Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.hns1.01 7.994204
2G.s1h1.04 7.44254179
3G.S2.06 7.01754139
4G.S3.03 7.135408
5G.S3.06 8.002527
6G.s3h2.03 6.8625429
7G.H2.03 10429
8G.H2.06 6.515429
9G.H2.07 6.96571729
10G.h2s4.01 9.106529
11G.s4h3.04 6.945408
12G.H3.09 6.89254159
13G.H3.13 9.7745156
14G.S5.05 7.06754229
15G.S5.07 4.704509
16G.HG.01 5.3446
17G.HG.03 5.265406
18G.hgh4.02 3.385218
19G.hgh4.05 8.89406
20G.hgh4.20 6.474543
21G.H4.07 8.6175445
22G.H4.08 7.61443
23G.H4.10 10.6654217
24G.H4.12 6.838544
25G.H4.14 9.444215
26G.H4.15 8.665408
27G.H4.16 6.1425444
28G.S6.02 8.3925438
29G.S6.05 8.944545
30G.H5.08 4.44538
31G.H5.13 5.1175438
32G.H5.16 5.2125436
33G.H5.17 7.03167635
34b.1x19 7.2486
35b.lhb1x3 3.942502
36b.lhb1x6 3.26754163
37b.l1x3 8.9325109
38b.b2x1 10.4583698
39b.b2x5 6.25167667
40b.l2x5 11.0625465
41b.b3x4 6.0954109
42b.l3x2 6.51254209
43b.b4x4 9.474108
44b.b4x6 9.673336109
45b.l4x2 9.685464
46b.b5x3 6.3625109
47b.b5x5 6.09254195
48b.l5x1 4.9025408
49b.l5x5 10.23529
50b.b6x5 4.324506
51b.b7x1 6.235404
52b.l7x2 4.772529
53b.b8x3 4.025476
54b.b8x4 5.416506
55b.b9x4 6.058579
56b.l9x3 8.922579
57b.l9x6 5.36222928
58b.b10x3 3.4175478
59b.b10x5 5.086509
60b.b11x4 5.8275479
61b.l11x2 9.84479
62b.b12x6 9.46678
63b.b13x7 7.474557
64b.l13x3 4.98167659
65b.l13x6 5.32167629
66b.l13x7 4.3775459
67b.l15x1 5.685427
68b.l15x2 6.94459
69b.b16x4 7.38456
70b.b16x6 6.69714758
71b.b17x5 4.82833687
72b.b17x7 7.476588
73b.l17x3 8.186676269
74b.l17x6 7.9225429
75b.b18x3 6.2475488
76b.b18x5 4.388505
77b.l18x1 8.3056276
78b.b19x2 7.21833686
79b.l19x2 9.274269
80b.b20x6 8.0825486
81b.l20x1 6.8925486
82b.l20x2 6.33254289
83b.b21x1 8.328587
84b.b21x7 5.345605
85b.b22x5 6.62407
86b.l22x5 4.856676169
87b.b23x6 6.6745297
88b.l23x1 6.87496
89b.l25x3 10.1845129
90b.l25x6 14.16598
91b.l26x5 4.76405
92b.l27x1 12.5871799
93b.l27x2 8.2754129
94b.b28x2 6.3625404
95b.b28x3 5.2885107
96b.b28x4 10.0154126
97b.b28x5 3.905465
98b.b28x6 12.58754129
991x39 7.44833617
1002x38 3.965406
1012x40 6.458577118
1022x60 6.75415
1032x61 5.525415
1043x25 7.54413
1053x29 8.816514
1063x32 8.1575414
1073x33 3.87414
1083x49 5.0554189
1093x50 7.374149
1103x53 7.1954188
1113x55 10.076536
112I2x53 6.8525188
1134x60 5.48333603
1144x61 5.966515
1155x47 8.318507
1165x58 4.561437149
1175x68 7.8975437
118I3.P225 7.1675443
1196x37 2.8025407
1206x41 2.875407
1216x48 7.41714718
1226x51 6.53415
1236x54 9415
1246x61 3.4365304
1257x37 8.2075405
1267x52 3.865149
1277x53 5.2556149
1288x49 4.484116
129g.h1x1 2.815402
130g.h1x8 2.6125407
131g.h1x14 4.18489
132g.ctx3 6.275409
133g.ctx4 3.9425407
134g.ctx6 3.85506
135g.ctx16 5.01429768
136Lig 10.91332110
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b3x1 b.b6x5 77.17945.86NoYes056
2b.b3x1 b.l2x5 77.44993.64NoYes655
3b.l2x5 b.l4x2 77.948714.4YesYes654
4b.l4x2 g.ctx16 75.94217.22YesYes648
5b.l4x1 g.ctx16 45.44533.96NoYes658
6b.b2x5 b.l4x1 45.55424.94YesNo675
7b.b2x5 b.b3x2 89.022810.25YesNo075
8b.b3x2 b.b4x6 89.11173.42NoYes059
9b.b28x5 g.ctx16 45.51923.77YesYes658
10b.b28x5 b.b2x5 45.84614.7YesYes657
11b.b3x4 b.b4x6 44.32273.71YesYes1099
12b.b3x4 b.l1x3 44.60476.97YesYes1099
13b.b4x2 b.l1x3 45.13873.93NoYes089
14b.b4x4 b.b4x6 44.333619.97YesYes1089
15b.b4x4 b.l1x3 44.865211.93YesYes1089
16b.b3x6 b.l1x3 44.704812.55NoYes099
17b.b3x6 b.l3x2 44.608310.31NoYes099
18b.l1x4 b.l3x2 86.54138.14NoYes2069
19G.HN.51 b.l1x4 92.79665.64NoNo046
20b.b4x2 b.l3x2 44.75274.15NoYes089
21G.HN.51 G.hns1.02 92.28134.95NoNo044
22G.hns1.02 I2x54 92.02783.39NoNo045
23I2x53 I2x54 91.77747.62YesNo085
243x53 I2x53 93.92089.99YesYes1888
253x53 G.H5.23 1006.24YesNo084
263x54 G.H5.23 52.03924.84NoNo094
273x54 3x55 47.83237.54NoYes096
283x55 5x64 45.36737.5YesNo365
295x64 G.H5.16 13.43179.37NoYes356
30G.H5.12 G.H5.16 12.59313.5NoYes376
31G.H5.08 G.H5.12 11.48454.28YesNo387
32G.H5.08 G.S2.08 10.38225.24YesNo086
33G.S2.08 G.S3.03 10.01375.24NoYes068
34b.b27x2 b.b2x5 12.25683.89NoYes057
35b.b27x2 b.b2x3 12.06194.83NoNo056
36b.b26x2 b.b2x3 12.12614.86NoNo076
37b.b26x1 b.b26x2 11.99393.44NoNo097
38b.b26x1 b.b2x1 10.55896.36NoYes998
39G.S1.05 G.h2s4.01 11.048818.27NoYes099
40G.S1.05 G.S4.02 10.85955.71NoNo098
415x64 5x68 31.582810.18NoYes357
425x68 G.H5.13 15.01136.3YesYes378
43G.H5.13 G.S6.02 13.92223.45YesYes388
44G.H5.10 G.S6.02 25.666413.79NoYes078
45G.H5.10 G.S6.04 24.935810.08NoNo079
46G.S5.05 G.S6.04 21.28075.66YesNo099
47G.S5.05 G.s6h5.01 18.351510.38YesNo2299
48G.S5.07 G.s6h5.01 17.62145.85YesNo099
49G.S5.07 G.s5hg.01 11.02445.6YesNo099
505x68 G.H5.17 16.475810.16YesYes375
51G.H5.17 G.S6.02 13.934710.29YesYes358
52G.S4.02 G.S5.02 10.36833.07NoNo086
532x40 I1x50 19.89149.38YesNo1188
541x60 I1x50 20.28719.61NoNo078
551x60 b.l25x4 20.57745.39NoNo075
56b.l25x4 b.l27x2 20.67843.99NoYes059
57b.l25x3 b.l27x2 20.636810.08YesYes1299
58b.b27x3 b.l25x3 10.4876.85NoYes089
59b.b27x3 b.b28x6 10.50428.49NoYes089
60b.b25x7 b.b28x6 21.539920.5NoYes079
61b.b25x7 b.lhb1x11 21.55184.24NoNo074
62b.lhb1x11 g.ctx5 21.60655.65NoNo049
63b.l22x1 g.ctx5 21.64976.01NoNo099
64b.l22x1 g.ctx3 14.013510.31NoYes099
65g.ctx3 g.ctx4 31.59234.83YesYes097
66b.l26x5 g.ctx4 33.75363.35YesYes057
67b.b28x4 b.l25x3 10.611213.1YesYes1269
68b.b28x4 b.b28x6 10.929210.44YesYes1269
69b.l26x5 g.ctx16 21.76293.73YesYes058
703x50 G.H5.23 52.358713.38YesNo094
713x50 5x58 42.88376.17YesYes1499
72b.b2x4 b.b6x5 67.78663.27NoYes066
73b.b10x4 b.b2x4 67.49039.03NoNo066
74b.b10x2 b.b10x4 67.19398.36NoNo066
75b.b10x2 b.b14x3 50.0294.76NoNo065
76b.b11x5 b.b14x3 49.72316.01NoNo065
77b.b11x5 b.l13x7 49.4174.85NoYes069
78b.l13x3 b.l13x7 44.01854.15YesYes599
79b.b16x4 b.l13x3 38.67575.24YesYes569
80b.b16x4 b.b17x6 37.920112.01YesNo067
81b.b17x6 g.h1x14 37.60834.23NoYes079
82b.b21x1 g.h1x14 10.61013.9YesYes879
83g.ctx3 g.ctx6 31.98654.07YesYes096
84b.l22x5 g.ctx6 37.39513.64YesYes096
85b.l22x5 b.lhb1x3 33.1093.76YesYes092
86b.h2x5 b.lhb1x3 30.95663.04NoYes052
87b.h2x1 b.h2x5 30.41812.95NoNo055
88b.b21x5 b.h2x1 29.34059.9NoNo045
89b.b21x5 b.b21x7 28.80154.79NoYes045
90b.b21x7 b.b23x2 19.07143.52YesNo056
91b.b22x5 b.b23x2 17.98713.4YesNo076
92b.b22x5 b.l18x1 15.27327.5YesYes076
93b.l18x1 b.l18x3 10.91716.04YesNo065
94b.b10x2 b.b6x2 18.30763.38NoNo068
95b.b10x3 b.b6x2 17.98523.38YesNo088
96b.b17x5 g.h1x14 17.38585.1YesYes879
97b.b17x7 b.b21x1 10.05349.55YesYes887
98b.b17x7 b.b20x6 10.990111.79YesYes886
995x54 5x58 34.77055.99NoYes089
1005x54 6x44 34.423111.2NoNo088
1016x44 6x48 34.07735.01NoYes088
1026x48 7x41 25.9218.22YesNo186
1036x51 7x41 25.57875.02YesNo156
1046x51 Lig 25.22684.29YesYes150
1052x37 2x38 15.19223.56NoYes076
1062x38 I2x57 16.30995.03YesNo068
1072x37 2x40 14.95663.82NoYes1178
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
LigNT.Q376.531YesNo0301
1x39NT.I405.021YesNo7512
1x392x619.081YesYes7511
1x397x383.651YesNo7312
1x397x426.221YesNo7612
1x39Lig18.11YesYes7010
1x402x614.420NoYes5521
2x563x324.640NoYes5421
2x573x3211.330NoYes6421
2x577x428.410NoNo6622
2x603x256.51YesYes5321
2x603x299.091YesYes5421
2x603x324.11YesYes5421
2x60Ca57.311YesNo5022
2x61Lig6.851YesYes5010
2x64Lig15.810NoYes4010
3x21Lig10.921NoYes8010
3x22Lig11.271NoYes5010
3x253x295.321YesYes3411
3x25Lig10.851YesYes3010
3x25Ca57.491YesNo3012
3x264x614.251NoYes4511
3x26Lig6.031NoYes4010
3x294x614.21YesYes4511
3x29Lig15.491YesYes4010
3x29Ca59.981YesNo4012
3x304x614.640NoYes4521
3x32Lig12.561YesYes4010
3x334x573.921YesNo4612
3x334x604.191YesYes4312
3x334x613.271YesYes4511
3x33Lig4.11YesYes4010
4x61Lig13.471YesYes5010
4x64Lig13.761NoYes5010
5x376x598.721NoNo4311
5x37Lig6.21NoYes4010
5x406x557.141NoNo6512
5x406x5910.31NoNo6311
5x40Lig8.471NoYes6010
6x516x5210.721YesNo5612
6x516x556.091YesNo5512
6x517x415.021YesNo5612
6x51Lig4.291YesYes5010
6x546x589.281YesNo5321
6x54E3.T2785.481YesNo5322
6x547x3414.711YesNo5321
6x58E3.T2784.561NoNo3312
6x58Lig3.771NoYes3010
6x59Lig3.771NoYes3010
7x347x386.091NoNo3312
7x34Lig18.981NoYes3010
3x213x242.921NoNo8512
5x375x382.881NoNo4512
4x64E2.E1842.871NoNo5412
1x397x392.621YesNo7512
3x193x222.560NoNo2521
1x362x611.750NoYes4521
3x183x211.40NoNo6821

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
94.74Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
61.90Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
61.54Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
60.87Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
60.71Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
60.71Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
59.09Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
58.33Single6W25SHU91196W25-MC4-SHU9119-Ca
58.33Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
56.52Single8KIGSHU91198KIG-MC3-SHU9119-Ca
56.52Single8WKYPG-9348WKY-MC4-PG-934
56.52Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
54.17Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
53.57Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
50.00Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
50.00Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
48.15Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
48.00Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
46.15Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
44.44Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
44.44Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
44.12Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
44.12Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
44.00Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
44.00Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
42.86Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
42.86Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
40.00Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
35.29Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
34.62Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single8QJ2pN1628QJ2-MC4-pN162-Gs
34.62Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
34.15Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
33.33Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
33.33Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
32.14Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
30.77Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
30.77Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
29.63Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
29.63Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
29.63Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
29.63Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
29.17Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
29.17Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
29.17Single6HLPNetupitant6HLP-NK1-Netupitant
29.17Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
29.03Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
28.57Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
28.57Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
28.57Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
28.12Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
28.00Single5TZRMK86665TZR-FFA1-MK8666
28.00Single5XR8AM8415XR8-CB1-AM841
28.00Single5XRAAM115425XRA-CB1-AM11542
28.00Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
28.00Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
28.00Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
27.59Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
27.59Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
27.27Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
27.27Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
27.27Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
27.27Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
27.27Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
27.27Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
27.27Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
26.92Single4RWADIPP-NH24RWA-δ-DIPP-NH2
26.92Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
26.92Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.92Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
26.92Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
26.92Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
26.92Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.92Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
26.67Single3OE0CVX153OE0-CXCR4-CVX15
26.67Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
26.67Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
26.47Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
26.09Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
26.09Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
25.93Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
25.93Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
25.93Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
25.81Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
25.81Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
25.81Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
25.81Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
25.81Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
25.00Single4YAYZD-71554YAY-AT1-ZD-7155
25.00Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
25.00Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
25.00Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7V3ZCP559407V3Z-CB1-CP55940
25.00Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
25.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
25.00Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
25.00Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.00Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
25.00Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
25.00Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
25.00Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
25.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
25.00Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensuscck_offOrthosteric Ligandccka_off
25.00Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
25.00Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
24.24Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
24.24Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
24.14Single4XT1Fractalkine4XT1-US28-Fractalkine
24.14Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
24.14Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
24.14Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
24.14Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
24.00Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
24.00Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
24.00Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.00Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
24.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
24.00Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
24.00Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
23.81Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.53Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
23.33Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
23.33Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
23.33Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
23.33Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
23.33Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
23.33Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
23.08Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
23.08Single6E59L-7607356E59-NK1-L-760735
23.08Single6J20Aprepitant6J20-NK1-Aprepitant
23.08Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
23.08Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
23.08Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
23.08Single7FEECP559407FEE-CB1-CP55940-ZCZ011
23.08Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
23.08Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
23.08Single8E0GBU728E0G-μ-BU72
23.08Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
23.08Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
23.08Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
23.08Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
23.08Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
23.08Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
23.08Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
23.08Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
23.08Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
23.08Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
22.73Single6HLLCP999946HLL-NK1-CP99994
22.73Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
22.73Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
22.73Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
22.73Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
22.58Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
22.58Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.58Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
22.58Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
22.58Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
22.22Single4PY02MeSATP4PY0-P2Y12-2MeSATP
22.22Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
22.22Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
22.22Single6KQICP559406KQI-CB1-CP55940-Org27569
22.22Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
22.22Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
22.22Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
22.22Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
22.22Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
22.22Single7YITNalfurafine7YIT-κ-Nalfurafine
22.22Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
22.22Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
22.22Single8XYIVUF106618XYI-CXCR3-VUF10661
22.22Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
22.22Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
22.22Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
22.22Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
22.22Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
22.22Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
22.22Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
22.22Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
22.22Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
22.22Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
22.22Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
22.22Consensuslpa_offOrthosteric Ligandlpa1_off
22.22Consensuslpl_offOrthosteric Ligands1p_off lpa_off
22.22Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
22.22Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
22.22Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
22.22Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
22.22Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
21.88Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
21.88Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
21.88Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
21.88Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
21.88Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
21.88Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
21.88Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
21.88Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
21.88Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
21.74Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
21.74Single7BR3Elagolix7BR3-GnRH1-Elagolix
21.74Single7F8ULintitript7F8U-CCKA-Lintitript
21.74Single7F8YDevazepide7F8Y-CCKA-Devazepide
21.74Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
21.74Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
21.74Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
21.74Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
21.74Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
21.74Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
21.74Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
21.74Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
21.74Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
21.74Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
21.43Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
21.43Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
21.43Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
21.43Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
21.43Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
21.43Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
21.43Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
21.43Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
21.43Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
21.43Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
21.43Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
21.43Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
21.43Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
21.43Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
21.43Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
21.43Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
21.43Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
21.21Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
21.21Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
21.21Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
21.21Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
20.83Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
20.83Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
20.83Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
20.83Single6TPKRetosiban6TPK-OT-Retosiban
20.83Single6TPNHTL66416TPN-OX2-HTL6641
20.83Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
20.83Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
20.83Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.83Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
20.83Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
20.83Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
20.83Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
20.83Consensusgrh_offOrthosteric Ligandgnrh1_off
20.83Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
20.83Consensusvasop-oxy_offOrthosteric Ligandot_off
20.69Single5ZTYAM102575ZTY-CB2-AM10257
20.69Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
20.69Single6PT3DPI-2876PT3-δ-DPI-287
20.69Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
20.69Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
20.69Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
20.69Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
20.69Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
20.69Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
20.59Single4XT3Fractalkine4XT3-US28-Fractalkine
20.59Single7SK3CXCL127SK3-ACKR3-CXCL12
20.59Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
20.59Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
20.59Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
20.59Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
20.59Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
20.00Single4EJ4Naltrindole4EJ4-δ-Naltrindole
20.00Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
20.00Single5UIGCmpd-15UIG-A2A-Cmpd-1
20.00Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
20.00Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
20.00Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
20.00Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
20.00Single7F8XNN90567F8X-CCKA-NN9056
20.00Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
20.00Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
20.00Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
20.00Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
20.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
20.00Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
20.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
20.00Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
20.00Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
20.00Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
20.00Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
20.00Single8RLNLUF58348RLN-A2A-LUF5834
20.00Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
20.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
20.00Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
20.00Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
20.00Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
20.00Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
20.00Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
20.00Consensusa3_onOrthosteric Liganda3a_on
20.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
20.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
20.00Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
20.00Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
20.00Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
20.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
20.00Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
20.00Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
20.00Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
20.00Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
20.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
20.00Consensuslpl_onOrthosteric Ligands1p_on lpa_on
20.00Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
20.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
20.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
20.00Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
19.44Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
19.35Single3QAKUK-4320973QAK-A2A-UK-432097
19.35Single6HLOAprepitant6HLO-NK1-Aprepitant
19.35Single7SK5CXCL127SK5-ACKR3-CXCL12
19.35Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
19.35Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
19.35Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
19.35Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
19.35Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
19.35Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
19.35Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
19.23Single4NTJAZD12834NTJ-P2Y12-AZD1283
19.23Single5C1MBU725C1M-μ-BU72
19.23Single5N2RPSB-365N2R-A2A-PSB-36-Na
19.23Single5N2SPSB365N2S-A1-PSB36
19.23Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
19.23Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
19.23Single7C4SS1P7C4S-S1P3-S1P
19.23Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
19.23Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
19.23Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
19.23Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
19.23Single7SINNPS-21437SIN-CaS-NPS-2143
19.23Single7SINNPS-21437SIN-CaS-NPS-2143
19.23Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
19.23Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
19.23Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
19.23Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
19.23Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
19.23Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
19.23Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
19.23Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
19.23Single8JXSPF-61428JXS-D1-PF-6142
19.23Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
19.23Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
19.23Single8QOTNanobody-E8QOT-μ-Nanobody-E
19.23Single8S4DCMF-0198S4D-Apelin-CMF-019
19.23Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
19.23Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
19.23Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
19.23Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
19.23Consensusa3_on_gpOrthosteric Liganda3a_on_gp
19.23Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
19.23Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
19.23Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
19.23Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
19.23Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
19.23Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
19.23Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
19.23Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
18.92Single5GLHEndothelin-15GLH-ETB-Endothelin-1
18.92Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
18.75Single5WF5UK-4320975WF5-A2A-UK-432097
18.75Single6PT2KGCHM076PT2-δ-KGCHM07
18.75Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
18.75Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.75Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
18.75Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
18.75Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
18.75Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.75Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
18.75Consensusangiotensin_onOrthosteric Ligandat1_on
18.75Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
18.75Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
18.52Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
18.52Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
18.52Single4BV0Neurotensin4BV0-NTS1-Neurotensin
18.52Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
18.52Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
18.52Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
18.52Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
18.52Single6TQ7SB-3348676TQ7-OX1-SB-334867
18.52Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
18.52Single7B6WCyclazosin7B6W-α1b-Cyclazosin
18.52Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
18.52Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
18.52Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
18.52Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
18.52Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
18.52Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
18.52Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
18.52Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
18.52Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
18.52Single7TUYGSK682753A7TUY-GPR183-GSK682753A
18.52Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
18.52Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
18.52Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
18.52Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
18.52Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
18.52Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
18.52Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
18.52Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
18.52Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
18.52Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
18.52Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
18.52Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
18.52Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
18.52Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
18.52Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
18.52Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
18.52Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
18.52Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
18.52Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
18.52Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
18.52Consensuslpa_onOrthosteric Ligandlpa1_on
18.52Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
18.52Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Consensusneurotensin_onOrthosteric Ligandnts1_on
18.52Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
18.52Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
18.52Consensustachykinin_offOrthosteric Ligandnk1_off
18.42Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
18.18Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
18.18Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
18.18Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
18.18Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
18.18Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.18Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.18Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
18.18Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
18.18Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
18.18Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
17.95Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
17.86Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
17.86Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
17.86Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
17.86Single4XEENeurotensin4XEE-NTS1-Neurotensin
17.86Single4XESNeurotensin4XES-NTS1-Neurotensin
17.86Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
17.86Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
17.86Single6MXTSalmeterol6MXT-β2-Salmeterol
17.86Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
17.86Single6YVRNTS8-136YVR-NTS1-NTS8-13
17.86Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
17.86Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
17.86Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
17.86Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
17.86Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.86Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
17.86Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
17.86Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
17.86Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
17.86Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.86Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
17.86Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
17.86Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
17.86Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
17.86Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
17.86Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
17.86Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
17.86Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.86Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
17.86Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
17.86Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
17.86Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
17.86Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
17.86Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
17.86Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
17.86Consensusorexin_onOrthosteric Ligandox2_on
17.86Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
17.65Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
17.65Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
17.65Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
17.65Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
17.65Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
17.65Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
17.65Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
17.65Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
17.65Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
17.65Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
17.65Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
17.50Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
17.39Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
17.39Single6TP4ACT-4622066TP4-OX1-ACT-462206
17.39Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
17.39Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
17.39Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
17.39Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
17.24Single4BUONeurotensin4BUO-NTS1-Neurotensin
17.24Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
17.24Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
17.24Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
17.24Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
17.24Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
17.24Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.24Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
17.24Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
17.24Single7UM4AS26747237UM4-5-HT5A-AS2674723
17.24Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
17.24Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
17.24Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
17.24Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
17.24Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
17.24Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
17.24Consensuscck_onOrthosteric Ligandccka_on cckb_on
17.24Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
17.24Consensuschemerin_onOrthosteric Ligandcml1_on
17.24Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
17.24Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
17.14Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
17.14Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
17.14Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
17.14Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
17.14Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
16.67Single3NY9ICI118-5513NY9-β2-ICI118-551
16.67Single3PWHZM-2413853PWH-A2A-ZM-241385
16.67Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
16.67Single4S0VSuvorexant4S0V-OX2-Suvorexant
16.67Single4UG2CGS216804UG2-A2A-CGS21680
16.67Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
16.67Single5WS3EMPA5WS3-OX2-EMPA
16.67Single5ZKQABT-4915ZKQ-PAF-ABT-491
16.67Single6AKXA4R6AKX-CCR5-A4R
16.67Single6AKYMaraviroc6AKY-CCR5-Maraviroc
16.67Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
16.67Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
16.67Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
16.67Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
16.67Single6TODEMPA6TOD-OX1-EMPA-Na
16.67Single6TPJSuvorexant6TPJ-OX2-Suvorexant
16.67Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
16.67Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
16.67Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
16.67Single7SK9CCX6627SK9-ACKR3-CCX662
16.67Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
16.67Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
16.67Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
16.67Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
16.67Single7XRRLemborexant7XRR-OX2-Lemborexant
16.67Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
16.67Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
16.67Single8IWESpermidine8IWE-TA9-Spermidine
16.67Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
16.67Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
16.67Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
16.67Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
16.67Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
16.67Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
16.67Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
16.67Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
16.67Consensusangiotensin_offOrthosteric Ligandat1_off
16.67Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
16.67Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
16.67Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
16.67Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
16.67Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
16.67Consensusorexin_offOrthosteric Ligandox2_off ox1_off
16.67Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
16.67Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
16.67Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
16.67Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
16.22Single6IGLIRL16206IGL-ETB-IRL1620
16.22Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
16.22Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
16.22Single8IY6Endothelin-18IY6-ETB-Endothelin-1
16.22Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
16.22Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
16.22Consensusbradykinin_onOrthosteric Ligandbk2_on
16.22Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
16.22Consensusendothelin_onOrthosteric Ligandetb_on eta_on
16.22Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
16.13Single4IARErgotamine4IAR-5-HT1B-Ergotamine
16.13Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
16.13Single7QA8Peptide7QA8-STE2-Peptide
16.13Single7QA8Peptide7QA8-STE2-Peptide
16.13Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
16.13Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
16.13Single8IEBA1LYA8IEB-GPR156-A1LYA
16.13Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
16.13Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
16.13Single8XWNCXCL88XWN-CXCR2-CXCL8
16.13Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.13Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
16.13Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
16.00Single3REYXAC3REY-A2A-XAC
16.00Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
16.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
16.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
16.00Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
16.00Single6IQLL7458706IQL-D4-L745870
16.00Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
16.00Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
16.00Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
16.00Single6TP3Nemorexant6TP3-OX1-Nemorexant
16.00Single6V9SGTPL114036V9S-OX1-GTPL11403
16.00Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
16.00Single7AROLUF58337ARO-A2A-LUF5833-Na
16.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
16.00Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.00Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
16.00Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
16.00Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
16.00Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
16.00Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
16.00Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
16.00Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
16.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
16.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
16.00Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
16.00Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
16.00Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
16.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.00Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
16.00Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
16.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
16.00Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
16.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
16.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
16.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
16.00Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
15.79Single6IGKEndothelin-36IGK-ETB-Endothelin-3
15.79Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
15.79Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
15.79Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
15.79Consensusbombesin_onOrthosteric Ligandbb2_on
15.79Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
15.79Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
15.62Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
15.62Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
15.62Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
15.62Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
15.62Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
15.62Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
15.62Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
15.62Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
15.62Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
15.62Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.62Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
15.62Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
15.62Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
15.62Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.62Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
15.62Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
15.62Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
15.38Single2Y04Salbutamol2Y04-β1-Salbutamol
15.38Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
15.38Single5T04Neurotensin5T04-NTS1-Neurotensin
15.38Single5TGZAM65385TGZ-CB1-AM6538
15.38Single5UENDU1725UEN-A1-DU172
15.38Single6D27CAY104716D27-DP2-CAY10471
15.38Single6DRXLisuride6DRX-5-HT2B-Lisuride
15.38Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
15.38Single6PS1Timolol6PS1-β2-Timolol
15.38Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
15.38Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
15.38Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
15.38Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
15.38Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
15.38Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
15.38Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
15.38Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
15.38Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
15.38Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
15.38Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
15.38Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
15.38Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
15.38Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
15.38Single7YXAONO-54306087YXA-S1P5-ONO-5430608
15.38Single8CU6LJ-45178CU6-A2A-LJ-4517
15.38Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
15.38Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
15.38Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
15.38Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
15.38Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
15.38Single8JXRLSD8JXR-D1-LSD
15.38Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
15.38Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
15.38Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
15.38Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
15.38Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
15.38Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
15.38Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
15.38Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
15.38Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
15.38Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
15.38Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
15.38Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
15.38Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
15.38Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
15.38Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
15.38Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
15.38Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
15.38Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
15.38Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
15.38Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
15.38Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
15.15Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
15.15Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
15.15Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
15.15Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
15.15Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
15.15Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
15.15Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
15.15Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
15.15Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
15.15Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
15.15Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.15Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
15.15Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
15.15Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
15.15Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
15.15Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
15.00Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
15.00Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
15.00Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single2Y03Isoprenaline2Y03-β1-Isoprenaline
14.81Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
14.81Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
14.81Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
14.81Single5WQCEMPA5WQC-OX2-EMPA
14.81Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
14.81Single5XPRBosentan5XPR-ETB-Bosentan
14.81Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
14.81Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
14.81Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
14.81Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
14.81Single6TP6Filorexant6TP6-OX1-Filorexant
14.81Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
14.81Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
14.81Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
14.81Single6Z4SSR486926Z4S-NTS1-SR48692
14.81Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
14.81Single7C61Ergotamine7C61-5-HT1B-Ergotamine
14.81Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
14.81Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
14.81Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
14.81Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
14.81Single7W41PD1762527W41-BB2-PD176252
14.81Single7WC6LSD7WC6-5-HT2A-LSD
14.81Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
14.81Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
14.81Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
14.81Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
14.81Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GNEKW-63568GNE-A2A-KW-6356-Na
14.81Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
14.81Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
14.81Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
14.81Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
14.81Single8ZMFA1L108ZMF-5-HT2C-A1L10
14.81Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
14.81Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
14.81Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
14.81Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
14.81Consensusadenosine_offOrthosteric Liganda1_off a2_off
14.81Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
14.81Consensusbombesin_offOrthosteric Ligandbb2_off
14.81Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
14.81Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
14.81Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
14.81Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.81Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
14.81Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
14.81Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
14.71Single6JODAngiotensin II6JOD-AT2-Angiotensin II
14.71Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
14.71Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
14.71Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
14.71Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
14.71Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
14.71Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
14.71Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
14.71Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
14.71Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
14.71Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
14.71Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.71Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
14.71Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
14.71Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
14.71Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
14.71Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
14.71Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
14.71Consensusvasop-oxy_onOrthosteric Ligandv2_on
14.71Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
14.63Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single3P0GBI1671073P0G-β2-BI167107
14.29Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
14.29Single5V54Methiothepin5V54-5-HT1B-Methiothepin
14.29Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
14.29Single6H7JIsoprenaline6H7J-β1-Isoprenaline
14.29Single6J21Aprepitant6J21-NK1-Aprepitant
14.29Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
14.29Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
14.29Single6OS1TRV0266OS1-AT1-TRV026
14.29Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
14.29Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
14.29Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
14.29Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
14.29Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
14.29Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
14.29Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
14.29Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
14.29Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
14.29Single7R0CAVP7R0C-V2-AVP-Arrestin2
14.29Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
14.29Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
14.29Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
14.29Single7WC4Serotonin7WC4-5-HT2A-Serotonin
14.29Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
14.29Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
14.29Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
14.29Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
14.29Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
14.29Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
14.29Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
14.29Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
14.29Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
14.29Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
14.29Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
14.29Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
14.29Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
14.29Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
14.29Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
14.29Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
14.29Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
14.29Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single8XVLZibotentan8XVL-ETA-Zibotentan
14.29Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
14.29Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
14.29Single8ZRTET-18ZRT-ETB-ET-1
14.29Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
14.29Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
14.29Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensus5ht1_offOrthosteric Ligand5ht1b_off
14.29Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
14.29Consensusa2_onOrthosteric Liganda2b_on
14.29Consensusa2_on_gpOrthosteric Liganda2b_on_gp
14.29Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.29Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.29Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
14.29Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
14.29Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
14.29Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
14.29Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
14.29Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
14.29Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
14.29Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.89Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
13.89Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
13.89Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
13.89Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
13.89Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
13.89Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
13.89Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
13.89Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
13.89Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
13.89Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
13.79Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
13.79Single4LDEBI1671074LDE-β2-BI167107
13.79Single6A93Risperidone6A93-5-HT2A-Risperidone
13.79Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
13.79Single6CM4Risperidone6CM4-D2-Risperidone
13.79Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
13.79Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
13.79Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
13.79Single6ZG4HTL00099366ZG4-M1-HTL0009936
13.79Single7DFPSpiperone7DFP-D2-Spiperone
13.79Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
13.79Single7K15MKD0467K15-BLT1-MKD046-Na
13.79Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
13.79Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
13.79Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
13.79Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
13.79Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
13.79Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
13.79Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
13.79Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
13.79Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
13.79Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
13.79Single8JJ8Formoterol8JJ8-β2-Formoterol
13.79Single8JJLOlodaterol8JJL-β2-Olodaterol
13.79Single8JWY2-1188JWY-A2A-2-118
13.79Single8JWZAB9288JWZ-A2A-AB928-Na
13.79Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
13.79Single8XWACXCL18XWA-CXCR2-CXCL1
13.79Single8XWMCXCL68XWM-CXCR2-CXCL6
13.79Single8XWSCXCL58XWS-CXCR2-CXCL5
13.79Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
13.79Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
13.79Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
13.79Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
13.79Consensusalpha1_offOrthosteric Ligandalpha1a_off
13.79Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
13.79Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
13.79Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
13.79Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
13.79Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
13.79Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
13.79Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
13.79Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
13.79Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
13.64Single3RFMCaffeine3RFM-A2A-Caffeine
13.64Single6TQ9SB-4081246TQ9-OX1-SB-408124
13.64Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
13.64Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
13.64Single9CHUNoradrenaline9CHU-β2-Noradrenaline
13.64Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
13.64Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
13.64Consensusp2y_offOrthosteric Ligandp2y1_off
13.51Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
13.51Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
13.51Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
13.51Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
13.51Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
13.51Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
13.51Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
13.51Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
13.51Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
13.51Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
13.33Single5X93K-87945X93-ETB-K-8794
13.33Single7EZCUKA7EZC-A2A-UKA
13.33Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
13.33Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
13.33Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
13.33Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
13.33Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
13.33Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
13.33Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
13.33Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
13.33Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
13.33Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
13.33Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
13.33Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
13.33Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
13.33Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
13.33Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.33Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8XVUCXCL28XVU-CXCR2-CXCL2
13.33Single8XWFCXCL38XWF-CXCR2-CXCL3
13.33Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
13.33Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
13.33Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
13.33Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
13.33Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
13.33Consensusendothelin_offOrthosteric Ligandetb_off
13.33Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
13.33Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Consensusprostanoid_offOrthosteric Ligandep_off dp_off
13.16Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
13.16Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
13.16Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
13.16Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
13.16Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
13.16Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
13.16Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
13.16Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
13.16Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
13.16Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
13.04Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
13.04Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
13.04Single4XNWMRS25004XNW-P2Y1-MRS2500
13.04Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
13.04Single6ME5Agomelatine6ME5-MT1-Agomelatine
13.04Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
13.04Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
13.04Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
13.04Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
13.04Single7WC5Psilocin7WC5-5-HT2A-Psilocin
13.04Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
13.04Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.04Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
13.04Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
13.04Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
13.04Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
13.04Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
13.04Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
13.04Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
13.04Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
13.04Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
13.04Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
13.04Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
13.04Consensus5ht2_onOrthosteric Ligand5ht2b_on
13.04Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
13.04Consensusgi_sensoryOrthosteric Ligandgi_opsins
13.04Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
13.04Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
13.04Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
13.04Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
13.04Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
13.04Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
12.90Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
12.90Single6KNMJN241-96KNM-Apelin-JN241-9
12.90Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
12.90Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
12.90Single7XN9L-054,5227XN9-SST2-L-054,522
12.90Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
12.90Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
12.90Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
12.90Single8XQJJN2418XQJ-Apelin-JN241
12.90Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
12.90Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
12.90Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
12.90Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
12.90Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.90Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.82Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
12.82Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
12.50Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
12.50Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
12.50Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
12.50Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
12.50Single3PBLEticlopride3PBL-D3-Eticlopride
12.50Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
12.50Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
12.50Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
12.50Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.50Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
12.50Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
12.50Single7SRQLSD7SRQ-5-HT2B-LSD
12.50Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
12.50Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
12.50Single7UL2SR486927UL2-NTS1-SR48692-Na
12.50Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
12.50Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
12.50Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
12.50Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
12.50Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
12.50Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
12.50Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
12.50Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
12.50Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
12.50Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
12.50Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
12.50Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
12.50Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
12.50Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
12.50Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
12.50Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
12.50Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
12.50Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
12.50Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
12.50Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
12.50Single8WDTphotoNECA8WDT-A2A-photoNECA
12.50Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
12.50Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
12.50Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
12.50Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
12.50Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
12.50Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
12.50Single9B9Y7DY9B9Y-CB1-7DY
12.50Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
12.50Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
12.50Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
12.50Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
12.50Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
12.50Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
12.50Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
12.50Consensusneurotensin_offOrthosteric Ligandnts1_off
12.50Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
12.50Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
12.50Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
12.50Consensussomatostatin_offOrthosteric Ligandsst2_off
12.20Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
12.20Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.12Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
12.12Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
12.12Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
12.12Single7XNACYN1548067XNA-SST2-CYN154806
12.12Single8IEBA1LYA8IEB-GPR156-A1LYA
12.12Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
12.12Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
12.12Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
12.00Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
12.00Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
12.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
12.00Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
12.00Single4BWBNeurotensin4BWB-NTS1-Neurotensin
12.00Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
12.00Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
12.00Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
12.00Single5U09Taranabant5U09-CB1-Taranabant
12.00Single6B73MP11046B73-κ-MP1104
12.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
12.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
12.00Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
12.00Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
12.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
12.00Single6ME9Ramelteon6ME9-MT2-Ramelteon
12.00Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
12.00Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
12.00Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
12.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
12.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
12.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
12.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
12.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
12.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
12.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.00Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
12.00Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
12.00Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
12.00Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
12.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
12.00Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
12.00Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
12.00Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
12.00Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
12.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
12.00Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
12.00Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
12.00Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
12.00Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
12.00Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
12.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
12.00Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
12.00Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
12.00Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
12.00Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
12.00Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
12.00Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
12.00Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
12.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
12.00Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
12.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
12.00Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
12.00Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
12.00Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
12.00Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
12.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
12.00Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
12.00Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
12.00Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
12.00Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
12.00Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
12.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
12.00Single8Y0HVUF114188Y0H-CXCR3-VUF11418
12.00Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
12.00Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
12.00Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
12.00Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
12.00Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
12.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
12.00Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
12.00Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
12.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
12.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
12.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
12.00Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
12.00Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
12.00Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
12.00Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
12.00Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
12.00Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
12.00Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
12.00Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
12.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
12.00Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
12.00Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
12.00Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
11.90Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
11.90Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
11.76Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
11.76Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
11.76Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
11.76Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
11.76Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
11.76Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
11.76Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
11.63Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
11.54Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
11.54Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
11.54Single3RZECidoxepin3RZE-H1-Cidoxepin
11.54Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
11.54Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
11.54Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
11.54Single5IU7Q274563465IU7-A2A-Q27456346-Na
11.54Single5IUBQ274563445IUB-A2A-Q27456344-Na
11.54Single5JTBZM-2413855JTB-A2A-ZM-241385
11.54Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
11.54Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
11.54Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
11.54Single5UVIZM-2413855UVI-A2A-ZM-241385
11.54Single6A94Zotepine6A94-5-HT2A-Zotepine
11.54Single6AQFZM-2413856AQF-A2A-ZM-241385
11.54Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
11.54Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
11.54Single6KUXRS-799486KUX-α2a-RS-79948
11.54Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
11.54Single6MH8ZM-2413856MH8-A2A-ZM-241385
11.54Single6PS0S-Carazolol6PS0-β2-S-Carazolol
11.54Single6PS4ICI118-5516PS4-β2-ICI118-551
11.54Single6PS5S-Propranolol6PS5-β2-S-Propranolol
11.54Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
11.54Single6TPGEMPA6TPG-OX2-EMPA
11.54Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
11.54Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
11.54Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
11.54Single6ZINSR486926ZIN-NTS1-SR48692
11.54Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
11.54Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
11.54Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
11.54Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
11.54Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
11.54Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
11.54Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
11.54Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
11.54Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
11.54Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
11.54Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
11.54Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
11.54Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single7T32ZM-2413857T32-A2A-ZM-241385
11.54Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
11.54Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
11.54Single7UL3Famotidine7UL3-H2-Famotidine
11.54Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
11.54Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
11.54Single7VV6C48/807VV6-MRGPRX2-C48/80
11.54Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
11.54Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
11.54Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
11.54Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
11.54Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
11.54Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
11.54Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
11.54Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
11.54Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
11.54Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
11.54Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
11.54Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
11.54Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
11.54Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
11.54Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
11.54Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
11.54Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
11.54Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
11.54Single8K2WAMG4878K2W-CXCR3-AMG487
11.54Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
11.54Single8K5CAcipimox8K5C-HCA2-Acipimox
11.54Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
11.54Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
11.54Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
11.54Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
11.54Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
11.54Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.54Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
11.54Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
11.54Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
11.54Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
11.54Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
11.54Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
11.54Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
11.54Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
11.54Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
11.54Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
11.54Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single9BJKNaloxone9BJK-μ-Naloxone-NAM
11.54Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
11.54Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
11.54Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
11.54Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
11.54Consensusa2_offOrthosteric Liganda2a_off
11.54Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
11.54Consensusalpha1_onOrthosteric Ligandalpha1a_on
11.54Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
11.54Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
11.54Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
11.54Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
11.54Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
11.54Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
11.54Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
11.54Consensushca_onOrthosteric Ligandhca2_on
11.54Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
11.54Consensusopsins_offOrthosteric Ligandrhodopsin_off
11.54Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
11.54Consensussensory_offOrthosteric Ligandopsins_off
11.43Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
11.43Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
11.43Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
11.43Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
11.43Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.43Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
11.43Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
11.43Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
11.43Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
11.43Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
11.11Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
11.11Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
11.11Single2Y01Dobutamine2Y01-β1-Dobutamine
11.11Single2Y02Carmoterol2Y02-β1-Carmoterol
11.11Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
11.11Single3EMLZM-2413853EML-A2A-ZM-241385
11.11Single3NY8ICI118-5513NY8-β2-ICI118-551
11.11Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
11.11Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
11.11Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
11.11Single4DAJTiotropium4DAJ-M3-Tiotropium
11.11Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
11.11Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
11.11Single4GBRS-Carazolol4GBR-β2-S-Carazolol
11.11Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
11.11Single4MQSIperoxo4MQS-M2-Iperoxo
11.11Single4QIMANTA XV4QIM-SMO-ANTA XV
11.11Single4QKX35V4QKX-β2-35V
11.11Single4U14Tiotropium4U14-M3-Tiotropium
11.11Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
11.11Single5DHGC-355DHG-NOP-C-35
11.11Single5IU8Q274563475IU8-A2A-Q27456347-Na
11.11Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
11.11Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
11.11Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
11.11Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
11.11Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
11.11Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
11.11Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
11.11Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
11.11Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
11.11Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
11.11Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
11.11Single6GPSMK08126GPS-CCR2-MK0812
11.11Single6H7MSalbutamol6H7M-β1-Salbutamol
11.11Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
11.11Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
11.11Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
11.11Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
11.11Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
11.11Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
11.11Single6S0LZM-2413856S0L-A2A-ZM-241385
11.11Single6TOTLemborexant6TOT-OX1-Lemborexant
11.11Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
11.11Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
11.11Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
11.11Single7BU7BI1671077BU7-β1-BI167107
11.11Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
11.11Single7F83PF-051904577F83-Ghrelin-PF-05190457
11.11Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
11.11Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
11.11Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
11.11Single7PYRPSB-21157PYR-A2A-PSB-2115
11.11Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
11.11Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
11.11Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
11.11Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
11.11Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
11.11Single7UL4Alvimopan7UL4-μ-Alvimopan
11.11Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
11.11Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
11.11Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
11.11Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
11.11Single7WC7Lisuride7WC7-5-HT2A-Lisuride
11.11Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
11.11Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
11.11Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
11.11Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
11.11Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
11.11Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
11.11Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
11.11Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
11.11Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
11.11Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
11.11Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
11.11Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
11.11Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
11.11Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
11.11Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
11.11Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
11.11Single8JJOAlprenolol8JJO-β2-Alprenolol
11.11Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
11.11Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
11.11Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
11.11Single8K5DGSK2560738K5D-HCA2-GSK256073
11.11Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
11.11Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
11.11Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
11.11Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
11.11Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
11.11Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
11.11Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
11.11Single8X63Mepyramine8X63-H1-Mepyramine
11.11Single8X64Desloratadine8X64-H1-Desloratadine
11.11Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
11.11Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
11.11Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
11.11Single9B9ZA1AKO9B9Z-CB1-A1AKO
11.11Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
11.11Single9CHXS-Carazolol9CHX-β2-S-Carazolol
11.11Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
11.11Single9IYAONO-97105319IYA-GPR55-ONO-9710531
11.11Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
11.11Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
11.11Consensus5ht5_onOrthosteric Ligand5ht5a_on
11.11Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
11.11Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
11.11Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
11.11Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
11.11Consensusalpha2_onOrthosteric Ligandalpha2b_on
11.11Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
11.11Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
11.11Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
11.11Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
11.11Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
11.11Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
11.11Consensusblt_onOrthosteric Ligandblt1_on
11.11Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
11.11Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
11.11Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
11.11Consensusdopamine_offOrthosteric Ligandd2_off d3_off
11.11Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
11.11Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
11.11Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
11.11Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
11.11Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
11.11Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
11.11Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
11.11Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
11.11Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
11.11Consensushca_on_gpOrthosteric Ligandhca2_on_gp
11.11Consensushistamine_offOrthosteric Ligandh1_off
11.11Consensusleukotriene_onOrthosteric Ligandblt_on
11.11Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
11.11Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
11.11Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
11.11Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
10.81Single6FJ3PTH6FJ3-PTH1-PTH
10.81Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
10.81Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
10.81Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
10.81Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
10.71Single2RH1S-Carazolol2RH1-β2-S-Carazolol
10.71Single2Y00Dobutamine2Y00-β1-Dobutamine
10.71Single2YCWS-Carazolol2YCW-β1-S-Carazolol
10.71Single5D6LS-Carazolol5D6L-β2-S-Carazolol
10.71Single5IUAQ274563485IUA-A2A-Q27456348-Na
10.71Single5JQHS-Carazolol5JQH-β2-S-Carazolol
10.71Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
10.71Single5TVNLSD5TVN-5-HT2B-LSD
10.71Single5WIUNemonapride5WIU-D4-Nemonapride
10.71Single5WIVNemonapride5WIV-D4-Nemonapride-Na
10.71Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
10.71Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
10.71Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
10.71Single6D26Fevipiprant6D26-DP2-Fevipiprant
10.71Single6E67BI1671076E67-β2-BI167107-Gs (fused)
10.71Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
10.71Single6GPXMK08126GPX-CCR2-MK0812
10.71Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
10.71Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
10.71Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
10.71Single6LUQHaloperidol6LUQ-D2-Haloperidol
10.71Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
10.71Single6PS6Timolol6PS6-β2-Timolol
10.71Single6S0QZM-2413856S0Q-A2A-ZM-241385
10.71Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
10.71Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
10.71Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
10.71Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
10.71Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
10.71Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
10.71Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
10.71Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
10.71Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
10.71Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
10.71Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
10.71Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
10.71Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
10.71Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
10.71Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
10.71Single8TF5Oleic acid8TF5-GPR6-Oleic acid
10.71Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
10.71Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
10.71Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
10.71Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
10.71Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
10.71Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
10.71Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
10.71Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
10.71Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
10.71Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
10.71Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
10.71Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
10.71Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
10.71Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
10.71Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
10.71Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
10.71Consensusamine_offonOrthosteric Ligandamine_off amine_on
10.71Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
10.71Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
10.71Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
10.71Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
10.71Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
10.71Consensusblt_offOrthosteric Ligandblt1_off
10.71Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
10.71Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
10.71Consensusdp_offOrthosteric Liganddp2_off
10.71Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
10.71Consensusep_offOrthosteric Ligandep4_off
10.71Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
10.71Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.71Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
10.71Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
10.71Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.71Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
10.71Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.71Consensustrace-amine_onOrthosteric Ligandta1_on
10.53Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
10.53Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
10.53Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
10.53Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
10.53Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
10.34Single2YDVNECA2YDV-A2A-NECA
10.34Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
10.34Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
10.34Single4DJHJDTic4DJH-κ-JDTic
10.34Single4U15Tiotropium4U15-M3-Tiotropium
10.34Single4UHRCGS216804UHR-A2A-CGS21680
10.34Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
10.34Single5D5AS-Carazolol5D5A-β2-S-Carazolol
10.34Single5D5BS-Carazolol5D5B-β2-S-Carazolol
10.34Single5G53NECA5G53-A2A-NECA-Gs
10.34Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
10.34Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.34Single6OL9Tiotropium6OL9-M5-Tiotropium
10.34Single6WGTLSD6WGT-5-HT2A-LSD
10.34Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
10.34Single7F1TMIP-1a7F1T-CCR5-MIP-1a
10.34Single7PX4PSB-21137PX4-A2A-PSB-2113
10.34Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
10.34Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
10.34Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
10.34Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
10.34Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
10.34Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
10.34Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
10.34Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
10.34Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
10.34Single8EA0Iperoxo8EA0-M3-Iperoxo
10.34Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
10.34Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
10.34Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
10.34Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
10.34Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
10.34Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
10.34Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
10.34Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
10.34Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
10.34Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
10.34Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
10.34Single9BJKNAM9BJK-μ-Naloxone-NAM
10.34Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
10.34Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
10.34Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
10.34Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
10.34Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
10.34Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
10.34Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
10.34Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
10.34Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
10.34Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
10.34Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.34Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
10.34Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
10.34Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
10.34Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
10.26Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
10.26Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
10.26Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
10.26Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
10.26Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
10.00Single3D4STimolol3D4S-β2-Timolol
10.00Single4AMIBucindolol4AMI-β1-Bucindolol
10.00Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
10.00Single5CXVTiotropium5CXV-M1-Tiotropium
10.00Single5X33BIIL2605X33-BLT1-BIIL260
10.00Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
10.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
10.00Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
10.00Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
10.00Single6IIURamatroban6IIU-TP-Ramatroban
10.00Single6OS2TRV0266OS2-AT1-TRV026
10.00Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
10.00Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
10.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
10.00Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
10.00Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
10.00Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
10.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
10.00Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
10.00Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
10.00Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
10.00Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
10.00Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
10.00Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
10.00Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
10.00Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8XQJJN2418XQJ-Apelin-JN241
10.00Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
10.00Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
10.00Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
10.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
10.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
10.00Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
10.00Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
10.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
10.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
9.76Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
9.68Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
9.68Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
9.68Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
9.68Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
9.68Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
9.68Single6H7LDobutamine6H7L-β1-Dobutamine
9.68Single6IBLArformoterol6IBL-β1-Arformoterol
9.68Single6K1QIRL25006K1Q-ETB-IRL2500
9.68Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
9.68Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
9.68Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
9.68Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
9.68Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
9.68Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
9.68Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
9.68Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
9.68Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
9.68Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
9.68Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
9.68Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
9.68Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
9.68Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
9.68Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
9.52Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
9.52Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
9.52Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
9.52Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single5EE7MK08935EE7-Glucagon-MK0893
9.38Single5WF6UK-4320975WF6-A2A-UK-432097
9.38Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
9.38Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
9.38Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
9.38Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
9.38Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
9.38Single8IEIA1LYA8IEI-GPR156-A1LYA
9.38Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single8X5YAstemizole8X5Y-H1-Astemizole
9.38Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
9.38Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
9.38Consensuskisspeptin_onOrthosteric Ligandkiss1_on
9.30Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
9.09Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
9.09Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
9.09Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
9.09Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
9.09Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.09Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
9.09Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
9.09Single8IEPA1LYA8IEP-GPR156-A1LYA
9.09Single8IEPA1LYA8IEP-GPR156-A1LYA
9.09Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
9.09Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
9.09Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
9.09Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
9.09Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
9.09Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.09Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
9.09Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
9.09Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
9.09Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
9.09Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
8.82Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
8.82Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
8.70Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
8.70Single3OE8IT1t3OE8-CXCR4-IT1t
8.70Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
8.70Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
8.70Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
8.70Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
8.70Single8A2OTheophylline8A2O-A2A-Theophylline-Na
8.70Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
8.70Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
8.70Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
8.70Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
8.70Consensussensory_onOrthosteric Ligandopsins_on
8.33Single3OE6IT1t3OE6-CXCR4-IT1t
8.33Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
8.33Single3UZAGTPL92363UZA-A2A-GTPL9236
8.33Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
8.33Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
8.33Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
8.33Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
8.33Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
8.33Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
8.33Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
8.33Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
8.33Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
8.33Single8JPSCCL78JPS-ACKR1-CCL7
8.33Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
8.33Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
8.33Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
8.33Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
8.33Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
8.33Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
8.33Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
8.00Single3OE9IT1t3OE9-CXCR4-IT1t
8.00Single4O9RCyclopamine4O9R-SMO-Cyclopamine
8.00Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
8.00Single6LI0C176LI0-GPR52-C17
8.00Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
8.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
8.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
8.00Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
8.00Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
8.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
8.00Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
8.00Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
8.00Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
8.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
8.00Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
8.00Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
8.00Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
8.00Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
8.00Single8K5BNiacin8K5B-HCA2-Niacin
8.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
8.00Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
8.00Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
8.00Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
8.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
8.00Consensusgq_nucleotideOrthosteric Ligandgq_p2y
8.00Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
8.00Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
7.89Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
7.89Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
7.89Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
7.69Single3ODUIT1t3ODU-CXCR4-IT1t
7.69Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
7.69Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
7.69Single4QINSAG1.54QIN-SMO-SAG1.5
7.69Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
7.69Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
7.69Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
7.69Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
7.69Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
7.69Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
7.69Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
7.69Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
7.69Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
7.69Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
7.69Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
7.69Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
7.69Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
7.69Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
7.69Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
7.69Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
7.69Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.69Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
7.69Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
7.69Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.69Single9BA0A1AKN9BA0-CB1-A1AKN
7.69Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
7.69Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
7.69Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
7.50Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
7.50Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
7.41Single2YDOAdenosine2YDO-A2A-Adenosine
7.41Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
7.41Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
7.41Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
7.41Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
7.41Single6VI4JDTic6VI4-κ-JDTic
7.41Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
7.41Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
7.41Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
7.41Single6ZG9GSK10347026ZG9-M1-GSK1034702
7.41Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.41Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
7.41Single7VODCariprazine7VOD-5-HT2A-Cariprazine
7.41Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
7.41Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
7.41Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
7.41Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.41Single8IHKAcifran8IHK-HCA3-Acifran
7.41Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
7.41Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.41Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
7.41Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
7.41Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
7.41Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
7.41Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
7.41Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
7.14Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
7.14Single5DHHSB-6121115DHH-NOP-SB-612111
7.14Single5DSGTiotropium5DSG-M4-Tiotropium
7.14Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
7.14Single6IIVDaltroban6IIV-TP-Daltroban
7.14Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
7.14Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
7.14Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
7.14Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
7.14Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
7.14Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
7.14Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
7.14Single8T1WCVN4248T1W-GPR6-CVN424
7.14Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
7.14Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
6.90Single4JKVTaladegib4JKV-SMO-Taladegib
6.90Single5CGCHTL142425CGC-mGlu5-HTL14242
6.90Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
6.90Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
6.90Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
6.90Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
6.90Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
6.90Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
6.90Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
6.90Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
6.90Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
6.82Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
6.82Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
6.67Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
6.67Single5V56TC1145V56-SMO-TC114
6.67Single5V57TC1145V57-SMO-TC114
6.67Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
6.67Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
6.67Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
6.67Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
6.67Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
6.67Consensusrelaxin_onOrthosteric Ligandrxfp4_on
6.67Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
6.45Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
6.45Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
6.45Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
6.45Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
6.25Single5CGDHTL142425CGD-mGlu5-HTL14242
6.25Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
6.25Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
6.25Single8XVJMacitentan8XVJ-ETA-Macitentan
5.88Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
5.88Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
5.88Single8IEIA1LYA8IEI-GPR156-A1LYA
5.71Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
5.71Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
5.41Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
5.41Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
5.26Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.26Single6D35Cholesterol6D35-SMO-Cholesterol
5.26Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.26Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.26Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
5.26Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
5.26Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
5.26Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
5.26Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
5.26Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
5.26Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
5.26Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
5.26Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.26Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
5.26Single7DTTCa7DTT-CaS-Ca-Ca
5.26Single7DTTCa7DTT-CaS-Ca-Ca
5.26Single7DTUTryptophan7DTU-CaS-Tryptophan
5.26Single7DTUTryptophan7DTU-CaS-Tryptophan
5.26Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.26Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.26Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.26Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.26Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.26Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.26Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.26Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.26Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
5.26Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.26Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.26Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.26Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.26Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.26Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.26Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
5.26Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
5.26Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.26Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.26Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.26Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.26Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.26Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.26Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.26Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.26Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.26Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.26Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.26Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.26Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.26Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.26Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.26Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
5.26Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
5.26Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.26Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.26Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.26Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.26Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.26Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.26Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
5.26Single7XW7K1-707XW7-TSH-K1-70
5.26Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
5.26Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.26Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.26Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.26Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.26Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.26Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.26Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.26Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.26Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.26Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.26Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.26Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.26Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
5.26Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.26Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.26Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.26Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.26Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
5.26Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
5.26Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.26Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.26Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
5.26Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
5.26Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
5.26Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
5.26Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.26Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.26Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
5.26Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
5.26Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
5.26Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
5.26Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
5.26Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.26Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
5.26Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.26Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.26Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.26Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.26Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.26Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.26Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.26Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.26Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.26Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.26Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.26Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.26Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.26Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.26Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.26Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.26Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
5.26Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
5.26Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
5.26Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
5.26Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
5.26Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
5.26Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.26Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.26Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.26Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.26Single8WVXNorrin8WVX-LGR4-Norrin
5.26Single8WVYNorrin8WVY-LGR4-Norrin
5.26Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.26Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.26Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.26Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.26Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.26Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.26Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.26Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
5.26Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.26Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.26Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.26Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.26Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.26Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.26Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.26Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.26Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.26Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.26Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.26Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
5.26Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.26Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.26Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.26Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.13Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
5.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.00Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.00Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.00Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
5.00Single8W8SAA-148W8S-GPR101-AA-14
5.00Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.00Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.88Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
4.76Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.76Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.76Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
4.76Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.76Single8W8RAA-148W8R-GPR101-AA-14-chim(NtGi1-Gs)/β1/γ2
4.65Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
4.65Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
4.55Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
4.55Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
4.55Single5MZPCaffeine5MZP-A2A-Caffeine-Na
4.55Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.55Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.55Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
4.55Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.55Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.55Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
4.55Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
4.44Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
4.35Single5L7DCholesterol5L7D-SMO-Cholesterol
4.35Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
4.35Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.35Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
4.35Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
4.35Single8HS2Fab0468HS2-GPR20-Fab046
4.35Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.35Single8PWNTheophylline8PWN-A2A-Theophylline
4.35Single9GE2Cholesterol9GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
4.17Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
4.17Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
4.17Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
4.17Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
4.08Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
4.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
4.00Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
4.00Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
4.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
4.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
4.00Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
4.00Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
4.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
3.85Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
3.85Single5L7IVismodegib5L7I-SMO-Vismodegib
3.85Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
3.85Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
3.85Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
3.85Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
3.85Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.85Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
3.85Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.85Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
3.70Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
3.70Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
3.70Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
3.70Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
3.70Single8G94CD698G94-S1P1-CD69-Gi1/β1/γ2
3.70Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
3.70Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
3.70Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
3.70Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
3.57Single6FFIMMPEP6FFI-mGlu5-MMPEP
3.57Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
3.57Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
3.57Single8IYXYL-3658IYX-GPR34-YL-365
3.45Single6FFHFenobam6FFH-mGlu5-Fenobam
3.45Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
3.45Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
3.33Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
3.33Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
3.23Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
3.23Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
3.23Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.23Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.12Single4N4WSANT-14N4W-SMO-SANT-1
3.12Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
2.94Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
2.86Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.86Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.78Single7SHEPI; PE7SHE-GPR158-PI; PE
2.70Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.70Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
2.63Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
2.63Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.56Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
2.44Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
2.44Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
8IOC 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
Net Summary
Imin 3.27
Number of Linked Nodes 847
Number of Links 986
Number of Hubs 136
Number of Links mediated by Hubs 525
Number of Communities 30
Number of Nodes involved in Communities 216
Number of Links involved in Communities 300
Path Summary
Number Of Nodes in MetaPath 108
Number Of Links MetaPath 107
Number of Shortest Paths 1807928
Length Of Smallest Path 3
Average Path Length 33.4724
Length of Longest Path 55
Minimum Path Strength 1.43
Average Path Strength 6.77758
Maximum Path Strength 22.94
Minimum Path Correlation 0.7
Average Path Correlation 0.980993
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.32558
Average % Of Corr. Nodes 40.9513
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 48.369
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
melanocortin_on_gpmc1_on_gp
mc4_on_gp
mc2_on_gp
mc3_on_gp
mc5_on_gp



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