Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.33 1.845404
2G.S1.02 5.818585
3G.S1.06 3.5125408
4G.H1.04 4.3875497
5G.H1.07 4.848599
6G.S2.01 5419
7G.S2.05 5.295413
8G.S2.08 8.0825485
9G.S3.01 4.7025484
10G.S3.03 7.34587
11G.S3.04 5.342516
12G.S3.05 3.31667687
13G.S3.06 6.26333615
14G.S3.08 3.7419
15G.s3h2.03 4.01833619
16G.H2.04 3.58419
17G.H2.06 5.6619
18G.H2.07 4.8875419
19G.h2s4.01 5.48519
20G.S4.03 3.515497
21G.s4h3.01 7.1475427
22G.s4h3.04 7.455428
23G.H3.01 7.2425429
24G.H3.02 3.07428
25G.H3.09 5.4925409
26G.H3.13 4.40254195
27G.H3.14 6.8925408
28G.H3.17 5.9345165
29G.S5.03 3.44598
30G.S5.05 3.88333699
31G.S5.07 6.0125499
32G.HG.03 5.5354186
33G.HG.14 2.1375405
34G.hgh4.01 3.67426
35G.hgh4.02 3.47625827
36G.H4.11 3.335427
37G.H4.15 3.4925428
38G.h4s6.02 5.394198
39G.h4s6.04 2.84404
40G.h4s6.11 5.4254197
41G.S6.02 5.465227
42G.s6h5.01 5.428599
43G.H5.03 4.755498
44G.H5.20 5.285439
45G.H5.23 4.3825404
46G.H5.25 4.0675437
47b.1x1 2.742504
48b.h2x1 2.8854175
49b.h2x5 4.85754175
50b.l1x3 7.083336129
51b.b2x1 6.29254168
52b.b2x5 4.976507
53b.b4x4 8.62754128
54b.b4x5 3.414267
55b.b4x6 8.227147129
56b.b5x3 5.647147129
57b.b5x5 4.3125405
58b.b5x7 3.624137
59b.l5x1 4.81754138
60b.l5x5 6.84619
61b.b6x5 4.2445266
62b.b7x1 5.54404
63b.b7x4 3.31754138
64b.b8x4 3.715136
65b.l8x8 3.5654134
66b.l9x3 7.366676119
67b.l9x6 4.01571718
68b.l9x7 3.5654117
69b.b10x5 3.9975409
70b.b11x4 5.0754119
71b.b11x5 4.4475446
72b.l11x2 7.354119
73b.b12x6 9.286118
74b.l12x1 3.79406
75b.b13x7 5.916547
76b.l13x3 8.15549
77b.b14x3 4.244545
78b.b15x1 5.945649
79b.b16x4 10.8775446
80b.b16x5 3.296505
81b.b16x6 8.71648
82b.b17x7 8.61458
83b.l17x3 5.34571759
84b.l17x6 5.6225419
85b.l17x7 3.64457
86b.b18x3 2.9425458
87b.l18x1 4.834297146
88b.l18x2 5.66754147
89b.b19x2 5.582556
90b.b19x4 4.994558
91b.l19x2 5.374559
92b.b20x2 5.67456
93b.b20x4 7.70333658
94b.b20x6 7.63556
95b.l20x2 8.745409
96b.b21x1 4.3275457
97b.b21x7 5.40167605
98b.l21x5 3.74754104
99b.b22x5 4.6025147
100b.l22x5 6.6475409
101b.b23x6 6.726107
102b.b24x4 8.424106
103b.b24x6 5.54754108
104b.l24x3 6.03254175
105b.b25x3 7.4225105
106b.l25x3 7.376579
107b.l26x5 4.0254255
108b.l27x1 7.781437169
109b.l27x2 9.15479
110b.b28x3 4.4054127
111b.b28x6 8.664579
112b.b28x7 4.794259
113g.ntx3 3.04754244
114g.h1x1 4.8654242
115g.l1x4 4.475458
116g.h2x11 5.55754146
117g.ctx3 6.703336289
118g.ctx14 2.7654259
119g.ctx16 4.994508
120NT.H18 8.4454298
121NT.Y19 8.9825469
1221x46 4.5975407
1231x50 5.28539
1241x57 4.49407
1252x38 5.23754315
1262x46 3.97439
1272x57 8.88407
1282x61 4.5825406
1293x25 5.04571769
1303x26 4.66465
1313x28 8.1675465
1323x29 7.6425465
1333x33 5.545465
1343x43 2.846538
1353x46 3.9875439
1363x50 4.614539
1373x54 4.415408
1383x56 7.67505
1394x42 3.54406
1404x50 3.08754209
1414x53 3.084207
1424x56 1.315406
143E2.Y189 7665
1445x39 7.11833667
1455x58 5.16509
1466x33 4.2875438
1476x44 5.7125439
1486x48 8.595439
1496x52 5.94327
150E3.C282 4.27254154
1517x31 3.85151
1527x33 5.57754304
1537x45 8.932539
1547x49 3.5525439
1557x50 3.636539
1567x53 4.136539
157Lig 7.122311300
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1G.HN.47 b.b5x3 52.63192.82NoYes069
2G.HN.47 b.b4x2 52.48524.23NoNo068
3b.b28x7 g.ctx16 66.61794.83YesYes098
4b.b28x7 b.l26x5 66.95194.21YesYes2595
5b.l26x5 g.ctx4 68.3195.03YesNo057
6g.ctx3 g.ctx4 68.45754.83YesNo097
7g.ctx3 g.ctx6 69.42468.14YesNo096
8b.l22x5 g.ctx6 69.83792.43YesNo096
9b.l22x5 b.l24x2 69.97214.86YesNo096
10b.h2x1 b.l24x2 70.09162.77YesNo1756
11b.b21x5 b.h2x1 72.24844.24NoYes045
12b.b21x5 b.b21x7 72.79239.58NoYes045
13b.b21x7 b.b24x6 77.89736.75YesYes058
14b.b23x6 b.b24x6 78.0635.79YesYes1078
15b.b23x6 b.l23x2 79.88154.6YesNo078
16b.l21x7 b.l23x2 80.40764.67NoNo058
17b.l21x7 b.l23x1 80.67027.78NoNo056
18b.l23x1 b.l25x6 80.93253.57NoNo068
19b.l25x6 b.l27x1 81.06369NoYes089
20b.b2x1 b.l27x1 79.19475.79YesYes1689
21b.b2x1 b.l3x1 79.98635.64YesNo089
22b.l3x1 b.l5x5 80.11129.86NoYes099
23G.S2.03 b.l5x5 35.39523.27NoYes199
24G.S2.03 G.S3.04 35.42016.75NoYes196
25G.S3.06 b.l5x5 35.39899.02YesYes159
26G.S3.04 G.S3.06 64.67022.48YesYes165
27G.S2.05 G.S3.04 99.91427.86YesYes136
28G.H1.12 G.S2.05 99.98972.39NoYes083
29G.H1.10 G.H1.12 99.99242.65NoNo088
30G.H1.10 G.S2.04 99.9953.04NoNo086
31G.S2.04 G.S3.05 1004.52NoYes067
32G.S1.04 G.S3.05 49.66614.24NoYes077
33G.S1.04 G.S3.03 48.92562.44NoYes077
34G.S2.06 G.S3.05 47.57442.49NoYes897
35G.S2.06 G.S3.03 47.630213.93NoYes897
36G.H5.11 G.S3.03 95.30083.93NoYes887
37G.S1.05 G.h2s4.01 11.019510.96NoYes199
38G.S1.05 G.S1.07 10.94966.92NoNo099
39G.S2.01 G.S3.08 13.86663.07YesYes199
40G.S3.08 G.h2s4.01 13.86622.62YesYes199
41G.H3.12 G.S1.07 13.17885.71NoNo089
42G.H2.07 G.S3.08 27.57886.13YesYes199
43G.H2.04 G.H2.07 21.4123YesYes199
44G.H2.04 G.H3.08 21.06694.86YesNo199
45G.H3.08 G.H3.12 13.06522.85NoNo198
46G.H3.08 G.S4.04 33.86014.87NoNo099
47G.S4.04 G.S4.06 25.29392.62NoNo097
48G.H4.15 G.S4.06 20.23915.24YesNo087
49G.H5.11 G.H5.15 95.61633.07NoNo087
50G.H5.15 G.H5.19 95.98922.83NoNo078
513x53 G.H5.23 95.30186.76NoYes084
523x53 3x56 95.40037.76NoYes085
533x56 G.H5.19 95.89137.23YesNo058
543x50 G.H5.23 93.15885.57YesYes094
553x50 5x58 16.94385.14YesYes099
56b.b4x2 b.b5x8 52.45085.02NoNo085
57b.b5x7 b.b5x8 52.30363.39YesNo075
58b.b4x3 b.b5x7 48.59252.85NoYes077
59b.b3x3 b.b4x3 47.42724.47NoNo087
60b.b3x3 b.b6x5 47.11677.57NoYes2686
61b.b2x4 b.b6x5 47.27124.36NoYes066
62b.b10x4 b.b2x4 47.1210.16NoNo066
63b.b10x4 b.b14x3 46.80632.43NoYes465
64b.b14x3 b.b15x1 45.05944.87YesYes459
65b.b15x1 b.b16x6 12.270112.03YesYes498
66g.h1x11 g.h1x14 10.04061.33NoNo099
67b.b15x1 b.l16x1 23.66152.62YesNo094
68b.l16x1 b.l16x2 23.1446.54NoNo049
69b.l14x5 b.l16x2 11.75424.26NoNo059
70b.l14x5 b.l14x6 10.57632.43NoNo053
71b.b16x5 b.l14x6 10.41222.77YesNo053
72b.b16x5 b.b17x5 11.83162.66YesNo057
73b.b16x7 b.l16x2 11.2393.57NoNo099
74b.b16x7 b.b17x4 10.742313.1NoNo095
75b.b16x5 b.b17x4 10.54522.43YesNo055
76b.b4x6 b.b5x3 53.1099.28YesYes1299
77b.b1x6 b.b4x6 54.95089.11NoYes1299
78b.b1x6 b.b5x1 55.57042.95NoNo095
79b.b1x4 b.b5x1 55.71482.59NoNo075
80b.b28x5 g.ctx16 56.14853.77NoYes058
813x25 NT.Y19 12.47593.86YesYes699
823x25 3x29 16.38863.27YesYes695
833x29 Lig 19.00969.65YesYes050
843x36 Lig 32.11947.33NoYes070
853x36 6x48 32.37696.83NoYes079
866x44 6x48 32.32887.02YesYes399
873x43 6x44 32.69252.44YesYes389
883x43 7x53 68.98213.52YesYes389
893x50 7x53 68.98956.17YesYes399
903x40 Lig 47.99277.89NoYes080
913x40 6x48 32.37922.45NoYes089
926x48 7x45 32.679518.08YesYes399
933x43 7x45 33.20982.75YesYes389
943x40 5x50 16.01163.07NoNo088
953x44 5x50 16.13447.14NoNo078
963x44 5x54 16.3815.71NoNo078
975x54 5x58 16.50772.42NoYes089
986x57 E3.C282 13.13333.17NoYes054
996x54 6x57 14.44494.15NoNo055
1006x54 6x55 17.72262.77NoNo056
1016x51 6x55 18.37795.54NoNo076
1026x51 Lig 19.68836.42NoYes070
1033x37 Lig 10.506910.74NoYes060
104b.b1x4 b.b28x5 56.00362.51NoNo075
105G.S3.06 G.h2s4.01 18.83034.29YesYes159
106G.S2.01 G.S3.06 10.47315.02YesYes195
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
NT.K24NT.T2230NoNo6812
LigNT.K244.670YesNo0601
2x563x323.390NoNo5521
2x577x3815.240YesNo7521
2x603x283.620NoYes5512
2x60Lig11.820NoYes5010
3x253x2886YesYes9522
3x253x293.276YesYes9521
3x25E2.L1864.566YesNo9722
3x25E2.Y1895.796YesYes9522
3x29E2.L1865.36YesNo5712
3x29E2.Y18912.356YesYes5512
3x29Lig9.656YesYes5010
3x33E2.Y1894.136YesYes5512
3x335x399.286YesYes5712
3x33Lig7.266YesYes5010
3x366x486.830NoYes7912
3x36Lig7.330NoYes7010
3x374x533.20NoYes6712
3x37Lig10.740NoYes6010
3x405x503.070NoNo8812
3x406x482.450NoYes8912
3x40Lig7.890NoYes8010
E2.L186E2.Y1898.216NoYes7522
5x39E2.Y1895.966YesYes7522
5x43Lig11.560NoYes5010
5x475x482.6232NoNo8412
5x476x529.6532NoYes8712
5x47Lig4.8432NoYes8010
5x486x523.9332NoYes4722
6x516x555.540NoNo7612
6x51Lig6.420NoYes7010
7x387x422.830NoNo5712
7x38Lig7.330NoYes5010
7x34Lig2.090NoYes4010
6x517x411.580NoNo7712
3x334x571.516YesNo5812
3x373x411.470NoNo6512
3x32Lig0.990NoYes5010

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
100.00Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
70.59Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
70.59Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
64.71Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
64.71Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
62.50Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
62.50Single8E0GBU728E0G-μ-BU72
60.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
58.82Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
58.82Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
58.82Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
58.82Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
57.14Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
56.25Single5C1MBU725C1M-μ-BU72
56.25Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
56.25Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
56.25Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
55.56Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
55.56Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
55.00Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
53.33Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
53.33Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
50.00Single7DFPSpiperone7DFP-D2-Spiperone
50.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
50.00Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
50.00Single7V68Iperoxo7V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
50.00Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
50.00Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
50.00Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
50.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
50.00Single7YITNalfurafine7YIT-κ-Nalfurafine
50.00Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
50.00Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
50.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
50.00Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
50.00Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
50.00Consensuslpl_onOrthosteric Ligands1p_on lpa_on
50.00Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
50.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
50.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
50.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
47.37Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
47.37Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
47.37Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
47.37Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
47.37Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
47.06Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
47.06Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
47.06Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
47.06Single8JXSPF-61428JXS-D1-PF-6142
47.06Single8TF5Oleic acid8TF5-GPR6-Oleic acid
47.06Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
47.06Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
47.06Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
47.06Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
47.06Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
47.06Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
46.67Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
46.67Single6AKXA4R6AKX-CCR5-A4R
46.67Single6AKYMaraviroc6AKY-CCR5-Maraviroc
46.67Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
46.67Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
46.67Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
46.67Consensusorexin_offOrthosteric Ligandox2_off ox1_off
46.67Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
46.67Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
45.45Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
45.45Consensusangiotensin_onOrthosteric Ligandat1_on
45.45Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
45.00Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
45.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
44.44Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
44.44Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
44.44Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
44.44Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
44.44Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
44.44Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
44.44Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
44.44Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
44.44Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
44.44Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
44.44Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
44.44Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
44.44Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
44.44Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
44.44Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
44.44Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
44.44Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
44.44Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
44.44Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
43.75Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
43.75Single4MBSMaraviroc4MBS-CCR5-Maraviroc
43.75Single4ZJCSB-6740424ZJC-OX1-SB-674042
43.75Single6TPGEMPA6TPG-OX2-EMPA
43.75Single7UL3Famotidine7UL3-H2-Famotidine
43.75Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
43.75Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
43.75Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
43.75Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
43.75Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.75Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
43.75Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
43.75Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
43.48Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
43.48Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
43.48Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
43.48Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
43.48Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
42.86Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
42.86Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
42.86Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.86Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
42.86Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
42.11Single4RWADIPP-NH24RWA-δ-DIPP-NH2
42.11Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
42.11Single6A93Risperidone6A93-5-HT2A-Risperidone
42.11Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
42.11Single6ZG4HTL00099366ZG4-M1-HTL0009936
42.11Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
42.11Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
42.11Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
42.11Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
42.11Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
42.11Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
42.11Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
42.11Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
42.11Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
42.11Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
42.11Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
42.11Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
42.11Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
42.11Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
42.11Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
42.11Consensuslpa_offOrthosteric Ligandlpa1_off
42.11Consensuslpl_offOrthosteric Ligands1p_off lpa_off
42.11Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
42.11Consensusorexin_onOrthosteric Ligandox2_on
41.67Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
41.18Single2Y04Salbutamol2Y04-β1-Salbutamol
41.18Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
41.18Single6DRXLisuride6DRX-5-HT2B-Lisuride
41.18Single6TOTLemborexant6TOT-OX1-Lemborexant
41.18Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
41.18Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
41.18Single7UL4Alvimopan7UL4-μ-Alvimopan
41.18Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
41.18Single7V3ZCP559407V3Z-CB1-CP55940
41.18Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
41.18Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
41.18Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
41.18Single8JXRLSD8JXR-D1-LSD
41.18Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
41.18Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
41.18Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
41.18Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
41.18Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
41.18Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
41.18Consensus5ht5_onOrthosteric Ligand5ht5a_on
41.18Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
41.18Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
41.18Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
40.91Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
40.91Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
40.00Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
40.00Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
40.00Single5X93K-87945X93-ETB-K-8794
40.00Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
40.00Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
40.00Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
40.00Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
40.00Single7SRQLSD7SRQ-5-HT2B-LSD
40.00Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
40.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
40.00Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
40.00Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
40.00Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
40.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
40.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
40.00Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
40.00Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
40.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
40.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
40.00Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
40.00Consensusendothelin_offOrthosteric Ligandetb_off
40.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
40.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
40.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
40.00Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
40.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
40.00Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
39.13Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
39.13Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
39.13Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
39.13Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
39.13Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
39.13Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
38.89Single2Y03Isoprenaline2Y03-β1-Isoprenaline
38.89Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
38.89Single5WQCEMPA5WQC-OX2-EMPA
38.89Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
38.89Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
38.89Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
38.89Single6TP6Filorexant6TP6-OX1-Filorexant
38.89Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
38.89Single7C4SS1P7C4S-S1P3-S1P
38.89Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
38.89Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
38.89Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
38.89Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
38.89Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
38.89Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.89Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
38.89Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
38.89Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.89Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
38.89Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
38.89Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
38.89Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
38.89Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.89Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.89Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.89Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
38.89Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.89Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
38.89Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
38.89Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
38.89Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
38.89Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
38.89Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
38.89Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
38.89Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
38.89Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
38.89Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
38.89Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
38.89Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
38.89Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
38.46Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
38.46Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
38.46Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
38.46Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
38.10Single5ZTYAM102575ZTY-CB2-AM10257
38.10Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
38.10Single7SK9CCX6627SK9-ACKR3-CCX662
38.10Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
38.10Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
38.10Single8QJ2pN1628QJ2-MC4-pN162-Gs
38.10Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
38.10Single8X5YAstemizole8X5Y-H1-Astemizole
38.10Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
38.10Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
38.10Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
38.10Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
37.50Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
37.50Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
37.50Single5WS3EMPA5WS3-OX2-EMPA
37.50Single6B73MP11046B73-κ-MP1104
37.50Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
37.50Single6TODEMPA6TOD-OX1-EMPA-Na
37.50Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
37.50Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
37.50Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
37.50Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
37.50Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
37.50Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
37.50Single7XRRLemborexant7XRR-OX2-Lemborexant
37.50Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
37.50Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
37.50Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
37.50Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
37.50Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
37.50Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
37.50Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
37.50Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
37.50Single8Y0HVUF114188Y0H-CXCR3-VUF11418
37.50Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
37.50Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
37.50Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
37.50Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
37.50Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
37.50Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
37.50Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
37.50Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
37.50Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
37.50Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
37.50Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
36.84Single3P0GBI1671073P0G-β2-BI167107
36.84Single4DJHJDTic4DJH-κ-JDTic
36.84Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
36.84Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
36.84Single4U15Tiotropium4U15-M3-Tiotropium
36.84Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
36.84Single5V54Methiothepin5V54-5-HT1B-Methiothepin
36.84Single5XR8AM8415XR8-CB1-AM841
36.84Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
36.84Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
36.84Single6H7JIsoprenaline6H7J-β1-Isoprenaline
36.84Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
36.84Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
36.84Single6OL9Tiotropium6OL9-M5-Tiotropium
36.84Single6TQ7SB-3348676TQ7-OX1-SB-334867
36.84Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
36.84Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
36.84Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
36.84Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
36.84Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
36.84Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
36.84Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
36.84Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
36.84Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
36.84Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
36.84Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
36.84Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
36.84Single8EA0Iperoxo8EA0-M3-Iperoxo
36.84Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
36.84Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
36.84Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
36.84Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
36.84Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
36.84Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
36.84Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
36.84Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
36.84Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
36.84Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
36.84Consensus5ht1_offOrthosteric Ligand5ht1b_off
36.84Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
36.84Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
36.84Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
36.84Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
36.84Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
36.84Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
36.84Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
36.84Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
36.84Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
36.84Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
36.84Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
36.84Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
36.84Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
36.36Single4IARErgotamine4IAR-5-HT1B-Ergotamine
36.36Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
36.36Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
36.36Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
36.36Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
36.36Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
36.36Single8PKMBefiradol8PKM-5-HT1A-Befiradol-t7m-Gi1/β1/γ1
36.36Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
36.00Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
35.71Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.71Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
35.71Single9CHUNoradrenaline9CHU-β2-Noradrenaline
35.71Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
35.71Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
35.29Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
35.29Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
35.29Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
35.29Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
35.29Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
35.29Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
35.29Single6PS0S-Carazolol6PS0-β2-S-Carazolol
35.29Single6PS4ICI118-5516PS4-β2-ICI118-551
35.29Single6PS5S-Propranolol6PS5-β2-S-Propranolol
35.29Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
35.29Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
35.29Single6TPNHTL66416TPN-OX2-HTL6641
35.29Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
35.29Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
35.29Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
35.29Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
35.29Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
35.29Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
35.29Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
35.29Single7F61PF-036547467F61-H3-PF-03654746-Cholesterol
35.29Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.29Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
35.29Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
35.29Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
35.29Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
35.29Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.29Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
35.29Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
35.29Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
35.29Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
35.29Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
35.29Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
35.29Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
35.29Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
35.29Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.29Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.29Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
35.29Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
35.29Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
35.29Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
35.29Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
35.29Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
35.29Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
35.29Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
35.29Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
35.29Single8K9LDamgo8K9L-μ-Damgo-VV9-Gi3/β1/γ1
35.29Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
35.29Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.29Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
35.29Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.29Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
35.29Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
35.29Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
35.29Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
35.29Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
35.29Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
35.29Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
35.29Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
35.29Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
35.29Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
35.29Consensusalpha1_onOrthosteric Ligandalpha1a_on
35.29Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
35.29Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
35.29Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
35.29Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
35.29Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
35.00Single3D4STimolol3D4S-β2-Timolol
35.00Single4LDEBI1671074LDE-β2-BI167107
35.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
35.00Single5CXVTiotropium5CXV-M1-Tiotropium
35.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
35.00Single6CM4Risperidone6CM4-D2-Risperidone
35.00Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
35.00Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
35.00Single6MXTSalmeterol6MXT-β2-Salmeterol
35.00Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
35.00Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
35.00Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
35.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
35.00Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
35.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
35.00Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
35.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
35.00Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
35.00Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
35.00Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
35.00Single8JD3HZR; PEF8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
35.00Single8JJ8Formoterol8JJ8-β2-Formoterol
35.00Single8JJLOlodaterol8JJL-β2-Olodaterol
35.00Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
35.00Single8XYIVUF106618XYI-CXCR3-VUF10661
35.00Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
35.00Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
35.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
35.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
35.00Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
35.00Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
35.00Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
35.00Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
35.00Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
35.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
35.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
34.78Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
34.78Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
34.78Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
34.78Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
34.78Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
34.78Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
34.78Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
34.62Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
34.62Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
34.62Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
34.48Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
33.33Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
33.33Single3NY8ICI118-5513NY8-β2-ICI118-551
33.33Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
33.33Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
33.33Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
33.33Single4EJ4Naltrindole4EJ4-δ-Naltrindole
33.33Single4GBRS-Carazolol4GBR-β2-S-Carazolol
33.33Single4MQSIperoxo4MQS-M2-Iperoxo
33.33Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
33.33Single4QKX35V4QKX-β2-35V
33.33Single4U14Tiotropium4U14-M3-Tiotropium
33.33Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
33.33Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
33.33Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
33.33Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
33.33Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
33.33Single6H7MSalbutamol6H7M-β1-Salbutamol
33.33Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
33.33Single6PS1Timolol6PS1-β2-Timolol
33.33Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
33.33Single6PT2KGCHM076PT2-δ-KGCHM07
33.33Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
33.33Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
33.33Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
33.33Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
33.33Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
33.33Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
33.33Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
33.33Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
33.33Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
33.33Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
33.33Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
33.33Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
33.33Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
33.33Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
33.33Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
33.33Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
33.33Single7UM4AS26747237UM4-5-HT5A-AS2674723
33.33Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
33.33Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
33.33Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
33.33Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Single7WC7Lisuride7WC7-5-HT2A-Lisuride
33.33Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
33.33Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
33.33Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
33.33Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
33.33Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
33.33Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
33.33Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
33.33Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
33.33Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
33.33Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
33.33Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
33.33Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
33.33Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
33.33Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
33.33Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
33.33Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
33.33Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
33.33Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
33.33Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
33.33Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
33.33Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
33.33Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
33.33Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
33.33Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
33.33Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
33.33Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
33.33Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
33.33Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
33.33Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
33.33Single8PJKST1718PJK-5-HT1A-ST171-t7m-Gi1/β1/γ1
33.33Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
33.33Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
33.33Single8T1WCVN4248T1W-GPR6-CVN424
33.33Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
33.33Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
33.33Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
33.33Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
33.33Single8X63Mepyramine8X63-H1-Mepyramine
33.33Single8X64Desloratadine8X64-H1-Desloratadine
33.33Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
33.33Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
33.33Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
33.33Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
33.33Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
33.33Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
33.33Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
33.33Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
33.33Single9CHXS-Carazolol9CHX-β2-S-Carazolol
33.33Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
33.33Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
33.33Consensus5ht2_onOrthosteric Ligand5ht2b_on
33.33Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
33.33Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
33.33Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
33.33Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
33.33Consensusalpha2_onOrthosteric Ligandalpha2b_on
33.33Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
33.33Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
33.33Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
33.33Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
33.33Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusblt_onOrthosteric Ligandblt1_on
33.33Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
33.33Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
33.33Consensusdopamine_offOrthosteric Ligandd2_off d3_off
33.33Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
33.33Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
33.33Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
33.33Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
33.33Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
33.33Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
33.33Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
33.33Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
33.33Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
33.33Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
33.33Consensushistamine_offOrthosteric Ligandh1_off
33.33Consensusleukotriene_onOrthosteric Ligandblt_on
33.33Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
33.33Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
33.33Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
33.33Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
33.33Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
32.26Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
32.26Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
32.14Single6IGLIRL16206IGL-ETB-IRL1620
32.14Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
32.00Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
32.00Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
32.00Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
32.00Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
32.00Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
32.00Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
32.00Consensusvasop-oxy_onOrthosteric Ligandv2_on
32.00Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
31.82Single3NY9ICI118-5513NY9-β2-ICI118-551
31.82Single4UG2CGS216804UG2-A2A-CGS21680
31.82Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
31.82Single6PT3DPI-2876PT3-δ-DPI-287
31.82Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
31.82Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
31.82Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
31.82Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
31.82Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
31.82Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
31.82Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
31.58Single2RH1S-Carazolol2RH1-β2-S-Carazolol
31.58Single2YCWS-Carazolol2YCW-β1-S-Carazolol
31.58Single5D6LS-Carazolol5D6L-β2-S-Carazolol
31.58Single5JQHS-Carazolol5JQH-β2-S-Carazolol
31.58Single5TVNLSD5TVN-5-HT2B-LSD
31.58Single5WIUNemonapride5WIU-D4-Nemonapride
31.58Single5WIVNemonapride5WIV-D4-Nemonapride-Na
31.58Single5X7DS-Carazolol5X7D-β2-S-Carazolol-PubChem 129318963
31.58Single5XPRBosentan5XPR-ETB-Bosentan
31.58Single6E67BI1671076E67-β2-BI167107-Gs (fused)
31.58Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
31.58Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
31.58Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
31.58Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
31.58Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
31.58Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
31.58Single7C61Ergotamine7C61-5-HT1B-Ergotamine
31.58Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
31.58Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
31.58Single7LD3Adenosine7LD3-A1-Adenosine-PubChem 25263603-Gi2/β1/γ2
31.58Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
31.58Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
31.58Single7WC6LSD7WC6-5-HT2A-LSD
31.58Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
31.58Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
31.58Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
31.58Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
31.58Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
31.58Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
31.58Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
31.58Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
31.58Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
31.58Single8S4DCMF-0198S4D-Apelin-CMF-019
31.58Single8XYKVUF106618XYK-CXCR3-VUF10661-Go1/β1/γ2
31.58Single8ZMFA1L108ZMF-5-HT2C-A1L10
31.58Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
31.58Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
31.58Single9F34FOB02-04A9F34-D3-FOB02-04A-Go1/β1/γ2
31.58Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
31.58Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
31.58Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
31.58Consensusa3_on_gpOrthosteric Liganda3a_on_gp
31.58Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
31.58Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
31.58Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
31.58Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
31.58Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
31.58Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
31.58Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
31.58Consensusamine_offonOrthosteric Ligandamine_off amine_on
31.58Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
31.58Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
31.58Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
31.58Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
31.58Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
31.58Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
31.58Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
31.58Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
31.58Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.58Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.58Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
31.58Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
31.58Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.58Consensustrace-amine_onOrthosteric Ligandta1_on
31.25Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
31.25Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
31.25Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
31.25Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
31.25Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
31.25Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
31.25Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
31.25Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
31.25Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
31.25Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
31.25Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
31.25Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
31.25Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
31.25Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
31.25Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
31.25Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
31.25Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go1/β1/γ2
31.25Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
31.25Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.25Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.25Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
31.25Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
31.25Single8YN7Immethridine8YN7-H3-Immethridine-Go1/β1/γ2
31.25Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
31.25Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
31.25Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
31.25Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
31.25Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
31.03Single5GLHEndothelin-15GLH-ETB-Endothelin-1
31.03Single6IGKEndothelin-36IGK-ETB-Endothelin-3
30.77Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
30.77Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
30.77Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
30.77Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
30.77Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
30.77Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
30.77Single8ZRTET-18ZRT-ETB-ET-1
30.77Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
30.77Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
30.43Single4XT1Fractalkine4XT1-US28-Fractalkine
30.43Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
30.43Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
30.43Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
30.43Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
30.43Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
30.43Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
30.43Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
30.43Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
30.43Single8WDTphotoNECA8WDT-A2A-photoNECA
30.43Single8WKYPG-9348WKY-MC4-PG-934
30.43Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
30.43Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
30.43Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.43Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.43Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
30.43Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
30.43Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
30.00Single2YDVNECA2YDV-A2A-NECA
30.00Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
30.00Single4UHRCGS216804UHR-A2A-CGS21680
30.00Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
30.00Single5D5AS-Carazolol5D5A-β2-S-Carazolol
30.00Single5D5BS-Carazolol5D5B-β2-S-Carazolol
30.00Single5G53NECA5G53-A2A-NECA-Gs
30.00Single5XRAAM115425XRA-CB1-AM11542
30.00Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
30.00Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
30.00Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
30.00Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
30.00Single6WGTLSD6WGT-5-HT2A-LSD
30.00Single7B6WCyclazosin7B6W-α1b-Cyclazosin
30.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
30.00Single7FEECP559407FEE-CB1-CP55940-ZCZ011
30.00Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
30.00Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
30.00Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
30.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
30.00Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
30.00Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
30.00Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
30.00Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
30.00Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
30.00Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
30.00Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
30.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
30.00Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
30.00Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
30.00Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
30.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
30.00Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
30.00Single8XVLZibotentan8XVL-ETA-Zibotentan
30.00Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
30.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
30.00Single9F33FOB02-04A9F33-D3-FOB02-04A-Go1/β1/γ2
30.00Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
30.00Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
30.00Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
30.00Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
30.00Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
30.00Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
30.00Consensuslpa_onOrthosteric Ligandlpa1_on
30.00Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
30.00Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
30.00Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
30.00Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
30.00Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
29.63Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
29.63Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
29.63Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
29.63Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
29.63Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.63Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
29.63Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
29.41Single4S0VSuvorexant4S0V-OX2-Suvorexant
29.41Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
29.41Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
29.41Single6TPJSuvorexant6TPJ-OX2-Suvorexant
29.41Single7BR3Elagolix7BR3-GnRH1-Elagolix
29.41Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
29.41Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
29.41Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
29.41Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
29.41Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.41Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
29.41Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
29.41Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
29.41Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
29.41Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
29.41Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
29.41Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
29.41Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
29.41Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
29.41Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
29.41Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.41Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
29.41Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
29.41Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
29.41Single8IWESpermidine8IWE-TA9-Spermidine
29.41Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
29.41Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
29.41Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
29.41Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
29.41Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.41Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
29.41Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
29.41Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
29.41Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
29.41Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ
29.41Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
29.41Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
29.41Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
29.41Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
29.41Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
29.41Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.41Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
29.41Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
29.41Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
29.41Consensusalpha2_offOrthosteric Ligandalpha2c_off
29.41Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
29.41Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
29.41Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
29.41Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
29.41Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
29.41Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
29.41Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
29.41Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
29.41Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
29.41Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
29.17Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
29.17Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
29.17Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
29.17Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
29.17Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
29.17Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
29.17Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
29.17Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
29.17Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
29.17Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
29.17Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
29.17Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
29.17Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
29.17Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
29.17Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
29.17Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
29.17Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
29.03Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
29.03Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
29.03Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
28.57Single4AMIBucindolol4AMI-β1-Bucindolol
28.57Single5TZYMK8666; PubChem 1270535975TZY-FFA1-MK8666; PubChem 127053597
28.57Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
28.57Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
28.57Single6KQICP559406KQI-CB1-CP55940-Org27569
28.57Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
28.57Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
28.57Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
28.57Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
28.57Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
28.57Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
28.57Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
28.57Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
28.57Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
28.57Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
28.57Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
28.57Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
28.57Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
28.57Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.57Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
28.57Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
28.57Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
28.57Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
28.57Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
28.57Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
28.57Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
28.57Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
28.57Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
28.57Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
28.57Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
28.57Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
28.57Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.12Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
28.00Single5WF5UK-4320975WF5-A2A-UK-432097
28.00Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
28.00Single6W25SHU91196W25-MC4-SHU9119-Ca
28.00Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
28.00Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
28.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
28.00Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
28.00Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
28.00Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
28.00Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
27.78Single3RZECidoxepin3RZE-H1-Cidoxepin
27.78Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
27.78Single6A94Zotepine6A94-5-HT2A-Zotepine
27.78Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
27.78Single6IQLL7458706IQL-D4-L745870
27.78Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
27.78Single6KUXRS-799486KUX-α2a-RS-79948
27.78Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
27.78Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
27.78Single6TP3Nemorexant6TP3-OX1-Nemorexant
27.78Single6V9SGTPL114036V9S-OX1-GTPL11403
27.78Single6VI4JDTic6VI4-κ-JDTic
27.78Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
27.78Single6ZG9GSK10347026ZG9-M1-GSK1034702
27.78Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
27.78Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
27.78Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
27.78Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
27.78Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
27.78Single7T94Acetylcholine7T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
27.78Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
27.78Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
27.78Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
27.78Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
27.78Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.78Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
27.78Single8IHKAcifran8IHK-HCA3-Acifran
27.78Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
27.78Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
27.78Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
27.78Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
27.78Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.78Single8K5CAcipimox8K5C-HCA2-Acipimox
27.78Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
27.78Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.78Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.78Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
27.78Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
27.78Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
27.78Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.78Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
27.78Single8YN8Proxyfan8YN8-H3-Proxyfan-Go1/β1/γ2
27.78Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
27.78Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
27.78Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
27.78Single9BJKNaloxone9BJK-μ-Naloxone-NAM
27.78Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
27.78Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
27.78Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
27.78Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
27.78Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
27.78Consensusgrh_offOrthosteric Ligandgnrh1_off
27.78Consensushca_onOrthosteric Ligandhca2_on
27.78Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
27.78Consensusopsins_offOrthosteric Ligandrhodopsin_off
27.78Consensussensory_offOrthosteric Ligandopsins_off
27.59Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
27.59Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
27.59Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
27.59Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
27.59Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
27.59Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
27.59Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
27.59Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
27.59Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
27.59Consensusbradykinin_onOrthosteric Ligandbk2_on
27.59Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
27.59Consensusendothelin_onOrthosteric Ligandetb_on eta_on
27.59Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
27.59Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
27.27Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
27.27Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
27.27Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
27.27Single6H7LDobutamine6H7L-β1-Dobutamine
27.27Single6IBLArformoterol6IBL-β1-Arformoterol
27.27Single6K1QIRL25006K1Q-ETB-IRL2500
27.27Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
27.27Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
27.27Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
27.27Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
27.27Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
27.27Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
27.27Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
27.27Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(CtGi1-G13)/β1/γ2
27.27Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
27.27Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
27.27Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
26.92Single6JODAngiotensin II6JOD-AT2-Angiotensin II
26.92Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
26.92Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
26.92Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
26.92Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
26.92Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
26.92Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
26.92Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
26.92Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
26.92Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
26.67Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
26.67Single3OE8IT1t3OE8-CXCR4-IT1t
26.67Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
26.67Single6TQ9SB-4081246TQ9-OX1-SB-408124
26.67Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
26.67Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
26.67Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
26.67Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
26.67Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
26.67Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
26.67Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
26.47Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
26.47Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
26.32Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
26.32Single2Y01Dobutamine2Y01-β1-Dobutamine
26.32Single2Y02Carmoterol2Y02-β1-Carmoterol
26.32Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
26.32Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
26.32Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
26.32Single4DAJTiotropium4DAJ-M3-Tiotropium
26.32Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
26.32Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
26.32Single4YAYZD-71554YAY-AT1-ZD-7155
26.32Single5DHGC-355DHG-NOP-C-35
26.32Single5DHHSB-6121115DHH-NOP-SB-612111
26.32Single5TGZAM65385TGZ-CB1-AM6538
26.32Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
26.32Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
26.32Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
26.32Single6D27CAY104716D27-DP2-CAY10471
26.32Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
26.32Single6GPSMK08126GPS-CCR2-MK0812
26.32Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
26.32Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
26.32Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.32Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
26.32Single7BU7BI1671077BU7-β1-BI167107
26.32Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
26.32Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
26.32Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
26.32Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
26.32Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
26.32Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
26.32Single7YXAONO-54306087YXA-S1P5-ONO-5430608
26.32Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
26.32Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
26.32Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
26.32Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
26.32Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
26.32Single8JJOAlprenolol8JJO-β2-Alprenolol
26.32Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
26.32Single8K5DGSK2560738K5D-HCA2-GSK256073
26.32Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
26.32Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
26.32Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
26.32Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
26.32Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
26.32Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
26.32Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
26.32Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
26.32Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
26.32Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
26.32Consensusa3_onOrthosteric Liganda3a_on
26.32Consensuscck_offOrthosteric Ligandccka_off
26.32Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
26.32Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
26.32Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
26.32Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
26.32Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
26.32Consensushca_on_gpOrthosteric Ligandhca2_on_gp
26.32Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
26.32Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
26.09Single5EE7MK08935EE7-Glucagon-MK0893
26.09Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
26.09Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
26.09Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
26.09Single7XN9L-054,5227XN9-SST2-L-054,522
26.09Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
26.09Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
26.09Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
25.93Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
25.93Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
25.93Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
25.93Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
25.93Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
25.93Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
25.93Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
25.93Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
25.93Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
25.93Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
25.93Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
25.93Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
25.93Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.81Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
25.00Single2Y00Dobutamine2Y00-β1-Dobutamine
25.00Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
25.00Single3OE6IT1t3OE6-CXCR4-IT1t
25.00Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
25.00Single4NTJAZD12834NTJ-P2Y12-AZD1283
25.00Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
25.00Single4XT3Fractalkine4XT3-US28-Fractalkine
25.00Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
25.00Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
25.00Single6D26Fevipiprant6D26-DP2-Fevipiprant
25.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
25.00Single6GPXMK08126GPX-CCR2-MK0812
25.00Single6LUQHaloperidol6LUQ-D2-Haloperidol
25.00Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
25.00Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
25.00Single6PS6Timolol6PS6-β2-Timolol
25.00Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
25.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
25.00Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
25.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
25.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
25.00Single7QA8Peptide7QA8-STE2-Peptide
25.00Single7QA8Peptide7QA8-STE2-Peptide
25.00Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
25.00Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
25.00Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
25.00Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
25.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
25.00Single8IEBA1LYA8IEB-GPR156-A1LYA
25.00Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
25.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
25.00Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
25.00Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
25.00Single8KIGSHU91198KIG-MC3-SHU9119-Ca
25.00Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
25.00Single8U4OCXCL128U4O-CXCR4-CXCL12-Cholesterol-Gi1/β1/γ2
25.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
25.00Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
25.00Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
25.00Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
25.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
25.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
25.00Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
25.00Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
25.00Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
25.00Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
25.00Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
25.00Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
25.00Consensusdp_offOrthosteric Liganddp2_off
25.00Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
25.00Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
25.00Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
25.00Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
25.00Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
25.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
25.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
25.00Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
25.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
25.00Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.14Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
24.14Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
24.14Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
24.14Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
24.14Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
24.14Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
24.14Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
24.14Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
24.14Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
24.00Single3QAKUK-4320973QAK-A2A-UK-432097
24.00Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
24.00Single7CUMPhospholipid7CUM-GABAB1, GABAB2-CGP54626-Phospholipid
24.00Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
24.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
24.00Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
23.81Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
23.81Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
23.81Single5TZRMK86665TZR-FFA1-MK8666
23.81Single6E59L-7607356E59-NK1-L-760735
23.81Single6J20Aprepitant6J20-NK1-Aprepitant
23.81Single6J21Aprepitant6J21-NK1-Aprepitant
23.81Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
23.81Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
23.81Single7TUYGSK682753A7TUY-GPR183-GSK682753A
23.81Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
23.81Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
23.81Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
23.81Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
23.81Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
23.81Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
23.81Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.81Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
23.81Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
23.81Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
23.81Single9GE2ML1849GE2-GPR55-ML184-Cholesterol-chim(CtGi1-G13)/β1/γ2
23.81Consensusa2_onOrthosteric Liganda2b_on
23.81Consensusa2_on_gpOrthosteric Liganda2b_on_gp
23.81Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
23.81Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
23.81Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
23.81Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
23.81Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
23.81Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
23.53Single3OE9IT1t3OE9-CXCR4-IT1t
23.53Single3PBLEticlopride3PBL-D3-Eticlopride
23.53Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
23.53Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
23.53Single6HLLCP999946HLL-NK1-CP99994
23.53Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
23.53Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
23.53Single6TP4ACT-4622066TP4-OX1-ACT-462206
23.53Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
23.53Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
23.53Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
23.53Single7XP6Strychnine7XP6-T2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
23.53Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
23.53Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
23.53Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
23.53Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
23.53Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
23.53Single8K5BNiacin8K5B-HCA2-Niacin
23.53Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
23.53Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.53Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
23.53Single9B9Y7DY9B9Y-CB1-7DY
23.53Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
23.53Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
23.53Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
23.53Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
23.53Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
23.33Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
23.33Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
23.33Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
23.33Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
23.33Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
23.33Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
23.33Single8IY6Endothelin-18IY6-ETB-Endothelin-1
23.33Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
23.08Single3OE0CVX153OE0-CXCR4-CVX15
23.08Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
23.08Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
23.08Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
23.08Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
23.08Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
23.08Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
23.08Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
23.08Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
23.08Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
23.08Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
23.08Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
23.08Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
23.08Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
22.73Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
22.73Single4N4WSANT-14N4W-SMO-SANT-1
22.73Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
22.73Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
22.73Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
22.73Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
22.73Single7K15MKD0467K15-BLT1-MKD046-Na
22.73Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
22.73Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
22.73Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
22.73Single8JWZAB9288JWZ-A2A-AB928-Na
22.73Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
22.73Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
22.73Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
22.73Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
22.73Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
22.58Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
22.58Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
22.58Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
22.58Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
22.58Consensusbombesin_onOrthosteric Ligandbb2_on
22.58Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
22.58Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
22.58Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
22.58Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
22.58Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
22.58Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
22.50Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
22.22Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
22.22Single3ODUIT1t3ODU-CXCR4-IT1t
22.22Single6DS0Ly2660976DS0-5-HT2B-Ly266097
22.22Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
22.22Single6ME2Ramelteon6ME2-MT1-Ramelteon
22.22Single6ME9Ramelteon6ME9-MT2-Ramelteon
22.22Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
22.22Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
22.22Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
22.22Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
22.22Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
22.22Single7F8ULintitript7F8U-CCKA-Lintitript
22.22Single7F8YDevazepide7F8Y-CCKA-Devazepide
22.22Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
22.22Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
22.22Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
22.22Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
22.22Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
22.22Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
22.22Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
22.22Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
22.22Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
22.22Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
22.22Single8GNGIstradefylline8GNG-A2A-Istradefylline
22.22Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
22.22Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
22.22Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
22.22Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
22.22Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
22.22Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
22.22Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
22.22Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
22.22Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8U4PAMD31008U4P-CXCR4-AMD3100-Cholesterol-Gi1/β1/γ2
22.22Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
22.22Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.22Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
22.22Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
22.22Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ22
22.22Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
22.22Consensusangiotensin_offOrthosteric Ligandat1_off
22.22Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.22Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.22Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
21.88Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
21.88Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
21.88Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
21.88Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
21.74Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
21.74Single5CGDHTL142425CGD-mGlu5-HTL14242
21.74Single7EZCUKA7EZC-A2A-UKA
21.74Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
21.74Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
21.74Single8T3OTUG-8918T3O-FFA4-TUG-891-2Y5-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8XVJMacitentan8XVJ-ETA-Macitentan
21.74Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
21.74Consensuschemerin_onOrthosteric Ligandcml1_on
21.74Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Consensusprostanoid_offOrthosteric Ligandep_off dp_off
21.43Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
21.43Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
21.43Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
21.43Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
21.43Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
21.43Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
21.43Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
21.43Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
21.43Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
21.43Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
21.43Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
21.43Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
21.43Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
21.43Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
21.05Single2YDOAdenosine2YDO-A2A-Adenosine
21.05Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
21.05Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
21.05Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
21.05Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
21.05Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
21.05Single6TPKRetosiban6TPK-OT-Retosiban
21.05Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
21.05Single7AROLUF58337ARO-A2A-LUF5833-Na
21.05Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
21.05Single7T32ZM-2413857T32-A2A-ZM-241385
21.05Single7VODCariprazine7VOD-5-HT2A-Cariprazine
21.05Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
21.05Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
21.05Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
21.05Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
21.05Single8K2WAMG4878K2W-CXCR3-AMG487
21.05Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
21.05Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
21.05Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
21.05Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
21.05Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
21.05Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
21.05Single8ZPMAMD0708ZPM-CXCR4-AMD070-Cholesterol
21.05Single8ZPNAMD31008ZPN-CXCR4-AMD3100-Cholesterol
21.05Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
21.05Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Cholesterol-Gi1/β1/γ2
21.05Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
21.05Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
21.05Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
21.05Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
21.05Consensusvasop-oxy_offOrthosteric Ligandot_off
20.83Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
20.83Single5WF6UK-4320975WF6-A2A-UK-432097
20.83Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
20.83Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
20.83Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
20.83Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
20.83Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
20.83Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
20.83Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
20.83Single8IEIA1LYA8IEI-GPR156-A1LYA
20.83Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
20.83Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
20.83Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
20.83Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.83Consensuskisspeptin_onOrthosteric Ligandkiss1_on
20.69Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
20.69Single6FJ3PTH6FJ3-PTH1-PTH
20.69Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
20.69Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
20.69Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
20.69Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
20.69Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
20.69Single7SK3CXCL127SK3-ACKR3-CXCL12
20.69Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
20.69Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
20.69Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
20.69Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
20.69Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
20.59Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
20.00Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
20.00Single5DSGTiotropium5DSG-M4-Tiotropium
20.00Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
20.00Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
20.00Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
20.00Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
20.00Single5UENDU1725UEN-A1-DU172
20.00Single5UIGCmpd-15UIG-A2A-Cmpd-1
20.00Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
20.00Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
20.00Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
20.00Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
20.00Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7F83PF-051904577F83-Ghrelin-PF-05190457
20.00Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
20.00Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
20.00Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
20.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
20.00Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
20.00Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
20.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
20.00Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
20.00Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
20.00Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7WC4Serotonin7WC4-5-HT2A-Serotonin
20.00Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
20.00Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
20.00Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
20.00Single8CU6LJ-45178CU6-A2A-LJ-4517
20.00Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
20.00Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8IEIA1LYA8IEI-GPR156-A1LYA
20.00Single8IEPA1LYA8IEP-GPR156-A1LYA
20.00Single8IEPA1LYA8IEP-GPR156-A1LYA
20.00Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
20.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
20.00Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
20.00Single8RLNLUF58348RLN-A2A-LUF5834
20.00Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
20.00Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
20.00Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
20.00Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
20.00Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
20.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
20.00Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
20.00Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.00Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9IYAONO-97105319IYA-GPR55-ONO-9710531
20.00Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
20.00Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
20.00Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.00Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.00Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
20.00Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
20.00Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
19.35Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
19.35Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
19.35Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
19.35Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
19.35Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
19.23Single6HLOAprepitant6HLO-NK1-Aprepitant
19.23Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
19.23Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
19.23Single7SK5CXCL127SK5-ACKR3-CXCL12
19.23Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
19.23Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
19.23Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single8IEBA1LYA8IEB-GPR156-A1LYA
19.23Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.23Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
19.23Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
19.05Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
19.05Single5CGCHTL142425CGC-mGlu5-HTL14242
19.05Single5N2RPSB-365N2R-A2A-PSB-36-Na
19.05Single5N2SPSB365N2S-A1-PSB36
19.05Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
19.05Single5T1APubChem 68764898; PubChem 120931705T1A-CCR2-PubChem 68764898; PubChem 12093170
19.05Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
19.05Single6HLPNetupitant6HLP-NK1-Netupitant
19.05Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
19.05Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
19.05Single6W2XPubChem 237279706W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
19.05Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
19.05Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
19.05Single7SINNPS-21437SIN-CaS-NPS-2143
19.05Single7SINNPS-21437SIN-CaS-NPS-2143
19.05Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
19.05Single7W41PD1762527W41-BB2-PD176252
19.05Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.05Single8WGBW9R8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
19.05Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
19.05Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
19.05Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
19.05Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
19.05Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
19.05Consensusadenosine_offOrthosteric Liganda1_off a2_off
19.05Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
19.05Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
19.05Consensusblt_offOrthosteric Ligandblt1_off
19.05Consensusbombesin_offOrthosteric Ligandbb2_off
19.05Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
19.05Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
19.05Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
19.05Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
18.75Single3RFMCaffeine3RFM-A2A-Caffeine
18.75Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
18.75Single7RBTTirzepatide7RBT-GIP-Tirzepatide-PubChem 163183774-chim(NtGi1-Gs)/β1/γ2
18.75Single8A2OTheophylline8A2O-A2A-Theophylline-Na
18.75Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
18.75Consensussensory_onOrthosteric Ligandopsins_on
18.52Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
18.52Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
18.52Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
18.52Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
18.42Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
18.18Single6OS1TRV0266OS1-AT1-TRV026
18.18Single7R0CAVP7R0C-V2-AVP-Arrestin2
18.18Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
18.18Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
18.18Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
18.18Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
18.18Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8JD5BQI; HZE; PEF8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
18.18Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
18.18Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
18.18Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
18.18Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
18.18Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
18.18Single9AUCCalcitonin gene-related peptide-19AUC-CT-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
18.18Single9BJKNAM9BJK-μ-Naloxone-NAM
18.18Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
18.18Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
18.18Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
18.18Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
18.18Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
18.18Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
18.18Consensusrelaxin_onOrthosteric Ligandrxfp4_on
18.18Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
18.18Consensustachykinin_offOrthosteric Ligandnk1_off
17.95Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
17.86Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
17.86Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
17.86Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
17.86Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
17.86Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
17.86Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
17.86Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
17.65Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
17.65Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
17.65Single6ME5Agomelatine6ME5-MT1-Agomelatine
17.65Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
17.65Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
17.65Single7WC5Psilocin7WC5-5-HT2A-Psilocin
17.65Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
17.65Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
17.65Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
17.65Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
17.65Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
17.65Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
17.65Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
17.65Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
17.65Consensusgi_sensoryOrthosteric Ligandgi_opsins
17.65Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
17.65Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
17.39Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
17.39Single4PY02MeSATP4PY0-P2Y12-2MeSATP
17.39Single5X33BIIL2605X33-BLT1-BIIL260
17.39Single6OS2TRV0266OS2-AT1-TRV026
17.39Single6W2YPubChem 237279706W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
17.39Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
17.39Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
17.39Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
17.39Single8JWY2-1188JWY-A2A-2-118
17.39Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
17.39Single8ZPLHF511168ZPL-CXCR4-HF51116-Cholesterol
17.39Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
17.39Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
17.39Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
17.24Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
17.24Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
17.24Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.24Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
17.14Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
16.67Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
16.67Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
16.67Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
16.67Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
16.67Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
16.67Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
16.67Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
16.67Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
16.67Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
16.67Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
16.67Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
16.67Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
16.67Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
16.67Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
16.67Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
16.67Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
16.67Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab-Cholesterol
16.67Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
16.67Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
16.67Consensuscck_onOrthosteric Ligandccka_on cckb_on
16.67Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
16.67Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
16.67Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
16.13Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
16.13Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
16.00Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
16.00Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
16.00Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
16.00Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
16.00Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
16.00Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
16.00Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
15.79Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
15.79Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
15.79Single3PWHZM-2413853PWH-A2A-ZM-241385
15.79Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
15.79Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
15.79Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
15.79Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
15.79Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
15.79Single5U09Taranabant5U09-CB1-Taranabant
15.79Single5ZKQABT-4915ZKQ-PAF-ABT-491
15.79Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
15.79Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
15.79Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
15.79Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
15.79Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
15.79Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
15.79Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
15.79Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
15.79Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
15.79Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
15.79Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
15.79Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
15.79Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
15.79Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
15.79Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
15.79Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.79Single9BA0A1AKN9BA0-CB1-A1AKN
15.79Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
15.79Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
15.79Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
15.62Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
15.62Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
15.38Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
15.38Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
15.38Single7F8XNN90567F8X-CCKA-NN9056
15.38Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
15.38Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
15.38Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Consensussomatostatin_offOrthosteric Ligandsst2_off
15.00Single3REYXAC3REY-A2A-XAC
15.00Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
15.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
15.00Single5IUBQ274563445IUB-A2A-Q27456344-Na
15.00Single5JTBZM-2413855JTB-A2A-ZM-241385
15.00Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
15.00Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
15.00Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
15.00Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
15.00Single6AQFZM-2413856AQF-A2A-ZM-241385
15.00Single6FFIMMPEP6FFI-mGlu5-MMPEP
15.00Single6MH8ZM-2413856MH8-A2A-ZM-241385
15.00Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
15.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
15.00Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
15.00Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
15.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
15.00Single7T94PubChem 576644067T94-M2-Acetylcholine-PubChem 57664406-chim(NtGi1-Go)/β1/γ2
15.00Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
15.00Consensusa2_offOrthosteric Liganda2a_off
15.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
15.00Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
15.00Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.81Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
14.81Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
14.81Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
14.81Single7XNACYN1548067XNA-SST2-CYN154806
14.81Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
14.81Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
14.81Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
14.81Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
14.71Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
14.29Single3EMLZM-2413853EML-A2A-ZM-241385
14.29Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
14.29Single5IU8Q274563475IU8-A2A-Q27456347-Na
14.29Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
14.29Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
14.29Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
14.29Single6FFHFenobam6FFH-mGlu5-Fenobam
14.29Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
14.29Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
14.29Single6S0LZM-2413856S0L-A2A-ZM-241385
14.29Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
14.29Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
14.29Single7PYRPSB-21157PYR-A2A-PSB-2115
14.29Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
14.29Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
14.29Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.29Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
14.29Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
14.29Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
14.29Single9B9ZA1AKO9B9Z-CB1-A1AKO
14.29Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
14.29Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
14.29Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.29Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.29Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
14.29Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
14.29Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
13.89Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.89Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
13.89Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
13.79Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
13.79Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.79Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
13.64Single5IUAQ274563485IUA-A2A-Q27456348-Na
13.64Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
13.64Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
13.64Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
13.64Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
13.64Single6S0QZM-2413856S0Q-A2A-ZM-241385
13.64Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
13.64Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
13.64Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
13.64Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
13.64Single8GNEKW-63568GNE-A2A-KW-6356-Na
13.64Single8QOTNanobody-E8QOT-μ-Nanobody-E
13.64Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
13.64Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
13.64Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
13.64Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
13.64Consensusep_offOrthosteric Ligandep4_off
13.33Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
13.33Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
13.33Single5MZPCaffeine5MZP-A2A-Caffeine-Na
13.33Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
13.04Single4BV0Neurotensin4BV0-NTS1-Neurotensin
13.04Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
13.04Single7F1TMIP-1a7F1T-CCR5-MIP-1a
13.04Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
13.04Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
13.04Single7P2L4YI7P2L-mGlu5-4YI
13.04Single7PX4PSB-21137PX4-A2A-PSB-2113
13.04Single7T9NPubChem 6440787T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
13.04Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
13.04Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
13.04Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
13.04Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
13.04Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
13.04Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.04Consensusneurotensin_onOrthosteric Ligandnts1_on
13.04Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
13.04Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.90Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
12.50Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
12.50Single4XEENeurotensin4XEE-NTS1-Neurotensin
12.50Single4XESNeurotensin4XES-NTS1-Neurotensin
12.50Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
12.50Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
12.50Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
12.50Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
12.50Single6YVRNTS8-136YVR-NTS1-NTS8-13
12.50Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.50Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
12.50Single7V68PubChem 576644067V68-M4-Iperoxo-PubChem 57664406-Gi1/β1/γ2
12.50Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
12.50Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
12.50Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
12.50Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
12.50Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-PubChem 118610427; GDP; Mg-Gq; GRK2
12.50Single8PWNTheophylline8PWN-A2A-Theophylline
12.50Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
12.50Single8XJNCloprosetnol8XJN-TP-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
12.50Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
12.50Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.50Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
12.50Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
12.00Single4BUONeurotensin4BUO-NTS1-Neurotensin
12.00Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
12.00Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
12.00Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
12.00Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
12.00Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
12.00Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
12.00Single8JPFNeurotensin8JPF-NTS1-Neurotensin-PubChem 118610427
12.00Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
12.00Single8XJOU466198XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single8XVUCXCL28XVU-CXCR2-CXCL2
12.00Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
12.00Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
12.00Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
12.00Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
12.00Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
12.00Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
12.00Consensustp_onOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Consensustp_on_gpOrthosteric Ligand8XJO-TP-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
11.76Consensusp2y_offOrthosteric Ligandp2y1_off
11.54Single6KNMJN241-96KNM-Apelin-JN241-9
11.54Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
11.54Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
11.54Single8XQJJN2418XQJ-Apelin-JN241
11.54Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
11.54Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
11.54Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
11.54Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
11.54Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
11.11Single3UZAGTPL92363UZA-A2A-GTPL9236
11.11Single4XNWMRS25004XNW-P2Y1-MRS2500
11.11Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
11.11Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
11.11Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
11.11Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
11.11Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
11.11Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
11.11Single8XWNCXCL88XWN-CXCR2-CXCL8
11.11Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
10.71Single7SHEPI; PE7SHE-GPR158-PI; PE
10.71Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
10.71Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
10.53Single6LI0C176LI0-GPR52-C17
10.53Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
10.53Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
10.34Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
10.00Single4BWBNeurotensin4BWB-NTS1-Neurotensin
10.00Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
10.00Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
10.00Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
10.00Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
10.00Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
10.00Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.00Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
10.00Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
10.00Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.68Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
9.68Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
9.68Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
9.52Single5UVIZM-2413855UVI-A2A-ZM-241385
9.52Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
9.52Single6ZINSR486926ZIN-NTS1-SR48692
9.52Single7UTZPubChem 6440787UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
9.52Single8IYXYL-3658IYX-GPR34-YL-365
9.52Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
9.09Single4QIMANTA XV4QIM-SMO-ANTA XV
9.09Single5T04Neurotensin5T04-NTS1-Neurotensin
9.09Single6IIVDaltroban6IIV-TP-Daltroban
9.09Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
9.09Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
9.09Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
9.09Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
9.09Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
9.09Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
9.09Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
8.70Single4JKVTaladegib4JKV-SMO-Taladegib
8.70Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
8.70Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
8.70Single6Z4SSR486926Z4S-NTS1-SR48692
8.70Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
8.70Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
8.70Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
8.70Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
8.70Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
8.70Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single5V56TC1145V56-SMO-TC114
8.33Single5V57TC1145V57-SMO-TC114
8.33Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
8.33Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
8.33Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
8.33Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Cholesterol-Gi1/β1/γ1
8.33Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
8.00Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
8.00Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
8.00Single6IIURamatroban6IIU-TP-Ramatroban
8.00Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
8.00Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
8.00Single8XQJJN2418XQJ-Apelin-JN241
8.00Single8XWACXCL18XWA-CXCR2-CXCL1
8.00Single8XWMCXCL68XWM-CXCR2-CXCL6
8.00Single8XWSCXCL58XWS-CXCR2-CXCL5
8.00Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
7.69Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
7.69Single6D35Cholesterol6D35-SMO-Cholesterol
7.69Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
7.69Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
7.69Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
7.69Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
7.69Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
7.69Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042-PubChem 23727970
7.69Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
7.69Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042-PubChem 23727970
7.69Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-PubChem 7023848
7.69Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
7.69Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626-Phospholipid
7.69Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.69Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.69Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.69Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
7.69Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
7.69Single7DTTCa7DTT-CaS-Ca-Ca
7.69Single7DTTCa7DTT-CaS-Ca-Ca
7.69Single7DTUTryptophan7DTU-CaS-Tryptophan
7.69Single7DTUTryptophan7DTU-CaS-Tryptophan
7.69Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
7.69Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
7.69Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
7.69Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
7.69Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.69Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.69Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.69Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.69Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
7.69Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
7.69Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
7.69Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
7.69Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
7.69Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
7.69Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
7.69Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
7.69Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
7.69Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
7.69Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
7.69Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
7.69Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
7.69Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
7.69Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
7.69Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.69Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.69Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.69Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.69Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.69Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.69Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
7.69Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
7.69Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
7.69Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
7.69Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
7.69Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
7.69Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
7.69Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.69Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.69Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.69Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.69Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.69Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.69Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.69Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
7.69Single7T9NM22 Fab7T9N-TSH-M22 Fab-PubChem 644078-Gs/β1/γ2
7.69Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
7.69Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
7.69Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
7.69Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
7.69Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
7.69Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
7.69Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
7.69Single7XW7K1-707XW7-TSH-K1-70
7.69Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-PubChem 118610427-chim(NtGi1-Go)/β1/γ2
7.69Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
7.69Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
7.69Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
7.69Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
7.69Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
7.69Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
7.69Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
7.69Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
7.69Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
7.69Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
7.69Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
7.69Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
7.69Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
7.69Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
7.69Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
7.69Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
7.69Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
7.69Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
7.69Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-HZR; PEF-Gi1/β1/γ2
7.69Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
7.69Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
7.69Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
7.69Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-BQI; HZE; PEF-Gi1/β1/γ2
7.69Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
7.69Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-N-(3-chlorophenyl)pyridine-2-carboxamide-Gi3/β1/γ2
7.69Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
7.69Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
7.69Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW
7.69Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
7.69Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-chim(NtGi1-Gq)/β1/γ2
7.69Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
7.69Single8SZHCa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZH-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi1/β1/γ2
7.69Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
7.69Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
7.69Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
7.69Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
7.69Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
7.69Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
7.69Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
7.69Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
7.69Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
7.69Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
7.69Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
7.69Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
7.69Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
7.69Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
7.69Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
7.69Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
7.69Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
7.69Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
7.69Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
7.69Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
7.69Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-W9R-Gi3/β1/γ2
7.69Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
7.69Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
7.69Single8WGDWAG/WA68WGD-mGlu4; mGlu2-WAG/WA6
7.69Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
7.69Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
7.69Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8WVXNorrin8WVX-LGR4-Norrin
7.69Single8WVYNorrin8WVY-LGR4-Norrin
7.69Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
7.69Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
7.69Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
7.69Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
7.69Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
7.69Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
7.69Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
7.69Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
7.69Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
7.69Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
7.69Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
7.69Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
7.69Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
7.69Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
7.69Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
7.69Single8XWFCXCL38XWF-CXCR2-CXCL3
7.69Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
7.69Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
7.69Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
7.69Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.69Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.69Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.69Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.69Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.69Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.69Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.69Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.69Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.69Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.69Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
7.69Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
7.69Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
7.69Single9C2FCa; Ca; Tryptophan; '6218; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '6218; PO4
7.69Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
7.69Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
7.69Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
7.69Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
7.41Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
7.41Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
7.14Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
7.14Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
7.14Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
7.14Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
7.14Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
7.14Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
7.14Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
7.14Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
7.14Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.14Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
7.14Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
7.14Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.14Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
7.14Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.14Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
6.90Single7SHFPI; PE7SHF-GPR158-PI; PE-B5; RGS7
6.67Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
6.67Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
6.67Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
6.45Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
6.25Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
6.25Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
6.25Single7UTZTR14027UTZ-TSH-TR1402-PubChem 644078-Gs/β1/γ2
6.25Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
6.25Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
5.88Single5L7DCholesterol5L7D-SMO-Cholesterol
5.88Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
5.88Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
5.88Single8HS2Fab0468HS2-GPR20-Fab046
5.88Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
5.88Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
5.56Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
5.56Single6XBM25(S)-Epoxycholesterol6XBM-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
5.56Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Cholesterol-Gi1/β1/γ2
5.26Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.26Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
5.26Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
5.26Single8JPSCCL78JPS-ACKR1-CCL7
5.26Single8ZPLCholesterol8ZPL-CXCR4-HF51116-Cholesterol
5.26Single8ZPMCholesterol8ZPM-CXCR4-AMD070-Cholesterol
5.00Single4O9RCyclopamine4O9R-SMO-Cyclopamine
5.00Single5L7IVismodegib5L7I-SMO-Vismodegib
5.00Single7UL2SR486927UL2-NTS1-SR48692-Na
5.00Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
5.00Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
5.00Single8HNNSCH5467388HNN-CXCR3-SCH546738
5.00Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
5.00Consensusgq_nucleotideOrthosteric Ligandgq_p2y
5.00Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
5.00Consensusneurotensin_offOrthosteric Ligandnts1_off
5.00Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
4.76Single4K5YCP-3763954K5Y-CRF1-CP-376395
4.76Single4QINSAG1.54QIN-SMO-SAG1.5
4.76Single6C1QNDT95137276C1Q-C5a1-PMX53-NDT9513727
4.76Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
4.76Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
4.76Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
4.76Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
4.76Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
4.55Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
4.55Single7VV6C48/807VV6-MRGPRX2-C48/80
4.55Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
4.55Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
4.35Single4Z9GCP-3763954Z9G-CRF1-CP-376395
4.35Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.35Single8GTIBMK-C2058GTI-CRF1-BMK-C205
4.35Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
4.35Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
4.17Single8GTGBMK-I1528GTG-CRF1-BMK-I152
4.17Single8SZICa; Ca; Tryptophan; Cinacalcet; PO4; PCW8SZI-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; PCW-Gi3/β1/γ2
4.17Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
4.17Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
3.85Single7SHEPI; PE7SHE-GPR158-PI; PE
3.85Single8GTMBMK-C2038GTM-CRF1-BMK-C203
3.70Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
3.45Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
3.45Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
3.45Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
3.23Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
3.23Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-Cholesterol-ZNRF3
3.12Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.86Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
7EW1 7EW1-S1P5-Siponimod-Gi1/β1/γ2
Net Summary
Imin 2.39
Number of Linked Nodes 828
Number of Links 1005
Number of Hubs 157
Number of Links mediated by Hubs 571
Number of Communities 32
Number of Nodes involved in Communities 247
Number of Links involved in Communities 350
Path Summary
Number Of Nodes in MetaPath 107
Number Of Links MetaPath 106
Number of Shortest Paths 3231581
Length Of Smallest Path 3
Average Path Length 48.1635
Length of Longest Path 85
Minimum Path Strength 1.13
Average Path Strength 5.19913
Maximum Path Strength 16.885
Minimum Path Correlation 0.7
Average Path Correlation 0.990974
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.63934
Average % Of Corr. Nodes 32.9263
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 48.3885
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following differences:
Id1st Network2nd Network
s1p5_off_on_gps1p5_on_gps1p5_off
This network is also present in following consensuses:
IdComponents
s1p_on_gps1p1_on_gp
s1p3_on_gp
s1p5_on_gp



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