Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 1.65471502
2G.HN.48 1.57647403
3G.S1.02 5.2599485
4G.S1.06 5.89367448
5G.H1.07 2.22082409
6G.S2.08 8.72506485
7G.S3.01 3.95633584
8G.S3.03 7.36805587
9G.S3.04 5.83922516
10G.S3.06 5.98936615
11G.S3.07 4.73747449
12G.s3h2.03 4.28912419
13G.H2.02 4.27489418
14G.H2.03 4.12838419
15G.H2.04 4.31205409
16G.H2.06 4.70533719
17G.H2.07 4.49456719
18G.H2.09 5.17168418
19G.h2s4.01 6.18151519
20G.S4.02 4.55144418
21G.S4.03 3.56055547
22G.S4.04 5.70228409
23G.s4h3.04 5.36023698
24G.s4h3.10 0.541955409
25G.H3.01 6.175125169
26G.H3.09 6.66053409
27G.H3.15 4.89083418
28G.H3.17 7.04108615
29G.H3.18 6.98769419
30G.S5.03 3.40433548
31G.S5.05 3.78228749
32G.S5.07 3.61128449
33G.HG.03 2.55864596
34G.HG.04 5.01776599
35G.HG.07 5.2228499
36G.hgh4.02 3.871195187
37G.hgh4.05 7.24582407
38G.H4.03 4.61449404
39G.H4.10 6.889155186
40G.H4.15 3.82226508
41G.h4s6.02 6.121784138
42G.S6.02 5.71864647
43G.H5.03 4.99043448
44G.H5.08 7.26034488
45b.1x4 1.61244408
46b.1x15 2.98676417
47b.h2x5 3.28107405
48b.lhb1x3 2.66801502
49b.lhb1x6 4.225384123
50b.b1x3 3.18444557
51b.b1x4 3.29343457
52b.l1x3 8.748295109
53b.b2x1 6.03549518
54b.b2x5 6.22815657
55b.b3x3 2.77704408
56b.l3x2 4.89229409
57b.b4x2 5.55532408
58b.b4x3 4.10734477
59b.b4x6 8.595457109
60b.l4x2 8.96264454
61b.b5x2 5.38269407
62b.b5x3 5.877327109
63b.b5x5 4.80373405
64b.b5x7 5.35404477
65b.l5x1 4.31768578
66b.l5x5 7.51439619
67b.b6x5 3.70345606
68b.l6x5 6.288144144
69b.b7x1 5.631245144
70b.b8x4 4.57242776
71b.b9x3 4.78845476
72b.l9x3 6.71296619
73b.l9x6 4.62735818
74b.b10x5 4.05428509
75b.l11x2 6.75335519
76b.b12x6 7.8494718
77b.b13x7 7.77227567
78b.l13x3 7.84681669
79b.l13x6 4.85864519
80b.l13x7 4.15268569
81b.b15x1 6.87474469
82b.b15x2 6.03623416
83b.l15x1 4.933517
84b.l15x2 5.0076569
85b.b16x4 8.80836566
86b.b16x5 5.00322515
87b.b16x6 8.62144668
88b.b16x7 6.84407419
89b.l16x3 6.30864413
90b.b17x4 4.88218415
91b.b17x5 6.99727517
92b.b17x7 8.56202418
93b.l17x3 7.64908719
94b.l17x6 6.0259419
95b.b18x3 4.54313418
96b.l18x1 6.12155736
97b.l18x2 5.17891437
98b.b19x2 5.33549716
99b.b19x4 5.19195518
100b.l19x2 5.54876519
101b.b20x2 5.63835416
102b.b20x4 8.00225618
103b.b20x6 6.62651616
104b.b20x7 4.24628409
105b.l20x2 6.48756409
106b.b21x1 9.75471417
107b.b21x5 4.94877434
108b.b21x7 3.96554735
109b.l21x2 4.80454404
110b.b22x5 5.16563537
111b.l22x5 6.70915129
112b.b23x1 3.93737405
113b.b23x6 6.0153737
114b.b24x4 7.03872436
115b.b24x6 4.98149438
116b.b24x7 6.890344129
117b.l24x3 5.014864125
118b.b25x3 6.04984435
119b.l25x3 8.522285119
120b.l27x1 9.60584719
121b.l27x2 7.667824119
122b.b28x3 3.717195107
123b.b28x4 4.854425116
124b.b28x6 9.182884119
125g.h1x11 2.46407409
126g.l1x4 4.00616718
127g.h2x11 7.98962436
128g.ctx3 6.42214509
129g.ctx6 3.182186126
130g.ctx14 4.55745559
131g.ctx15 5.98308459
132g.ctx16 4.49266858
133Lig 6.495212420
1341x35 3.34691526
1351x36 3.95622405
1361x39 4.13276527
1371x43 3.56032406
1382x42 5.44068507
1392x44 4.78229406
1402x46 3.68046529
1412x50 4.65882529
1422x64 4.58335525
143E1x50 6.94435728
144E1x52 8.30181526
1453x34 4.924235155
1463x35 4.63189408
1473x37 4.16029406
1483x38 5.844444157
1493x51 7.318464238
150I2x57 5.332446207
1514x50 8.665624159
152E2 10.23591423
153E2x50 6.43051429
1545x40 4.1299424
1555x44 5.95264426
1565x47 4.88749528
1575x58 5.497116229
158I3 7.68027643
1596x30 2.78306406
1606x48 5.03181628
1616x52 4.78928527
1626x58 3.66755423
163E3 4.17332722
1647x34 5.70474424
1657x35 6.55495424
1667x42 7.30526427
1677x45 6.64466429
1687x47 2.13138408
1697x49 5.23202429
1707x53 4.33367629
1718x50 3.316508
172g.h1x1 1.06941400
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b4x6 b.b5x3 17.313311.3844YesYes1099
2b.b3x2 b.b4x6 21.7973.4391NoYes059
3b.b2x5 b.b3x2 22.07948.31481YesNo075
4b.b2x3 b.b2x5 79.32615.54654NoYes567
5b.b26x2 b.b2x3 79.8754.73538NoNo076
6b.b26x1 b.b26x2 80.14563.27462NoNo097
7b.b26x1 b.l27x1 80.41655.37756NoYes099
8G.H2.09 b.l27x1 35.71446.0107YesYes189
9G.H2.09 G.H2.10 44.84322.84385YesNo187
10G.H2.10 b.l5x5 80.9843.05378NoYes179
11G.h2s4.01 b.l5x5 53.293911.7819YesYes199
12G.H2.07 G.h2s4.01 53.76683.5075YesYes199
13G.H2.04 G.H2.07 96.46955.09615YesYes099
14G.H2.04 G.H3.08 1003.64962YesNo099
15G.H3.08 G.S4.04 99.95486.09019NoYes099
16G.S4.04 G.s1h1.01 94.43932.56929YesNo099
17G.H1.01 G.s1h1.01 94.38673.16449NoNo099
18G.H1.01 G.S1.06 94.08427.82731NoYes498
19G.S1.06 G.S3.05 31.44126.87859YesNo087
20G.S1.04 G.S3.05 31.08332.86276NoNo077
21G.S1.04 G.S3.03 62.09183.4275NoYes077
22G.H5.11 G.S3.03 58.87366.14263NoYes887
23G.H5.11 G.H5.15 58.89482.81417NoNo087
24G.H5.15 G.H5.19 56.66953.17609NoNo078
25G.H5.19 I2x57 56.33993.03897NoYes2087
263x49 I2x57 55.080411.0492NoYes087
27b.b2x1 b.l27x1 71.41864.33987YesYes189
28G.H2.10 b.b2x1 36.07244.775NoYes178
29b.b2x1 b.l3x1 36.072710.3205YesNo089
30b.l3x1 b.l5x5 36.15418.82647NoYes099
31b.l5x5 b.l7x2 63.48976.59878YesNo199
32G.H2.07 b.l7x2 53.24222.7607YesNo199
33G.S1.06 G.S4.03 62.70472.82288YesYes487
34G.S1.04 G.S4.03 31.18934.56603NoYes077
35G.H4.15 G.S4.06 10.53375.51115YesNo087
36G.S4.04 G.S4.06 10.75093.23301YesNo097
37G.H2.07 b.l9x6 30.22272.76263YesYes198
38G.s3h2.03 b.l7x2 10.26263.9991YesNo199
39G.s3h2.03 b.l9x6 10.09793.09186YesYes198
40G.H2.06 b.l9x6 32.93513.53423YesYes198
41G.H2.06 b.l17x6 32.12736.96603YesYes199
42G.S4.03 G.S5.03 29.61184.92462YesYes478
43b.l25x6 b.l27x1 26.460220.0479NoYes189
44G.S5.03 G.S6.02 29.59412.73718YesYes487
45G.S6.02 I3 29.038510.9322YesYes473
465x65 I3 26.97654.7216NoYes083
472x42 3x49 53.97537.21679YesNo078
483x50 5x58 25.6277.2291NoYes099
495x58 5x61 26.15493.3216YesNo098
503x54 5x61 26.23037.1009NoNo088
513x54 5x65 26.30643.11942NoNo088
52b.l17x5 b.l17x6 32.19262.80064NoYes169
53b.l17x5 b.l19x2 32.07033.25442NoYes169
54b.l17x3 b.l19x2 30.67393.82038YesYes199
55b.b20x6 b.l17x3 19.98014.36904YesYes169
56b.b17x7 b.b20x6 13.662710.5175YesYes186
57b.b17x7 b.b21x1 10.72557.73731YesYes187
58b.l23x1 b.l25x6 38.04120.3032NoNo068
59b.l21x7 b.l23x1 37.2354.28679NoNo056
60b.b23x6 b.l21x7 35.19913.56481YesNo375
61b.b23x6 b.b24x6 29.92976.87154YesYes378
62b.b21x7 b.b24x6 29.184.30872YesYes358
63b.l2x5 b.l4x2 29.109815.0568NoYes054
64b.l26x5 g.ctx4 22.28795.41833NoNo057
65g.ctx3 g.ctx4 21.73714.80936YesNo097
66b.b21x5 b.h2x1 11.1436.96673YesNo045
67b.b21x5 b.b21x7 12.69457.41494YesYes345
68b.l2x3 b.l2x5 28.19863.12776NoNo085
69b.b3x1 b.l2x3 27.91644.90885NoNo058
70b.b3x1 b.b6x5 26.21133.98904NoYes056
71b.b2x4 b.b6x5 16.12393.82897NoYes066
72b.b10x4 b.b2x4 15.83757.44436NoNo066
73b.b2x5 b.l26x1 23.135912.0352YesNo577
74b.l26x1 b.l26x3 22.00935.80045NoNo577
75b.l26x3 b.l26x5 21.76666.99288NoNo075
76b.l4x1 b.l4x2 28.90043.51532NoYes554
77b.b10x2 b.b10x4 11.52175.76603NoNo066
78b.b10x2 b.b14x3 10.66044.08962NoNo065
79b.b21x7 b.b23x2 10.8433.75942YesNo356
80b.b22x5 b.b23x2 10.00938.25917YesNo376
812x42 3x45 44.25853.41808YesNo077
823x45 4x49 43.92963.45609NoNo077
833x41 4x49 43.76543.09026NoNo057
843x37 3x41 43.4382.82596YesNo065
853x36 3x37 19.64552.77487NoYes076
863x36 Lig 29.60788.55199NoYes270
873x50 7x53 25.4033.54917NoYes099
887x49 7x53 24.39423.56122YesYes299
897x45 7x49 24.21317.53641YesYes299
906x48 7x45 22.70998.475YesYes289
913x36 6x48 10.27115.80314NoYes278
923x37 5x43 22.84023.51481YesNo065
935x43 Lig 19.46724.08603NoYes250
946x48 6x52 11.87874.17378YesYes287
956x52 Lig 10.23243.76141YesYes270
967x38 Lig 18.07675.18737NoYes250
971x39 7x38 17.56564.53756YesNo275
98b.b2x5 b.l4x1 33.90474.67256YesNo575
99G.H3.17 b.l25x6 11.98574.75YesNo158
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
3x33Lig9.874042NoYes4010
3x36Lig8.551992NoYes7010
5x40Lig3.560582YesYes4010
5x43Lig4.086032NoYes5010
6x52Lig3.761412YesYes7010
6x55Lig6.05432NoYes5010
6x51Lig2.866150NoYes6010
7x34Lig5.413592YesYes4010
7x38Lig5.187372NoYes5010
2x60Lig11.97852NoYes6010
2x63Lig6.240392NoYes4010
E1x50Lig2.627372YesYes8010
3x28Lig3.020962NoYes5010
3x29Lig5.549552NoYes4010
3x32Lig7.369872NoYes5010
E2x50Lig3.793332YesYes9010
1x392x572.622952YesNo7722
1x397x384.537562YesNo7521
2x562x603.452560NoNo6621
2x563x326.031280NoNo6521
2x577x4211.07780NoYes7721
2x59E1x502.618782NoYes6821
2x59E1x528.553722NoYes6622
2x593x285.451732NoNo6521
2x607x427.652762NoYes6711
2x63E1x505.873852NoYes4811
E1x49E25.004492NoYes5321
E1x50E1x5218.23982YesYes8612
3x25E1x505.264872NoYes9821
E1x50E2x5012.02222YesYes8911
3x22E28.062632NoYes3321
3x25E23.4552NoYes9321
3x25E2x507.1752NoYes9921
3x29E2x502.731542NoYes4911
3x29E2x522.81412NoNo4412
3x327x426.877692NoYes5711
3x334x605.060192NoNo4512
3x33E2x522.891352NoNo4412
3x363x372.774872NoYes7612
3x366x485.803142NoYes7812
3x375x433.514810YesNo6521
4x60E2x522.806472NoNo5422
4x63E23.562050NoYes5321
E2E238.56972YesYes3311
E2E2x514.296732YesNo3412
5x32E23.499870NoYes3321
5x35E26.52842NoYes1321
5x36E28.420062NoYes4321
5x39E23.447182NoYes6321
5x31E23.996472NoYes4321
5x315x352.600642NoNo4122
5x365x405.297122NoYes4421
5x395x432.903972NoNo6521
5x406x594.273782YesNo4412
5x445x475.881152YesYes6822
5x446x526.603532YesYes6721
5x4616x523.193590NoYes5721
5x476x526.21412YesYes8721
6x486x524.173782YesYes8721
6x547x349.29072NoYes5421
6x587x342.677122YesYes3411
E3E35.464742YesYes2211
7x30E34.217122NoYes3221
7x347x385.437562YesNo4511
7x42Lig3.612822YesYes7010
5x406x553.388142YesNo4511
6x546x583.975962NoYes5321
6x58E33.785192YesYes3211
E2Lig12.11082YesYes3010
6x58Lig4.231922YesYes3010
E2E33.779172YesYes3211
E3Lig4.55252YesYes2010
3x21E1x501.963590NoYes7821
6x61E31.949810NoYes2221
2x67Lig0.4755770NoYes2010
LigNT0.06846152YesNo0701

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
95.45Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
73.08Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
70.83Single6PT2KGCHM076PT2-δ-KGCHM07
69.57Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
69.57Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
68.18Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
68.00Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
66.67Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
66.67Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
65.22Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
64.00Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
64.00Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
62.50Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
62.50Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
59.09Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
59.09Single8E0GBU728E0G-μ-BU72
59.09Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
59.09Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
58.33Single8QJ2pN1628QJ2-MC4-pN162-Gs
57.69Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
57.69Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
57.69Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
56.52Single4RWADIPP-NH24RWA-δ-DIPP-NH2
56.52Single7YITNalfurafine7YIT-κ-Nalfurafine
56.52Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
56.52Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
56.52Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
56.52Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
56.52Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
56.52Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
56.00Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
56.00Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
56.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
56.00Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
55.56Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
55.17Single9KDFRES-701-39KDF-ETB-RES-701-3
55.17Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
54.55Single5C1MBU725C1M-μ-BU72
54.55Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
54.55Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
54.55Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
54.55Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
54.17Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
54.17Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
54.17Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
53.85Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
53.85Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
53.85Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
52.17Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
52.17Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
52.00Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
52.00Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
52.00Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
51.85Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
51.85Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
51.85Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
51.85Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
51.72Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
51.72Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
50.00Single5DHHSB-6121115DHH-NOP-SB-612111
50.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
50.00Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
50.00Single7F8XNN90567F8X-CCKA-NN9056
50.00Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
50.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
50.00Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
50.00Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
50.00Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
50.00Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
50.00Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
50.00Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
50.00Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
50.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
50.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
50.00Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
50.00Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
50.00Consensuslpl_onOrthosteric Ligands1p_on lpa_on
50.00Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
50.00Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
50.00Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
50.00Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
48.28Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
48.28Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
48.28Single8ZRTET-18ZRT-ETB-ET-1
48.28Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
48.15Single3QAKUK-4320973QAK-A2A-UK-432097
48.15Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
48.15Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
48.15Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
48.00Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
48.00Single5X93K-87945X93-ETB-K-8794
48.00Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
48.00Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
48.00Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
48.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
48.00Consensusendothelin_offOrthosteric Ligandetb_off
48.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
48.00Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
47.83Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
47.83Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
47.83Single7WC6LSD7WC6-5-HT2A-LSD
47.83Single8JXSPF-61428JXS-D1-PF-6142
47.83Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
47.83Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
47.83Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
47.06Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
46.88Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
46.88Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
46.88Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
46.88Consensusbombesin_onOrthosteric Ligandbb2_on
46.88Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
46.88Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
46.67Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
46.67Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
46.43Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
46.43Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
46.43Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
46.43Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
46.43Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
46.43Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
46.43Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
46.15Single3NY9ICI118-5513NY9-β2-ICI118-551
46.15Single4UG2CGS216804UG2-A2A-CGS21680
46.15Single6PT3DPI-2876PT3-δ-DPI-287
46.15Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
46.15Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
46.15Single8X5YAstemizole8X5Y-H1-Astemizole
46.15Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
46.15Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
46.15Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
46.15Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
46.15Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
45.83Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
45.83Single4DJHJDTic4DJH-κ-JDTic
45.83Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
45.83Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
45.83Single6H7JIsoprenaline6H7J-β1-Isoprenaline
45.83Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
45.83Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
45.83Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
45.83Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
45.83Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
45.83Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
45.83Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
45.83Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
45.83Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
45.83Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
45.83Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
45.83Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
45.83Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
45.83Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
45.83Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
45.83Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
45.83Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
45.83Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
45.83Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
45.83Single8XVLZibotentan8XVL-ETA-Zibotentan
45.83Single9BJKNaloxone9BJK-μ-Naloxone-NAM
45.83Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
45.83Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
45.83Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
45.83Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
45.83Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
45.83Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
45.83Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
45.83Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
45.83Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
45.83Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
45.83Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
45.83Consensuslpa_onOrthosteric Ligandlpa1_on
45.83Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
45.45Single6IQLL7458706IQL-D4-L745870
45.45Single6TPGEMPA6TPG-OX2-EMPA
45.45Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
45.45Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
45.45Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
45.45Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
45.45Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
44.83Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
44.83Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
44.83Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
44.44Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
44.44Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
44.44Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
44.44Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
44.44Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
44.12Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
44.00Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
44.00Single4LDEBI1671074LDE-β2-BI167107
44.00Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
44.00Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
44.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
44.00Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
44.00Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
44.00Single8JJ8Formoterol8JJ8-β2-Formoterol
44.00Single8JJLOlodaterol8JJL-β2-Olodaterol
44.00Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
44.00Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
44.00Consensusorexin_onOrthosteric Ligandox2_on
44.00Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
43.75Single6IGLIRL16206IGL-ETB-IRL1620
43.75Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
43.75Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
43.48Single2Y04Salbutamol2Y04-β1-Salbutamol
43.48Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
43.48Single4EJ4Naltrindole4EJ4-δ-Naltrindole
43.48Single5DHGC-355DHG-NOP-C-35
43.48Single6TOTLemborexant6TOT-OX1-Lemborexant
43.48Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
43.48Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
43.48Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
43.48Single7UL4Alvimopan7UL4-μ-Alvimopan
43.48Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
43.48Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
43.48Single8JXRLSD8JXR-D1-LSD
43.48Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.48Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.48Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
43.48Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
43.48Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
43.48Consensusa3_onOrthosteric Liganda3a_on
43.48Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
43.48Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
43.33Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
43.33Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
43.33Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
43.33Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.86Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
42.86Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
42.86Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
42.86Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
42.86Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
42.86Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
42.86Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
42.86Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
42.42Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
42.42Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
42.42Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
42.42Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
42.42Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
42.31Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
42.31Single6H7LDobutamine6H7L-β1-Dobutamine
42.31Single7EZCUKA7EZC-A2A-UKA
42.31Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
42.31Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
42.31Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
42.31Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
42.31Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
42.31Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
42.31Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
42.31Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
42.31Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
42.31Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
42.31Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
42.31Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
42.31Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
42.31Consensuscck_onOrthosteric Ligandccka_on cckb_on
42.31Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
42.31Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
42.31Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
42.31Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
42.31Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
41.94Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
41.94Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
41.94Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
41.67Single2Y03Isoprenaline2Y03-β1-Isoprenaline
41.67Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
41.67Single5JQHS-Carazolol5JQH-β2-S-Carazolol
41.67Single5N2SPSB365N2S-A1-PSB36
41.67Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
41.67Single5WIUNemonapride5WIU-D4-Nemonapride
41.67Single5WIVNemonapride5WIV-D4-Nemonapride-Na
41.67Single5WQCEMPA5WQC-OX2-EMPA
41.67Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
41.67Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
41.67Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
41.67Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
41.67Single6TP6Filorexant6TP6-OX1-Filorexant
41.67Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
41.67Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
41.67Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
41.67Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
41.67Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
41.67Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
41.67Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
41.67Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
41.67Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
41.67Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
41.67Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
41.67Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
41.67Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
41.67Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
41.67Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
41.67Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
41.67Single8GNEKW-63568GNE-A2A-KW-6356-Na
41.67Single8S4DCMF-0198S4D-Apelin-CMF-019
41.67Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
41.67Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
41.67Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
41.67Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
41.67Consensusa3_on_gpOrthosteric Liganda3a_on_gp
41.67Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
41.67Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
41.67Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
41.67Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
41.67Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
41.67Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
41.67Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
41.67Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
41.67Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
41.38Single5WF5UK-4320975WF5-A2A-UK-432097
41.38Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
41.38Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
41.38Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
41.38Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
41.38Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
41.38Consensusangiotensin_onOrthosteric Ligandat1_on
41.38Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
41.38Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
41.38Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
41.18Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
41.18Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
40.91Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
40.91Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
40.91Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
40.91Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
40.91Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
40.74Single5WF6UK-4320975WF6-A2A-UK-432097
40.74Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
40.74Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
40.74Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
40.74Single7XN9L-054,5227XN9-SST2-L-054,522
40.74Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
40.74Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
40.74Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
40.74Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
40.74Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
40.74Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
40.74Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
40.74Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
40.74Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
40.74Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
40.74Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
40.62Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
40.62Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
40.62Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
40.62Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
40.62Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
40.62Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
40.62Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
40.54Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
40.54Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
40.00Single2YDVNECA2YDV-A2A-NECA
40.00Single3P0GBI1671073P0G-β2-BI167107
40.00Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
40.00Single4UHRCGS216804UHR-A2A-CGS21680
40.00Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
40.00Single5G53NECA5G53-A2A-NECA-Gs
40.00Single6J21Aprepitant6J21-NK1-Aprepitant
40.00Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
40.00Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
40.00Single6TQ7SB-3348676TQ7-OX1-SB-334867
40.00Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
40.00Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
40.00Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
40.00Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
40.00Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
40.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
40.00Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
40.00Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
40.00Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
40.00Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
40.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
40.00Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
40.00Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
40.00Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
40.00Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
40.00Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
40.00Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
40.00Single8ZWFJR14a8ZWF-C3aB-JR14a
40.00Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
40.00Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
40.00Consensusa2_onOrthosteric Liganda2b_on
40.00Consensusa2_on_gpOrthosteric Liganda2b_on_gp
40.00Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
40.00Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
40.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
40.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
40.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
40.00Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
40.00Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
40.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
40.00Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
40.00Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
40.00Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
40.00Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
39.39Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
39.39Single8IY6Endothelin-18IY6-ETB-Endothelin-1
39.39Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
39.39Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
39.39Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
39.39Consensusbradykinin_onOrthosteric Ligandbk2_on
39.39Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
39.39Consensusendothelin_onOrthosteric Ligandetb_on eta_on
39.39Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
39.39Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
39.29Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
39.29Single4IARErgotamine4IAR-5-HT1B-Ergotamine
39.29Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
39.29Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
39.29Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
39.29Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
39.29Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
39.29Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
39.29Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
39.29Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
39.29Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
39.29Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
39.29Single8WDTphotoNECA8WDT-A2A-photoNECA
39.29Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
39.29Single9M4TSilodosin9M4T-Alpha1A-Silodosin
39.29Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
39.29Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
39.13Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
39.13Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
39.13Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
39.13Single4ZJCSB-6740424ZJC-OX1-SB-674042
39.13Single6PS0S-Carazolol6PS0-β2-S-Carazolol
39.13Single6PS4ICI118-5516PS4-β2-ICI118-551
39.13Single6VI4JDTic6VI4-κ-JDTic
39.13Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
39.13Single6ZG9GSK10347026ZG9-M1-GSK1034702
39.13Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
39.13Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
39.13Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
39.13Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
39.13Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
39.13Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
39.13Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
39.13Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
39.13Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
39.13Single8IHKAcifran8IHK-HCA3-Acifran
39.13Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
39.13Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
39.13Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
39.13Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
39.13Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
39.13Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
39.13Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
39.13Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
39.13Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
39.13Consensusalpha1_onOrthosteric Ligandalpha1a_on
39.13Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
39.13Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
39.13Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
39.13Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
39.13Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
39.13Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
39.13Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
38.71Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
38.71Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
38.71Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
38.71Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.71Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
38.71Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
38.71Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
38.71Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
38.46Single4AMIBucindolol4AMI-β1-Bucindolol
38.46Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
38.46Single6MXTSalmeterol6MXT-β2-Salmeterol
38.46Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
38.46Single6ZG4HTL00099366ZG4-M1-HTL0009936
38.46Single7DFPSpiperone7DFP-D2-Spiperone
38.46Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
38.46Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
38.46Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
38.46Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
38.46Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
38.46Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
38.46Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
38.46Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
38.46Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
38.46Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
38.46Single9DGIZ85267113509DGI-CB1-Z8526711350
38.46Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
38.46Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
38.46Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
38.46Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
38.46Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
38.46Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
38.46Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
38.46Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
38.46Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
38.46Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
38.46Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
38.46Consensuslpa_offOrthosteric Ligandlpa1_off
38.46Consensuslpl_offOrthosteric Ligands1p_off lpa_off
38.46Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
38.46Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
38.24Single5GLHEndothelin-15GLH-ETB-Endothelin-1
38.24Single6IGKEndothelin-36IGK-ETB-Endothelin-3
38.24Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
37.93Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
37.93Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
37.93Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
37.93Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
37.93Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
37.93Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
37.93Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
37.93Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
37.93Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
37.93Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
37.50Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
37.50Single3NY8ICI118-5513NY8-β2-ICI118-551
37.50Single4GBRS-Carazolol4GBR-β2-S-Carazolol
37.50Single4QKX35V4QKX-β2-35V
37.50Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
37.50Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
37.50Single6H7MSalbutamol6H7M-β1-Salbutamol
37.50Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
37.50Single6PS1Timolol6PS1-β2-Timolol
37.50Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
37.50Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
37.50Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
37.50Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
37.50Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
37.50Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
37.50Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
37.50Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
37.50Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
37.50Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
37.50Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
37.50Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
37.50Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
37.50Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
37.50Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
37.50Single8CU6LJ-45178CU6-A2A-LJ-4517
37.50Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
37.50Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
37.50Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
37.50Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
37.50Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
37.50Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
37.50Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
37.50Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
37.50Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
37.50Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
37.50Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
37.50Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
37.50Single8T1WCVN4248T1W-GPR6-CVN424
37.50Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
37.50Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
37.50Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
37.50Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
37.50Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
37.50Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
37.50Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
37.50Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
37.50Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
37.50Single9CHXS-Carazolol9CHX-β2-S-Carazolol
37.50Single9H37A1IR09H37-A2A-A1IR0-Na
37.50Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
37.50Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
37.50Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
37.50Consensus5ht5_onOrthosteric Ligand5ht5a_on
37.50Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
37.50Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
37.50Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
37.50Consensuscck_offOrthosteric Ligandccka_off
37.50Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
37.50Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
37.50Consensusdopamine_offOrthosteric Ligandd2_off d3_off
37.50Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
37.50Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
37.50Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
37.50Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
37.50Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
37.04Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
37.04Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
37.04Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
37.04Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
37.04Single6IBLArformoterol6IBL-β1-Arformoterol
37.04Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
37.04Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
37.04Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
37.04Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
37.04Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
37.04Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
37.04Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
37.04Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
37.04Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.04Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
37.04Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
37.04Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
37.04Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
37.04Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
37.04Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
37.04Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
37.04Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
37.04Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
37.04Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
37.04Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
37.04Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
36.67Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
36.67Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
36.67Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
36.67Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
36.36Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
36.36Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
36.36Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
36.36Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
36.36Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
36.36Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
36.36Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
36.36Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
36.00Single2RH1S-Carazolol2RH1-β2-S-Carazolol
36.00Single2Y00Dobutamine2Y00-β1-Dobutamine
36.00Single2YCWS-Carazolol2YCW-β1-S-Carazolol
36.00Single5D6LS-Carazolol5D6L-β2-S-Carazolol
36.00Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
36.00Single5TVNLSD5TVN-5-HT2B-LSD
36.00Single6E67BI1671076E67-β2-BI167107-Gs(CT)
36.00Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
36.00Single7C4SS1P7C4S-S1P3-S1P
36.00Single7C61Ergotamine7C61-5-HT1B-Ergotamine
36.00Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
36.00Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
36.00Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
36.00Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
36.00Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
36.00Single8QOTNanobody-E8QOT-μ-Nanobody-E
36.00Single8TF5Oleic acid8TF5-GPR6-Oleic acid
36.00Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
36.00Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
36.00Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
36.00Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
36.00Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
36.00Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
36.00Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
36.00Single9HAPTolvaptan9HAP-V2-Tolvaptan
36.00Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
36.00Consensusadenosine_offOrthosteric Liganda1_off a2_off
36.00Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
36.00Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
36.00Consensusamine_offonOrthosteric Ligandamine_off amine_on
36.00Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
36.00Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
36.00Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
36.00Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
36.00Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
36.00Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
36.00Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
36.00Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
36.00Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
36.00Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
36.00Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
36.00Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
36.00Consensustrace-amine_onOrthosteric Ligandta1_on
35.71Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
35.71Single5ZTYAM102575ZTY-CB2-AM10257
35.71Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
35.71Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
35.71Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
35.71Single9IPYJR14a9IPY-C3aB-JR14a
35.71Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
35.71Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
35.48Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
35.48Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
35.48Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
35.48Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
35.48Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
35.48Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
35.48Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
35.48Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
35.48Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
35.48Consensusvasop-oxy_onOrthosteric Ligandv2_on
35.48Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
35.29Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
34.88Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
34.78Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
34.78Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
34.78Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
34.78Single5WS3EMPA5WS3-OX2-EMPA
34.78Single6AKXA4R6AKX-CCR5-A4R
34.78Single6B73MP11046B73-κ-MP1104
34.78Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
34.78Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
34.78Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
34.78Single6TODEMPA6TOD-OX1-EMPA-Na
34.78Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
34.78Single7F8ULintitript7F8U-CCKA-Lintitript
34.78Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
34.78Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
34.78Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
34.78Single7XRRLemborexant7XRR-OX2-Lemborexant
34.78Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
34.78Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
34.78Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
34.78Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
34.78Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
34.78Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
34.78Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
34.78Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
34.78Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
34.78Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
34.78Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
34.78Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
34.78Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
34.78Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
34.78Consensusalpha2_offOrthosteric Ligandalpha2c_off
34.78Consensusorexin_offOrthosteric Ligandox2_off ox1_off
34.78Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
34.78Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
34.62Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
34.62Single5D5AS-Carazolol5D5A-β2-S-Carazolol
34.62Single5D5BS-Carazolol5D5B-β2-S-Carazolol
34.62Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
34.62Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
34.62Single6WGTLSD6WGT-5-HT2A-LSD
34.62Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
34.62Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
34.62Single7TUYGSK682753A7TUY-GPR183-GSK682753A
34.62Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
34.62Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
34.62Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
34.62Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
34.62Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
34.62Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
34.62Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
34.62Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
34.62Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
34.62Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
34.62Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
34.62Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.62Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
34.62Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
34.62Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
34.62Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
34.62Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
34.62Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
34.62Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
34.62Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
34.62Consensusrelaxin_onOrthosteric Ligandrxfp4_on
34.62Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
34.62Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.62Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
34.48Single4XT1Fractalkine4XT1-US28-Fractalkine
34.48Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
34.48Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
34.48Single7QA8Peptide7QA8-STE2-Peptide
34.48Single7QA8Peptide7QA8-STE2-Peptide
34.48Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
34.48Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
34.48Single8WKYPG-9348WKY-MC4-PG-934
34.48Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.48Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
34.48Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
34.48Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
34.48Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
34.48Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
34.48Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
34.48Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
34.48Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
34.48Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
34.48Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
34.48Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
34.38Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
34.38Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
34.38Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
34.38Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
34.38Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
34.38Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
34.38Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
34.38Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
34.38Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
34.38Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
34.38Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
34.38Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
34.38Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
33.33Single3D4STimolol3D4S-β2-Timolol
33.33Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
33.33Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
33.33Single4MBSMaraviroc4MBS-CCR5-Maraviroc
33.33Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
33.33Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
33.33Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
33.33Single5IU7Q274563465IU7-A2A-Q27456346-Na
33.33Single5IUBQ274563445IUB-A2A-Q27456344-Na
33.33Single5JTBZM-2413855JTB-A2A-ZM-241385
33.33Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
33.33Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
33.33Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
33.33Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
33.33Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
33.33Single6A93Risperidone6A93-5-HT2A-Risperidone
33.33Single6CM4Risperidone6CM4-D2-Risperidone
33.33Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
33.33Single6HLOAprepitant6HLO-NK1-Aprepitant
33.33Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
33.33Single6KUXRS-799486KUX-α2a-RS-79948
33.33Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
33.33Single6PS5S-Propranolol6PS5-β2-S-Propranolol
33.33Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
33.33Single6TP3Nemorexant6TP3-OX1-Nemorexant
33.33Single6TPNHTL66416TPN-OX2-HTL6641
33.33Single6V9SGTPL114036V9S-OX1-GTPL11403
33.33Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
33.33Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
33.33Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
33.33Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
33.33Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
33.33Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
33.33Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
33.33Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
33.33Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
33.33Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
33.33Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
33.33Single7F61PF-036547467F61-H3-PF-03654746
33.33Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
33.33Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
33.33Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
33.33Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
33.33Single7SK3CXCL127SK3-ACKR3-CXCL12
33.33Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
33.33Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
33.33Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
33.33Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
33.33Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
33.33Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
33.33Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
33.33Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
33.33Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
33.33Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
33.33Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
33.33Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
33.33Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
33.33Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
33.33Single8JWY2-1188JWY-A2A-2-118
33.33Single8JWZAB9288JWZ-A2A-AB928-Na
33.33Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
33.33Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
33.33Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
33.33Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
33.33Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
33.33Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
33.33Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
33.33Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
33.33Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
33.33Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
33.33Single8XYIVUF106618XYI-CXCR3-VUF10661
33.33Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
33.33Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
33.33Single9ARXSerotonin9ARX-5-HT2A-Serotonin
33.33Single9AS3LSD9AS3-5-HT2A-LSD
33.33Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9AS5Mescaline9AS5-5-HT2A-Mescaline
33.33Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
33.33Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
33.33Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
33.33Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
33.33Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
33.33Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
33.33Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
33.33Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
33.33Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
33.33Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
33.33Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
33.33Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
33.33Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
33.33Consensusa2_offOrthosteric Liganda2a_off
33.33Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
33.33Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
33.33Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
33.33Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
33.33Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
33.33Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
33.33Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
33.33Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
33.33Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
33.33Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
33.33Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
33.33Consensusgrh_offOrthosteric Ligandgnrh1_off
33.33Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
33.33Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
33.33Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
33.33Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
32.35Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
32.35Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
32.35Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
32.35Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
32.26Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
32.26Single6W25SHU91196W25-MC4-SHU9119-Ca
32.26Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
32.26Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.26Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
32.26Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
32.14Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
32.14Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
32.14Single6K1QIRL25006K1Q-ETB-IRL2500
32.14Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Single7UM4AS26747237UM4-5-HT5A-AS2674723
32.14Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
32.14Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
32.14Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
32.14Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.14Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
32.14Single8ZPLHF511168ZPL-CXCR4-HF51116
32.14Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
32.00Single2Y01Dobutamine2Y01-β1-Dobutamine
32.00Single2Y02Carmoterol2Y02-β1-Carmoterol
32.00Single3EMLZM-2413853EML-A2A-ZM-241385
32.00Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
32.00Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
32.00Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
32.00Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
32.00Single5IU8Q274563475IU8-A2A-Q27456347-Na
32.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
32.00Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
32.00Single5UIGCmpd-15UIG-A2A-Cmpd-1
32.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
32.00Single6DRXLisuride6DRX-5-HT2B-Lisuride
32.00Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
32.00Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
32.00Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
32.00Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
32.00Single6S0LZM-2413856S0L-A2A-ZM-241385
32.00Single7BU7BI1671077BU7-β1-BI167107
32.00Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
32.00Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
32.00Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
32.00Single7PYRPSB-21157PYR-A2A-PSB-2115
32.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
32.00Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
32.00Single7V3ZCP559407V3Z-CB1-CP55940
32.00Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
32.00Single7WC7Lisuride7WC7-5-HT2A-Lisuride
32.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
32.00Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
32.00Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
32.00Single8JJOAlprenolol8JJO-β2-Alprenolol
32.00Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
32.00Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
32.00Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
32.00Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
32.00Single8X64Desloratadine8X64-H1-Desloratadine
32.00Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
32.00Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
32.00Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
32.00Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
32.00Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
32.00Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
32.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
32.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
32.00Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
32.00Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
32.00Consensusalpha2_onOrthosteric Ligandalpha2b_on
32.00Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
32.00Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
32.00Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
32.00Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
32.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
32.00Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
32.00Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
32.00Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
31.82Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
31.82Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
31.82Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
31.58Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
31.43Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
31.25Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
31.25Single6JODAngiotensin II6JOD-AT2-Angiotensin II
31.25Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
31.25Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
31.25Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
31.25Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.25Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
31.25Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
31.25Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
31.25Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
31.25Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
31.03Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
31.03Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
31.03Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
31.03Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
31.03Single7SK9CCX6627SK9-ACKR3-CCX662
31.03Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
31.03Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
31.03Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
31.03Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
31.03Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
31.03Consensuskisspeptin_onOrthosteric Ligandkiss1_on
31.03Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single5IUAQ274563485IUA-A2A-Q27456348-Na
30.77Single5N2RPSB-365N2R-A2A-PSB-36-Na
30.77Single5XPRBosentan5XPR-ETB-Bosentan
30.77Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
30.77Single6HLPNetupitant6HLP-NK1-Netupitant
30.77Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
30.77Single6LUQHaloperidol6LUQ-D2-Haloperidol
30.77Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
30.77Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
30.77Single6PS6Timolol6PS6-β2-Timolol
30.77Single6S0QZM-2413856S0Q-A2A-ZM-241385
30.77Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
30.77Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
30.77Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
30.77Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
30.77Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
30.77Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
30.77Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
30.77Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
30.77Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
30.77Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
30.77Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
30.77Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
30.77Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
30.77Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
30.77Single9EHSLUF76029EHS-A3A-LUF7602
30.77Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
30.77Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.77Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
30.77Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
30.77Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
30.77Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
30.77Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
30.77Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
30.77Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
30.77Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
30.77Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
30.77Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
30.56Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
30.43Single3PBLEticlopride3PBL-D3-Eticlopride
30.43Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
30.43Single6TP4ACT-4622066TP4-OX1-ACT-462206
30.43Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
30.43Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
30.43Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
30.43Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
30.43Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
30.43Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
30.43Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
30.43Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
30.43Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
30.43Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
30.43Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
30.43Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
30.30Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
30.30Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
30.30Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
30.30Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
30.30Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.30Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
30.00Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
30.00Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
30.00Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
30.00Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
30.00Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
30.00Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
30.00Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
30.00Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
30.00Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
30.00Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.00Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
30.00Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
29.63Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
29.63Single4U15Tiotropium4U15-M3-Tiotropium
29.63Single5V54Methiothepin5V54-5-HT1B-Methiothepin
29.63Single5XR8AM8415XR8-CB1-AM841
29.63Single5XRAAM115425XRA-CB1-AM11542
29.63Single6E59L-7607356E59-NK1-L-760735
29.63Single6J20Aprepitant6J20-NK1-Aprepitant
29.63Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
29.63Single6OL9Tiotropium6OL9-M5-Tiotropium
29.63Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
29.63Single7B6WCyclazosin7B6W-α1b-Cyclazosin
29.63Single7FEECP559407FEE-CB1-CP55940-ZCZ011
29.63Single7PX4PSB-21137PX4-A2A-PSB-2113
29.63Single7R0CAVP7R0C-V2-AVP-Arrestin2
29.63Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
29.63Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.63Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
29.63Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
29.63Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
29.63Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
29.63Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
29.63Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
29.63Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
29.63Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
29.63Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
29.63Consensus5ht1_offOrthosteric Ligand5ht1b_off
29.63Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
29.63Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
29.63Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
29.63Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
29.63Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
29.63Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
29.63Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
29.63Consensustachykinin_offOrthosteric Ligandnk1_off
29.41Single4XT3Fractalkine4XT3-US28-Fractalkine
29.41Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
29.41Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
29.17Single3ODUIT1t3ODU-CXCR4-IT1t
29.17Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
29.17Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
29.17Single4S0VSuvorexant4S0V-OX2-Suvorexant
29.17Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
29.17Single6AKYMaraviroc6AKY-CCR5-Maraviroc
29.17Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
29.17Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
29.17Single6TPJSuvorexant6TPJ-OX2-Suvorexant
29.17Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
29.17Single7BR3Elagolix7BR3-GnRH1-Elagolix
29.17Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
29.17Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
29.17Single7F8YDevazepide7F8Y-CCKA-Devazepide
29.17Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
29.17Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.17Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
29.17Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
29.17Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
29.17Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
29.17Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
29.17Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
29.17Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
29.17Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
29.17Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
29.17Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
29.17Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.17Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
29.17Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
29.17Single8Y0HVUF114188Y0H-CXCR3-VUF11418
29.17Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
29.17Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
29.17Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
29.17Single9H2XA1IR19H2X-A2A-A1IR1-Na
29.17Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
29.17Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
29.17Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.17Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
29.17Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
29.17Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
29.17Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
29.17Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
29.17Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
29.17Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
29.17Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
29.03Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
29.03Single7SK5CXCL127SK5-ACKR3-CXCL12
29.03Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
29.03Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
29.03Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
29.03Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
29.03Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
28.95Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
28.57Single4PY02MeSATP4PY0-P2Y12-2MeSATP
28.57Single5CXVTiotropium5CXV-M1-Tiotropium
28.57Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
28.57Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
28.57Single6KQICP559406KQI-CB1-CP55940-Org27569
28.57Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
28.57Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
28.57Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
28.57Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
28.57Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
28.57Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
28.57Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
28.57Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
28.57Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
28.57Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
28.57Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
28.57Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
28.57Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
28.12Single3OE0CVX153OE0-CXCR4-CVX15
28.12Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
28.12Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
28.12Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
28.12Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
28.12Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
28.12Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
28.12Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
28.00Single2YDOAdenosine2YDO-A2A-Adenosine
28.00Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
28.00Single5UVIZM-2413855UVI-A2A-ZM-241385
28.00Single6AQFZM-2413856AQF-A2A-ZM-241385
28.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
28.00Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
28.00Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
28.00Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
28.00Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
28.00Single7AROLUF58337ARO-A2A-LUF5833-Na
28.00Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
28.00Single7T32ZM-2413857T32-A2A-ZM-241385
28.00Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
28.00Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
28.00Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
28.00Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
28.00Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
28.00Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
28.00Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
28.00Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
28.00Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
28.00Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
28.00Single8K5CAcipimox8K5C-HCA2-Acipimox
28.00Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
28.00Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
28.00Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
28.00Single8ZPNAMD31008ZPN-CXCR4-AMD3100
28.00Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
28.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
28.00Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
28.00Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
28.00Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
28.00Consensushca_onOrthosteric Ligandhca2_on
28.00Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
28.00Consensusopsins_offOrthosteric Ligandrhodopsin_off
28.00Consensussensory_offOrthosteric Ligandopsins_off
27.78Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
27.59Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
27.59Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
27.59Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
27.59Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
27.59Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
27.59Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
27.59Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
27.59Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
27.59Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
27.59Consensusprostanoid_offOrthosteric Ligandep_off dp_off
27.50Consensuspth_onOrthosteric Ligandpth1_on pth2_on
27.27Single3OE8IT1t3OE8-CXCR4-IT1t
27.27Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
27.27Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
27.27Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
27.27Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
27.27Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
27.27Single9CHUNoradrenaline9CHU-β2-Noradrenaline
27.27Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
27.27Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
27.27Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.27Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.27Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
27.27Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
27.27Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
27.27Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
27.27Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
26.92Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
26.92Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
26.92Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
26.92Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
26.92Single5TGZAM65385TGZ-CB1-AM6538
26.92Single5UENDU1725UEN-A1-DU172
26.92Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
26.92Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
26.92Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
26.92Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
26.92Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
26.92Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
26.92Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
26.92Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
26.92Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
26.92Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
26.92Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
26.92Single7YXAONO-54306087YXA-S1P5-ONO-5430608
26.92Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
26.92Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
26.92Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
26.92Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
26.92Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
26.92Single8K5DGSK2560738K5D-HCA2-GSK256073
26.92Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
26.92Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
26.92Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
26.92Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
26.92Single8X63Mepyramine8X63-H1-Mepyramine
26.92Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
26.92Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
26.92Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
26.92Single9JEAAtropine9JEA-M1-Atropine
26.92Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
26.92Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
26.92Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
26.92Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
26.92Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
26.92Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
26.92Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
26.92Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
26.92Consensushca_on_gpOrthosteric Ligandhca2_on_gp
26.92Consensushistamine_offOrthosteric Ligandh1_off
26.67Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
26.67Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.67Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
26.67Single9JF4PD1683689JF4-BB1-PD168368
26.47Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
26.47Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
26.47Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
26.47Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
26.32Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
26.19Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
26.09Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
26.09Single3OE6IT1t3OE6-CXCR4-IT1t
26.09Single3UZAGTPL92363UZA-A2A-GTPL9236
26.09Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
26.09Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
26.09Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
26.09Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
26.09Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
26.09Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
26.09Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
26.09Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
26.09Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
26.09Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
26.09Single9LRCHistamine9LRC-H4-Histamine
26.09Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
26.09Consensus5ht2_onOrthosteric Ligand5ht2b_on
26.09Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.09Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
26.09Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
26.09Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
26.09Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
26.09Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
25.93Single4NTJAZD12834NTJ-P2Y12-AZD1283
25.93Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
25.93Single6D26Fevipiprant6D26-DP2-Fevipiprant
25.93Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
25.93Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
25.93Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
25.93Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
25.93Single7SINNPS-21437SIN-CaS-NPS-2143
25.93Single7SINNPS-21437SIN-CaS-NPS-2143
25.93Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.93Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
25.93Single7W41PD1762527W41-BB2-PD176252
25.93Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
25.93Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
25.93Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
25.93Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
25.93Single8ZMFA1L108ZMF-5-HT2C-A1L10
25.93Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
25.93Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
25.93Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
25.93Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
25.93Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
25.93Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
25.93Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
25.93Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
25.93Consensusbombesin_offOrthosteric Ligandbb2_off
25.93Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
25.93Consensusdp_offOrthosteric Liganddp2_off
25.93Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.93Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
25.93Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
25.93Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.81Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
25.81Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
25.81Single8IEBA1LYA8IEB-GPR156-A1LYA
25.71Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
25.71Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
25.71Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
25.71Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
25.71Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
25.64Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
25.64Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
25.00Single3OE9IT1t3OE9-CXCR4-IT1t
25.00Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
25.00Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
25.00Single4BV0Neurotensin4BV0-NTS1-Neurotensin
25.00Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
25.00Single6HLLCP999946HLL-NK1-CP99994
25.00Single6OS1TRV0266OS1-AT1-TRV026
25.00Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
25.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
25.00Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
25.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
25.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
25.00Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
25.00Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
25.00Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
25.00Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
25.00Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
25.00Single7SRQLSD7SRQ-5-HT2B-LSD
25.00Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
25.00Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
25.00Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
25.00Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
25.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
25.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
25.00Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
25.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
25.00Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
25.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8EA0Iperoxo8EA0-M3-Iperoxo
25.00Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
25.00Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
25.00Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
25.00Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
25.00Single8IEBA1LYA8IEB-GPR156-A1LYA
25.00Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8K5BNiacin8K5B-HCA2-Niacin
25.00Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
25.00Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
25.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
25.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
25.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
25.00Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
25.00Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
25.00Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
25.00Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
25.00Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
25.00Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
25.00Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
25.00Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
25.00Consensusneurotensin_onOrthosteric Ligandnts1_on
25.00Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
25.00Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
25.00Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
25.00Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
24.32Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
24.32Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
24.32Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
24.32Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
24.32Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
24.32Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
24.32Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
24.32Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
24.32Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
24.24Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
24.24Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
24.24Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
24.24Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
24.14Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
24.14Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
24.14Single4XEENeurotensin4XEE-NTS1-Neurotensin
24.14Single4XESNeurotensin4XES-NTS1-Neurotensin
24.14Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
24.14Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
24.14Single6OS2TRV0266OS2-AT1-TRV026
24.14Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
24.14Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
24.14Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
24.14Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
24.14Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.14Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
24.14Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
24.14Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
24.14Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
24.14Single9BJKNAM9BJK-μ-Naloxone-NAM
24.14Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
24.14Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
24.14Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
24.14Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
24.14Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
24.14Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
24.14Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
24.14Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
24.14Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
24.14Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
24.00Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
24.00Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
24.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
24.00Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
24.00Single3PWHZM-2413853PWH-A2A-ZM-241385
24.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
24.00Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
24.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
24.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
24.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
24.00Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
24.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
24.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
24.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
24.00Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
24.00Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
24.00Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
24.00Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
24.00Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
24.00Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
24.00Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
24.00Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
24.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
24.00Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
24.00Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
24.00Single8IWESpermidine8IWE-TA9-Spermidine
24.00Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
24.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
24.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
24.00Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
24.00Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
24.00Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
24.00Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
24.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
24.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
24.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
24.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
24.00Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
24.00Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
24.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
24.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
24.00Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
24.00Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
24.00Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
24.00Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
24.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
24.00Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
24.00Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
24.00Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
24.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
24.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
23.68Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
23.53Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
23.53Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
23.53Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
23.53Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
23.33Single4BUONeurotensin4BUO-NTS1-Neurotensin
23.33Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
23.33Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
23.33Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
23.33Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
23.33Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
23.33Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
23.33Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
23.33Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
23.33Single8XVJMacitentan8XVJ-ETA-Macitentan
23.33Single8XVUCXCL28XVU-CXCR2-CXCL2
23.33Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
23.33Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
23.33Consensuschemerin_onOrthosteric Ligandcml1_on
23.26Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
23.26Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
23.08Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
23.08Single3REYXAC3REY-A2A-XAC
23.08Single3RZECidoxepin3RZE-H1-Cidoxepin
23.08Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
23.08Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
23.08Single6A94Zotepine6A94-5-HT2A-Zotepine
23.08Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
23.08Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
23.08Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
23.08Single6MH8ZM-2413856MH8-A2A-ZM-241385
23.08Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
23.08Single6TPKRetosiban6TPK-OT-Retosiban
23.08Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
23.08Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
23.08Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
23.08Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
23.08Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
23.08Single7UL3Famotidine7UL3-H2-Famotidine
23.08Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
23.08Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
23.08Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
23.08Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
23.08Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
23.08Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
23.08Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
23.08Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
23.08Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
23.08Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
23.08Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
23.08Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
23.08Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
23.08Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.08Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
23.08Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
23.08Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
23.08Single8ZPMAMD0708ZPM-CXCR4-AMD070
23.08Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
23.08Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
23.08Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
23.08Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
23.08Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
23.08Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
23.08Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
23.08Consensusvasop-oxy_offOrthosteric Ligandot_off
22.86Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
22.86Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
22.86Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
22.86Consensuspac_onOrthosteric Ligandpac1_on
22.86Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
22.58Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
22.58Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
22.58Single8XQJJN2418XQJ-Apelin-JN241
22.58Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
22.58Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
22.50Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
22.50Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.22Single4DAJTiotropium4DAJ-M3-Tiotropium
22.22Single4MQSIperoxo4MQS-M2-Iperoxo
22.22Single4QIMANTA XV4QIM-SMO-ANTA XV
22.22Single4U14Tiotropium4U14-M3-Tiotropium
22.22Single4YAYZD-71554YAY-AT1-ZD-7155
22.22Single5DSGTiotropium5DSG-M4-Tiotropium
22.22Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
22.22Single6D27CAY104716D27-DP2-CAY10471
22.22Single6FJ3PTH6FJ3-PTH1-PTH
22.22Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
22.22Single6GPSMK08126GPS-CCR2-MK0812
22.22Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
22.22Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
22.22Single7F83PF-051904577F83-Ghrelin-PF-05190457
22.22Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
22.22Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
22.22Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
22.22Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
22.22Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
22.22Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
22.22Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
22.22Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
22.22Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
22.22Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
22.22Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
22.22Single9AS1DMT9AS1-5-HT2A-DMT
22.22Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
22.22Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
22.22Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
22.22Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
22.22Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Consensusblt_onOrthosteric Ligandblt1_on
22.22Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
22.22Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
22.22Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
22.22Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
22.22Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
22.22Consensusleukotriene_onOrthosteric Ligandblt_on
22.22Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
22.22Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
22.22Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
22.22Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
21.88Single8IEIA1LYA8IEI-GPR156-A1LYA
21.88Single8IEPA1LYA8IEP-GPR156-A1LYA
21.88Single8IEPA1LYA8IEP-GPR156-A1LYA
21.88Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
21.88Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
21.88Single8KIGSHU91198KIG-MC3-SHU9119-Ca
21.88Single8XWNCXCL88XWN-CXCR2-CXCL8
21.74Single3RFMCaffeine3RFM-A2A-Caffeine
21.74Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
21.74Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
21.74Single6TQ9SB-4081246TQ9-OX1-SB-408124
21.74Single8A2OTheophylline8A2O-A2A-Theophylline-Na
21.74Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
21.74Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
21.74Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
21.62Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
21.62Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
21.62Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
21.62Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
21.62Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
21.62Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
21.62Consensusglp_onOrthosteric Ligandglp1_on glp2_on
21.62Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
21.62Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
21.43Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
21.43Single6GPXMK08126GPX-CCR2-MK0812
21.43Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
21.43Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
21.43Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
21.43Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
21.43Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
21.43Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
21.43Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
21.43Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
21.43Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
21.43Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
21.43Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
21.43Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
21.43Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
21.43Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
21.28Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
21.21Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
21.21Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
21.21Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
21.21Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
21.05Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
21.05Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
21.05Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
21.05Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
20.83Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
20.83Single4XNWMRS25004XNW-P2Y1-MRS2500
20.83Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
20.83Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
20.83Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
20.83Single7WC5Psilocin7WC5-5-HT2A-Psilocin
20.83Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.83Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
20.83Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
20.83Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
20.83Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
20.69Single5TZRMK86665TZR-FFA1-MK8666
20.69Single5V56TC1145V56-SMO-TC114
20.69Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
20.69Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
20.69Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
20.69Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
20.69Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
20.69Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
20.69Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
20.69Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
20.69Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
20.69Single9AS9RS130-1809AS9-5-HT2A-RS130-180
20.69Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
20.69Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
20.69Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
20.59Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
20.59Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
20.59Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
20.51Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
20.51Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
20.00Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
20.00Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
20.00Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
20.00Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
20.00Single4N4WSANT-14N4W-SMO-SANT-1
20.00Single5L7IVismodegib5L7I-SMO-Vismodegib
20.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
20.00Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
20.00Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
20.00Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
20.00Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
20.00Single6YVRNTS8-136YVR-NTS1-NTS8-13
20.00Single7K15MKD0467K15-BLT1-MKD046-Na
20.00Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
20.00Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
20.00Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
20.00Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
20.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
20.00Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
20.00Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
20.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
20.00Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
20.00Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
20.00Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
20.00Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
20.00Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
20.00Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
20.00Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
20.00Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
20.00Single8XWACXCL18XWA-CXCR2-CXCL1
20.00Single8XWMCXCL68XWM-CXCR2-CXCL6
20.00Single8XWSCXCL58XWS-CXCR2-CXCL5
20.00Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
20.00Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
20.00Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
20.00Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
20.00Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9AS7Psilocin9AS7-5-HT2A-Psilocin
20.00Single9B9Y7DY9B9Y-CB1-7DY
20.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
20.00Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
20.00Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
20.00Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
20.00Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
20.00Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
19.51Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
19.51Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
19.44Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
19.44Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
19.44Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
19.35Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
19.35Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
19.35Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single8XWFCXCL38XWF-CXCR2-CXCL3
19.35Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
19.35Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single5ZKQABT-4915ZKQ-PAF-ABT-491
19.23Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
19.23Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
19.23Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
19.23Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
19.23Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
19.23Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
19.23Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
19.23Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
19.23Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
19.23Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
19.23Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
19.23Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
19.23Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
19.23Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
19.23Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
19.23Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
19.23Consensusangiotensin_offOrthosteric Ligandat1_off
19.23Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
19.23Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
19.23Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
19.23Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
19.23Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
19.05Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
18.92Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
18.92Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
18.92Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
18.92Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
18.92Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
18.92Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
18.92Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
18.92Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
18.75Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
18.75Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
18.75Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
18.75Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
18.75Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
18.75Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
18.75Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
18.75Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
18.60Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
18.60Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
18.52Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
18.52Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
18.52Single7VODCariprazine7VOD-5-HT2A-Cariprazine
18.52Single7VV6C48/807VV6-MRGPRX2-C48/80
18.52Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
18.52Single8K2WAMG4878K2W-CXCR3-AMG487
18.52Single8RLNLUF58348RLN-A2A-LUF5834
18.52Single9BA0A1AKN9BA0-CB1-A1AKN
18.52Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
18.52Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
18.52Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
18.52Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
18.52Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
18.42Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
18.42Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
18.42Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
18.42Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
18.42Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
18.42Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
18.18Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
18.18Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
18.18Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8IEIA1LYA8IEI-GPR156-A1LYA
18.18Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
18.18Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
17.95Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
17.95Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
17.95Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
17.95Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
17.95Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
17.95Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.95Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
17.95Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
17.86Single5T04Neurotensin5T04-NTS1-Neurotensin
17.86Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
17.86Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
17.86Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
17.86Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
17.86Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
17.86Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
17.86Single9IYAONO-97105319IYA-GPR55-ONO-9710531
17.65Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
17.65Single7XNACYN1548067XNA-SST2-CYN154806
17.65Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
17.50Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
17.50Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
17.50Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
17.39Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
17.39Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
17.39Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
17.39Single7WC4Serotonin7WC4-5-HT2A-Serotonin
17.39Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
17.39Single8PWNTheophylline8PWN-A2A-Theophylline
17.39Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
17.24Single4JKVTaladegib4JKV-SMO-Taladegib
17.24Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
17.24Single5CGCHTL142425CGC-mGlu5-HTL14242
17.24Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
17.24Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
17.24Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
17.24Single6Z4SSR486926Z4S-NTS1-SR48692
17.24Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.24Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
17.24Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
17.24Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
17.24Single9B9ZA1AKO9B9Z-CB1-A1AKO
17.24Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
17.24Consensusblt_offOrthosteric Ligandblt1_off
17.24Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
17.24Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
17.24Consensusep_offOrthosteric Ligandep4_off
17.14Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
17.14Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
17.14Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
17.07Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
17.07Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
17.02Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
16.67Single5V57TC1145V57-SMO-TC114
16.67Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
16.67Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
16.67Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
16.67Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
16.67Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
16.67Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
16.67Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
16.67Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
16.67Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
16.67Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
16.67Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
16.67Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
16.67Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
16.67Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
16.67Consensusp2y_offOrthosteric Ligandp2y1_off
16.67Consensussensory_onOrthosteric Ligandopsins_on
16.28Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
16.22Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
16.22Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
16.22Consensuscalcitonin_onOrthosteric Ligandctlike_on
16.13Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
16.13Single5X33BIIL2605X33-BLT1-BIIL260
16.13Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
16.13Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
16.13Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
16.13Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8XQJJN2418XQJ-Apelin-JN241
16.13Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
16.13Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
16.13Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.13Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
16.00Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
16.00Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
16.00Single6ME5Agomelatine6ME5-MT1-Agomelatine
16.00Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
16.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
16.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
16.00Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
16.00Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
16.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
16.00Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
16.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
16.00Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
16.00Consensusgi_sensoryOrthosteric Ligandgi_opsins
16.00Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
16.00Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
16.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
16.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
16.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
15.79Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
15.79Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
15.79Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
15.79Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
15.79Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
15.79Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
15.79Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
15.62Single5CGDHTL142425CGD-mGlu5-HTL14242
15.62Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
15.62Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
15.62Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
15.62Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
15.62Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
15.62Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single4O9RCyclopamine4O9R-SMO-Cyclopamine
15.38Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
15.38Single6LI0C176LI0-GPR52-C17
15.38Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
15.38Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
15.38Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
15.38Single7UL2SR486927UL2-NTS1-SR48692-Na
15.38Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
15.38Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
15.38Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
15.38Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
15.38Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
15.38Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
15.38Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
15.38Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
15.38Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
15.38Consensusneurotensin_offOrthosteric Ligandnts1_off
15.38Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
15.15Single6KNMJN241-96KNM-Apelin-JN241-9
15.15Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
15.15Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
15.15Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
15.15Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
15.15Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
15.00Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
15.00Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
14.81Single4BWBNeurotensin4BWB-NTS1-Neurotensin
14.81Single4QINSAG1.54QIN-SMO-SAG1.5
14.81Single5U09Taranabant5U09-CB1-Taranabant
14.81Single6ME9Ramelteon6ME9-MT2-Ramelteon
14.81Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
14.81Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
14.81Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
14.81Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
14.81Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
14.81Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
14.81Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
14.81Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
14.81Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
14.71Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
14.71Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
14.71Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
14.71Consensussomatostatin_offOrthosteric Ligandsst2_off
14.63Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
14.29Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
14.29Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
14.29Single6ZINSR486926ZIN-NTS1-SR48692
14.29Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
14.29Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
14.29Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
14.29Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
14.29Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
14.29Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
13.95Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
13.79Single6IIVDaltroban6IIV-TXA2-Daltroban
13.79Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
13.79Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
13.79Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
13.79Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
13.79Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
13.79Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
13.64Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
13.64Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
13.51Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
13.51Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
13.51Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
13.33Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
13.33Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
13.33Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
13.33Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
13.33Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
13.33Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
13.33Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
13.33Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
13.33Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
13.33Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
13.33Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9HC04YI9HC0-mGlu5-4YI
13.33Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
13.04Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
13.04Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
13.04Single5MZPCaffeine5MZP-A2A-Caffeine-Na
13.04Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
13.04Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
12.90Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
12.90Single7F1TMIP-1a7F1T-CCR5-MIP-1a
12.90Single7P2L4YI7P2L-mGlu5-4YI
12.90Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
12.90Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
12.90Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
12.90Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
12.50Single6IIURamatroban6IIU-TXA2-Ramatroban
12.50Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
12.50Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
12.50Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
12.50Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
12.20Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
12.12Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
12.12Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
12.12Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
12.00Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
11.54Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
11.54Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
11.54Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
11.54Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
11.54Single8JPSCCL78JPS-ACKR1-CCL7
11.54Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
11.54Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
11.43Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
11.43Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
11.11Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
11.11Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
11.11Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
11.11Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
11.11Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
11.11Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
11.11Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
11.11Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
11.11Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
11.11Consensusgq_nucleotideOrthosteric Ligandgq_p2y
11.11Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
10.71Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
10.71Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
10.71Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
10.71Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
10.53Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
10.34Single6FFIMMPEP6FFI-mGlu5-MMPEP
10.34Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
10.34Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
10.26Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
10.00Single6FFHFenobam6FFH-mGlu5-Fenobam
10.00Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
10.00Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
10.00Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
10.00Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
9.68Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
9.52Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
9.38Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
9.38Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
8.82Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
8.70Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
8.57Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
8.33Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
8.33Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
8.00Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.00Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
7.69Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
7.69Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
7.69Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
7.41Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
7.41Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
7.14Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
6.90Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
6.90Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
6.45Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
6.25Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.25Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
6.25Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
6.25Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
6.25Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
4.55Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.55Single6D35Cholesterol6D35-SMO-Cholesterol
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.55Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.55Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.55Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.55Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.55Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
4.55Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.55Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.55Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTTCa7DTT-CaS-Ca-Ca
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTUTryptophan7DTU-CaS-Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.55Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.55Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.55Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.55Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.55Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.55Single7XW7K1-707XW7-TSH-K1-70
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.55Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.55Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.55Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.55Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.55Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.55Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.55Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.55Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.55Single8WVXNorrin8WVX-LGR4-Norrin
4.55Single8WVYNorrin8WVY-LGR4-Norrin
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.55Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.55Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.55Single9KHHNorrin9KHH-LGR4-Norrin
4.55Single9S37NB219S37-LGR4-NB21
4.55Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.35Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.35Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.35Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.35Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.35Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.17Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.17Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.17Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.00Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.00Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.00Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.00Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.00Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.00Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
3.85Single5L7DCholesterol5L7D-SMO-Cholesterol
3.85Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.85Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
3.85Single8HS2Fab0468HS2-GPR20-Fab046
3.85Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.85Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
3.70Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
3.57Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
3.57Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
3.45Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
3.45Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.45Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
3.45Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
3.45Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
3.33Single4XNVBPTU4XNV-P2Y1-BPTU
3.33Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
3.33Single7WV9ZCZ0117WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
3.23Single8IYXYL-3658IYX-GPR34-YL-365
3.23Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
2.94Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
2.63Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.63Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.50Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.50Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.44Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.27Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
mop_on_gp 8F7R-μ-Endomorphin-Gi1/β1/γ2
8EF5-μ-Fentanyl-Gi1/β1/γ2
7SCG-μ-FH210-Gi1/β1/γ2
7T2H-μ-Lofentanil-Gi1/β1/γ2
7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
8EF6-μ-Morphine-Gi1/β1/γ2
8EFB-μ-Oliceridine-Gi1/β1/γ2
7U2L-μ-PubChem 163201242-Gi1/β1/γ2
8EFO-μ-PZM21-Gi1/β1/γ2
8EFL-μ-SR17018-Gi1/β1/γ2
8F7Q-μ-β-Endorphin-Gi1/β1/γ2
7U2K-μ-C6-guano-Gi1/β1/γ2
8EFQ-μ-Damgo-Gi1/β1/γ2
nop_on_gp 8F7X-NOP-Nociceptin-Gi1/β1/γ2
dop_on_gp 8F7S-δ-Deltorphin-Gi1/β1/γ2
kop_on_gp 8F7W-κ-Dynorphin-Gi1/β1/γ2
8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
8DZP-κ-momSalB-Gi1/β1/γ2
Net Summary
Imin 2.55083
Number of Linked Nodes 890
Number of Links 1105
Number of Hubs 172
Number of Links mediated by Hubs 684
Number of Communities 23
Number of Nodes involved in Communities 265
Number of Links involved in Communities 406
Path Summary
Number Of Nodes in MetaPath 100
Number Of Links MetaPath 99
Number of Shortest Paths 5259962
Length Of Smallest Path 3
Average Path Length 34.5531
Length of Longest Path 60
Minimum Path Strength 0.171699
Average Path Strength 5.32563
Maximum Path Strength 20.2193
Minimum Path Correlation 0.700064
Average Path Correlation 0.992664
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 2.04082
Average % Of Corr. Nodes 35.605
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 49.9483
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following differences:
Id1st Network2nd Network
opioid_off_on_gpopioid_on_gpopioid_off
This network is also present in following consensuses:
IdComponents
peptide_on_gpcck_on_gp
angiotensin_on_gp
apelin_on_gp
bombesin_on_gp
bradykinin_on_gp
compl-peptide_on_gp
endothelin_on_gp
formylpeptide_on_gp
galanin_on_gp
ghrelin_on_gp
kisspeptin_on_gp
melanocortin_on_gp
motilin_on_gp
neuromedin-u_on_gp
npy_on_gp
neurotensin_on_gp
opioid_on_gp
orexin_on_gp
relaxin_on_gp
somatostatin_on_gp
tachykinin_on_gp
trh_on_gp
vasop-oxy_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download opioid_on_gp.zip



You can click to copy the link of this page to easily come back here later

or use this QR code to link and share this page.



You can also  read or  download a guide explaining the meaning of all files and numerical data.