Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 3.4175402
2G.HN.52 3.80667404
3G.S1.02 5.61833475
4G.S1.05 6.33167419
5G.H1.01 4.89667589
6G.S2.08 6.9675475
7G.S3.01 5.4375474
8G.S3.03 7.58467577
9G.S3.04 9.225416
10G.S3.06 9.26515
11G.S3.08 4.44833419
12G.s3h2.03 4.90889619
13G.H2.02 4.96167418
14G.H2.03 5.88467519
15G.H2.04 4.875419
16G.H2.06 6.2881719
17G.H2.07 5.47792819
18G.H2.08 3.596518
19G.h2s4.01 7.33667519
20G.S4.05 3.2425487
21G.s4h3.04 4.5275898
22G.s4h3.05 4.85417499
23G.s4h3.08 3.23583408
24G.H3.01 5.70167409
25G.H3.09 6.89833669
26G.H3.13 4.8575465
27G.H3.17 7.47715
28G.S5.03 3.38667408
29G.S5.04 4.89569
30G.S5.05 4.53083489
31G.S5.07 4.38333489
32G.HG.04 4.85667409
33G.HG.15 5.81333497
34G.hgh4.01 6.16167406
35G.hgh4.02 6.92667697
36G.hgh4.05 10.3583407
37G.H4.03 7.34867504
38G.H4.10 10.6042496
39G.H4.11 3.65917497
40G.H4.15 5.23733568
41G.h4s6.02 5.64333468
42G.h4s6.11 4.78933567
43G.h4s6.12 6.75134
44G.S6.02 7.260675137
45G.S6.04 8.1625489
46G.s6h5.01 6.44083489
47G.s6h5.02 3.58833407
48G.s6h5.05 4.5409
49G.H5.08 6.34667578
50G.H5.17 4.116674135
51G.H5.26 7.993334235
52b.1x1 1.64917404
53b.1x7 3.67417408
54b.h2x1 4.09083405
55b.lhb1x11 4.335834124
56b.b1x6 7.24667439
57b.l1x3 9.28667639
58b.b2x1 10.5993518
59b.b2x3 3.9775406
60b.b2x5 7.19507
61b.b3x4 5.72167439
62b.l3x2 5.71267539
63b.b4x3 4.5625407
64b.b4x4 9.19583438
65b.b4x5 4.3565147
66b.b4x6 8.62476739
67b.l4x2 13.1025434
68b.b5x2 5.55583407
69b.b5x3 6.78278639
70b.b5x5 6.0754145
71b.b5x7 5.98083407
72b.l5x1 4.584258
73b.l5x5 8.86056619
74b.b6x5 4.193337146
75b.l6x5 6.155834104
76b.b7x1 6.583335104
77b.l7x2 4.496519
78b.l7x4 3.60167419
79b.b8x3 4.3225406
80b.b8x4 5.1425256
81b.l8x1 4.28754145
82b.l8x3 3.558334103
83b.l8x5 3.35754103
84b.l9x3 8.43933519
85b.l9x6 5.67074918
86b.b10x5 5.19609
87b.b11x4 5.85083419
88b.l11x2 9.71917419
89b.b12x3 4.35167458
90b.b12x6 9.65722618
91b.b12x7 6.789174219
92b.b13x7 8.162557
93b.l13x3 7.58759
94b.l13x6 6.31333419
95b.l13x7 4.45333459
96b.b14x3 4.368555
97b.b15x1 8.428559
98b.b15x2 8.92667446
99b.b15x3 5.13417459
100b.l15x1 5.76083417
101b.l15x2 6.41533559
102b.b16x4 11.9575456
103b.b16x5 4.9675405
104b.b16x6 9.135658
105b.b16x7 7.691674269
106b.b17x5 8.085447
107b.b17x7 9.3125448
108b.l17x3 8.52809749
109b.l17x6 6.548519
110b.b18x3 5.9225448
111b.b18x5 6.40833405
112b.l18x1 7.039527156
113b.l18x2 7.444174157
114b.b19x2 8.86067546
115b.b19x4 6.53167448
116b.l19x2 8.93167449
117b.b20x2 4.95533546
118b.b20x4 8.00143748
119b.b20x6 8.92733546
120b.b21x1 8.61533547
121b.b21x4 4.73333405
122b.b21x7 6.75667505
123b.l21x2 4.625414
124b.l21x5 3.66083414
125b.b22x5 5.645335157
126b.l22x5 5.514297179
127b.b23x6 7.32095717
128b.l23x1 8.90833416
129b.b24x4 8.27083416
130b.b24x5 3.68833405
131b.b24x6 7.32667418
132b.b25x3 7.10917415
133b.b25x7 7.61754127
134b.l25x3 8.885335129
135b.l25x6 12.5692418
136b.l27x1 12.3619719
137b.l27x2 8.004174129
138b.b28x3 4.12133537
139b.b28x4 8.725834126
140b.b28x5 4.04833435
141b.b28x6 7.794446129
142g.h1x11 3.37917409
143g.l1x2 4.17917442
144g.l1x4 6.38167448
145g.h2x11 11.1654156
146g.ctx3 6.328336279
147g.ctx6 4.03667406
148g.ctx14 5.96583439
149g.ctx15 5.57133539
150g.ctx16 5.67095738
151Lig 13.30832720
1521x32 2.25833404
1531x39 5.24222627
1541x43 4.82167427
1551x46 4.60833408
1561x50 5.215409
1571x56 4.394167
158I1x48 6.65254165
1592x37 4.0554117
1602x38 5.188675116
1612x42 7.148675117
1622x44 4.185406
1632x50 5.1125429
1642x53 5.644526
1652x57 7.95427
1662x60 9.29833426
167E1x50 6.25852929
168E1x52 8.49833427
1693x28 4.57917425
1703x32 7.84133526
1713x33 7.14667625
1723x36 5.912528
1733x37 6.25778627
1743x38 4.4754187
1753x41 4.50917425
1763x42 8.183896188
1773x50 8.15083409
1783x51 7.996675208
179I2x57 7.334174117
1804x65 7.7225424
181E2.Q182 5.63667424
182E2x51 5.96167422
183E2.F186 3.64417404
184E2.Y187 5.80333405
1855x36 4.19405
1865x51 5.14917407
1875x54 5.666198
1885x55 3.275834194
1895x58 7.151676199
190I3.N230 5.133334134
1916x45 2.92417406
1926x47 4.23278628
1936x48 8.84778629
1946x51 5.812527
1957x26 2.42833403
1967x38 7.76333425
1977x42 8.134527
1987x45 5.96476729
1997x53 6.00933509
2007x55 4.46917406
2018x48 6.0554234
2028x50 6.161335168
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
12x37 2x38 80.2932.58333YesYes1176
22x37 2x40 80.85242.94667YesNo078
31x57 2x40 81.59613.61667NoNo078
41x57 2x44 81.78163.69NoYes076
51x54 2x44 83.0764.28NoYes076
61x54 2x47 83.81233.25NoNo079
71x53 2x47 83.9963.39NoNo099
81x53 8x50 84.17953.93NoYes098
91x56 8x50 85.73128.74YesYes1678
101x56 8x53 86.70132.76667YesNo1674
118x53 I1x48 86.819412.6633NoYes1645
128x56 I1x48 87.60384.95NoYes055
138x52 8x56 87.78412.7NoNo055
148x48 8x52 87.96442.7YesNo045
158x48 G.H5.26 88.292214.77YesYes2345
166x29 G.H5.26 89.40056.04333NoYes055
176x29 G.H5.17 89.57944.19667NoYes055
18G.H5.17 G.h4s6.12 89.56163.15YesYes1354
19G.S6.02 G.h4s6.12 90.971414.2167YesYes1374
20G.H5.10 G.S6.02 92.73187.11667NoYes067
21G.H5.10 G.S5.03 92.90823.79NoYes068
22G.S4.03 G.S5.03 93.43633.43333NoYes078
23G.S4.03 G.S5.05 98.1263.76667NoYes079
24G.S5.05 G.S6.04 48.94624.52667YesYes899
25G.H5.02 G.S6.04 49.07893.05667NoYes049
26G.H5.02 G.s6h5.05 49.14397.37333NoYes049
27G.s6h5.02 G.s6h5.05 99.88874.14667YesYes079
28G.HG.01 G.s6h5.02 99.97247.00667NoYes077
29G.H4.03 G.HG.01 1009.95YesNo047
30G.H4.03 G.HG.04 53.07123.78333YesYes049
31G.HG.04 G.s4h3.01 49.2787.71333YesNo097
32G.S5.06 G.s4h3.01 48.287811.0733NoNo087
33G.S5.04 G.S5.06 94.93783.69YesNo098
34G.S4.04 G.S5.04 93.48673.65NoYes699
35G.H3.08 G.S4.04 97.9916.09NoNo099
36G.H2.04 G.H3.08 97.8695.67YesNo099
37G.H2.04 G.H2.08 62.07853.75667YesYes198
38G.H2.08 G.H3.17 63.76093.13YesYes185
39G.H3.17 b.l27x1 29.59134.37333YesYes159
40b.b26x1 b.l27x1 29.71054.94NoYes099
41b.b26x1 b.b26x2 29.54263.44NoNo097
42b.b26x2 b.b2x3 29.37516.48NoYes076
43b.b28x3 b.b2x3 11.68193.3YesYes076
44G.S5.05 G.s6h5.01 49.08986.48333YesYes899
45G.H5.03 G.s6h5.01 50.42729.26NoYes089
46G.H5.03 G.s6h5.05 50.68894.93667NoYes089
47G.H4.03 G.H4.07 47.06053.55667YesNo045
48G.H4.07 G.S6.05 47.02913.69667NoNo054
49G.S5.06 G.S6.05 46.7797.71667NoNo084
50G.H2.07 b.l9x6 29.69954.18YesYes198
513x50 7x53 12.87766.85667YesYes099
523x46 7x53 75.23096.78333NoYes099
532x42 3x46 75.42395.19YesNo079
542x38 2x42 75.33369.26667YesYes1167
55b.l26x5 g.ctx4 12.5376.15NoNo057
56g.ctx3 g.ctx4 12.18574.29333YesNo097
57b.b21x4 g.h2x1 19.13692.48333YesNo058
58b.b21x2 g.h2x1 18.93814.29667NoNo068
59b.1x19 b.b21x2 18.53994.28333NoNo066
60b.1x19 b.b21x1 11.897210.3233NoYes067
61b.b27x2 b.b2x5 17.20314.32333NoYes057
62b.b27x2 b.b2x3 17.36713.22NoYes056
63b.b2x4 b.b6x5 11.48253.27NoYes066
64b.b10x4 b.b2x4 11.632915.7967NoNo066
65b.b2x5 b.l26x1 10.308712.13YesNo077
66b.b10x2 b.b10x4 10.38165.10667NoNo566
67b.b10x2 b.b6x2 19.8083.38NoNo068
68b.b10x3 b.b6x2 19.96866.19667NoNo088
69b.b10x3 b.b8x1 20.13853.64NoNo088
70b.b11x4 b.b8x1 19.72613.38YesNo098
71b.b11x4 b.l9x3 19.79296.39333YesYes199
72b.b11x6 b.l9x3 25.90515.3433NoYes199
73b.l11x1 b.l9x6 27.17478.20667NoYes198
74b.l23x1 b.l25x6 33.628621.8367YesYes168
75b.l21x7 b.l23x1 33.29315.70333NoYes156
76b.b23x6 b.l21x7 32.33963.58333YesNo175
77b.b23x6 b.b24x6 29.75478.04YesYes178
78b.b21x7 b.b24x6 29.567411.2533YesYes058
79b.b20x5 b.b21x7 18.05416.64333NoYes075
80b.b20x5 b.b21x4 17.89344.15NoYes075
812x53 7x45 34.04453.39333YesYes269
827x45 7x49 45.59914.67667YesNo299
837x49 7x53 50.04216.97667NoYes099
842x53 3x32 26.908810.6567YesYes266
853x32 Lig 22.457913.8067YesYes260
863x50 5x58 11.729210.6333YesYes099
875x58 6x40 11.71673.36667YesNo098
886x40 7x53 12.40583.78667NoYes089
895x54 5x58 10.782812.0367YesYes1989
90G.H2.04 G.H2.07 35.55517YesYes199
91b.b11x6 b.l11x1 27.08223.71NoNo199
92G.H3.17 b.l25x6 32.93654.66667YesYes158
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
1x39Lig3.492YesYes7010
2x60Lig21.62332YesYes6010
E1x50Lig3.722YesYes9010
3x28Lig3.633332YesYes5010
3x32Lig13.80672YesYes6010
3x33Lig5.743332YesYes5010
4x65Lig6.72YesYes4010
E2x50Lig3.466672NoYes9010
6x51Lig4.22YesYes7010
6x55Lig4.382NoYes5010
7x34Lig4.366672NoYes4010
7x38Lig15.262YesYes5010
1x351x393.906670NoYes6721
1x392x607.513332YesYes7611
1x392x613.333332YesNo7712
1x397x395.643332YesNo7512
1x397x427.566672YesYes7712
2x533x3210.65672YesYes6621
2x537x425.716672YesYes6722
2x563x323.390NoYes7621
2x59E1x527.143330NoYes6722
2x593x287.863330NoYes6521
2x602x634.512YesNo6512
2x602x643.546672YesNo6512
2x63E1x507.393330NoYes5921
2x63E2.Q1827.516670NoYes5021
E1x50E1x5213.69672YesYes9712
3x25E1x504.353332NoYes9921
3x28E1x503.272YesYes5911
E1x50E2.V1743.682YesNo9012
E1x50E2x5015.23672YesNo9911
3x25E2.V1743.422NoNo9022
3x25E2x507.282NoNo9921
3x294x6511.44330NoYes5421
3x323x337.613332YesYes6511
3x327x383.742YesYes6511
3x334x6113.28332YesNo5412
3x334x658.933332YesYes5411
3x335x434.392YesNo5512
4x65E2x523.813332YesNo4412
E2.E177E2.Q1828.070NoYes0021
E2.E177E2x516.736670NoYes0221
E2.Q182E2.V1803.822YesNo0012
E2.F186E2x516.190YesYes0221
E2.Y187E2x525.933330YesNo0422
5x32E2.Y1873.746672NoYes3012
6x517x383.52YesYes7511
6x517x4110.572YesNo7812
6x547x343.170NoNo5421
6x547x377.933330NoNo5622
7x387x428.553332YesYes5712
7x397x424.186672NoYes5722
LigNT.E285.362YesNo0001
E2x51Lig7.953332YesYes2010
E2.Q182Lig3.142YesYes0010
LigNT.D265.163332YesNo0001
E2.D178Lig8.430NoYes0010
LigNT.P249.056672YesNo0001
LigNT.S224.466672YesNo0001
LigNT.I207.542YesNo0001
5x32Lig4.692NoYes3010
3x243x283.552NoYes6521
E2x51E2x522.966672YesNo2412
6x516x556.92YesNo7511
6x517x373.892YesNo7612
3x24E1x503.103332NoYes6921
3x334x572.916672YesNo5712
5x33Lig2.503332NoYes1010
LigNT.C212.426672YesNo0001
7x24NT.C252.426672NoNo8012
7x24Lig2.326672NoYes8010
7x247x282.033332NoNo8312
3x21E1x501.873330NoYes8921
5x33E2.Q1891.773332NoNo1012
NT.P24NT.S231.186672NoNo0012
LigNT.A270.572YesNo0001

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
77.78Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
50.00Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
50.00Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
50.00Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
48.28Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
47.83Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
47.62Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
47.62Single8ZWFJR14a8ZWF-C3aB-JR14a
45.45Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
45.45Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
44.44Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
44.44Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
43.48Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
43.48Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
43.48Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
42.86Single8S4DCMF-0198S4D-Apelin-CMF-019
42.86Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
42.31Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
42.31Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
42.11Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
41.67Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
41.67Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
41.67Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
40.91Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
40.91Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
40.91Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
40.91Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
40.74Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
40.74Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
40.74Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
40.00Single4XT1Fractalkine4XT1-US28-Fractalkine
40.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
40.00Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
40.00Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
40.00Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
40.00Consensuslpl_onOrthosteric Ligands1p_on lpa_on
40.00Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
39.29Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
39.29Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
39.29Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
39.29Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
39.13Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
39.13Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
39.13Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
39.13Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
39.13Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
39.13Consensuslpl_offOrthosteric Ligands1p_off lpa_off
38.46Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
38.46Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
38.46Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
38.10Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
38.10Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
37.93Single7SK3CXCL127SK3-ACKR3-CXCL12
37.93Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
37.93Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
37.50Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
37.50Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
37.50Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
37.50Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
37.50Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
37.50Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
37.04Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
37.04Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
37.04Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
37.04Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
37.04Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
37.04Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
37.04Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
37.04Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
37.04Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
36.67Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
36.36Single5C1MBU725C1M-μ-BU72
36.36Single6D26Fevipiprant6D26-DP2-Fevipiprant
36.36Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
36.36Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
36.36Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
36.36Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
36.36Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
36.36Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
36.36Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
36.36Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
36.36Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
36.36Consensusdp_offOrthosteric Liganddp2_off
36.00Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
36.00Single6KNMJN241-96KNM-Apelin-JN241-9
36.00Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
36.00Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
36.00Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
36.00Single8QJ2pN1628QJ2-MC4-pN162-Gs
36.00Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
36.00Single9IPYJR14a9IPY-C3aB-JR14a
35.71Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
35.71Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
35.71Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
35.71Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
35.71Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
35.71Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
35.71Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
35.48Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
35.48Consensusendothelin_onOrthosteric Ligandetb_on eta_on
35.00Single6AKXA4R6AKX-CCR5-A4R
35.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
35.00Single8GNGIstradefylline8GNG-A2A-Istradefylline
35.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
35.00Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
34.78Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
34.78Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
34.78Single7TUYGSK682753A7TUY-GPR183-GSK682753A
34.78Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
34.78Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
34.78Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
34.78Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
34.78Single8E0GBU728E0G-μ-BU72
34.78Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
34.78Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
34.78Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
34.78Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
34.78Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
34.78Consensuslpa_onOrthosteric Ligandlpa1_on
34.78Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
34.62Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
34.62Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
34.62Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
34.62Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
34.62Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
34.48Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
34.48Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
34.48Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
34.48Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
34.48Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
34.48Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
34.38Single5GLHEndothelin-15GLH-ETB-Endothelin-1
34.38Single6IGKEndothelin-36IGK-ETB-Endothelin-3
34.38Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
33.33Single4MBSMaraviroc4MBS-CCR5-Maraviroc
33.33Single4XT3Fractalkine4XT3-US28-Fractalkine
33.33Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
33.33Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
33.33Single7F61PF-036547467F61-H3-PF-03654746
33.33Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
33.33Single7SK5CXCL127SK5-ACKR3-CXCL12
33.33Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
33.33Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
33.33Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
33.33Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
33.33Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
33.33Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
33.33Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
33.33Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
33.33Single8JJLOlodaterol8JJL-β2-Olodaterol
33.33Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
33.33Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
33.33Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
33.33Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
33.33Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
33.33Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
33.33Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
33.33Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
33.33Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
33.33Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
33.33Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
33.33Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
33.33Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
33.33Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
33.33Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
33.33Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
33.33Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
33.33Consensuslpa_offOrthosteric Ligandlpa1_off
33.33Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
33.33Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
33.33Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
32.26Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
32.26Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
32.26Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
32.26Single9KDFRES-701-39KDF-ETB-RES-701-3
32.26Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
32.26Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
32.26Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
32.14Single6PT2KGCHM076PT2-δ-KGCHM07
32.14Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
32.14Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
32.14Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
32.14Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
32.14Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
32.14Consensusangiotensin_onOrthosteric Ligandat1_on
32.14Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
32.14Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
32.14Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
32.14Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
32.00Single5X93K-87945X93-ETB-K-8794
32.00Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.00Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
32.00Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
32.00Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
32.00Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
32.00Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
32.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
32.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
32.00Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
32.00Consensusprostanoid_offOrthosteric Ligandep_off dp_off
31.82Single2Y02Carmoterol2Y02-β1-Carmoterol
31.82Single5DHHSB-6121115DHH-NOP-SB-612111
31.82Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
31.82Single6D27CAY104716D27-DP2-CAY10471
31.82Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
31.82Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
31.82Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
31.82Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
31.82Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
31.82Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
31.82Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
31.82Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
31.82Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
31.82Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
31.82Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
31.82Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
31.58Single7WC5Psilocin7WC5-5-HT2A-Psilocin
31.43Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
31.25Single6IGLIRL16206IGL-ETB-IRL1620
31.25Single8IY6Endothelin-18IY6-ETB-Endothelin-1
31.25Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
31.25Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
31.25Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
31.25Consensusbradykinin_onOrthosteric Ligandbk2_on
31.25Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
31.25Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
31.03Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
31.03Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
31.03Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
31.03Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
31.03Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
31.03Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
31.03Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
31.03Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
30.77Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
30.77Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
30.77Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
30.77Single8XQJJN2418XQJ-Apelin-JN241
30.77Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
30.77Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
30.77Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
30.77Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
30.77Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
30.77Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
30.77Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
30.43Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
30.43Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
30.43Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
30.43Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
30.43Single7C4SS1P7C4S-S1P3-S1P
30.43Single7C61Ergotamine7C61-5-HT1B-Ergotamine
30.43Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
30.43Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
30.43Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
30.43Single8JXSPF-61428JXS-D1-PF-6142
30.43Single8TF5Oleic acid8TF5-GPR6-Oleic acid
30.43Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
30.43Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
30.43Single9EHSLUF76029EHS-A3A-LUF7602
30.43Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
30.43Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
30.43Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
30.43Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
30.30Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
30.30Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
30.30Consensusbombesin_onOrthosteric Ligandbb2_on
30.30Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
30.30Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
30.30Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
30.00Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
30.00Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
30.00Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
30.00Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
30.00Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
30.00Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
30.00Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
30.00Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
30.00Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
29.63Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
29.63Single7F8XNN90567F8X-CCKA-NN9056
29.63Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
29.63Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
29.63Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
29.63Single8WDTphotoNECA8WDT-A2A-photoNECA
29.63Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.63Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
29.63Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
29.63Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.63Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.63Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
29.63Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
29.63Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
29.63Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
29.63Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
29.41Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
29.41Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
29.41Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
29.41Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
29.41Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
29.17Single3P0GBI1671073P0G-β2-BI167107
29.17Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
29.17Single4DJHJDTic4DJH-κ-JDTic
29.17Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
29.17Single6WGTLSD6WGT-5-HT2A-LSD
29.17Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
29.17Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
29.17Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
29.17Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
29.17Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
29.17Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
29.17Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
29.17Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
29.17Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
29.17Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
29.17Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
29.17Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
29.17Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
29.17Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
29.17Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
29.17Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
29.17Single8XVLZibotentan8XVL-ETA-Zibotentan
29.17Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
29.17Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
29.17Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
29.17Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
29.17Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
29.17Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
29.17Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
29.17Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
29.17Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
29.17Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
29.17Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
29.03Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
29.03Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
29.03Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
29.03Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
29.03Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
28.57Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
28.57Single3ODUIT1t3ODU-CXCR4-IT1t
28.57Single3QAKUK-4320973QAK-A2A-UK-432097
28.57Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
28.57Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
28.57Single5ZKQABT-4915ZKQ-PAF-ABT-491
28.57Single6AKYMaraviroc6AKY-CCR5-Maraviroc
28.57Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
28.57Single7BR3Elagolix7BR3-GnRH1-Elagolix
28.57Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
28.57Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
28.57Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
28.57Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
28.57Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
28.57Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
28.57Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
28.57Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
28.57Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
28.57Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
28.57Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
28.57Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
28.57Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
28.57Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
28.57Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
28.57Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
28.57Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
28.57Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
28.57Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.57Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
28.57Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
28.57Consensusangiotensin_offOrthosteric Ligandat1_off
28.57Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
28.57Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
28.57Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
28.57Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
28.57Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
28.57Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
28.57Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
28.57Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
28.57Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
28.12Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
28.12Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
28.12Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
28.12Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
28.12Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
28.00Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
28.00Single4AMIBucindolol4AMI-β1-Bucindolol
28.00Single4RWADIPP-NH24RWA-δ-DIPP-NH2
28.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
28.00Single6A93Risperidone6A93-5-HT2A-Risperidone
28.00Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
28.00Single6MXTSalmeterol6MXT-β2-Salmeterol
28.00Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
28.00Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
28.00Single7DFPSpiperone7DFP-D2-Spiperone
28.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
28.00Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
28.00Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
28.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
28.00Single7YITNalfurafine7YIT-κ-Nalfurafine
28.00Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
28.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
28.00Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
28.00Single8JJ8Formoterol8JJ8-β2-Formoterol
28.00Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
28.00Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.00Single8XQJJN2418XQJ-Apelin-JN241
28.00Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
28.00Consensusalpha1_offOrthosteric Ligandalpha1a_off
28.00Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
28.00Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
28.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
28.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
28.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
28.00Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
27.78Single7WC4Serotonin7WC4-5-HT2A-Serotonin
27.59Single3OE0CVX153OE0-CXCR4-CVX15
27.59Single5WF5UK-4320975WF5-A2A-UK-432097
27.59Single6W25SHU91196W25-MC4-SHU9119-Ca
27.59Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
27.59Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
27.59Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
27.59Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
27.59Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
27.59Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
27.59Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
27.59Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
27.59Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
27.59Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
27.59Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
27.59Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
27.27Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
27.27Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
27.27Single6IQLL7458706IQL-D4-L745870
27.27Single6KUXRS-799486KUX-α2a-RS-79948
27.27Single6MH8ZM-2413856MH8-A2A-ZM-241385
27.27Single6TP3Nemorexant6TP3-OX1-Nemorexant
27.27Single6V9SGTPL114036V9S-OX1-GTPL11403
27.27Single6VI4JDTic6VI4-κ-JDTic
27.27Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
27.27Single7AROLUF58337ARO-A2A-LUF5833-Na
27.27Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
27.27Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
27.27Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
27.27Single8IHKAcifran8IHK-HCA3-Acifran
27.27Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
27.27Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
27.27Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
27.27Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
27.27Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
27.27Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
27.27Single8ZPMAMD0708ZPM-CXCR4-AMD070
27.27Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
27.27Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
27.27Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
27.27Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
27.27Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
27.27Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
27.27Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
27.27Consensusgrh_offOrthosteric Ligandgnrh1_off
27.27Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
27.27Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
26.92Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
26.92Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
26.92Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
26.92Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
26.92Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
26.92Single6IBLArformoterol6IBL-β1-Arformoterol
26.92Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
26.92Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
26.92Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
26.92Single7EZCUKA7EZC-A2A-UKA
26.92Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
26.92Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
26.92Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
26.92Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
26.92Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
26.92Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
26.92Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
26.92Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
26.92Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
26.92Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
26.92Consensuscck_onOrthosteric Ligandccka_on cckb_on
26.92Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
26.92Consensusendothelin_offOrthosteric Ligandetb_off
26.92Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
26.67Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
26.67Single6JODAngiotensin II6JOD-AT2-Angiotensin II
26.67Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.67Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
26.67Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
26.67Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
26.67Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
26.67Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
26.67Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.67Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
26.67Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
26.67Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.67Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
26.67Consensusvasop-oxy_onOrthosteric Ligandv2_on
26.67Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
26.47Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
26.32Single8A2OTheophylline8A2O-A2A-Theophylline-Na
26.32Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
26.32Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
26.09Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
26.09Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
26.09Single4YAYZD-71554YAY-AT1-ZD-7155
26.09Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
26.09Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
26.09Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
26.09Single5UENDU1725UEN-A1-DU172
26.09Single6DRXLisuride6DRX-5-HT2B-Lisuride
26.09Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
26.09Single6PS1Timolol6PS1-β2-Timolol
26.09Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
26.09Single7BU7BI1671077BU7-β1-BI167107
26.09Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
26.09Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
26.09Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
26.09Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
26.09Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
26.09Single7UL4Alvimopan7UL4-μ-Alvimopan
26.09Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
26.09Single7V3ZCP559407V3Z-CB1-CP55940
26.09Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
26.09Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
26.09Single8CU6LJ-45178CU6-A2A-LJ-4517
26.09Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
26.09Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
26.09Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
26.09Single8JXRLSD8JXR-D1-LSD
26.09Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
26.09Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
26.09Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
26.09Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
26.09Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
26.09Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
26.09Single9CHXS-Carazolol9CHX-β2-S-Carazolol
26.09Single9H37A1IR09H37-A2A-A1IR0-Na
26.09Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
26.09Consensus5ht5_onOrthosteric Ligand5ht5a_on
26.09Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
26.09Consensusa3_onOrthosteric Liganda3a_on
26.09Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
26.09Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
26.09Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
26.09Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
25.93Single3NY9ICI118-5513NY9-β2-ICI118-551
25.93Single4UG2CGS216804UG2-A2A-CGS21680
25.93Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
25.93Single5ZTYAM102575ZTY-CB2-AM10257
25.93Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
25.93Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
25.93Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
25.93Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
25.93Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
25.93Single8X5YAstemizole8X5Y-H1-Astemizole
25.93Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
25.93Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
25.93Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
25.93Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
25.93Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
25.93Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
25.93Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
25.81Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
25.81Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
25.81Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
25.81Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.81Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
25.81Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
25.81Single8ZRTET-18ZRT-ETB-ET-1
25.81Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
25.81Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
25.81Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
25.81Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
25.00Single3OE6IT1t3OE6-CXCR4-IT1t
25.00Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
25.00Single4IARErgotamine4IAR-5-HT1B-Ergotamine
25.00Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
25.00Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
25.00Single5JQHS-Carazolol5JQH-β2-S-Carazolol
25.00Single5N2RPSB-365N2R-A2A-PSB-36-Na
25.00Single5N2SPSB365N2S-A1-PSB36
25.00Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
25.00Single5TVNLSD5TVN-5-HT2B-LSD
25.00Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
25.00Single5WQCEMPA5WQC-OX2-EMPA
25.00Single6E67BI1671076E67-β2-BI167107-Gs(CT)
25.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
25.00Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
25.00Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
25.00Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
25.00Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
25.00Single6TP6Filorexant6TP6-OX1-Filorexant
25.00Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
25.00Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
25.00Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
25.00Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
25.00Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
25.00Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
25.00Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
25.00Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
25.00Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
25.00Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
25.00Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
25.00Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
25.00Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
25.00Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.00Single7WC6LSD7WC6-5-HT2A-LSD
25.00Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
25.00Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
25.00Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
25.00Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
25.00Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
25.00Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
25.00Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
25.00Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
25.00Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
25.00Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
25.00Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8WKYPG-9348WKY-MC4-PG-934
25.00Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single9B9ZA1AKO9B9Z-CB1-A1AKO
25.00Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
25.00Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
25.00Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
25.00Single9HAPTolvaptan9HAP-V2-Tolvaptan
25.00Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
25.00Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
25.00Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
25.00Consensus5ht2_onOrthosteric Ligand5ht2b_on
25.00Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
25.00Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
25.00Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
25.00Consensusa3_on_gpOrthosteric Liganda3a_on_gp
25.00Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
25.00Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
25.00Consensusadenosine_offOrthosteric Liganda1_off a2_off
25.00Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
25.00Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
25.00Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
25.00Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
25.00Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
25.00Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
25.00Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
25.00Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
25.00Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
25.00Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
25.00Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
25.00Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
25.00Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
25.00Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
25.00Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
25.00Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.32Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
24.24Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
24.24Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
24.24Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
24.24Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
24.24Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
24.24Consensusglp_onOrthosteric Ligandglp1_on glp2_on
24.24Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
24.14Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
24.14Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
24.14Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
24.14Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
24.14Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
24.14Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
24.14Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
24.14Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
24.14Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
24.14Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
24.14Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
24.00Single2YDVNECA2YDV-A2A-NECA
24.00Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
24.00Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
24.00Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
24.00Single4UHRCGS216804UHR-A2A-CGS21680
24.00Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
24.00Single5G53NECA5G53-A2A-NECA-Gs
24.00Single5XRAAM115425XRA-CB1-AM11542
24.00Single6H7JIsoprenaline6H7J-β1-Isoprenaline
24.00Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
24.00Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
24.00Single6OS1TRV0266OS1-AT1-TRV026
24.00Single6TQ7SB-3348676TQ7-OX1-SB-334867
24.00Single7B6WCyclazosin7B6W-α1b-Cyclazosin
24.00Single7F1TMIP-1a7F1T-CCR5-MIP-1a
24.00Single7FEECP559407FEE-CB1-CP55940-ZCZ011
24.00Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
24.00Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
24.00Single7PX4PSB-21137PX4-A2A-PSB-2113
24.00Single7R0CAVP7R0C-V2-AVP-Arrestin2
24.00Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
24.00Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
24.00Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
24.00Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
24.00Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
24.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
24.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
24.00Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.00Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
24.00Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
24.00Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
24.00Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
24.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
24.00Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
24.00Single9BJKNaloxone9BJK-μ-Naloxone-NAM
24.00Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
24.00Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
24.00Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
24.00Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
24.00Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
24.00Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
24.00Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
24.00Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
24.00Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
24.00Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
23.81Single3OE9IT1t3OE9-CXCR4-IT1t
23.81Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
23.81Single6LI0C176LI0-GPR52-C17
23.81Single7SRQLSD7SRQ-5-HT2B-LSD
23.81Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
23.81Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
23.81Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
23.81Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
23.81Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
23.81Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
23.81Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
23.81Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
23.81Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
23.81Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
23.81Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
23.81Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
23.81Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
23.81Single9B9Y7DY9B9Y-CB1-7DY
23.81Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
23.81Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
23.81Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
23.81Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
23.53Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
23.53Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
23.53Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
23.53Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
23.53Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
23.53Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
23.33Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
23.33Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.33Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
23.33Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
23.33Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
23.33Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
23.08Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
23.08Single4LDEBI1671074LDE-β2-BI167107
23.08Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
23.08Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
23.08Single6CM4Risperidone6CM4-D2-Risperidone
23.08Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
23.08Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
23.08Single6KQICP559406KQI-CB1-CP55940-Org27569
23.08Single6OS2TRV0266OS2-AT1-TRV026
23.08Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
23.08Single6ZG4HTL00099366ZG4-M1-HTL0009936
23.08Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
23.08Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
23.08Single7K15MKD0467K15-BLT1-MKD046-Na
23.08Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
23.08Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
23.08Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
23.08Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
23.08Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
23.08Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
23.08Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
23.08Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
23.08Single9DGIZ85267113509DGI-CB1-Z8526711350
23.08Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
23.08Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
23.08Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
23.08Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
23.08Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
23.08Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
23.08Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
23.08Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
23.08Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
23.08Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
23.08Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
23.08Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
23.08Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
23.08Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
23.08Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
23.08Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
23.08Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
23.08Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
23.08Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
23.08Consensusorexin_onOrthosteric Ligandox2_on
23.08Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.86Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
22.86Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
22.86Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
22.86Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
22.73Single3PWHZM-2413853PWH-A2A-ZM-241385
22.73Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
22.73Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
22.73Single4S0VSuvorexant4S0V-OX2-Suvorexant
22.73Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
22.73Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
22.73Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
22.73Single5U09Taranabant5U09-CB1-Taranabant
22.73Single5WS3EMPA5WS3-OX2-EMPA
22.73Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
22.73Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
22.73Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
22.73Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
22.73Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
22.73Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
22.73Single6TPJSuvorexant6TPJ-OX2-Suvorexant
22.73Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
22.73Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
22.73Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
22.73Single7F8ULintitript7F8U-CCKA-Lintitript
22.73Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
22.73Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
22.73Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
22.73Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
22.73Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
22.73Single7XRRLemborexant7XRR-OX2-Lemborexant
22.73Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
22.73Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
22.73Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
22.73Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
22.73Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
22.73Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
22.73Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
22.73Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
22.73Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
22.73Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
22.73Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
22.73Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
22.73Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
22.73Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
22.73Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
22.73Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.73Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
22.73Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
22.73Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
22.73Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
22.73Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
22.73Consensusalpha2_offOrthosteric Ligandalpha2c_off
22.73Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
22.73Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
22.73Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
22.73Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.73Consensusorexin_offOrthosteric Ligandox2_off ox1_off
22.73Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
22.73Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
22.73Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
22.73Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.73Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
22.58Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
22.58Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
22.58Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
22.58Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
22.58Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
22.22Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
22.22Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
22.22Single6H7LDobutamine6H7L-β1-Dobutamine
22.22Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
22.22Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
22.22Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
22.22Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
22.22Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
22.22Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
22.22Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
22.22Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
22.22Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
22.22Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
22.22Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
22.22Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
22.22Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
22.22Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
22.22Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
22.22Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
22.22Single8XVUCXCL28XVU-CXCR2-CXCL2
22.22Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
22.22Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
22.22Single8ZPLHF511168ZPL-CXCR4-HF51116
22.22Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
22.22Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
22.22Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
22.22Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
22.22Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
22.22Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
22.22Consensuschemerin_onOrthosteric Ligandcml1_on
22.22Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
22.22Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
22.22Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
21.88Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
21.88Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
21.88Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
21.88Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
21.88Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
21.88Consensuspac_onOrthosteric Ligandpac1_on
21.88Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
21.74Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
21.74Single2YDOAdenosine2YDO-A2A-Adenosine
21.74Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
21.74Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
21.74Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
21.74Single4ZJCSB-6740424ZJC-OX1-SB-674042
21.74Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
21.74Single5IU7Q274563465IU7-A2A-Q27456346-Na
21.74Single5IUBQ274563445IUB-A2A-Q27456344-Na
21.74Single5JTBZM-2413855JTB-A2A-ZM-241385
21.74Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
21.74Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
21.74Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
21.74Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
21.74Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
21.74Single6AQFZM-2413856AQF-A2A-ZM-241385
21.74Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
21.74Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
21.74Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
21.74Single6PS0S-Carazolol6PS0-β2-S-Carazolol
21.74Single6PS4ICI118-5516PS4-β2-ICI118-551
21.74Single6PS5S-Propranolol6PS5-β2-S-Propranolol
21.74Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
21.74Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
21.74Single6TPGEMPA6TPG-OX2-EMPA
21.74Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
21.74Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
21.74Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
21.74Single6ZG9GSK10347026ZG9-M1-GSK1034702
21.74Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
21.74Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
21.74Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
21.74Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
21.74Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
21.74Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
21.74Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
21.74Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single7T32ZM-2413857T32-A2A-ZM-241385
21.74Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
21.74Single7UL3Famotidine7UL3-H2-Famotidine
21.74Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
21.74Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
21.74Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
21.74Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.74Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
21.74Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
21.74Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
21.74Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
21.74Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
21.74Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
21.74Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
21.74Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
21.74Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
21.74Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
21.74Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
21.74Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
21.74Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
21.74Single8RLNLUF58348RLN-A2A-LUF5834
21.74Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
21.74Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.74Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.74Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
21.74Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
21.74Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
21.74Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
21.74Single9AS3LSD9AS3-5-HT2A-LSD
21.74Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single9AS5Mescaline9AS5-5-HT2A-Mescaline
21.74Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
21.74Single9BA0A1AKN9BA0-CB1-A1AKN
21.74Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
21.74Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
21.74Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
21.74Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
21.74Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
21.74Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
21.74Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
21.74Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
21.74Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
21.74Consensusa2_offOrthosteric Liganda2a_off
21.74Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
21.74Consensusalpha1_onOrthosteric Ligandalpha1a_on
21.74Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
21.74Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
21.74Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
21.74Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
21.74Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
21.74Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
21.74Consensushca_onOrthosteric Ligandhca2_on
21.74Consensusopsins_offOrthosteric Ligandrhodopsin_off
21.74Consensussensory_offOrthosteric Ligandopsins_off
21.43Single5WF6UK-4320975WF6-A2A-UK-432097
21.43Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
21.43Single6PT3DPI-2876PT3-δ-DPI-287
21.43Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
21.43Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.43Single7SK9CCX6627SK9-ACKR3-CCX662
21.43Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
21.43Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
21.43Single7XN9L-054,5227XN9-SST2-L-054,522
21.43Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
21.43Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
21.43Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
21.43Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
21.43Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
21.43Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
21.43Consensuskisspeptin_onOrthosteric Ligandkiss1_on
21.43Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
21.43Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
21.21Single6FJ3PTH6FJ3-PTH1-PTH
21.21Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
21.21Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
21.21Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
21.21Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
21.21Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
21.21Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
21.21Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
21.21Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
21.05Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
21.05Single8PWNTheophylline8PWN-A2A-Theophylline
21.05Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
20.83Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
20.83Single2Y01Dobutamine2Y01-β1-Dobutamine
20.83Single2Y04Salbutamol2Y04-β1-Salbutamol
20.83Single3EMLZM-2413853EML-A2A-ZM-241385
20.83Single3NY8ICI118-5513NY8-β2-ICI118-551
20.83Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
20.83Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
20.83Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
20.83Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
20.83Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
20.83Single4EJ4Naltrindole4EJ4-δ-Naltrindole
20.83Single4GBRS-Carazolol4GBR-β2-S-Carazolol
20.83Single4QIMANTA XV4QIM-SMO-ANTA XV
20.83Single4QKX35V4QKX-β2-35V
20.83Single5DHGC-355DHG-NOP-C-35
20.83Single5IU8Q274563475IU8-A2A-Q27456347-Na
20.83Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
20.83Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
20.83Single5TGZAM65385TGZ-CB1-AM6538
20.83Single5UIGCmpd-15UIG-A2A-Cmpd-1
20.83Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
20.83Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
20.83Single6H7MSalbutamol6H7M-β1-Salbutamol
20.83Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
20.83Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
20.83Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
20.83Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
20.83Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
20.83Single6S0LZM-2413856S0L-A2A-ZM-241385
20.83Single6TOTLemborexant6TOT-OX1-Lemborexant
20.83Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
20.83Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
20.83Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
20.83Single7PYRPSB-21157PYR-A2A-PSB-2115
20.83Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
20.83Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
20.83Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
20.83Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
20.83Single7WC7Lisuride7WC7-5-HT2A-Lisuride
20.83Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
20.83Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
20.83Single7YXAONO-54306087YXA-S1P5-ONO-5430608
20.83Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
20.83Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
20.83Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
20.83Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
20.83Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
20.83Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
20.83Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
20.83Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
20.83Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
20.83Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
20.83Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
20.83Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
20.83Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
20.83Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
20.83Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
20.83Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
20.83Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
20.83Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
20.83Single8JJOAlprenolol8JJO-β2-Alprenolol
20.83Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
20.83Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
20.83Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
20.83Single8T1WCVN4248T1W-GPR6-CVN424
20.83Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
20.83Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
20.83Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
20.83Single8X63Mepyramine8X63-H1-Mepyramine
20.83Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
20.83Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
20.83Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
20.83Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
20.83Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
20.83Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
20.83Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
20.83Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
20.83Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
20.83Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
20.83Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
20.83Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
20.83Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
20.83Consensusalpha2_onOrthosteric Ligandalpha2b_on
20.83Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
20.83Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
20.83Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
20.83Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
20.83Consensuscck_offOrthosteric Ligandccka_off
20.83Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
20.83Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
20.83Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
20.83Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
20.83Consensusdopamine_offOrthosteric Ligandd2_off d3_off
20.83Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
20.83Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
20.83Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
20.83Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
20.83Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
20.83Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
20.83Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
20.83Consensushca_on_gpOrthosteric Ligandhca2_on_gp
20.83Consensushistamine_offOrthosteric Ligandh1_off
20.69Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
20.69Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
20.69Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
20.69Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
20.69Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
20.69Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
20.69Single8IEBA1LYA8IEB-GPR156-A1LYA
20.69Single8KIGSHU91198KIG-MC3-SHU9119-Ca
20.69Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
20.69Single8XWNCXCL88XWN-CXCR2-CXCL8
20.69Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
20.69Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.69Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
20.69Single9M4TSilodosin9M4T-Alpha1A-Silodosin
20.69Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
20.69Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.69Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
20.69Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
20.59Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
20.59Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
20.59Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
20.59Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
20.59Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
20.59Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
20.59Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
20.59Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
20.51Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
20.00Single2RH1S-Carazolol2RH1-β2-S-Carazolol
20.00Single2Y00Dobutamine2Y00-β1-Dobutamine
20.00Single2Y03Isoprenaline2Y03-β1-Isoprenaline
20.00Single2YCWS-Carazolol2YCW-β1-S-Carazolol
20.00Single3OE8IT1t3OE8-CXCR4-IT1t
20.00Single3RFMCaffeine3RFM-A2A-Caffeine
20.00Single5D6LS-Carazolol5D6L-β2-S-Carazolol
20.00Single5IUAQ274563485IUA-A2A-Q27456348-Na
20.00Single5WIUNemonapride5WIU-D4-Nemonapride
20.00Single5WIVNemonapride5WIV-D4-Nemonapride-Na
20.00Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
20.00Single5XPRBosentan5XPR-ETB-Bosentan
20.00Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
20.00Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
20.00Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
20.00Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
20.00Single6HLOAprepitant6HLO-NK1-Aprepitant
20.00Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
20.00Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
20.00Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
20.00Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
20.00Single6PS6Timolol6PS6-β2-Timolol
20.00Single6S0QZM-2413856S0Q-A2A-ZM-241385
20.00Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
20.00Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
20.00Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
20.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
20.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
20.00Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
20.00Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
20.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.00Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
20.00Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
20.00Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
20.00Single7W41PD1762527W41-BB2-PD176252
20.00Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
20.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
20.00Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
20.00Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GNEKW-63568GNE-A2A-KW-6356-Na
20.00Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
20.00Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
20.00Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
20.00Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
20.00Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
20.00Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.00Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
20.00Single8QOTNanobody-E8QOT-μ-Nanobody-E
20.00Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
20.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
20.00Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
20.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
20.00Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
20.00Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
20.00Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
20.00Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
20.00Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
20.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9CHUNoradrenaline9CHU-β2-Noradrenaline
20.00Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
20.00Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
20.00Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
20.00Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
20.00Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
20.00Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
20.00Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
20.00Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
20.00Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
20.00Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
20.00Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
20.00Consensusamine_offonOrthosteric Ligandamine_off amine_on
20.00Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
20.00Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
20.00Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
20.00Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
20.00Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
20.00Consensusbombesin_offOrthosteric Ligandbb2_off
20.00Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
20.00Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
20.00Consensusep_offOrthosteric Ligandep4_off
20.00Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
20.00Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
20.00Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
20.00Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.00Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
20.00Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
20.00Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
20.00Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Consensustrace-amine_onOrthosteric Ligandta1_on
19.51Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
19.44Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
19.35Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
19.35Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
19.35Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
19.35Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
19.35Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
19.35Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.35Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
19.23Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
19.23Single4BV0Neurotensin4BV0-NTS1-Neurotensin
19.23Single5D5AS-Carazolol5D5A-β2-S-Carazolol
19.23Single5D5BS-Carazolol5D5B-β2-S-Carazolol
19.23Single5TZRMK86665TZR-FFA1-MK8666
19.23Single5V56TC1145V56-SMO-TC114
19.23Single5XR8AM8415XR8-CB1-AM841
19.23Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
19.23Single6J21Aprepitant6J21-NK1-Aprepitant
19.23Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
19.23Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
19.23Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
19.23Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
19.23Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
19.23Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
19.23Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
19.23Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
19.23Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
19.23Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
19.23Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
19.23Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.23Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
19.23Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
19.23Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
19.23Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
19.23Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
19.23Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
19.23Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
19.23Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
19.23Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
19.23Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
19.23Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
19.23Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
19.23Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
19.23Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Consensusa2_onOrthosteric Liganda2b_on
19.23Consensusa2_on_gpOrthosteric Liganda2b_on_gp
19.23Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
19.23Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
19.23Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
19.23Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
19.23Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
19.23Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
19.23Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
19.23Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
19.23Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
19.23Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
19.23Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
19.23Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
19.23Consensusneurotensin_onOrthosteric Ligandnts1_on
19.23Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
19.23Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.23Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
19.05Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
19.05Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
19.05Single6ME5Agomelatine6ME5-MT1-Agomelatine
19.05Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
19.05Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
19.05Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
19.05Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
19.05Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
19.05Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.05Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
19.05Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
19.05Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
19.05Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
19.05Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
19.05Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
19.05Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
19.05Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
19.05Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
19.05Single9LRCHistamine9LRC-H4-Histamine
19.05Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
19.05Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
19.05Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
19.05Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
19.05Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
18.92Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
18.92Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
18.92Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
18.92Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
18.75Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
18.75Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
18.75Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
18.75Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
18.75Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
18.75Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
18.75Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.75Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.75Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
18.75Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
18.75Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
18.52Single3D4STimolol3D4S-β2-Timolol
18.52Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
18.52Single4N4WSANT-14N4W-SMO-SANT-1
18.52Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
18.52Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
18.52Single4XEENeurotensin4XEE-NTS1-Neurotensin
18.52Single4XESNeurotensin4XES-NTS1-Neurotensin
18.52Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
18.52Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
18.52Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
18.52Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
18.52Single6YVRNTS8-136YVR-NTS1-NTS8-13
18.52Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
18.52Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
18.52Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
18.52Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
18.52Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
18.52Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
18.52Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
18.52Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
18.52Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
18.52Single8JWY2-1188JWY-A2A-2-118
18.52Single8JWZAB9288JWZ-A2A-AB928-Na
18.52Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
18.52Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
18.52Single8XWACXCL18XWA-CXCR2-CXCL1
18.52Single8XWSCXCL58XWS-CXCR2-CXCL5
18.52Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
18.52Single8XYIVUF106618XYI-CXCR3-VUF10661
18.52Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
18.52Single9BJKNAM9BJK-μ-Naloxone-NAM
18.52Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
18.52Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
18.52Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
18.52Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
18.52Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
18.52Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
18.42Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
18.42Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
18.42Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
18.42Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
18.42Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.42Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
18.42Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
18.18Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
18.18Single3PBLEticlopride3PBL-D3-Eticlopride
18.18Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
18.18Single6HLLCP999946HLL-NK1-CP99994
18.18Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
18.18Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
18.18Single6TP4ACT-4622066TP4-OX1-ACT-462206
18.18Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
18.18Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
18.18Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
18.18Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
18.18Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
18.18Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
18.18Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
18.18Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
18.18Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
18.18Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
18.18Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
18.18Single8K5BNiacin8K5B-HCA2-Niacin
18.18Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
18.18Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
18.18Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
18.18Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
18.18Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
18.18Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
18.18Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
18.18Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
18.18Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
18.18Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
18.18Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
18.18Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
18.18Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
18.18Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
18.18Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
17.95Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
17.95Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
17.95Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Single4BUONeurotensin4BUO-NTS1-Neurotensin
17.86Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
17.86Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
17.86Single6K1QIRL25006K1Q-ETB-IRL2500
17.86Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
17.86Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
17.86Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
17.86Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
17.86Single7UM4AS26747237UM4-5-HT5A-AS2674723
17.86Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
17.86Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
17.86Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
17.86Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
17.86Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
17.86Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8XWFCXCL38XWF-CXCR2-CXCL3
17.86Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
17.86Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
17.86Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
17.86Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
17.86Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.86Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.78Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
17.65Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
17.65Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
17.65Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
17.65Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
17.65Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
17.65Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
17.65Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
17.50Consensuspth_onOrthosteric Ligandpth1_on pth2_on
17.39Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
17.39Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
17.39Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
17.39Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
17.39Single6B73MP11046B73-κ-MP1104
17.39Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
17.39Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
17.39Single6ME9Ramelteon6ME9-MT2-Ramelteon
17.39Single6TODEMPA6TOD-OX1-EMPA-Na
17.39Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
17.39Single7F8YDevazepide7F8Y-CCKA-Devazepide
17.39Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
17.39Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
17.39Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
17.39Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
17.39Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
17.39Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
17.39Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
17.39Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
17.39Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
17.39Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
17.39Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
17.39Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
17.39Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
17.39Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
17.39Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
17.39Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
17.39Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
17.39Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
17.39Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
17.39Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
17.39Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
17.39Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
17.39Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
17.39Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
17.39Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
17.39Single8IWESpermidine8IWE-TA9-Spermidine
17.39Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
17.39Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.39Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
17.39Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
17.39Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
17.39Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
17.39Single8Y0HVUF114188Y0H-CXCR3-VUF11418
17.39Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
17.39Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
17.39Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
17.39Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
17.39Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
17.39Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
17.39Single9H2XA1IR19H2X-A2A-A1IR1-Na
17.39Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
17.39Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
17.39Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
17.39Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
17.39Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
17.39Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
17.39Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
17.39Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
17.39Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
17.39Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
17.39Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
17.24Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
17.24Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
17.24Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
17.24Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
17.24Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
17.24Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
17.24Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
17.24Single9JF4PD1683689JF4-BB1-PD168368
17.24Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
17.24Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
17.14Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
17.14Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
17.14Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
17.14Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
17.14Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
17.14Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
17.14Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
16.67Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
16.67Single3REYXAC3REY-A2A-XAC
16.67Single3RZECidoxepin3RZE-H1-Cidoxepin
16.67Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
16.67Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
16.67Single5UVIZM-2413855UVI-A2A-ZM-241385
16.67Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
16.67Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
16.67Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
16.67Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
16.67Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
16.67Single6TPKRetosiban6TPK-OT-Retosiban
16.67Single6TPNHTL66416TPN-OX2-HTL6641
16.67Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
16.67Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
16.67Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
16.67Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
16.67Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
16.67Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
16.67Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
16.67Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
16.67Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
16.67Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
16.67Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
16.67Single7QA8Peptide7QA8-STE2-Peptide
16.67Single7QA8Peptide7QA8-STE2-Peptide
16.67Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
16.67Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
16.67Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
16.67Single7VODCariprazine7VOD-5-HT2A-Cariprazine
16.67Single7VV6C48/807VV6-MRGPRX2-C48/80
16.67Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
16.67Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
16.67Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
16.67Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
16.67Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
16.67Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
16.67Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
16.67Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
16.67Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
16.67Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
16.67Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
16.67Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
16.67Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
16.67Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
16.67Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
16.67Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
16.67Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
16.67Single8K2WAMG4878K2W-CXCR3-AMG487
16.67Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
16.67Single8K5CAcipimox8K5C-HCA2-Acipimox
16.67Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
16.67Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
16.67Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
16.67Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
16.67Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
16.67Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
16.67Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
16.67Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
16.67Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
16.67Single8ZPNAMD31008ZPN-CXCR4-AMD3100
16.67Single9ARXSerotonin9ARX-5-HT2A-Serotonin
16.67Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
16.67Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
16.67Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
16.67Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
16.67Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
16.67Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
16.67Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
16.67Consensusvasop-oxy_offOrthosteric Ligandot_off
16.67Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
16.67Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
16.22Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
16.22Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
16.22Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
16.13Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
16.13Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
16.13Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
16.13Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
16.13Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
16.00Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
16.00Single4DAJTiotropium4DAJ-M3-Tiotropium
16.00Single4MQSIperoxo4MQS-M2-Iperoxo
16.00Single4U14Tiotropium4U14-M3-Tiotropium
16.00Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
16.00Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
16.00Single5T04Neurotensin5T04-NTS1-Neurotensin
16.00Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
16.00Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
16.00Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
16.00Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
16.00Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
16.00Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
16.00Single6GPSMK08126GPS-CCR2-MK0812
16.00Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
16.00Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
16.00Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
16.00Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
16.00Single7F83PF-051904577F83-Ghrelin-PF-05190457
16.00Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
16.00Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
16.00Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
16.00Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
16.00Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
16.00Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
16.00Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
16.00Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
16.00Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
16.00Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
16.00Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
16.00Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
16.00Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
16.00Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
16.00Single8K5DGSK2560738K5D-HCA2-GSK256073
16.00Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
16.00Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
16.00Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
16.00Single8X64Desloratadine8X64-H1-Desloratadine
16.00Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
16.00Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
16.00Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
16.00Single9AS1DMT9AS1-5-HT2A-DMT
16.00Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
16.00Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
16.00Single9JEAAtropine9JEA-M1-Atropine
16.00Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
16.00Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
16.00Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
16.00Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
16.00Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
16.00Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
16.00Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
16.00Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
16.00Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
16.00Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
16.00Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
16.00Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
15.91Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
15.79Single5MZPCaffeine5MZP-A2A-Caffeine-Na
15.79Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
15.79Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
15.62Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
15.62Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
15.38Single4JKVTaladegib4JKV-SMO-Taladegib
15.38Single4NTJAZD12834NTJ-P2Y12-AZD1283
15.38Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
15.38Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
15.38Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
15.38Single6GPXMK08126GPX-CCR2-MK0812
15.38Single6HLPNetupitant6HLP-NK1-Netupitant
15.38Single6LUQHaloperidol6LUQ-D2-Haloperidol
15.38Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
15.38Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
15.38Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
15.38Single7SINNPS-21437SIN-CaS-NPS-2143
15.38Single7SINNPS-21437SIN-CaS-NPS-2143
15.38Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
15.38Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
15.38Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.38Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
15.38Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
15.38Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
15.38Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
15.38Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
15.38Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
15.38Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
15.38Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
15.38Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
15.38Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
15.38Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
15.38Consensusblt_offOrthosteric Ligandblt1_off
15.38Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
15.38Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
15.38Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
15.38Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
15.38Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
15.38Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
15.38Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
15.15Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
15.15Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
15.15Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
15.15Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
15.15Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
15.15Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
15.00Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
15.00Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
15.00Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
15.00Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
15.00Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
15.00Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
14.81Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
14.81Single4U15Tiotropium4U15-M3-Tiotropium
14.81Single5V57TC1145V57-SMO-TC114
14.81Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
14.81Single6E59L-7607356E59-NK1-L-760735
14.81Single6J20Aprepitant6J20-NK1-Aprepitant
14.81Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
14.81Single6OL9Tiotropium6OL9-M5-Tiotropium
14.81Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
14.81Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
14.81Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
14.81Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
14.81Single8EA0Iperoxo8EA0-M3-Iperoxo
14.81Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.81Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
14.81Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
14.81Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
14.81Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
14.81Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
14.81Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
14.81Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
14.81Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.81Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
14.81Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
14.81Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
14.81Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
14.81Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
14.81Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
14.81Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
14.81Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
14.81Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
14.81Consensusrelaxin_onOrthosteric Ligandrxfp4_on
14.81Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
14.81Consensustachykinin_offOrthosteric Ligandnk1_off
14.71Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
14.63Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
14.29Single4PY02MeSATP4PY0-P2Y12-2MeSATP
14.29Single5CXVTiotropium5CXV-M1-Tiotropium
14.29Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
14.29Single6IIURamatroban6IIU-TXA2-Ramatroban
14.29Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
14.29Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
14.29Single6TQ9SB-4081246TQ9-OX1-SB-408124
14.29Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
14.29Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
14.29Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
14.29Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
14.29Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
14.29Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
14.29Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
14.29Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
14.29Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
14.29Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
14.29Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
14.29Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
14.29Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
14.29Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
14.29Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8XWMCXCL68XWM-CXCR2-CXCL6
14.29Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
14.29Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
14.29Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
14.29Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
14.29Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
14.29Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
14.29Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
14.29Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
14.29Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
14.29Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
14.29Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
14.29Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
14.29Consensusp2y_offOrthosteric Ligandp2y1_off
14.29Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
13.95Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
13.89Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
13.89Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
13.89Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
13.89Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
13.89Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
13.89Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
13.79Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
13.79Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
13.79Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
13.79Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Single8XVJMacitentan8XVJ-ETA-Macitentan
13.79Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
13.79Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
13.79Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
13.79Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single3UZAGTPL92363UZA-A2A-GTPL9236
13.64Single4XNWMRS25004XNW-P2Y1-MRS2500
13.64Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
13.64Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
13.64Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
13.64Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.64Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.64Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
13.64Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
13.64Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
13.64Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
13.64Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
13.64Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
13.64Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
13.51Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
13.51Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
13.51Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
13.33Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
13.33Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
13.33Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
13.33Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
13.33Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
13.16Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
13.04Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
13.04Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
13.04Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
13.04Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
13.04Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
13.04Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
13.04Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
13.04Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
13.04Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
13.04Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
13.04Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
13.04Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
13.04Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
13.04Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
13.04Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
13.04Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
13.04Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
13.04Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.04Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
13.04Single9AS7Psilocin9AS7-5-HT2A-Psilocin
13.04Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
13.04Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
13.04Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
13.04Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
12.90Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
12.90Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single8IEIA1LYA8IEI-GPR156-A1LYA
12.90Single8IEIA1LYA8IEI-GPR156-A1LYA
12.90Single8IEPA1LYA8IEP-GPR156-A1LYA
12.90Single8IEPA1LYA8IEP-GPR156-A1LYA
12.90Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
12.82Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
12.82Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
12.50Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
12.50Single4BWBNeurotensin4BWB-NTS1-Neurotensin
12.50Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
12.50Single6ME2Ramelteon6ME2-MT1-Ramelteon
12.50Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.50Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
12.50Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
12.50Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.50Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
12.50Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
12.50Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
12.50Single7XNACYN1548067XNA-SST2-CYN154806
12.50Single8IEBA1LYA8IEB-GPR156-A1LYA
12.50Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
12.50Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
12.50Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
12.50Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
12.50Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
12.50Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
12.50Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.50Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
12.50Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
12.50Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
12.20Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
12.20Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
12.20Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
12.20Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
12.12Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
12.00Single6A94Zotepine6A94-5-HT2A-Zotepine
12.00Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
12.00Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
12.00Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
12.00Single6ZINSR486926ZIN-NTS1-SR48692
12.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
12.00Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
12.00Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
12.00Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.00Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
12.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
12.00Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
12.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
12.00Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
11.90Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
11.76Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
11.76Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
11.76Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
11.63Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
11.54Single5DSGTiotropium5DSG-M4-Tiotropium
11.54Single6IIVDaltroban6IIV-TXA2-Daltroban
11.54Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
11.54Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
11.54Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
11.54Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
11.54Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
11.54Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.54Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
11.54Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
11.54Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
11.54Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
11.54Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
11.54Single9IYAONO-97105319IYA-GPR55-ONO-9710531
11.54Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
11.54Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
11.54Consensusblt_onOrthosteric Ligandblt1_on
11.54Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
11.54Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
11.54Consensusleukotriene_onOrthosteric Ligandblt_on
11.54Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
11.54Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
11.43Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
11.43Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
11.43Consensuscalcitonin_onOrthosteric Ligandctlike_on
11.11Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
11.11Single5CGCHTL142425CGC-mGlu5-HTL14242
11.11Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
11.11Single6Z4SSR486926Z4S-NTS1-SR48692
11.11Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
11.11Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
11.11Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
11.11Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
11.11Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
11.11Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
11.11Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
11.11Single8ZMFA1L108ZMF-5-HT2C-A1L10
11.11Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
11.11Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
11.11Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
11.11Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
11.11Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
10.87Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
10.81Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
10.81Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
10.71Single5V54Methiothepin5V54-5-HT1B-Methiothepin
10.71Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
10.71Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
10.71Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
10.71Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
10.71Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
10.71Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
10.71Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
10.71Single9AS9RS130-1809AS9-5-HT2A-RS130-180
10.71Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Consensus5ht1_offOrthosteric Ligand5ht1b_off
10.71Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
10.71Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
10.53Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
10.53Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
10.53Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
10.34Single5X33BIIL2605X33-BLT1-BIIL260
10.34Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
10.34Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
10.00Single5CGDHTL142425CGD-mGlu5-HTL14242
10.00Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
10.00Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
10.00Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
10.00Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
9.68Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
9.52Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
9.52Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
9.52Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
9.38Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
9.38Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
9.38Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
9.38Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
9.38Consensussomatostatin_offOrthosteric Ligandsst2_off
9.09Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
9.09Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
9.09Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
9.09Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
9.09Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
9.09Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
9.09Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
9.09Consensussensory_onOrthosteric Ligandopsins_on
8.70Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
8.70Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
8.70Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
8.70Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
8.70Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
8.70Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
8.70Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
8.70Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
8.70Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.70Single8JPSCCL78JPS-ACKR1-CCL7
8.70Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
8.70Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
8.70Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
8.70Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.70Consensusgi_sensoryOrthosteric Ligandgi_opsins
8.70Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.70Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
8.70Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
8.70Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
8.70Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
8.57Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
8.57Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
8.57Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
8.33Single4O9RCyclopamine4O9R-SMO-Cyclopamine
8.33Single5L7IVismodegib5L7I-SMO-Vismodegib
8.33Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
8.33Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.33Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
8.33Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
8.33Consensusgq_nucleotideOrthosteric Ligandgq_p2y
8.33Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
8.11Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
8.11Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
8.00Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
8.00Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
8.00Single4QINSAG1.54QIN-SMO-SAG1.5
8.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
8.00Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
8.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
8.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
8.00Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
7.89Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
7.69Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
7.69Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
7.69Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
7.69Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
7.50Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
7.41Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
7.41Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
7.14Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
7.14Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
7.14Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
7.14Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
7.14Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
7.14Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
7.14Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
7.14Single9HC04YI9HC0-mGlu5-4YI
7.14Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
6.90Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
6.90Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
6.90Single7P2L4YI7P2L-mGlu5-4YI
6.90Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
6.90Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
6.90Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
6.45Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.56Single6D35Cholesterol6D35-SMO-Cholesterol
5.56Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.56Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.56Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
5.56Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
5.56Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
5.56Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
5.56Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
5.56Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
5.56Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
5.56Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
5.56Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.56Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
5.56Single7DTTCa7DTT-CaS-Ca-Ca
5.56Single7DTTCa7DTT-CaS-Ca-Ca
5.56Single7DTUTryptophan7DTU-CaS-Tryptophan
5.56Single7DTUTryptophan7DTU-CaS-Tryptophan
5.56Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.56Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.56Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.56Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.56Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.56Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.56Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.56Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.56Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
5.56Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.56Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.56Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.56Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.56Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.56Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.56Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
5.56Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
5.56Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.56Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.56Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.56Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.56Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.56Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.56Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.56Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.56Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.56Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.56Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.56Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.56Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.56Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.56Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.56Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.56Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
5.56Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.56Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.56Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.56Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.56Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.56Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.56Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
5.56Single7XW7K1-707XW7-TSH-K1-70
5.56Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.56Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.56Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.56Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.56Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.56Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.56Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.56Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.56Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.56Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.56Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.56Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.56Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
5.56Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.56Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.56Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.56Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.56Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.56Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.56Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.56Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.56Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.56Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.56Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.56Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.56Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.56Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.56Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
5.56Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.56Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.56Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.56Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.56Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.56Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.56Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.56Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.56Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.56Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.56Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.56Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.56Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.56Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.56Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.56Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.56Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
5.56Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
5.56Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
5.56Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
5.56Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
5.56Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
5.56Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.56Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.56Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.56Single8WVXNorrin8WVX-LGR4-Norrin
5.56Single8WVYNorrin8WVY-LGR4-Norrin
5.56Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.56Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.56Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.56Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.56Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.56Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.56Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.56Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
5.56Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.56Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.56Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.56Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.56Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.56Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.56Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.56Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.56Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.56Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.56Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.56Single9KHHNorrin9KHH-LGR4-Norrin
5.56Single9S37NB219S37-LGR4-NB21
5.56Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
5.26Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.26Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.26Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.26Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
5.26Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.26Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.26Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.26Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
5.26Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.26Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.26Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.26Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.26Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
5.26Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
5.26Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
5.00Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
5.00Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
5.00Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
5.00Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
4.76Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
4.76Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
4.76Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.76Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.76Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.76Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.76Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.76Single8JGBConorfamide-Tx28JGB-MRGPRX1-Conorfamide-Tx2-Gi1/β1/γ2
4.55Single5L7DCholesterol5L7D-SMO-Cholesterol
4.55Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.55Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
4.55Single8HS2Fab0468HS2-GPR20-Fab046
4.55Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.35Single7Y14Beta-Alanine7Y14-MRGPRD-β-Alanine
4.17Single7Y12Beta-Alanine7Y12-MRGPRD-β-Alanine-Gi1/β1/γ2
4.17Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
4.00Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
4.00Single7UL2SR486927UL2-NTS1-SR48692-Na
4.00Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
4.00Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.00Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
4.00Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
4.00Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
4.00Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
4.00Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
4.00Consensusneurotensin_offOrthosteric Ligandnts1_off
4.00Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
3.85Single4XNVBPTU4XNV-P2Y1-BPTU
3.85Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
3.85Single7WV9ZCZ0117WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
3.70Single6FFIMMPEP6FFI-mGlu5-MMPEP
3.70Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.70Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single8IYXYL-3658IYX-GPR34-YL-365
3.57Single6FFHFenobam6FFH-mGlu5-Fenobam
3.45Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.33Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.33Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
2.94Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.94Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.78Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.78Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.70Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.50Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
8KFX 8KFX-CCR8-LMD-009-Gi1/β1/γ2
8KFY 8KFY-CCR8-ZK-756326-Gi1/β1/γ2
8U1U 8U1U-CCR8-CCL1-Gi1/β1/γ2
Net Summary
Imin 2.96333
Number of Linked Nodes 905
Number of Links 1139
Number of Hubs 202
Number of Links mediated by Hubs 739
Number of Communities 27
Number of Nodes involved in Communities 287
Number of Links involved in Communities 427
Path Summary
Number Of Nodes in MetaPath 93
Number Of Links MetaPath 92
Number of Shortest Paths 1709042
Length Of Smallest Path 3
Average Path Length 43.8974
Length of Longest Path 78
Minimum Path Strength 0.701667
Average Path Strength 5.86468
Maximum Path Strength 24.4733
Minimum Path Correlation 0.71
Average Path Correlation 0.983676
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.47059
Average % Of Corr. Nodes 35.691
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 53.9065
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
ccr_on_gpccr6_on_gp
ccr8_on_gp
ccr2_on_gp
ccr1_on_gp
ccr5_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download ccr8_on_gp.zip



You can click to copy the link of this page to easily come back here later

or use this QR code to link and share this page.



You can also  read or  download a guide explaining the meaning of all files and numerical data.