Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.11 1.14082603
2G.HN.37 1.47711402
3G.S2.08 3.66028405
4G.S3.03 4.39861407
5G.S3.06 4.21886406
6G.H2.07 3.1059409
7G.H3.09 3.37971509
8G.H3.17 4.48802404
9G.H3.18 3.18529409
10G.S5.05 1.98495609
11G.hgh4.02 2.42528608
12G.hgh4.05 4.33104406
13G.H4.12 3.53529405
14G.S6.02 3.89534408
15b.1x4 0.942635408
16b.h2x1 1.72465405
17b.l1x3 5.35413409
18b.b2x5 3.51173507
19b.l3x2 2.72386409
20b.b4x2 2.68934408
21b.b4x3 2.89424407
22b.b4x6 6.1518409
23b.b5x2 3.04281407
24b.b5x3 4.00823409
25b.b5x5 2.86117405
26b.l5x5 4.20251609
27b.b6x5 2.22159506
28b.b7x1 3.15742404
29b.l7x4 1.7925409
30b.l9x6 3.42448508
31b.b10x5 2.44408609
32b.b12x6 4.68879508
33b.b13x7 4.08938567
34b.l13x3 4.8556409
35b.b16x4 4.51704506
36b.b16x5 2.21653405
37b.b16x6 5.3914468
38b.b17x5 3.53612407
39b.l17x3 4.83323509
40b.l17x6 3.71781509
41b.b18x5 2.81427405
42b.l18x1 2.73255606
43b.b19x2 4.13955576
44b.l19x2 3.2036409
45b.b20x4 6.01356408
46b.b20x7 2.21602409
47b.l20x2 2.48434509
48b.b21x1 3.71821407
49b.b21x2 1.66481406
50b.b21x5 3.11133404
51b.b21x7 2.92185505
52b.l22x5 3.01207509
53b.b23x6 3.69209607
54b.l23x1 3.92476406
55b.l24x2 2.06598406
56b.l24x3 1.95125405
57b.l25x3 4.38203529
58b.l25x4 1.79581405
59b.b27x1 1.46122406
60b.l27x1 6.10696659
61b.l27x2 4.03621429
62b.b28x4 4.26771426
63b.b28x6 4.40533529
64g.h1x8 1.6126407
65g.h1x11 1.32318409
66g.l1x4 2.00151508
67g.ctx3 3.29858409
68g.ctx4 2.00753407
69g.ctx6 1.95568406
70g.ctx16 3.13891408
71Lig 17.98312210
72NT 6.98394713
731x39 4.2888408
741x43 3.67595406
751x53 3.66146408
761x59 1.69275504
771x60 2.56178505
782x38 4.22181546
792x40 2.34871408
802x42 4.90953547
812x50 5.75474539
822x53 4.78312506
83E1x50 6.49837718
84E1x52 6.00949407
853x37 4.62903407
863x42 4.61533437
873x50 3.34783509
883x51 4.73308408
893x54 2.56359408
904x50 4.78349539
91E2 13.41161414
925x35 5.19734412
935x58 5.19878609
946x48 6.98489509
956x51 5.81272517
966x59 3.19366405
97E3 4.18744914
987x30 1.84888414
997x42 5.43808407
1007x53 3.50846609
1017x56 2.28985607
102I2x57 3.81006540
103g.ntx4 0.418417400
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
15x58 6x40 34.05493.88954YesNo097
26x40 7x53 35.2753.62617NoYes079
36x36 7x53 1002.61188NoYes079
46x36 7x56 99.91452.71642NoYes077
57x56 8x48 98.25822.05787YesNo075
68x48 I1 98.09824.0775NoNo050
7I1 b.l1x4 97.1382.115NoNo006
8b.l1x4 b.l3x2 96.81791.85259NoYes069
9b.b3x6 b.l3x2 95.85784.20595NoYes099
10b.b3x6 b.l1x3 95.69776.38205NoYes099
11b.b4x4 b.l1x3 95.21766.38789NoYes089
12b.b4x4 b.b4x6 95.05767.21589NoYes089
13b.b3x2 b.b4x6 93.45733.0695NoYes059
14b.b2x5 b.b3x2 93.29734.27084YesNo075
15b.b2x5 b.l26x1 92.33715.57669YesNo077
16b.l26x1 b.l26x3 92.17713.46857NoNo077
17b.l26x3 b.l26x5 91.8572.73229NoNo075
18b.l26x5 g.ctx15 23.20433.95456NoNo059
19b.l4x2 g.ctx15 22.40425.61065NoNo049
20b.l2x5 b.l4x2 21.123914.0709NoNo054
216x51 Lig 23.157810.4792YesYes170
226x48 6x51 25.19923.62226YesYes097
236x44 6x48 26.42389.32928NoYes099
245x54 6x44 27.21156.04484NoNo079
253x47 5x54 27.34315.1551NoNo097
263x47 5x58 31.5979.14929NoYes099
272x53 7x46 62.34044.20868YesNo068
282x50 7x46 67.70884.57013YesNo098
291x50 2x50 29.95018.49033NoYes099
301x50 7x50 30.5999.20958NoNo099
311x53 7x50 72.78253.57042YesNo089
321x53 7x53 72.64364.14146YesYes089
332x50 7x49 29.35887.4032YesNo399
347x49 7x50 42.13323.84575NoNo099
352x42 3x45 17.14066.1414YesNo076
363x45 4x49 17.43913.29556NoNo066
373x42 4x49 17.73685.63634YesNo076
382x46 3x42 22.39773.35162NoYes397
392x46 7x49 12.64426.02551NoNo399
402x53 3x32 49.7395.54567YesNo067
41E1x50 E2 12.46424.17915YesYes184
42E2 Lig 25.03519.1031YesYes140
433x32 Lig 46.30426.8928NoYes170
443x37 5x43 15.11354.7093YesNo075
455x43 Lig 15.20323.33811NoYes150
466x59 6x60 13.27912.629YesNo055
476x60 E3 15.09275.59673NoYes154
483x53 I2x57 11.48053.10325NoYes080
493x53 G.H5.19 11.03072.8275NoNo088
50G.H5.15 G.H5.19 10.85291.32727NoNo088
51G.H5.11 G.H5.15 10.49421.34969NoNo088
52G.H5.11 G.S1.02 10.31642.88508NoNo084
53b.l26x5 g.ctx4 68.49273.40412NoYes057
54g.ctx3 g.ctx4 67.37251.87833YesYes097
55g.ctx3 g.ctx6 57.93073.7573YesYes096
56b.l22x5 g.ctx6 57.29062.66618YesYes096
57b.l22x5 b.l24x2 54.41012.7635YesYes096
58b.h2x5 b.l24x2 53.932.66831NoYes056
59b.h2x1 b.h2x5 53.28991.85772YesNo055
60b.b21x5 b.h2x1 52.00963.67921YesYes045
61b.b21x5 b.b21x7 51.04955.51798YesYes045
62b.b21x7 b.b24x6 44.96833.0158YesNo058
63b.b23x6 b.b24x6 44.80833.52831YesNo078
64b.b23x6 b.l23x2 42.72791.94661YesNo078
65b.l21x7 b.l23x2 42.24783.49071NoNo058
66b.l21x7 b.l23x1 42.08782.81558NoYes056
67b.l23x1 b.l25x6 41.28779.34976YesNo068
68b.l25x6 b.l27x1 41.127610.5565NoYes089
69b.b2x1 b.l27x1 38.72724.36053NoYes589
70b.b2x1 b.l3x1 38.56718.2579NoNo089
71b.l3x1 b.l5x5 38.24713.26061NoYes099
722x46 2x50 10.0383.60825NoYes399
73b.l5x5 b.l7x2 35.20653.13566YesNo099
74G.H2.07 b.l7x2 35.04652.18242YesNo099
75G.H2.07 G.s3h2.03 19.20363.83208YesNo099
76G.s3h2.03 b.l9x6 18.08343.25225NoYes098
77b.l13x6 b.l9x6 10.24194.24474NoYes098
78G.H2.03 b.l13x6 10.08192.42375NoNo099
79G.H2.04 G.H2.07 15.52292.87812NoYes099
80G.H2.04 G.H3.08 15.20282.39616NoNo099
81G.H3.08 G.S4.04 15.04282.88313NoNo099
82G.H3.09 G.S4.04 14.88286.90334YesNo099
83b.l2x3 b.l2x5 17.92331.85566NoNo085
84b.b3x1 b.l2x3 17.76333.02087NoNo058
85b.b3x1 b.b6x5 17.60332.10384NoYes056
86b.b2x4 b.b6x5 12.64231.55325NoYes066
87b.b10x4 b.b2x4 12.48238.37726NoNo066
88b.b10x2 b.b10x4 12.32232.16951NoNo066
89b.b10x2 b.b14x3 12.16232.68869NoNo065
90b.b11x5 b.b14x3 11.84222.83958NoNo065
91b.b11x5 b.l13x7 11.52212.40412NoNo069
92b.l13x3 b.l13x7 11.36213.70602YesNo099
93b.b16x4 b.l13x3 10.24197.89275YesYes069
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
7x34Lig5.823091NoYes5010
LigNT21.70111YesYes0301
E2Lig19.10311YesYes4010
E2x51Lig10.8811NoYes3010
NTNT8.098491YesYes3311
1x357x355.923430NoNo5521
2x533x325.545670YesNo6721
2x537x424.583230YesYes6722
2x603x325.661681NoNo6711
E1x49E28.035061NoYes4421
E1x50E24.179151YesYes8421
3x22E26.470781NoYes4421
4x64E213.89691NoYes4421
4x645x353.994691NoYes4222
4x65E2x526.776930NoNo5521
E2E246.32331YesYes4411
E2E2x5110.50441YesNo4311
E2E2x526.920861YesNo4511
5x35E26.94281YesYes2421
5x36E28.675040NoYes4421
5x39E25.036051NoYes5421
6x517x384.834821YesNo7611
6x547x344.207660NoNo5521
6x61E35.946991NoYes4412
7x387x424.968591NoYes6712
2x60Lig11.02951NoYes6010
3x32Lig6.89281NoYes7010
6x516x556.906291YesNo7612
6x51Lig10.47921YesYes7010
6x58Lig6.611471NoYes4010
6x61Lig4.862831NoYes4010
7x35Lig3.92451NoYes5010
7x38Lig5.581731NoYes6010
E2x52Lig4.011631NoYes5010
3x375x434.70930YesNo7521
6x486x513.622260YesYes9721
E3E34.143431YesYes4422
E3NT3.5921YesYes4321
E2NT3.969691YesYes4311
7x357x393.569381NoNo5412
6x58E34.181881NoYes4412
7x30Lig3.410261YesYes4010
2x562x603.365450NoNo6621
5x43Lig3.338111NoYes5010
6x517x373.220961YesNo7612
7x27Lig3.027450NoYes4010
E1Lig2.6850NoYes0010
7x31Lig2.676520NoYes5010
5x32Lig2.490620NoYes2010
7x24NT2.201060NoYes7321
7x307x332.021YesNo4512
7x307x321.78251YesNo4212
6x62Lig1.479890NoYes5010
2x67E21.38251NoYes4421
7x28NT1.226811NoYes3321
1x28Lig1.11650NoYes4010
6x657x300.182750NoYes1421

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
100.00Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
81.82Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
75.00Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
75.00Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
65.22Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
65.22Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
65.22Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
64.00Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
62.96Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
62.96Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
62.96Consensusbradykinin_onOrthosteric Ligandbk2_on
62.96Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
62.96Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
62.50Consensusangiotensin_onOrthosteric Ligandat1_on
62.50Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
61.90Single6OS2TRV0266OS2-AT1-TRV026
60.87Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
60.00Single6JODAngiotensin II6JOD-AT2-Angiotensin II
60.00Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
60.00Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
60.00Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
60.00Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
57.69Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
57.69Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
56.52Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
56.00Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
55.17Single5GLHEndothelin-15GLH-ETB-Endothelin-1
55.17Single6IGKEndothelin-36IGK-ETB-Endothelin-3
55.17Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
54.55Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
54.55Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
54.17Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
54.17Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
54.17Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
54.17Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
53.57Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
53.33Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
52.00Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
52.00Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
52.00Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
51.85Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
51.85Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
51.72Single8IY6Endothelin-18IY6-ETB-Endothelin-1
51.72Consensusendothelin_onOrthosteric Ligandetb_on eta_on
51.61Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
50.00Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
50.00Single6OS1TRV0266OS1-AT1-TRV026
50.00Single7F1TMIP-1a7F1T-CCR5-MIP-1a
50.00Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
50.00Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
50.00Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
50.00Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
50.00Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
50.00Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
50.00Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
50.00Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
48.39Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
48.28Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
48.28Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
48.28Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
48.15Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
48.00Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
48.00Single8XWNCXCL88XWN-CXCR2-CXCL8
47.83Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
46.67Single6IGLIRL16206IGL-ETB-IRL1620
46.67Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
46.43Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
46.43Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
46.43Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
46.43Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
46.43Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
46.43Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
46.43Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
46.15Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
46.15Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
46.15Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
45.83Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
45.83Consensuschemerin_onOrthosteric Ligandcml1_on
45.16Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
45.16Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
45.00Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
44.83Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
44.83Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
44.83Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
44.44Single3OE0CVX153OE0-CXCR4-CVX15
44.44Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
44.44Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
44.44Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
44.00Single6KNMJN241-96KNM-Apelin-JN241-9
44.00Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
44.00Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
44.00Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
43.75Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
43.48Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
43.48Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
43.33Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
43.33Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
42.86Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
42.86Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
42.86Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
42.86Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
42.86Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
42.86Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
42.31Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
42.31Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
42.31Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
41.94Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
41.67Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
41.67Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
41.67Single8XWSCXCL58XWS-CXCR2-CXCL5
41.67Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
41.38Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
41.38Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
41.38Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
41.38Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
41.38Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
41.38Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
41.38Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
41.38Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
41.38Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
40.91Single6D27CAY104716D27-DP2-CAY10471
40.91Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
40.91Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
40.91Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
40.91Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
40.91Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
40.74Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
40.74Single7SK5CXCL127SK5-ACKR3-CXCL12
40.74Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
40.74Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
40.74Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
40.74Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
40.74Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
40.74Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
40.62Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
40.62Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
40.62Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
40.00Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
40.00Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
40.00Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
40.00Single7SK3CXCL127SK3-ACKR3-CXCL12
40.00Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
40.00Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
40.00Single8XVUCXCL28XVU-CXCR2-CXCL2
40.00Single8XWFCXCL38XWF-CXCR2-CXCL3
40.00Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
40.00Single8ZPLHF511168ZPL-CXCR4-HF51116
40.00Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
40.00Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
39.39Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
39.29Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
39.29Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
39.29Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
39.29Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
39.29Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
39.29Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
39.29Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
39.29Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
39.29Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
39.29Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
39.13Single6D26Fevipiprant6D26-DP2-Fevipiprant
39.13Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
39.13Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
39.13Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
39.13Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
39.13Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
39.13Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
39.13Consensusdp_offOrthosteric Liganddp2_off
38.71Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
38.71Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
38.71Single9KDFRES-701-39KDF-ETB-RES-701-3
38.46Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
38.46Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
38.46Single8XQJJN2418XQJ-Apelin-JN241
38.46Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
38.10Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
38.10Single8GNGIstradefylline8GNG-A2A-Istradefylline
38.10Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
38.10Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
38.10Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
37.93Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
37.93Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
37.93Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
37.50Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
37.50Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
37.50Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
37.50Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
37.50Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
37.14Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
37.04Single4IARErgotamine4IAR-5-HT1B-Ergotamine
37.04Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
37.04Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
37.04Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
37.04Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
37.04Single8WDTphotoNECA8WDT-A2A-photoNECA
37.04Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
37.04Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
37.04Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
37.04Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
37.04Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.67Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
36.67Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
36.67Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
36.67Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
36.67Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
36.36Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
36.36Single7AROLUF58337ARO-A2A-LUF5833-Na
36.36Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
36.36Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
36.36Single8ZPNAMD31008ZPN-CXCR4-AMD3100
36.00Single4XEENeurotensin4XEE-NTS1-Neurotensin
36.00Single4XESNeurotensin4XES-NTS1-Neurotensin
36.00Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
36.00Single6MXTSalmeterol6MXT-β2-Salmeterol
36.00Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
36.00Single6YVRNTS8-136YVR-NTS1-NTS8-13
36.00Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
36.00Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
36.00Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
36.00Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
36.00Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
36.00Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
36.00Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
36.00Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
36.00Single8XQJJN2418XQJ-Apelin-JN241
36.00Single8XWACXCL18XWA-CXCR2-CXCL1
36.00Single8XWMCXCL68XWM-CXCR2-CXCL6
36.00Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
36.00Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
36.00Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
36.00Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
36.00Consensuslpa_offOrthosteric Ligandlpa1_off
36.00Consensuslpl_offOrthosteric Ligands1p_off lpa_off
36.00Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
36.00Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
35.71Single7XNACYN1548067XNA-SST2-CYN154806
35.71Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
35.71Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
35.71Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
35.71Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
35.71Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
35.71Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
35.71Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
35.71Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
35.71Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
35.48Single4XT3Fractalkine4XT3-US28-Fractalkine
35.48Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
35.48Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
34.78Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
34.78Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
34.78Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
34.78Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
34.78Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
34.78Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
34.78Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
34.78Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
34.62Single4BUONeurotensin4BUO-NTS1-Neurotensin
34.62Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
34.62Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
34.62Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
34.62Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
34.62Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
34.62Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
34.62Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
34.62Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
34.62Consensusprostanoid_offOrthosteric Ligandep_off dp_off
34.48Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
34.48Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
34.48Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
34.48Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
34.38Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
34.38Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
34.38Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
34.38Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
33.33Single5N2RPSB-365N2R-A2A-PSB-36-Na
33.33Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
33.33Single5WF6UK-4320975WF6-A2A-UK-432097
33.33Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
33.33Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
33.33Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
33.33Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
33.33Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
33.33Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
33.33Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
33.33Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
33.33Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
33.33Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
33.33Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
33.33Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
33.33Single8TF5Oleic acid8TF5-GPR6-Oleic acid
33.33Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
33.33Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
33.33Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
33.33Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
33.33Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
33.33Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
33.33Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
33.33Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
33.33Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
33.33Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
33.33Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
33.33Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
33.33Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
33.33Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
33.33Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
33.33Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
33.33Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
33.33Consensusvasop-oxy_onOrthosteric Ligandv2_on
33.33Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
32.35Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
32.26Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
32.26Single8ZRTET-18ZRT-ETB-ET-1
32.26Consensuspac_onOrthosteric Ligandpac1_on
32.14Single4XT1Fractalkine4XT1-US28-Fractalkine
32.14Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
32.14Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
32.14Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
32.14Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
32.14Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
32.14Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
32.14Consensuslpl_onOrthosteric Ligands1p_on lpa_on
32.14Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
32.14Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
32.14Consensussomatostatin_offOrthosteric Ligandsst2_off
32.00Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
32.00Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
32.00Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
32.00Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
32.00Single7PX4PSB-21137PX4-A2A-PSB-2113
32.00Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
32.00Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
32.00Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
32.00Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
32.00Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
32.00Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
32.00Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
32.00Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
32.00Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
32.00Consensusneurotensin_onOrthosteric Ligandnts1_on
32.00Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
31.82Single4BWBNeurotensin4BWB-NTS1-Neurotensin
31.82Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
31.82Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
31.82Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
31.82Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
31.82Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
31.82Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
31.82Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
31.43Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
31.25Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
31.25Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
31.25Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
31.25Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
31.25Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
31.25Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
31.25Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
31.03Single3QAKUK-4320973QAK-A2A-UK-432097
31.03Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
31.03Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
31.03Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
31.03Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
31.03Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
30.77Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
30.77Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
30.77Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
30.77Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
30.77Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
30.77Single8JJLOlodaterol8JJL-β2-Olodaterol
30.77Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
30.77Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
30.77Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
30.77Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
30.77Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
30.77Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
30.77Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
30.77Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
30.77Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
30.77Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
30.56Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
30.43Single6MH8ZM-2413856MH8-A2A-ZM-241385
30.43Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
30.43Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
30.43Single7F61PF-036547467F61-H3-PF-03654746
30.43Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
30.43Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
30.43Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
30.43Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
30.43Single8ZPMAMD0708ZPM-CXCR4-AMD070
30.43Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
30.43Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
30.43Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
30.43Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
30.43Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
30.30Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
30.30Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
30.00Single5WF5UK-4320975WF5-A2A-UK-432097
30.00Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
30.00Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
30.00Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
30.00Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
30.00Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
30.00Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
30.00Consensusp2y_offOrthosteric Ligandp2y1_off
29.63Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
29.63Single6IBLArformoterol6IBL-β1-Arformoterol
29.63Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
29.63Single7EZCUKA7EZC-A2A-UKA
29.63Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
29.63Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
29.63Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.63Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
29.63Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
29.63Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
29.63Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.63Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
29.41Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
29.41Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
29.41Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
29.41Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
29.41Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
29.17Single4QIMANTA XV4QIM-SMO-ANTA XV
29.17Single5UENDU1725UEN-A1-DU172
29.17Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
29.17Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
29.17Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
29.17Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
29.17Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
29.17Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
29.17Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
29.17Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
29.17Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
29.17Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
29.17Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
29.17Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
29.17Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
29.17Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
29.17Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
29.17Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
29.17Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
29.17Consensushca_on_gpOrthosteric Ligandhca2_on_gp
29.03Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
29.03Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
29.03Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
29.03Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
29.03Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
29.03Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
29.03Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
29.03Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
28.57Single4XNWMRS25004XNW-P2Y1-MRS2500
28.57Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
28.57Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
28.57Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
28.57Single7XN9L-054,5227XN9-SST2-L-054,522
28.57Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
28.57Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
28.57Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
28.57Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
28.57Single8QJ2pN1628QJ2-MC4-pN162-Gs
28.57Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
28.57Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
28.57Single9IPYJR14a9IPY-C3aB-JR14a
28.57Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
28.57Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
28.57Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
28.21Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
28.21Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
28.12Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
28.12Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
28.12Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
28.12Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
28.12Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
28.00Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
28.00Single5C1MBU725C1M-μ-BU72
28.00Single5IUAQ274563485IUA-A2A-Q27456348-Na
28.00Single5N2SPSB365N2S-A1-PSB36
28.00Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
28.00Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
28.00Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
28.00Single6S0QZM-2413856S0Q-A2A-ZM-241385
28.00Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
28.00Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
28.00Single7C61Ergotamine7C61-5-HT1B-Ergotamine
28.00Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
28.00Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
28.00Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
28.00Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
28.00Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
28.00Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
28.00Single8S4DCMF-0198S4D-Apelin-CMF-019
28.00Single9EHSLUF76029EHS-A3A-LUF7602
28.00Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
28.00Consensusadenosine_offOrthosteric Liganda1_off a2_off
28.00Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
28.00Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
28.00Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
27.78Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
27.78Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
27.59Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
27.59Single7F8XNN90567F8X-CCKA-NN9056
27.59Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
27.59Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
27.59Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
27.59Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
27.59Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
27.59Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
27.59Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.59Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
27.59Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
27.59Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
27.50Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
27.27Single3OE9IT1t3OE9-CXCR4-IT1t
27.27Single4O9RCyclopamine4O9R-SMO-Cyclopamine
27.27Single6FJ3PTH6FJ3-PTH1-PTH
27.27Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
27.27Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
27.27Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
27.27Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
27.27Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
26.92Single3P0GBI1671073P0G-β2-BI167107
26.92Single4BV0Neurotensin4BV0-NTS1-Neurotensin
26.92Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
26.92Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
26.92Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
26.92Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
26.92Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
26.92Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
26.92Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
26.92Single7TUYGSK682753A7TUY-GPR183-GSK682753A
26.92Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
26.92Single8E0GBU728E0G-μ-BU72
26.92Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
26.92Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
26.92Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
26.92Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
26.92Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
26.92Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
26.92Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
26.92Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
26.92Single8ZWFJR14a8ZWF-C3aB-JR14a
26.92Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
26.92Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
26.92Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
26.92Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
26.92Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
26.92Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
26.92Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
26.92Consensuslpa_onOrthosteric Ligandlpa1_on
26.92Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
26.92Consensusrelaxin_onOrthosteric Ligandrxfp4_on
26.92Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
26.92Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
26.92Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
26.67Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
26.67Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
26.67Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
26.67Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
26.67Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
26.67Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
26.67Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
26.67Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
26.47Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
26.47Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
26.47Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
26.47Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
26.47Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
26.47Consensusglp_onOrthosteric Ligandglp1_on glp2_on
26.47Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
26.09Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
26.09Single3PWHZM-2413853PWH-A2A-ZM-241385
26.09Single4QINSAG1.54QIN-SMO-SAG1.5
26.09Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
26.09Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
26.09Single7BR3Elagolix7BR3-GnRH1-Elagolix
26.09Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
26.09Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
26.09Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
26.09Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
26.09Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
26.09Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
26.09Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
26.09Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
26.09Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
26.09Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
26.09Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
26.09Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
26.09Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
25.93Single4RWADIPP-NH24RWA-δ-DIPP-NH2
25.93Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
25.93Single6A93Risperidone6A93-5-HT2A-Risperidone
25.93Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
25.93Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
25.93Single7K15MKD0467K15-BLT1-MKD046-Na
25.93Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
25.93Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
25.93Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
25.93Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
25.93Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
25.93Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
25.93Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
25.93Single8JJ8Formoterol8JJ8-β2-Formoterol
25.93Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
25.93Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
25.93Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
25.93Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
25.93Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
25.93Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
25.93Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
25.93Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
25.93Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
25.93Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
25.93Consensusorexin_onOrthosteric Ligandox2_on
25.81Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
25.81Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
25.81Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
25.81Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
25.81Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
25.81Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.81Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
25.71Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
25.71Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
25.71Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
25.71Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
25.71Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
25.71Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
25.71Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
25.71Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
25.64Consensuspth_onOrthosteric Ligandpth1_on pth2_on
25.00Single3REYXAC3REY-A2A-XAC
25.00Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
25.00Single5IUBQ274563445IUB-A2A-Q27456344-Na
25.00Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
25.00Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
25.00Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
25.00Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
25.00Single6AQFZM-2413856AQF-A2A-ZM-241385
25.00Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
25.00Single6KUXRS-799486KUX-α2a-RS-79948
25.00Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
25.00Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
25.00Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
25.00Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
25.00Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
25.00Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
25.00Single7T32ZM-2413857T32-A2A-ZM-241385
25.00Single7UL3Famotidine7UL3-H2-Famotidine
25.00Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
25.00Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
25.00Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
25.00Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
25.00Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
25.00Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
25.00Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
25.00Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
25.00Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
25.00Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
25.00Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
25.00Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
25.00Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
25.00Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
25.00Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
25.00Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
25.00Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
25.00Single8K5CAcipimox8K5C-HCA2-Acipimox
25.00Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
25.00Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
25.00Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
25.00Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
25.00Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
25.00Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
25.00Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
25.00Single9BA0A1AKN9BA0-CB1-A1AKN
25.00Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
25.00Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
25.00Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
25.00Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
25.00Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.00Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.00Consensusbombesin_onOrthosteric Ligandbb2_on
25.00Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
25.00Consensuscck_onOrthosteric Ligandccka_on cckb_on
25.00Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
25.00Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
25.00Consensusgrh_offOrthosteric Ligandgnrh1_off
25.00Consensushca_onOrthosteric Ligandhca2_on
25.00Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
25.00Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
25.00Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
24.44Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
24.39Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
24.32Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
24.24Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
24.24Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
24.24Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
24.24Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
24.24Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
24.24Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
24.24Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
24.14Single3NY9ICI118-5513NY9-β2-ICI118-551
24.14Single4UG2CGS216804UG2-A2A-CGS21680
24.14Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
24.14Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single7SK9CCX6627SK9-ACKR3-CCX662
24.14Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
24.14Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
24.14Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
24.14Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
24.14Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
24.14Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
24.14Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
24.14Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
24.14Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
24.00Single2Y01Dobutamine2Y01-β1-Dobutamine
24.00Single2Y02Carmoterol2Y02-β1-Carmoterol
24.00Single3EMLZM-2413853EML-A2A-ZM-241385
24.00Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
24.00Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
24.00Single5IU8Q274563475IU8-A2A-Q27456347-Na
24.00Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
24.00Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
24.00Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
24.00Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
24.00Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
24.00Single5T04Neurotensin5T04-NTS1-Neurotensin
24.00Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
24.00Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
24.00Single6S0LZM-2413856S0L-A2A-ZM-241385
24.00Single7BU7BI1671077BU7-β1-BI167107
24.00Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
24.00Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
24.00Single7PYRPSB-21157PYR-A2A-PSB-2115
24.00Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
24.00Single7UL4Alvimopan7UL4-μ-Alvimopan
24.00Single7V3ZCP559407V3Z-CB1-CP55940
24.00Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
24.00Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
24.00Single8CU6LJ-45178CU6-A2A-LJ-4517
24.00Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
24.00Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
24.00Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
24.00Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
24.00Single8K5DGSK2560738K5D-HCA2-GSK256073
24.00Single8T1WCVN4248T1W-GPR6-CVN424
24.00Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
24.00Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
24.00Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
24.00Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
24.00Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
24.00Single9CHXS-Carazolol9CHX-β2-S-Carazolol
24.00Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
24.00Single9H37A1IR09H37-A2A-A1IR0-Na
24.00Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
24.00Consensusa3_onOrthosteric Liganda3a_on
24.00Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
24.00Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
24.00Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
24.00Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
24.00Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
24.00Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
23.81Single8A2OTheophylline8A2O-A2A-Theophylline-Na
23.68Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
23.68Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
23.68Consensuscrf_on_gpOrthosteric Ligandcrf2_on_gp crf1_on_gp
23.53Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
23.53Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
23.53Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
23.53Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
23.53Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
23.53Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
23.53Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
23.53Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
23.53Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
23.33Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
23.33Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
23.33Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
23.33Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.33Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
23.33Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
23.33Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
23.33Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
23.33Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
23.33Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
23.26Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
23.08Single2Y00Dobutamine2Y00-β1-Dobutamine
23.08Single4JKVTaladegib4JKV-SMO-Taladegib
23.08Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
23.08Single6E67BI1671076E67-β2-BI167107-Gs(CT)
23.08Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
23.08Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
23.08Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
23.08Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
23.08Single6Z4SSR486926Z4S-NTS1-SR48692
23.08Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
23.08Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
23.08Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
23.08Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
23.08Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
23.08Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
23.08Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
23.08Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
23.08Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
23.08Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
23.08Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
23.08Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
23.08Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8GNEKW-63568GNE-A2A-KW-6356-Na
23.08Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
23.08Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
23.08Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
23.08Single8JXSPF-61428JXS-D1-PF-6142
23.08Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
23.08Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
23.08Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
23.08Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
23.08Single9B9ZA1AKO9B9Z-CB1-A1AKO
23.08Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
23.08Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
23.08Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
23.08Consensusa3_on_gpOrthosteric Liganda3a_on_gp
23.08Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.08Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
23.08Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
23.08Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
23.08Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
23.08Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
23.08Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
23.08Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
23.08Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
23.08Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
23.08Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
23.08Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.08Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
23.08Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
23.08Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
23.08Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
23.08Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
23.08Consensustrace-amine_onOrthosteric Ligandta1_on
22.86Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
22.86Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
22.86Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
22.86Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
22.86Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
22.86Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
22.86Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
22.86Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
22.86Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
22.73Single3OE6IT1t3OE6-CXCR4-IT1t
22.73Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
22.73Single6ME5Agomelatine6ME5-MT1-Agomelatine
22.73Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
22.73Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
22.73Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
22.73Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.73Single8JPSCCL78JPS-ACKR1-CCL7
22.73Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
22.73Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
22.58Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
22.58Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
22.58Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
22.58Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
22.58Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
22.58Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
22.58Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
22.58Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
22.58Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
22.50Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
22.22Single2YDVNECA2YDV-A2A-NECA
22.22Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
22.22Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
22.22Single4UHRCGS216804UHR-A2A-CGS21680
22.22Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
22.22Single5G53NECA5G53-A2A-NECA-Gs
22.22Single5V56TC1145V56-SMO-TC114
22.22Single5V57TC1145V57-SMO-TC114
22.22Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
22.22Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
22.22Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
22.22Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
22.22Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
22.22Single6WGTLSD6WGT-5-HT2A-LSD
22.22Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
22.22Single7B6WCyclazosin7B6W-α1b-Cyclazosin
22.22Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
22.22Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
22.22Single7R0CAVP7R0C-V2-AVP-Arrestin2
22.22Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
22.22Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
22.22Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
22.22Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
22.22Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
22.22Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
22.22Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
22.22Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
22.22Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
22.22Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
22.22Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
22.22Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
22.22Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
22.22Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
22.22Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
22.22Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
22.22Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
22.22Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.22Consensusa2_onOrthosteric Liganda2b_on
22.22Consensusa2_on_gpOrthosteric Liganda2b_on_gp
22.22Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
22.22Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
22.22Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
22.22Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
22.22Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
22.22Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
22.22Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
22.22Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
22.22Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
22.22Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
22.22Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
21.88Single6PT2KGCHM076PT2-δ-KGCHM07
21.88Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
21.88Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
21.88Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
21.88Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
21.88Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.88Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
21.88Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
21.88Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
21.88Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
21.74Single5L7IVismodegib5L7I-SMO-Vismodegib
21.74Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
21.74Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
21.74Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
21.74Single8K5BNiacin8K5B-HCA2-Niacin
21.74Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
21.74Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
21.74Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
21.74Single9B9Y7DY9B9Y-CB1-7DY
21.74Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
21.74Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
21.74Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
21.74Consensusgq_nucleotideOrthosteric Ligandgq_p2y
21.74Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
21.62Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
21.62Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
21.43Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
21.43Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
21.43Single4AMIBucindolol4AMI-β1-Bucindolol
21.43Single4LDEBI1671074LDE-β2-BI167107
21.43Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
21.43Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
21.43Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
21.43Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
21.43Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
21.43Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
21.43Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
21.43Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.43Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
21.43Single7YITNalfurafine7YIT-κ-Nalfurafine
21.43Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
21.43Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
21.43Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
21.43Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
21.43Single8XYIVUF106618XYI-CXCR3-VUF10661
21.43Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
21.43Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
21.43Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
21.43Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
21.43Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
21.43Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
21.43Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
21.43Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
21.43Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
21.43Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
21.43Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
21.43Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
21.43Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
21.43Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
21.43Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
21.43Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.43Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.21Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
21.21Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
21.21Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
21.21Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
21.21Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
21.21Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
21.05Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
21.05Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
21.05Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
21.05Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.83Single3ODUIT1t3ODU-CXCR4-IT1t
20.83Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
20.83Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
20.83Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
20.83Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
20.83Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
20.83Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
20.83Single5WS3EMPA5WS3-OX2-EMPA
20.83Single5ZKQABT-4915ZKQ-PAF-ABT-491
20.83Single6AKXA4R6AKX-CCR5-A4R
20.83Single6AKYMaraviroc6AKY-CCR5-Maraviroc
20.83Single6DS0Ly2660976DS0-5-HT2B-Ly266097
20.83Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
20.83Single6ME9Ramelteon6ME9-MT2-Ramelteon
20.83Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
20.83Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
20.83Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.83Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
20.83Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
20.83Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
20.83Single7F8ULintitript7F8U-CCKA-Lintitript
20.83Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
20.83Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
20.83Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
20.83Single7XRRLemborexant7XRR-OX2-Lemborexant
20.83Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
20.83Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
20.83Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.83Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
20.83Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
20.83Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
20.83Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
20.83Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
20.83Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.83Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
20.83Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
20.83Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
20.83Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
20.83Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
20.83Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
20.83Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
20.83Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
20.83Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
20.83Consensusorexin_offOrthosteric Ligandox2_off ox1_off
20.83Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
20.83Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
20.83Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
20.83Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
20.83Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
20.69Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
20.69Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
20.69Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
20.69Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
20.69Single6H7LDobutamine6H7L-β1-Dobutamine
20.69Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
20.69Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
20.69Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
20.69Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
20.69Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
20.69Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
20.69Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
20.69Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
20.69Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
20.69Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
20.69Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
20.69Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
20.69Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.69Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
20.69Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
20.69Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.69Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
20.69Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
20.69Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
20.69Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
20.69Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
20.69Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
20.69Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
20.59Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
20.59Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
20.59Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
20.59Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
20.51Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
20.51Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
20.51Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.51Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
20.00Single2YDOAdenosine2YDO-A2A-Adenosine
20.00Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
20.00Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
20.00Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
20.00Single4MBSMaraviroc4MBS-CCR5-Maraviroc
20.00Single4ZJCSB-6740424ZJC-OX1-SB-674042
20.00Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
20.00Single5IU7Q274563465IU7-A2A-Q27456346-Na
20.00Single5JTBZM-2413855JTB-A2A-ZM-241385
20.00Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
20.00Single5UVIZM-2413855UVI-A2A-ZM-241385
20.00Single5ZTYAM102575ZTY-CB2-AM10257
20.00Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
20.00Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
20.00Single6PS0S-Carazolol6PS0-β2-S-Carazolol
20.00Single6PS4ICI118-5516PS4-β2-ICI118-551
20.00Single6PS5S-Propranolol6PS5-β2-S-Propranolol
20.00Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
20.00Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
20.00Single6PT3DPI-2876PT3-δ-DPI-287
20.00Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
20.00Single6TPGEMPA6TPG-OX2-EMPA
20.00Single6V9SGTPL114036V9S-OX1-GTPL11403
20.00Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
20.00Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
20.00Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
20.00Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
20.00Single6ZINSR486926ZIN-NTS1-SR48692
20.00Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
20.00Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
20.00Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
20.00Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
20.00Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
20.00Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
20.00Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
20.00Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
20.00Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
20.00Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
20.00Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
20.00Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
20.00Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
20.00Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
20.00Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
20.00Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
20.00Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
20.00Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
20.00Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
20.00Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
20.00Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
20.00Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
20.00Single8IHKAcifran8IHK-HCA3-Acifran
20.00Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
20.00Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
20.00Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
20.00Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
20.00Single8RLNLUF58348RLN-A2A-LUF5834
20.00Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
20.00Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
20.00Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
20.00Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
20.00Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
20.00Single8X5YAstemizole8X5Y-H1-Astemizole
20.00Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
20.00Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
20.00Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
20.00Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
20.00Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
20.00Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
20.00Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
20.00Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
20.00Consensusa2_offOrthosteric Liganda2a_off
20.00Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
20.00Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
20.00Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
20.00Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
20.00Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
20.00Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
19.51Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
19.51Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
19.44Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
19.44Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
19.44Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
19.44Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
19.35Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
19.35Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
19.35Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
19.35Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
19.35Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
19.35Single8WKYPG-9348WKY-MC4-PG-934
19.35Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
19.23Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
19.23Single2Y04Salbutamol2Y04-β1-Salbutamol
19.23Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
19.23Single3NY8ICI118-5513NY8-β2-ICI118-551
19.23Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
19.23Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
19.23Single4EJ4Naltrindole4EJ4-δ-Naltrindole
19.23Single4GBRS-Carazolol4GBR-β2-S-Carazolol
19.23Single4QKX35V4QKX-β2-35V
19.23Single5TGZAM65385TGZ-CB1-AM6538
19.23Single5UIGCmpd-15UIG-A2A-Cmpd-1
19.23Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
19.23Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
19.23Single6H7MSalbutamol6H7M-β1-Salbutamol
19.23Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
19.23Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
19.23Single6PS1Timolol6PS1-β2-Timolol
19.23Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
19.23Single6TOTLemborexant6TOT-OX1-Lemborexant
19.23Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
19.23Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
19.23Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
19.23Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
19.23Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
19.23Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
19.23Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
19.23Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
19.23Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
19.23Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
19.23Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
19.23Single7WC7Lisuride7WC7-5-HT2A-Lisuride
19.23Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
19.23Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
19.23Single7YXAONO-54306087YXA-S1P5-ONO-5430608
19.23Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
19.23Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
19.23Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
19.23Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
19.23Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
19.23Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
19.23Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
19.23Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
19.23Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
19.23Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
19.23Single8JXRLSD8JXR-D1-LSD
19.23Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
19.23Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.23Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
19.23Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
19.23Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
19.23Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
19.23Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
19.23Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
19.23Consensus5ht5_onOrthosteric Ligand5ht5a_on
19.23Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
19.23Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
19.23Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
19.23Consensuscck_offOrthosteric Ligandccka_off
19.23Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
19.23Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
19.23Consensusdopamine_offOrthosteric Ligandd2_off d3_off
19.23Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
19.23Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
19.23Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
19.23Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
19.05Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
19.05Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
19.05Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
19.05Single8PWNTheophylline8PWN-A2A-Theophylline
19.05Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
18.92Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
18.92Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
18.92Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
18.92Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
18.92Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
18.75Single6HLOAprepitant6HLO-NK1-Aprepitant
18.75Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
18.75Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
18.75Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
18.75Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
18.75Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
18.60Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
18.52Single2RH1S-Carazolol2RH1-β2-S-Carazolol
18.52Single2Y03Isoprenaline2Y03-β1-Isoprenaline
18.52Single2YCWS-Carazolol2YCW-β1-S-Carazolol
18.52Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
18.52Single5D6LS-Carazolol5D6L-β2-S-Carazolol
18.52Single5JQHS-Carazolol5JQH-β2-S-Carazolol
18.52Single5TVNLSD5TVN-5-HT2B-LSD
18.52Single5WIUNemonapride5WIU-D4-Nemonapride
18.52Single5WIVNemonapride5WIV-D4-Nemonapride-Na
18.52Single5WQCEMPA5WQC-OX2-EMPA
18.52Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
18.52Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
18.52Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
18.52Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
18.52Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
18.52Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
18.52Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
18.52Single6TP6Filorexant6TP6-OX1-Filorexant
18.52Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
18.52Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
18.52Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
18.52Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
18.52Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
18.52Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
18.52Single7W41PD1762527W41-BB2-PD176252
18.52Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
18.52Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
18.52Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.52Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
18.52Single8QOTNanobody-E8QOT-μ-Nanobody-E
18.52Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
18.52Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
18.52Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
18.52Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
18.52Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
18.52Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
18.52Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.52Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
18.52Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
18.52Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
18.52Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
18.52Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
18.52Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
18.52Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
18.52Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
18.52Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
18.52Consensusamine_offonOrthosteric Ligandamine_off amine_on
18.52Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
18.52Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
18.52Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
18.52Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
18.52Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
18.52Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
18.52Consensusblt_offOrthosteric Ligandblt1_off
18.52Consensusbombesin_offOrthosteric Ligandbb2_off
18.52Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
18.52Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
18.52Consensusep_offOrthosteric Ligandep4_off
18.52Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
18.42Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
18.42Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
18.42Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
18.42Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
18.18Single3RFMCaffeine3RFM-A2A-Caffeine
18.18Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
18.18Single6W25SHU91196W25-MC4-SHU9119-Ca
18.18Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
18.18Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
18.18Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
18.18Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
18.18Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
18.18Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
18.18Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
18.18Consensussensory_onOrthosteric Ligandopsins_on
17.95Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
17.95Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
17.86Single5D5AS-Carazolol5D5A-β2-S-Carazolol
17.86Single5D5BS-Carazolol5D5B-β2-S-Carazolol
17.86Single5XR8AM8415XR8-CB1-AM841
17.86Single5XRAAM115425XRA-CB1-AM11542
17.86Single6H7JIsoprenaline6H7J-β1-Isoprenaline
17.86Single6J21Aprepitant6J21-NK1-Aprepitant
17.86Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
17.86Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
17.86Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
17.86Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
17.86Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
17.86Single7FEECP559407FEE-CB1-CP55940-ZCZ011
17.86Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
17.86Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
17.86Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
17.86Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
17.86Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
17.86Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
17.86Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
17.86Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
17.86Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
17.86Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
17.86Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
17.86Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
17.86Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
17.86Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.86Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
17.86Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
17.86Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
17.86Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
17.86Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
17.86Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
17.86Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
17.86Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.86Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
17.86Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
17.86Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
17.86Single9BJKNaloxone9BJK-μ-Naloxone-NAM
17.86Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
17.86Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
17.86Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
17.86Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
17.86Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
17.86Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
17.86Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.86Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
17.86Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
17.86Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
17.86Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
17.78Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
17.65Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
17.65Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
17.65Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
17.50Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
17.50Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
17.39Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
17.39Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
17.39Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
17.39Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
17.39Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
17.39Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
17.39Single7WC5Psilocin7WC5-5-HT2A-Psilocin
17.39Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.39Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
17.39Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
17.39Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
17.39Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
17.39Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
17.39Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
17.39Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
17.39Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
17.24Single3D4STimolol3D4S-β2-Timolol
17.24Single4N4WSANT-14N4W-SMO-SANT-1
17.24Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
17.24Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
17.24Single4PY02MeSATP4PY0-P2Y12-2MeSATP
17.24Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
17.24Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
17.24Single6CM4Risperidone6CM4-D2-Risperidone
17.24Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
17.24Single6KQICP559406KQI-CB1-CP55940-Org27569
17.24Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
17.24Single7DFPSpiperone7DFP-D2-Spiperone
17.24Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
17.24Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
17.24Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
17.24Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
17.24Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
17.24Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
17.24Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
17.24Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
17.24Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
17.24Single8JWY2-1188JWY-A2A-2-118
17.24Single8JWZAB9288JWZ-A2A-AB928-Na
17.24Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
17.24Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
17.24Single9DGIZ85267113509DGI-CB1-Z8526711350
17.24Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
17.24Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
17.24Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
17.24Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
17.24Consensusalpha1_offOrthosteric Ligandalpha1a_off
17.24Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
17.24Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
17.24Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
17.14Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
17.14Consensuscalcitonin_onOrthosteric Ligandctlike_on
17.14Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
17.14Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
17.14Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
17.14Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
17.07Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
17.07Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
17.07Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.07Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
16.67Single3PBLEticlopride3PBL-D3-Eticlopride
16.67Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
16.67Single5X93K-87945X93-ETB-K-8794
16.67Single6HLLCP999946HLL-NK1-CP99994
16.67Single6LI0C176LI0-GPR52-C17
16.67Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
16.67Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
16.67Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
16.67Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
16.67Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
16.67Single7UL2SR486927UL2-NTS1-SR48692-Na
16.67Single7UM4AS26747237UM4-5-HT5A-AS2674723
16.67Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
16.67Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
16.67Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
16.67Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
16.67Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
16.67Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
16.67Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
16.67Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
16.67Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
16.67Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
16.67Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
16.67Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
16.67Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
16.67Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
16.67Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
16.67Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
16.67Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
16.67Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
16.67Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
16.67Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
16.67Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
16.67Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
16.67Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
16.67Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
16.67Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
16.67Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
16.67Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
16.67Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
16.67Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
16.67Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
16.67Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
16.67Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
16.67Consensusendothelin_offOrthosteric Ligandetb_off
16.67Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
16.67Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusneurotensin_offOrthosteric Ligandnts1_off
16.67Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
16.67Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
16.67Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
16.22Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
16.22Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
16.22Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
16.22Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
16.13Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
16.13Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
16.13Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
16.13Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
16.13Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
16.13Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
16.00Single4S0VSuvorexant4S0V-OX2-Suvorexant
16.00Single5U09Taranabant5U09-CB1-Taranabant
16.00Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
16.00Single6ME2Ramelteon6ME2-MT1-Ramelteon
16.00Single6TODEMPA6TOD-OX1-EMPA-Na
16.00Single6TPJSuvorexant6TPJ-OX2-Suvorexant
16.00Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
16.00Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
16.00Single7F8YDevazepide7F8Y-CCKA-Devazepide
16.00Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.00Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
16.00Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
16.00Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
16.00Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
16.00Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
16.00Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
16.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
16.00Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
16.00Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
16.00Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
16.00Single8IWESpermidine8IWE-TA9-Spermidine
16.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
16.00Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
16.00Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
16.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
16.00Single8Y0HVUF114188Y0H-CXCR3-VUF11418
16.00Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
16.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
16.00Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
16.00Single9H2XA1IR19H2X-A2A-A1IR1-Na
16.00Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
16.00Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
16.00Consensusalpha2_offOrthosteric Ligandalpha2c_off
16.00Consensusangiotensin_offOrthosteric Ligandat1_off
16.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
16.00Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
16.00Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
16.00Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
16.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
16.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
15.79Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
15.79Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
15.79Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
15.79Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
15.62Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
15.62Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
15.62Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
15.62Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
15.62Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.62Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
15.62Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
15.62Single8KIGSHU91198KIG-MC3-SHU9119-Ca
15.62Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
15.56Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
15.38Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
15.38Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
15.38Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
15.38Single6A94Zotepine6A94-5-HT2A-Zotepine
15.38Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
15.38Single6TP3Nemorexant6TP3-OX1-Nemorexant
15.38Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
15.38Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
15.38Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
15.38Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
15.38Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
15.38Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
15.38Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
15.38Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
15.38Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
15.38Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.38Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
15.38Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
15.38Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
15.38Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
15.38Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
15.38Single8K2WAMG4878K2W-CXCR3-AMG487
15.38Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
15.38Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
15.38Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.38Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
15.38Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
15.38Single9AS5Mescaline9AS5-5-HT2A-Mescaline
15.38Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
15.38Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
15.38Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
15.38Consensusalpha1_onOrthosteric Ligandalpha1a_on
15.38Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
15.38Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
15.38Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
15.38Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
15.38Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
15.38Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
15.38Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
15.38Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
15.38Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
15.15Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
15.15Single8IEBA1LYA8IEB-GPR156-A1LYA
15.15Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.81Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
14.81Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
14.81Single4YAYZD-71554YAY-AT1-ZD-7155
14.81Single6DRXLisuride6DRX-5-HT2B-Lisuride
14.81Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
14.81Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
14.81Single6GPSMK08126GPS-CCR2-MK0812
14.81Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
14.81Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
14.81Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
14.81Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
14.81Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
14.81Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
14.81Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
14.81Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
14.81Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
14.81Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
14.81Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
14.81Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
14.81Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
14.81Single8JJOAlprenolol8JJO-β2-Alprenolol
14.81Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
14.81Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
14.81Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
14.81Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
14.81Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
14.81Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
14.81Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
14.81Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
14.81Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
14.81Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
14.81Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
14.81Single9AS1DMT9AS1-5-HT2A-DMT
14.81Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
14.81Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
14.81Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
14.81Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
14.81Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
14.81Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
14.81Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
14.81Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
14.81Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
14.81Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
14.81Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
14.81Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
14.81Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
14.81Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
14.81Consensusblt_onOrthosteric Ligandblt1_on
14.81Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
14.81Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
14.81Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
14.81Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
14.81Consensusleukotriene_onOrthosteric Ligandblt_on
14.81Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
14.71Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
14.71Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.71Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.63Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
14.29Single4NTJAZD12834NTJ-P2Y12-AZD1283
14.29Single5MZPCaffeine5MZP-A2A-Caffeine-Na
14.29Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
14.29Single5XPRBosentan5XPR-ETB-Bosentan
14.29Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
14.29Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
14.29Single6GPXMK08126GPX-CCR2-MK0812
14.29Single6LUQHaloperidol6LUQ-D2-Haloperidol
14.29Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
14.29Single6PS6Timolol6PS6-β2-Timolol
14.29Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
14.29Single7C4SS1P7C4S-S1P3-S1P
14.29Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
14.29Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
14.29Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
14.29Single7SINNPS-21437SIN-CaS-NPS-2143
14.29Single7SINNPS-21437SIN-CaS-NPS-2143
14.29Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
14.29Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
14.29Single7WC6LSD7WC6-5-HT2A-LSD
14.29Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
14.29Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
14.29Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
14.29Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
14.29Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
14.29Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
14.29Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
14.29Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
14.29Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
14.29Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
14.29Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
14.29Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
14.29Single8ZMFA1L108ZMF-5-HT2C-A1L10
14.29Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
14.29Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
14.29Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
14.29Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
14.29Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
14.29Single9HAPTolvaptan9HAP-V2-Tolvaptan
14.29Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
14.29Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
14.29Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
14.29Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
14.29Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
14.29Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
13.89Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
13.79Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
13.79Single4DJHJDTic4DJH-κ-JDTic
13.79Single4U15Tiotropium4U15-M3-Tiotropium
13.79Single5TZRMK86665TZR-FFA1-MK8666
13.79Single5V54Methiothepin5V54-5-HT1B-Methiothepin
13.79Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
13.79Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
13.79Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
13.79Single6OL9Tiotropium6OL9-M5-Tiotropium
13.79Single6TQ7SB-3348676TQ7-OX1-SB-334867
13.79Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
13.79Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
13.79Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
13.79Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.79Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
13.79Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
13.79Single8XVLZibotentan8XVL-ETA-Zibotentan
13.79Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
13.79Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
13.79Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.79Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
13.79Consensus5ht1_offOrthosteric Ligand5ht1b_off
13.79Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
13.79Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
13.79Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
13.79Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.79Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
13.79Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
13.79Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
13.79Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
13.79Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
13.79Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
13.79Consensustachykinin_offOrthosteric Ligandnk1_off
13.64Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
13.64Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
13.64Single7WC4Serotonin7WC4-5-HT2A-Serotonin
13.64Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
13.64Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
13.51Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
13.51Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
13.33Single5CXVTiotropium5CXV-M1-Tiotropium
13.33Single5X33BIIL2605X33-BLT1-BIIL260
13.33Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
13.33Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
13.33Single6ZG4HTL00099366ZG4-M1-HTL0009936
13.33Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
13.33Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
13.33Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
13.33Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
13.33Single9BJKNAM9BJK-μ-Naloxone-NAM
13.33Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.33Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
13.33Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
13.33Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
13.33Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
13.16Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
13.16Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
13.16Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
13.04Single3OE8IT1t3OE8-CXCR4-IT1t
13.04Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
13.04Single6TQ9SB-4081246TQ9-OX1-SB-408124
13.04Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
13.04Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
13.04Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.04Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
13.04Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
13.04Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
13.04Single9CHUNoradrenaline9CHU-β2-Noradrenaline
13.04Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
13.04Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
12.90Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
12.90Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
12.90Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
12.90Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.90Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
12.82Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
12.82Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
12.50Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
12.50Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
12.50Single3UZAGTPL92363UZA-A2A-GTPL9236
12.50Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
12.50Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
12.50Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
12.50Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.50Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
12.50Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
12.50Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
12.50Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
12.50Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
12.50Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
12.50Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
12.50Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
12.50Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
12.50Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
12.50Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
12.50Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
12.50Single9LRCHistamine9LRC-H4-Histamine
12.50Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
12.50Consensus5ht2_onOrthosteric Ligand5ht2b_on
12.50Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
12.50Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
12.50Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Consensusgi_sensoryOrthosteric Ligandgi_opsins
12.50Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
12.50Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.50Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
12.50Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
12.50Consensuskisspeptin_onOrthosteric Ligandkiss1_on
12.50Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.50Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
12.12Single7QA8Peptide7QA8-STE2-Peptide
12.12Single7QA8Peptide7QA8-STE2-Peptide
12.12Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single8IEBA1LYA8IEB-GPR156-A1LYA
12.12Single8IEIA1LYA8IEI-GPR156-A1LYA
12.12Single8IEIA1LYA8IEI-GPR156-A1LYA
12.12Single8IEPA1LYA8IEP-GPR156-A1LYA
12.12Single8IEPA1LYA8IEP-GPR156-A1LYA
12.12Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
12.12Single9M4TSilodosin9M4T-Alpha1A-Silodosin
12.12Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
12.12Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
12.12Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
12.00Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
12.00Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
12.00Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
12.00Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
12.00Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
12.00Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
12.00Single6TP4ACT-4622066TP4-OX1-ACT-462206
12.00Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
12.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.00Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
12.00Single7SRQLSD7SRQ-5-HT2B-LSD
12.00Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
12.00Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
12.00Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
12.00Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
12.00Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.00Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
12.00Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
12.00Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
12.00Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.00Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
12.00Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
12.00Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
12.00Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
12.00Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
12.00Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
11.54Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
11.54Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
11.54Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
11.54Single6B73MP11046B73-κ-MP1104
11.54Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
11.54Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
11.54Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
11.54Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
11.54Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
11.54Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
11.54Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
11.54Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
11.54Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
11.54Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.54Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.54Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
11.54Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
11.54Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
11.54Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
11.54Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
11.54Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
11.54Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
11.54Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
11.54Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
11.54Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
11.54Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
11.54Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
11.54Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
11.54Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
11.54Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
11.54Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
11.54Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
11.54Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
11.54Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.54Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.54Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
11.54Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
11.54Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
11.54Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.54Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
11.11Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
11.11Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
11.11Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
11.11Single6IQLL7458706IQL-D4-L745870
11.11Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
11.11Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
11.11Single6TPNHTL66416TPN-OX2-HTL6641
11.11Single6VI4JDTic6VI4-κ-JDTic
11.11Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
11.11Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
11.11Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
11.11Single6ZG9GSK10347026ZG9-M1-GSK1034702
11.11Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
11.11Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
11.11Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
11.11Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
11.11Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
11.11Single7VODCariprazine7VOD-5-HT2A-Cariprazine
11.11Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
11.11Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
11.11Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
11.11Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
11.11Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
11.11Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
11.11Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
11.11Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
11.11Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
11.11Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
11.11Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
11.11Single9ARXSerotonin9ARX-5-HT2A-Serotonin
11.11Single9AS3LSD9AS3-5-HT2A-LSD
11.11Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
11.11Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
11.11Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
11.11Consensusopsins_offOrthosteric Ligandrhodopsin_off
11.11Consensussensory_offOrthosteric Ligandopsins_off
10.81Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
10.71Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
10.71Single4DAJTiotropium4DAJ-M3-Tiotropium
10.71Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
10.71Single4MQSIperoxo4MQS-M2-Iperoxo
10.71Single4U14Tiotropium4U14-M3-Tiotropium
10.71Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
10.71Single5DHHSB-6121115DHH-NOP-SB-612111
10.71Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
10.71Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
10.71Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
10.71Single6IIVDaltroban6IIV-TXA2-Daltroban
10.71Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.71Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
10.71Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.71Single7F83PF-051904577F83-Ghrelin-PF-05190457
10.71Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
10.71Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
10.71Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
10.71Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
10.71Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.71Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
10.71Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
10.71Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
10.71Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
10.71Single8X63Mepyramine8X63-H1-Mepyramine
10.71Single8X64Desloratadine8X64-H1-Desloratadine
10.71Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
10.71Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
10.71Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
10.71Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
10.71Single9IYAONO-97105319IYA-GPR55-ONO-9710531
10.71Single9JEAAtropine9JEA-M1-Atropine
10.71Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
10.71Consensusalpha2_onOrthosteric Ligandalpha2b_on
10.71Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
10.71Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.71Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
10.71Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
10.71Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
10.71Consensushistamine_offOrthosteric Ligandh1_off
10.71Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
10.71Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
10.71Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
10.53Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
10.34Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
10.34Single5CGCHTL142425CGC-mGlu5-HTL14242
10.34Single6HLPNetupitant6HLP-NK1-Netupitant
10.34Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
10.34Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
10.34Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
10.34Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
10.34Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
10.34Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
10.34Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
10.34Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
10.34Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
10.34Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
10.34Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
10.34Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.34Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.34Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
10.34Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.34Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.34Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
10.34Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.34Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.26Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
10.26Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
10.00Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
10.00Single6J20Aprepitant6J20-NK1-Aprepitant
10.00Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.00Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
10.00Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
10.00Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
10.00Single8EA0Iperoxo8EA0-M3-Iperoxo
10.00Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
10.00Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
10.00Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
10.00Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
10.00Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
10.00Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
9.68Single6IIURamatroban6IIU-TXA2-Ramatroban
9.68Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
9.68Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
9.68Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
9.68Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
9.68Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
9.68Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
9.68Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
9.68Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
9.38Single5CGDHTL142425CGD-mGlu5-HTL14242
9.38Single6K1QIRL25006K1Q-ETB-IRL2500
9.38Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
9.38Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
9.38Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Single8XVJMacitentan8XVJ-ETA-Macitentan
9.38Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
9.38Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
9.38Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
9.38Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
9.38Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
9.09Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
9.09Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
9.09Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
9.09Single9JF4PD1683689JF4-BB1-PD168368
9.09Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
8.82Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
8.82Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
8.82Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
8.70Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
8.70Single8HS2Fab0468HS2-GPR20-Fab046
8.70Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
8.33Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
8.33Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
8.33Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
8.11Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
8.11Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
8.00Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
8.00Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
8.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
8.00Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.00Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
8.00Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
7.69Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
7.69Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
7.69Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
7.69Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
7.69Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
7.69Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.69Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
7.69Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
7.69Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
7.69Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.69Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
7.69Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
7.69Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.69Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
7.69Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.69Single9AS7Psilocin9AS7-5-HT2A-Psilocin
7.69Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.69Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
7.69Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
7.69Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
7.69Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
7.41Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
7.41Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
7.41Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.41Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
7.41Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.41Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
7.41Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
7.41Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
7.41Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
7.41Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
7.41Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.41Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
7.41Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
7.41Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
7.41Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
7.14Single3RZECidoxepin3RZE-H1-Cidoxepin
7.14Single6TPKRetosiban6TPK-OT-Retosiban
7.14Single7VV6C48/807VV6-MRGPRX2-C48/80
7.14Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.14Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
7.14Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
7.14Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
7.14Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
7.14Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
7.14Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
7.14Consensusvasop-oxy_offOrthosteric Ligandot_off
6.90Single5DHGC-355DHG-NOP-C-35
6.90Single5DSGTiotropium5DSG-M4-Tiotropium
6.90Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
6.90Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
6.67Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
6.67Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
6.67Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
6.67Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
6.67Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
6.67Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
6.45Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
6.45Single6E59L-7607356E59-NK1-L-760735
6.45Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
6.45Single9AS9RS130-1809AS9-5-HT2A-RS130-180
6.45Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
6.06Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
5.00Single6D35Cholesterol6D35-SMO-Cholesterol
5.00Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.00Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
5.00Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
5.00Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
5.00Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
5.00Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
5.00Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
5.00Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
5.00Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
5.00Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
5.00Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.00Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.00Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
5.00Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
5.00Single7DTTCa7DTT-CaS-Ca-Ca
5.00Single7DTTCa7DTT-CaS-Ca-Ca
5.00Single7DTUTryptophan7DTU-CaS-Tryptophan
5.00Single7DTUTryptophan7DTU-CaS-Tryptophan
5.00Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.00Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.00Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
5.00Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
5.00Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.00Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
5.00Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.00Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
5.00Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
5.00Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.00Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
5.00Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.00Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
5.00Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.00Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
5.00Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
5.00Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
5.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
5.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
5.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.00Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
5.00Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.00Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
5.00Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.00Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
5.00Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.00Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
5.00Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.00Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.00Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
5.00Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
5.00Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
5.00Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.00Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
5.00Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.00Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
5.00Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.00Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
5.00Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
5.00Single7XW7K1-707XW7-TSH-K1-70
5.00Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.00Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
5.00Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.00Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
5.00Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.00Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
5.00Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.00Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
5.00Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.00Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
5.00Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.00Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
5.00Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
5.00Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.00Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
5.00Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.00Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
5.00Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.00Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
5.00Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.00Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
5.00Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.00Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
5.00Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.00Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.00Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
5.00Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
5.00Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.00Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
5.00Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.00Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
5.00Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.00Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
5.00Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.00Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
5.00Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.00Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
5.00Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.00Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
5.00Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.00Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
5.00Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.00Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
5.00Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
5.00Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
5.00Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
5.00Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
5.00Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
5.00Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
5.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.00Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
5.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.00Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
5.00Single8WVXNorrin8WVX-LGR4-Norrin
5.00Single8WVYNorrin8WVY-LGR4-Norrin
5.00Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.00Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
5.00Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
5.00Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.00Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
5.00Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.00Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
5.00Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
5.00Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.00Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
5.00Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.00Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
5.00Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.00Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.00Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
5.00Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
5.00Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.00Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.00Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
5.00Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.00Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
5.00Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.00Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
5.00Single9KHHNorrin9KHH-LGR4-Norrin
5.00Single9S37NB219S37-LGR4-NB21
5.00Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
4.76Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.76Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.76Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.76Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
4.76Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.76Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
4.76Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
4.76Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
4.76Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.76Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
4.76Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
4.76Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
4.55Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
4.55Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
4.55Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
4.55Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
4.35Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
4.35Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
4.35Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
4.35Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
4.35Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
4.17Single5L7DCholesterol5L7D-SMO-Cholesterol
4.17Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
4.17Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
4.00Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
4.00Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
3.85Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
3.85Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.70Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
3.70Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
3.70Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
3.70Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.57Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.45Single6FFIMMPEP6FFI-mGlu5-MMPEP
3.45Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.45Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
3.33Single6FFHFenobam6FFH-mGlu5-Fenobam
3.23Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.23Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.23Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.23Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
3.23Single9HC04YI9HC0-mGlu5-4YI
3.12Single7P2L4YI7P2L-mGlu5-4YI
3.12Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.12Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.12Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.12Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
2.78Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.78Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.63Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.63Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.56Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.38Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
protein_on_gp chemokine_on_gp
chemerin_on_gp
protein_off chemokine_off
grh_off
Net Summary
Imin 3.44285
Number of Linked Nodes 952
Number of Links 982
Number of Hubs 103
Number of Links mediated by Hubs 455
Number of Communities 7
Number of Nodes involved in Communities 54
Number of Links involved in Communities 69
Path Summary
Number Of Nodes in MetaPath 94
Number Of Links MetaPath 93
Number of Shortest Paths 347145
Length Of Smallest Path 3
Average Path Length 37.4961
Length of Longest Path 77
Minimum Path Strength 0.627172
Average Path Strength 4.33458
Maximum Path Strength 16.5
Minimum Path Correlation 0.700563
Average Path Correlation 0.887906
Maximum Path Correlation 0.987073
Minimum % Of Corr. Nodes 1.33333
Average % Of Corr. Nodes 13.8417
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 40.8759
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .




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