Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1NT 42.25321215
21x39 3.58172417
31x43 4.40302406
41x50 4.82076409
51x60 3.02543405
62x39 3.91091508
72x40 2.89585508
82x42 3.77884407
92x44 3.14146405
102x45 5.19364479
112x46 3.88859579
122x50 5.78235679
132x60 3.96906417
14E1x52 2.08603407
153x32 4.71933415
163x34 3.81553405
173x42 5.63816578
183x44 3.37997407
193x46 5.16198409
203x49 4.13102508
214x53 3.19022408
224x60 3.42738515
23E2 6.359832114
245x40 1.46646504
255x44 3.38265415
265x47 3.9493408
275x58 3.57723509
286x32 1.52596407
296x48 6.40196578
306x49 2.13143406
316x51 2.96859516
32E3 2.126071012
337x38 4.32794415
347x45 5.30954479
357x47 2.56687407
367x53 4.68222509
378x58 1.06182406
38Lig 9.074943010
39G.HN.33 2.02742404
40G.S1.06 4.432694179
41G.s1h1.04 1.6287409
42G.H1.01 2.552325179
43G.H1.07 1.19348509
44G.S2.02 0.827737405
45G.S2.03 5.22937439
46G.S2.04 1.59136407
47G.S2.06 3.80825508
48G.S2.08 4.44065565
49G.S3.01 3.65111465
50G.S3.03 5.70135667
51G.S3.04 8.66077437
52G.S3.06 7.85981536
53G.S3.07 3.177884179
54G.H2.06 5.8252529
55G.H2.07 4.80971629
56G.h2s4.01 7.95721409
57G.h2s4.02 4.69755437
58G.H3.01 2.44972709
59G.H3.09 5.16882609
60G.H3.13 6.38271405
61G.H3.17 6.29033734
62G.H3.18 5.100144169
63G.S5.05 3.120257189
64G.S5.07 3.11618509
65G.hgh4.02 4.196055199
66G.hgh4.05 6.0192607
67G.hgh4.08 4.84504403
68G.H4.05 3.06167604
69G.H4.10 7.890115197
70G.H4.12 5.66222485
71G.H4.15 6.18961408
72G.H4.16 2.43077483
73G.S6.02 5.72672508
74G.S6.05 5.23717585
75G.H5.03 3.156775188
76G.H5.08 4.78353668
77G.H5.17 4.635144206
78G.H5.20 3.49859408
79b.1x1 1.21631504
80b.1x3 1.23904401
81b.1x4 1.50011608
82b.lh12x2 3.35867408
83b.h2x1 3.06088405
84b.lhb1x3 2.80615402
85b.lhb1x6 4.280014133
86b.lhb1x11 3.15999404
87b.b1x4 3.475464107
88b.l1x3 8.95098549
89b.l1x6 8.48228539
90b.b2x1 6.24458538
91b.b2x5 6.24812647
92b.b3x3 3.55333598
93b.l3x1 7.10649439
94b.l3x2 6.27312409
95b.b4x2 4.94923408
96b.b4x3 4.29978497
97b.b4x6 8.64033749
98b.l4x2 9.117554104
99b.b5x2 6.56433407
100b.b5x3 6.17408649
101b.b5x5 4.62464405
102b.b5x7 5.35308407
103b.l5x1 3.98863598
104b.l5x5 8.06709639
105b.b6x5 3.75164696
106b.l6x5 4.933044144
107b.b7x1 5.211485144
108b.l7x4 3.3105409
109b.b8x4 5.32989596
110b.l9x3 6.44786629
111b.l9x6 4.7065828
112b.b10x5 4.58744509
113b.b11x4 5.27853429
114b.l11x2 7.7195429
115b.b12x6 8.52378628
116b.b13x7 7.57982557
117b.l13x3 7.35127659
118b.l13x6 4.921529
119b.l13x7 4.50424459
120b.b14x3 3.85659455
121b.b15x1 6.45005559
122b.b15x3 4.58938459
123b.l15x1 5.25956427
124b.l15x2 6.21031459
125b.b16x4 9.79486456
126b.b16x6 7.61063758
127b.b17x5 6.87955427
128b.b17x7 8.11484428
129b.l17x3 7.90822729
130b.l17x6 6.54416529
131b.b18x3 4.79511428
132b.l18x1 5.562588126
133b.l18x2 5.27414127
134b.l18x3 6.083595125
135b.b19x2 6.44144626
136b.b19x4 6.0572428
137b.l19x2 6.67329529
138b.b20x4 10.4896528
139b.b20x6 5.91474726
140b.l20x2 4.25854609
141b.b21x1 5.7016627
142b.b21x2 2.85311406
143b.b21x5 5.19794404
144b.b21x7 5.59459605
145b.l21x2 4.95368404
146b.b22x5 5.391295127
147b.l22x1 3.49839409
148b.l22x5 5.848346139
149b.b23x6 7.030596157
150b.l23x1 6.81288436
151b.b24x4 7.472244156
152b.b24x6 6.749464158
153b.l24x2 3.33675506
154b.b25x3 4.784335155
155b.l25x3 8.565375119
156b.l25x4 3.04673405
157b.l25x6 13.0124438
158b.l26x5 4.12784405
159b.l27x1 8.95289839
160b.l27x2 7.703314119
161b.b28x2 4.57513404
162b.b28x3 4.14958547
163b.b28x4 7.198044116
164b.b28x6 8.355245119
165g.h2x11 8.247394129
166g.ctx3 5.76269504
167g.ctx6 3.05255135
168G.HN.11 0.576906600
169G.HN.37 2.00488400
170g.h1x1 1.19723500
171g.h1x12 1.45432400
172g.l1x4 4.32619400
173g.ctx14 4.938784100
174g.ctx15 6.102514100
175g.ctx16 4.596748100
176E1 3.956651010
1774x64 5.11517410
178G.hgh4.13 0.445793400
179G.hgh4.20 2.35564500
180I2 3.59792860
181H.HA.07 0.0451177400
182H.HA.16 0.0505188400
183H.HB.02 0.0551862400
184H.HB.05 0.0640579400
185H.hbhc.14 0.077558400
186H.hchd.01 0.0615495400
187H.HD.07 0.0755815400
188H.hdhe.01 0.0583264600
189H.HE.04 0.134482400
190H.HE.05 0.0552476500
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
12x50 3x39 17.666510.2983YesNo099
22x53 3x39 17.39655.52128NoNo079
32x53 3x36 17.26144.83461NoNo077
43x36 Lig 17.12516.61854NoYes170
52x40 I1x50 95.21382.90556YesNo087
62x39 2x40 94.05193.80311YesYes088
72x39 2x43 34.50273.62041YesNo088
82x43 3x46 28.45926.63773NoYes089
92x46 3x46 29.23284.71802YesYes099
102x46 2x50 22.66725.26347YesYes799
111x60 I1x50 97.52892.43674YesNo057
121x60 8x53 97.99065.36005YesNo055
13b.l2x5 b.l4x2 11.755119.7286NoYes054
14b.l4x2 g.ctx15 11.86779.92443YesYes1040
15b.l26x5 g.ctx15 14.58255.54226YesYes050
16b.l26x5 g.ctx4 17.93834.30451YesNo056
17g.ctx3 g.ctx4 18.09714.40769YesNo046
18b.l22x1 g.ctx3 1007.74924YesYes094
19b.b23x1 b.l22x1 24.96443.01648NoYes059
20b.b23x1 b.b24x5 24.94654.89406NoNo055
21b.b23x3 b.b24x5 24.91144.42847NoNo075
22b.b23x3 b.b26x3 49.78652.96669NoNo076
23b.b26x3 b.b27x3 49.68793.45306NoNo068
24b.b27x3 b.l25x3 74.50887.54332NoYes089
25b.l25x3 b.l27x2 99.06767.6938YesYes1199
26b.l25x4 b.l27x2 98.70084.81277YesYes059
27I1x49 b.l25x4 98.19124.58827NoYes055
288x53 I1x49 98.10422.76029NoNo055
29b.l22x1 g.ctx5 75.06152.89214YesNo095
30b.b27x1 g.ctx5 24.97883.00798NoNo065
31b.b23x3 b.b27x1 24.92524.34951NoNo076
32b.lhb1x11 g.ctx5 50.09473.97794YesNo045
33b.b25x7 b.lhb1x11 50.06965.80004NoYes074
34b.b25x7 b.b28x6 50.056816.66NoYes079
35b.b27x3 b.b28x6 24.9057.65675NoYes089
36b.b28x4 b.b28x6 25.11326.23605YesYes1169
37b.b28x4 b.l25x3 24.91349.96134YesYes1169
38b.l3x1 b.l5x5 10.7757.35799YesYes399
39b.l25x6 b.l27x1 26.457420.2457YesYes389
40b.l23x1 b.l25x6 26.680316.3453YesYes368
41b.l21x7 b.l23x1 84.37523.76599NoYes056
42b.l21x7 b.l23x2 84.58946.91907NoNo058
43b.b23x6 b.l23x2 84.8983.67758YesNo078
44b.b23x6 b.b24x6 85.1987.41419YesYes1578
45b.b21x7 b.b24x6 86.39198.78775YesYes058
46b.b21x5 b.b21x7 91.69589.32416YesYes045
47b.b21x5 b.h2x1 92.73186.15071YesYes045
48b.h2x1 b.h2x5 93.13943.43691YesNo055
49b.h2x5 b.lhb1x3 46.63363.19987NoYes052
50b.l22x5 b.lhb1x3 46.90464.20117YesYes092
51b.l22x5 g.ctx6 93.80594.19147YesYes1395
52g.ctx3 g.ctx6 94.35415.71724YesYes045
53b.b2x1 b.l27x1 47.10616.39155YesYes389
54G.H3.17 b.l27x1 26.44963.45848YesYes349
55G.H3.17 b.l23x1 57.47844.74258YesYes346
56b.h2x5 b.l24x2 46.61094.2555NoYes056
57b.l22x5 b.l24x2 46.7568.25172YesYes096
58G.S3.01 G.S3.03 23.49435.18205YesYes657
59G.S3.01 I2 24.00964.14171YesYes650
602x38 I2 52.25573.25576NoYes660
612x38 3x49 52.84134.66692NoYes068
62G.H5.08 G.S3.03 23.5293.48135YesYes687
63G.H5.08 I2 25.04193.21573YesYes680
64G.S1.04 G.S3.03 38.3723.39403NoYes077
65G.S1.04 G.S4.03 38.10894.2978NoNo077
66G.H3.15 G.H3.18 28.02718.29671NoYes089
67G.H3.15 G.H3.17 28.13973.45009NoYes084
68G.H2.07 G.H2.08 26.97983.18932YesNo099
69G.H2.08 G.H3.18 27.09193.69918NoYes099
70G.S5.07 G.s6h5.01 28.51315.21632YesNo099
71G.S5.05 G.s6h5.01 28.75625.0202YesNo1899
72G.S4.03 G.S5.05 34.842.96673NoYes079
73b.b6x1 b.l9x6 41.66365.07875NoYes098
74b.b2x1 b.b6x1 42.12783.62252YesNo089
75G.H2.06 b.l17x6 26.06657.6922YesYes299
76G.H2.06 b.l9x6 27.03963.5466YesYes298
77G.H2.04 G.H2.07 26.83366.04826NoYes099
78G.H2.04 G.H3.08 26.59435.86785NoNo099
79G.H3.08 G.S4.04 26.47585.80715NoNo099
80G.H3.09 G.S4.04 16.89027.79467YesNo099
81G.S4.07 G.s5hg.01 25.59063.99767NoNo089
82G.S5.07 G.s5hg.01 26.65372.93533YesNo099
83G.H3.06 G.hgh4.02 17.13532.93235NoYes069
84G.H3.06 G.H4.15 11.67637.30657NoYes068
85G.H4.10 G.hgh4.02 12.87145.96794YesYes1979
86b.l17x5 b.l17x6 25.43713.22605NoYes269
87b.l17x5 b.l19x2 25.19653.65352NoYes269
88b.l17x3 b.l19x2 23.23364.25532YesYes299
89b.b20x6 b.l17x3 19.06092.89136YesYes269
90b.b17x7 b.b20x6 14.154310.1632YesYes286
91b.b17x7 b.b21x1 11.70484.62913YesYes287
92b.l11x1 b.l9x6 11.67766.24772NoYes298
93b.b11x6 b.l11x1 11.51913.32514NoNo299
94b.b11x6 b.l9x3 10.156514.1809NoYes299
95G.H3.01 G.s4h3.03 25.11514.82571YesNo098
96G.S4.07 G.s4h3.03 25.32472.26887NoNo088
97G.H3.01 G.s1h1.04 23.11615.4502YesYes099
98G.s1h1.04 H.hehf.07 22.42890.0404167YesNo090
99H.HF.03 H.hehf.07 22.21930.102795NoNo000
100H.HF.03 H.hehf.04 18.23660.0765923NoNo000
101H.hehf.04 H.hehf.06 17.81740.105377NoNo000
102H.HA.08 H.hehf.06 17.18850.0677699NoNo000
103H.HA.08 H.HA.12 16.97890.0440087NoNo000
104H.HA.12 H.hbhc.14 16.76930.127165NoYes000
105H.HA.16 H.hbhc.14 15.09230.053948YesYes000
106H.HA.16 H.HB.12 14.46350.0639973YesNo000
107H.HB.08 H.HB.12 14.25390.0505214NoNo000
108H.HB.08 H.HC.06 12.78660.0486961NoNo000
109H.HB.05 H.HC.06 12.36730.0794409YesNo000
1102x39 3x49 57.82073.19602YesYes088
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
NTNT224.5181YesYes5511
E2NT8.863191YesYes4511
1x392x613.809751YesNo7612
1x397x424.563971YesNo7712
2x533x364.834610NoNo7721
3x26E24.630461NoYes7421
3x32Lig6.817931YesYes5010
3x33Lig5.946681NoYes4010
3x36Lig6.618541NoYes7010
5x39E23.518620NoYes6421
5x36E24.35680NoYes4421
E2E231.97371YesYes4411
E2E2x523.73871YesNo4411
E2E2x516.547481YesNo4512
E2x52Lig8.428761NoYes4010
E2Lig13.1491YesYes4010
5x43Lig3.553881NoYes5010
6x517x373.911831YesNo6611
6x51Lig3.528391YesYes6010
E3E35.024091YesYes2211
1x291x332.926831NoNo3212
2x573x322.996140NoYes7521
2x603x282.99191YesNo7512
3x22E23.135131NoYes3421
1x39Lig2.961141YesYes7010
2x60Lig5.115771YesYes7010
7x38Lig8.178211YesYes5010
1x357x382.951640NoYes5521
1x397x382.992041YesYes7511
2x563x323.694750NoYes6521
2x572x613.107940NoNo7622
4x64E24.495961YesYes0421
4x68E25.695450NoYes0421
7x347x383.189851NoYes4511
7x34Lig5.350051NoYes4010
E1NT4.515431YesYes0511
2x603x325.368481YesYes7511
E1Lig10.67331YesYes0010
3x334x603.614981NoYes4512
5x41E24.026251NoYes5411
E1E23.59491YesYes0411
3x335x434.296661NoNo4511
5x44Lig4.818021YesYes5010
7x337x374.330331NoNo4621
5x415x443.888911NoYes5511
4x604x644.89171YesYes5022
4x605x435.033131YesNo5521
E3Lig2.913121YesYes2010
LigNT40.83181YesYes0501
E1E19.82941YesYes0011
7x37Lig3.906241NoYes6010
5x41Lig3.0071NoYes5010
1x32Lig7.544680NoYes5010
1x29Lig3.826221NoYes3010
3x26E2x5111.87931NoNo7522
4x64E2x518.903361YesNo0522
5x425x443.37830NoYes4521
6x517x333.133121YesNo6412
7x30Lig2.749830NoYes4010
6x516x552.607511YesNo6512
2x602x642.400091YesNo7512
3x29Lig2.328311NoYes5010
1x25Lig2.216780NoYes0010
6x61E32.189561NoYes3221
6x54E31.964490NoYes5221
3x294x651.963241NoNo5012
6x506x511.662080NoYes9621
7x29E31.653341NoYes0221
1x28Lig1.592880NoYes3010
6x587x341.578410NoNo4421
2x65Lig1.534820NoYes4010
5x446x561.445351YesNo5612
5x38E21.339220NoYes4421
5x35E21.250331NoYes3421
1x24NT1.192751NoYes0521
2x68Lig1.076460NoYes0010
1x21Lig1.05290NoYes0010
7x27E31.051930NoYes0221
7x28NT0.9018910NoYes0521
1x26Lig0.8600350NoYes0010
2x67E10.8447290NoYes4021
7x32NT0.8409690NoYes1521
6x60E30.7890051NoYes5221
6x62E20.6123211NoYes0421
5x32E20.597761NoYes0421
1x22Lig0.5470170NoYes0010
7x26E30.5057241NoYes0221
7x24NT0.4337020NoYes0521
1x19NT0.21750NoYes0521
3x20E10.1771360NoYes0021
E1x501NT0.1465160NoYes0521
6x65E30.1453490NoYes0221
E1x48NT0.05789291NoYes0521
2x69E10.05341350NoYes0021
3x19E10.04833331NoYes0021
5x27E20.02804351NoYes0421
5x28E20.0184111NoYes0421
3x29Ca50.0178231NoNo5012
4x69E20.01090770NoYes0421
2x70E10.0004037270NoYes0021

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
89.29Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
73.53Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
67.65Consensuspth_onOrthosteric Ligandpth1_on pth2_on
65.79Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
62.07Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
62.07Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
60.53Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
59.46Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
59.38Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
58.06Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
57.58Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
57.58Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
57.58Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
56.25Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
55.56Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
55.56Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
54.84Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
54.84Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
54.55Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
54.55Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
54.55Consensusglp_onOrthosteric Ligandglp1_on glp2_on
54.55Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
54.29Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
54.29Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
54.05Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
53.12Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
53.12Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
53.12Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
53.12Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
52.94Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
52.94Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
52.94Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
52.94Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
52.94Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
52.94Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
52.94Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
52.78Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
51.52Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
51.52Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
51.52Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
51.52Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
51.52Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
51.52Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
51.52Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
51.43Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
51.35Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
51.35Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
50.00Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
50.00Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
50.00Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
50.00Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
50.00Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
50.00Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
50.00Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
50.00Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
50.00Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
50.00Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
50.00Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
48.65Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
48.65Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
48.65Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
48.57Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
48.57Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
48.48Consensuspac_onOrthosteric Ligandpac1_on
48.39Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
47.06Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
47.06Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
47.06Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
47.06Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
46.88Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
46.88Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
46.88Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
46.15Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
45.71Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
45.45Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
45.45Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
45.45Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
45.16Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
44.74Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
44.74Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
44.74Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
44.44Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
44.44Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
44.12Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
44.12Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
43.75Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
43.59Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
43.33Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
43.24Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
42.86Single6FJ3PTH6FJ3-PTH1-PTH
42.86Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
42.86Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
42.42Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
42.42Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
42.11Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
41.67Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
41.67Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
41.67Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
41.67Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
41.18Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
41.18Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
41.18Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
41.18Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
40.54Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
40.00Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
40.00Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
40.00Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
40.00Consensuscalcitonin_onOrthosteric Ligandctlike_on
39.47Single6IGKEndothelin-36IGK-ETB-Endothelin-3
38.89Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
38.89Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
38.89Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
38.89Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
38.89Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
38.71Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
38.71Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
38.46Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
38.24Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
37.84Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
37.14Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
37.14Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
37.14Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
37.14Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
37.14Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
36.84Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
36.84Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
36.84Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
36.59Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
36.36Single4XT1Fractalkine4XT1-US28-Fractalkine
36.36Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
36.11Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
35.90Single5GLHEndothelin-15GLH-ETB-Endothelin-1
35.90Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
35.90Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
35.29Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
35.14Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
35.14Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
35.14Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
35.14Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
35.14Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
35.00Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
34.38Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
34.38Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
34.29Consensusangiotensin_onOrthosteric Ligandat1_on
34.29Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
34.29Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
34.21Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
34.21Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
34.21Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
34.15Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
33.33Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
33.33Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
33.33Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
33.33Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
33.33Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
33.33Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
32.50Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
32.43Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
32.43Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
32.43Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
32.43Single8ZRTET-18ZRT-ETB-ET-1
32.43Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
32.43Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
32.43Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
32.35Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
32.35Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
32.35Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
32.35Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
32.35Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
32.35Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
32.35Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
32.35Consensuslpl_onOrthosteric Ligands1p_on lpa_on
32.35Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
32.35Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
32.26Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
32.26Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
32.26Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
32.26Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
32.26Single8E0GBU728E0G-μ-BU72
32.26Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
32.26Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
31.58Single4XT3Fractalkine4XT3-US28-Fractalkine
31.58Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
31.58Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
31.58Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
31.43Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
31.43Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
31.43Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
31.43Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
31.43Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
31.43Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
31.43Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
31.43Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
31.43Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
31.43Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
31.43Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
31.25Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
31.25Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
31.25Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
31.25Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
31.25Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
31.25Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
31.25Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
31.25Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
31.25Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
31.25Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
31.25Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
31.25Consensuslpa_offOrthosteric Ligandlpa1_off
31.25Consensuslpl_offOrthosteric Ligands1p_off lpa_off
31.11Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
30.95Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
30.95Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
30.77Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
30.77Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
30.77Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
30.77Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
30.77Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
30.77Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
30.56Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
30.56Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
30.56Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
30.56Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
30.56Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
30.56Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
30.56Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
30.56Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
30.56Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
30.56Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
30.30Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
30.30Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
30.30Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
30.30Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
30.30Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
30.30Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
30.30Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
30.23Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
30.00Single6IGLIRL16206IGL-ETB-IRL1620
30.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
30.00Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
30.00Single8IY6Endothelin-18IY6-ETB-Endothelin-1
30.00Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
30.00Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
30.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
30.00Consensusendothelin_onOrthosteric Ligandetb_on eta_on
30.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
30.00Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
30.00Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
30.00Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
29.79Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
29.73Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
29.73Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
29.73Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
29.73Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
29.73Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
29.73Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
29.73Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
29.73Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
29.73Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
29.73Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
29.73Consensusvasop-oxy_onOrthosteric Ligandv2_on
29.73Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
29.41Single3NY9ICI118-5513NY9-β2-ICI118-551
29.41Single4UG2CGS216804UG2-A2A-CGS21680
29.41Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
29.41Single8QJ2pN1628QJ2-MC4-pN162-Gs
29.41Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
29.41Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
29.41Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
29.41Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
29.41Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
29.41Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
29.41Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
29.27Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
29.27Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
29.27Consensusbombesin_onOrthosteric Ligandbb2_on
29.27Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
29.27Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
29.03Single5C1MBU725C1M-μ-BU72
29.03Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
29.03Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
29.03Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
29.03Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
29.03Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
29.03Single8JXSPF-61428JXS-D1-PF-6142
29.03Single8TF5Oleic acid8TF5-GPR6-Oleic acid
29.03Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
29.03Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
29.03Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
29.03Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
29.03Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
29.03Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
29.03Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
29.03Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
28.95Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
28.95Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
28.95Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
28.95Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
28.95Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
28.95Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
28.95Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
28.95Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
28.95Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
28.95Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
28.95Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
28.95Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
28.57Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
28.57Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
28.57Single7QA8Peptide7QA8-STE2-Peptide
28.57Single7QA8Peptide7QA8-STE2-Peptide
28.57Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
28.57Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
28.57Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
28.57Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
28.57Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
28.57Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
28.57Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
28.57Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
28.57Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
28.57Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
28.57Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.21Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
28.21Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
28.21Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
28.21Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
28.21Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
28.21Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
28.12Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
28.12Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
28.12Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
28.12Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
28.12Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.12Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
28.12Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
28.12Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
28.12Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
28.12Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
28.12Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
28.12Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
28.12Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.12Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
28.12Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
28.12Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
28.12Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
27.78Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
27.78Single7XNACYN1548067XNA-SST2-CYN154806
27.78Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
27.78Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
27.78Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
27.78Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
27.78Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
27.66Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
27.59Single6AKXA4R6AKX-CCR5-A4R
27.59Single6AKYMaraviroc6AKY-CCR5-Maraviroc
27.59Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.59Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
27.50Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
27.50Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
27.50Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
27.50Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
27.50Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
27.50Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
27.50Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
27.50Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
27.50Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
27.50Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
27.50Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
27.27Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
27.27Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
27.27Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
27.27Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
27.27Single7YITNalfurafine7YIT-κ-Nalfurafine
27.27Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
27.27Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
27.27Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
27.27Single8XYIVUF106618XYI-CXCR3-VUF10661
27.27Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
27.27Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
27.27Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
27.27Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
27.27Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
27.27Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
27.27Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
27.27Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
27.27Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
27.27Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
27.27Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
27.27Consensusorexin_onOrthosteric Ligandox2_on
27.27Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
27.27Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
27.03Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
27.03Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
27.03Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.03Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
27.03Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.03Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
26.83Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
26.83Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
26.83Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
26.83Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
26.83Consensusbradykinin_onOrthosteric Ligandbk2_on
26.83Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
26.83Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
26.83Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
26.67Single4MBSMaraviroc4MBS-CCR5-Maraviroc
26.67Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.67Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
26.67Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
26.67Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
26.67Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
26.67Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
26.67Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.47Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
26.47Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
26.47Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
26.47Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
26.47Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
26.47Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
26.47Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
26.47Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
26.47Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
26.47Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
26.47Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
26.47Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
26.47Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
26.47Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
26.47Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
26.47Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
26.47Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
26.47Consensuschemerin_onOrthosteric Ligandcml1_on
26.47Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
26.47Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
26.32Single6JODAngiotensin II6JOD-AT2-Angiotensin II
26.32Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
26.32Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
26.32Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
26.32Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
26.32Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
26.32Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
26.32Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
26.32Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
26.19Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
26.19Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
26.19Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
26.19Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
26.19Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
26.09Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
26.09Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
25.81Single2Y04Salbutamol2Y04-β1-Salbutamol
25.81Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
25.81Single7UL4Alvimopan7UL4-μ-Alvimopan
25.81Single7V3ZCP559407V3Z-CB1-CP55940
25.81Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
25.81Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
25.81Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
25.81Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
25.81Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
25.81Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
25.81Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
25.81Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
25.81Single8T1WCVN4248T1W-GPR6-CVN424
25.81Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.81Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.81Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.81Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
25.81Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
25.81Single9CHXS-Carazolol9CHX-β2-S-Carazolol
25.81Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
25.81Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
25.81Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
25.81Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
25.81Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
25.81Consensushca_on_gpOrthosteric Ligandhca2_on_gp
25.71Single5ZTYAM102575ZTY-CB2-AM10257
25.71Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
25.71Single7SK9CCX6627SK9-ACKR3-CCX662
25.71Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
25.71Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
25.71Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
25.71Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
25.71Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
25.71Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
25.71Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.71Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
25.71Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
25.71Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
25.71Single9IPYJR14a9IPY-C3aB-JR14a
25.71Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
25.71Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
25.71Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
25.64Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
25.64Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
25.64Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
25.64Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
25.64Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
25.64Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
25.64Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
25.64Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
25.64Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
25.64Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
25.64Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
25.64Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
25.58Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
25.58Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
25.58Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
25.00Single2Y03Isoprenaline2Y03-β1-Isoprenaline
25.00Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
25.00Single5JQHS-Carazolol5JQH-β2-S-Carazolol
25.00Single5TVNLSD5TVN-5-HT2B-LSD
25.00Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
25.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
25.00Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
25.00Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
25.00Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
25.00Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
25.00Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
25.00Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
25.00Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
25.00Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
25.00Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
25.00Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
25.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
25.00Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
25.00Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
25.00Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
25.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
25.00Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
25.00Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
25.00Single8WDTphotoNECA8WDT-A2A-photoNECA
25.00Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
25.00Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
25.00Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
25.00Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
25.00Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
25.00Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
25.00Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
25.00Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
25.00Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
25.00Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
25.00Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
25.00Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
25.00Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
25.00Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
25.00Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensussomatostatin_offOrthosteric Ligandsst2_off
25.00Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Consensustrace-amine_onOrthosteric Ligandta1_on
24.44Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
24.39Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
24.39Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
24.32Single3QAKUK-4320973QAK-A2A-UK-432097
24.32Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
24.32Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
24.32Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
24.32Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
24.32Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
24.32Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
24.32Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
24.32Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
24.32Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
24.32Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
24.32Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
24.32Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
24.32Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
24.32Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
24.24Single2YDVNECA2YDV-A2A-NECA
24.24Single3P0GBI1671073P0G-β2-BI167107
24.24Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
24.24Single4UHRCGS216804UHR-A2A-CGS21680
24.24Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
24.24Single5G53NECA5G53-A2A-NECA-Gs
24.24Single5XR8AM8415XR8-CB1-AM841
24.24Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
24.24Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
24.24Single6H7JIsoprenaline6H7J-β1-Isoprenaline
24.24Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
24.24Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
24.24Single6WGTLSD6WGT-5-HT2A-LSD
24.24Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
24.24Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
24.24Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
24.24Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
24.24Single7TUYGSK682753A7TUY-GPR183-GSK682753A
24.24Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
24.24Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
24.24Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
24.24Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
24.24Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
24.24Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
24.24Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
24.24Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
24.24Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
24.24Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
24.24Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
24.24Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
24.24Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
24.24Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
24.24Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
24.24Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
24.24Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
24.24Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
24.24Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
24.24Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
24.24Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
24.24Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
24.24Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
24.24Consensuslpa_onOrthosteric Ligandlpa1_on
24.24Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
24.24Consensusrelaxin_onOrthosteric Ligandrxfp4_on
24.24Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
24.24Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.24Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
24.14Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
24.14Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
24.14Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
23.81Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
23.81Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
23.81Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
23.81Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
23.68Single3OE0CVX153OE0-CXCR4-CVX15
23.68Single5WF5UK-4320975WF5-A2A-UK-432097
23.68Single6PT2KGCHM076PT2-δ-KGCHM07
23.68Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
23.68Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
23.68Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
23.68Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
23.68Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
23.68Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
23.68Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
23.68Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
23.68Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
23.68Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
23.68Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
23.53Single4LDEBI1671074LDE-β2-BI167107
23.53Single4RWADIPP-NH24RWA-δ-DIPP-NH2
23.53Single4XEENeurotensin4XEE-NTS1-Neurotensin
23.53Single4XESNeurotensin4XES-NTS1-Neurotensin
23.53Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
23.53Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
23.53Single6KQICP559406KQI-CB1-CP55940-Org27569
23.53Single6MXTSalmeterol6MXT-β2-Salmeterol
23.53Single6OS2TRV0266OS2-AT1-TRV026
23.53Single6YVRNTS8-136YVR-NTS1-NTS8-13
23.53Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
23.53Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
23.53Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
23.53Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
23.53Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
23.53Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
23.53Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
23.53Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
23.53Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
23.53Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
23.53Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
23.53Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
23.53Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
23.53Single8JJ8Formoterol8JJ8-β2-Formoterol
23.53Single8JJLOlodaterol8JJL-β2-Olodaterol
23.53Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
23.53Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
23.53Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
23.53Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
23.53Single9DGIZ85267113509DGI-CB1-Z8526711350
23.53Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
23.53Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
23.53Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
23.53Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
23.53Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
23.53Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
23.40Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
23.33Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
23.33Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
23.33Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
23.33Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
23.33Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
23.33Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
23.33Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
23.33Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
23.33Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.33Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
23.33Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
23.33Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
23.33Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
23.33Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
23.33Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
23.33Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
23.33Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
23.33Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
23.33Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
23.33Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
23.33Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
23.33Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
23.33Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
23.33Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
23.33Consensusorexin_offOrthosteric Ligandox2_off ox1_off
23.33Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
23.33Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
23.33Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
23.33Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
23.26Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
23.26Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
23.26Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
23.08Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
23.08Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
23.08Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
23.08Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
23.08Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
23.08Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
23.08Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
23.08Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
23.08Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
22.86Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
22.86Single4BUONeurotensin4BUO-NTS1-Neurotensin
22.86Single5X93K-87945X93-ETB-K-8794
22.86Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
22.86Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
22.86Single7EZCUKA7EZC-A2A-UKA
22.86Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
22.86Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
22.86Single7UM4AS26747237UM4-5-HT5A-AS2674723
22.86Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
22.86Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.86Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
22.86Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
22.86Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
22.86Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
22.86Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
22.86Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
22.86Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
22.86Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.86Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
22.86Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
22.86Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
22.86Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
22.86Consensusendothelin_offOrthosteric Ligandetb_off
22.86Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
22.86Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.86Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.86Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
22.86Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
22.86Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
22.86Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
22.73Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
22.58Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
22.58Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
22.58Single4ZJCSB-6740424ZJC-OX1-SB-674042
22.58Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
22.58Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
22.58Single6PS0S-Carazolol6PS0-β2-S-Carazolol
22.58Single6PS4ICI118-5516PS4-β2-ICI118-551
22.58Single6PS5S-Propranolol6PS5-β2-S-Propranolol
22.58Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
22.58Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
22.58Single6TPGEMPA6TPG-OX2-EMPA
22.58Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
22.58Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
22.58Single7F61PF-036547467F61-H3-PF-03654746
22.58Single7T32ZM-2413857T32-A2A-ZM-241385
22.58Single7UL3Famotidine7UL3-H2-Famotidine
22.58Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
22.58Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
22.58Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
22.58Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
22.58Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
22.58Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
22.58Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
22.58Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
22.58Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
22.58Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.58Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.58Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
22.58Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
22.58Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
22.58Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
22.58Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
22.58Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
22.58Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
22.58Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
22.58Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
22.58Single8K5CAcipimox8K5C-HCA2-Acipimox
22.58Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
22.58Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
22.58Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.58Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.58Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
22.58Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
22.58Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
22.58Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
22.58Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
22.58Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
22.58Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
22.58Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
22.58Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
22.58Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
22.58Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
22.58Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
22.58Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
22.58Consensusgrh_offOrthosteric Ligandgnrh1_off
22.58Consensushca_onOrthosteric Ligandhca2_on
22.50Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
22.50Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
22.50Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
22.22Single5WF6UK-4320975WF6-A2A-UK-432097
22.22Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
22.22Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
22.22Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
22.22Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
22.22Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
22.22Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
22.22Single7XN9L-054,5227XN9-SST2-L-054,522
22.22Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
22.22Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
22.22Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
22.22Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
22.22Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
22.22Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
21.95Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
21.95Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
21.95Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
21.95Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
21.95Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
21.88Single3NY8ICI118-5513NY8-β2-ICI118-551
21.88Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
21.88Single4GBRS-Carazolol4GBR-β2-S-Carazolol
21.88Single4QKX35V4QKX-β2-35V
21.88Single4YAYZD-71554YAY-AT1-ZD-7155
21.88Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
21.88Single6H7MSalbutamol6H7M-β1-Salbutamol
21.88Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
21.88Single6PS1Timolol6PS1-β2-Timolol
21.88Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
21.88Single6TOTLemborexant6TOT-OX1-Lemborexant
21.88Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
21.88Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
21.88Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
21.88Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
21.88Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
21.88Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
21.88Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
21.88Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
21.88Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
21.88Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
21.88Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
21.88Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
21.88Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
21.88Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
21.88Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
21.88Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
21.88Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
21.88Single7WC7Lisuride7WC7-5-HT2A-Lisuride
21.88Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
21.88Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
21.88Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
21.88Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
21.88Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
21.88Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
21.88Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
21.88Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
21.88Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
21.88Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
21.88Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
21.88Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
21.88Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
21.88Single8JXRLSD8JXR-D1-LSD
21.88Single8K5DGSK2560738K5D-HCA2-GSK256073
21.88Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
21.88Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
21.88Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
21.88Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
21.88Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
21.88Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
21.88Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
21.88Single9AS1DMT9AS1-5-HT2A-DMT
21.88Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
21.88Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
21.88Consensus5ht5_onOrthosteric Ligand5ht5a_on
21.88Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
21.88Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
21.88Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
21.88Consensusa3_onOrthosteric Liganda3a_on
21.88Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
21.88Consensusdopamine_offOrthosteric Ligandd2_off d3_off
21.88Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
21.88Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
21.88Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
21.88Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
21.88Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
21.88Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
21.88Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
21.62Single4IARErgotamine4IAR-5-HT1B-Ergotamine
21.62Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
21.62Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
21.62Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
21.62Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
21.62Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
21.62Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
21.62Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
21.62Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
21.62Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
21.62Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
21.62Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
21.62Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.62Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
21.62Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
21.62Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
21.62Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
21.62Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
21.62Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
21.62Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
21.62Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
21.43Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
21.43Single9KDFRES-701-39KDF-ETB-RES-701-3
21.43Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
21.43Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
21.28Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
21.21Single2RH1S-Carazolol2RH1-β2-S-Carazolol
21.21Single2YCWS-Carazolol2YCW-β1-S-Carazolol
21.21Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
21.21Single5D6LS-Carazolol5D6L-β2-S-Carazolol
21.21Single5N2RPSB-365N2R-A2A-PSB-36-Na
21.21Single5N2SPSB365N2S-A1-PSB36
21.21Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
21.21Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
21.21Single5WIUNemonapride5WIU-D4-Nemonapride
21.21Single5WIVNemonapride5WIV-D4-Nemonapride-Na
21.21Single5WQCEMPA5WQC-OX2-EMPA
21.21Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
21.21Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
21.21Single6D26Fevipiprant6D26-DP2-Fevipiprant
21.21Single6E67BI1671076E67-β2-BI167107-Gs(CT)
21.21Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
21.21Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
21.21Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
21.21Single6PS6Timolol6PS6-β2-Timolol
21.21Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
21.21Single6TP6Filorexant6TP6-OX1-Filorexant
21.21Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
21.21Single7C4SS1P7C4S-S1P3-S1P
21.21Single7C61Ergotamine7C61-5-HT1B-Ergotamine
21.21Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
21.21Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
21.21Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
21.21Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
21.21Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
21.21Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
21.21Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
21.21Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.21Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.21Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
21.21Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
21.21Single8S4DCMF-0198S4D-Apelin-CMF-019
21.21Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
21.21Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
21.21Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
21.21Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
21.21Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
21.21Single9EHSLUF76029EHS-A3A-LUF7602
21.21Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
21.21Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
21.21Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.21Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
21.21Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
21.21Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
21.21Consensusa3_on_gpOrthosteric Liganda3a_on_gp
21.21Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
21.21Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
21.21Consensusadenosine_offOrthosteric Liganda1_off a2_off
21.21Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
21.21Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
21.21Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
21.21Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
21.21Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
21.21Consensusamine_offonOrthosteric Ligandamine_off amine_on
21.21Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
21.21Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
21.21Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
21.21Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
21.21Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
21.21Consensusdp_offOrthosteric Liganddp2_off
21.21Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
21.21Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
21.21Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
21.21Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.21Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.21Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
21.21Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.21Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.21Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
21.05Single6HLOAprepitant6HLO-NK1-Aprepitant
21.05Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
21.05Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
21.05Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
21.05Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
21.05Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
21.05Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
21.05Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
21.05Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
21.05Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
21.05Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
21.05Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
20.69Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
20.69Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
20.69Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
20.69Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
20.59Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
20.59Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
20.59Single4BV0Neurotensin4BV0-NTS1-Neurotensin
20.59Single4DJHJDTic4DJH-κ-JDTic
20.59Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
20.59Single5D5AS-Carazolol5D5A-β2-S-Carazolol
20.59Single5D5BS-Carazolol5D5B-β2-S-Carazolol
20.59Single5V54Methiothepin5V54-5-HT1B-Methiothepin
20.59Single5XRAAM115425XRA-CB1-AM11542
20.59Single6J21Aprepitant6J21-NK1-Aprepitant
20.59Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
20.59Single6TQ7SB-3348676TQ7-OX1-SB-334867
20.59Single7B6WCyclazosin7B6W-α1b-Cyclazosin
20.59Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
20.59Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
20.59Single7FEECP559407FEE-CB1-CP55940-ZCZ011
20.59Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
20.59Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
20.59Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
20.59Single7PX4PSB-21137PX4-A2A-PSB-2113
20.59Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
20.59Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
20.59Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
20.59Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
20.59Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.59Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
20.59Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
20.59Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
20.59Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
20.59Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
20.59Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
20.59Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
20.59Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
20.59Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
20.59Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.59Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
20.59Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.59Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
20.59Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
20.59Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
20.59Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
20.59Single8ZWFJR14a8ZWF-C3aB-JR14a
20.59Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
20.59Single9BJKNaloxone9BJK-μ-Naloxone-NAM
20.59Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
20.59Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
20.59Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
20.59Consensus5ht1_offOrthosteric Ligand5ht1b_off
20.59Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
20.59Consensusa2_onOrthosteric Liganda2b_on
20.59Consensusa2_on_gpOrthosteric Liganda2b_on_gp
20.59Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
20.59Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
20.59Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
20.59Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
20.59Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
20.59Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
20.59Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
20.59Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
20.59Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
20.59Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
20.59Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
20.59Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
20.59Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
20.59Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
20.59Consensusneurotensin_onOrthosteric Ligandnts1_on
20.59Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.51Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
20.51Single6W25SHU91196W25-MC4-SHU9119-Ca
20.51Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.51Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
20.51Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
20.51Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
20.51Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
20.45Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
20.00Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
20.00Single3D4STimolol3D4S-β2-Timolol
20.00Single3OE9IT1t3OE9-CXCR4-IT1t
20.00Single4AMIBucindolol4AMI-β1-Bucindolol
20.00Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
20.00Single5CXVTiotropium5CXV-M1-Tiotropium
20.00Single6A93Risperidone6A93-5-HT2A-Risperidone
20.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
20.00Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
20.00Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
20.00Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
20.00Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
20.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
20.00Single6ZG4HTL00099366ZG4-M1-HTL0009936
20.00Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
20.00Single7DFPSpiperone7DFP-D2-Spiperone
20.00Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
20.00Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.00Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
20.00Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
20.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
20.00Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
20.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
20.00Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
20.00Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
20.00Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
20.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
20.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
20.00Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
20.00Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
20.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
20.00Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
20.00Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
20.00Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
20.00Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
20.00Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
20.00Single8K5BNiacin8K5B-HCA2-Niacin
20.00Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
20.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
20.00Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
20.00Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
20.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
20.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
20.00Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
20.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
20.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
20.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
20.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.00Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.00Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.00Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
20.00Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
20.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
20.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
20.00Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
20.00Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
20.00Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
20.00Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
20.00Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
20.00Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
20.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
20.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
20.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
20.00Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
20.00Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
20.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.00Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.51Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
19.51Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
19.51Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
19.51Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.51Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
19.44Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
19.44Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
19.44Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
19.44Single6H7LDobutamine6H7L-β1-Dobutamine
19.44Single6IBLArformoterol6IBL-β1-Arformoterol
19.44Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
19.44Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
19.44Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
19.44Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
19.44Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
19.44Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
19.44Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
19.44Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
19.44Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
19.44Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
19.44Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
19.44Consensuscck_onOrthosteric Ligandccka_on cckb_on
19.44Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
19.44Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Consensusprostanoid_offOrthosteric Ligandep_off dp_off
19.35Single3ODUIT1t3ODU-CXCR4-IT1t
19.35Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
19.35Single4BWBNeurotensin4BWB-NTS1-Neurotensin
19.35Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
19.35Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
19.35Single5WS3EMPA5WS3-OX2-EMPA
19.35Single6B73MP11046B73-κ-MP1104
19.35Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
19.35Single6ME2Ramelteon6ME2-MT1-Ramelteon
19.35Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
19.35Single6TODEMPA6TOD-OX1-EMPA-Na
19.35Single7BR3Elagolix7BR3-GnRH1-Elagolix
19.35Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
19.35Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
19.35Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
19.35Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
19.35Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
19.35Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
19.35Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
19.35Single7XRRLemborexant7XRR-OX2-Lemborexant
19.35Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
19.35Single8GNGIstradefylline8GNG-A2A-Istradefylline
19.35Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
19.35Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
19.35Single8IWESpermidine8IWE-TA9-Spermidine
19.35Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
19.35Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
19.35Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.35Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.35Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.35Single8Y0HVUF114188Y0H-CXCR3-VUF11418
19.35Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
19.35Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
19.35Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
19.35Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
19.35Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
19.35Consensusalpha2_offOrthosteric Ligandalpha2c_off
19.35Consensusangiotensin_offOrthosteric Ligandat1_off
19.35Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
19.35Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
19.35Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
19.05Single7SK3CXCL127SK3-ACKR3-CXCL12
19.05Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
19.05Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
18.92Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
18.92Single6PT3DPI-2876PT3-δ-DPI-287
18.92Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
18.92Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
18.92Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
18.92Single8X5YAstemizole8X5Y-H1-Astemizole
18.92Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
18.92Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
18.92Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
18.92Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
18.92Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
18.92Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
18.92Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.92Consensuskisspeptin_onOrthosteric Ligandkiss1_on
18.75Single2YDOAdenosine2YDO-A2A-Adenosine
18.75Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
18.75Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
18.75Single5IU7Q274563465IU7-A2A-Q27456346-Na
18.75Single5IUBQ274563445IUB-A2A-Q27456344-Na
18.75Single5JTBZM-2413855JTB-A2A-ZM-241385
18.75Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
18.75Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
18.75Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
18.75Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
18.75Single6A94Zotepine6A94-5-HT2A-Zotepine
18.75Single6KUXRS-799486KUX-α2a-RS-79948
18.75Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
18.75Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
18.75Single6TPNHTL66416TPN-OX2-HTL6641
18.75Single6V9SGTPL114036V9S-OX1-GTPL11403
18.75Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
18.75Single7AROLUF58337ARO-A2A-LUF5833-Na
18.75Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
18.75Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
18.75Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
18.75Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
18.75Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
18.75Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
18.75Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
18.75Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
18.75Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
18.75Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
18.75Single8IHKAcifran8IHK-HCA3-Acifran
18.75Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
18.75Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
18.75Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
18.75Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
18.75Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
18.75Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
18.75Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
18.75Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
18.75Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
18.75Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
18.75Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
18.75Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
18.75Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
18.75Single9ARXSerotonin9ARX-5-HT2A-Serotonin
18.75Single9AS5Mescaline9AS5-5-HT2A-Mescaline
18.75Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
18.75Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
18.75Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
18.75Consensusa2_offOrthosteric Liganda2a_off
18.75Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
18.75Consensusalpha1_onOrthosteric Ligandalpha1a_on
18.75Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
18.75Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
18.75Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
18.75Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
18.75Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
18.75Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
18.75Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
18.75Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
18.60Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
18.60Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
18.42Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
18.42Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
18.42Single7F8XNN90567F8X-CCKA-NN9056
18.42Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
18.42Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
18.42Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
18.42Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
18.42Single8IEBA1LYA8IEB-GPR156-A1LYA
18.42Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
18.42Single8KIGSHU91198KIG-MC3-SHU9119-Ca
18.42Single8WKYPG-9348WKY-MC4-PG-934
18.42Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
18.42Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
18.42Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.42Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
18.42Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.42Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.42Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
18.18Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
18.18Single2Y01Dobutamine2Y01-β1-Dobutamine
18.18Single2Y02Carmoterol2Y02-β1-Carmoterol
18.18Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
18.18Single3EMLZM-2413853EML-A2A-ZM-241385
18.18Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
18.18Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
18.18Single4DAJTiotropium4DAJ-M3-Tiotropium
18.18Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
18.18Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
18.18Single4EJ4Naltrindole4EJ4-δ-Naltrindole
18.18Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
18.18Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
18.18Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
18.18Single5IU8Q274563475IU8-A2A-Q27456347-Na
18.18Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
18.18Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
18.18Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
18.18Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
18.18Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
18.18Single5T04Neurotensin5T04-NTS1-Neurotensin
18.18Single5TGZAM65385TGZ-CB1-AM6538
18.18Single5UENDU1725UEN-A1-DU172
18.18Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
18.18Single6D27CAY104716D27-DP2-CAY10471
18.18Single6DRXLisuride6DRX-5-HT2B-Lisuride
18.18Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
18.18Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
18.18Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
18.18Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
18.18Single6S0LZM-2413856S0L-A2A-ZM-241385
18.18Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
18.18Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
18.18Single7BU7BI1671077BU7-β1-BI167107
18.18Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
18.18Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.18Single7PYRPSB-21157PYR-A2A-PSB-2115
18.18Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
18.18Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
18.18Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
18.18Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
18.18Single8CU6LJ-45178CU6-A2A-LJ-4517
18.18Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
18.18Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
18.18Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
18.18Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
18.18Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
18.18Single8JJOAlprenolol8JJO-β2-Alprenolol
18.18Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
18.18Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
18.18Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
18.18Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
18.18Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
18.18Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
18.18Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
18.18Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
18.18Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
18.18Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
18.18Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
18.18Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
18.18Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
18.18Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
18.18Single9H37A1IR09H37-A2A-A1IR0-Na
18.18Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
18.18Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
18.18Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
18.18Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.18Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.18Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
18.18Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
18.18Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
18.18Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
18.18Consensuscck_offOrthosteric Ligandccka_off
18.18Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
18.18Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
17.95Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
17.95Single7SK5CXCL127SK5-ACKR3-CXCL12
17.95Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
17.95Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
17.95Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
17.95Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
17.95Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.95Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
17.86Single8HS2Fab0468HS2-GPR20-Fab046
17.65Single2Y00Dobutamine2Y00-β1-Dobutamine
17.65Single5IUAQ274563485IUA-A2A-Q27456348-Na
17.65Single5XPRBosentan5XPR-ETB-Bosentan
17.65Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
17.65Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
17.65Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
17.65Single6S0QZM-2413856S0Q-A2A-ZM-241385
17.65Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
17.65Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
17.65Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
17.65Single7SINNPS-21437SIN-CaS-NPS-2143
17.65Single7SINNPS-21437SIN-CaS-NPS-2143
17.65Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
17.65Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
17.65Single7W41PD1762527W41-BB2-PD176252
17.65Single7WC6LSD7WC6-5-HT2A-LSD
17.65Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
17.65Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
17.65Single8GNEKW-63568GNE-A2A-KW-6356-Na
17.65Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
17.65Single8QOTNanobody-E8QOT-μ-Nanobody-E
17.65Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
17.65Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
17.65Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
17.65Single8ZMFA1L108ZMF-5-HT2C-A1L10
17.65Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
17.65Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
17.65Single9B9ZA1AKO9B9Z-CB1-A1AKO
17.65Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
17.65Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
17.65Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
17.65Single9HAPTolvaptan9HAP-V2-Tolvaptan
17.65Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
17.65Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
17.65Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
17.65Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
17.65Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
17.65Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
17.65Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
17.65Consensusbombesin_offOrthosteric Ligandbb2_off
17.65Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
17.65Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
17.65Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
17.65Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
17.50Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
17.50Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.50Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.24Single8A2OTheophylline8A2O-A2A-Theophylline-Na
17.24Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
17.24Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
17.24Single9CHUNoradrenaline9CHU-β2-Noradrenaline
17.24Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
17.24Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
17.24Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
17.14Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
17.14Single4U15Tiotropium4U15-M3-Tiotropium
17.14Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
17.14Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
17.14Single6J20Aprepitant6J20-NK1-Aprepitant
17.14Single6OL9Tiotropium6OL9-M5-Tiotropium
17.14Single6OS1TRV0266OS1-AT1-TRV026
17.14Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
17.14Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
17.14Single7F1TMIP-1a7F1T-CCR5-MIP-1a
17.14Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
17.14Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.14Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
17.14Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
17.14Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
17.14Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
17.14Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.14Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.14Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
17.14Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
17.14Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
17.14Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.14Single8XVLZibotentan8XVL-ETA-Zibotentan
17.14Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
17.14Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
17.14Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
17.14Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.07Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
17.07Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
17.07Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
17.07Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
16.67Single3OE6IT1t3OE6-CXCR4-IT1t
16.67Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
16.67Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
16.67Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
16.67Single6CM4Risperidone6CM4-D2-Risperidone
16.67Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
16.67Single6ME5Agomelatine6ME5-MT1-Agomelatine
16.67Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
16.67Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
16.67Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
16.67Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7K15MKD0467K15-BLT1-MKD046-Na
16.67Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
16.67Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
16.67Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
16.67Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
16.67Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
16.67Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
16.67Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
16.67Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
16.67Single8JWY2-1188JWY-A2A-2-118
16.67Single8JWZAB9288JWZ-A2A-AB928-Na
16.67Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
16.67Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
16.67Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
16.67Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
16.67Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
16.67Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
16.67Single9LRCHistamine9LRC-H4-Histamine
16.67Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
16.67Consensus5ht2_onOrthosteric Ligand5ht2b_on
16.67Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
16.67Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
16.67Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
16.67Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
16.67Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
16.67Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
16.67Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
16.67Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
16.67Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
16.67Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.22Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
16.22Single6K1QIRL25006K1Q-ETB-IRL2500
16.22Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
16.22Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.22Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
16.22Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.22Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
16.22Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.22Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
16.22Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
16.22Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
16.22Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.22Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single8XVUCXCL28XVU-CXCR2-CXCL2
16.22Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
16.22Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
16.22Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
16.22Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.22Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
16.22Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
16.22Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
16.22Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single3PBLEticlopride3PBL-D3-Eticlopride
16.13Single6HLLCP999946HLL-NK1-CP99994
16.13Single6LI0C176LI0-GPR52-C17
16.13Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
16.13Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
16.13Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
16.13Single7SRQLSD7SRQ-5-HT2B-LSD
16.13Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
16.13Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
16.13Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
16.13Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
16.13Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
16.13Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
16.13Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
16.13Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
16.13Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.13Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
16.13Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
16.13Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
16.13Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single9AS7Psilocin9AS7-5-HT2A-Psilocin
16.13Single9B9Y7DY9B9Y-CB1-7DY
16.13Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
16.13Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
15.79Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
15.79Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
15.79Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.79Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
15.79Single8XQJJN2418XQJ-Apelin-JN241
15.79Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
15.62Single3PWHZM-2413853PWH-A2A-ZM-241385
15.62Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
15.62Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
15.62Single4S0VSuvorexant4S0V-OX2-Suvorexant
15.62Single5U09Taranabant5U09-CB1-Taranabant
15.62Single5ZKQABT-4915ZKQ-PAF-ABT-491
15.62Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
15.62Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
15.62Single6ME9Ramelteon6ME9-MT2-Ramelteon
15.62Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
15.62Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
15.62Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
15.62Single6TPJSuvorexant6TPJ-OX2-Suvorexant
15.62Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
15.62Single7F8ULintitript7F8U-CCKA-Lintitript
15.62Single7F8YDevazepide7F8Y-CCKA-Devazepide
15.62Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
15.62Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
15.62Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
15.62Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
15.62Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
15.62Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
15.62Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
15.62Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
15.62Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
15.62Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
15.62Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
15.62Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
15.62Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
15.62Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
15.62Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
15.62Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
15.62Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
15.62Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
15.62Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
15.62Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
15.62Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
15.62Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
15.62Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
15.62Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
15.62Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
15.62Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
15.62Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
15.62Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
15.62Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
15.62Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
15.62Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
15.62Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
15.62Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
15.62Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
15.62Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
15.62Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
15.62Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
15.62Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
15.62Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
15.62Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
15.62Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
15.62Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
15.62Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
15.62Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
15.62Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
15.62Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
15.62Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
15.62Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
15.62Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
15.62Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
15.38Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8IEIA1LYA8IEI-GPR156-A1LYA
15.38Single8IEIA1LYA8IEI-GPR156-A1LYA
15.38Single8IEPA1LYA8IEP-GPR156-A1LYA
15.38Single8IEPA1LYA8IEP-GPR156-A1LYA
15.38Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
15.38Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
15.38Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
15.38Single9M4TSilodosin9M4T-Alpha1A-Silodosin
15.38Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
15.15Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
15.15Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
15.15Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
15.15Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
15.15Single5UVIZM-2413855UVI-A2A-ZM-241385
15.15Single6AQFZM-2413856AQF-A2A-ZM-241385
15.15Single6IQLL7458706IQL-D4-L745870
15.15Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
15.15Single6MH8ZM-2413856MH8-A2A-ZM-241385
15.15Single6TP3Nemorexant6TP3-OX1-Nemorexant
15.15Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
15.15Single6VI4JDTic6VI4-κ-JDTic
15.15Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
15.15Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
15.15Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
15.15Single6ZG9GSK10347026ZG9-M1-GSK1034702
15.15Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
15.15Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
15.15Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
15.15Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
15.15Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
15.15Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
15.15Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
15.15Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
15.15Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
15.15Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
15.15Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.15Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
15.15Single8K2WAMG4878K2W-CXCR3-AMG487
15.15Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.15Single8RLNLUF58348RLN-A2A-LUF5834
15.15Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
15.15Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
15.15Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
15.15Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
15.15Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
15.15Single8ZPMAMD0708ZPM-CXCR4-AMD070
15.15Single9AS3LSD9AS3-5-HT2A-LSD
15.15Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
15.15Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single9BA0A1AKN9BA0-CB1-A1AKN
15.15Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
15.15Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
15.15Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
15.15Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
15.15Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
15.15Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
15.15Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
15.15Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.00Single8IEBA1LYA8IEB-GPR156-A1LYA
15.00Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.00Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
15.00Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
14.71Single4MQSIperoxo4MQS-M2-Iperoxo
14.71Single4U14Tiotropium4U14-M3-Tiotropium
14.71Single5DHGC-355DHG-NOP-C-35
14.71Single5DHHSB-6121115DHH-NOP-SB-612111
14.71Single5DSGTiotropium5DSG-M4-Tiotropium
14.71Single5UIGCmpd-15UIG-A2A-Cmpd-1
14.71Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
14.71Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
14.71Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
14.71Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
14.71Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
14.71Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
14.71Single6GPSMK08126GPS-CCR2-MK0812
14.71Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
14.71Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
14.71Single7F83PF-051904577F83-Ghrelin-PF-05190457
14.71Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
14.71Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
14.71Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
14.71Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
14.71Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
14.71Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
14.71Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.71Single7YXAONO-54306087YXA-S1P5-ONO-5430608
14.71Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
14.71Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
14.71Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
14.71Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
14.71Single8X63Mepyramine8X63-H1-Mepyramine
14.71Single8X64Desloratadine8X64-H1-Desloratadine
14.71Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
14.71Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
14.71Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
14.71Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
14.71Single9IYAONO-97105319IYA-GPR55-ONO-9710531
14.71Single9JEAAtropine9JEA-M1-Atropine
14.71Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
14.71Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
14.71Consensusalpha2_onOrthosteric Ligandalpha2b_on
14.71Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
14.71Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
14.71Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
14.71Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
14.71Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
14.71Consensusblt_onOrthosteric Ligandblt1_on
14.71Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
14.71Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
14.71Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.71Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.71Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.71Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
14.71Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
14.71Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
14.71Consensushistamine_offOrthosteric Ligandh1_off
14.71Consensusleukotriene_onOrthosteric Ligandblt_on
14.71Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
14.71Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
14.71Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
14.71Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
14.71Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
14.63Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.63Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
14.63Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.63Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
14.63Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
14.63Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
14.29Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
14.29Single5CGCHTL142425CGC-mGlu5-HTL14242
14.29Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
14.29Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
14.29Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
14.29Single6GPXMK08126GPX-CCR2-MK0812
14.29Single6LUQHaloperidol6LUQ-D2-Haloperidol
14.29Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
14.29Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
14.29Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
14.29Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
14.29Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
14.29Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
14.29Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
14.29Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
14.29Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
14.29Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
14.29Consensusblt_offOrthosteric Ligandblt1_off
14.29Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
14.29Consensusep_offOrthosteric Ligandep4_off
14.29Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
14.29Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
14.29Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.89Single5TZRMK86665TZR-FFA1-MK8666
13.89Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
13.89Single6E59L-7607356E59-NK1-L-760735
13.89Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.89Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
13.89Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
13.89Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
13.89Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
13.89Single8EA0Iperoxo8EA0-M3-Iperoxo
13.89Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
13.89Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
13.89Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
13.89Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
13.89Single9AS9RS130-1809AS9-5-HT2A-RS130-180
13.89Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
13.89Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.89Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
13.89Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
13.89Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.89Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
13.89Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
13.89Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
13.89Consensustachykinin_offOrthosteric Ligandnk1_off
13.79Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
13.79Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
13.79Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
13.79Single8PWNTheophylline8PWN-A2A-Theophylline
13.79Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
13.51Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
13.51Single4PY02MeSATP4PY0-P2Y12-2MeSATP
13.51Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
13.51Single6IIURamatroban6IIU-TXA2-Ramatroban
13.51Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
13.51Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.51Single8XWMCXCL68XWM-CXCR2-CXCL6
13.51Single8XWSCXCL58XWS-CXCR2-CXCL5
13.51Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
13.51Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
13.51Single9BJKNAM9BJK-μ-Naloxone-NAM
13.33Single3OE8IT1t3OE8-CXCR4-IT1t
13.33Single3RFMCaffeine3RFM-A2A-Caffeine
13.33Single6TQ9SB-4081246TQ9-OX1-SB-408124
13.33Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
13.33Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
13.33Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
13.33Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
13.33Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
13.33Consensussensory_onOrthosteric Ligandopsins_on
13.16Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
13.16Single5CGDHTL142425CGD-mGlu5-HTL14242
13.16Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
13.16Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
13.16Single8XVJMacitentan8XVJ-ETA-Macitentan
13.16Single8XWFCXCL38XWF-CXCR2-CXCL3
13.16Single8ZPLHF511168ZPL-CXCR4-HF51116
13.16Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
12.90Single4XNWMRS25004XNW-P2Y1-MRS2500
12.90Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
12.90Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
12.90Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
12.90Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
12.90Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
12.90Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.90Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
12.90Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
12.90Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
12.90Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
12.90Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
12.90Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
12.90Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
12.90Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
12.90Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
12.90Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
12.90Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
12.90Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
12.90Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.90Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
12.82Single6KNMJN241-96KNM-Apelin-JN241-9
12.82Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
12.82Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
12.82Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
12.82Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
12.82Single9JF4PD1683689JF4-BB1-PD168368
12.82Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
12.82Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single4O9RCyclopamine4O9R-SMO-Cyclopamine
12.50Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
12.50Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
12.50Single6TP4ACT-4622066TP4-OX1-ACT-462206
12.50Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
12.50Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.50Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
12.50Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
12.50Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
12.50Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
12.50Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
12.50Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
12.50Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
12.50Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
12.50Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
12.50Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
12.50Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8XWNCXCL88XWN-CXCR2-CXCL8
12.50Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
12.50Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
12.50Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
12.50Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
12.50Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
12.50Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
12.50Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
12.12Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
12.12Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
12.12Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
12.12Single4QINSAG1.54QIN-SMO-SAG1.5
12.12Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
12.12Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
12.12Single6DS0Ly2660976DS0-5-HT2B-Ly266097
12.12Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
12.12Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
12.12Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
12.12Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
12.12Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
12.12Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
12.12Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.12Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.12Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
12.12Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
12.12Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
12.12Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
12.12Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
12.12Single9H2XA1IR19H2X-A2A-A1IR1-Na
12.12Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
12.12Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
12.12Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
12.12Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
12.12Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
12.12Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
11.76Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
11.76Single3REYXAC3REY-A2A-XAC
11.76Single3RZECidoxepin3RZE-H1-Cidoxepin
11.76Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
11.76Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
11.76Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
11.76Single6TPKRetosiban6TPK-OT-Retosiban
11.76Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
11.76Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
11.76Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
11.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
11.76Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
11.76Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
11.76Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
11.76Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
11.76Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
11.76Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
11.76Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single8ZPNAMD31008ZPN-CXCR4-AMD3100
11.76Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
11.76Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
11.76Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
11.76Consensusopsins_offOrthosteric Ligandrhodopsin_off
11.76Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
11.76Consensussensory_offOrthosteric Ligandopsins_off
11.76Consensusvasop-oxy_offOrthosteric Ligandot_off
11.43Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
11.43Single6IIVDaltroban6IIV-TXA2-Daltroban
11.43Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
11.43Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.43Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
11.43Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
11.43Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
11.43Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.43Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
11.43Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.43Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
11.43Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
11.43Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
11.43Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
11.43Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.11Single4JKVTaladegib4JKV-SMO-Taladegib
11.11Single4NTJAZD12834NTJ-P2Y12-AZD1283
11.11Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
11.11Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
11.11Single6HLPNetupitant6HLP-NK1-Netupitant
11.11Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
11.11Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
11.11Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
11.11Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
11.11Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
11.11Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
11.11Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
11.11Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.11Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
11.11Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
11.11Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
11.11Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
11.11Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
11.11Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
11.11Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
10.81Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
10.81Single5V56TC1145V56-SMO-TC114
10.81Single5V57TC1145V57-SMO-TC114
10.81Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
10.81Single7R0CAVP7R0C-V2-AVP-Arrestin2
10.81Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
10.81Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
10.81Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
10.81Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
10.81Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
10.81Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
10.53Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
10.53Single4N4WSANT-14N4W-SMO-SANT-1
10.53Single5X33BIIL2605X33-BLT1-BIIL260
10.53Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
10.53Single8XQJJN2418XQJ-Apelin-JN241
10.53Single8XWACXCL18XWA-CXCR2-CXCL1
10.53Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
10.53Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single5MZPCaffeine5MZP-A2A-Caffeine-Na
10.34Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
10.26Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
10.26Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
10.00Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
10.00Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
10.00Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
10.00Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
10.00Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
10.00Single7WC4Serotonin7WC4-5-HT2A-Serotonin
10.00Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
10.00Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
10.00Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
10.00Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
10.00Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
9.76Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
9.76Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
9.76Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.76Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.76Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.68Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
9.68Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
9.68Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
9.68Consensusp2y_offOrthosteric Ligandp2y1_off
9.38Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
9.38Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
9.38Single3UZAGTPL92363UZA-A2A-GTPL9236
9.38Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
9.38Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
9.38Single7WC5Psilocin7WC5-5-HT2A-Psilocin
9.38Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
9.38Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
9.38Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
9.38Consensusgi_sensoryOrthosteric Ligandgi_opsins
9.38Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
9.38Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
9.09Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
9.09Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
9.09Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
9.09Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
9.09Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
9.09Single5L7IVismodegib5L7I-SMO-Vismodegib
9.09Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
9.09Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
9.09Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
9.09Single7UL2SR486927UL2-NTS1-SR48692-Na
9.09Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
9.09Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
9.09Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
9.09Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
9.09Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.09Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
9.09Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
9.09Consensusgq_nucleotideOrthosteric Ligandgq_p2y
9.09Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.09Consensusneurotensin_offOrthosteric Ligandnts1_off
9.09Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
8.82Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
8.82Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
8.82Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
8.82Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
8.82Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
8.82Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
8.82Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
8.82Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.82Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.82Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
8.82Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
8.82Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
8.57Single7VODCariprazine7VOD-5-HT2A-Cariprazine
8.57Single7VV6C48/807VV6-MRGPRX2-C48/80
8.57Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
8.57Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
8.57Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single4QIMANTA XV4QIM-SMO-ANTA XV
8.33Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
8.11Single6Z4SSR486926Z4S-NTS1-SR48692
8.11Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
8.11Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
8.11Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
8.11Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
8.11Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
8.11Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
8.11Single9HC04YI9HC0-mGlu5-4YI
8.11Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.11Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
7.89Single7P2L4YI7P2L-mGlu5-4YI
7.89Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
7.89Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
7.89Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
7.89Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.89Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
7.69Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
7.69Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
7.69Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
7.69Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
7.50Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
7.50Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
6.67Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
6.67Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
6.25Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
6.25Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
6.25Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
6.06Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
6.06Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
6.06Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
6.06Single8JPSCCL78JPS-ACKR1-CCL7
5.88Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
5.88Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
5.88Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
5.88Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
5.88Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
5.56Single6FFIMMPEP6FFI-mGlu5-MMPEP
5.56Single6ZINSR486926ZIN-NTS1-SR48692
5.56Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.41Single6FFHFenobam6FFH-mGlu5-Fenobam
5.26Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
5.26Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
5.13Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.88Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
3.57Single6D35Cholesterol6D35-SMO-Cholesterol
3.57Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
3.57Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
3.57Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
3.57Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
3.57Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
3.57Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
3.57Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
3.57Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
3.57Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
3.57Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
3.57Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.57Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.57Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.57Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.57Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
3.57Single7DTTCa7DTT-CaS-Ca-Ca
3.57Single7DTTCa7DTT-CaS-Ca-Ca
3.57Single7DTUTryptophan7DTU-CaS-Tryptophan
3.57Single7DTUTryptophan7DTU-CaS-Tryptophan
3.57Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
3.57Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
3.57Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
3.57Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
3.57Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.57Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.57Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.57Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.57Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
3.57Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
3.57Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
3.57Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
3.57Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
3.57Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
3.57Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
3.57Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
3.57Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
3.57Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
3.57Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
3.57Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
3.57Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
3.57Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.57Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.57Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
3.57Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
3.57Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.57Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.57Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.57Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.57Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
3.57Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
3.57Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
3.57Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
3.57Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
3.57Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
3.57Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.57Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.57Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.57Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.57Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.57Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.57Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.57Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.57Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
3.57Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
3.57Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
3.57Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
3.57Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
3.57Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
3.57Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
3.57Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
3.57Single7XW7K1-707XW7-TSH-K1-70
3.57Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
3.57Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
3.57Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
3.57Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
3.57Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
3.57Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
3.57Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
3.57Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
3.57Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
3.57Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
3.57Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
3.57Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
3.57Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
3.57Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
3.57Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
3.57Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
3.57Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
3.57Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
3.57Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
3.57Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
3.57Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
3.57Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.57Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.57Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.57Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.57Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.57Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.57Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
3.57Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
3.57Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
3.57Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
3.57Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
3.57Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.57Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.57Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
3.57Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
3.57Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
3.57Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
3.57Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
3.57Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
3.57Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
3.57Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
3.57Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
3.57Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
3.57Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
3.57Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
3.57Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
3.57Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
3.57Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
3.57Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
3.57Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.57Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.57Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.57Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.57Single8WVXNorrin8WVX-LGR4-Norrin
3.57Single8WVYNorrin8WVY-LGR4-Norrin
3.57Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.57Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.57Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.57Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.57Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.57Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.57Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
3.57Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
3.57Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.57Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.57Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
3.57Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
3.57Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
3.57Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
3.57Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
3.57Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.57Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.57Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.57Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.57Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.57Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.57Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.57Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.57Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.57Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.57Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.57Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.57Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.57Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.57Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.57Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.57Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
3.57Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
3.57Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
3.57Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
3.57Single9KHHNorrin9KHH-LGR4-Norrin
3.57Single9S37NB219S37-LGR4-NB21
3.57Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
3.45Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.45Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.45Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.45Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.45Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.45Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.45Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.45Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.45Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.45Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.45Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.45Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.45Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.45Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.45Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.45Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
3.45Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
3.33Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
3.33Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
3.33Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
3.33Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
3.23Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
3.23Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
3.23Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
3.23Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
3.23Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.12Single5L7DCholesterol5L7D-SMO-Cholesterol
3.12Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
3.12Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.12Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.03Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
3.03Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
2.86Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.86Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
2.70Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
2.70Single8IYXYL-3658IYX-GPR34-YL-365
2.70Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
2.27Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.27Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.17Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.17Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.13Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.00Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
class-a_on_gp sensory_on_gp
alicarboxylic_on_gp
amine_on_gp
lipid_on_gp
nucleotide_on_gp
peptide_on_gp
protein_on_gp
class-b1_on_gp glucagon_on_gp
vip-pacap_on_gp
pth_on_gp
crf_on_gp
calcitonin_on_gp
Net Summary
Imin 2.89027
Number of Linked Nodes 1213
Number of Links 1369
Number of Hubs 190
Number of Links mediated by Hubs 788
Number of Communities 21
Number of Nodes involved in Communities 202
Number of Links involved in Communities 293
Path Summary
Number Of Nodes in MetaPath 111
Number Of Links MetaPath 110
Number of Shortest Paths 7403843
Length Of Smallest Path 3
Average Path Length 47.1329
Length of Longest Path 89
Minimum Path Strength 0.181851
Average Path Strength 5.06223
Maximum Path Strength 20.9066
Minimum Path Correlation 0.700725
Average Path Correlation 0.976504
Maximum Path Correlation 0.996875
Minimum % Of Corr. Nodes 1.42857
Average % Of Corr. Nodes 20.8063
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 59.1856
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .




You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download class-a_class-b1_cons_on_gp.zip



You can click to copy the link of this page to easily come back here later

or use this QR code to link and share this page.



You can also  read or  download a guide explaining the meaning of all files and numerical data.