apelin; Apelin-WN561-Gi1/β1/γ2
15.62Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
15.62Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
15.62Single9IPYJR14a9IPY-C3aB-JR14a
15.62Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
15.62Single9KX6C5a-des-Arg9KX6-C5a1-C5a-des-Arg-Go/β1/γ2
15.62Single9M0RNeuropeptide-VF9M0R-NPFF1-Neuropeptide-VF-Gi1/β1/γ2
15.62Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
15.62Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
15.62Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
15.62Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
15.62Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
15.38Single3ODUIT1t3ODU-CXCR4-IT1t
15.38Single3PWHZM-2413853PWH-A2A-ZM-241385
15.38Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
15.38Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
15.38Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
15.38Single4BWBNeurotensin-(8-12)4BWB-NTS1-Neurotensin-(8-12)
15.38Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
15.38Single4S0VSuvorexant4S0V-OX2-Suvorexant
15.38Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
15.38Single6IGLIRL16206IGL-ETB-IRL1620
15.38Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
15.38Single6TPJSuvorexant6TPJ-OX2-Suvorexant
15.38Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
15.38Single7BR3Elagolix7BR3-GnRH1-Elagolix
15.38Single7EJ0Norepinephrine7EJ0-α2a-Norepinephrine-Go/β1/γ2
15.38Single7F8ULintitript7F8U-CCKA-Lintitript
15.38Single7F8YDevazepide7F8Y-CCKA-Devazepide
15.38Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
15.38Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS; CaS-Ca; Ca; Tryptophan; NPS-2143
15.38Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS; CaS-Ca; Ca; Tryptophan; NPS-2143
15.38Single7M3FCa; Ca; Tryptophan; Cinacalcet7M3F-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet
15.38Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
15.38Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
15.38Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
15.38Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
15.38Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
15.38Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
15.38Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
15.38Single8IW4Spermidine8IW4-TAA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
15.38Single8IWESpermidine8IWE-TAA9-Spermidine
15.38Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
15.38Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
15.38Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
15.38Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
15.38Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
15.38Single8Y0HVUF114188Y0H-CXCR3-VUF11418
15.38Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
15.38Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.38Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
15.38Single8Z87CHBA8Z87-HCA1-CHBA-Gi1/β1/γ2
15.38Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS; CaS-Ca-Ca; Tryptophan; '6218; PO4
15.38Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
15.38Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
15.38Single9KO2CCL199KO2-CCR7-CCL19-Gi1/β1
15.38Single9KO6CCL199KO6-CCR7-CCL19
15.38Single9KPESalicin9KPE-TAS2R16-Salicin-Gi1/β1/γ2
15.38Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
15.38Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
15.38Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
15.38Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
15.38Consensusbradykinin_onOrthosteric Ligandbk2_on
15.38Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
15.38Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
15.38Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
15.38Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-CXCL8-Gi1/β1/γ2
15.38Consensusendothelin_onOrthosteric Ligandetb_on eta_on
15.38Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.38Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
15.38Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
15.38Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.38Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
15.38Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
15.38Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.38Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.15Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
15.15Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
15.15Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
15.15Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
15.15Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
15.15Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
15.15Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
15.15Single8IEBPubChem 1347468948IEB-GPR156; GPR156-PubChem 134746894
15.15Single8IEIPubChem 1347468948IEI-GPR156; GPR156-PubChem 134746894
15.15Single8IEPPubChem 1347468948IEP-GPR156; GPR156-PubChem 134746894
15.15Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
15.15Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
15.15Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.15Single8XWNCXCL88XWN-CXCR2-CXCL8
15.15Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
15.15Single9UMRC5a-pep9UMR-C5a1-C5a-pep-Go/β1/γ2
15.15Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
15.15Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
15.15Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
15.15Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
15.15Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
15.15Consensuslpl_onOrthosteric Ligands1p_on lpa_on
15.15Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
15.15Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
15.15Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-14-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.00Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
15.00Single8ZJETAK4488ZJE-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ1
14.81Single3UZCPubChem 1355666093UZC-A2A-PubChem 135566609
14.81Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
14.81Single5UVIZM-2413855UVI-A2A-ZM-241385
14.81Single6AQFZM-2413856AQF-A2A-ZM-241385
14.81Single6MH8ZM-2413856MH8-A2A-ZM-241385
14.81Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
14.81Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
14.81Single6TP3Nemorexant6TP3-OX1-Nemorexant
14.81Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
14.81Single6V9SGTPL114036V9S-OX1-GTPL11403
14.81Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
14.81Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
14.81Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
14.81Single7UTZDPPC7UTZ-TSH-TSH-DPPC-Gs/β1/γ2
14.81Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
14.81Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
14.81Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
14.81Single8IHKAcifran8IHK-HCA3-Acifran
14.81Single8JEIPubChem 117155568JEI-HCAR3-PubChem 11715556-Gi1/β1/γ2
14.81Single8K9KDAMGO8K9K-μ-DAMGO-Gi3/β1/γ1
14.81Single8PM2DMCHA8PM2-TA7-DMCHA-Gs/β1/γ2
14.81Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
14.81Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
14.81Single8Y01All-trans-Retinal8Y01-Opsin1MW-All-trans-Retinal-Gi1/β1/γ2
14.81Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
14.81Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
14.81Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
14.81Single9BA0MRI-18919BA0-CB1-MRI-1891
14.81Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
14.81Single9JKYAcifran9JKY-HCA2-Acifran-Gi1/β1/γ2
14.81Single9KUWCMPD6449KUW-Apelin; Apelin-CMPD644-Arrestin2 ; Arrestin2
14.81Single9L8LBI1671079L8L-β2-BI167107-Atazanavir-Gs/β1/γ2 ; Arrestin2
14.81Single9LKBPL459LKB-OR5V1-PL45-chim(NtGi1-Gs)/β1
14.81Single9PXXNaloxone9PXX-μ-Naloxone-GDPβS-Gi1/β1/γ2
14.81Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
14.81Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
14.81Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.71Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
14.71Single7W0NElabela7W0N-Apelin; Apelin-Elabela-Gi1/β1/γ2
14.71Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
14.71Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
14.71Single8IEBPubChem 1347468948IEB-GPR156; GPR156-PubChem 134746894
14.71Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
14.71Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
14.71Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
14.71Single9E82CXCL12 (fragment)9E82-ACKR3-CXCL12 (fragment)-Arrestin2
14.71Single9KT7MK68929KT7-HCA2-MK6892-Gi1/β1/γ2
14.71Single9L60Dynorphin9L60-κ-Dynorphin-MPAM-15-Gi1/β1/γ2
14.71Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
14.71Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
14.71Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
14.71Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
14.71Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
14.63Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
14.63Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
14.29Single2Y04Salbutamol2Y04-β1-Salbutamol
14.29Single4DAJTiotropium4DAJ-M3-Tiotropium
14.29Single4U16N-methyl-Scopolamine4U16-M3-N-methyl-Scopolamine
14.29Single4YAYZD-71554YAY-AT1-ZD-7155
14.29Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
14.29Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
14.29Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
14.29Single5T04Neurotensin-(8-13)5T04-NTS1-Neurotensin-(8-13)
14.29Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
14.29Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
14.29Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
14.29Single6IIVDaltroban6IIV-TXA2-Daltroban
14.29Single6KPFAM120336KPF-CB2-AM12033-Gi1/β1/γ2
14.29Single6PS1Timolol6PS1-β2-Timolol
14.29Single6TOTLemborexant6TOT-OX1-Lemborexant
14.29Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
14.29Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
14.29Single7F83PF-051904577F83-Ghrelin-PF-05190457
14.29Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
14.29Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
14.29Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
14.29Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
14.29Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
14.29Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
14.29Single7UL4Alvimopan7UL4-μ-Alvimopan
14.29Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
14.29Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.29Single7XJHIsoprenaline7XJH-β3-Isoprenaline-Gs/β1/γ2
14.29Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
14.29Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
14.29Single7YXAONO-54306087YXA-S1P5-ONO-5430608
14.29Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8IC0CXCL88IC0-CXCR1-CXCL8-Gi1/β1/γ2
14.29Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
14.29Single8JHNMonomethyl fumarate8JHN-HCA2-Monomethyl fumarate-Go/β1/γ2
14.29Single8K5DGSK2560738K5D-HCA2-GSK256073
14.29Single8T1WCVN4248T1W-GPR6-CVN424
14.29Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
14.29Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
14.29Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
14.29Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
14.29Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
14.29Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
14.29Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
14.29Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
14.29Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single8XZHMM078XZH-Apelin; Apelin-MM07-Gi1/β1/γ2
14.29Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
14.29Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
14.29Single8ZQEGPR15L(CT)8ZQE-GPR15-GPR15L(CT)-Gi1/β1/γ1
14.29Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
14.29Single8ZYYNeurotensin-(8-13)8ZYY-NTS1-Neurotensin-(8-13)-SBI-553-Arrestin2
14.29Single9AS1DMT9AS1-5-HT2A-DMT
14.29Single9B54VIP369B54-CB1-VIP36-Gi1/β1/γ2
14.29Single9CHXCarazolol9CHX-β2-Carazolol
14.29Single9H37PubChem 1756706469H37-A2A-PubChem 175670646-Na
14.29Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
14.29Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
14.29Single9M1ONeuropeptide-FF9M1O-NPFF2-Neuropeptide-FF-Gi1/β1/γ2
14.29Single9VMYTMU41429VMY-5-HT1A-TMU4142-Go/β1/γ2
14.29Consensusa3_onOrthosteric Liganda3a_on
14.29Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-C5a-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a-Gi1/β1/γ2
14.29Consensuscck_offOrthosteric Ligandccka_off
14.29Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
14.29Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-CXCL8-Gi1/β1/γ2
14.29Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
14.29Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.29Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.29Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.29Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.00Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
13.89Single7AD3Alpha-factor mating pheromone7AD3-STE2; STE2-α-factor mating pheromone-Gi1/STE4/γ2
13.89Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
13.89Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
13.89Single8IEDPubChem 1347468948IED-GPR156; GPR156-PubChem 134746894-Go/β1/γ2
13.89Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
13.89Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
13.89Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMIFL-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-TC-FPR 43-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
13.89Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
13.79Single2Y03Isoprenaline2Y03-β1-Isoprenaline
13.79Single4JKVTaladegib4JKV-SMO-Taladegib
13.79Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
13.79Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
13.79Single5C1MBU725C1M-μ-BU72
13.79Single5CGCHTL142425CGC-mGlu5-HTL14242
13.79Single5JQHCarazolol5JQH-β2-Carazolol
13.79Single5TVNLSD5TVN-5-HT2B-LSD
13.79Single5XPRBosentan5XPR-ETB-Bosentan
13.79Single6D26Fevipiprant6D26-DP2-Fevipiprant
13.79Single6LUQHaloperidol6LUQ-D2-Haloperidol
13.79Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
13.79Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
13.79Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
13.79Single6PS6Timolol6PS6-β2-Timolol
13.79Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
13.79Single6TP6Filorexant6TP6-OX1-Filorexant
13.79Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
13.79Single7C4SS1P7C4S-S1P3-S1P
13.79Single7C61Ergotamine7C61-5-HT1B-Ergotamine
13.79Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
13.79Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
13.79Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
13.79Single7WIGL-0542647WIG-SST2-L-054264-Gi1/β1/γ2
13.79Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
13.79Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
13.79Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
13.79Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
13.79Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
13.79Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
13.79Single8JXSPF-61428JXS-D1-PF-6142
13.79Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
13.79Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
13.79Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
13.79Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
13.79Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
13.79Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
13.79Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
13.79Single9IYBPGD29IYB-DP2-PGD2-A1D5Q-Gi1/β1/γ2
13.79Single9KT6Acifran9KT6-HCA3-Acifran-Gi1/β1/γ2
13.79Single9KUTJR14a9KUT-C3aB-JR14a-Go/β1/γ2
13.79Single9KUVCMPD6449KUV-Apelin-CMPD644-Arrestin2
13.79Single9L74S1P d16:19L74-S1P3-S1P d16:1-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single9M8POleic monoethanolamide9M8P-GPR3 ; GPR3-Oleic monoethanolamide-AF64394
13.79Single9PXYNaloxone9PXY-μ-Naloxone-GDPβS-Gi1/β1/γ2
13.79Consensusa3_on_gpOrthosteric Liganda3a_on_gp
13.79Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
13.79Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
13.79Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
13.79Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
13.79Consensusdp_offOrthosteric Liganddp2_off
13.79Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.79Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
13.79Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
13.79Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
13.79Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
13.79Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
13.79Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.79Consensusm2_offOrthosteric Ligand5ZKC-M2-N-methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
13.79Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
13.79Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
13.79Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
13.79Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-2-Phenylethylamine-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs)/β1/γ2
13.79Consensustrace-amine_onOrthosteric Ligandta1_on
13.64Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
13.51Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
13.51Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
13.51Single7P02Substance-P7P02-NK1-Substance-P-chim(NtGi1-Gs)/β1/γ2
13.51Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.51Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single3P0GBI1671073P0G-β2-BI167107
13.33Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
13.33Single4LDLHydroxybenzyl Isoproterenol4LDL-β2-Hydroxybenzyl Isoproterenol
13.33Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
13.33Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
13.33Single5V56TC1145V56-SMO-TC114
13.33Single5V57TC1145V57-SMO-TC114
13.33Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
13.33Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
13.33Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
13.33Single6H7JIsoprenaline6H7J-β1-Isoprenaline
13.33Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
13.33Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.33Single6WGTLSD6WGT-5-HT2A-LSD
13.33Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
13.33Single7B6WCyclazosin7B6W-α1b-Cyclazosin
13.33Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
13.33Single7FEECP559407FEE-CB1-CP55940-ZCZ011
13.33Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
13.33Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
13.33Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
13.33Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
13.33Single7TUYGSK682753A7TUY-GPR183-GSK682753A
13.33Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
13.33Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
13.33Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
13.33Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
13.33Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
13.33Single8EA0Iperoxo8EA0-M3-Iperoxo
13.33Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
13.33Single8HPTC5a (C-terminal peptide)8HPT-C5a1-C5a (C-terminal peptide)-Go/β1/γ2
13.33Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
13.33Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.33Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
13.33Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-PtdIns4P-Gi1/β1/γ2
13.33Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
13.33Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
13.33Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.33Single8JZPC5a8JZP-C5a1-C5a-Go/β1/γ2
13.33Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
13.33Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
13.33Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
13.33Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
13.33Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
13.33Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
13.33Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
13.33Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
13.33Single8ZWFJR14a8ZWF-C3aB-JR14a
13.33Single9AS9RS130-1809AS9-5-HT2A-RS130-180
13.33Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9B65MDMB-Fubinaca9B65-CB1-MDMB-Fubinaca-Gi1/β1/γ2
13.33Single9E9SPGD29E9S-DP1-PGD2-Gs/β1/γ1
13.33Single9EGOZ85267113509EGO-CB1-Z8526711350-Gi1/β1/γ2
13.33Single9I54PubChem 1764520919I54-D1-PubChem 176452091-Gs/β1/γ2
13.33Single9IK9Lanreotide9IK9-SST1-Lanreotide-Gi1/β1/γ2
13.33Single9KUXCMPD6449KUX-Apelin; Apelin-CMPD644-Arrestin2
13.33Single9MENGp120 (V3 loop)9MEN-CXCR4-Gp120 (V3 loop)
13.33Single9RHGC4079RHG-FZD7-C407
13.33Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9WSTDAMGO9WST-μ-DAMGO-chim(NtGi1-Gz)/β1/γ2
13.33Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
13.33Consensusa2_onOrthosteric Liganda2b_on
13.33Consensusa2_on_gpOrthosteric Liganda2b_on_gp
13.33Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
13.33Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
13.33Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.33Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
13.33Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
13.33Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
13.33Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
13.33Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.33Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.33Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-methyl-Scopolamine 5ZHP-M3-PubChem 134828589
13.33Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
13.33Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
13.33Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-2-Phenylethylamine-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs)/β1/γ2
13.33Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
13.16Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
13.16Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
13.16Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.16Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
13.04Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
13.04Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
13.04Single7XKDDehydroepiandrosterone7XKD-ADGRG2-Dehydroepiandrosterone-Gs/β1/γ2
13.04Single8PWNTheophylline8PWN-A2A-Theophylline
13.04Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.90Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
12.90Single4LDEBI1671074LDE-β2-BI167107
12.90Single4RWADIPP-NH24RWA-δ-DIPP-NH2
12.90Single5CXVTiotropium5CXV-M1-Tiotropium
12.90Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
12.90Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
12.90Single5X33BIIL2605X33-BLT1-BIIL260
12.90Single6AK3PGE26AK3-EP3-PGE2
12.90Single6CM4Risperidone6CM4-D2-Risperidone
12.90Single6MXTSalmeterol6MXT-β2-Salmeterol
12.90Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
12.90Single7DFPSpiperone7DFP-D2-Spiperone
12.90Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
12.90Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single7W0NElabela7W0N-Apelin; Apelin-Elabela-Gi1/β1/γ2
12.90Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
12.90Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.90Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
12.90Single7YITNalfurafine7YIT-κ-Nalfurafine
12.90Single8DWCBAM8-228DWC-MRGPRX1-BAM8-22-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-PtdIns4P-Gi1/β1/γ1
12.90Single8FYTLSD8FYT-5-HT1A-LSD-PtdIns4P-Gi1/β1/γ1
12.90Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
12.90Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8JJ8Arformoterol8JJ8-β2-Arformoterol
12.90Single8JJLOlodaterol8JJL-β2-Olodaterol
12.90Single8JJPChemerin-98JJP-CML2-Chemerin-9-Gi1/β1/γ2
12.90Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
12.90Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
12.90Single8XWACXCL18XWA-CXCR2-CXCL1
12.90Single8XWSCXCL58XWS-CXCR2-CXCL5
12.90Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
12.90Single8XYIVUF106618XYI-CXCR3-VUF10661
12.90Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
12.90Single9DGIZ85267113509DGI-CB1-Z8526711350
12.90Single9ECJS-geranylgeranyl-L-glutathione9ECJ-P2Y8-S-geranylgeranyl-L-glutathione-G13/β1/γ2
12.90Single9EK0Iperoxo9EK0-M5-Iperoxo-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
12.90Single9KVG5-MeO-DMT9KVG-5-HT1A-5-MeO-DMT-PtdIns4P-Gi1/β1/γ2
12.90Single9L3WChemerin9L3W-CML1-Chemerin-Gi1/β1/γ2
12.90Single9V6ONalfurafine9V6O-κ-Nalfurafine-Gi1/β1/γ2
12.90Single9VJ6F-155999VJ6-5-HT1A-F-15599-Gi3/β1/γ2
12.90Single9WSVDAMGO9WSV-μ-DAMGO-Arrestin2
12.90Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoprenaline-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
12.90Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoprenaline-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
12.90Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
12.90Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
12.90Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
12.90Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
12.90Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-C5-guano-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-DAMGO-Gi1/β1/γ2
12.90Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-C5-guano-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-DAMGO-Gi1/β1/γ2
12.90Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
12.90Consensusorexin_onOrthosteric Ligandox2_on
12.90Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.90Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.82Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
12.82Single9KDFRES-701-39KDF-ETB-RES-701-3
12.50Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
12.50Single3OE8IT1t3OE8-CXCR4-IT1t
12.50Single3RFMCaffeine3RFM-A2A-Caffeine
12.50Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
12.50Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
12.50Single5CGDHTL142425CGD-mGlu5-HTL14242
12.50Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
12.50Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
12.50Single5X93K-87945X93-ETB-K-8794
12.50Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
12.50Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
12.50Single6DDFDAMGO6DDF-μ-DAMGO-Gi1/β1/γ2
12.50Single6UP7Neurotensin-(8-13)6UP7-NTS1-Neurotensin-(8-13)-Arrestin2
12.50Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS; CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.50Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
12.50Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
12.50Single7UM4AS26747237UM4-5-HT5A-AS2674723
12.50Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
12.50Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
12.50Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
12.50Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
12.50Single8GAGZ85267113508GAG-CB1-Z8526711350-Gi1/β1/γ2
12.50Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
12.50Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
12.50Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8IY6Endothelin-18IY6-ETB-Endothelin-1
12.50Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
12.50Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
12.50Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
12.50Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
12.50Single8Z8ALactate8Z8A-HCA1-Lactate-Gi1/β1/γ2
12.50Single8ZPLHF511168ZPL-CXCR4-HF51116
12.50Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
12.50Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
12.50Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
12.50Single9M54Neuropeptide-VF9M54-NPFF2-Neuropeptide-VF-Gi1/β1/γ2
12.50Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
12.50Consensusendothelin_offOrthosteric Ligandetb_off
12.50Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
12.50Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
12.50Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
12.50Consensusp2y_offOrthosteric Ligandp2y1_off
12.50Consensusprostanoid_offOrthosteric Ligandep_off dp_off
12.20Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
12.12Single5VBLAMG3054 5VBL-Apelin-AMG3054
12.12Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
12.12Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
12.12Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
12.12Single6PT3DPI-2876PT3-δ-DPI-287
12.12Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
12.12Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
12.12Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8XQJJN2418XQJ-Apelin; Apelin-JN241
12.12Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
12.12Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
12.12Single9JF4PD1683689JF4-BB1-PD168368
12.12Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.12Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
12.00Single6PWCNeurotensin-(9-13)6PWC-NTS1-Neurotensin-(9-13)-Arrestin2
12.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
12.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
12.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
12.00Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
12.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
12.00Single8ITFDMCHA8ITF-TAA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
12.00Single8IU2All-trans-Retinal8IU2-Opsin1LW-All-trans-Retinal-Gi1/β1/γ2
12.00Single8J6QPubChem 251012238J6Q-HCA2-β-Hydroxybutyrate-PubChem 25101223-Gi1/β1/γ2
12.00Single8JEFPubChem 113671668JEF-HCA3-PubChem 11367166-Gi1/β1/γ2
12.00Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
12.00Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
12.00Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
12.00Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
12.00Single9JG1Adriforant9JG1-H4-Adriforant
12.00Single9LRCHistamine9LRC-H4-Histamine
12.00Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
12.00Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-All-trans-Retinal-Gi1/β1/γ2
12.00Consensusgi_sensoryOrthosteric Ligandgi_opsins
12.00Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.00Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.00Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-All-trans-Retinal-Gi1/β1/γ2
12.00Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-All-trans-Retinal-Gi1/β1/γ2
11.90Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
11.90Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
11.76Single4IARErgotamine4IAR-5-HT1B-Ergotamine
11.76Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
11.76Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
11.76Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
11.76Single7NA7Ghrelin7NA7-Ghrelin-Ghrelin-Gi1/β1/γ2
11.76Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
11.76Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.76Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single8DWGBAM8-228DWG-MRGPRX1-BAM8-22-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.76Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.76Single8KIGSHU91198KIG-MC3-SHU9119-Ca
11.76Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
11.76Single8WKYPG-9348WKY-MC4-PG-934
11.76Single8XBHPubChem 1626566368XBH-GPR34-PubChem 162656636-Gi1/β1/γ2
11.76Single9MEJGp1209MEJ-CXCR4-Gp120
11.76Single9UYLChemerin-99UYL-CML2-Chemerin-9-Arrestin2
11.76Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.76Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
11.76Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
11.54Single4O9RCyclopamine4O9R-SMO-Cyclopamine
11.54Single5L7IVismodegib5L7I-SMO-Vismodegib
11.54Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
11.54Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
11.54Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
11.54Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS; CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
11.54Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
11.54Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
11.54Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
11.54Single7XKFDehydroepiandrosterone7XKF-ADGRG2-Dehydroepiandrosterone-Gs/β1/γ2
11.54Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
11.54Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
11.54Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
11.54Single8J6PPubChem 251012238J6P-HCA2-Niacin-PubChem 25101223-Gi1/β1/γ2
11.54Single8JHYPubChem 251012238JHY-HCA2-PubChem 25101223-Gi1/β1/γ2
11.54Single8JIIPubChem 251012238JII-HCA2-Niacin-PubChem 25101223-Gi1/β1/γ2
11.54Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
11.54Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
11.54Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
11.54Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
11.54Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
11.54Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
11.54Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
11.54Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
11.54Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.54Single9JEDHistamine9JED-H4-Histamine-PO4-Gi1/β1/γ2
11.54Single9JEQHistamine9JEQ-H3-Histamine-Gi1/β1/γ2
11.54Single9JLCAVE 09919JLC-MAS1-AVE 0991-Gi1/β1/γ2
11.54Single9KUWCMPD6449KUW-Apelin; Apelin-CMPD644-Arrestin2 ; Arrestin2
11.54Single9L42Histamine9L42-H4-Histamine-Gi1/β1/γ2
11.54Single9U9VMETH9U9V-β2-METH-Gs/β1/γ2
11.54Single9YDAAll-trans-Retinal9YDA-Opsin1MW-All-trans-Retinal-chim(NtGi1L-Gs-CtGt)/β1/γ2
11.54Consensusgq_nucleotideOrthosteric Ligandgq_p2y
11.54Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
11.54Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
11.43Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
11.43Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
11.43Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
11.43Single7PIVAfamelanotide7PIV-MC4-Afamelanotide-Gs/β1/γ2
11.43Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.43Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
11.43Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
11.43Single9IK8Pasireotide9IK8-SST1-Pasireotide-Gi1/β1/γ2
11.43Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
11.43Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-Ibutamoren-Gi1/β1/γ2
11.43Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-Ibutamoren-Gi1/β1/γ2
11.43Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
11.43Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
11.11Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
11.11Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
11.11Single4QINSAG1.54QIN-SMO-SAG1.5
11.11Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
11.11Single5WS3EMPA5WS3-OX2-EMPA
11.11Single5ZKQABT-4915ZKQ-PAF-ABT-491
11.11Single6LFOCXCL86LFO-CXCR2-CXCL8-Gi1/β1/γ2
11.11Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
11.11Single6OBAAlprenolol6OBA-β2-Alprenolol-GTPL11074
11.11Single6PT2KGCHM076PT2-δ-KGCHM07
11.11Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
11.11Single6TODEMPA6TOD-OX1-EMPA-Na
11.11Single6W25SHU91196W25-MC4-SHU9119-Ca
11.11Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
11.11Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
11.11Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
11.11Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
11.11Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
11.11Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
11.11Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
11.11Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
11.11Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
11.11Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
11.11Single7XRRLemborexant7XRR-OX2-Lemborexant
11.11Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
11.11Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
11.11Single8DWGML3828DWG-MRGPRX1-BAM8-22-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
11.11Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
11.11Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
11.11Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
11.11Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
11.11Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
11.11Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
11.11Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
11.11Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
11.11Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
11.11Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
11.11Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
11.11Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
11.11Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
11.11Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
11.11Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
11.11Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
11.11Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
11.11Single8XZGApelin-138XZG-Apelin; Apelin-Apelin-13-Gi1/β1/γ2
11.11Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
11.11Single8YNFCXCL88YNF-ACKR1-CXCL8
11.11Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
11.11Single9H2XPubChem 1756706449H2X-A2A-PubChem 175670644-Na
11.11Single9LKDPL459LKD-OR5V1-PL45
11.11Single9M88Oleic monoethanolamide9M88-GPR3 ; GPR3-Oleic monoethanolamide-AF64394
11.11Consensusalpha2_offOrthosteric Ligandalpha2c_off
11.11Consensusangiotensin_offOrthosteric Ligandat1_off
11.11Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-TC-FPR 43-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
11.11Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
11.11Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
11.11Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.11Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
11.11Consensusorexin_offOrthosteric Ligandox2_off ox1_off
11.11Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
11.11Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
11.11Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
11.11Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
11.11Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
10.81Single6JODAngiotensin II6JOD-AT2-Angiotensin II
10.81Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
10.81Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-TC-FPR 43-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
10.81Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
10.71Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
10.71Single3REYPubChem 56973REY-A2A-PubChem 5697
10.71Single4LDOEpinephrine4LDO-β2-Epinephrine
10.71Single4ZJCSB-6740424ZJC-OX1-SB-674042
10.71Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
10.71Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
10.71Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
10.71Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
10.71Single6KUXRS799486KUX-α2a-RS79948
10.71Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
10.71Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
10.71Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
10.71Single6PS0Carazolol6PS0-β2-Carazolol
10.71Single6PS4ICI118-5516PS4-β2-ICI118-551
10.71Single6PS5Propranolol6PS5-β2-Propranolol
10.71Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
10.71Single6TPGEMPA6TPG-OX2-EMPA
10.71Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
10.71Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
10.71Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
10.71Single6ZG9GSK10347026ZG9-M1-GSK1034702
10.71Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
10.71Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
10.71Single7F61PF-036547467F61-H3-PF-03654746
10.71Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS; CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
10.71Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.71Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
10.71Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
10.71Single7UL3Famotidine7UL3-H2-Famotidine
10.71Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
10.71Single7VV6C48/807VV6-MRGPRX2-C48/80
10.71Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
10.71Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
10.71Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
10.71Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
10.71Single8GE5Constrained Epinephrine8GE5-β2-Constrained Epinephrine-Gs/β1/γ1
10.71Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
10.71Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
10.71Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
10.71Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
10.71Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
10.71Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
10.71Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
10.71Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
10.71Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
10.71Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
10.71Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
10.71Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
10.71Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
10.71Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
10.71Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
10.71Single8K2WAMG4878K2W-CXCR3-AMG487
10.71Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.71Single8RLNLUF58348RLN-A2A-LUF5834
10.71Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
10.71Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
10.71Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
10.71Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single8ZPMAMD0708ZPM-CXCR4-AMD070
10.71Single8ZPNAMD31008ZPN-CXCR4-AMD3100
10.71Single9AS5Mescaline9AS5-5-HT2A-Mescaline
10.71Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single9AS8Psilocin9AS8-5-HT2A-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single9JH3CMF-0199JH3-Apelin; Apelin-CMF-019-Gi1/β1/γ2
10.71Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
10.71Single9L84Epinephrine9L84-β1-Epinephrine-Atazanavir-Gs/β1/γ2
10.71Single9LL8Psilocin9LL8-5-HT2A-Psilocin-Gi1/β1/γ2
10.71Single9VNFPindolol9VNF-5-HT1A-Pindolol-Go/β1/γ2
10.71Single9W33S5A19W33-SST5-S5A1
10.71Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
10.71Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
10.71Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
10.71Consensusopsins_offOrthosteric Ligandrhodopsin_off
10.71Consensussensory_offOrthosteric Ligandopsins_off
10.53Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
10.34Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
10.34Single2Y01Dobutamine2Y01-β1-Dobutamine
10.34Single2Y02Carmoterol2Y02-β1-Carmoterol
10.34Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
10.34Single3NY8ICI118-5513NY8-β2-ICI118-551
10.34Single3NYAAlprenolol3NYA-β2-Alprenolol
10.34Single3ZPQPubChem 5945903ZPQ-β1-PubChem 594590-Na
10.34Single3ZPRPubChem 5987543ZPR-β1-PubChem 598754-Na
10.34Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
10.34Single4GBRCarazolol4GBR-β2-Carazolol
10.34Single4MQSIperoxo4MQS-M2-Iperoxo
10.34Single4QIMANTA XV4QIM-SMO-ANTA XV
10.34Single4QKXPubChem 762106284QKX-β2-PubChem 76210628
10.34Single4U14Tiotropium4U14-M3-Tiotropium
10.34Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
10.34Single5DSGTiotropium5DSG-M4-Tiotropium
10.34Single5UIGPubChem 1240811965UIG-A2A-PubChem 124081196
10.34Single5YC8N-methyl-Scopolamine5YC8-M2-N-methyl-Scopolamine
10.34Single5ZK8N-methyl-Scopolamine5ZK8-M2-N-methyl-Scopolamine
10.34Single5ZKCN-methyl-Scopolamine5ZKC-M2-N-methyl-Scopolamine
10.34Single5ZKPSR274175ZKP-PAF-SR27417
10.34Single6DRXLisuride6DRX-5-HT2B-Lisuride
10.34Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
10.34Single6GPSMK08126GPS-CCR2-MK0812
10.34Single6H7MSalbutamol6H7M-β1-Salbutamol
10.34Single6PRZAlprenolol6PRZ-β2-Alprenolol
10.34Single6PS2Alprenolol6PS2-β2-Alprenolol
10.34Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
10.34Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
10.34Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
10.34Single7BTSEpinephrine7BTS-β1-Epinephrine
10.34Single7BU6Norepinephrine7BU6-β1-Norepinephrine
10.34Single7BU7BI1671077BU7-β1-BI167107
10.34Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
10.34Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
10.34Single7JOZPubChem 752020227JOZ-D1-PubChem 75202022-Gs/β1/γ2
10.34Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
10.34Single7LJCSKF812977LJC-D1-SKF81297-Mevidalen-Gs/β1/γ2
10.34Single7NA8Ibutamoren7NA8-Ghrelin-Ibutamoren-Gi1/β1/γ2
10.34Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
10.34Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
10.34Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
10.34Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
10.34Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
10.34Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
10.34Single7VGZRamelteon7VGZ-MT1-Ramelteon-Gi1/β1/γ2
10.34Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
10.34Single7VIFFTY720-P7VIF-S1P1-FTY720-P-Gi1/β1/γ2
10.34Single7WC7Lisuride7WC7-5-HT2A-Lisuride
10.34Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
10.34Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
10.34Single8GCML-9026888GCM-EP4-L-902688-Gi1/β1/γ2
10.34Single8GE2Constrained Epinephrine8GE2-β2-Constrained Epinephrine-Gs/β1/γ1
10.34Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
10.34Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
10.34Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
10.34Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
10.34Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
10.34Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
10.34Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
10.34Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
10.34Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
10.34Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
10.34Single8JJOAlprenolol8JJO-β2-Alprenolol
10.34Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
10.34Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
10.34Single8JXRLSD8JXR-D1-LSD
10.34Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
10.34Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
10.34Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
10.34Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.34Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
10.34Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
10.34Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
10.34Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
10.34Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
10.34Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
10.34Single9IMATalquetamab9IMA-GPRC5D; GPRC5D-Talquetamab
10.34Single9IYAONO-97105319IYA-GPR55-ONO-9710531
10.34Single9JEAAtropine9JEA-M1-Atropine
10.34Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
10.34Single9METGp120; CD49MET-CXCR4-Gp120; CD4
10.34Single9PXWNaloxone9PXW-μ-Naloxone-GDPβS-Gi1/β1/γ2
10.34Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
10.34Consensus5ht5_onOrthosteric Ligand5ht5a_on
10.34Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
10.34Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
10.34Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
10.34Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
10.34Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
10.34Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
10.34Consensusdopamine_offOrthosteric Ligandd2_off d3_off
10.34Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
10.34Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
10.34Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
10.34Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
10.34Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-2-Phenylethylamine-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
10.34Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
10.34Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
10.34Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
10.34Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
10.00Single2RH1Carazolol2RH1-β2-Carazolol
10.00Single2Y00Dobutamine2Y00-β1-Dobutamine
10.00Single2YCWCarazolol2YCW-β1-Carazolol
10.00Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
10.00Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
10.00Single5D6LCarazolol5D6L-β2-Carazolol
10.00Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
10.00Single5WQCEMPA5WQC-OX2-EMPA
10.00Single5X7DCarazolol5X7D-β2-Carazolol-PubChem 129318963
10.00Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
10.00Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
10.00Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
10.00Single6E67BI1671076E67-β2-BI167107-Gs(CT)
10.00Single6GPXMK08126GPX-CCR2-MK0812
10.00Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
10.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
10.00Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
10.00Single6PS3Carvedilol6PS3-β2-Carvedilol
10.00Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
10.00Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
10.00Single7BVQCarazolol7BVQ-β1-Carazolol
10.00Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
10.00Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
10.00Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
10.00Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
10.00Single7VFXfMIFL7VFX-FPR1-ALX-fMIFL-Gi1/β1/γ2
10.00Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
10.00Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
10.00Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
10.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
10.00Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
10.00Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
10.00Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.00Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.00Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
10.00Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
10.00Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
10.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
10.00Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
10.00Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
10.00Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
10.00Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
10.00Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
10.00Single9EKHONO-30302979EKH-DP1-ONO-3030297
10.00Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
10.00Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
10.00Single9HAPTolvaptan9HAP-V2-Tolvaptan
10.00Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single9U81Tolvaptan9U81-V2-Tolvaptan
10.00Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
10.00Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
10.00Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
10.00Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-Dehydroepiandrosterone-Gs/β1/γ2
10.00Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-Dehydroepiandrosterone-Gs/β1/γ2
10.00Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
10.00Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
10.00Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
10.00Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
10.00Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
10.00Consensusamine_offonOrthosteric Ligandamine_off amine_on
10.00Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
10.00Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
10.00Consensusbeta2_offOrthosteric Ligand2RH1-β2-Carazolol 6PS3-β2-Carvedilol 6PS5-β2-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-PubChem 913103 6PRZ-β2-Alprenolol
10.00Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
10.00Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
10.00Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
10.00Consensusep_offOrthosteric Ligandep4_off
10.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMIFL-Gi1/β1/γ2
10.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMIFL-Gi1/β1/γ2
10.00Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
10.00Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-Lysophosphatidylserine (WJS)-chim(NtGi2-G13)/β1/γ2
9.76Single8KGGLysophosphatidylserine (WJS)8KGG-P2Y10-Lysophosphatidylserine (WJS)-chim(NtGi2-G13)/β1/γ2
9.76Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
9.68Single3PDSFAUC503PDS-β2-FAUC50
9.68Single4DJHJDTic4DJH-κ-JDTic
9.68Single4U15Tiotropium4U15-M3-Tiotropium
9.68Single5D5ACarazolol5D5A-β2-Carazolol
9.68Single5D5BCarazolol5D5B-β2-Carazolol
9.68Single5TZRMK86665TZR-FFA1-MK8666
9.68Single5V54Methiothepin5V54-5-HT1B-Methiothepin
9.68Single6DDEDAMGO6DDE-μ-DAMGO-Gi1/β1/γ2
9.68Single6J20Aprepitant6J20-NK1-Aprepitant
9.68Single6J21Aprepitant6J21-NK1-Aprepitant
9.68Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
9.68Single6OL9Tiotropium6OL9-M5-Tiotropium
9.68Single6OS1TRV0266OS1-AT1-TRV026
9.68Single6TQ7SB-3348676TQ7-OX1-SB-334867
9.68Single7EW4CYM-55417EW4-S1P3-CYM-5541-Gi1/β1/γ2
9.68Single7P2L4YI7P2L-mGlu5-4YI
9.68Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
9.68Single7U2LC5-guano7U2L-μ-C5-guano-Gi1/β1/γ2
9.68Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
9.68Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
9.68Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
9.68Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
9.68Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
9.68Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
9.68Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
9.68Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
9.68Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
9.68Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
9.68Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
9.68Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
9.68Single8XBIPubChem 1626566368XBI-GPR34-PubChem 162656636
9.68Single8XVLZibotentan8XVL-ETA-Zibotentan
9.68Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
9.68Single9BJKNaloxone9BJK-μ-Naloxone-PubChem 171642066
9.68Single9BS9LSD9BS9-D2-LSD
9.68Single9BSBLSD9BSB-D2-LSD-chim(NtGi1-Go)/β1/γ2
9.68Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
9.68Single9PY3Loperamide9PY3-μ-Loperamide-GDPβS-Gi1/β1/γ2
9.68Single9UCPIperoxo9UCP-M1-Iperoxo-G11(CT)
9.68Consensus5ht1_offOrthosteric Ligand5ht1b_off
9.68Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
9.68Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
9.68Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-PubChem 594590-Na 3ZPR-β1-PubChem 598754-Na
9.68Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
9.68Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
9.68Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
9.68Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
9.68Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-PtdIns4P-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-PtdIns4P-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-PtdIns4P-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-PtdIns4P-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-PtdIns4P-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-PtdIns4P-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-PtdIns4P-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-PtdIns4P-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
9.68Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoprenaline-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
9.68Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
9.68Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
9.68Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
9.38Single3D4STimolol3D4S-β2-Timolol
9.38Single4AMIBucindolol4AMI-β1-Bucindolol
9.38Single4N4WSANT-14N4W-SMO-SANT-1
9.38Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
9.38Single4PY02MeSATP4PY0-P2Y12-2MeSATP
9.38Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
9.38Single6A93Risperidone6A93-5-HT2A-Risperidone
9.38Single6DRYMethylergometrine6DRY-5-HT2B-Methylergometrine
9.38Single6H7NXamoterol6H7N-β1-Xamoterol
9.38Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
9.38Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
9.38Single6ZG4HTL00099366ZG4-M1-HTL0009936
9.38Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
9.38Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
9.38Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
9.38Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
9.38Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
9.38Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
9.38Single8JWY2-1188JWY-A2A-2-118
9.38Single8T3QDoconexent8T3Q-FFA4-Doconexent-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Single8WRBLysophosphatidylserine (UBL)8WRB-GPR34-Lysophosphatidylserine (UBL)-Gi1/β1/γ2
9.38Single8XQJJN2418XQJ-Apelin; Apelin-JN241
9.38Single9BJKPubChem 1716420669BJK-μ-Naloxone-PubChem 171642066
9.38Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
9.38Single9VIFNeuropeptide-VF9VIF-NPFF1-Neuropeptide-VF-Gi1/β1/γ2
9.38Single9W32SSTR5 antagonist 19W32-SST5-SSTR5 antagonist 1
9.38Single9WSWEndomorphin9WSW-μ-Endomorphin-chim(NtGi1-Gz)/β1/γ2
9.38Single9YDQDADLE9YDQ-δ-DADLE-MIPS3614-chim(NtGi1L-Gs-CtGi1)/β1/γ2
9.38Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-PtdIns4P-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-PtdIns4P-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-PtdIns4P-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-PtdIns4P-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-PtdIns4P-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-PtdIns4P-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-PtdIns4P-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-PtdIns4P-Gi1/β1/γ1
9.38Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-PtdIns4P-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-PtdIns4P-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-PtdIns4P-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-PtdIns4P-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-PtdIns4P-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-PtdIns4P-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-PtdIns4P-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-PtdIns4P-Gi1/β1/γ1
9.38Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
9.38Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
9.38Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
9.38Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
9.38Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
9.38Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
9.09Single6H7LDobutamine6H7L-β1-Dobutamine
9.09Single6IBLArformoterol6IBL-β1-Arformoterol
9.09Single6K1QIRL25006K1Q-ETB-IRL2500
9.09Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
9.09Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
9.09Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.09Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
9.09Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
9.09Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8XVJMacitentan8XVJ-ETA-Macitentan
9.09Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
9.09Single9DYEBuspirone9DYE-5-HT1A-Buspirone-PtdIns4P-Go/β1/γ2
9.09Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single9HYIDP819HYI-5-HT1A-DP81-Gi1/β1/γ2
9.09Single9J0BUDP-Glucose9J0B-P2Y14-UDP-Glucose-Gi1/β1/γ2
9.09Single9YDPDADLE9YDP-δ-DADLE-chim(NtGi1L-Gs-CtGi1)/β1/γ2
9.09Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
9.09Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
9.09Consensuschemerin_onOrthosteric Ligandcml1_on
9.09Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
8.82Single6KNMJN241-96KNM-Apelin-JN241-9
8.82Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
8.82Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
8.82Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
8.82Single7SK9CCX6627SK9-ACKR3-CCX662
8.82Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
8.82Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
8.82Single8SAILysophosphatidylserine (S12)8SAI-GPR34-Lysophosphatidylserine (S12)-Gi1/β1/γ2
8.82Single8Z74JN241-98Z74-Apelin; Apelin-JN241-9
8.82Single8Z74JN241-98Z74-Apelin; Apelin-JN241-9
8.82Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
8.82Single9MD1Buspirone9MD1-5-HT1A-Buspirone-PtdIns4P-Gz/β1/γ2
8.82Single9WSXEndomorphin9WSX-μ-Endomorphin-Arrestin2
8.82Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-1-chim(NtGi1-Gq)/β1/γ1
8.82Consensuskisspeptin_onOrthosteric Ligandkiss1_on
8.70Single5MZPCaffeine5MZP-A2A-Caffeine-Na
8.70Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
8.70Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
8.57Single4AMJCarvedilol4AMJ-β1-Carvedilol
8.57Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
8.57Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
8.57Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
8.57Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-PtdIns4P-Gi1/β1/γ1
8.57Single8IZBLysophosphatidylserine (UBL)8IZB-GPR174-Lysophosphatidylserine (UBL)-Gs/β1/γ2
8.57Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
8.57Single8ZJDKisspeptin-18ZJD-Kiss1-Kisspeptin-1-chim(NtGi1-Gq)/β1/γ1
8.57Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
8.57Single9M4TSilodosin9M4T-Alpha1A-Silodosin
8.57Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-1-chim(NtGi1-Gq)/β1/γ1
8.57Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-1-chim(NtGi1-Gq)/β1/γ1
8.57Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
8.57Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
8.57Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
8.33Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
8.33Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
8.33Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
8.33Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
8.33Single8K6ONeuropeptide-Y8K6O-Y1-Neuropeptide-Y-Gi2/β1/γ1
8.33Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
8.33Single9JIDNiacin9JID-HCA3-Niacin-Gi1/β1/γ2
8.33Single9JKVPubChem 27366909JKV-HCA3-PubChem 2736690-Gi1/β1/γ2
8.11Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
8.11Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
8.11Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
8.00Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
8.00Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
8.00Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
8.00Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
8.00Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
8.00Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single9CHUNorepinephrine9CHU-β2-Norepinephrine
8.00Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
8.00Single9L0HJR14a9L0H-C3aB-JR14a-Go/β1/γ2
8.00Single9M42A1L8O9M42-GPR139-A1L8O-chim(Gs-CtGq)/β1/γ2
8.00Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
8.00Consensussensory_onOrthosteric Ligandopsins_on
7.69Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
7.69Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
7.69Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
7.69Single3UZAGTPL92363UZA-A2A-GTPL9236
7.69Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
7.69Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
7.69Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
7.69Single6ME5Agomelatine6ME5-MT1-Agomelatine
7.69Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
7.69Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
7.69Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
7.69Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
7.69Single7XV3Lysophosphatidylserine (WJS)7XV3-GPR174-Lysophosphatidylserine (WJS)-chim(NtGi1-Gs)/β1/γ2
7.69Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8IW72-Phenylethylamine8IW7-TAA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
7.69Single8JPSCCL78JPS-ACKR1-CCL7
7.69Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
7.69Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
7.69Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
7.69Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
7.69Single9JKT(2R)-2-hydroxy-3-phenylpropanoic acid9JKT-HCA3-(2R)-2-hydroxy-3-phenylpropanoic acid-Gi1/β1/γ2
7.69Consensus5ht2_onOrthosteric Ligand5ht2b_on
7.69Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
7.69Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-Lysophosphatidylserine (WJS)-chim(NtGi2-G13)/β1/γ2
7.69Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
7.69Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
7.41Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
7.41Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
7.41Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
7.41Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
7.41Single3PBLEticlopride3PBL-D3-Eticlopride
7.41Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
7.41Single6HLLCP999946HLL-NK1-CP99994
7.41Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
7.41Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
7.41Single6TP4ACT-4622066TP4-OX1-ACT-462206
7.41Single7SRQLSD7SRQ-5-HT2B-LSD
7.41Single7UL2SR486927UL2-NTS1-SR48692-Na
7.41Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
7.41Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
7.41Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
7.41Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
7.41Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
7.41Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
7.41Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
7.41Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
7.41Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
7.41Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
7.41Single8W892-Phenylethylamine8W89-TA1-2-Phenylethylamine-chim(NtGi1L-Gs)/β1/γ2
7.41Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
7.41Single8ZYUNeurotensin-(8-13)8ZYU-NTS1-Neurotensin-(8-13)-SBI-553-Arrestin2
7.41Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single9AS7Psilocin9AS7-5-HT2A-Psilocin
7.41Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
7.41Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
7.41Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
7.41Single9M88Oleic monoethanolamide9M88-GPR3 ; GPR3-Oleic monoethanolamide-AF64394
7.41Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
7.41Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
7.41Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
7.41Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
7.41Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
7.41Consensusneurotensin_offOrthosteric Ligandnts1_off
7.41Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
7.14Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
7.14Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
7.14Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
7.14Single5OLVLUAA470705OLV-A2A-LUAA47070-Na
7.14Single6AKXA4R6AKX-CCR5-A4R
7.14Single6AKYMaraviroc6AKY-CCR5-Maraviroc
7.14Single6B73MP11046B73-κ-MP1104
7.14Single6DS0LY2660976DS0-5-HT2B-LY266097
7.14Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
7.14Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
7.14Single6ME2Ramelteon6ME2-MT1-Ramelteon
7.14Single6ME9Ramelteon6ME9-MT2-Ramelteon
7.14Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
7.14Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
7.14Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
7.14Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
7.14Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
7.14Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
7.14Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
7.14Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
7.14Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
7.14Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
7.14Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
7.14Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8FYXBuspirone8FYX-5-HT1A-Buspirone-PtdIns4P-Gi1/β1/γ1
7.14Single8T3VDoconexent8T3V-FFA1-Doconexent-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
7.14Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
7.14Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
7.14Single9K6LSalicin9K6L-TAS2R16-Salicin-Gi2/β1/γ2
7.14Single9LL9DOI9LL9-5-HT2A-DOI-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single9LLBDOI-NBOMe9LLB-5-HT2A-DOI-NBOMe-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
7.14Single9PEEPF-07054894; OXM29PEE-CCR6-PF-07054894; OXM2
7.14Single9PXUNaloxone9PXU-μ-Naloxone-Na
7.14Single9VJ5Gepirone9VJ5-5-HT1A-Gepirone-Go/β1/γ2
7.14Single9VJEBuspirone9VJE-5-HT1A-Buspirone-Go/β1/γ2
7.14Single9W49U-50488H9W49-κ-U-50488H-Gi1/β1/γ2
7.14Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
7.14Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
7.14Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
7.14Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.14Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
7.14Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.14Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
6.90Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
6.90Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
6.90Single4MBSMaraviroc4MBS-CCR5-Maraviroc
6.90Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
6.90Single6A94Zotepine6A94-5-HT2A-Zotepine
6.90Single6IQLL7458706IQL-D4-L745870
6.90Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
6.90Single6TPKRetosiban6TPK-OT-Retosiban
6.90Single6TPNHTL66416TPN-OX2-HTL6641
6.90Single6VI4JDTic6VI4-κ-JDTic
6.90Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
6.90Single6ZDVPubChem 9840736ZDV-A2A-PubChem 984073-Na
6.90Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
6.90Single6ZINSR486926ZIN-NTS1-SR48692
6.90Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
6.90Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
6.90Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
6.90Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
6.90Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
6.90Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
6.90Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
6.90Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
6.90Single7VODCariprazine7VOD-5-HT2A-Cariprazine
6.90Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
6.90Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
6.90Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
6.90Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
6.90Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
6.90Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
6.90Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
6.90Single8K9LDAMGO8K9L-μ-DAMGO-BMS-986122-Gi3/β1/γ1
6.90Single8THKA-616038THK-Alpha1A-A-61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
6.90Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
6.90Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
6.90Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
6.90Single8ZBWQuin-C18ZBW-FPR2-ALX-Quin-C1-Gi2/β1/γ2
6.90Single9ARXSerotonin9ARX-5-HT2A-Serotonin
6.90Single9AS3LSD9AS3-5-HT2A-LSD
6.90Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
6.90Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
6.90Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
6.90Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
6.90Single9ODJMitragynine Pseudoindoxyl9ODJ-μ-Mitragynine Pseudoindoxyl-GTP; Mg-Gi1/β1/γ2
6.90Single9ODLMitragynine Pseudoindoxyl9ODL-μ-Mitragynine Pseudoindoxyl-GTP; Mg-Gi1/β1/γ2
6.90Single9PXVNaloxone9PXV-μ-Naloxone-Gi1/β1/γ2
6.90Single9PY2Loperamide9PY2-μ-Loperamide-GDPβS-Gi1/β1/γ2
6.90Single9U80Conivaptan9U80-V2-Conivaptan
6.90Single9VJG8-OH-DPAT9VJG-5-HT1A-8-OH-DPAT-chim(NtGi2-Gz)/β1/γ2
6.90Single9W6W5-CT9W6W-5-HT5A-5-CT-Gi1/β1/γ2
6.90Consensusalpha1_onOrthosteric Ligandalpha1a_on
6.90Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
6.90Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
6.90Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
6.90Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
6.90Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
6.90Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
6.90Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
6.90Consensusvasop-oxy_offOrthosteric Ligandot_off
6.67Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
6.67Single4EJ4Naltrindole4EJ4-δ-Naltrindole
6.67Single5DHGC-355DHG-NOP-C-35
6.67Single5DHHSB-6121115DHH-NOP-SB-612111
6.67Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
6.67Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
6.67Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
6.67Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
6.67Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
6.67Single8EFQDAMGO8EFQ-μ-DAMGO-Gi1/β1/γ2
6.67Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.67Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-PtdIns4P-Gi1/β1/γ1
6.67Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
6.67Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
6.67Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
6.67Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
6.67Single8X63Mepyramine8X63-H1-Mepyramine
6.67Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
6.67Single8Y71A1D6F8Y71-δ-A1D6F-BMS986187-Gi1/β1/γ2
6.67Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
6.67Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
6.67Single9DYFAsenapine9DYF-5-HT1A-Asenapine-PtdIns4P-Gi1/β1/γ2
6.67Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
6.67Single9JROPF-044189489JRO-EP2-PF-04418948
6.67Single9PLNPubChem 1682595949PLN-α2a-PubChem 168259594
6.67Single9PLOPubChem 1682595949PLO-α2a-PubChem 168259594-Go/β1/γ2
6.67Single9PQDPubChem 1764919279PQD-α2a-PubChem 176491927
6.67Single9UAZAtropine9UAZ-M1-Atropine
6.67Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
6.67Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
6.67Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
6.67Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
6.67Consensusalpha2_onOrthosteric Ligandalpha2b_on
6.67Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
6.67Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
6.67Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
6.67Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
6.67Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
6.67Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
6.67Consensushistamine_offOrthosteric Ligandh1_off
6.45Single5WIUNemonapride5WIU-D4-Nemonapride
6.45Single5WIVNemonapride5WIV-D4-Nemonapride-Na
6.45Single6Z4SSR486926Z4S-NTS1-SR48692
6.45Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
6.45Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS; CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
6.45Single7WC6LSD7WC6-5-HT2A-LSD
6.45Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
6.45Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
6.45Single8IZ4Lysophosphatidylserine (TJR)8IZ4-GPR34-Lysophosphatidylserine (TJR)-Gi1/β1/γ2
6.45Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
6.45Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.45Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.45Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
6.45Single8ZMFPubChem 1719206738ZMF-5-HT2C-PubChem 171920673
6.45Single9DYDAsenapine9DYD-5-HT1A-Asenapine-PtdIns4P-Go/β1/γ2
6.45Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
6.45Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
6.45Single9HC04YI9HC0-mGlu5-4YI
6.45Single9JRTTG6-1299JRT-EP2-TG6-129
6.45Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
6.45Single9VJFBuspirone9VJF-5-HT1A-Buspirone-Gi3/β1/γ2
6.45Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
6.45Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
6.45Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
6.45Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
6.45Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
6.45Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
6.25Single6E59L-7607356E59-NK1-L-760735
6.25Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
6.25Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-PtdIns4P-Gi1/β1/γ2
6.25Single7R0CAVP7R0C-V2-AVP-Arrestin2
6.25Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
6.25Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
6.25Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
6.25Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
6.25Single8X0FVU298X0F-mGlu5; mGlu5-Quisqualate-VU29
6.25Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
6.25Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
6.25Single9PY4Loperamide9PY4-μ-Loperamide-GDPβS-Gi1/β1/γ2
6.25Single9YDVMRS29059YDV-P2Y14-MRS2905-Gi1/β1/γ2
6.25Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
6.25Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
6.25Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
6.25Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
6.25Consensustachykinin_offOrthosteric Ligandnk1_off
6.06Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
6.06Single4PXFOctyl-Beta-D-Glucopyranoside4PXF-Rhodopsin-Octyl-β-D-Glucopyranoside-Arrestin1 Finger Loop
6.06Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
6.06Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
6.06Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
6.06Single8JWZEtrumadenant8JWZ-A2A-Etrumadenant-Na
6.06Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
6.06Single9YDUUDP-Glucose9YDU-P2Y14-UDP-Glucose-Gi1/β1/γ2
6.06Consensusalpha1_offOrthosteric Ligandalpha1a_off
6.06Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
6.06Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
6.06Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
6.06Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
5.88Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
5.88Single7D7MPGE27D7M-EP4-PGE2-Gs/β1/γ1
5.88Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
5.88Single8XBES3E-Lysophosphatidylserine 8XBE-GPR34-S3E-Lysophosphatidylserine-Gi1/β1/γ1
5.88Single9VI9RFRP-39VI9-NPFF1-RFRP-3-Gi1/β1/γ2
5.88Single9YDRDADLE9YDR-δ-DADLE-MIPS3983-chim(NtGi1L-Gs-CtGi1)/β1/γ2
5.88Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
5.71Single8X5YAstemizole8X5Y-H1-Astemizole
5.71Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.71Single9NS9TUG-13759NS9-FFA2-TUG-1375-PubChem 118615810-Gi1/β1/γ2
5.56Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
4.76Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.76Single6D35Cholesterol6D35-SMO-Cholesterol
4.76Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.76Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.76Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.76Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.76Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
4.76Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.76Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.76Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
4.76Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.76Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
4.76Single7DD5Ca7DD5-CaS; CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS; CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DD5Ca7DD5-CaS; CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS; CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.76Single7DTTCa7DTT-CaS; CaS-Ca-Ca
4.76Single7DTTCa7DTT-CaS; CaS-Ca-Ca
4.76Single7DTUTryptophan7DTU-CaS; CaS-Tryptophan
4.76Single7DTUTryptophan7DTU-CaS; CaS-Tryptophan
4.76Single7DTVCa7DTV-CaS; CaS-Ca-Ca; Tryptophan
4.76Single7DTVCa; Tryptophan7DTV-CaS; CaS-Ca-Ca; Tryptophan
4.76Single7DTVCa7DTV-CaS; CaS-Ca-Ca; Tryptophan
4.76Single7DTVCa; Tryptophan7DTV-CaS; CaS-Ca-Ca; Tryptophan
4.76Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E6TCa7E6T-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E6TCa7E6T-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.76Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.76Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.76Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.76Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.76Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.76Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.76Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.76Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.76Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.76Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.76Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.76Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.76Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS; CaS-Ca; Ca; Tryptophan; NPS-2143
4.76Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS; CaS-Ca; Ca; Tryptophan; NPS-2143
4.76Single7M3FCa; Ca; Tryptophan; Cinacalcet7M3F-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet
4.76Single7M3FCa; Ca; Tryptophan; Cinacalcet7M3F-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS; CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS; CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS; CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS; CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.76Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.76Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.76Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.76Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.76Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.76Single7SILCa7SIL-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4
4.76Single7SILCa; Ca; Ca; Cyclomethyltryptophan; R-568; PO47SIL-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4
4.76Single7SILCa7SIL-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4
4.76Single7SILCa; Ca; Ca; Cyclomethyltryptophan; R-568; PO47SIL-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4
4.76Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7SIMCa7SIM-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7SIMCa7SIM-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
4.76Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.76Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.76Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.76Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.76Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.76Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.76Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.76Single7XW7K1-707XW7-TSH-K1-70
4.76Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.76Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.76Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.76Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.76Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.76Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.76Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.76Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.76Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.76Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.76Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.76Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.76Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.76Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.76Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.76Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.76Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.76Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.76Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.76Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.76Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.76Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.76Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.76Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.76Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.76Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.76Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.76Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.76Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.76Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.76Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.76Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.76Single8TQBCa; LY3792688TQB-mGlu3; mGlu3-Ca; LY379268-Ca
4.76Single8TQBCa; LY3792688TQB-mGlu3; mGlu3-Ca; LY379268-Ca
4.76Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.76Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.76Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.76Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.76Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.76Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.76Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.76Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.76Single8WG9PubChem 1793948WG9-mGlu4; mGlu2-PubChem 179394
4.76Single8WGBGlutamate8WGB-mGlu4; mGlu2-Glutamate-VU0155041-Gi3/β1/γ2
4.76Single8WGBGlutamate8WGB-mGlu4; mGlu2-Glutamate-VU0155041-Gi3/β1/γ2
4.76Single8WGCLY3792688WGC-mGlu2; mGlu4-LY379268
4.76Single8WGDLY341495; CPPG8WGD-mGlu4; mGlu2-LY341495; CPPG
4.76Single8WGDLY341495; CPPG8WGD-mGlu4; mGlu2-LY341495; CPPG
4.76Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS; CaS-Tryptophan; Cinacalcet; PO4; Ca
4.76Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS; CaS-Tryptophan; Cinacalcet; PO4; Ca
4.76Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS; CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS; CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8WVXNorrin8WVX-LGR4-Norrin
4.76Single8WVYNorrin8WVY-LGR4-Norrin
4.76Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.76Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.76Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU29
4.76Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU29
4.76Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.76Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.76Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.76Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.76Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.76Single9ASBCa9ASB-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9ASBCa; Ca; Cyclomethyltryptophan; R-568; PO49ASB-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AVGCa9AVG-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AVGCa; Ca; Cyclomethyltryptophan; R-568; PO49AVG-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AVLCa9AVL-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-Gi3/β2/γ2
4.76Single9AVLCa; Ca; Cyclomethyltryptophan; R-568; PO49AVL-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-Gi3/β2/γ2
4.76Single9AVLCa9AVL-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-Gi3/β2/γ2
4.76Single9AVLCa; Ca; Cyclomethyltryptophan; R-568; PO49AVL-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-Gi3/β2/γ2
4.76Single9AXFCa9AXF-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; R-568; PO49AXF-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AXFCa9AXF-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; R-568; PO49AXF-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AYFCa9AYF-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4-Gi1/β1/γ2
4.76Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; R-568; PO49AYF-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4-Gi1/β1/γ2
4.76Single9C1PCa9C1P-CaS; CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS; CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C1PCa9C1P-CaS; CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS; CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C2FCa9C2F-CaS; CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.76Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS; CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.76Single9C2FCa9C2F-CaS; CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.76Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS; CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.76Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2; Arrestin2
4.76Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2; Arrestin2
4.76Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single9KB7R-spondin-29KB7-LGR4-R-spondin-2
4.76Single9KGKNB189KGK-LGR4-NB18
4.76Single9KHHNorrin9KHH-LGR4-Norrin
4.76Single9MBAGlutamate9MBA-mGlu8; mGlu8-Glutamate-Arrestin2 ; Arrestin2
4.76Single9MBAGlutamate9MBA-mGlu8; mGlu8-Glutamate-Arrestin2 ; Arrestin2
4.76Single9MBBLY3414959MBB-mGlu8; mGlu8-LY341495
4.76Single9MBBLY3414959MBB-mGlu8; mGlu8-LY341495
4.76Single9MBCDCPG9MBC-mGlu8; mGlu8-DCPG-AZ12216052
4.76Single9MBCDCPG9MBC-mGlu8; mGlu8-DCPG-AZ12216052
4.76Single9S37NB219S37-LGR4-NB21
4.76Single9S38NB219S38-LGR4-NB21
4.76Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.55Single7DD6Ca7DD6-CaS; CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD6Ca; Ca; Tryptophan7DD6-CaS; CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD6Ca7DD6-CaS; CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD6Ca; Ca; Tryptophan7DD6-CaS; CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD7Ca7DD7-CaS; CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS; CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single7DD7Ca7DD7-CaS; CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS; CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single9ASBCa9ASB-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9ASBCa; Ca; Cyclomethyltryptophan; R-568; PO49ASB-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AVGCa9AVG-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVGCa; Ca; Cyclomethyltryptophan; R-568; PO49AVG-CaS; CaS-Ca-Ca; Ca; Cyclomethyltryptophan; R-568; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AYFCa9AYF-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4-Gi1/β1/γ2
4.55Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; R-568; PO49AYF-CaS; CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; R-568; PO4-Gi1/β1/γ2
4.55Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.55Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.35Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.35Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.35Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS; CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.35Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.17Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.17Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.17Single7UTZTSH7UTZ-TSH-TSH-DPPC-Gs/β1/γ2
4.17Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.17Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.00Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
4.00Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
4.00Single5L7DCholesterol5L7D-SMO-Cholesterol
4.00Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.00Single7WC4Serotonin7WC4-5-HT2A-Serotonin
4.00Single8I2GFSH8I2G-FSH-FSH-PubChem 67530240-Gs/β1/γ2
4.00Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
3.85Single6TQ9SB-4081246TQ9-OX1-SB-408124
3.85Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
3.85Single8IWM2-Phenylethylamine8IWM-TAA9-2-Phenylethylamine
3.85Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
3.85Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
3.70Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
3.70Single7WC5Psilocin7WC5-5-HT2A-Psilocin
3.70Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.70Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
3.70Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
3.70Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
3.70Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
3.70Single9LL7DOI9LL7-5-HT2A-DOI-Gi1/β1/γ2
3.70Single9MBCAZ122160529MBC-mGlu8; mGlu8-DCPG-AZ12216052
3.70Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
3.70Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
3.70Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
3.57Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
3.57Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-PtdIns4P-Gi1/β1/γ2
3.57Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.57Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
3.57Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
3.57Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
3.57Single8HNNSCH5467388HNN-CXCR3-SCH546738
3.57Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.57Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.57Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
3.57Single9MBCAZ122160529MBC-mGlu8; mGlu8-DCPG-AZ12216052
3.57Single9MNIdC2_059MNI-CTLike-dC2_05-RAMP1
3.57Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
3.45Single4XNVBPTU4XNV-P2Y1-BPTU
3.45Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
3.45Single7T6STC-FPR 437T6S-FPR2-ALX-TC-FPR 43-Gi1/β1/γ2
3.45Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
3.45Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
3.45Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.45Single8TZQDopamine8TZQ-D2-Dopamine-Go/β1/γ2
3.45Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
3.45Single9KVHCinobufotenine9KVH-5-HT1A-Cinobufotenine-PtdIns4P-Gi1/β1/γ2
3.45Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
3.33Single3RZECidoxepin3RZE-H1-Cidoxepin
3.33Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
3.33Single6FFIMPEP6FFI-mGlu5-MPEP
3.33Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
3.33Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
3.33Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
3.33Single8K4NPubChem 1687197658K4N-GPR34-PubChem 168719765-Gi1/β1/γ2
3.33Single8U02Dopamine8U02-D2-Dopamine-Go/β1/γ2
3.33Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
3.33Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
3.33Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single9JQYTG6-1299JQY-EP4-TG6-129
3.33Single9K1DButyric acid9K1D-FFA2-Butyric acid-Gi1/β1/γ2
3.33Single9KVIBufotenin9KVI-5-HT1A-Bufotenin-PtdIns4P-Gi1/β1/γ2
3.33Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
3.23Single6FFHFenobam6FFH-mGlu5-Fenobam
3.23Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
3.23Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
3.23Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
3.23Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
3.23Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
3.23Single8X64Desloratadine8X64-H1-Desloratadine
3.23Single8XBGS3E-Lysophosphatidylserine 8XBG-GPR34-S3E-Lysophosphatidylserine
3.23Single9KFTfMLFC9KFT-FPR1-ALX-fMLFC-Gi1/β1/γ2
3.23Single9LLAAriadne9LLA-5-HT2A-Ariadne-chim(NtGi1L-Gs-CtGq)/β1/γ2
3.23Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
3.23Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
3.23Consensusblt_onOrthosteric Ligandblt1_on
3.23Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
3.23Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
3.23Consensusleukotriene_onOrthosteric Ligandblt_on
3.23Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
3.12Single4NTJAZD12834NTJ-P2Y12-AZD1283
3.12Single6HLPNetupitant6HLP-NK1-Netupitant
3.12Single9EE5ONO-25502899EE5-DP1-ONO-2550289
2.94Single9CM3TUG-13759CM3-FFA2-TUG-1375-PubChem 118615810-chim(NtGi1L-Gs-CtGq)/β1/γ2
2.94Single9WXMGPR15L(CT)9WXM-GPR15-GPR15L(CT)-Gi3/β1/γ2
2.86Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
2.86Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
2.78Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
2.70Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3; ZNRF3
2.70Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.70Single8Y69R-spondin-28Y69-LGR4; LGR4-R-spondin-2-ZNRF3
2.63Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3; ZNRF3
2.63Single9KB8R-spondin-29KB8-LGR4-R-spondin-2-ZNRF3; ZNRF3
2.63Single9KB9R-spondin-29KB9-LGR4; LGR4-R-spondin-2-ZNRF3; ZNRF3
2.56Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.56Single8Y69R-spondin-28Y69-LGR4; LGR4-R-spondin-2-ZNRF3
2.56Single9KB9R-spondin-29KB9-LGR4; LGR4-R-spondin-2-ZNRF3; ZNRF3

PDB Summary
PDB 8YG4
Class B1
SubFamily Peptide
Type Parathyroid Hormone
SubType PTH1
Species Homo Sapiens
Ligand LA-PTH Analog
Other Ligand(s) -
Protein Partners chim(NtGi1-Gs)/Beta1/Gamma2
PDB Resolution 2.59
Date 2025-09-03
D.O.I. To be published
Net Summary
Imin 2.94
Number of Linked Nodes 890
Number of Links 1116
Number of Hubs 200
Number of Links mediated by Hubs 707
Number of Communities 23
Number of Nodes involved in Communities 284
Number of Links involved in Communities 425
Path Summary
Number Of Nodes in MetaPath 114
Number Of Links MetaPath 113
Number of Shortest Paths 1276193
Length Of Smallest Path 3
Average Path Length 31.1757
Length of Longest Path 64
Minimum Path Strength 1.31
Average Path Strength 7.38498
Maximum Path Strength 25.035
Minimum Path Correlation 0.7
Average Path Correlation 0.983671
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.38095
Average % Of Corr. Nodes 48.0649
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 46.137
Maximum Path Hubs % 100
AnnotationTypeLinks
Gene OntologyMolecular Function
Gene OntologyBiological Process• fibroblast proliferation   • cell population proliferation   • cellular process   • cellular response to nitrogen compound   • cellular response to stimulus   • response to dopamine   • regulation of cellular process   • response to stimulus   • signaling   • cellular response to dopamine   • response to monoamine   • cell communication   • response to catecholamine   • adenylate cyclase-activating dopamine receptor signaling pathway   • cellular response to catecholamine stimulus   • signal transduction   • regulation of biological process   • G protein-coupled dopamine receptor signaling pathway   • biological regulation   • response to oxygen-containing compound   • response to nitrogen compound   • adenylate cyclase-activating G protein-coupled receptor signaling pathway   • cellular response to oxygen-containing compound   • cellular response to chemical stimulus   • cellular response to monoamine stimulus   • response to chemical   • adenylate cyclase-modulating G protein-coupled receptor signaling pathway   • G protein-coupled receptor signaling pathway   • response to ketone   • response to prostaglandin   • response to lipid   • response to endogenous stimulus   • response to alcohol   • cellular response to prostaglandin stimulus   • cellular response to endogenous stimulus   • cellular response to prostaglandin E stimulus   • cellular response to alcohol   • response to hormone   • cellular response to lipid   • response to prostaglandin E   • cellular response to ketone   • cellular response to hormone stimulus   • cellular anatomical structure   • membrane   • protein-containing complex   • extrinsic component of plasma membrane   • catalytic complex   • plasma membrane protein complex   • cytoplasmic side of membrane   • plasma membrane   • membrane protein complex   • heterotrimeric G-protein complex   • side of membrane   • cell periphery   • cytoplasmic side of plasma membrane   • GTPase complex
Gene OntologyCellular Component• cellular anatomical structure   • membrane   • protein-containing complex   • extrinsic component of plasma membrane   • catalytic complex   • plasma membrane protein complex   • cytoplasmic side of membrane   • plasma membrane   • membrane protein complex   • heterotrimeric G-protein complex   • side of membrane   • cell periphery   • cytoplasmic side of plasma membrane   • GTPase complex   • extrinsic component of membrane   • extrinsic component of cytoplasmic side of plasma membrane   • extracellular exosome   • membrane-bounded organelle   • extracellular vesicle   • extracellular organelle   • extracellular region   • organelle   • extracellular space   • vesicle   • extracellular membrane-bounded organelle   • synapse   • cell junction   • molecular transducer activity   • G protein-coupled receptor activity   • transmembrane signaling receptor activity   • signaling receptor activity   • identical protein binding   • protein binding   • binding   • protein homodimerization activity   • protein dimerization activity   • peptide hormone binding   • hormone binding   • peptide receptor activity   • G protein-coupled peptide receptor activity   • parathyroid hormone receptor activity   • developmental process   • multicellular organismal process   • ossification   • bone mineralization   • animal organ development   • anatomical structure development   • biomineral tissue development   • tissue development   • multicellular organism development   • skeletal system development   • system development   • cell population proliferation   • cellular process   • cellular response to stimulus   • regulation of biological process   • regulation of cellular process   • response to stimulus   • signaling   • biological regulation   • cell communication   • adenylate cyclase-modulating G protein-coupled receptor signaling pathway   • G protein-coupled receptor signaling pathway   • signal transduction   • inorganic ion homeostasis   • intracellular calcium ion homeostasis   • homeostatic process   • calcium ion homeostasis   • cellular homeostasis   • chemical homeostasis   • intracellular monoatomic cation homeostasis   • monoatomic ion homeostasis   • intracellular chemical homeostasis   • monoatomic cation homeostasis   • intracellular monoatomic ion homeostasis   • osteoblast development   • cellular developmental process   • cell differentiation   • cell development   • osteoblast differentiation   • embryo development ending in birth or egg hatching   • chordate embryonic development   • embryo development   • in utero embryonic development   • anatomical structure maturation   • cell maturation   • developmental maturation   • adenylate cyclase-activating G protein-coupled receptor signaling pathway   • positive regulation of cell population proliferation   • regulation of cell population proliferation   • positive regulation of biological process   • positive regulation of cellular process   • cell surface receptor signaling pathway   • negative regulation of cell population proliferation   • negative regulation of cellular process   • negative regulation of biological process   • phospholipase C-activating G protein-coupled receptor signaling pathway   • connective tissue development   • chondrocyte differentiation   • cartilage development   • regulation of inositol phosphate biosynthetic process   • alcohol metabolic process   • positive regulation of phosphate metabolic process   • inositol phosphate metabolic process   • regulation of primary metabolic process   • positive regulation of metabolic process   • regulation of small molecule metabolic process   • positive regulation of biosynthetic process   • phosphate-containing compound metabolic process   • polyol biosynthetic process   • small molecule metabolic process   • phosphorus metabolic process   • regulation of carbohydrate metabolic process   • regulation of biosynthetic process   • carbohydrate metabolic process   • polyol metabolic process   • positive regulation of phosphorus metabolic process   • regulation of alcohol biosynthetic process   • small molecule biosynthetic process   • carbohydrate biosynthetic process   • primary metabolic process   • positive regulation of inositol phosphate biosynthetic process   • biosynthetic process   • organophosphate metabolic process   • organophosphate biosynthetic process   • inositol phosphate biosynthetic process   • alcohol biosynthetic process   • metabolic process   • regulation of phosphorus metabolic process   • positive regulation of carbohydrate metabolic process   • regulation of carbohydrate biosynthetic process   • positive regulation of small molecule metabolic process   • regulation of metabolic process   • positive regulation of alcohol biosynthetic process   • multicellular organismal-level homeostasis   • tissue remodeling   • bone remodeling   • anatomical structure homeostasis   • tissue homeostasis   • bone resorption   • G protein-coupled receptor signaling pathway, coupled to cyclic nucleotide second messenger   • intracellular anatomical structure   • nucleus   • membrane-enclosed lumen   • intracellular membraneless organelle   • intracellular membrane-bounded organelle   • nucleolus   • intracellular organelle lumen   • intracellular organelle   • organelle lumen   • membraneless organelle   • nuclear lumen   • apical part of cell   • plasma membrane region   • apical plasma membrane   • cytoplasm   • cytosol   • basal part of cell   • basal plasma membrane   • basolateral plasma membrane   • receptor complex   • enzyme binding   • GTPase binding   • protein-containing complex binding   • pyrophosphatase activity   • GTPase activity   • ribonucleoside triphosphate phosphatase activity   • hydrolase activity, acting on acid anhydrides, in phosphorus-containing anhydrides   • hydrolase activity   • hydrolase activity, acting on acid anhydrides   • catalytic activity   • signaling receptor complex adaptor activity   • protein-macromolecule adaptor activity   • molecular adaptor activity   • signaling adaptor activity   • system process   • sensory perception of chemical stimulus   • sensory perception   • nervous system process   • sensory perception of taste   • sensory organ development   • eye development   • retina development in camera-type eye   • visual system development   • camera-type eye development   • sensory system development   • response to ketone   • response to prostaglandin   • response to lipid   • response to endogenous stimulus   • response to alcohol   • cellular response to prostaglandin stimulus   • response to oxygen-containing compound   • cellular response to oxygen-containing compound   • cellular response to endogenous stimulus   • cellular response to prostaglandin E stimulus   • cellular response to chemical stimulus   • cellular response to alcohol   • response to hormone   • response to chemical   • cellular response to lipid   • response to prostaglandin E   • cellular response to ketone   • cellular response to hormone stimulus   • small GTPase-mediated signal transduction   • Ras protein signal transduction   • intracellular signal transduction   • intracellular signaling cassette   • cellular response to nitrogen compound   • response to dopamine   • cellular response to dopamine   • response to monoamine   • response to catecholamine   • adenylate cyclase-activating dopamine receptor signaling pathway   • cellular response to catecholamine stimulus   • G protein-coupled dopamine receptor signaling pathway   • response to nitrogen compound   • cellular response to monoamine stimulus   • synaptic signaling   • cellular response to acetylcholine   • cell-cell signaling   • acetylcholine receptor signaling pathway   • postsynaptic signal transduction   • G protein-coupled acetylcholine receptor signaling pathway   • response to acetylcholine   • non-motile cilium   • 9+0 non-motile cilium   • cilium   • neuron projection   • photoreceptor disc membrane   • photoreceptor outer segment   • plasma membrane bounded cell projection   • cell projection   • photoreceptor cell cilium   • organelle membrane   • vacuolar membrane   • lytic vacuole   • vacuole   • lytic vacuole membrane   • bounding membrane of organelle   • lysosomal membrane   • lysosome
SCOP2Domain Identifier• Transducin (heterotrimeric G protein), gamma chain   • G protein-coupled receptor-like
SCOP2Family Identifier• Transducin (heterotrimeric G protein), gamma chain   • G protein-coupled receptor-like
Membrane Protein Annotations-• Orientations of Proteins in Membranes database (OPM)   • Protein Data Bank of Transmembrane Proteins (PDBTM)   • MemProtMD


Details about the values in these tables can be found in the corresponding documentation page .
PDBsumOpen PDBsum Page
ChainA
ProteinG Protein α Sub unit
UniProtP63092
Sequence
>8YG4_Chain_A
LSAEDKAAV ERSKMIEKQ LQKDKQVYR ATHRLLLLG ADNSGKSTI 
VKQMRIYHV TSGIFETKF QVDKVNFHM FDVGAQRDE RRKWIQCFN 
DVTAIIFVV DSSDYNRLQ EALNDFKSI WNNRWLRTI SVILFLNKQ 
DLLAEKVLA GKSKIEDYF PEFARYTTP EDATPEPGE DPRVTRAKY 
FIRDEFLRI STASGDGRH YCYPHFTCS VDTENARRI FNDCRDIIQ 
RMHLRQYEL L


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainB
ProteinG Protein β Sub unit
UniProtP62873
Sequence
>8YG4_Chain_B
ELDQLRQEA EQLKNQIRD ARKACADAT LSQITNNID PVGRIQMRT 
RRTLRGHLA KIYAMHWGT DSRLLVSAS QDGKLIIWD SYTTNKVHA 
IPLRSSWVM TCAYAPSGN YVACGGLDN ICSIYNLKT REGNVRVSR 
ELAGHTGYL SCCRFLDDN QIVTSSGDT TCALWDIET GQQTTTFTG 
HTGDVMSLS LAPDTRLFV SGACDASAK LWDVREGMC RQTFTGHES 
DINAICFFP NGNAFATGS DDATCRLFD LRADQELMT YSHDNIICG 
ITSVSFSKS GRLLLAGYD DFNCNVWDA LKADRAGVL AGHDNRVSC 
LGVTDDGMA VATGSWDSF LKIWN


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainG
ProteinG Protein γ Sub unit
UniProtP59768
Sequence
>8YG4_Chain_G
TASIAQARK LVEQLKMEA NIDRIKVSK AAADLMAYC EAHAKEDPL 
LTPVPASEN PFR


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

ChainR
ProteinReceptor
UniProtQ03431
Sequence
>8YG4_Chain_R
VMTKEEQIF LLHRAQAQT REREVFDRL GMIYTVGYS VSLASLTVA 
VLILAYFRR LHCTRNYIH MHLFLSFML RAVSIFVKD AVLYSAGYA 
GCRVAVTFF LYFLATNYY WILVEGLYL HSLIFMAFF SEKKYLWGF 
TVFGWGLPA VFVAVWVSV RATLANTGC WDLSSGNKK WIIQVPILA 
SIVLNFILF INIVRVLAT KLRETNTRQ QYRKLLKST LVLMPLFGV 
HYIVFMATP YTEVSGTLW QVQMHYEML FNSFQGFFV AIIYCFCNG 
EVQAEIKKS WSRWTLAL


Click on each residue to open a popup with some information about it.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  




This receptor, from the same or other species and bound to the same or other ligands, is also present in the following networks:
Show PDB Class SubFamily Type SubType Species Orthosteric Ligand Other Ligand(s) Protein Partners Resolution Date DOI
6FJ3B1PeptideParathyroid HormonePTH1Homo sapiensPTH--2.52018-11-21doi.org/10.1038/s41594-018-0151-4
6NBFB1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-Gs/β1/γ232019-04-17doi.org/10.1126/science.aav7942
6NBF (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-32019-04-17doi.org/10.1126/science.aav7942
6NBHB1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-Gs/β1/γ23.52019-04-17doi.org/10.1126/science.aav7942
6NBH (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-3.52019-04-17doi.org/10.1126/science.aav7942
6NBIB1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-Gs/β1/γ242019-04-17doi.org/10.1126/science.aav7942
6NBI (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-42019-04-17doi.org/10.1126/science.aav7942
7VVJB1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-Gs/β1/γ23.22022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVJ (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-3.22022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVKB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ23.32022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVK (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.32022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVLB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ22.82022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVL (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVMB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ23.22022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVM (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.22022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVNB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ23.82022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVN (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.82022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVOB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ24.12022-08-03doi.org/10.1016/j.molcel.2022.07.003
7VVO (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-4.12022-08-03doi.org/10.1016/j.molcel.2022.07.003
8HA0B1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1-Gs)/β1/γ22.622022-12-21doi.org/10.1038/s41401-022-01032-z
8HA0 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.622022-12-21doi.org/10.1038/s41401-022-01032-z
8HAFB1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-chim(NtGi1-Gs)/β1/γ23.252022-12-21doi.org/10.1038/s41401-022-01032-z
8HAF (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-3.252022-12-21doi.org/10.1038/s41401-022-01032-z
8HAOB1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1-Gs)/β1/γ23.762022-12-21doi.org/10.1038/s41401-022-01032-z
8HAO (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-3.762022-12-21doi.org/10.1038/s41401-022-01032-z
8FLQB1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ22.552023-04-26doi.org/10.1016/j.str.2023.04.002
8FLQ (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.552023-04-26doi.org/10.1016/j.str.2023.04.002
8FLRB1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-Gs/β1/γ22.942023-04-26doi.org/10.1016/j.str.2023.04.002
8FLR (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTHrP(1-36)-2.942023-04-26doi.org/10.1016/j.str.2023.04.002
8FLSB1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-Gs/β1/γ23.092023-04-26doi.org/10.1016/j.str.2023.04.002
8FLS (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-3.092023-04-26doi.org/10.1016/j.str.2023.04.002
8FLTB1PeptideParathyroid HormonePTH1Homo sapiensM-PTH(1-14)-Gs/β1/γ23.032023-04-26doi.org/10.1016/j.str.2023.04.002
8FLT (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensM-PTH(1-14)-3.032023-04-26doi.org/10.1016/j.str.2023.04.002
8FLUB1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-Gs/β1/γ22.762023-04-26doi.org/10.1016/j.str.2023.04.002
8FLU (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-2.762023-04-26doi.org/10.1016/j.str.2023.04.002
8GW8B1PeptideParathyroid HormonePTH1Homo sapiens-PCO371Gs/β1/γ22.92023-06-14doi.org/10.1038/s41586-023-06169-3
8GW8 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiens-PCO3712.92023-06-14doi.org/10.1038/s41586-023-06169-3
7Y35B1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-Gs/β1/γ22.92023-07-05To be published
7Y35 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensAbaloparatide-2.92023-07-05To be published
7Y36B1PeptideParathyroid HormonePTH1Homo sapiensPTH-Gs/β1/γ22.82023-07-05To be published
7Y36 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82023-07-05To be published
8JR9B1PeptideParathyroid HormonePTH1Homo sapiens-PCO371chim(NtGi1-Gs)/β1/γ22.572023-08-02doi.org/10.1038/s41586-023-06467-w
8JR9 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiens-PCO3712.572023-08-02doi.org/10.1038/s41586-023-06467-w
9LXRB1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-Arrestin23.072025-09-10To be published
9JR2B1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1L-Gs-CtGq)/β1/γ22.82024-10-16doi.org/10.1038/s41589-025-01957-6
9JR2 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82024-10-16doi.org/10.1038/s41589-025-01957-6
9JR3B1PeptideParathyroid HormonePTH1Homo sapiensPTH-chim(NtGi1L-Gs-CtGq)/β1/γ22.82024-10-16doi.org/10.1038/s41589-025-01957-6
9JR3 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensPTH-2.82024-10-16doi.org/10.1038/s41589-025-01957-6
9B5YB1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-chim(NtGi1-Gq)/β1/γ23.492025-03-19doi.org/10.1073/pnas.2426178122
9B5Y (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-3.492025-03-19doi.org/10.1073/pnas.2426178122
8YFOB1PeptideParathyroid HormonePTH1Homo sapiensAc-LA-PTH Analog-chim(NtGi1-Gs)/β1/γ22.712025-09-03To be published
8YFO (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensAc-LA-PTH Analog-2.712025-09-03To be published
8YG4B1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-chim(NtGi1-Gs)/β1/γ22.592025-09-03To be published
8YG4 (No Gprot) B1PeptideParathyroid HormonePTH1Homo sapiensLA-PTH Analog-2.592025-09-03To be published




You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download 8YG4.zip



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