Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 1.52055503
2G.HN.37 2.18094402
3G.HN.52 1.82622404
4G.S1.02 5.01251544
5G.S1.05 5.24502409
6G.S1.06 3.65357548
7G.S1.07 3.92177409
8G.S2.03 5.25684418
9G.S2.05 6.28691413
10G.S2.08 7.05363445
11G.S3.03 7.44379547
12G.S3.04 7.04216516
13G.S3.06 8.11688516
14G.S3.07 4.63633449
15G.s3h2.03 4.4256519
16G.H2.06 4.93342719
17G.H2.07 4.65508719
18G.H2.09 6.01885418
19G.h2s4.01 6.18467519
20G.S4.03 3.49076447
21G.S4.04 5.18145589
22G.s4h3.04 4.57556678
23G.H3.01 5.63624409
24G.H3.09 5.64502689
25G.H3.13 3.94914585
26G.H3.14 5.45483408
27G.H3.17 5.97563614
28G.H3.18 5.811164179
29G.S5.03 3.04367448
30G.S5.04 3.62472589
31G.S5.05 3.61525849
32G.S5.07 3.79905449
33G.HG.03 3.30134476
34G.HG.04 5.25805578
35G.HG.07 3.89897479
36G.HG.14 2.63746405
37G.hgh4.01 4.12139474
38G.hgh4.02 5.24286778
39G.hgh4.05 6.81668406
40G.H4.03 6.48673403
41G.H4.10 8.46751476
42G.H4.12 5.96367485
43G.H4.15 4.83399488
44G.h4s6.02 5.03471487
45G.S6.02 6.098355138
46G.S6.04 7.77796448
47G.s6h5.01 4.79357549
48G.H5.03 5.14205448
49G.H5.08 5.39939448
50G.H5.20 3.47595508
51G.H5.25 4.22556406
52G.H5.26 5.08183505
53b.1x4 1.66452608
54b.h2x1 2.88609405
55b.lhb1x3 2.35278502
56b.b1x4 3.75531457
57b.b1x6 7.84562459
58b.l1x3 7.23321759
59b.b2x1 7.93548518
60b.b2x5 6.5056607
61b.l3x2 4.64184559
62b.b4x2 4.35988408
63b.b4x3 4.231954147
64b.b4x5 4.07784107
65b.b4x6 8.6491759
66b.l4x2 11.1591454
67b.b5x2 5.13624407
68b.b5x3 6.31767659
69b.b5x5 5.149694105
70b.b5x7 5.42452407
71b.l5x1 4.001925148
72b.l5x5 6.61439719
73b.b6x5 3.794867106
74b.l6x5 5.400364154
75b.b7x1 5.364115154
76b.b7x4 3.398514148
77b.l7x2 3.32284619
78b.l7x4 3.30501409
79b.b8x4 5.308275146
80b.l8x1 3.779374105
81b.l8x3 3.45915403
82b.l9x3 5.72799719
83b.l9x6 4.293181018
84b.b10x5 4.21133609
85b.l10x1 4.31375403
86b.b11x4 4.75042519
87b.l11x2 8.38273419
88b.b12x3 3.34332468
89b.b12x6 7.32061718
90b.b13x7 7.6815567
91b.l13x3 7.08644669
92b.l13x6 4.71835519
93b.l13x7 4.13746469
94b.b14x3 4.0679465
95b.b15x1 5.62023769
96b.b15x2 7.0156416
97b.b15x3 4.53848469
98b.l15x1 5.26659417
99b.l15x2 5.17218569
100b.b16x4 10.0758466
101b.b16x5 4.24318515
102b.b16x6 8.105668
103b.b17x4 5.07231415
104b.b17x5 6.58449417
105b.b17x7 7.87703418
106b.l17x3 7.39972719
107b.l17x6 6.01925519
108b.b18x3 4.89356418
109b.b18x5 5.17458405
110b.l18x1 5.580168126
111b.l18x2 5.478734127
112b.l18x3 7.23374125
113b.b19x2 6.10158716
114b.b19x4 5.31763518
115b.l19x2 5.27478519
116b.b20x2 4.57391516
117b.b20x4 10.4061518
118b.b20x6 7.27186516
119b.b20x7 4.46406409
120b.l20x2 5.05936509
121b.b21x1 6.32304517
122b.b21x2 2.80175406
123b.b21x5 5.07783404
124b.b21x7 5.97432505
125b.b22x5 4.50046127
126b.l22x5 5.21229799
127b.b23x1 3.4889405
128b.b23x6 7.210016167
129b.l23x1 7.51405406
130b.b24x4 8.193054166
131b.b24x6 7.117234168
132b.b24x7 7.49481499
133b.l24x2 3.92392496
134b.l24x3 3.64602595
135b.l25x3 8.696135119
136b.b26x3 4.15291406
137b.b27x1 2.80737406
138b.l27x1 10.2805719
139b.l27x2 7.032354119
140b.b28x3 3.86289557
141b.b28x4 7.953334116
142b.b28x6 9.751984119
143g.h1x1 0.628942502
144g.h1x8 2.4204407
145g.l1x4 3.49806508
146g.h2x11 9.196224126
147g.ctx3 5.560696199
148g.ctx5 3.48474199
149g.ctx6 3.1712506
150g.ctx14 4.95959459
151g.ctx15 6.26204459
152g.ctx16 4.77902758
153Lig 36.3222320
154NT 18.0456523
1551x30 2.29837405
1561x35 4.38729405
1571x39 4.72217528
1581x50 5.79431409
1591x57 3.15868407
1601x59 2.82796404
1612x38 4.76656436
1622x42 4.99244637
1632x46 3.89195439
1642x50 6.17899439
1652x53 5.71923426
166E1x50 7.62695528
167E1x52 4.59554607
1683x32 5.41699627
1693x33 4.40792405
1703x37 4.09926537
1713x42 5.23902437
1723x49 6.38561438
1733x50 5.68889539
1743x51 6.849424228
175I2x52 2.82399404
1764x41 1.301402
1774x50 5.12976439
178E2 14.34091424
179E2x52 4.67654425
1805x47 5.37698408
1815x50 2.99103409
1825x58 5.79839739
183I3 4.539784134
1846x30 1.9916407
1856x44 4.27721539
1866x48 7.01634539
1876x49 3.62916406
1886x51 5.47618527
189E3 3.92959724
1907x42 5.34732527
1917x43 2.11672405
1927x45 5.97647539
1937x49 4.71835639
1947x52 2.62265438
1957x53 4.96292639
1968x50 5.725435218
1978x54 2.06978406
198I2x57 5.17385430
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b2x3 b.b2x5 24.40214.58983NoYes067
2b.b26x2 b.b2x3 24.59744.9005NoNo076
3b.b26x1 b.b26x2 24.79743.01NoNo097
4b.b26x1 b.l27x1 24.9995.15725NoYes099
5b.b2x1 b.l27x1 16.39336.83213YesYes189
6b.b2x1 b.l3x1 16.757814.9916YesNo189
7b.l3x1 b.l5x5 17.09525.37246NoYes199
8G.h2s4.01 b.l5x5 12.974910.4911YesYes199
9G.S1.05 G.h2s4.01 14.86649.581YesYes099
10G.S1.05 G.S1.07 50.64345.64667YesYes099
11G.S1.07 G.S4.04 50.74813.01725YesYes099
12G.S4.04 G.S5.04 94.60982.99938YesYes899
13G.S5.04 G.S5.06 94.93253.57025YesNo098
14G.S5.06 G.s4h3.01 95.35265.89921NoNo087
15G.HG.04 G.s4h3.01 96.374210.3763YesNo087
16G.H4.03 G.HG.04 98.96973.10046YesYes038
17G.H4.03 G.HG.01 99.76827.21925YesNo035
18G.HG.01 G.s6h5.02 99.7864.70079NoNo057
19G.s6h5.02 G.s6h5.05 99.80372.82667NoNo079
20G.s6h5.01 G.s6h5.05 99.89062.31325YesNo099
21G.S5.05 G.s6h5.01 99.57685.70583YesYes499
22G.S4.03 G.S5.05 99.43093.13917YesYes479
23G.S1.04 G.S4.03 1005.38204NoYes477
24G.S1.02 G.S1.04 49.91733.02346YesNo447
25G.H5.11 G.S1.02 49.5965.13033NoYes484
26G.H5.11 G.H5.15 99.66842.32875NoNo088
27G.H5.15 G.H5.19 99.48012.47908NoNo088
283x53 G.H5.19 99.38583.86NoNo088
293x53 I2x57 99.29133.688NoYes080
302x38 I2x57 49.6955.98825YesYes360
312x38 2x42 49.06574.08217YesYes367
32G.H3.17 b.l27x1 11.6672.81633YesYes149
33G.H3.15 G.H3.17 38.33494.11696NoYes084
34G.H3.15 G.H3.18 38.43084.14767NoYes089
35G.H3.18 G.S4.02 35.60857.87925YesNo1797
36G.S1.05 G.S4.02 35.77253.69125YesNo097
37G.S1.04 G.S3.03 50.09573.11217NoYes477
38G.H5.11 G.S3.03 50.16634.42125NoYes487
393x49 I2x57 49.31248.82492YesYes380
402x42 3x49 49.08496.63646YesYes378
41b.b2x4 b.b6x5 11.35422.943NoYes066
42b.b10x4 b.b2x4 11.443114.329NoNo066
43b.b10x2 b.b10x4 10.9644.49804NoNo066
44b.b10x2 b.b14x3 10.50414.40475NoYes065
45b.b11x5 b.b14x3 13.06245.34833NoYes065
46b.b10x1 b.b11x5 16.98433.423NoNo096
47b.b10x1 b.l9x6 17.09723.2585NoYes098
482x42 3x46 90.15244.3805YesNo379
493x46 3x50 31.09853.005NoYes399
503x50 5x58 14.72457.01771YesYes399
51G.H2.07 b.l9x6 50.6373.29925YesYes198
52G.H2.06 b.l9x6 37.01713.10275YesYes198
53G.H2.04 G.H2.07 48.80244.5125NoYes099
54G.H2.04 G.H3.08 48.85484.72463NoNo099
55G.H2.06 b.l17x6 36.34347.22633YesYes199
56G.H5.20 G.H5.25 14.11843.23438YesYes086
573x50 G.H5.25 16.93668.97321YesYes096
58G.H5.20 G.H5.26 11.19155.24617YesYes085
59b.l17x5 b.l17x6 37.25994.35504NoYes169
60b.l17x5 b.l19x2 37.1763.398NoYes169
61b.l17x3 b.l19x2 28.83633.36625YesYes199
62b.b19x4 b.l17x3 20.88327.69933YesYes189
63b.b19x2 b.b19x4 10.96972.59YesYes168
64b.b17x7 b.b21x1 26.93294.23388YesYes187
65b.1x19 b.b21x1 22.91116.71958NoYes067
66b.1x15 b.1x19 20.37513.06296NoNo076
67b.1x12 b.1x15 18.3111.7545NoNo067
68b.1x12 g.h1x11 17.79471.79775NoNo069
69b.1x11 g.h1x11 16.76183.55917NoNo089
70b.1x11 g.h1x12 16.24522.068NoNo086
71g.h1x12 g.h1x8 14.17782.15842NoYes067
72b.b17x7 b.b20x6 21.29938.64383YesYes186
73b.b20x4 b.b20x6 14.45294.50346YesYes186
74g.ctx3 g.ctx6 13.20866.88921YesYes096
75b.l22x5 g.ctx6 13.20743.37471YesYes096
76b.l23x1 b.l25x6 29.266618.339YesNo068
77b.l21x7 b.l23x1 13.63875.04233NoYes056
78b.l21x7 b.l23x2 13.49456.18283NoNo058
79b.b23x6 b.l23x2 12.77334.33646YesNo078
80b.b23x6 b.b24x6 11.03397.36325YesYes1678
81b.b22x1 b.l23x1 15.56983.168NoYes086
82b.b22x1 b.b22x2 15.42862.59333NoNo088
833x46 7x53 58.80414.10508NoYes399
847x49 7x53 57.70075.00067YesYes399
852x50 7x49 40.84076.05363YesYes399
862x50 7x46 38.57045.62133YesNo098
872x53 7x46 38.30163.73221YesNo068
882x53 3x32 29.2768.37767YesYes267
893x32 Lig 26.18737.03704YesYes270
907x45 7x49 13.57845.42704YesYes399
91G.H3.08 G.S4.04 48.88765.4425NoYes099
92b.b21x7 b.b24x6 10.80398.20321YesYes058
93b.b22x2 b.b26x3 15.29366.45613NoYes086
94G.H3.17 b.l25x6 26.22433.52917YesNo148
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
7x34Lig4.936542NoYes5010
LigNT45.15842YesYes0301
1x28Lig3.40852NoYes4010
7x31Lig3.774422NoYes5010
E2Lig42.01312YesYes4010
E2x51Lig8.900832NoYes3010
E3Lig3.469422YesYes4010
5x32Lig4.022NoYes2010
NTNT17.98232YesYes3311
7x24NT5.770920NoYes7321
1x357x353.698710YesNo5521
2x533x328.377672YesYes6721
2x537x425.822922YesYes6722
2x603x326.438372NoYes6711
2x63E1x507.078582NoYes5812
E1x49E24.303582NoYes4421
E1x50E24.715752YesYes8421
3x22E26.008132NoYes4421
3x294x659.406832NoNo5512
3x327x423.27152YesYes7712
3x334x617.105080YesNo5422
4x614x652.852252NoNo4522
4x64E210.47352NoYes4421
4x645x353.749582NoNo4222
4x65E2x525.895212NoYes5521
E2E247.70582YesYes4411
E2E2x517.775082YesNo4311
E2E2x524.888462YesYes4511
5x35E29.610372NoYes2421
5x36E23.3562NoYes4411
5x39E24.758382NoYes5421
5x32E23.796712NoYes2411
5x406x555.26850NoNo5622
5x406x583.74750NoNo5421
6x516x523.354792YesNo7812
6x517x375.52052YesNo7612
6x517x387.310132YesNo7611
6x547x343.318130NoNo5521
6x547x373.815960NoNo5622
6x61E34.778790NoYes4421
6x64E32.530460NoYes1421
7x387x426.375212NoYes6712
1x247x312.59750NoNo0521
2x562x603.320132NoNo6621
2x563x322.707882NoYes6721
2x60Lig13.22882NoYes6010
2x63E23.662422NoYes5411
2x63Lig3.719082NoYes5010
3x29Lig3.359632NoYes5010
3x323x334.669462YesYes7512
3x32Lig7.037042YesYes7010
6x516x558.2162YesNo7612
6x51Lig2.97952YesYes7010
6x587x302.600422NoNo4412
6x58Lig3.033382NoYes4010
7x26E35.248292NoYes1421
7x27Lig8.508120NoYes4010
7x35Lig3.661332NoYes5010
7x38Lig7.105252NoYes6010
E2x52Lig2.89152YesYes5010
1x277x312.60250NoNo3521
5x36Lig4.342372NoYes4010
6x62Lig3.484542NoYes5010
4x61E2x525.0312NoYes4521
E3E33.442872YesYes4411
5x376x623.039670NoNo3521
6x60E34.594422NoYes5421
7x28NT3.333922NoYes3321
5x36E2x513.631832NoNo4311
5x336x621.952750NoNo1521
1x251x280.7420NoNo4421
2x67Lig0.7170NoYes4010

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
90.91Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
80.95Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
75.00Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
73.91Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
64.29Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
64.00Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
64.00Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
62.50Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
60.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
60.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
60.00Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
60.00Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
59.26Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
59.26Single7SK3CXCL127SK3-ACKR3-CXCL12
59.26Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
59.26Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
59.26Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
59.09Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
56.67Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
56.00Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
56.00Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
56.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
55.56Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
55.56Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
54.17Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
54.17Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
54.17Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
53.85Single3OE0CVX153OE0-CXCR4-CVX15
53.85Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
53.57Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
53.57Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
53.57Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
53.33Single5GLHEndothelin-15GLH-ETB-Endothelin-1
53.33Single6IGKEndothelin-36IGK-ETB-Endothelin-3
52.17Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
52.17Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
52.00Single8XWNCXCL88XWN-CXCR2-CXCL8
52.00Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
51.85Single6JODAngiotensin II6JOD-AT2-Angiotensin II
51.85Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
51.85Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
51.85Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
51.85Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
51.72Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
51.72Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
51.61Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
50.00Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
50.00Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
50.00Single6IGLIRL16206IGL-ETB-IRL1620
50.00Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
50.00Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
50.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
50.00Single7SK5CXCL127SK5-ACKR3-CXCL12
50.00Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
50.00Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
50.00Single8IY6Endothelin-18IY6-ETB-Endothelin-1
50.00Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
50.00Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
50.00Single8XVUCXCL28XVU-CXCR2-CXCL2
50.00Single8XWFCXCL38XWF-CXCR2-CXCL3
50.00Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
50.00Single8ZPLHF511168ZPL-CXCR4-HF51116
50.00Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
50.00Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
50.00Consensusbradykinin_onOrthosteric Ligandbk2_on
50.00Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
50.00Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
50.00Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
50.00Consensusendothelin_onOrthosteric Ligandetb_on eta_on
50.00Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
48.39Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
48.39Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
48.39Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
48.28Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
48.28Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
48.15Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
48.15Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
48.15Consensusangiotensin_onOrthosteric Ligandat1_on
48.15Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
48.00Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
47.83Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
47.83Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
47.62Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
47.62Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
46.67Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
46.67Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
46.43Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
46.43Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
46.43Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
46.43Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
46.43Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
46.43Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
46.43Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
46.15Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
46.15Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
46.15Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
46.15Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
46.15Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
45.83Single6OS2TRV0266OS2-AT1-TRV026
45.83Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
45.83Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
45.45Single6D27CAY104716D27-DP2-CAY10471
45.45Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
45.45Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
45.16Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
44.83Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
44.83Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
44.83Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
44.83Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
44.83Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
44.83Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
44.83Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
44.83Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
44.44Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
44.44Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
44.44Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
44.44Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
44.44Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
44.44Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
44.44Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
44.44Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
44.44Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
44.12Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
44.00Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
43.75Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
43.75Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
43.48Single6D26Fevipiprant6D26-DP2-Fevipiprant
43.48Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
43.48Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
43.48Consensusdp_offOrthosteric Liganddp2_off
43.33Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
43.33Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
42.86Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
42.86Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
42.86Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
42.86Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
42.86Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
42.86Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
42.86Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
42.86Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
42.86Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
42.42Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
42.42Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
42.31Single6KNMJN241-96KNM-Apelin-JN241-9
42.31Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
42.31Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
42.31Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
42.31Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
42.31Single8QJ2pN1628QJ2-MC4-pN162-Gs
42.31Single8XQJJN2418XQJ-Apelin-JN241
42.31Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
42.31Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
41.94Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
41.94Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
41.94Single9KDFRES-701-39KDF-ETB-RES-701-3
41.67Single6OS1TRV0266OS1-AT1-TRV026
41.67Single7F1TMIP-1a7F1T-CCR5-MIP-1a
41.67Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
41.67Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
41.67Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
41.67Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.67Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
41.67Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
41.67Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
41.38Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
41.38Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
41.38Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
41.38Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
41.18Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
40.91Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
40.91Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
40.91Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
40.91Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
40.74Single4XT1Fractalkine4XT1-US28-Fractalkine
40.74Single7F8XNN90567F8X-CCKA-NN9056
40.74Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
40.74Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
40.74Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
40.74Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
40.74Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
40.74Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
40.74Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
40.74Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
40.62Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
40.62Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
40.00Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
40.00Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
40.00Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
40.00Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
40.00Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
40.00Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
40.00Single8XWACXCL18XWA-CXCR2-CXCL1
40.00Single8XWMCXCL68XWM-CXCR2-CXCL6
40.00Single8XWSCXCL58XWS-CXCR2-CXCL5
40.00Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Single8ZRTET-18ZRT-ETB-ET-1
40.00Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
40.00Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
40.00Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
40.00Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
40.00Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
39.29Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
39.29Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
39.29Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
39.29Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
39.29Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
39.13Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
39.13Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
39.13Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
39.13Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
39.13Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
39.13Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
39.13Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
39.13Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
39.13Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
38.71Single4XT3Fractalkine4XT3-US28-Fractalkine
38.71Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
38.71Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
38.71Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
38.71Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
38.71Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
38.46Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
38.46Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
38.46Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
38.46Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.46Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
38.46Consensusprostanoid_offOrthosteric Ligandep_off dp_off
38.10Single3OE9IT1t3OE9-CXCR4-IT1t
38.10Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
38.10Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
37.93Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
37.93Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
37.93Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
37.93Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
37.93Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
37.93Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
37.93Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
37.93Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
37.93Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
37.84Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
37.84Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
37.50Single5N2RPSB-365N2R-A2A-PSB-36-Na
37.50Single5N2SPSB365N2S-A1-PSB36
37.50Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
37.50Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
37.50Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
37.50Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
37.50Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
37.50Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
37.50Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
37.50Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
37.04Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
37.04Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
37.04Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
37.04Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
37.04Single7XN9L-054,5227XN9-SST2-L-054,522
37.04Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
37.04Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
37.04Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
37.04Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.04Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
37.04Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
37.04Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
37.04Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
36.67Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
36.67Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
36.67Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
36.67Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
36.67Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
36.67Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
36.67Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
36.67Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
36.67Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
36.67Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
36.67Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
36.67Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
36.67Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
36.67Consensusvasop-oxy_onOrthosteric Ligandv2_on
36.67Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
36.36Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
36.36Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
36.36Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
36.36Single8GNGIstradefylline8GNG-A2A-Istradefylline
36.36Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
36.36Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
36.36Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
36.36Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
36.36Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
36.00Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
36.00Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
36.00Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
36.00Single7PX4PSB-21137PX4-A2A-PSB-2113
36.00Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
36.00Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
36.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
36.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
36.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
35.71Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
35.71Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
35.71Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
35.71Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
35.71Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
35.71Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
35.71Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
35.71Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
35.48Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
35.48Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
35.48Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
35.48Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
35.48Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
35.48Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
35.48Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.78Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
34.78Single7AROLUF58337ARO-A2A-LUF5833-Na
34.78Single7F61PF-036547467F61-H3-PF-03654746
34.78Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
34.78Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
34.78Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
34.78Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
34.78Single8ZPMAMD0708ZPM-CXCR4-AMD070
34.78Single8ZPNAMD31008ZPN-CXCR4-AMD3100
34.78Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
34.78Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
34.78Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
34.62Single4XEENeurotensin4XEE-NTS1-Neurotensin
34.62Single4XESNeurotensin4XES-NTS1-Neurotensin
34.62Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
34.62Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
34.62Single6YVRNTS8-136YVR-NTS1-NTS8-13
34.62Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
34.62Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
34.62Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
34.62Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
34.62Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
34.62Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
34.62Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
34.62Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.62Single8XQJJN2418XQJ-Apelin-JN241
34.62Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
34.62Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
34.62Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
34.62Consensuslpl_offOrthosteric Ligands1p_off lpa_off
34.62Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
34.62Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
34.62Consensusorexin_onOrthosteric Ligandox2_on
34.48Single3QAKUK-4320973QAK-A2A-UK-432097
34.48Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
34.48Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
34.48Single7XNACYN1548067XNA-SST2-CYN154806
34.48Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
34.48Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
34.48Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
34.48Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
34.48Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
34.48Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
34.48Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
34.48Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
34.48Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
34.48Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
34.48Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
34.48Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
34.38Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
34.29Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
34.29Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
33.33Single3OE6IT1t3OE6-CXCR4-IT1t
33.33Single4BUONeurotensin4BUO-NTS1-Neurotensin
33.33Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
33.33Single4XNWMRS25004XNW-P2Y1-MRS2500
33.33Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
33.33Single5WF5UK-4320975WF5-A2A-UK-432097
33.33Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
33.33Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
33.33Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
33.33Single7EZCUKA7EZC-A2A-UKA
33.33Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
33.33Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
33.33Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
33.33Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
33.33Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
33.33Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
33.33Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
33.33Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
33.33Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
33.33Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
33.33Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
33.33Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
33.33Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
33.33Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
33.33Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
33.33Consensuscck_onOrthosteric Ligandccka_on cckb_on
33.33Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
33.33Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
33.33Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
33.33Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
33.33Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
33.33Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
33.33Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
32.56Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
32.26Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
32.26Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
32.14Single5WF6UK-4320975WF6-A2A-UK-432097
32.14Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
32.14Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
32.14Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
32.14Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
32.14Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
32.14Single9IPYJR14a9IPY-C3aB-JR14a
32.14Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
32.14Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Single5IUAQ274563485IUA-A2A-Q27456348-Na
32.00Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
32.00Single6S0QZM-2413856S0Q-A2A-ZM-241385
32.00Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
32.00Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
32.00Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
32.00Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
32.00Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
32.00Single8GNEKW-63568GNE-A2A-KW-6356-Na
32.00Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
32.00Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
32.00Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
32.00Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
32.00Single9EHSLUF76029EHS-A3A-LUF7602
32.00Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
32.00Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
32.00Consensusadenosine_offOrthosteric Liganda1_off a2_off
31.82Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
31.82Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.82Consensusgq_nucleotideOrthosteric Ligandgq_p2y
31.82Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
31.25Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
31.03Single4IARErgotamine4IAR-5-HT1B-Ergotamine
31.03Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
31.03Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
31.03Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
31.03Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
31.03Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
31.03Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
31.03Single8WDTphotoNECA8WDT-A2A-photoNECA
31.03Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.03Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
31.03Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
31.03Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
31.03Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
31.03Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
31.03Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
31.03Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
31.03Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
31.03Consensussomatostatin_offOrthosteric Ligandsst2_off
30.77Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
30.77Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
30.77Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
30.77Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
30.77Single7R0CAVP7R0C-V2-AVP-Arrestin2
30.77Single7TUYGSK682753A7TUY-GPR183-GSK682753A
30.77Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.77Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
30.77Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
30.77Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.77Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
30.77Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
30.77Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
30.77Single8ZWFJR14a8ZWF-C3aB-JR14a
30.77Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
30.77Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
30.77Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
30.77Consensusneurotensin_onOrthosteric Ligandnts1_on
30.77Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
30.77Consensusrelaxin_onOrthosteric Ligandrxfp4_on
30.77Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
30.43Single3ODUIT1t3ODU-CXCR4-IT1t
30.43Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
30.43Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
30.43Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
30.43Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
30.43Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
30.43Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
30.43Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
30.43Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
30.43Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
30.43Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
30.30Single6FJ3PTH6FJ3-PTH1-PTH
30.30Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
30.30Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
30.00Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
30.00Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
30.00Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
30.00Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
30.00Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
30.00Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
29.63Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
29.63Single6MXTSalmeterol6MXT-β2-Salmeterol
29.63Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
29.63Single7K15MKD0467K15-BLT1-MKD046-Na
29.63Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
29.63Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
29.63Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
29.63Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
29.63Single8JJLOlodaterol8JJL-β2-Olodaterol
29.63Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
29.63Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
29.63Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
29.63Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
29.63Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
29.63Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
29.63Consensuslpa_offOrthosteric Ligandlpa1_off
29.41Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
29.17Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
29.17Single5IUBQ274563445IUB-A2A-Q27456344-Na
29.17Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
29.17Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
29.17Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
29.17Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
29.17Single6MH8ZM-2413856MH8-A2A-ZM-241385
29.17Single7T32ZM-2413857T32-A2A-ZM-241385
29.17Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
29.17Single8IHKAcifran8IHK-HCA3-Acifran
29.17Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
29.17Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
29.17Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
29.17Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
29.17Single8K5CAcipimox8K5C-HCA2-Acipimox
29.17Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
29.17Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
29.17Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
29.17Consensusgrh_offOrthosteric Ligandgnrh1_off
29.17Consensushca_onOrthosteric Ligandhca2_on
29.03Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
29.03Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
29.03Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
29.03Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
29.03Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
29.03Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
28.95Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
28.57Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
28.57Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
28.57Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
28.57Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
28.57Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
28.57Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.57Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
28.57Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
28.57Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
28.57Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
28.57Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
28.57Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
28.57Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
28.57Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
28.57Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
28.57Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
28.57Consensusp2y_offOrthosteric Ligandp2y1_off
28.57Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
28.12Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
28.12Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
28.12Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
28.12Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
28.00Single3EMLZM-2413853EML-A2A-ZM-241385
28.00Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
28.00Single4QIMANTA XV4QIM-SMO-ANTA XV
28.00Single5IU8Q274563475IU8-A2A-Q27456347-Na
28.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
28.00Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
28.00Single5UENDU1725UEN-A1-DU172
28.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
28.00Single6S0LZM-2413856S0L-A2A-ZM-241385
28.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
28.00Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
28.00Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
28.00Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
28.00Single7PYRPSB-21157PYR-A2A-PSB-2115
28.00Single8CU6LJ-45178CU6-A2A-LJ-4517
28.00Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
28.00Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
28.00Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
28.00Single8K5DGSK2560738K5D-HCA2-GSK256073
28.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
28.00Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
28.00Single9H37A1IR09H37-A2A-A1IR0-Na
28.00Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
28.00Consensuscck_offOrthosteric Ligandccka_off
28.00Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
28.00Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
28.00Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
28.00Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
28.00Consensushca_on_gpOrthosteric Ligandhca2_on_gp
28.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
27.78Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
27.78Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
27.78Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
27.78Consensusbombesin_onOrthosteric Ligandbb2_on
27.78Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
27.78Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
27.78Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
27.59Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.59Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
27.59Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
27.59Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
27.59Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
27.59Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
27.59Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
27.59Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
27.27Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
27.27Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
27.27Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
27.27Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
27.27Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
27.27Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
27.27Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
27.27Consensuspac_onOrthosteric Ligandpac1_on
26.92Single4JKVTaladegib4JKV-SMO-Taladegib
26.92Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
26.92Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
26.92Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
26.92Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
26.92Single7C61Ergotamine7C61-5-HT1B-Ergotamine
26.92Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
26.92Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
26.92Single7W41PD1762527W41-BB2-PD176252
26.92Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
26.92Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
26.92Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
26.92Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
26.92Single8QOTNanobody-E8QOT-μ-Nanobody-E
26.92Single8S4DCMF-0198S4D-Apelin-CMF-019
26.92Single8TF5Oleic acid8TF5-GPR6-Oleic acid
26.92Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
26.92Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
26.92Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
26.92Consensusbombesin_offOrthosteric Ligandbb2_off
26.92Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
26.92Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
26.92Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
26.92Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
26.67Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
26.67Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
26.67Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
26.67Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
26.67Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
26.67Consensuslpl_onOrthosteric Ligands1p_on lpa_on
26.67Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
26.67Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
26.67Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
26.47Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
26.47Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
26.47Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
26.47Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
26.09Single4O9RCyclopamine4O9R-SMO-Cyclopamine
26.09Single5L7IVismodegib5L7I-SMO-Vismodegib
26.09Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
26.09Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
26.09Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
26.09Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
26.09Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
25.93Single4BV0Neurotensin4BV0-NTS1-Neurotensin
25.93Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
25.93Single5V56TC1145V56-SMO-TC114
25.93Single5V57TC1145V57-SMO-TC114
25.93Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
25.93Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
25.93Single7B6WCyclazosin7B6W-α1b-Cyclazosin
25.93Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
25.93Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
25.93Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
25.93Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
25.93Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
25.93Single8E0GBU728E0G-μ-BU72
25.93Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
25.93Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
25.93Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
25.93Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
25.93Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
25.93Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
25.93Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
25.81Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
25.81Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
25.81Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
25.81Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
25.71Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
25.71Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
25.71Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
25.71Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
25.64Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
25.64Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
25.00Single3PWHZM-2413853PWH-A2A-ZM-241385
25.00Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
25.00Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
25.00Single4BWBNeurotensin4BWB-NTS1-Neurotensin
25.00Single4QINSAG1.54QIN-SMO-SAG1.5
25.00Single4RWADIPP-NH24RWA-δ-DIPP-NH2
25.00Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
25.00Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
25.00Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
25.00Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
25.00Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
25.00Single6A93Risperidone6A93-5-HT2A-Risperidone
25.00Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
25.00Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
25.00Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
25.00Single6PT2KGCHM076PT2-δ-KGCHM07
25.00Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
25.00Single7BR3Elagolix7BR3-GnRH1-Elagolix
25.00Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
25.00Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
25.00Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
25.00Single7F8ULintitript7F8U-CCKA-Lintitript
25.00Single7F8YDevazepide7F8Y-CCKA-Devazepide
25.00Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
25.00Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
25.00Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
25.00Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
25.00Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
25.00Single7XRRLemborexant7XRR-OX2-Lemborexant
25.00Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
25.00Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
25.00Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
25.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
25.00Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
25.00Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
25.00Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.00Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
25.00Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
25.00Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
25.00Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
25.00Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
25.00Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
25.00Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
25.00Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
25.00Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
25.00Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
25.00Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
25.00Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
25.00Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
25.00Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
25.00Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
25.00Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
25.00Consensuspth_onOrthosteric Ligandpth1_on pth2_on
25.00Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
25.00Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
24.24Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
24.24Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
24.24Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
24.24Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
24.24Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
24.24Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
24.24Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
24.14Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
24.14Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
24.14Single6IBLArformoterol6IBL-β1-Arformoterol
24.14Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
24.14Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
24.14Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
24.14Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
24.14Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
24.14Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
24.14Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
24.14Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
24.14Consensuschemerin_onOrthosteric Ligandcml1_on
24.14Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
24.14Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
24.14Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
24.14Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
24.00Single3REYXAC3REY-A2A-XAC
24.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
24.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
24.00Single5JTBZM-2413855JTB-A2A-ZM-241385
24.00Single5UVIZM-2413855UVI-A2A-ZM-241385
24.00Single6AQFZM-2413856AQF-A2A-ZM-241385
24.00Single6V9SGTPL114036V9S-OX1-GTPL11403
24.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
24.00Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
24.00Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
24.00Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
24.00Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
24.00Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
24.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
24.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
24.00Single9BA0A1AKN9BA0-CB1-A1AKN
24.00Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
24.00Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
24.00Consensusa2_offOrthosteric Liganda2a_off
24.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
24.00Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
23.81Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
23.68Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
23.68Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
23.68Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
23.53Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
23.53Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
23.53Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
23.33Single4UG2CGS216804UG2-A2A-CGS21680
23.33Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
23.33Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
23.33Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
23.33Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
23.33Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
23.33Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
23.33Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
23.33Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
23.33Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
23.08Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
23.08Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
23.08Single5T04Neurotensin5T04-NTS1-Neurotensin
23.08Single5TGZAM65385TGZ-CB1-AM6538
23.08Single5UIGCmpd-15UIG-A2A-Cmpd-1
23.08Single6TOTLemborexant6TOT-OX1-Lemborexant
23.08Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
23.08Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
23.08Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
23.08Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
23.08Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
23.08Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
23.08Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
23.08Single7UL4Alvimopan7UL4-μ-Alvimopan
23.08Single7V3ZCP559407V3Z-CB1-CP55940
23.08Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
23.08Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
23.08Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
23.08Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
23.08Single7YXAONO-54306087YXA-S1P5-ONO-5430608
23.08Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
23.08Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
23.08Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
23.08Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
23.08Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
23.08Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
23.08Consensusa3_onOrthosteric Liganda3a_on
23.08Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
23.08Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
23.08Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
23.08Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
22.86Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
22.86Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
22.73Single3OE8IT1t3OE8-CXCR4-IT1t
22.73Single8A2OTheophylline8A2O-A2A-Theophylline-Na
22.73Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
22.58Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
22.58Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
22.58Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
22.58Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
22.58Single8WKYPG-9348WKY-MC4-PG-934
22.22Single2Y00Dobutamine2Y00-β1-Dobutamine
22.22Single5C1MBU725C1M-μ-BU72
22.22Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
22.22Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
22.22Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
22.22Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
22.22Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
22.22Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
22.22Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
22.22Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
22.22Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
22.22Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
22.22Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
22.22Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
22.22Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
22.22Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
22.22Single8JXSPF-61428JXS-D1-PF-6142
22.22Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
22.22Single9B9ZA1AKO9B9Z-CB1-A1AKO
22.22Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
22.22Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
22.22Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
22.22Consensusa3_on_gpOrthosteric Liganda3a_on_gp
22.22Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
22.22Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
22.22Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
22.22Consensusblt_offOrthosteric Ligandblt1_off
22.22Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
22.22Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
22.22Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
22.22Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
22.22Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
22.22Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
22.22Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
22.22Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
22.22Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
21.88Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
21.88Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
21.74Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
21.74Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
21.74Single8JPSCCL78JPS-ACKR1-CCL7
21.62Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
21.62Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
21.62Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
21.62Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
21.62Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
21.62Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
21.62Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
21.62Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
21.62Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
21.43Single3P0GBI1671073P0G-β2-BI167107
21.43Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
21.43Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
21.43Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
21.43Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
21.43Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
21.43Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
21.43Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
21.43Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
21.43Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
21.43Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
21.43Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
21.43Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
21.43Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
21.43Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
21.43Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
21.43Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
21.43Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
21.43Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
21.43Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
21.43Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
21.43Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
21.43Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
21.43Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
21.43Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
21.43Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
21.43Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
21.43Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
21.43Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
21.43Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
21.43Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.43Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
21.43Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
21.43Consensuslpa_onOrthosteric Ligandlpa1_on
21.43Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
21.43Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
21.21Single6W25SHU91196W25-MC4-SHU9119-Ca
21.21Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
21.05Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
20.93Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
20.93Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
20.83Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
20.83Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
20.83Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
20.83Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
20.83Single8K5BNiacin8K5B-HCA2-Niacin
20.83Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
20.83Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
20.83Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
20.83Single9B9Y7DY9B9Y-CB1-7DY
20.83Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
20.69Single4LDEBI1671074LDE-β2-BI167107
20.69Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
20.69Single4PY02MeSATP4PY0-P2Y12-2MeSATP
20.69Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
20.69Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
20.69Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
20.69Single6ZG4HTL00099366ZG4-M1-HTL0009936
20.69Single7DFPSpiperone7DFP-D2-Spiperone
20.69Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
20.69Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.69Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
20.69Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
20.69Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
20.69Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
20.69Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
20.69Single7YITNalfurafine7YIT-κ-Nalfurafine
20.69Single8JJ8Formoterol8JJ8-β2-Formoterol
20.69Single8JWY2-1188JWY-A2A-2-118
20.69Single8JWZAB9288JWZ-A2A-AB928-Na
20.69Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
20.69Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
20.69Single8XYIVUF106618XYI-CXCR3-VUF10661
20.69Single9BJKNAM9BJK-μ-Naloxone-NAM
20.69Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
20.69Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.69Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
20.69Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
20.69Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
20.69Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
20.69Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
20.69Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
20.69Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
20.69Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
20.69Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
20.69Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
20.69Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
20.59Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
20.59Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
20.59Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
20.59Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
20.51Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
20.51Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
20.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
20.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
20.00Single4S0VSuvorexant4S0V-OX2-Suvorexant
20.00Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
20.00Single5WS3EMPA5WS3-OX2-EMPA
20.00Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
20.00Single5ZKQABT-4915ZKQ-PAF-ABT-491
20.00Single6AKYMaraviroc6AKY-CCR5-Maraviroc
20.00Single6DS0Ly2660976DS0-5-HT2B-Ly266097
20.00Single6H7LDobutamine6H7L-β1-Dobutamine
20.00Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
20.00Single6TPJSuvorexant6TPJ-OX2-Suvorexant
20.00Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
20.00Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
20.00Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
20.00Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
20.00Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
20.00Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
20.00Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
20.00Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
20.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
20.00Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
20.00Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
20.00Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
20.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
20.00Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
20.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
20.00Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
20.00Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
20.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
20.00Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
20.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
20.00Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
20.00Single8Y0HVUF114188Y0H-CXCR3-VUF11418
20.00Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
20.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
20.00Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
20.00Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
20.00Single9H2XA1IR19H2X-A2A-A1IR1-Na
20.00Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
20.00Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
20.00Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
20.00Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
20.00Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.00Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.00Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.00Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
20.00Consensusendothelin_offOrthosteric Ligandetb_off
20.00Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
20.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusorexin_offOrthosteric Ligandox2_off ox1_off
20.00Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
20.00Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
20.00Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
20.00Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
20.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
19.51Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
19.51Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.44Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
19.44Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
19.44Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
19.44Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
19.44Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
19.44Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
19.44Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
19.44Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
19.35Single3NY9ICI118-5513NY9-β2-ICI118-551
19.35Single5ZTYAM102575ZTY-CB2-AM10257
19.35Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
19.35Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
19.35Single8X5YAstemizole8X5Y-H1-Astemizole
19.35Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
19.35Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
19.35Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
19.23Single2YDOAdenosine2YDO-A2A-Adenosine
19.23Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
19.23Single4MBSMaraviroc4MBS-CCR5-Maraviroc
19.23Single4ZJCSB-6740424ZJC-OX1-SB-674042
19.23Single6IQLL7458706IQL-D4-L745870
19.23Single6KUXRS-799486KUX-α2a-RS-79948
19.23Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
19.23Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
19.23Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
19.23Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
19.23Single6TP3Nemorexant6TP3-OX1-Nemorexant
19.23Single6TPGEMPA6TPG-OX2-EMPA
19.23Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
19.23Single6ZG9GSK10347026ZG9-M1-GSK1034702
19.23Single6ZINSR486926ZIN-NTS1-SR48692
19.23Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
19.23Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.23Single7UL3Famotidine7UL3-H2-Famotidine
19.23Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
19.23Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
19.23Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
19.23Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
19.23Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
19.23Single8K2WAMG4878K2W-CXCR3-AMG487
19.23Single8RLNLUF58348RLN-A2A-LUF5834
19.23Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
19.23Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
19.23Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
19.23Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
19.23Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
19.23Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
19.23Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
19.23Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
19.23Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
19.23Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
19.23Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
19.23Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
19.23Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
19.15Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
19.05Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
18.92Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
18.92Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
18.92Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
18.92Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
18.92Consensusglp_onOrthosteric Ligandglp1_on glp2_on
18.92Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
18.92Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
18.75Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
18.75Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
18.75Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
18.75Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
18.75Single8IEBA1LYA8IEB-GPR156-A1LYA
18.75Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
18.75Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
18.75Single8KIGSHU91198KIG-MC3-SHU9119-Ca
18.75Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
18.75Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.75Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.75Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
18.75Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
18.52Single2Y01Dobutamine2Y01-β1-Dobutamine
18.52Single2Y02Carmoterol2Y02-β1-Carmoterol
18.52Single2Y04Salbutamol2Y04-β1-Salbutamol
18.52Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
18.52Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
18.52Single4QKX35V4QKX-β2-35V
18.52Single4YAYZD-71554YAY-AT1-ZD-7155
18.52Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
18.52Single6DRXLisuride6DRX-5-HT2B-Lisuride
18.52Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
18.52Single6GPSMK08126GPS-CCR2-MK0812
18.52Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
18.52Single6PS1Timolol6PS1-β2-Timolol
18.52Single7BU7BI1671077BU7-β1-BI167107
18.52Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
18.52Single7F83PF-051904577F83-Ghrelin-PF-05190457
18.52Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
18.52Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
18.52Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
18.52Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
18.52Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
18.52Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
18.52Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
18.52Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
18.52Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
18.52Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
18.52Single8T1WCVN4248T1W-GPR6-CVN424
18.52Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
18.52Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
18.52Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
18.52Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
18.52Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
18.52Single9CHXS-Carazolol9CHX-β2-S-Carazolol
18.52Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
18.52Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
18.52Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
18.52Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
18.52Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
18.52Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
18.52Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
18.52Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
18.52Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
18.52Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
18.42Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
18.42Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
18.42Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
18.42Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
18.42Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
18.42Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
18.18Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
18.18Single6HLOAprepitant6HLO-NK1-Aprepitant
18.18Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
18.18Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
18.18Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
18.18Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
18.18Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
18.18Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
18.18Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
18.18Single8IEBA1LYA8IEB-GPR156-A1LYA
18.18Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
18.18Single8PWNTheophylline8PWN-A2A-Theophylline
18.18Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
17.95Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
17.95Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
17.95Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
17.86Single2Y03Isoprenaline2Y03-β1-Isoprenaline
17.86Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
17.86Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
17.86Single5WIUNemonapride5WIU-D4-Nemonapride
17.86Single5WIVNemonapride5WIV-D4-Nemonapride-Na
17.86Single5WQCEMPA5WQC-OX2-EMPA
17.86Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
17.86Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
17.86Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
17.86Single6E67BI1671076E67-β2-BI167107-Gs(CT)
17.86Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
17.86Single6GPXMK08126GPX-CCR2-MK0812
17.86Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
17.86Single6LUQHaloperidol6LUQ-D2-Haloperidol
17.86Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
17.86Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
17.86Single6TP6Filorexant6TP6-OX1-Filorexant
17.86Single6Z4SSR486926Z4S-NTS1-SR48692
17.86Single7C4SS1P7C4S-S1P3-S1P
17.86Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
17.86Single7SINNPS-21437SIN-CaS-NPS-2143
17.86Single7SINNPS-21437SIN-CaS-NPS-2143
17.86Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
17.86Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
17.86Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
17.86Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
17.86Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
17.86Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
17.86Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
17.86Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
17.86Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.86Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
17.86Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
17.86Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
17.86Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
17.86Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
17.86Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
17.86Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
17.86Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.86Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
17.86Consensusep_offOrthosteric Ligandep4_off
17.86Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
17.86Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
17.86Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.86Consensustrace-amine_onOrthosteric Ligandta1_on
17.65Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
17.65Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
17.65Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
17.65Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
17.65Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.65Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
17.50Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
17.50Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
17.50Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.39Single3RFMCaffeine3RFM-A2A-Caffeine
17.39Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
17.39Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
17.39Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
17.39Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
17.24Single2YDVNECA2YDV-A2A-NECA
17.24Single4UHRCGS216804UHR-A2A-CGS21680
17.24Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
17.24Single5G53NECA5G53-A2A-NECA-Gs
17.24Single5TZRMK86665TZR-FFA1-MK8666
17.24Single5XR8AM8415XR8-CB1-AM841
17.24Single5XRAAM115425XRA-CB1-AM11542
17.24Single6H7JIsoprenaline6H7J-β1-Isoprenaline
17.24Single6J20Aprepitant6J20-NK1-Aprepitant
17.24Single6J21Aprepitant6J21-NK1-Aprepitant
17.24Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
17.24Single6TQ7SB-3348676TQ7-OX1-SB-334867
17.24Single6WGTLSD6WGT-5-HT2A-LSD
17.24Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
17.24Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
17.24Single7FEECP559407FEE-CB1-CP55940-ZCZ011
17.24Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
17.24Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
17.24Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
17.24Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
17.24Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
17.24Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
17.24Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
17.24Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
17.24Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.24Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
17.24Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.24Single8XVLZibotentan8XVL-ETA-Zibotentan
17.24Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
17.24Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
17.24Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
17.24Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
17.24Consensusa2_onOrthosteric Liganda2b_on
17.24Consensusa2_on_gpOrthosteric Liganda2b_on_gp
17.24Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.24Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
17.24Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
17.24Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
17.24Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
17.24Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.24Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
17.24Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
17.24Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
17.24Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
17.24Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
17.24Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
17.24Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.24Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
17.14Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
17.14Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
17.14Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
17.14Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
17.14Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
17.07Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
17.07Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
16.67Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
16.67Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
16.67Single4AMIBucindolol4AMI-β1-Bucindolol
16.67Single4N4WSANT-14N4W-SMO-SANT-1
16.67Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
16.67Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
16.67Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
16.67Single5X33BIIL2605X33-BLT1-BIIL260
16.67Single6CM4Risperidone6CM4-D2-Risperidone
16.67Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
16.67Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
16.67Single6KQICP559406KQI-CB1-CP55940-Org27569
16.67Single6ME5Agomelatine6ME5-MT1-Agomelatine
16.67Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
16.67Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
16.67Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
16.67Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
16.67Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
16.67Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
16.67Single7WC5Psilocin7WC5-5-HT2A-Psilocin
16.67Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
16.67Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
16.67Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.67Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
16.67Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
16.67Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
16.67Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.67Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
16.67Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
16.67Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
16.67Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
16.67Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
16.67Single9DGIZ85267113509DGI-CB1-Z8526711350
16.67Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
16.67Consensusalpha1_offOrthosteric Ligandalpha1a_off
16.67Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
16.67Consensuscalcitonin_onOrthosteric Ligandctlike_on
16.67Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
16.67Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.67Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
16.67Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.67Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
16.67Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
16.67Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
16.28Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
16.22Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
16.22Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
16.22Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
16.22Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
16.22Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
16.22Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
16.22Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
16.22Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
16.22Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
16.13Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
16.13Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
16.13Single5X93K-87945X93-ETB-K-8794
16.13Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
16.13Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
16.13Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
16.13Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
16.13Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
16.13Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
16.13Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
16.13Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
16.13Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
16.13Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
16.13Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
16.13Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
16.13Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
16.13Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
16.13Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.00Single6LI0C176LI0-GPR52-C17
16.00Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
16.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
16.00Single7UL2SR486927UL2-NTS1-SR48692-Na
16.00Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
16.00Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
16.00Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
16.00Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
16.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
16.00Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
16.00Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
16.00Consensusneurotensin_offOrthosteric Ligandnts1_off
16.00Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
15.79Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
15.79Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
15.79Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
15.79Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
15.79Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
15.79Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
15.79Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
15.62Single6PT3DPI-2876PT3-δ-DPI-287
15.62Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
15.62Single7SK9CCX6627SK9-ACKR3-CCX662
15.62Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
15.62Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
15.62Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
15.62Single9JF4PD1683689JF4-BB1-PD168368
15.62Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
15.62Consensuskisspeptin_onOrthosteric Ligandkiss1_on
15.56Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
15.38Single5U09Taranabant5U09-CB1-Taranabant
15.38Single6AKXA4R6AKX-CCR5-A4R
15.38Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
15.38Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
15.38Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
15.38Single6ME9Ramelteon6ME9-MT2-Ramelteon
15.38Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
15.38Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
15.38Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
15.38Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
15.38Single6TODEMPA6TOD-OX1-EMPA-Na
15.38Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
15.38Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
15.38Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
15.38Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
15.38Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
15.38Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
15.38Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
15.38Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
15.38Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
15.38Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
15.38Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
15.38Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
15.38Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
15.38Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
15.38Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
15.38Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
15.38Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
15.38Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
15.38Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
15.38Single8IWESpermidine8IWE-TA9-Spermidine
15.38Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
15.38Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
15.38Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
15.38Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
15.38Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
15.38Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
15.38Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
15.38Consensusalpha2_offOrthosteric Ligandalpha2c_off
15.38Consensusangiotensin_offOrthosteric Ligandat1_off
15.38Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
15.22Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
15.15Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
15.15Single7QA8Peptide7QA8-STE2-Peptide
15.15Single7QA8Peptide7QA8-STE2-Peptide
15.15Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
15.15Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Single8IEIA1LYA8IEI-GPR156-A1LYA
15.15Single8IEIA1LYA8IEI-GPR156-A1LYA
15.15Single8IEPA1LYA8IEP-GPR156-A1LYA
15.15Single8IEPA1LYA8IEP-GPR156-A1LYA
15.15Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
15.15Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
15.15Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
15.15Single9M4TSilodosin9M4T-Alpha1A-Silodosin
15.00Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
15.00Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
14.81Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
14.81Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
14.81Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
14.81Single6PS0S-Carazolol6PS0-β2-S-Carazolol
14.81Single6PS4ICI118-5516PS4-β2-ICI118-551
14.81Single6PS5S-Propranolol6PS5-β2-S-Propranolol
14.81Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
14.81Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
14.81Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
14.81Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
14.81Single7VV6C48/807VV6-MRGPRX2-C48/80
14.81Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
14.81Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
14.81Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
14.81Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
14.81Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
14.81Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
14.81Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
14.81Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
14.81Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
14.81Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
14.81Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
14.81Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
14.81Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
14.81Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
14.81Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.81Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
14.81Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
14.81Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single9AS5Mescaline9AS5-5-HT2A-Mescaline
14.81Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.81Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
14.81Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
14.81Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
14.81Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
14.29Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
14.29Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
14.29Single3NY8ICI118-5513NY8-β2-ICI118-551
14.29Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
14.29Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
14.29Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
14.29Single4EJ4Naltrindole4EJ4-δ-Naltrindole
14.29Single4GBRS-Carazolol4GBR-β2-S-Carazolol
14.29Single5DHGC-355DHG-NOP-C-35
14.29Single5DHHSB-6121115DHH-NOP-SB-612111
14.29Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
14.29Single6H7MSalbutamol6H7M-β1-Salbutamol
14.29Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
14.29Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
14.29Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
14.29Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
14.29Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
14.29Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
14.29Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
14.29Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
14.29Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
14.29Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
14.29Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
14.29Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
14.29Single7WC7Lisuride7WC7-5-HT2A-Lisuride
14.29Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
14.29Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
14.29Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
14.29Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
14.29Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
14.29Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
14.29Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
14.29Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
14.29Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
14.29Single8JJOAlprenolol8JJO-β2-Alprenolol
14.29Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
14.29Single8JXRLSD8JXR-D1-LSD
14.29Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
14.29Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
14.29Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
14.29Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
14.29Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single9AS1DMT9AS1-5-HT2A-DMT
14.29Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
14.29Consensus5ht5_onOrthosteric Ligand5ht5a_on
14.29Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
14.29Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
14.29Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
14.29Consensusdopamine_offOrthosteric Ligandd2_off d3_off
14.29Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
14.29Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
14.29Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
13.95Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
13.95Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
13.89Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
13.89Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
13.89Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
13.89Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
13.79Single2RH1S-Carazolol2RH1-β2-S-Carazolol
13.79Single2YCWS-Carazolol2YCW-β1-S-Carazolol
13.79Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
13.79Single5D6LS-Carazolol5D6L-β2-S-Carazolol
13.79Single5JQHS-Carazolol5JQH-β2-S-Carazolol
13.79Single5TVNLSD5TVN-5-HT2B-LSD
13.79Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
13.79Single5XPRBosentan5XPR-ETB-Bosentan
13.79Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
13.79Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
13.79Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
13.79Single6PS6Timolol6PS6-β2-Timolol
13.79Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
13.79Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
13.79Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.79Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
13.79Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
13.79Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
13.79Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
13.79Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.79Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
13.79Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
13.79Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
13.79Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
13.79Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
13.79Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
13.79Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
13.79Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
13.79Single9HAPTolvaptan9HAP-V2-Tolvaptan
13.79Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.79Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
13.79Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
13.79Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
13.79Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
13.79Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
13.79Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
13.79Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
13.79Consensusamine_offonOrthosteric Ligandamine_off amine_on
13.79Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
13.79Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
13.79Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
13.79Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
13.79Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
13.64Single5MZPCaffeine5MZP-A2A-Caffeine-Na
13.64Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
13.64Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
13.64Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
13.51Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
13.51Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.33Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
13.33Single4DJHJDTic4DJH-κ-JDTic
13.33Single5D5AS-Carazolol5D5A-β2-S-Carazolol
13.33Single5D5BS-Carazolol5D5B-β2-S-Carazolol
13.33Single6E59L-7607356E59-NK1-L-760735
13.33Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
13.33Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
13.33Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
13.33Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
13.33Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
13.33Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
13.33Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
13.33Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
13.33Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
13.33Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
13.33Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
13.33Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
13.33Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
13.33Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
13.33Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
13.33Single9BJKNaloxone9BJK-μ-Naloxone-NAM
13.33Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.33Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
13.33Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
13.33Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
13.33Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
13.33Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
13.33Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
13.33Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.33Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
13.33Consensustachykinin_offOrthosteric Ligandnk1_off
13.16Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
13.16Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
13.16Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
13.16Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
13.04Single7WC4Serotonin7WC4-5-HT2A-Serotonin
13.04Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
13.04Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
12.90Single3D4STimolol3D4S-β2-Timolol
12.90Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
12.90Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
12.90Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
12.90Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
12.90Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
12.90Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
12.90Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
12.90Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.90Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.90Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
12.90Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
12.90Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
12.82Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
12.82Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
12.82Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
12.82Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
12.82Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
12.82Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
12.50Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
12.50Single6K1QIRL25006K1Q-ETB-IRL2500
12.50Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
12.50Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
12.50Single6TQ9SB-4081246TQ9-OX1-SB-408124
12.50Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
12.50Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.50Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
12.50Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
12.50Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
12.50Single7UM4AS26747237UM4-5-HT5A-AS2674723
12.50Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
12.50Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
12.50Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
12.50Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
12.50Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
12.50Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
12.50Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
12.50Single9CHUNoradrenaline9CHU-β2-Noradrenaline
12.50Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
12.50Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
12.50Consensussensory_onOrthosteric Ligandopsins_on
12.12Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
12.12Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
12.12Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
12.12Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
12.00Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
12.00Single3UZAGTPL92363UZA-A2A-GTPL9236
12.00Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
12.00Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
12.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
12.00Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
12.00Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
12.00Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
12.00Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
12.00Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
12.00Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
12.00Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
12.00Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.00Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
12.00Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
12.00Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
12.00Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
12.00Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
12.00Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
12.00Single9LRCHistamine9LRC-H4-Histamine
12.00Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
12.00Consensus5ht2_onOrthosteric Ligand5ht2b_on
12.00Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.00Consensusgi_sensoryOrthosteric Ligandgi_opsins
12.00Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.00Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.00Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.00Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.00Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
12.00Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
12.00Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
11.76Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
11.76Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
11.76Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
11.63Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
11.54Single3PBLEticlopride3PBL-D3-Eticlopride
11.54Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
11.54Single6HLLCP999946HLL-NK1-CP99994
11.54Single6TP4ACT-4622066TP4-OX1-ACT-462206
11.54Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
11.54Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
11.54Single7SRQLSD7SRQ-5-HT2B-LSD
11.54Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
11.54Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.54Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
11.54Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
11.54Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
11.54Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
11.54Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
11.54Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
11.54Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
11.54Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
11.54Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
11.54Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
11.54Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
11.54Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
11.54Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
11.54Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.54Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
11.54Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
11.36Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
11.11Single6B73MP11046B73-κ-MP1104
11.11Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
11.11Single6ME2Ramelteon6ME2-MT1-Ramelteon
11.11Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
11.11Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
11.11Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
11.11Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
11.11Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
11.11Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
11.11Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
11.11Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
11.11Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
11.11Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
11.11Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
11.11Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
11.11Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
11.11Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
11.11Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
11.11Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
11.11Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
11.11Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
11.11Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
11.11Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
11.11Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
11.11Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
11.11Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
11.11Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
11.11Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.11Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
11.11Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.11Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
11.11Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
11.11Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
11.11Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
10.87Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
10.81Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
10.81Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
10.81Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
10.81Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
10.81Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
10.71Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
10.71Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
10.71Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
10.71Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
10.71Single6A94Zotepine6A94-5-HT2A-Zotepine
10.71Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
10.71Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
10.71Single6TPKRetosiban6TPK-OT-Retosiban
10.71Single6TPNHTL66416TPN-OX2-HTL6641
10.71Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
10.71Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
10.71Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
10.71Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
10.71Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
10.71Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
10.71Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
10.71Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
10.71Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
10.71Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
10.71Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
10.71Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
10.71Single7VODCariprazine7VOD-5-HT2A-Cariprazine
10.71Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
10.71Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
10.71Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
10.71Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
10.71Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.71Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
10.71Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
10.71Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
10.71Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
10.71Single9AS3LSD9AS3-5-HT2A-LSD
10.71Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
10.71Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
10.71Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
10.71Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
10.71Consensusalpha1_onOrthosteric Ligandalpha1a_on
10.71Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
10.71Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
10.71Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
10.71Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
10.71Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
10.71Consensusopsins_offOrthosteric Ligandrhodopsin_off
10.71Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
10.71Consensussensory_offOrthosteric Ligandopsins_off
10.71Consensusvasop-oxy_offOrthosteric Ligandot_off
10.34Single4DAJTiotropium4DAJ-M3-Tiotropium
10.34Single4MQSIperoxo4MQS-M2-Iperoxo
10.34Single4U14Tiotropium4U14-M3-Tiotropium
10.34Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
10.34Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
10.34Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
10.34Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
10.34Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
10.34Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
10.34Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
10.34Single6IIVDaltroban6IIV-TXA2-Daltroban
10.34Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.34Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
10.34Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.34Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
10.34Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
10.34Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
10.34Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
10.34Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
10.34Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
10.34Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
10.34Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
10.34Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
10.34Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
10.34Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
10.34Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
10.34Single8X63Mepyramine8X63-H1-Mepyramine
10.34Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
10.34Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
10.34Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
10.34Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
10.34Single9IYAONO-97105319IYA-GPR55-ONO-9710531
10.34Single9JEAAtropine9JEA-M1-Atropine
10.34Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
10.34Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
10.34Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
10.34Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.34Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
10.34Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
10.34Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
10.34Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
10.34Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
10.34Consensusalpha2_onOrthosteric Ligandalpha2b_on
10.34Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
10.34Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.34Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.34Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
10.34Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
10.34Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
10.34Consensusblt_onOrthosteric Ligandblt1_on
10.34Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
10.34Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
10.34Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
10.34Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
10.34Consensushistamine_offOrthosteric Ligandh1_off
10.34Consensusleukotriene_onOrthosteric Ligandblt_on
10.34Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
10.34Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
10.34Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
10.00Single4NTJAZD12834NTJ-P2Y12-AZD1283
10.00Single5CGCHTL142425CGC-mGlu5-HTL14242
10.00Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
10.00Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
10.00Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
10.00Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
10.00Single7WC6LSD7WC6-5-HT2A-LSD
10.00Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
10.00Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
10.00Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
10.00Single8ZMFA1L108ZMF-5-HT2C-A1L10
10.00Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
10.00Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
10.00Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
10.00Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
10.00Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
10.00Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
10.00Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
10.00Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.00Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.00Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
10.00Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
10.00Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.00Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
10.00Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.00Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
10.00Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single4U15Tiotropium4U15-M3-Tiotropium
9.68Single5V54Methiothepin5V54-5-HT1B-Methiothepin
9.68Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
9.68Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
9.68Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
9.68Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
9.68Single6OL9Tiotropium6OL9-M5-Tiotropium
9.68Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
9.68Single8EA0Iperoxo8EA0-M3-Iperoxo
9.68Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
9.68Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
9.68Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
9.68Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
9.68Consensus5ht1_offOrthosteric Ligand5ht1b_off
9.68Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
9.68Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
9.68Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
9.68Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
9.68Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
9.68Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
9.52Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
9.38Single5CXVTiotropium5CXV-M1-Tiotropium
9.38Single6IIURamatroban6IIU-TXA2-Ramatroban
9.38Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
9.38Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.38Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
9.38Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
9.38Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
9.38Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
9.09Single5CGDHTL142425CGD-mGlu5-HTL14242
9.09Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
9.09Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
9.09Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
9.09Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
9.09Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
9.09Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
9.09Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
9.09Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
8.82Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
8.57Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
8.33Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
8.33Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
8.33Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.33Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.33Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
8.00Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
8.00Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
8.00Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
8.00Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
8.00Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
7.69Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
7.69Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
7.69Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
7.69Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
7.69Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
7.69Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
7.69Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
7.69Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
7.69Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
7.69Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
7.69Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
7.69Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
7.69Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
7.69Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
7.69Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
7.41Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
7.41Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
7.41Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
7.41Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
7.41Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
7.41Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
7.41Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
7.41Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
7.41Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
7.41Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.41Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
7.41Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
7.41Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
7.41Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
7.41Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
7.41Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
7.41Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
7.41Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.41Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
7.41Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.41Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
7.41Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
7.41Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.41Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.41Single9AS7Psilocin9AS7-5-HT2A-Psilocin
7.41Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
7.41Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
7.41Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
7.41Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
7.41Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.41Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
7.14Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
7.14Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
7.14Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
7.14Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
7.14Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
7.14Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
7.14Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
7.14Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.14Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
7.14Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
7.14Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
7.14Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
7.14Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
7.14Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
7.14Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.14Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
7.14Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
7.14Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
7.14Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
7.14Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
6.90Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
6.90Single3RZECidoxepin3RZE-H1-Cidoxepin
6.90Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
6.90Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
6.90Single6VI4JDTic6VI4-κ-JDTic
6.90Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
6.90Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
6.90Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
6.90Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
6.90Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
6.90Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
6.90Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
6.90Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
6.90Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
6.90Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
6.90Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
6.90Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
6.90Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
6.90Single9ARXSerotonin9ARX-5-HT2A-Serotonin
6.90Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
6.67Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
6.67Single5DSGTiotropium5DSG-M4-Tiotropium
6.67Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
6.67Single8X64Desloratadine8X64-H1-Desloratadine
6.67Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
6.67Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
6.45Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
6.45Single6HLPNetupitant6HLP-NK1-Netupitant
6.45Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
6.45Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
6.45Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
6.45Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.45Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.45Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.45Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
6.45Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
6.25Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
6.25Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
6.25Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
6.25Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
6.25Single9AS9RS130-1809AS9-5-HT2A-RS130-180
6.25Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
6.06Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.88Single8XVJMacitentan8XVJ-ETA-Macitentan
5.71Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
4.76Single6D35Cholesterol6D35-SMO-Cholesterol
4.76Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.76Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
4.76Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
4.76Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
4.76Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
4.76Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.76Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
4.76Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
4.76Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
4.76Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
4.76Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
4.76Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
4.76Single7DTTCa7DTT-CaS-Ca-Ca
4.76Single7DTTCa7DTT-CaS-Ca-Ca
4.76Single7DTUTryptophan7DTU-CaS-Tryptophan
4.76Single7DTUTryptophan7DTU-CaS-Tryptophan
4.76Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.76Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.76Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
4.76Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
4.76Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.76Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
4.76Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.76Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
4.76Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
4.76Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.76Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
4.76Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.76Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
4.76Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.76Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
4.76Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
4.76Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
4.76Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.76Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
4.76Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.76Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
4.76Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.76Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
4.76Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.76Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
4.76Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.76Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
4.76Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.76Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.76Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.76Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
4.76Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
4.76Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
4.76Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.76Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
4.76Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.76Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
4.76Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.76Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
4.76Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
4.76Single7XW7K1-707XW7-TSH-K1-70
4.76Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.76Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
4.76Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.76Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
4.76Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.76Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
4.76Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.76Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
4.76Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.76Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
4.76Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.76Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
4.76Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
4.76Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.76Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
4.76Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.76Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
4.76Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.76Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
4.76Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.76Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
4.76Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.76Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
4.76Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.76Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.76Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.76Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.76Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
4.76Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.76Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
4.76Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.76Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
4.76Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.76Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
4.76Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.76Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
4.76Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.76Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
4.76Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.76Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
4.76Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.76Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
4.76Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
4.76Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.76Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
4.76Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
4.76Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.76Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
4.76Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.76Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
4.76Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
4.76Single8WVXNorrin8WVX-LGR4-Norrin
4.76Single8WVYNorrin8WVY-LGR4-Norrin
4.76Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.76Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
4.76Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
4.76Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.76Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
4.76Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.76Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
4.76Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
4.76Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.76Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.76Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.76Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
4.76Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.76Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.76Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
4.76Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.76Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.76Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.76Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
4.76Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
4.76Single9KHHNorrin9KHH-LGR4-Norrin
4.76Single9S37NB219S37-LGR4-NB21
4.76Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.55Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.55Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.55Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.55Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.55Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.55Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.55Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.35Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.35Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.35Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.17Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
4.17Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
4.17Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.17Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.17Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.17Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.17Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.00Single5L7DCholesterol5L7D-SMO-Cholesterol
4.00Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.00Single8HS2Fab0468HS2-GPR20-Fab046
4.00Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.85Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
3.85Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
3.70Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
3.57Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
3.57Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
3.33Single6FFIMMPEP6FFI-mGlu5-MMPEP
3.33Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.33Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Single6FFHFenobam6FFH-mGlu5-Fenobam
3.23Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
3.12Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.12Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.12Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.12Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
3.12Single9HC04YI9HC0-mGlu5-4YI
3.03Single7P2L4YI7P2L-mGlu5-4YI
3.03Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.03Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.03Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
2.70Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.70Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.56Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.56Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.50Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.33Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
ccr_on_gp ccr6_on_gp
ccr8_on_gp
ccr2_on_gp
ccr1_on_gp
ccr5_on_gp
cxcr_on_gp cxcr3_on_gp
cxcr4_on_gp
cxcr1_on_gp
cxcr2_on_gp
Net Summary
Imin 2.52225
Number of Linked Nodes 945
Number of Links 1178
Number of Hubs 198
Number of Links mediated by Hubs 771
Number of Communities 22
Number of Nodes involved in Communities 274
Number of Links involved in Communities 417
Path Summary
Number Of Nodes in MetaPath 95
Number Of Links MetaPath 94
Number of Shortest Paths 2753298
Length Of Smallest Path 3
Average Path Length 36.6186
Length of Longest Path 65
Minimum Path Strength 0.278
Average Path Strength 4.944
Maximum Path Strength 32.5483
Minimum Path Correlation 0.704792
Average Path Correlation 0.98299
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.81818
Average % Of Corr. Nodes 36.7208
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 53.0722
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following differences:
Id1st Network2nd Network
chemokine_off_on_gpchemokine_on_gpchemokine_off
This network is also present in following consensuses:
IdComponents
protein_on_gpchemokine_on_gp
chemerin_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download chemokine_on_gp.zip



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You can also  read or  download a guide explaining the meaning of all files and numerical data.