Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: hub id, click on each number to highlight the corresponding hub in the 3D visualization.

Hub: the hub being considered.

Avg Int. Strength: the average interaction strength of all the links of the corresponding hub.

Num Of Links: the number of links of the corresponding hub.

Community: the id of the community the link belong to, otherwise 0.

ConSurf: this column reports the ConSurf conservation grades of each hub.

Index Hub Avg. Int. Strength Num. Of Links Community ConSurf
1G.HN.45 2.28875404
2G.S1.02 3.6325424
3G.S1.06 4.19155168
4G.S3.01 4.68813424
5G.S3.03 5.99333627
6G.S3.04 10.0844446
7G.S3.06 10.9394446
8G.H2.06 5.2055559
9G.H2.07 5.5315509
10G.H2.10 4.44187446
11G.h2s4.01 9.3025409
12G.S4.02 4.78063407
13G.S4.04 4.7265179
14G.H3.01 5.4725409
15G.H3.03 3.20687404
16G.H3.09 5.6175609
17G.H3.13 5.8015505
18G.H3.17 5.39875644
19G.S5.05 4.3275509
20G.HG.04 2.8145508
21G.hgh4.02 4.0225198
22G.hgh4.08 3.792501
23G.H4.10 11.19814196
24G.H4.12 5.06754205
25G.H4.14 6.01254196
26G.H4.15 6.88188408
27G.h4s6.12 4.15188404
28G.S6.02 6.42625408
29G.H5.08 6.61458628
30G.H5.17 5.30625425
31G.H5.20 3.37812408
32b.1x15 3.39438407
33b.lhb1x6 4.47437463
34b.l1x3 8.01417699
35b.l1x6 9.3735549
36b.b2x1 8.25813448
37b.b2x5 5.85042607
38b.b3x3 3.993508
39b.l3x1 10.1562449
40b.l3x2 6.43313409
41b.b4x2 5.68187408
42b.b4x3 4.48407
43b.b4x6 8.87107799
44b.b4x7 7.1325408
45b.l4x2 9.10312474
46b.b5x2 5.7975407
47b.b5x3 5.78958699
48b.b5x7 5.95437407
49b.l5x1 4.14375408
50b.l5x5 10.5604649
51b.b6x5 3.83563406
52b.b7x1 5.5365504
53b.b8x4 6.65937406
54b.l9x3 6.9435559
55b.l9x6 5.04208658
56b.b10x5 5.08562409
57b.l10x1 4.39437403
58b.b11x4 5.37375459
59b.l11x2 7.125559
60b.b12x6 8.90375658
61b.b13x7 7.9575587
62b.l13x3 6.97333689
63b.l13x6 5.07188459
64b.l13x7 5.57125489
65b.b15x1 7.03875489
66b.l15x1 4.9595557
67b.l15x2 5.565489
68b.b16x4 8.11625486
69b.b16x6 8.01429788
70b.b17x5 6.10812437
71b.b17x7 7.29187438
72b.l17x3 8.64083639
73b.l17x6 6.1635559
74b.b18x3 4.64625438
75b.b18x5 3.88375405
76b.l18x1 5.990717136
77b.l18x3 9.248134135
78b.b19x2 6.2075636
79b.b19x4 6.77313438
80b.l19x2 6.163539
81b.b20x2 7.28125436
82b.b20x4 9.51167638
83b.b20x6 6.06214736
84b.b21x1 8.054537
85b.b21x5 6.23404
86b.b21x7 5.75208605
87b.b22x5 6.505407
88b.l22x5 7.3475669
89b.b23x6 7.498756157
90b.b24x4 8.155634156
91b.b24x6 5.164374158
92b.b25x3 8.15254155
93b.l25x3 8.85955119
94b.l25x6 10.9775448
95b.b26x3 3.3625466
96b.l26x5 4.88475
97b.b27x1 3.68937466
98b.l27x1 8.66844849
99b.l27x2 7.719374119
100b.b28x3 5.08375497
101b.b28x4 6.221254116
102b.b28x6 8.6045119
103b.b28x7 5.3775479
104g.h1x5 2.33438406
105g.h1x8 3.488754227
106g.h1x11 3.186509
107g.l1x4 7.2055538
108g.h2x9 3.325404
109g.h2x11 9.499384136
110g.ctx3 6.337569
111g.ctx5 3.98625469
112g.ctx6 3.266566
113g.ctx14 5.3955579
114g.ctx15 6.62312479
115g.ctx16 4.8825878
116Lig 12.09732910
117NT 17.4475415
1181x31 6.2275414
1191x39 4.99687417
1201x43 11.0494416
1211x50 4.73409
1222x38 4.668754106
1232x39 5.605426108
1242x40 5.23625407
1252x42 5.2255108
1262x44 8.21562406
1272x50 7.563509
1282x51 3.18687407
1292x53 6.06437418
1302x57 11.1789717
131E1 9.81722912
1323x26 8.65437416
1333x32 5.26125616
1343x34 6.79955128
1353x39 8.48813408
1363x40 7.22708618
1373x41 4.188754125
1383x42 8.643509
1393x43 4.21875409
1403x44 5.13313407
1413x46 7.15955109
1423x49 5.084384107
1433x54 3.803124217
144I2 6.42851025
1454x46 4.48255107
1464x52 3.541254123
1474x53 4.54755129
1484x60 7.184518
1494x64 6.7395515
150E2 15.7636914
151E2x51 7.94792619
1525x40 3.48188414
1535x41 5.64688416
1545x43 9.73518
1555x60 3.32375406
1565x68 5.08125427
157I3 4.0965524
1586x46 3.71155236
1596x48 7.1415519
1606x49 3.958754235
161E3 6.41031814
1627x33 6.4415517
1637x35 4.13437406
1647x43 5.138506
1657x45 5.3625419
1667x52 4.45625407
1677x53 7.33875408
1687x54 3.77875407
1698x58 3.2325404
   

Color ConSurf Grade
      No Conservation data available
      1
      2
      3
      4
      5
      6
      7
      8
      9

All columns can be sorted in ascending/descending alphabetical order, clicking on the corresponding column header.

Index: link id, click on each number to highlight the corresponding link in the 3D visualization.

Node1 Node2: the two nodes of the corresponding link.

Recurrence: the relative Recurrence in the pool of shortest paths.

Strength: the interaction strength between the two nodes.

Hub1?, Hub2?: "Yes" if the corresponding node has more than 3 links, otherwise "No".

Community: the id of the community the link belong to, otherwise 0.

ConSurf1, ConSurf2: these columns report the ConSurf conservation grades of the two nodes involved in a link.


Index Node1 Node2 Recurrence Int. Strength Hub1? Hub2? Community ConSurf1 ConSurf2
1b.b3x1 b.b4x7 75.50923.7325NoYes058
2b.b3x1 b.b5x4 75.65793.3525NoNo055
3b.b5x4 b.b5x5 75.80755.885NoNo055
4b.b4x5 b.b5x5 75.49878.285NoNo075
5b.b3x3 b.b4x5 75.7194.605YesNo087
6b.b3x3 b.b6x5 89.87854.1025YesYes086
7b.b2x4 b.b6x5 90.26353.27NoYes066
8b.b10x4 b.b2x4 90.391110.4375NoNo066
9b.b10x2 b.b10x4 95.61685.57NoNo066
10b.b10x2 b.b6x2 95.72683.38NoNo068
11b.b10x3 b.b6x2 95.83644.225NoNo088
12b.b10x3 b.b11x4 97.9462.9575NoYes089
13b.b11x4 b.l9x3 97.96055.8225YesYes599
14b.b11x6 b.l9x3 98.737313.9475NoYes599
15b.b11x6 b.l11x1 1003.71NoNo599
16b.l11x1 b.l9x6 84.68394.71NoYes598
17G.H2.07 b.l9x6 66.38912.895YesYes098
18G.H2.04 G.H2.07 65.08054.75NoYes099
19G.H2.04 G.H3.08 83.97253.9475NoNo099
20G.H3.08 G.S4.04 83.65456.395NoYes1799
21G.H3.09 G.S4.04 73.54656.165YesYes099
22G.H3.09 G.H3.13 80.53497.9475YesYes095
23G.H3.13 G.h4s6.13 80.136411.6375YesNo050
24G.h4s6.12 G.h4s6.13 80.04212.82YesNo040
25G.S6.02 G.h4s6.12 79.64534.49YesYes084
26G.H5.13 G.S6.02 74.19777.47NoYes078
275x68 G.H5.13 11.93386.2225YesNo277
285x68 G.H5.16 15.27726.9775YesNo277
29G.H5.16 I2 15.03094.605NoYes275
30G.HG.04 G.s4h3.01 10.22664.405YesNo087
31G.S5.06 G.s4h3.01 11.55545.595NoNo087
32G.S5.06 G.S6.05 11.88636.065NoNo085
33G.H4.12 G.S6.05 15.0452.8175YesNo055
34G.H4.12 G.S6.03 15.99398.5425YesNo2054
35G.S5.04 G.S6.03 16.6543.225NoNo094
36G.S4.04 G.S5.04 15.69723.0475YesNo099
37G.H5.10 G.S6.02 12.08096.795NoYes078
38b.l11x1 b.l13x6 15.40973.355NoYes599
39b.l13x6 b.l15x1 15.38563.8875YesYes597
40b.l15x1 b.l17x6 15.557711.67YesYes579
41G.H2.06 b.l9x6 15.64293.58YesYes598
42G.H3.09 G.H4.15 10.81674.5525YesYes098
43G.H3.03 G.H3.06 18.11712.9925YesNo047
44G.H3.06 G.H4.15 13.00929.7425NoYes078
45G.H3.03 G.hgh4.02 14.32163.2175YesYes048
46G.H5.13 G.H5.17 62.1444.765NoYes275
47G.H5.26 I3 63.79484.45NoYes054
48G.H5.17 I3 65.70073.655YesYes254
49G.H5.20 G.H5.26 63.3433.6975YesNo085
50G.H5.20 G.H5.25 36.4883.4625YesNo086
513x54 G.H5.20 26.95084.28YesYes078
523x50 3x54 24.67673.5675NoYes2187
533x50 G.H5.23 24.55768.0325NoNo084
546x40 G.H5.25 36.10564.155NoNo096
55G.H2.06 b.l17x6 15.40655.1875YesYes599
56b.l17x5 b.l17x6 48.04762.9425NoYes069
57b.l17x5 b.l19x2 47.69732.5725NoYes069
58b.b20x4 b.l19x2 43.34213.2725YesYes389
59b.b20x4 b.b20x6 40.04074.0125YesYes386
60b.b17x7 b.b20x6 31.41417.77YesYes386
61b.b17x7 b.b21x1 27.14753.285YesYes387
62b.1x19 b.b21x1 14.550210.4225NoYes067
63b.1x15 b.1x19 11.13765.95YesNo076
64b.1x15 g.h1x11 20.91351.43YesYes079
65b.1x11 g.h1x11 13.25335.5375NoYes089
66b.1x11 g.h1x8 11.85551.49NoYes087
67b.b21x1 g.l1x4 12.11712.8025YesYes378
68b.1x15 g.l1x4 11.17513.76YesYes078
69b.b4x7 b.l2x5 70.084516.08YesNo085
70b.l2x5 b.l4x2 69.7619.52NoYes054
71b.l4x2 g.ctx15 32.830110.435YesYes749
72b.l26x5 g.ctx15 31.2516.29YesYes759
73b.l26x5 g.ctx4 62.58644.6125YesNo057
74g.ctx3 g.ctx4 62.14444.83YesNo097
75g.ctx3 g.ctx5 48.68113.0525YesYes699
76b.b27x1 g.ctx5 41.70613.725YesYes669
77b.b26x5 b.b27x1 35.04043.21NoYes076
78b.b22x4 b.b26x5 34.57294.85NoNo057
79b.b18x4 b.b22x4 34.10513.01NoNo035
80b.b18x4 b.b22x5 33.63694.54NoYes037
81b.b22x5 b.b23x2 24.19038.525YesNo076
82b.b21x7 b.b23x2 23.71394.69YesNo056
83b.l4x2 g.ctx16 34.367112.6375YesYes748
84b.l26x5 g.ctx16 32.49773.42YesYes758
85g.ctx3 g.ctx6 13.2015.7675YesYes696
86b.b21x7 b.b24x6 14.55995.065YesYes058
87b.b3x3 b.b4x3 13.96572.98YesYes087
88b.b4x3 b.b5x7 11.03584.6375YesYes077
89b.b10x4 b.b14x5 12.32193.0375NoNo065
90b.b14x5 b.l10x1 12.04365.54NoYes053
913x40 Lig 25.933.4375YesYes180
923x40 5x51 33.50025.1775YesNo087
935x51 6x49 33.63813.8875NoYes075
946x46 6x49 33.83524.0075YesYes2365
955x58 6x46 35.7463.2075NoYes076
965x58 6x40 35.92434.4975NoNo079
972x39 3x46 10.58344.65YesYes1089
982x39 G.H5.23 24.38984.8875YesNo084
99G.H2.04 b.l17x6 20.61664.765NoYes099
Download PSN data

2D representation of the global metapath, ligand(s) interactions and
histograms of path distribution according to several parameters
(click on the image to enlarge it 🔍):

A 2D representation of the global communication in the network.

ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Number of shortest communication paths as a function of the average residue correlation.

Number of shortest communication paths as a function of the average interaction strength of their links.

Number of shortest communication paths as a function of the % of hub nodes in each path.

Number of shortest communication paths as a function of the number of nodes in each path.

Number of shortest communication paths as a function of the % of correlated nodes in each path.


2D representation of the interactions of this orthosteric/allosteric ligand.


Links and nodes colored according to ConSurf Conservation Grade (See documentation): 

 n/a   1    2    3    4    5    6    7    8    9  

Node1Node2LinkStrengthCommIsNode1Hub?IsNode2Hub?Node1ConsNode2ConsNode1ShellNode2Shell
7x33Lig6.15751YesYes7010
5x44Lig14.36251NoYes6010
6x52Lig9.64751NoYes5010
6x48Lig7.391YesYes9010
7x37Lig11.25751NoYes8010
3x40Lig3.43751YesYes8010
E2Lig15.88751YesYes4010
5x43Lig3.271YesYes8010
7x34Lig6.9851NoYes6010
7x38Lig5.251NoYes6010
7x41Lig7.471NoYes8010
2x57Lig5.461YesYes7010
3x32Lig11.641YesYes6010
2x60Lig3.311NoYes6010
3x29Lig2.921NoYes7010
3x33Lig7.55251NoYes8010
E2x52Lig19.95251NoYes7010
1x32Lig12.80751NoYes4010
2x61Lig6.00751NoYes6010
E1Lig14.0851YesYes2010
1x29Lig6.691NoYes3010
LigNT11.5851YesYes0501
1x21Lig3.570NoYes1010
NTNT28.0151YesYes5511
1x281x315.751NoYes3422
1x281x324.49251NoNo3421
1x291x338.4551NoNo3211
1x301x333.6450NoNo1221
1x391x435.10251YesYes7622
1x392x577.06251YesYes7721
1x402x576.511NoYes5721
1x402x618.7351NoNo5621
1x432x5726.1851YesYes6721
2x533x323.3651YesYes8621
2x533x368.23251YesNo8622
2x563x324.050NoYes5621
2x572x588.51751YesNo7612
2x572x6118.61751YesNo7611
2x573x325.91YesYes7611
2x603x282.941NoNo6612
2x603x323.721NoYes6611
E1E114.8651YesYes2211
3x22E16.61251NoYes3221
3x24E14.90251NoYes1221
3x25E15.041NoYes9221
E1E215.64751YesYes2411
E1E2x528.121YesNo2711
3x223x2411.991NoNo3122
3x26E26.631YesYes6421
3x26E2x5121.241YesYes6922
3x29E2x524.8651NoNo7711
3x323x362.89251YesNo6612
3x334x607.62751NoYes8812
3x335x4311.91751NoYes8811
3x363x405.55251NoYes6821
3x403x435.28751YesYes8912
3x405x4712.81751YesNo8712
3x405x515.17751YesNo8712
3x406x4811.091YesYes8911
3x437x454.760YesYes9922
4x605x414.46751YesYes8622
4x605x4311.5751YesYes8821
4x65E23.7751NoYes1421
4x65E2x514.841NoYes1922
4x68E221.2551NoYes6421
E2E2x516.781YesYes4912
E2E233.08251YesYes4411
5x42E25.73250NoYes6421
5x415x439.771YesYes6821
5x415x444.8951YesNo6621
5x435x4412.11751YesNo8611
5x486x526.59250NoNo4521
6x476x483.43751NoYes8921
6x477x453.541NoYes8922
6x487x415.61751YesNo9811
6x487x458.17251YesYes9912
6x51E36.64751NoYes8422
6x517x337.51NoYes8721
6x526x534.5851NoNo5512
E3E38.161YesYes4422
7x33E36.951YesYes7412
7x337x343.14251YesNo7611
7x337x378.45751YesNo7811
1x33Lig3.9051NoYes2010
1x397x383.35251YesNo7621
3x26E14.21751YesYes6221
1x311x324.3551YesNo4421
1x251x272.711NoNo2312
1x23Lig2.5151NoYes1010
1x261x292.380NoNo1321
1x19NT2.1750NoYes1521
1x25Lig2.0351NoYes2010
1x22Lig0.99750NoYes2010
1x231x240.691NoNo1312

Location and physicochemical properties of the interaction partners of this ligand

Interactions of this ligand

Similarities between the interactions of this ligand and those of other networks

ShowSimilarityNetwork TypeNameLigandDescription
85.19Consensuscrf_onOrthosteric Ligandcrf2_on crf1_on
75.86Single7TS0Urocortin7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
73.33Single6PB0Urocortin6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
56.25Single6P9XCorticoliberin6P9X-CRF1-Corticoliberin-Gs/β1/γ2
54.55Single6PB1Urocortin6PB1-CRF2-Urocortin-chim(NtGi1-Gs)/β1/γ2
53.85Consensuspth_on_gpOrthosteric Ligandpth1_on_gp pth2_on_gp
53.12Single9BLWCagrilintide backbone (non-acylated)9BLW-CT (AMY1)-Cagrilintide backbone (non-acylated)-Gs/β1/γ2; RAMP1
52.94Consensusclass-a_class-b1_cons_onOrthosteric Ligandclass-a_on class-b1_on
52.78Single7TYOCalcitonin7TYO-CT-Calcitonin-Gs/β1/γ2
52.78Single7Y36Teriparatide7Y36-PTH1-Teriparatide-Gs/β1/γ2
52.63Single7F16TIP397F16-PTH2-TIP39-Gs/β1/γ2
51.52Single6UVAAdrenomedullin-26UVA-CT Like (AM2)-Adrenomedullin-2-Gs/β1/γ2; RAMP3
51.52Single8HAOPTH8HAO-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
51.22Consensusclass-b1_on_gpOrthosteric Ligandglucagon_on_gp vip-pacap_on_gp pth_on_gp crf_on_gp calcitonin_on_gp
50.00Single6NBHLong-Acting PTH Analog6NBH-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
48.72Consensusclass-b1_onOrthosteric Ligandglucagon_on vip-pacap_on pth_on crf_on calcitonin_on
48.65Single7TYYCalcitonin-17TYY-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
48.65Single9JR3PTH9JR3-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
48.65Consensusclass-a_class-b1_cons_on_gpOrthosteric Ligandclass-a_on_gp class-b1_on_gp
48.39Consensusclass-b1_class-b2_cons_onOrthosteric Ligandclass-b1_on class-b2_on
48.39Consensusclass-b1_class-b2_cons_on_gpOrthosteric Ligandclass-b1_on_gp class-b2_on_gp
47.22Single6LPBPACAP6LPB-PAC1-PACAP-Gs/β1/γ1
47.06Single9BUCCagrilintide9BUC-CT-Cagrilintide-Gs/β1/γ2
45.95Single7VVMPTH7VVM-PTH1-PTH-Gs/β1/γ2
45.71Single6WZGSecretin6WZG-Secretin-Secretin-Gs/β1/γ2
45.45Single7TYWCalcitonin-17TYW-CT (AMY1)-Calcitonin-1-Gs/β1/γ2; RAMP1
45.45Single7WBJPACAP277WBJ-VPAC1-PACAP27-Gs/β1/γ2
44.74Single8FLQPTH8FLQ-PTH1-PTH-Gs/β1/γ2
44.44Single7RBTTirzepatide7RBT-GIP-Tirzepatide-LSN3556672-chim(NtGi1-Gs)/β1/γ2
44.12Single7VABNon-Acylated Tirzepatide7VAB-GIP-Non-Acylated Tirzepatide-chim(NtGi1-Gs)/β1/γ2
43.59Single6E3YCalcitonin gene-related peptide-16E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
43.59Consensuspth_onOrthosteric Ligandpth1_on pth2_on
43.24Single8F2APramlintide Analogue San3858F2A-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
43.24Single8FLSAbaloparatide8FLS-PTH1-Abaloparatide-Gs/β1/γ2
43.24Single8FLULong-Acting PTH8FLU-PTH1-Long-Acting PTH-Gs/β1/γ2
42.86Single7VQXPACAP277VQX-VPAC1-PACAP27-Gs/β1/γ2
42.42Single6WI9Secretin6WI9-Secretin-Secretin-Gs/β1/γ2
42.42Single8YW4Retatrutide8YW4-GIP-Retatrutide-chim(NtGi1-Gs)/β1/γ2
41.67Single6UUSAdrenomedullin6UUS-CT Like (AM2)-Adrenomedullin-Gs/β1/γ2; RAMP3
41.67Single7VVJPTHrP(1-36)7VVJ-PTH1-PTHrP(1-36)-Gs/β1/γ2
41.67Single7VVLPTH7VVL-PTH1-PTH-Gs/β1/γ2
41.67Single8F0KPramlintide Analogue San3858F0K-CT (AMY3)-Pramlintide Analogue San385-Gs/β1/γ2; RAMP3
41.67Consensusvip-pacap_onOrthosteric Ligandvpac_on pac_on
41.67Consensusvip-pacap_on_gpOrthosteric Ligandvpac_on_gp pac_on_gp
41.18Single8E3ZVIP8E3Z-VPAC1-VIP-Gs/β1/γ2
41.03Consensusglucagon_onOrthosteric Ligandglp_on gluc_on secretin_on gip_on
40.62Single7TRYUrocortin7TRY-CRF2-Urocortin-chim(NtGi1-G11)/β1/γ2
40.00Single6NBFLong-Acting PTH Analog6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
40.00Single6NBILong-Acting PTH Analog6NBI-PTH1-Long-Acting PTH Analog-Gs/β1/γ2
40.00Single8E3XPACAP278E3X-PAC1-PACAP27-Gs/β1/γ2
40.00Single8FLRPTHrP(1-36)8FLR-PTH1-PTHrP(1-36)-Gs/β1/γ2
40.00Single9BLBCagrilintide backbone (non-acylated)9BLB-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
40.00Single9BP3Cagrilintide9BP3-CT (AMY1)-Cagrilintide-Gs/β1/γ2; RAMP1
40.00Single9BUBCagrilintide9BUB-CT-Cagrilintide-Gs/β1/γ2
40.00Consensusglucagon_on_gpOrthosteric Ligandglp_on_gp gluc_on_gp secretin_on_gp gip_on_gp
40.00Consensuspac_on_gpOrthosteric Ligandpac1_on_gp
39.47Single7TZFAmylin7TZF-CT (AMY3)-Amylin-Gs/β1/γ2; RAMP3
38.89Single6B3JExendin-P56B3J-GLP-1-Exendin-P5-Gs/β1/γ2
38.89Single7DTYGIP7DTY-GIP-GIP-Gs/β1/γ2
38.89Single7TYNCalcitonin-17TYN-CT-Calcitonin-1-Gs/β1/γ2
38.89Consensusglp_onOrthosteric Ligandglp1_on glp2_on
38.89Consensusglp_on_gpOrthosteric Ligandglp1_on_gp glp2_on_gp
38.46Single6WPWGlucagon derivative ZP37806WPW-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
38.24Single6NIYAdrenomedullin6NIY-CT-Adrenomedullin-Gs/β1/γ2
38.24Single7TYIAmylin7TYI-CT-Amylin-Gs/β1/γ2
38.10Consensuspth2_on_gpOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
37.84Single5VAIGLP-15VAI-GLP-1-GLP-1-Gs/β1/γ2
37.84Single6LMLGlucagon6LML-Glucagon-Glucagon-Gi1/β1/γ1
37.84Single7D68GLP-27D68-GLP-2-GLP-2-Gs/β1/γ2
37.84Single7TYLAmylin7TYL-CT-Amylin-Gs/β1/γ2
37.84Single8FLTM-PTH(1-14)8FLT-PTH1-M-PTH(1-14)-Gs/β1/γ2
37.84Single9BQ3Cagrilintide9BQ3-CT (AMY2)-Cagrilintide-Gs/β1/γ2; RAMP2
37.84Single9BTWCagrilintide9BTW-CT (AMY3)-Cagrilintide-Gs/β1/γ2; RAMP3
37.50Consensuspth2_onOrthosteric Ligand7F16-PTH2-TIP39-Gs/β1/γ2
37.14Single7TYHCalcitonin-17TYH-CT (AMY2)-Calcitonin-1-Gs/β1/γ2; RAMP2
37.14Consensuscalcitonin_onOrthosteric Ligandctlike_on
37.14Consensuspac_onOrthosteric Ligandpac1_on
37.14Consensusvpac_onOrthosteric Ligandvpac1_on vpac2_on
36.84Single7DUQGLP-17DUQ-GLP-1-GLP-1-PubChem 156022738-Gs/β1/γ2
36.84Single7TYXAmylin7TYX-CT (AMY2)-Amylin-Gs/β1/γ2; RAMP2
36.67Consensuslpl_offOrthosteric Ligands1p_off lpa_off
36.11Single7CZ5Somatoliberin7CZ5-GHRH-Somatoliberin-Gs/β1/γ2
36.11Single7D3SSecretin7D3S-Secretin-Secretin-Gs/β1/γ2
36.11Single7RA3GIP7RA3-GIP-GIP-chim(NtGi1-Gs)/β1/γ2
36.11Consensuscalcitonin_on_gpOrthosteric Ligandctlike_on_gp
36.11Consensusvpac_on_gpOrthosteric Ligandvpac1_on_gp vpac2_on_gp
35.90Single9AUCCalcitonin gene-related peptide-19AUC-CT (AMY1)-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
35.71Single7V3ZCP559407V3Z-CB1-CP55940
35.48Single9C0KExendin-49C0K-GLP-1-Exendin-4-Gs/β1/γ2
35.29Single6UUNAdrenomedullin6UUN-CT Like (AM1)-Adrenomedullin-Gs/β1/γ2; RAMP2
35.14Single6VCBGLP-16VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
35.14Single7FIYTirzepatide7FIY-GIP-Tirzepatide-Gs/β1/γ2
35.14Single7S1MEx4-D-Ala7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2
35.14Single7TYFAmylin7TYF-CT (AMY1)-Amylin-Gs/β1/γ2; RAMP1
35.14Single7VVKPTH7VVK-PTH1-PTH-Gs/β1/γ2
35.00Single9JR2PTH9JR2-PTH1-PTH-chim(NtGi1L-Gs-CtGq)/β1/γ2
34.48Single9ERXD9-THC analog9ERX-CB1-D9-THC analog-Gi1/β1/γ2
34.48Consensuscb2_onOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
34.48Consensuscb2_on_gpOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2
34.38Single5ZTYAM102575ZTY-CB2-AM10257
34.38Single8X3LXWD8X3L-CB2-XWD-Gi1/β1/γ2
34.38Consensuscb2_offOrthosteric Ligand5ZTY-CB2-AM10257
34.29Single7FIMTirzepatide7FIM-GLP-1-Tirzepatide-Gs/β1/γ2
34.29Single7FINPeptide-20; GGL7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2
34.29Single8H4KGW95088H4K-FFA4-GW9508-chim(NtGi1-Gs-CtGq)/β1/γ2
34.29Single8HA0PTH8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2
34.29Single8YW3Retatrutide8YW3-GLP-1-Retatrutide-Gs/β1/γ2
34.29Single8YW5Retatrutide8YW5-Glucagon-Retatrutide-Gs/β1/γ2
34.29Single9BLCCagrilintide backbone (non-acylated)9BLC-CT-Cagrilintide backbone (non-acylated)-Gs/β1/γ2
34.29Consensusgi_class-aOrthosteric Ligandgi_peptide gi_sensory gi_alicarboxylic gi_amine gi_lipid gi_nucleotide gi_protein
34.21Single7KI1Taspoglutide7KI1-GLP-1-Taspoglutide-Gs/β1/γ2
34.21Single8HAFPTHrP(1-36)8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2
34.21Single9BYOExendin-39BYO-GLP-1-Exendin-3-Gs/β1/γ2
34.21Consensuspth1_onOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
34.21Consensusvpac2_onOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
34.21Consensusvpac2_on_gpOrthosteric Ligand7VQX-VPAC1-PACAP27-Gs/β1/γ2
34.09Single8F0JPramlintide Analogue San458F0J-CT-Pramlintide Analogue San45-Gs/β1/γ2
33.33Single5GLHEndothelin-15GLH-ETB-Endothelin-1
33.33Single5XRAAM115425XRA-CB1-AM11542
33.33Single6IGKEndothelin-36IGK-ETB-Endothelin-3
33.33Single7FEECP559407FEE-CB1-CP55940-ZCZ011
33.33Single7WV9CP559407WV9-CB1-CP55940-ZCZ011-Gi2/β1/γ2
33.33Single8E3YPACAP278E3Y-VPAC1-PACAP27-Gs/β1/γ2
33.33Single8YWFRetatrutide8YWF-GLP-1-Retatrutide-chim(NtGi1-Gs)/β1/γ2
33.33Single9BUECagrilintide9BUE-CT-Cagrilintide-Gs/β1/γ2
33.33Consensusgi_cannabinoidOrthosteric Ligand8GUR-CB2-CP55,940-Gi1/β1/γ2 8GUS-CB2-HU-308-Gi1/β1/γ2 8GUT-CB2-LEI-102-Gi1/β1/γ2 8GUQ-CB2-Olorinab-Gi1/β1/γ2 6KPF-CB2-PubChem 145915889-Gi1/β1/γ2 6PT0-CB2-WIN 55212-2-Gi1/β1/γ2 6KPG-CB1-AM841-Gi1/β1/γ2
33.33Consensusgi_opioidOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8F7X-NOP-Nociceptin-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2 8F7S-δ-Deltorphin-Gi1/β1/γ2 8F7W-κ-Dynorphin-Gi1/β1/γ2
32.43Single6FJ3PTH6FJ3-PTH1-PTH
32.43Single7RGPTirzepatide7RGP-GLP-1-Tirzepatide-chim(NtGi1-Gs)/β1/γ2
32.43Single8JISPeptide-158JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2
32.43Single9J1Pg1:Ox9J1P-GLP-1-g1:Ox-chim(NtGi1-Gs)/β1/γ2
32.43Consensusgi_peptideOrthosteric Ligandgi_cck gi_apelin gi_compl-pept gi_endothelin gi_formylpeptide gi_galanin gi_ghrelin gi_npy gi_neurotensin gi_opioid gi_orexin gi_relaxin gi_somatostatin
32.35Single8F7QBeta-Endorphin8F7Q-μ-β-Endorphin-Gi1/β1/γ2
32.26Single4Z36ONO-30805734Z36-LPA1-ONO-3080573
32.26Single6KPGAM8416KPG-CB1-AM841-Gi1/β1/γ2
32.26Single6KQICP559406KQI-CB1-CP55940-Org27569
32.26Consensuscannabinoid_offOrthosteric Ligandcb2_off cb1_off
32.26Consensuscannabinoid_onOrthosteric Ligandcb2_on cb1_on
32.26Consensuscannabinoid_on_gpOrthosteric Ligandcb2_on_gp cb1_on_gp
32.26Consensuslipid_offonOrthosteric Ligandlipid_off lipid_on
32.26Consensuslipid_offon_gpOrthosteric Ligandlipid_on_gp lipid_off
32.26Consensuslpa1_offOrthosteric Ligand4Z36-LPA1-ONO-3080573 4Z35-LPA1-ONO-9910539 4Z34-LPA1-ONO-9780307
32.26Consensuslpa_offOrthosteric Ligandlpa1_off
31.71Single6LRYSarafotoxin-B6LRY-ETB-Sarafotoxin-B
31.71Consensuspth1_on_gpOrthosteric Ligand6NBF-PTH1-Long-Acting PTH Analog-Gs/β1/γ2 8HA0-PTH1-PTH-chim(NtGi1-Gs)/β1/γ2 8HAF-PTH1-PTHrP(1-36)-chim(NtGi1-Gs)/β1/γ2 7Y36-PTH1-Teriparatide-Gs/β1/γ2 7Y35-PTH1-Abaloparatide-Gs/β1/γ2
31.58Single7WVYAmyloid-Beta427WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2
31.58Single8FU6Glucagon derivative ZP37808FU6-Glucagon-Glucagon derivative ZP3780-Gs/β1/γ2
31.58Consensuspeptide_onOrthosteric Ligandcck_on angiotensin_on apelin_on bombesin_on bradykinin_on compl-peptide_on endothelin_on formylpeptide_on galanin_on ghrelin_on kisspeptin_on melanocortin_on motilin_on neuromedin-u_on npy_on neurotensin_on opioid_on orexin_on relaxin_on somatostatin_on tachykinin_on trh_on vasop-oxy_on
31.58Consensuspeptide_on_gpOrthosteric Ligandcck_on_gp angiotensin_on_gp apelin_on_gp bombesin_on_gp bradykinin_on_gp compl-peptide_on_gp endothelin_on_gp formylpeptide_on_gp galanin_on_gp ghrelin_on_gp kisspeptin_on_gp melanocortin_on_gp motilin_on_gp neuromedin-u_on_gp npy_on_gp neurotensin_on_gp opioid_on_gp orexin_on_gp relaxin_on_gp somatostatin_on_gp tachykinin_on_gp trh_on_gp vasop-oxy_on_gp
31.43Single6VN7PACAP6VN7-VPAC1-PACAP-Gs/β1/γ2
31.43Single7TD0LPA7TD0-LPA1-LPA-Gi1/β1/γ2
31.43Single7TD2LPA7TD2-LPA1-LPA-Gi1/β1/γ2
31.43Single9B54A1AIW9B54-CB1-A1AIW-Gi1/β1/γ2
31.43Single9B5YLong-Acting PTH9B5Y-PTH1-Long-Acting PTH-chim(NtGi1-Gq)/β1/γ2
31.43Single9IVMGLP-1 (Truncated)9IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
31.43Consensuspeptide_offonOrthosteric Ligandpeptide_off peptide_on
31.25Single4Z35ONO-99105394Z35-LPA1-ONO-9910539
31.25Single6M1HMaxadilan6M1H-PAC1-Maxadilan-Gs/β1/γ2
31.25Single7VVNPTH7VVN-PTH1-PTH-Gs/β1/γ2
31.25Consensuscb1_on_gpOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
31.25Consensusclass-a_onOrthosteric Ligandsensory_on alicarboxylic_on amine_on lipid_on nucleotide_on peptide_on protein_on
30.95Single8JITMEDI03828JIT-Glucagon-MEDI0382-Gs/β1/γ2
30.95Single8JIUSAR4258998JIU-Glucagon-SAR425899-Gs/β1/γ2
30.77Single6LMKGlucagon6LMK-Glucagon-Glucagon-Gs/β1/γ2
30.56Single6M1IPACAP6M1I-PAC1-PACAP-Gs/β1/γ2
30.56Single7V9MSomatoliberin7V9M-GHRH (SV1)-Somatoliberin-Gs/β1/γ2
30.56Single9BUDCagrilintide9BUD-CT-Cagrilintide-Gs/β1/γ2
30.56Single9EBOGLP-1 (ACPC18)9EBO-GLP-1-GLP-1 (ACPC18)-Gs/β1/γ2
30.56Consensuspeptide_offon_gpOrthosteric Ligandpeptide_on_gp peptide_off
30.43Single8F2BPramlintide Analogue San458F2B-CT (AMY3)-Pramlintide Analogue San45-Gs/β1/γ2; RAMP3
30.30Single3NY9ICI118-5513NY9-β2-ICI118-551
30.30Single4UG2CGS216804UG2-A2A-CGS21680
30.30Single7XY6BAY 60-65837XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
30.30Consensuss1p_onOrthosteric Ligands1p1_on s1p3_on s1p5_on
30.30Consensuss1p_on_gpOrthosteric Ligands1p1_on_gp s1p3_on_gp s1p5_on_gp
30.00Single6KPCPubChem 1459158896KPC-CB2-PubChem 145915889
30.00Single7YU6ONO-07405567YU6-LPA1-ONO-0740556-Gi1/β1/γ2
30.00Single8ZRKGSK-12922638ZRK-GPR119-GSK-1292263-Gs/β1/γ2
30.00Single9KPFSA09KPF-TAS2R16-SA0-Gi1/β1/γ2
30.00Consensuss1p_offOrthosteric Ligands1p1_off s1p5_off
29.73Single5YQZGlucagon analogue5YQZ-Glucagon-Glucagon analogue
29.73Single6X18GLP-16X18-GLP-1-GLP-1-Gs/β1/γ2
29.73Single7LLYOxyntomodulin7LLY-GLP-1-Oxyntomodulin-Gs/β1/γ2
29.73Single7Y35Abaloparatide7Y35-PTH1-Abaloparatide-Gs/β1/γ2
29.73Single8XQEApelin-138XQE-Apelin-Apelin-13-Gi1/β1/γ2
29.73Single8ZRTET-18ZRT-ETB-ET-1
29.73Consensusvpac1_onOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
29.41Single4XT1Fractalkine4XT1-US28-Fractalkine
29.41Single8JIQPeptide-158JIQ-Glucagon-Peptide-15-Gs/β1/γ2
29.41Single8WDTphotoNECA8WDT-A2A-photoNECA
29.41Single8ZSPLSD8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
29.41Consensusclass-a_on_gpOrthosteric Ligandsensory_on_gp alicarboxylic_on_gp amine_on_gp lipid_on_gp nucleotide_on_gp peptide_on_gp protein_on_gp
29.41Consensusmop_offOrthosteric Ligand4DKL-μ-β-Funaltrexamine 8QOT-μ-Nanobody-E 7UL4-μ-Alvimopan
29.27Single7VBHPeptide-207VBH-GLP-1-Peptide-20-Gs/β1/γ2
29.03Single2YDVNECA2YDV-A2A-NECA
29.03Single4UHRCGS216804UHR-A2A-CGS21680
29.03Single4Z34ONO-97803074Z34-LPA1-ONO-9780307
29.03Single5G53NECA5G53-A2A-NECA-Gs
29.03Single5XR8AM8415XR8-CB1-AM841
29.03Single6GT3Imaradenant6GT3-A2A-Imaradenant-Na
29.03Single7CKYPW04647CKY-D1-PW0464-Gs/β1/γ2
29.03Single7EW1Siponimod7EW1-S1P5-Siponimod-Gi1/β1/γ2
29.03Single7JV5SKF812977JV5-D1-SKF81297-Gs/β1/γ2
29.03Single7JVPSKF839597JVP-D1-SKF83959-Gs/β1/γ2
29.03Single7T2HLofentanil7T2H-μ-Lofentanil-Gi1/β1/γ2
29.03Single7YU7ONO-07405567YU7-LPA1-ONO-0740556-Gi1/β1/γ2
29.03Single8E0GBU728E0G-μ-BU72
29.03Single8GUSHU-3088GUS-CB2-HU-308-Gi1/β1/γ2
29.03Single8WU1PubChem 1190256658WU1-CB1-PubChem 119025665-Arrestin2
29.03Single9EGOYVF9EGO-CB1-YVF-Gi1/β1/γ2
29.03Single9IZGNKP9IZG-LPA1-NKP-chim(NtGi1-Gs-CtGq)/β1/γ2
29.03Consensus5ht_offOrthosteric Ligand5ht2_off 5ht1_off
29.03Consensusclass-a_offOrthosteric Ligandsensory_off alicarboxylic_off amine_off lipid_off nucleotide_off peptide_off protein_off
29.03Consensuss1p5_onOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
29.03Consensuss1p5_on_gpOrthosteric Ligand7EW1-S1P5-Siponimod-Gi1/β1/γ2
28.95Single4XT3Fractalkine4XT3-US28-Fractalkine
28.95Single6P9YPACAP6P9Y-PAC1-PACAP-Gs/β1/γ2
28.95Single7KI0Semaglutide7KI0-GLP-1-Semaglutide-Gs/β1/γ2
28.95Consensuspac1_onOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
28.95Consensuspac1_on_gpOrthosteric Ligand8E3X-PAC1-PACAP27-Gs/β1/γ2 6M1H-PAC1-Maxadilan-Gs/β1/γ2
28.95Consensusvpac1_on_gpOrthosteric Ligand8E3Z-VPAC1-VIP-Gs/β1/γ2
28.57Single6HLOAprepitant6HLO-NK1-Aprepitant
28.57Single6WHCGlu16 analog of GCG6WHC-Glucagon-Glu16 analog of GCG-Gs/β1/γ2
28.57Single7V35Peptide-207V35-Glucagon-Peptide-20-Gs/β1/γ2
28.57Single8JIPMEDI03828JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2
28.57Single8JIRSAR4258998JIR-GLP-1-SAR425899-chim(NtGi1-Gs)/β1/γ2
28.57Single9J5VCpY9J5V-LPA1-CpY-Gi1/β1/γ2
28.57Consensusformylpeptide_on_gpOrthosteric Ligandfpr2-alx_on_gp fpr1-alx_on_gp
28.57Consensuss1p3_on_gpOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
28.21Single8XWPEndothelin-18XWP-ETB-Endothelin-1-Gi1/β1/γ2
28.21Consensusgq_peptideOrthosteric Ligandgq_cck gq_kisspeptin gq_bradykinin gq_bombesin gq_angiotensin
28.21Consensussecretin_on_gpOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
28.12Single5UNHPubChem 1264564065UNH-AT2-PubChem 126456406
28.12Single6OS0Angiotensinogen6OS0-AT1-Angiotensinogen
28.12Single7WCNAR2314537WCN-GPR119-AR231453-Gs/β1/γ2
28.12Single7YITNalfurafine7YIT-κ-Nalfurafine
28.12Single8VHFMBX-29828VHF-GPR119-MBX-2982-Gs/β1/γ2
28.12Single9DGIZ85267113509DGI-CB1-Z8526711350
28.12Single9IZHLPA9IZH-LPA1-LPA-chim(NtGi2-G13)/β1/γ2
28.12Consensuscb1_onOrthosteric Ligand6KPG-CB1-AM841-Gi1/β1/γ2 8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
28.12Consensusmop_onOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
28.12Consensusmop_on_gpOrthosteric Ligand8F7R-μ-Endomorphin-Gi1/β1/γ2 8EF5-μ-Fentanyl-Gi1/β1/γ2 7SCG-μ-FH210-Gi1/β1/γ2 7T2H-μ-Lofentanil-Gi1/β1/γ2 7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2 8EF6-μ-Morphine-Gi1/β1/γ2 8EFB-μ-Oliceridine-Gi1/β1/γ2 7U2L-μ-PubChem 163201242-Gi1/β1/γ2 8EFO-μ-PZM21-Gi1/β1/γ2 8EFL-μ-SR17018-Gi1/β1/γ2 8F7Q-μ-β-Endorphin-Gi1/β1/γ2 7U2K-μ-C6-guano-Gi1/β1/γ2 8EFQ-μ-Damgo-Gi1/β1/γ2
28.12Consensusopioid_offOrthosteric Ligandmop_off nop_off dop_off kop_off
27.78Consensusangiotensin_onOrthosteric Ligandat1_on
27.78Consensusat1_onOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
27.78Consensusgs_class-aOrthosteric Ligandgs_peptide gs_nucleotide gs_amine
27.59Single6PT0WIN 55212-26PT0-CB2-WIN 55212-2-Gi1/β1/γ2
27.59Single8GURCP55,9408GUR-CB2-CP55,940-Gi1/β1/γ2
27.50Consensusendothelin_onOrthosteric Ligandetb_on eta_on
27.27Single4BVNCyanopindolol4BVN-β1-Cyanopindolol-Na
27.27Single7EVZCenerimod7EVZ-S1P1-Cenerimod-Gi1/β1/γ2
27.27Single7LLLExendin-47LLL-GLP-1-Exendin-4-Gs/β1/γ2
27.27Single7SK7CCX6627SK7-ACKR3-CXCL12-CCX662
27.27Single7X2DTavapadon7X2D-D1-Tavapadon-Gs/β1/γ2
27.27Single7XJISolabegron7XJI-β3-Solabegron-Gs/β1/γ2
27.27Single7XZ6APD6687XZ6-GPR119-APD668-Gs/β1/γ2
27.27Single7Y65C5a peptide7Y65-C5a1-C5a peptide-Gi1/β1/γ2
27.27Single7YU8ONO-07405567YU8-LPA1-ONO-0740556-Gi1/β1/γ2
27.27Single8GAGPubChem 1708384908GAG-CB1-PubChem 170838490-Gi1/β1/γ2
27.27Single8GUTLEI-1028GUT-CB2-LEI-102-Gi1/β1/γ2
27.27Single8IJDMK68928IJD-HCA2-MK6892-Gi1/β1/γ2
27.27Single8J19LY2378J19-GPR84-LY237-Gi1/β1/γ2
27.27Single8WRZPubChem 1023367048WRZ-CB1-PubChem 102336704-Arrestin2
27.27Consensusgi_s1pOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7EW3-S1P3-S1P-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EW1-S1P5-Siponimod-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
27.27Consensuskop_on_gpOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
27.03Single7F6GSAR1-AngII7F6G-AT1-SAR1-AngII-Gq/β1/γ2
27.03Single8XWQEndothelin-18XWQ-ETB-Endothelin-1-Gi1/β1/γ2
27.03Consensusangiotensin_on_gpOrthosteric Ligandat1_on_gp
27.03Consensusat1_on_gpOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
27.03Consensusfpr2-alx_on_gpOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.03Consensusgi_formylpeptideOrthosteric Ligand7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
27.03Consensusgq_angiotensinOrthosteric Ligand7F6G-AT1-SAR1-AngII-Gq/β1/γ2
27.03Consensusprotein_onOrthosteric Ligandchemokine_on chemerin_on
26.83Consensusgi_endothelinOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
26.83Consensusgip_onOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
26.83Consensusgip_on_gpOrthosteric Ligand7FIN-GIP-Peptide-20; GGL-Gs/β1/γ2 7FIY-GIP-Tirzepatide-Gs/β1/γ2 7DTY-GIP-GIP-Gs/β1/γ2
26.67Single5TGZAM65385TGZ-CB1-AM6538
26.67Single6KPFPubChem 1459158896KPF-CB2-PubChem 145915889-Gi1/β1/γ2
26.67Single7YK7DC5910537YK7-RXFP4-DC591053-Gi2/β1/γ2
26.67Single7YU4ONO-07405567YU4-LPA1-ONO-0740556
26.67Single8T1WCVN4248T1W-GPR6-CVN424
26.67Single8X9TAP5038X9T-ADGRD1-AP503-chim(NtGi1-Gs)/β1/γ2
26.67Single8ZSSRO52633978ZSS-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
26.67Single9CHXS-Carazolol9CHX-β2-S-Carazolol
26.67Consensusgluc_on_gpOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
26.47Single7SK9CCX6627SK9-ACKR3-CCX662
26.47Single7XBXCX3CL17XBX-CX3CR1-CX3CL1-Gi1/β1/γ2
26.47Single8JLRA776368JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2
26.47Single8XQLCholesterol8XQL-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
26.47Single8XQOCholesterol8XQO-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
26.47Single8Y72Peptide8Y72-μ-Peptide-BMS-986122-Gi1/β1/γ2
26.47Consensusdop_onOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
26.32Single7Y64C5a anaphylatoxin7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
26.32Single8HCQEndothelin-18HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Single8HK5Complement C58HK5-C5a1-Complement C5-Gi1/β1/γ2
26.32Single8XVHEndothelin-18XVH-ETB-Endothelin-1-chim(Gs-CtGq)/β1/γ2
26.32Consensuseta_onOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Consensuseta_on_gpOrthosteric Ligand8HCQ-ETA-Endothelin-1-chim(NtGi1-Gs-CtGq)/β1/γ2
26.32Consensusopioid_onOrthosteric Ligandmop_on nop_on dop_on kop_on
26.19Single8HBDIRL16208HBD-ETB-IRL1620-Gi1/β1/γ2
26.19Consensusendothelin_on_gpOrthosteric Ligandetb_on_gp eta_on_gp
26.19Consensusetb_on_gpOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
26.19Consensusglp1_onOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
25.81Single5C1MBU725C1M-μ-BU72
25.81Single5OM4PubChem 1355666095OM4-A2A-PubChem 135566609-Na
25.81Single5ZK33-quinuclidinyl-benzilate5ZK3-M2-3-quinuclidinyl-benzilate
25.81Single7CKXA776367CKX-D1-A77636-Gs/β1/γ2
25.81Single7EPFNAM5977EPF-mGlu2; mGlu2-NAM597
25.81Single7YU3ONO-07405567YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.81Single8EFBOliceridine8EFB-μ-Oliceridine-Gi1/β1/γ2
25.81Single8J18(3R)-3-Hydroxydodecanoic acid8J18-GPR84-(3R)-3-Hydroxydodecanoic acid-Gi1/β1/γ2
25.81Single8J6JGSK2560738J6J-HCA2-GSK256073-Gi1/β1/γ2
25.81Single8JXSPF-61428JXS-D1-PF-6142
25.81Single8K8JFenofibrate8K8J-CB1-Fenofibrate-chim(Gs-CtGq)/β1/γ2
25.81Single9I52A1IZU9I52-D1-A1IZU-Gs/β1/γ2
25.81Consensusd1_onOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
25.81Consensuslipid_onOrthosteric Ligandcannabinoid_on ffa_on lpl_on prostanoid_on leukotriene_on
25.81Consensuslipid_on_gpOrthosteric Ligandcannabinoid_on_gp ffa_on_gp lpl_on_gp prostanoid_on_gp leukotriene_on_gp
25.81Consensuss1p5_offOrthosteric Ligand7YXA-S1P5-ONO-5430608
25.81Consensusta1_onOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.81Consensustrace-amine_onOrthosteric Ligandta1_on
25.71Single6X19CHU-1286X19-GLP-1-CHU-128-Gs/β1/γ2
25.71Single7QA8Peptide7QA8-STE2-Peptide
25.71Single7QA8Peptide7QA8-STE2-Peptide
25.71Single7RTBPeptide-197RTB-GLP-1-Peptide-19-Gs/β1/γ2
25.71Single7T6UCGEN-855A7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2
25.71Single7TD4Siponimod7TD4-S1P1-Siponimod-Gi1/β1/γ2
25.71Single7W0PElabela7W0P-Apelin-Elabela-Gi1/β1/γ2
25.71Single7WVWfMYFINILTL7WVW-FPR2-ALX-fMYFINILTL-Gi2/β1/γ2
25.71Single8G59TUG-8918G59-FFA4-TUG-891-chim(Gi1-CtGq)/β1/γ2
25.71Single8GHVAMG3158GHV-CB1-AMG315-Gi1/β1/γ2
25.71Single8PKMBefiradol8PKM-5-HT1A-Befiradol-Gi1/β1/γ1
25.71Consensuslpl_onOrthosteric Ligands1p_on lpa_on
25.71Consensuslpl_on_gpOrthosteric Ligands1p_on_gp lpa_on_gp
25.64Single7YKDChemerin-97YKD-CML1-Chemerin-9-Gi1/β1/γ2
25.64Single9KFKRelaxin-39KFK-RXFP4-Relaxin-3-Gi2/β1/γ2
25.64Consensusgi_compl-peptOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
25.64Consensusgi_proteinOrthosteric Ligandgi_chemokine gi_chemerin
25.64Consensusopioid_on_gpOrthosteric Ligandmop_on_gp nop_on_gp dop_on_gp kop_on_gp
25.64Consensusprotein_on_gpOrthosteric Ligandchemokine_on_gp chemerin_on_gp
25.64Consensussecretin_onOrthosteric Ligand7D3S-Secretin-Secretin-Gs/β1/γ2
25.58Consensusglp1_on_gpOrthosteric Ligand7S1M-GLP-1-Ex4-D-Ala-Gs/β1/γ2 7X8R-GLP-1-BOC5-Gs/β1/γ2 6X19-GLP-1-CHU-128-Gs/β1/γ2 6X1A-GLP-1-Danuglipron-Gs/β1/γ2 6X18-GLP-1-GLP-1-Gs/β1/γ2 8JIP-GLP-1-MEDI0382-chim(NtGi1-Gs)/β1/γ2 7C2E-GLP-1-PubChem 149050799-Gs/β1/γ2 7KI0-GLP-1-Semaglutide-Gs/β1/γ2 7KI1-GLP-1-Taspoglutide-Gs/β1/γ2 7X8S-GLP-1-WB4-24-Gs/β1/γ2 8JIS-GLP-1-Peptide-15-chim(NtGi1-Gs)/β1/γ2 7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
25.00Single3QAKUK-4320973QAK-A2A-UK-432097
25.00Single3SN6BI1671073SN6-β2-BI167107-Gs/β1/γ2
25.00Single3UON3-quinuclidinyl-benzilate3UON-M2-3-quinuclidinyl-benzilate
25.00Single5A8E7-Methylcyanopindolol5A8E-β1-7-Methylcyanopindolol-Na
25.00Single5NX2GLP-1 (Truncated)5NX2-GLP-1-GLP-1 (Truncated)
25.00Single5V54Methiothepin5V54-5-HT1B-Methiothepin
25.00Single6DO1Angiotensin-like peptide S1I86DO1-AT1-Angiotensin-like peptide S1I8
25.00Single6N4BMDMB-Fubinaca6N4B-CB1-MDMB-Fubinaca-Gi1/β1/γ2
25.00Single6NI3BI1671076NI3-β2-BI167107-Gs/β1/γ2
25.00Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
25.00Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
25.00Single7E14Orforglipron7E14-GLP-1-Orforglipron-PubChem 156022738-Gs/β1/γ2
25.00Single7EW7SEW28717EW7-S1P1-SEW2871-Gi1/β1/γ2
25.00Single7RKMFractalkine7RKM-US28-Fractalkine-Gi1/β1/γ2
25.00Single7VBINon-Acylated Tirzepatide7VBI-GLP-1-Non-Acylated Tirzepatide-Gs/β1/γ2
25.00Single7XMSSomatostatin-147XMS-SST4-Somatostatin-14-Gi1/β1/γ2
25.00Single7YU5ONO-07405567YU5-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Single8DZPmomSalB8DZP-κ-momSalB-Gi1/β1/γ2
25.00Single8EF5Fentanyl8EF5-μ-Fentanyl-Gi1/β1/γ2
25.00Single8F7SDeltorphin8F7S-δ-Deltorphin-Gi1/β1/γ2
25.00Single8ID39-Hydroxystearic acid8ID3-FFA4-9-Hydroxystearic acid-Gi1/β1/γ2
25.00Single8IRURotigotine8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Single8IRVRotigotine8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
25.00Single8JZZC5a-desArg8JZZ-C5a1-C5a-desArg-Go/β1/γ2
25.00Single8T1VPubChem 1183102098T1V-GPR6-PubChem 118310209-Na
25.00Single8Z7JAgonistic antibody8Z7J-Apelin-Agonistic antibody-Gi1/β1/γ2
25.00Single8ZH8QRF-Amide8ZH8-QRFP-QRF-Amide-Gq/β1/γ1
25.00Single8ZJGChemerin8ZJG-CML1-Chemerin-Gi1/β1/γ2
25.00Single9ASTLymphotactin9AST-XCR1-Lymphotactin-Gi1/β1/γ2
25.00Single9B65KCA9B65-CB1-KCA-Gi1/β1/γ2
25.00Single9I54A1IZV9I54-D1-A1IZV-Gs/β1/γ2
25.00Single9JMCDS-3801b9JMC-Motilin-DS-3801b-chim(Gs-CtGq)/β1/γ2
25.00Consensus5ht1_offOrthosteric Ligand5ht1b_off
25.00Consensus5ht1b_offOrthosteric Ligand5V54-5-HT1B-Methiothepin
25.00Consensuscompl-peptide_onOrthosteric Ligandc5a1_on c3a_on
25.00Consensusd1_on_gpOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2
25.00Consensusd4_on_gpOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
25.00Consensusd5_on_gpOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
25.00Consensusdop_on_gpOrthosteric Ligand8F7S-δ-Deltorphin-Gi1/β1/γ2
25.00Consensusgi_lpaOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
25.00Consensusglp2_onOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
25.00Consensusglp2_on_gpOrthosteric Ligand7D68-GLP-2-GLP-2-Gs/β1/γ2
25.00Consensusgq_class-aOrthosteric Ligandgq_peptide gq_amine gq_nucleotide
25.00Consensusgs_dopamineOrthosteric Ligand7F0T-D1-Dopamine-Gs/β1/γ2 7CKW-D1-Fenoldopam-Gs/β1/γ2 7CKY-D1-PW0464-Gs/β1/γ2 8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2 8IRR-D1-Rotigotine-Gs/β1/γ2 7JV5-D1-SKF81297-Gs/β1/γ2 7JVP-D1-SKF83959-Gs/β1/γ2 7X2D-D1-Tavapadon-Gs/β1/γ2 7CKX-D1-A77636-Gs/β1/γ2 7JVQ-D1-Apomorphine-Gs/β1/γ2
25.00Consensuslpa_onOrthosteric Ligandlpa1_on
25.00Consensuslpa_on_gpOrthosteric Ligandlpa1_on_gp
25.00Consensusm3_offOrthosteric Ligand4U15-M3-Tiotropium 4U16-M3-N-Methyl-Scopolamine 5ZHP-M3-PubChem 134828589
25.00Consensusmuscarinic_offOrthosteric Ligandm2_off m3_off m4_off m5_off m1_off
25.00Consensusta1_on_gpOrthosteric Ligand8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2 8W88-TA1-SEP-363856-Gs/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8ZSP-TA1-LSD-chim(NtGi1L-Gs-CtGq)/β1/γ2
25.00Consensustrace-amine_on_gpOrthosteric Ligandta1_on_gp
24.44Consensusgluc_onOrthosteric Ligand6LMK-Glucagon-Glucagon-Gs/β1/γ2 8JIT-Glucagon-MEDI0382-Gs/β1/γ2 7V35-Glucagon-Peptide-20-Gs/β1/γ2
24.39Single6IGLIRL16206IGL-ETB-IRL1620
24.39Single8IY5Endothelin-18IY5-ETB-Endothelin-1-Gi1/β1/γ2
24.39Single8IY6Endothelin-18IY6-ETB-Endothelin-1
24.39Consensusctlike_on_gpOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
24.39Consensusetb_onOrthosteric Ligand8IY5-ETB-Endothelin-1-Gi1/β1/γ2 8HBD-ETB-IRL1620-Gi1/β1/γ2
24.32Single5WF5UK-4320975WF5-A2A-UK-432097
24.32Single6LW5WKYMVm6LW5-FPR2-ALX-WKYMVm
24.32Consensuscompl-peptide_on_gpOrthosteric Ligandc5a1_on_gp c3a_on_gp
24.32Consensusfpr2-alx_onOrthosteric Ligand7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2 7T6U-FPR2-ALX-CGEN-855A-Gi1/β1/γ2 7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2 7WVY-FPR2-ALX-Amyloid-β42-Gi2/β1/γ2 7T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2 6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
24.24Single5CXVTiotropium5CXV-M1-Tiotropium
24.24Single5F8UCyanopindolol5F8U-β1-Cyanopindolol
24.24Single6A93Risperidone6A93-5-HT2A-Risperidone
24.24Single7BZ2Arformoterol7BZ2-β2-Arformoterol-Gs/β1/γ2
24.24Single7DFPSpiperone7DFP-D2-Spiperone
24.24Single7EO4BAF3127EO4-S1P1-BAF312-Gi1/β1/γ2
24.24Single7EPENAM5637EPE-mGlu2; mGlu2-NAM563
24.24Single7EVYSiponimod7EVY-S1P1-Siponimod-Gi1/β1/γ2
24.24Single7EW2Fingolimod7EW2-S1P3-Fingolimod-Gi1/β1/γ2
24.24Single7WCMMBX-29827WCM-GPR119-MBX-2982-Gs/β1/γ2
24.24Single8FYE4-F,5-MeO-PyrT8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1
24.24Single8FYTLSD8FYT-5-HT1A-LSD-Gi1/β1/γ1
24.24Single8I9AEP548I9A-C3aB-EP54-chim(NtGi1-Gs-CtGq)/β1/γ2
24.24Single8IA8E7 peptide8IA8-C3aB-E7 peptide-Gi1/β1/γ2
24.24Single8XQNCholesterol8XQN-TAS2R14-Cholesterol-Aristolochic acid A-Gi1/β1/γ1
24.24Single8XQSCholesterol8XQS-TAS2R14-Cholesterol-Flufenamic acid-Gi1/β1/γ1
24.24Single9GYOP3959GYO-GPBA-P395-chim(NtGi1-Gs)/β1/γ2
24.24Single9M4QDoxazosin9M4Q-Alpha1A-Doxazosin
24.24Single9MQLIsoquinuclidine9MQL-κ-Isoquinuclidine
24.24Consensusgi_lipidOrthosteric Ligandgi_cannabinoid gi_ffa gi_leukotriene gi_lpa gi_s1p
24.24Consensuskop_onOrthosteric Ligand8F7W-κ-Dynorphin-Gi1/β1/γ2 8DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2 8DZP-κ-momSalB-Gi1/β1/γ2
24.24Consensusm1_offOrthosteric Ligand5CXV-M1-Tiotropium
24.24Consensuss1p1_onOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
24.24Consensuss1p1_on_gpOrthosteric Ligand7VIE-S1P1-S1P-Gi1/β1/γ2 7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2 7VIG-S1P1-CBP-307-Gi1/β1/γ2 7EVY-S1P1-Siponimod-Gi1/β1/γ2 7EVZ-S1P1-Cenerimod-Gi1/β1/γ2 7EW0-S1P1-Ozanimod-Gi1/β1/γ2 7EW7-S1P1-SEW2871-Gi1/β1/γ2
24.14Single3V2WPubChem 518926453V2W-S1P1-PubChem 51892645
24.14Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
24.14Single7WF7S1P7WF7-S1P1-S1P-Gi1/β1/γ2
24.14Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
24.14Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
24.14Consensuss1p1_offOrthosteric Ligand3V2W-S1P1-PubChem 51892645
23.91Consensusmc2_onOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
23.91Consensusmc2_on_gpOrthosteric Ligand8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
23.81Consensusbb2_onOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
23.81Consensusbb2_on_gpOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
23.81Consensusbombesin_onOrthosteric Ligandbb2_on
23.81Consensusbombesin_on_gpOrthosteric Ligandbb2_on_gp
23.81Consensusccr5_on_gpOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
23.81Consensuscrf1_onOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
23.81Consensusgq_bombesinOrthosteric Ligand7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2 7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
23.68Single6JODAngiotensin II6JOD-AT2-Angiotensin II
23.68Single7AD3Alpha-factor mating pheromone7AD3-STE2-α-factor mating pheromone-Gi1/STE4/γ2
23.68Single8IHFMK68928IHF-HCA2-MK6892-Gi1/β1/γ2
23.68Single8XZJWN3538XZJ-Apelin-WN353-Gi1/β1/γ2
23.68Single9BKKCholecystokinin-89BKK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
23.68Consensusc5a1_on_gpOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
23.68Consensuscxcr3_on_gpOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
23.68Consensusprotein_offonOrthosteric Ligandprotein_off protein_on
23.68Consensusprotein_offon_gpOrthosteric Ligandprotein_on_gp protein_off
23.53Single2YCZIodocyanopindolol2YCZ-β1-Iodocyanopindolol
23.53Single5X93K-87945X93-ETB-K-8794
23.53Single6BQHRitanserin6BQH-5-HT2C-Ritanserin
23.53Single6DDFDamgo6DDF-μ-Damgo-Gi1/β1/γ2
23.53Single7EW0Ozanimod7EW0-S1P1-Ozanimod-Gi1/β1/γ2
23.53Single7MTSADX551647MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
23.53Single7SK8CCX6627SK8-ACKR3-CXCL12-CCX662
23.53Single7U2KC6-guano7U2K-μ-C6-guano-Gi1/β1/γ2
23.53Single7VGY2-Iodomelatonin7VGY-MT1-2-Iodomelatonin-Gi1/β1/γ2
23.53Single7X8RBOC57X8R-GLP-1-BOC5-Gs/β1/γ2
23.53Single7XK2MK68927XK2-HCA2-MK6892-Gi1/β1/γ2
23.53Single8E9X2-Deoxycytidine8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2
23.53Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
23.53Single8IYSTUG-8918IYS-FFA4-TUG-891-GDP-chim(NtGi1L-Gq)/β1/γ2
23.53Single8S2TIsoprenaline8S2T-β1-Isoprenaline-chim(NtGi1-Gs)/β1/γ2
23.53Single9AS02-bromo-LSD9AS0-5-HT2A-2-bromo-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
23.53Single9IZFNKP9IZF-LPA1-NKP-Gi1/β1/γ2
23.53Consensus5ht2c_offOrthosteric Ligand6BQH-5-HT2C-Ritanserin
23.53Consensusc3a_on_gpOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
23.53Consensusd2_offOrthosteric Ligand6CM4-D2-Risperidone 6LUQ-D2-Haloperidol 7DFP-D2-Spiperone
23.53Consensusendothelin_offOrthosteric Ligandetb_off
23.53Consensusetb_offOrthosteric Ligand5X93-ETB-K-8794 5XPR-ETB-Bosentan 6K1Q-ETB-IRL2500
23.33Single7T32ZM-2413857T32-A2A-ZM-241385
23.33Single7YK6PubChem 1383196747YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
23.33Single8GGSConstrained Epinephrine8GGS-β2-Constrained Epinephrine
23.33Single8GGTConstrained Epinephrine8GGT-β2-Constrained Epinephrine
23.33Single8GUQOlorinab8GUQ-CB2-Olorinab-Gi1/β1/γ2
23.33Single8JLQFenoldopam8JLQ-TA1-Fenoldopam-Gs/β1/γ2
23.33Single8K9KDamgo8K9K-μ-Damgo-Gi3/β1/γ1
23.33Single8W88SEP-3638568W88-TA1-SEP-363856-Gs/β1/γ2
23.33Single8WC8ZH86518WC8-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
23.33Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
23.33Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
23.33Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
23.33Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
23.33Single9KPDSA09KPD-TAS2R16-SA0-chim(Gs-CtGt3)/β1/γ2
23.33Consensusghrelin_offOrthosteric Ligand6KO5-Ghrelin-PubChem 57400002 7F83-Ghrelin-PF-05190457
23.26Consensusmelanocortin_onOrthosteric Ligandmc1_on mc4_on mc2_on mc3_on mc5_on
23.26Consensusmelanocortin_on_gpOrthosteric Ligandmc1_on_gp mc4_on_gp mc2_on_gp mc3_on_gp mc5_on_gp
23.08Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
23.08Single7X9BNeuropeptide-Y7X9B-Y2-Neuropeptide-Y-Gi1/β1/γ2
23.08Single8IA2C5a anaphylatoxin8IA2-C5a1-C5a anaphylatoxin-Go/β1/γ2
23.08Single8XGOTAK4488XGO-Kiss1-TAK448-chim(NtGi1-Gq)/β1/γ2
23.08Single8ZPSPrRP208ZPS-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
23.08Single9JFYhNPSF9JFY-NPFF2-hNPSF-Gi1/β1/γ2
23.08Consensuscml1_on_gpOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
23.08Consensusgi_apelinOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
22.86Single5WF6UK-4320975WF6-A2A-UK-432097
22.86Single6G79Donitriptan6G79-5-HT1B-Donitriptan-Go/β1/γ2
22.86Single7RKFFractalkine7RKF-US28-Fractalkine-GDP-chim(NtGi1-G11)/β1/γ2
22.86Single7YJ4INSL57YJ4-RXFP4-INSL5-Gi2/β1/γ2
22.86Single8H4IDoconexent8H4I-FFA4-Doconexent-chim(NtGi1-Gs)/β1/γ2
22.86Single8QJ2pN1628QJ2-MC4-pN162-Gs
22.86Single8X5YAstemizole8X5Y-H1-Astemizole
22.86Single9IPVJR14a9IPV-C3aB-JR14a-Gi1/β1/γ2
22.86Single9M0RNeuropeptide VF9M0R-NPFF1-Neuropeptide VF-Gi1/β1/γ2
22.86Single9V2NMacimorelin9V2N-Ghrelin-Macimorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
22.86Consensuscxcr3_onOrthosteric Ligand8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2
22.86Consensusformylpeptide_onOrthosteric Ligandfpr2-alx_on fpr1-alx_on
22.73Consensuscrf1_on_gpOrthosteric Ligand6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2 6P9X-CRF1-Corticoliberin-Gs/β1/γ2
22.58Single2Y04Salbutamol2Y04-β1-Salbutamol
22.58Single3NY8ICI118-5513NY8-β2-ICI118-551
22.58Single3ZPQ4-(piperazin-1- yl)-1H-indole3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na
22.58Single3ZPR4-methyl-2-(piperazin-1-yl)3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
22.58Single4DAJTiotropium4DAJ-M3-Tiotropium
22.58Single4GBRS-Carazolol4GBR-β2-S-Carazolol
22.58Single4U16N-Methyl-Scopolamine4U16-M3-N-Methyl-Scopolamine
22.58Single5OLZPubChem 1355666095OLZ-A2A-PubChem 135566609-Na
22.58Single5OM1PubChem 1355666095OM1-A2A-PubChem 135566609-Na
22.58Single6PS2S-Alprenolol6PS2-β2-S-Alprenolol
22.58Single7CRHSKF839597CRH-D1-SKF83959-Gs/β1/γ2
22.58Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
22.58Single7T6VfMLFII7T6V-FPR2-ALX-fMLFII-Gi1/β1/γ2
22.58Single7VIES1P7VIE-S1P1-S1P-Gi1/β1/γ2
22.58Single7WC7Lisuride7WC7-5-HT2A-Lisuride
22.58Single7XJHIsoproterenol7XJH-β3-Isoproterenol-Gs/β1/γ2
22.58Single7YXAONO-54306087YXA-S1P5-ONO-5430608
22.58Single8CU6LJ-45178CU6-A2A-LJ-4517
22.58Single8CU7LJ-45178CU7-A2A-LJ-4517-Na
22.58Single8GE9Constrained Epinephrine8GE9-β2-Constrained Epinephrine-Gs/β1/γ2
22.58Single8I7VAcipimox8I7V-HCA2-Acipimox-Gi1/β1/γ2
22.58Single8J6PNiacin8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
22.58Single8JXRLSD8JXR-D1-LSD
22.58Single8UH3Setiptiline8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
22.58Single8UNVConstrained Epinephrine8UNV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.58Single8UNZConstrained Epinephrine8UNZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.58Single8UO2Constrained Epinephrine8UO2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
22.58Single8VVGGB188VVG-κ-GB18-Gi1/β1/γ2
22.58Single8W87METH8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2
22.58Single8W8ARO52563908W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
22.58Single9AS1DMT9AS1-5-HT2A-DMT
22.58Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
22.58Single9BQJRO769BQJ-μ-RO76-Gi1/β1/γ2
22.58Single9H37A1IR09H37-A2A-A1IR0-Na
22.58Single9KFJPubChem 1383196749KFJ-RXFP3-PubChem 138319674-Gi2/β1/γ2
22.58Consensusalicarboxylic_on_gpOrthosteric Ligandsuccinate_on_gp hca_on_gp
22.58Consensusd5_onOrthosteric Ligand8IRV-D5-Rotigotine-chim(NtGi1-Gs)/β1/γ2
22.58Consensusdopamine_offOrthosteric Ligandd2_off d3_off
22.58Consensusgi_alicarboxylicOrthosteric Ligandgi_hca gi_succinate
22.58Consensusgi_hcaOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
22.58Consensusgs_trace-amineOrthosteric Ligand8W88-TA1-SEP-363856-Gs/β1/γ2 8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2 8JLO-TA1-Ulotaront-Gs/β1/γ2 8WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2 8WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2 8JLR-TA1-A77636-chim(NtGi1-Gs)/β1/γ2 8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2 8W87-TA1-METH-chim(NtGi1L-Gs)/β1/γ2 8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2 8JLP-TA1-Ralmitaront-Gs/β1/γ2 8W8A-TA1-RO5256390-chim(NtGi1L-Gs)/β1/γ2
22.58Consensushca2_onOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2
22.58Consensushca2_on_gpOrthosteric Ligand8J6R-HCA2-MK6892-Gi1/β1/γ2 8IHI-HCA2-Acifran-Gi1/β1/γ2 8IHH-HCA2-LUF6283-Gi1/β1/γ2 8I7V-HCA2-Acipimox-Gi1/β1/γ2 8JIM-HCA2-MMF-Gi1/β1/γ2 8I7W-HCA2-GSK256073-Gi1/β1/γ2
22.58Consensushca_on_gpOrthosteric Ligandhca2_on_gp
22.58Consensuslipid_offOrthosteric Ligandcannabinoid_off paf_off lpl_off prostanoid_off leukotriene_off
22.50Single7QBIAlpha-factor mating pheromone7QBI-STE2-α-factor mating pheromone
22.50Single8XQFApelin-138XQF-Apelin-Apelin-13-Gi1/β1/γ2
22.50Single8XVEBQ30208XVE-ETB-BQ3020-chim(Gs-CtGq)/β1/γ2
22.50Consensusctlike_onOrthosteric Ligand6E3Y-CT Like-Calcitonin gene-related peptide-1-Gs/β1/γ2; RAMP1
22.22Single7F4ISHU91197F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
22.22Single7W2ZGhrelin7W2Z-Ghrelin-Ghrelin-Go/β1/γ2
22.22Single8J6RMK68928J6R-HCA2-MK6892-Gi1/β1/γ2
22.22Single8XGMChemerin8XGM-CML2-Chemerin-Gi1/β1/γ2
22.22Single9L3YRetinoic acid receptor responder protein 29L3Y-CML2-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
22.22Consensuschemerin_on_gpOrthosteric Ligandcml1_on_gp
22.22Consensuscml1_onOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
22.22Consensusgi_chemerinOrthosteric Ligand7YKD-CML1-Chemerin-9-Gi1/β1/γ2
22.22Consensusp2y_onOrthosteric Ligandp2y1_on p2y10_on p2y12_on
21.95Single7F4FAfamelanotide7F4F-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
21.95Single7F53Alpha-MSH7F53-MC4-α-MSH-Gs/β1/γ2
21.95Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
21.95Single8FEG(DNCP)-Beta-Naloxamine8FEG-κ-(DNCP)-β-Naloxamine-Gi1/β1/γ2
21.95Single9K26PrRP319K26-PrRP-PrRP31-Gi1/β1/γ2
21.95Single9KDFRES-701-39KDF-ETB-RES-701-3
21.88Single2RH1S-Carazolol2RH1-β2-S-Carazolol
21.88Single2Y03Isoprenaline2Y03-β1-Isoprenaline
21.88Single2YCWS-Carazolol2YCW-β1-S-Carazolol
21.88Single4RWDDIPP-NH24RWD-δ-DIPP-NH2-Na
21.88Single5D6LS-Carazolol5D6L-β2-S-Carazolol
21.88Single5JQHS-Carazolol5JQH-β2-S-Carazolol
21.88Single5NM2ZM-2413855NM2-A2A-ZM-241385-Na
21.88Single5TVNLSD5TVN-5-HT2B-LSD
21.88Single5X7DS-Carazolol5X7D-β2-S-Carazolol-Cmpd-15
21.88Single5XPRBosentan5XPR-ETB-Bosentan
21.88Single6GDGNECA6GDG-A2A-NECA-Gs/β1/γ1
21.88Single6ME82-Phenylmelatonin6ME8-MT2-2-Phenylmelatonin
21.88Single6PS6Timolol6PS6-β2-Timolol
21.88Single7C4SS1P7C4S-S1P3-S1P
21.88Single7EO2FTY720-P7EO2-S1P1-FTY720-P-Gi1/β1/γ2
21.88Single7LD3Adenosine7LD3-A1-Adenosine-MIPS521-Gi2/β1/γ2
21.88Single7M3JNPS-2143; PO47M3J-CaS-NPS-2143; PO4
21.88Single7SBFPZM217SBF-μ-PZM21-Gi1/β1/γ2
21.88Single7TD3S1P7TD3-S1P1-S1P-Gi1/β1/γ2
21.88Single7TRKIperoxo7TRK-M4-Iperoxo-Gi1/β1/γ2
21.88Single7W41PD1762527W41-BB2-PD176252
21.88Single7XKAConstrained Epinephrine7XKA-β2-Constrained Epinephrine
21.88Single8DZQmomSalB8DZQ-κ-momSalB-Go/β1/γ2
21.88Single8DZRGR89,6968DZR-κ-GR89,696-chim(NtGi2-Gt3)/β1/γ2
21.88Single8E9ZIperoxo8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.88Single8GDZConstrained Epinephrine8GDZ-β2-Constrained Epinephrine-Gs/β1/γ2
21.88Single8GEBConstrained Epinephrine8GEB-β2-Constrained Epinephrine-Gs/β1/γ2
21.88Single8GEGConstrained Epinephrine8GEG-β2-Constrained Epinephrine-Gs/β1/γ2
21.88Single8GGBConstrained Epinephrine8GGB-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8QOTNanobody-E8QOT-μ-Nanobody-E
21.88Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
21.88Single8TF5Oleic acid8TF5-GPR6-Oleic acid
21.88Single8UNNConstrained Epinephrine8UNN-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8UNPConstrained Epinephrine8UNP-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.88Single8UUJFCH-22964138UUJ-HCA2-FCH-2296413-Gi1/β1/γ2
21.88Single8YICSAR2477998YIC-S1P1-SAR247799-Gi1/β1/γ2
21.88Single8ZMFA1L108ZMF-5-HT2C-A1L10
21.88Single8ZPTPrRP208ZPT-PrRP-PrRP20-chim(NtGi1-Gs-CtGq)/β1/γ2
21.88Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
21.88Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
21.88Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
21.88Single9CIBFCH-22964139CIB-HCA2-FCH-2296413
21.88Single9DYDAsenapine9DYD-5-HT1A-Asenapine-Go/β1/γ2
21.88Single9DYFAsenapine9DYF-5-HT1A-Asenapine-Gi1/β1/γ2
21.88Single9EAHOlmesartan9EAH-AT1-Olmesartan-Nanobody AT209
21.88Single9EE8Adenosine9EE8-A2A-Adenosine-Gs/β1/γ2
21.88Single9K07DSO-5a9K07-BB3-DSO-5a-chim(NtGi2L-Gs-CtGq)/β1/γ2
21.88Single9MQKIsoquinuclidine9MQK-κ-Isoquinuclidine
21.88Consensusadenosine_offOrthosteric Liganda1_off a2_off
21.88Consensusamine_offOrthosteric Ligand5ht_off adrenergic_off dopamine_off histamine_off muscarinic_off
21.88Consensusamine_offonOrthosteric Ligandamine_off amine_on
21.88Consensusamine_offon_gpOrthosteric Ligandamine_on_gp amine_off
21.88Consensusamine_onOrthosteric Ligand5ht_on adrenergic_on dopamine_on histamine_on muscarinic_on trace-amine_on
21.88Consensusbb2_offOrthosteric Ligand7W41-BB2-PD176252
21.88Consensusbeta2_offOrthosteric Ligand2RH1-β2-S-Carazolol 6PS3-β2-S-Carvedilol 6PS5-β2-S-Propranolol 3D4S-β2-Timolol 3NY8-β2-ICI118-551 3NY9-β2-ICI118-551 6PRZ-β2-S-Alprenolol
21.88Consensusbeta_offOrthosteric Ligandbeta1_off beta2_off
21.88Consensusbombesin_offOrthosteric Ligandbb2_off
21.88Consensusd2_onOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
21.88Consensusd4_onOrthosteric Ligand8IRU-D4-Rotigotine-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.88Consensusgi_adrenergicOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 6K42-α2b-Dexmedetomidine-Gi1/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
21.88Consensusgs_amineOrthosteric Ligandgs_5ht gs_adrenergic gs_dopamine gs_histamine gs_trace-amine
21.88Consensush1_offOrthosteric Ligand8X63-H1-Mepyramine 3RZE-H1-Cidoxepin 8X5Y-H1-Astemizole
21.88Consensuslpa1_onOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.88Consensuslpa1_on_gpOrthosteric Ligand7TD1-LPA1-LPA-Gi1/β1/γ2 7YU3-LPA1-ONO-0740556-Gi1/β1/γ2
21.88Consensusm2_offOrthosteric Ligand5ZKC-M2-N-Methyl-Scopolamine 5ZK3-M2-3-quinuclidinyl-benzilate 5ZKB-M2-AF-DX 384
21.88Consensusrxfp4_onOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.88Consensusrxfp4_on_gpOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.62Single7DDZJNJ-310200287DDZ-Y2-JNJ-31020028
21.62Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
21.62Single8F7WDynorphin8F7W-κ-Dynorphin-Gi1/β1/γ2
21.62Single8SG1Chemerin-98SG1-CML1-Chemerin-9-Gi1/β1/γ2
21.62Single9E82SDF-1-beta9E82-ACKR3-SDF-1-β-Arrestin2
21.62Consensusnpy2_offOrthosteric Ligand7DDZ-Y2-JNJ-31020028
21.62Consensussst4_onOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
21.62Consensussst4_on_gpOrthosteric Ligand7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2
21.43Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
21.43Single7QBCAlpha-factor mating pheromone7QBC-STE2-α-factor mating pheromone
21.43Single8GGEConstrained Epinephrine8GGE-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
21.43Single8RQLFlufenamic acid8RQL-TAS2R14-Flufenamic acid-Flufenamic acid-chim(NtGi1-Gt3)/β1/γ2
21.43Single8WWNMCH8WWN-MCH1-MCH-Gi1/β1/γ2
21.43Consensusbk2_onOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
21.43Consensusbk2_on_gpOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
21.43Consensusbradykinin_onOrthosteric Ligandbk2_on
21.43Consensusbradykinin_on_gpOrthosteric Ligandbk2_on_gp
21.43Consensusgq_bradykininOrthosteric Ligand7F6H-BK2-Bradykinin-Gq/β1/γ2 7F6I-BK2-Kallidin-Gq/β1/γ2
21.43Consensusgs_melanocortinOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2 8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1 8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2 7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2
21.21Single3P0GBI1671073P0G-β2-BI167107
21.21Single4DJHJDTic4DJH-κ-JDTic
21.21Single4IAQDihydroergotamine4IAQ-5-HT1B-Dihydroergotamine
21.21Single4LDLHydroxybenzylisoproterenol4LDL-β2-Hydroxybenzylisoproterenol
21.21Single4U15Tiotropium4U15-M3-Tiotropium
21.21Single5D5AS-Carazolol5D5A-β2-S-Carazolol
21.21Single5D5BS-Carazolol5D5B-β2-S-Carazolol
21.21Single5ZHPPubChem 1348285895ZHP-M3-PubChem 134828589
21.21Single5ZKBAF-DX 3845ZKB-M2-AF-DX 384
21.21Single6DDEDamgo6DDE-μ-Damgo-Gi1/β1/γ2
21.21Single6H7JIsoprenaline6H7J-β1-Isoprenaline
21.21Single6J21Aprepitant6J21-NK1-Aprepitant
21.21Single6KO5PubChem 574000026KO5-Ghrelin-PubChem 57400002
21.21Single6N48BI1671076N48-β2-BI167107-PubChem 138454256
21.21Single6OL9Tiotropium6OL9-M5-Tiotropium
21.21Single6TQ7SB-3348676TQ7-OX1-SB-334867
21.21Single6WGTLSD6WGT-5-HT2A-LSD
21.21Single7EW3S1P7EW3-S1P3-S1P-Gi1/β1/γ2
21.21Single7JJOIsoprenaline7JJO-β1-Isoprenaline-Gs/β1/γ2
21.21Single7TD1LPA7TD1-LPA1-LPA-Gi1/β1/γ2
21.21Single7TRQIperoxo7TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
21.21Single7U2LPubChem 1632012427U2L-μ-PubChem 163201242-Gi1/β1/γ2
21.21Single7VIGCBP-3077VIG-S1P1-CBP-307-Gi1/β1/γ2
21.21Single7W6PN-pyridin-4-ylisoquinolin-4-amine7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2
21.21Single7W7EPubChem 1649466767W7E-α2a-PubChem 164946676-Go/β1/γ2
21.21Single7WVXHumanin7WVX-FPR2-ALX-Humanin-Gi2/β1/γ2
21.21Single7XY7NECA7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2
21.21Single8DCSCyanopindolol8DCS-β1-Cyanopindolol-Gs/β1/γ2
21.21Single8EA0Iperoxo8EA0-M3-Iperoxo
21.21Single8HDOBAY 60-65838HDO-A2B-BAY 60-6583-Gs/β1/γ2
21.21Single8HPTC5a anaphylatoxin C-terminal peptide8HPT-C5a1-C5a anaphylatoxin C-terminal peptide-Go/β1/γ2
21.21Single8HQCC5a anaphylatoxin8HQC-C5a1-C5a anaphylatoxin-Go/β1/γ2
21.21Single8IHBGSK2560738IHB-HCA2-GSK256073-Gi1/β1/γ2
21.21Single8IHHLUF62838IHH-HCA2-LUF6283-Gi1/β1/γ2
21.21Single8IRRRotigotine8IRR-D1-Rotigotine-Gs/β1/γ2
21.21Single8JXXClobenpropit8JXX-H4-Clobenpropit-Gi1/β1/γ2
21.21Single8UGWPubChem 30865998UGW-A2A-PubChem 3086599
21.21Single8VVFJDTic8VVF-κ-JDTic-Gi1/β1/γ2
21.21Single8XVLZibotentan8XVL-ETA-Zibotentan
21.21Single8XZICMF-0198XZI-Apelin-CMF-019-Gi1/β1/γ2
21.21Single8Y73Peptide8Y73-μ-Peptide-MPAM-15-Gi1/β1/γ2
21.21Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
21.21Single9BJKNaloxone9BJK-μ-Naloxone-NAM
21.21Consensusa2_onOrthosteric Liganda2b_on
21.21Consensusa2_on_gpOrthosteric Liganda2b_on_gp
21.21Consensusa2b_onOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
21.21Consensusa2b_on_gpOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2
21.21Consensusamine_on_gpOrthosteric Ligand5ht_on_gp adrenergic_on_gp dopamine_on_gp histamine_on_gp muscarinic_on_gp trace-amine_on_gp
21.21Consensusbeta1_offOrthosteric Ligand2VT4-β1-Cyanopindolol 2YCW-β1-S-Carazolol 2YCZ-β1-Iodocyanopindolol 5A8E-β1-7-Methylcyanopindolol-Na 3ZPQ-β1-4-(piperazin-1- yl)-1H-indole-Na 3ZPR-β1-4-methyl-2-(piperazin-1-yl)-Na
21.21Consensusgi_dopamineOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 7CMV-D3-PD128907-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2
21.21Consensusgi_relaxinOrthosteric Ligand7YK7-RXFP4-DC591053-Gi2/β1/γ2 7YJ4-RXFP4-INSL5-Gi2/β1/γ2 7YK6-RXFP4-PubChem 138319674-Gi2/β1/γ2
21.21Consensusgs_adenosineOrthosteric Ligand8HDP-A2B-Adenosine-Gs/β1/γ2 8HDO-A2B-BAY 60-6583-Gs/β1/γ2 7XY7-A2B-NECA-chim(NtGi1-Gs)/β1/γ2 7XY6-A2B-BAY 60-6583-chim(NtGi1-Gs)/β1/γ2
21.21Consensusgs_nucleotideOrthosteric Ligandgs_adenosine
21.21Consensush4_on_gpOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
21.21Consensuskop_offOrthosteric Ligand4DJH-κ-JDTic
21.21Consensusm5_offOrthosteric Ligand6OL9-M5-Tiotropium
21.21Consensusmotilin_onOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
21.21Consensusprotein_offOrthosteric Ligandchemokine_off grh_off
21.21Consensusrelaxin_onOrthosteric Ligandrxfp4_on
21.21Consensusrelaxin_on_gpOrthosteric Ligandrxfp4_on_gp
21.15Single8GY7Corticotropin8GY7-MC2-Corticotropin-Ca-chim(NtGi1-Gs)/β1/γ2; MRAP1
21.05Single3OE0CVX153OE0-CXCR4-CVX15
21.05Single6PT2KGCHM076PT2-δ-KGCHM07
21.05Single6W25SHU91196W25-MC4-SHU9119-Ca
21.05Single7MBXCholecystokinin-87MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
21.05Single7O7F6P4-CCL57O7F-CCR5-6P4-CCL5-Gi1/β1/γ1
21.05Single7T6TfMLFII7T6T-FPR1-ALX-fMLFII-Gi1/β1/γ2
21.05Single7XA3CCL27XA3-CCR2-CCL2-Gi1/β1/γ2
21.05Single8K6NPro-neuropeptide-Y8K6N-Y2-Pro-neuropeptide-Y-Gi2/β1/γ1
21.05Single8XIQL7967788XIQ-SST3-L796778-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.05Single8XIRPasireotide8XIR-SST3-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
21.05Single8XZHMM078XZH-Apelin-MM07-Gi1/β1/γ2
21.05Single9K27PrRP319K27-PrRP-PrRP31-chim(NtGi1-Gq)/β1/γ2
21.05Single9U4WGonadoliberin-19U4W-GnRH1-Gonadoliberin-1-chim(NtGi1L-Gs-CtGq)/β1/γ2
21.05Consensusc5a1_onOrthosteric Ligand8HK5-C5a1-Complement C5-Gi1/β1/γ2 7Y66-C5a1-BM213-Gi1/β1/γ2 7Y67-C5a1-C089 peptide-Gi1/β1/γ2 7Y64-C5a1-C5a anaphylatoxin-Gi1/β1/γ2
21.05Consensusccr2_onOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
21.05Consensusccr2_on_gpOrthosteric Ligand7XA3-CCR2-CCL2-Gi1/β1/γ2
21.05Consensusccr_onOrthosteric Ligandccr6_on ccr8_on ccr2_on ccr1_on ccr5_on
21.05Consensusgs_cckOrthosteric Ligand7MBX-CCKA-Cholecystokinin-8-Gs/β1/γ1
20.69Single3OE9IT1t3OE9-CXCR4-IT1t
20.69Single7XP6Strychnine7XP6-TAS2R46-Strychnine-chim(Gs-CtGt3)/β1/γ2
20.69Single8JPNCis-Epoxysuccinic acid8JPN-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ1
20.69Single8WP1Cis-Epoxysuccinic acid8WP1-Succinate-Cis-Epoxysuccinic acid-Gi1/β1/γ2
20.69Single8ZSVRO52633978ZSV-TA1-RO5263397-chim(NtGi1-Gs)/β1/γ2
20.69Single9L3ZLRH7-C29L3Z-CML1-LRH7-C2
20.59Single2YCXCyanopindolol2YCX-β1-Cyanopindolol
20.59Single3D4STimolol3D4S-β2-Timolol
20.59Single4AMIBucindolol4AMI-β1-Bucindolol
20.59Single4LDEBI1671074LDE-β2-BI167107
20.59Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
20.59Single4RWADIPP-NH24RWA-δ-DIPP-NH2
20.59Single6C1RPMX536C1R-C5a1-PMX53-Avacopan; Na
20.59Single6H7NS-Xamoterol6H7N-β1-S-Xamoterol
20.59Single6H7OCyanopindolol6H7O-β1-Cyanopindolol
20.59Single6MXTSalmeterol6MXT-β2-Salmeterol
20.59Single6OS2TRV0266OS2-AT1-TRV026
20.59Single6XOXOrforglipron6XOX-GLP-1-Orforglipron-chim(NtGi1-Gs)/β1/γ2
20.59Single7DH5Mirabegron7DH5-β3-Mirabegron-Gs/β1/γ2
20.59Single7EXDLasmiditan7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.59Single7JNIOlodanrigan7JNI-AT2-Olodanrigan
20.59Single7K15MKD0467K15-BLT1-MKD046-Na
20.59Single7MTRADX551647MTR-mGlu2; mGlu2-Glutamate-ADX55164
20.59Single7SUSPubChem 1227019087SUS-Apelin-PubChem 122701908
20.59Single7T6BS1P7T6B-S1P2-S1P-chim(NtGi1L-G13)/β1/γ2
20.59Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
20.59Single7W0LPubChem 1227019087W0L-Apelin-PubChem 122701908-Gi1/β1/γ2
20.59Single7W0NElabela7W0N-Apelin-Elabela-Gi1/β1/γ2
20.59Single8E9W2-Deoxycytidine8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.59Single8G056-OAU8G05-GPR84-6-OAU-Gi1/β1/γ2
20.59Single8IBUErythromycin-A8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Single8ID9Eicosapentaenoic acid8ID9-FFA4-Eicosapentaenoic acid-Gi1/β1/γ2
20.59Single8IRSRotigotine8IRS-D2-Rotigotine-Gi1/β1/γ2
20.59Single8JJ8Formoterol8JJ8-β2-Formoterol
20.59Single8JJLOlodaterol8JJL-β2-Olodaterol
20.59Single8JZ7MK68928JZ7-HCA2-MK6892-Gi1/β1/γ2
20.59Single9EBIPiclidenoson9EBI-A3A-Piclidenoson-chim(NtGi1L-Gs-CtGi1)/β1/γ2
20.59Single9GL2Befiradol9GL2-5-HT1A-Befiradol-Gs/β1/γ2
20.59Consensus5ht1f_onOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.59Consensus5ht1f_on_gpOrthosteric Ligand7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2
20.59Consensusbeta3_onOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
20.59Consensusbeta3_on_gpOrthosteric Ligand7DH5-β3-Mirabegron-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2
20.59Consensusc3a_onOrthosteric Ligand8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2 8IA8-C3aB-E7 peptide-Gi1/β1/γ2
20.59Consensusccr8_onOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
20.59Consensusd2_on_gpOrthosteric Ligand7JVR-D2-Bromoergocryptine-Gi1/β1/γ2 8IRS-D2-Rotigotine-Gi1/β1/γ2
20.59Consensusgi_amineOrthosteric Ligandgi_5ht gi_muscarinic gi_adrenergic gi_dopamine gi_histamine
20.59Consensusleukotriene_offOrthosteric Ligandblt_off cyslt_off
20.59Consensusmotilin_on_gpOrthosteric Ligand8IBU-Motilin-Erythromycin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
20.59Consensuss1p3_onOrthosteric Ligand7EW3-S1P3-S1P-Gi1/β1/γ2 7EW4-S1P3-CYM5541-Gi1/β1/γ2 7EW2-S1P3-Fingolimod-Gi1/β1/γ2
20.51Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
20.51Single7W40Bombesin7W40-BB2-Bombesin-chim(NtGi1L-Gq)/β1/γ2
20.51Single7WUIIP157WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2
20.51Single7YONPeptide-YY(3-36)7YON-Y2-Peptide-YY(3-36)-Gi1/β1/γ2
20.51Single8J6IMK68928J6I-HCA2-MK6892-Gi1/β1/γ2
20.51Single8ZBISomatostatin-148ZBI-SST3-Somatostatin-14-Gi1/β1/γ2
20.51Consensusapelin_onOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
20.51Consensusapelin_on_gpOrthosteric Ligand8XZH-Apelin-MM07-Gi1/β1/γ2 7W0M-Apelin-PubChem 122701908-Gi1/β1/γ2 8XZJ-Apelin-WN353-Gi1/β1/γ2 8XZF-Apelin-WN561-Gi1/β1/γ2 8XZG-Apelin-Apelin-13-Gi1/β1/γ2
20.51Consensuscrf2_onOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
20.51Consensusp2y_on_gpOrthosteric Ligandp2y1_on_gp p2y10_on_gp p2y12_on_gp
20.00Single2X72All-trans-Retinal2X72-Rhodopsin-All-trans-Retinal-Gt(CT)
20.00Single3VGAZM-2413853VGA-A2A-ZM-241385-Antibody
20.00Single4OR2FITM4OR2-mGlu1; mGlu1-FITM
20.00Single5U09Taranabant5U09-CB1-Taranabant
20.00Single5UNGPubChem 157800525UNG-AT2-PubChem 15780052
20.00Single6B73MP11046B73-κ-MP1104
20.00Single6BQGErgotamine6BQG-5-HT2C-Ergotamine
20.00Single6NWEOctyl-Beta-D-Glucopyranoside6NWE-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
20.00Single6OBAS-Alprenolol6OBA-β2-S-Alprenolol-GTPL11074
20.00Single7EZCUKA7EZC-A2A-UKA
20.00Single7F6HBradykinin7F6H-BK2-Bradykinin-Gq/β1/γ2
20.00Single7JVRBromoergocryptine7JVR-D2-Bromoergocryptine-Gi1/β1/γ2
20.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
20.00Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
20.00Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
20.00Single7P00Substance-P7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Single7P02Protachykinin-17P02-NK1-Protachykinin-1-chim(NtGi1-Gs)/β1/γ2
20.00Single7UM4AS26747237UM4-5-HT5A-AS2674723
20.00Single7W0OElabela7W0O-Apelin-Elabela-Gi1/β1/γ2
20.00Single7WVVfMLFII7WVV-FPR2-ALX-fMLFII-Gi2/β1/γ2
20.00Single7X1UTRH7X1U-TRH-TRH-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single7YMHNorepinephrine7YMH-Alpha1A-Norepinephrine-chim(Gs-CtGq)
20.00Single8DU3PubChem 1055260648DU3-A2A-PubChem 105526064
20.00Single8E9YClozapine-N-oxide8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8EFOPZM218EFO-μ-PZM21-Gi1/β1/γ2
20.00Single8GGAConstrained Epinephrine8GGA-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GGCConstrained Epinephrine8GGC-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
20.00Single8GGRConstrained Epinephrine8GGR-β2-Constrained Epinephrine
20.00Single8GH0Constrained Epinephrine8GH0-β2-Constrained Epinephrine
20.00Single8HCXEndothelin-18HCX-ETB-Endothelin-1-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8I95EP548I95-C3aB-EP54-Go/β1/γ2
20.00Single8ID8TUG-8918ID8-FFA4-TUG-891-Gi1/β1/γ2
20.00Single8IJANiacin8IJA-HCA2-Niacin-Gi1/β1/γ2
20.00Single8JPPSuccinic acid8JPP-Succinate-Succinic acid-chim(Gs-CtGq)/β1/γ1
20.00Single8JSOAMPH8JSO-TA1-AMPH-chim(NtGi1-Gs)/β1/γ2
20.00Single8T3OTUG-8918T3O-FFA4-TUG-891-chim(NtGi2L-Gs-CtGq)/β1/γ2
20.00Single8WC4ZH86518WC4-TA1-ZH8651-chim(NtGi1-Gs)/β1/γ2
20.00Single8WCA2-Phenylethylamine8WCA-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
20.00Single8WOGSuccinic acid8WOG-Succinate-Succinic acid-Gi1/β1/γ2
20.00Single8WWKMCH8WWK-MCH1-MCH-Gi1/β1/γ2
20.00Single8XIOL7975918XIO-SST1-L797591-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.00Single8XVIEndothelin-18XVI-ETA-Endothelin-1-chim(Gs-CtGq)/β1/γ2
20.00Single8Y0HVUF114188Y0H-CXCR3-VUF11418
20.00Single8Y0NVUF114188Y0N-CXCR3-VUF11418-Go/β1/γ2
20.00Single8YKXMaleic acid8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Single8ZWGJR14a8ZWG-C3aB-JR14a-Gi1/β1/γ2
20.00Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
20.00Single9DYEBuspirone9DYE-5-HT1A-Buspirone-Go/β1/γ2
20.00Single9EAILosartan9EAI-AT1-Losartan-Nanobody AT209
20.00Single9EEAAdenosine9EEA-A2A-Adenosine-Gs/β1/γ2
20.00Single9GE3Lysophosphatidylinositol9GE3-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
20.00Single9K6LSA09K6L-TAS2R16-SA0-Gi2/β1/γ2
20.00Single9KPESA09KPE-TAS2R16-SA0-Gi1/β1/γ2
20.00Single9M54Neuropeptide VF9M54-NPFF2-Neuropeptide VF-Gi1/β1/γ2
20.00Consensusccr_on_gpOrthosteric Ligandccr6_on_gp ccr8_on_gp ccr2_on_gp ccr1_on_gp ccr5_on_gp
20.00Consensuschemokine_offOrthosteric Ligandccr_off cxcr_off
20.00Consensuschemokine_on_gpOrthosteric Ligandccr_on_gp cxcr_on_gp
20.00Consensuscxcr_offOrthosteric Ligandcxcr3_off cxcr4_off
20.00Consensusgi_chemokineOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2 8HNK-CXCR3-CXCL11-Gi1/β1/γ2 8K3Z-CXCR4-CXCL12-Gi1/β1/γ1 8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2 6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2 8KFX-CCR8-LMD-009-Gi1/β1/γ2 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2 8HNL-CXCR3-PS372424-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 8U1U-CCR8-CCL1-Gi1/β1/γ2 7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2 7XA3-CCR2-CCL2-Gi1/β1/γ2
20.00Consensusgi_succinateOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Consensusgs_peptideOrthosteric Ligandgs_cck gs_melanocortin gs_vasop-oxy
20.00Consensusmc1_onOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.00Consensusmc1_on_gpOrthosteric Ligand7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2 7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2 7F4I-MC1-SHU9119-chim(NtGi1-Gs)/β1/γ2
20.00Consensusnk1_onOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensusnk1_on_gpOrthosteric Ligand7P00-NK1-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
20.00Consensuspeptide_offOrthosteric Ligandcck_off angiotensin_off bombesin_off endothelin_off ghrelin_off npy_off opioid_off orexin_off somatostatin_off tachykinin_off vasop-oxy_off neurotensin_off
20.00Consensussst5_on_gpOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
20.00Consensussuccinate_onOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
20.00Consensussuccinate_on_gpOrthosteric Ligand8YKW-Succinate-Succinic acid-Gi1/β1/γ1 8YKX-Succinate-Maleic acid-Gi1/β1/γ1
19.51Single5UIW5P7-CCL55UIW-CCR5-5P7-CCL5
19.51Single7F8VGastrin-177F8V-CCKB-Gastrin-17-Gi2/β1/γ2
19.51Single7SK4CXCL12_LRHQ7SK4-ACKR3-CXCL12_LRHQ
19.51Single8H0PNMB308H0P-BB1-NMB30-chim(NtGi1-Gs-CtGq)/β1/γ2
19.51Consensusccr5_offOrthosteric Ligand5UIW-CCR5-5P7-CCL5
19.51Consensusccr5_onOrthosteric Ligand7O7F-CCR5-6P4-CCL5-Gi1/β1/γ1 7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
19.51Consensusccr_offOrthosteric Ligandccr2_off ccr5_off
19.51Consensuscrf2_on_gpOrthosteric Ligand7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
19.44Single6C1QPMX536C1Q-C5a1-PMX53-NDT9513727
19.44Single6OMMWKYMVX6OMM-FPR2-ALX-WKYMVX-Gi1/β1/γ2
19.44Single6PT3DPI-2876PT3-δ-DPI-287
19.44Single7AUESetmelanotide7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2
19.44Single7F9ZGHRP-67F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Single7RKNFractalkine7RKN-US28-Fractalkine-Gi1/β1/γ2
19.44Single7RMGSubstance-P7RMG-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
19.44Single7RMHSubstance-P7RMH-NK1-Substance-P-Gs/β1/γ2
19.44Single7X8SWB4-247X8S-GLP-1-WB4-24-Gs/β1/γ2
19.44Single7Y1FDynorphin7Y1F-κ-Dynorphin-Gi1/β1/γ2
19.44Single8JBFSenktide8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Single9CGKC5-Quino9CGK-δ-C5-Quino-Gi1/β1/γ2
19.44Single9IPYJR14a9IPY-C3aB-JR14a
19.44Single9IZASCH9002719IZA-HCA2-SCH900271-Gi1/β1/γ2
19.44Consensuscxcr4_offOrthosteric Ligand4RWS-CXCR4-vMIP-II 3OE0-CXCR4-CVX15 3OE6-CXCR4-IT1t
19.44Consensuscxcr_on_gpOrthosteric Ligandcxcr3_on_gp cxcr4_on_gp cxcr1_on_gp cxcr2_on_gp
19.44Consensusox2_onOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.44Consensusox2_on_gpOrthosteric Ligand7L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2 7SQO-OX2-TAK-925-Gi1/β1/γ2 7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single2YDOAdenosine2YDO-A2A-Adenosine
19.35Single3UZC4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol3UZC-A2A-4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol
19.35Single3V2YPubChem 518926453V2Y-S1P1-PubChem 51892645
19.35Single4LDOL-Epinephrine4LDO-β2-L-Epinephrine
19.35Single4ZUDOlmesartan4ZUD-AT1-Olmesartan
19.35Single5IU7Q274563465IU7-A2A-Q27456346-Na
19.35Single5JTBZM-2413855JTB-A2A-ZM-241385
19.35Single5K2BZM-2413855K2B-A2A-ZM-241385-Na
19.35Single5TE3Octyl-Beta-D-Glucopyranoside5TE3-Rhodopsin-Octyl-β-D-Glucopyranoside
19.35Single6A94Zotepine6A94-5-HT2A-Zotepine
19.35Single6AQFZM-2413856AQF-A2A-ZM-241385
19.35Single6KUXRS-799486KUX-α2a-RS-79948
19.35Single6ME42-Iodomelatonin6ME4-MT1-2-Iodomelatonin
19.35Single6PS0S-Carazolol6PS0-β2-S-Carazolol
19.35Single6PS4ICI118-5516PS4-β2-ICI118-551
19.35Single6PS5S-Propranolol6PS5-β2-S-Propranolol
19.35Single6TOSGSK10598656TOS-OX1-GSK1059865-Na
19.35Single6TPGEMPA6TPG-OX2-EMPA
19.35Single6TPNHTL66416TPN-OX2-HTL6641
19.35Single6WJCAtropine6WJC-M1-Atropine-Muscarinic toxin 7
19.35Single6ZDRHMS1413f126ZDR-A2A-HMS1413f12-Na
19.35Single7CKWFenoldopam7CKW-D1-Fenoldopam-Gs/β1/γ2
19.35Single7DHISalbutamol7DHI-β2-Salbutamol-Gs/β1/γ2
19.35Single7EJ8Brimonidine7EJ8-α2a-Brimonidine-Go/β1/γ2
19.35Single7SR8TAK-9257SR8-OX2-TAK-925-chim(NtGi1L-Gs-CtGq)/β1/γ2
19.35Single8GE1Constrained Epinephrine8GE1-β2-Constrained Epinephrine-Gs/β1/γ2
19.35Single8GE4Constrained Epinephrine8GE4-β2-Constrained Epinephrine-Gs/β1/γ2
19.35Single8GE6Constrained Epinephrine8GE6-β2-Constrained Epinephrine-Gs/β1/γ2
19.35Single8GE7Constrained Epinephrine8GE7-β2-Constrained Epinephrine-Gs/β1/γ2
19.35Single8GE8Constrained Epinephrine8GE8-β2-Constrained Epinephrine-Gs/β1/γ2
19.35Single8GEAConstrained Epinephrine8GEA-β2-Constrained Epinephrine-Gs/β1/γ2
19.35Single8GEFConstrained Epinephrine8GEF-β2-Constrained Epinephrine-Gs/β1/γ2
19.35Single8GG7Constrained Epinephrine8GG7-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.35Single8GG8Constrained Epinephrine8GG8-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.35Single8GGLConstrained Epinephrine8GGL-β2-Constrained Epinephrine
19.35Single8GGMConstrained Epinephrine8GGM-β2-Constrained Epinephrine
19.35Single8GGPConstrained Epinephrine8GGP-β2-Constrained Epinephrine
19.35Single8GGQConstrained Epinephrine8GGQ-β2-Constrained Epinephrine
19.35Single8GGVConstrained Epinephrine8GGV-β2-Constrained Epinephrine
19.35Single8GGXConstrained Epinephrine8GGX-β2-Constrained Epinephrine
19.35Single8IY9Niacin8IY9-HCA2-Niacin-Go/β1/γ2
19.35Single8JIMMMF8JIM-HCA2-MMF-Gi1/β1/γ2
19.35Single8JLKUlotaront8JLK-TA1-Ulotaront-chim(NtGi1-Gs)/β1/γ2
19.35Single8JLNT1AM8JLN-TA1-T1AM-Gs/β1/γ2
19.35Single8JSPUlotaront8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2
19.35Single8K5CAcipimox8K5C-HCA2-Acipimox
19.35Single8PM2DMCH8PM2-TA7-DMCH-Gs/β1/γ2
19.35Single8RQQZM-2413858RQQ-A2A-ZM-241385-Na
19.35Single8THKA616038THK-Alpha1A-A61603-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single8THLEpinephrine8THL-Alpha1A-Epinephrine-chim(NtGi2L-Gs-CtGq)/β1/γ2
19.35Single8UHBRO52563908UHB-TA1-RO5256390-Gs/β1/γ2
19.35Single8UNLConstrained Epinephrine8UNL-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.35Single8UNOConstrained Epinephrine8UNO-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.35Single8UO0Constrained Epinephrine8UO0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
19.35Single8UO1Constrained Epinephrine8UO1-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
19.35Single8Y01Retinal8Y01-Opsin1MW-Retinal-Gi1/β1/γ2
19.35Single8YKVPubChem 1375531688YKV-Succinate-PubChem 137553168-Gi1/β1/γ2
19.35Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
19.35Single9EPQ11,20-Ethanoretinal9EPQ-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
19.35Single9JKQMETH9JKQ-TA1-METH-Gs/β1/γ2
19.35Single9M2FNeuropeptide FF9M2F-NPFF1-Neuropeptide FF-Gi1/β1/γ2
19.35Consensus5ht_on_gpOrthosteric Ligand5ht1_on_gp 5ht2_on_gp 5ht4_on_gp 5ht5_on_gp 5ht6_on_gp 5ht7_on_gp
19.35Consensusa2_offOrthosteric Liganda2a_off
19.35Consensusa2a_offOrthosteric Ligand3RFM-A2A-Caffeine 8C9W-A2A-Etrumadenant 3UZA-A2A-GTPL9236 8GNG-A2A-Istradefylline 8CU6-A2A-LJ-4517 7PX4-A2A-PSB-2113 7PYR-A2A-PSB-2115 8DU3-A2A-PubChem 105526064 8JWY-A2A-2-118 8PWN-A2A-Theophylline 5IU4-A2A-ZM-241385-Na 5OLZ-A2A-PubChem 135566609-Na 6GT3-A2A-Imaradenant-Na 5OLV-A2A-LUAA41063-Na 5N2R-A2A-PSB-36-Na 5IU7-A2A-Q27456346-Na 5OLH-A2A-Vipadenant-Na 5OLO-A2A-Tozadenant-Na 6ZDR-A2A-HMS1413f12-Na 8GNE-A2A-KW-6356-Na 8JWZ-A2A-AB928-Na 5IU8-A2A-Q27456347-Na 5IUB-A2A-Q27456344-Na 6ZDV-A2A-Chromone 5d-Na 5IUA-A2A-Q27456348-Na 8A2P-A2A-LUAA47070-Na
19.35Consensusalpha1_onOrthosteric Ligandalpha1a_on
19.35Consensusalpha1_on_gpOrthosteric Ligandalpha1a_on_gp
19.35Consensusalpha1a_onOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
19.35Consensusalpha1a_on_gpOrthosteric Ligand7EJ0-α2a-L-Norepinephrine-Go/β1/γ2 7EJ8-α2a-Brimonidine-Go/β1/γ2 7EJA-α2a-Dexmedetomidine-Go/β1/γ2 7EJK-α2a-Oxymetazoline-Go/β1/γ2 7W6P-α2a-N-pyridin-4-ylisoquinolin-4-amine-Go/β1/γ2 7W7E-α2a-PubChem 164946676-Go/β1/γ2
19.35Consensusat1_offOrthosteric Ligand4YAY-AT1-ZD-7155 4ZUD-AT1-Olmesartan
19.35Consensuscb1_offOrthosteric Ligand5U09-CB1-Taranabant 5TGZ-CB1-AM6538
19.35Consensushca_onOrthosteric Ligandhca2_on
19.05Single7EIBDes-Arg10-Kallidin7EIB-BK1-Des-Arg10-Kallidin-chim(NtGi1-Gs-CtGq)/β1/γ2
19.05Single7XATSomatostatin-147XAT-SST2-Somatostatin-14-Gi1/β1/γ2
19.05Single7YOONeuropeptide-Y7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
19.05Single8WWLMCH8WWL-MCH1-MCH-Gi1/β1/γ2
19.05Consensusnpy2_onOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
19.05Consensusnpy2_on_gpOrthosteric Ligand7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
18.92Single4AMJS-Carvedilol4AMJ-β1-S-Carvedilol
18.92Single4IARErgotamine4IAR-5-HT1B-Ergotamine
18.92Single4IB4Ergotamine4IB4-5-HT2B-Ergotamine
18.92Single5UNFPubChem 157800525UNF-AT2-PubChem 15780052
18.92Single6WIVPubChem 52923113; PubChem 529246456WIV-GABAB1, GABAB2-PubChem 52923113; PubChem 52924645
18.92Single7WKDTRH7WKD-TRH-TRH-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Single8DCRDobutamine8DCR-β1-Dobutamine-Gs/β1/γ2
18.92Single8FYLVilazodone8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
18.92Single8K3ZCXCL128K3Z-CXCR4-CXCL12-Gi1/β1/γ1
18.92Single9BKJCholecystokinin-89BKJ-CCKA-Cholecystokinin-8-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Single9BUYLM1899BUY-β2-LM189-Gi1/β1/γ2
18.92Single9HB3Mambaquaretin-19HB3-V2-Mambaquaretin-1
18.92Consensusnk3_onOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
18.92Consensusnk3_on_gpOrthosteric Ligand8JBF-NK3-Senktide-chim(NtGi1-Gs-CtGq)/β1/γ2
18.75Single2VT4Cyanopindolol2VT4-β1-Cyanopindolol
18.75Single2Y01Dobutamine2Y01-β1-Dobutamine
18.75Single2Y02Carmoterol2Y02-β1-Carmoterol
18.75Single2YCYCyanopindolol2YCY-β1-Cyanopindolol
18.75Single3EMLZM-2413853EML-A2A-ZM-241385
18.75Single3NYAS-Alprenolol3NYA-β2-S-Alprenolol
18.75Single4EA3PubChem 102965614EA3-NOP-PubChem 10296561
18.75Single4EIYZM-2413854EIY-A2A-ZM-241385-Na
18.75Single4J4QOctyl Beta-D-Glucopyranoside4J4Q-Rhodopsin-Octyl β-D-Glucopyranoside-Gt(CT)
18.75Single4MQSIperoxo4MQS-M2-Iperoxo
18.75Single4U14Tiotropium4U14-M3-Tiotropium
18.75Single4YAYZD-71554YAY-AT1-ZD-7155
18.75Single5DSGTiotropium5DSG-M4-Tiotropium
18.75Single5IU8Q274563475IU8-A2A-Q27456347-Na
18.75Single5K2AZM-2413855K2A-A2A-ZM-241385-Na
18.75Single5OLGZM-2413855OLG-A2A-ZM-241385-Na
18.75Single5VRAZM-2413855VRA-A2A-ZM-241385-Na
18.75Single5YC8N-Methyl-Scopolamine5YC8-M2-N-Methyl-Scopolamine
18.75Single5ZK8N-Methyl-Scopolamine5ZK8-M2-N-Methyl-Scopolamine
18.75Single5ZKCN-Methyl-Scopolamine5ZKC-M2-N-Methyl-Scopolamine
18.75Single5ZKPForopafant (SR27417)5ZKP-PAF-Foropafant (SR27417)
18.75Single6FKDPubChem 1373491836FKD-Rhodopsin-PubChem 137349183
18.75Single6H7MSalbutamol6H7M-β1-Salbutamol
18.75Single6IIVDaltroban6IIV-TXA2-Daltroban
18.75Single6PRZS-Alprenolol6PRZ-β2-S-Alprenolol
18.75Single6PS1Timolol6PS1-β2-Timolol
18.75Single6S0LZM-2413856S0L-A2A-ZM-241385
18.75Single6TOTLemborexant6TOT-OX1-Lemborexant
18.75Single7BTSL-Epinephrine7BTS-β1-L-Epinephrine
18.75Single7BU6L-Norepinephrine7BU6-β1-L-Norepinephrine
18.75Single7E32Serotonin7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.75Single7F83PF-051904577F83-Ghrelin-PF-05190457
18.75Single7JOZVFP7JOZ-D1-VFP-Gs/β1/γ2
18.75Single7JVQApomorphine7JVQ-D1-Apomorphine-Gs/β1/γ2
18.75Single7LCIDanuglipron7LCI-GLP-1-Danuglipron-Gs/β1/γ2
18.75Single7LCKDanuglipron7LCK-GLP-1-Danuglipron
18.75Single7LJCSKF-812977LJC-D1-SKF-81297-Mevidalen-Gs/β1/γ2
18.75Single7PYRPSB-21157PYR-A2A-PSB-2115
18.75Single7S0GIsoprenaline7S0G-β1-Isoprenaline-chim(Gi1-CtGs)/β1/γ2
18.75Single7S15PubChem 1346112237S15-GLP-1-PubChem 134611223
18.75Single7TRPIperoxo7TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
18.75Single7UL4Alvimopan7UL4-μ-Alvimopan
18.75Single7UM55-CT7UM5-5-HT5A-5-CT-chim(NtGi1-Go)/β1/γ2
18.75Single7UM6Lisuride7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
18.75Single7VGZRemalteon7VGZ-MT1-Remalteon-Gi1/β1/γ2
18.75Single7VH0Ramelteon7VH0-MT2-Ramelteon-Gi1/β1/γ1
18.75Single7VIFS-FTY720-P7VIF-S1P1-S-FTY720-P-Gi1/β1/γ2
18.75Single7XTC5-CT7XTC-5-HT7-5-CT-Gs/β1/γ2
18.75Single7YACPaltusotine7YAC-SST2-Paltusotine-Gi1/β1/γ2
18.75Single8CICEtrumadenant8CIC-A2A-Etrumadenant-Na
18.75Single8DZSGR89,6968DZS-κ-GR89,696-chim(NtGi2-Gz)/β1/γ2
18.75Single8FY85-MeO-DMT8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1
18.75Single8GE3Constrained Epinephrine8GE3-β2-Constrained Epinephrine-Gs/β1/γ2
18.75Single8GECConstrained Epinephrine8GEC-β2-Constrained Epinephrine-Gs/β1/γ2
18.75Single8GEEConstrained Epinephrine8GEE-β2-Constrained Epinephrine-Gs/β1/γ2
18.75Single8GEHConstrained Epinephrine8GEH-β2-Constrained Epinephrine-Gs/β1/γ2
18.75Single8GFVConstrained Epinephrine8GFV-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8GFWConstrained Epinephrine8GFW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8GFXConstrained Epinephrine8GFX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8GFZConstrained Epinephrine8GFZ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8GG0Constrained Epinephrine8GG0-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8GG1Constrained Epinephrine8GG1-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8GG3Constrained Epinephrine8GG3-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8GG4Constrained Epinephrine8GG4-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8GG6Constrained Epinephrine8GG6-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8GG9Constrained Epinephrine8GG9-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8GGIConstrained Epinephrine8GGI-β2-Constrained Epinephrine
18.75Single8GGJConstrained Epinephrine8GGJ-β2-Constrained Epinephrine
18.75Single8GGKConstrained Epinephrine8GGK-β2-Constrained Epinephrine
18.75Single8GGNConstrained Epinephrine8GGN-β2-Constrained Epinephrine
18.75Single8GGOConstrained Epinephrine8GGO-β2-Constrained Epinephrine
18.75Single8GGUConstrained Epinephrine8GGU-β2-Constrained Epinephrine
18.75Single8JHNMMF8JHN-HCA2-MMF-Go/β1/γ2
18.75Single8JIINiacin8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
18.75Single8JJOAlprenolol8JJO-β2-Alprenolol
18.75Single8JLJT1AM8JLJ-TA1-T1AM-chim(NtGi1-Gs)/β1/γ2
18.75Single8JLZST19368JLZ-5-HT6-ST1936-Gs/β1/γ2
18.75Single8K5DGSK2560738K5D-HCA2-GSK256073
18.75Single8PJKST1718PJK-5-HT1A-ST171-Gi1/β1/γ1
18.75Single8UGYMianserin8UGY-5-HT1E-Mianserin-Gi1/β1/γ1
18.75Single8UNQConstrained Epinephrine8UNQ-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8UNRConstrained Epinephrine8UNR-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8UNUConstrained Epinephrine8UNU-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8UNYConstrained Epinephrine8UNY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.75Single8X63Mepyramine8X63-H1-Mepyramine
18.75Single8X64Desloratadine8X64-H1-Desloratadine
18.75Single8XVKAmbrisentan8XVK-ETA-Ambrisentan
18.75Single8YN8Proxyfan8YN8-H3-Proxyfan-Go/β1/γ2
18.75Single8ZQEGPR15L(C11)8ZQE-GPR15-GPR15L(C11)-Gi1/β1/γ1
18.75Single9CBMDexmedetomidine9CBM-α2a-Dexmedetomidine-Gi1/β1/γ2
18.75Single9D61JDTic9D61-κ-JDTic-Gi1/β1/γ2
18.75Single9EPP11,20-Ethanoretinal9EPP-Rhodopsin-11,20-Ethanoretinal-chim(Gi1-CtGq)/β1/γ2
18.75Single9IVGGLP-1 (Truncated)9IVG-GLP-1-GLP-1 (Truncated)-chim(NtGi1-Gs)/β1/γ2
18.75Single9IZCMK19039IZC-HCA2-MK1903-Gi1/β1/γ2
18.75Single9JEAAtropine9JEA-M1-Atropine
18.75Single9PLNN-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLN-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine
18.75Single9PLON-(5-methylnaphthalen-1-yl)pyridin-4-amine9PLO-α2a-N-(5-methylnaphthalen-1-yl)pyridin-4-amine-Go/β1/γ2
18.75Consensus5ht1d_onOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.75Consensus5ht1d_on_gpOrthosteric Ligand7E32-5-HT1D-Serotonin-Gi1/β1/γ2
18.75Consensus5ht5_onOrthosteric Ligand5ht5a_on
18.75Consensus5ht5a_onOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
18.75Consensus5ht6_onOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
18.75Consensus5ht6_on_gpOrthosteric Ligand7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2
18.75Consensus5ht7_onOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
18.75Consensus5ht7_on_gpOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2
18.75Consensusadenosine_on_gpOrthosteric Liganda1_on_gp a2_on_gp a3_on_gp
18.75Consensusadrenergic_onOrthosteric Ligandalpha_on beta_on
18.75Consensusalpha_onOrthosteric Ligandalpha1_on alpha2_on
18.75Consensusdopamine_onOrthosteric Ligandd2_on d1_on d3_on d4_on d5_on
18.75Consensusdopamine_on_gpOrthosteric Ligandd2_on_gp d1_on_gp d3_on_gp d4_on_gp d5_on_gp
18.75Consensushistamine_offOrthosteric Ligandh1_off
18.75Consensusm4_offOrthosteric Ligand5DSG-M4-Tiotropium
18.75Consensusnucleotide_offonOrthosteric Ligandnucleotide_off nucleotide_on
18.75Consensusnucleotide_offon_gpOrthosteric Ligandnucleotide_on_gp nucleotide_off
18.60Single8Y52BA18Y52-BB3-BA1-chim(NtGi1-Gs-CtGq)/β1/γ2
18.42Single5XJM(Sar1,Ile8)-Angiotensin II5XJM-AT2-(Sar1,Ile8)-Angiotensin II
18.42Single7C6A(Sar1,Ile8)-Angiotensin II7C6A-AT2-(Sar1,Ile8)-Angiotensin II
18.42Single7PIVSetmelanotide7PIV-MC4-Setmelanotide-Gs/β1/γ2
18.42Single7XNACYN1548067XNA-SST2-CYN154806
18.42Single8XYDPlatelet Activating Factor8XYD-PAF-Platelet Activating Factor-Gi1/β1/γ2
18.42Single9KFIRelaxin-39KFI-RXFP3-Relaxin-3-Gi2/β1/γ2
18.42Consensusccr8_on_gpOrthosteric Ligand8KFX-CCR8-LMD-009-Gi1/β1/γ2 8KFY-CCR8-ZK-756326-Gi1/β1/γ2 8U1U-CCR8-CCL1-Gi1/β1/γ2
18.42Consensusghrelin_onOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
18.42Consensusghrelin_on_gpOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7F9Z-Ghrelin-GHRP-6-chim(NtGi1-Gs-CtGq)/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
18.42Consensusgi_cckOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
18.42Consensusgi_ghrelinOrthosteric Ligand7NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2 7NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
18.42Consensusmc4_on_gpOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
18.42Consensussst2_offOrthosteric Ligand7XNA-SST2-CYN154806
18.18Single2Y00Dobutamine2Y00-β1-Dobutamine
18.18Single4WW3All-trans-Retinal4WW3-Rhodopsin-All-trans-Retinal
18.18Single4ZJ8Suvorexant4ZJ8-OX1-Suvorexant
18.18Single5IUAQ274563485IUA-A2A-Q27456348-Na
18.18Single5N2RPSB-365N2R-A2A-PSB-36-Na
18.18Single5N2SPSB365N2S-A1-PSB36
18.18Single5WIUNemonapride5WIU-D4-Nemonapride
18.18Single5WIVNemonapride5WIV-D4-Nemonapride-Na
18.18Single5WQCEMPA5WQC-OX2-EMPA
18.18Single6D26Fevipiprant6D26-DP2-Fevipiprant
18.18Single6E67BI1671076E67-β2-BI167107-Gs(CT)
18.18Single6HLPNetupitant6HLP-NK1-Netupitant
18.18Single6KUWPubChem 572132346KUW-α2c-PubChem 57213234
18.18Single6LPLZM-2413856LPL-A2A-ZM-241385-Na
18.18Single6ME62-Phenylmelatonin6ME6-MT2-2-Phenylmelatonin
18.18Single6ME72-Phenylmelatonin6ME7-MT2-2-Phenylmelatonin
18.18Single6PS3S-Carvedilol6PS3-β2-S-Carvedilol
18.18Single6S0QZM-2413856S0Q-A2A-ZM-241385
18.18Single6TO7Suvorexant6TO7-OX1-Suvorexant-Na
18.18Single6TP6Filorexant6TP6-OX1-Filorexant
18.18Single6WQAZM-2413856WQA-A2A-ZM-241385-Na
18.18Single7BB7AVP7BB7-V2-AVP-Gs/β1/γ2
18.18Single7BVQS-Carazolol7BVQ-β1-S-Carazolol
18.18Single7C61Ergotamine7C61-5-HT1B-Ergotamine
18.18Single7CFNINT-7777CFN-GPBA-INT-777-Gs/β1/γ2
18.18Single7E9GJNJ-404118137E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
18.18Single7RM5ZM-2413857RM5-A2A-ZM-241385-Na
18.18Single7S0FIsoprenaline7S0F-β1-Isoprenaline-Gi1/β1/γ2
18.18Single7SINNPS-21437SIN-CaS-NPS-2143
18.18Single7SINNPS-21437SIN-CaS-NPS-2143
18.18Single7VUHJNJ-635330547VUH-GPR139-JNJ-63533054-chim(Gs-CtGq)/β1/γ2
18.18Single7X1TTaltirelin7X1T-TRH-Taltirelin-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Single7XK9Constrained Isoproterenol7XK9-β2-Constrained Isoproterenol-Na
18.18Single8C9WEtrumadenant8C9W-A2A-Etrumadenant
18.18Single8FYNZM-2413858FYN-A2A-ZM-241385-Na
18.18Single8GFYConstrained Epinephrine8GFY-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GG2Constrained Epinephrine8GG2-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
18.18Single8GNEKW-63568GNE-A2A-KW-6356-Na
18.18Single8I7WGSK2560738I7W-HCA2-GSK256073-Gi1/β1/γ2
18.18Single8ID4Linoleic acid8ID4-FFA4-Linoleic acid-Gi1/β1/γ2
18.18Single8KFXLMD-0098KFX-CCR8-LMD-009-Gi1/β1/γ2
18.18Single8S4DCMF-0198S4D-Apelin-CMF-019
18.18Single8TH4Losartan8TH4-AT1-Losartan-AT118-L Nanobody
18.18Single8U1UCCL18U1U-CCR8-CCL1-Gi1/β1/γ2
18.18Single8WGBVU01550418WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
18.18Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
18.18Single8XQPCholesterol8XQP-TAS2R14-Cholesterol-Aristolochic acid A-Gt3/β1/γ1
18.18Single8YNSSNAP-948478YNS-MCH1-SNAP-94847
18.18Single8ZJETAK-4488ZJE-Kiss1-TAK-448-chim(NtGi1-Gq)/β1/γ1
18.18Single9ARYSerotonin9ARY-5-HT2A-Serotonin-chim(NtGi1-Gs-CtGq)/β1/γ2
18.18Single9ARZ2-bromo-LSD9ARZ-5-HT2A-2-bromo-LSD
18.18Single9B9ZA1AKO9B9Z-CB1-A1AKO
18.18Single9EHSLUF76029EHS-A3A-LUF7602
18.18Single9F33FOB02-04A9F33-D3-FOB02-04A-Go/β1/γ2
18.18Single9F34FOB02-04A9F34-D3-FOB02-04A-Go/β1/γ2
18.18Single9IYBProstaglandin9IYB-DP2-Prostaglandin-A1D5Q-Gi1/β1/γ2
18.18Consensus5ht1_onOrthosteric Ligand5ht1a_on 5ht1d_on 5ht1e_on 5ht1f_on
18.18Consensus5ht1_on_gpOrthosteric Ligand5ht1a_on_gp 5ht1d_on_gp 5ht1e_on_gp 5ht1f_on_gp
18.18Consensus5ht1e_on_gpOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
18.18Consensus5ht2_offOrthosteric Ligand5ht2a_off 5ht2b_off 5ht2c_off
18.18Consensus5ht5_on_gpOrthosteric Ligand5ht5a_on_gp
18.18Consensus5ht5a_on_gpOrthosteric Ligand7X5H-5-HT5A-5-CT-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
18.18Consensusa1_offOrthosteric Ligand5UEN-A1-DU172 5N2S-A1-PSB36
18.18Consensusadrenergic_offOrthosteric Ligandalpha_off beta_off
18.18Consensusadrenergic_on_gpOrthosteric Ligandalpha_on_gp beta_on_gp
18.18Consensusalpha2c_offOrthosteric Ligand6KUW-α2c-PubChem 57213234
18.18Consensusalpha_offOrthosteric Ligandalpha1_off alpha2_off
18.18Consensusalpha_on_gpOrthosteric Ligandalpha1_on_gp alpha2_on_gp
18.18Consensusblt1_offOrthosteric Ligand5X33-BLT1-BIIL260 7K15-BLT1-MKD046-Na
18.18Consensusblt_offOrthosteric Ligandblt1_off
18.18Consensusdp2_offOrthosteric Ligand6D26-DP2-Fevipiprant
18.18Consensusdp_offOrthosteric Liganddp2_off
18.18Consensusgi_npyOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1 7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2 7YOO-Y2-Neuropeptide-Y-Gi1/β1/γ2
18.18Consensusgq_muscarinicOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
18.18Consensusm1_onOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
18.18Consensusm3_onOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Consensusm3_on_gpOrthosteric Ligand8E9Z-M3-Iperoxo-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9W-M3-2-Deoxycytidine-chim(NtGi2L-Gs-CtGq)/β1/γ2 8E9Y-M3-Clozapine-N-oxide-chim(NtGi2L-Gs-CtGq)/β1/γ2
18.18Consensusnpy_onOrthosteric Ligandnpy1_on npy2_on npy4_on
18.18Consensusnpy_on_gpOrthosteric Ligandnpy1_on_gp npy2_on_gp npy4_on_gp
17.95Single7RYCOxytocin7RYC-OT-Oxytocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.95Single8W8YGamma-MSH8W8Y-MC3-γ-MSH-Ca-Gs/β1/γ2
17.95Single8WKZSBL-MC-318WKZ-MC4-SBL-MC-31
17.95Single8XGUTAK4488XGU-Kiss1-TAK448-Gi1/β1/γ2
17.95Single8XZGApelin-138XZG-Apelin-Apelin-13-Gi1/β1/γ2
17.95Single9M1OMorphine-Modulating Neuropeptide B9M1O-NPFF2-Morphine-Modulating Neuropeptide B-Gi1/β1/γ2
17.95Consensuscxcr4_on_gpOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
17.95Consensusgi_somatostatinOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7XMS-SST4-Somatostatin-14-Gi1/β1/γ2 8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 7XMT-SST4-J-2156-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
17.95Consensussomatostatin_onOrthosteric Ligandsst2_on sst4_on sst5_on
17.95Consensussomatostatin_on_gpOrthosteric Ligandsst2_on_gp sst4_on_gp sst5_on_gp
17.78Single7SK6CXCL12_LRHQ7SK6-ACKR3-CXCL12_LRHQ
17.65Single3PDSHydroxybenzylisoproterenol3PDS-β2-Hydroxybenzylisoproterenol
17.65Single6J20Aprepitant6J20-NK1-Aprepitant
17.65Single6OIJIperoxo6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.65Single6OS1TRV0266OS1-AT1-TRV026
17.65Single7B6WCyclazosin7B6W-α1b-Cyclazosin
17.65Single7EW4CYM55417EW4-S1P3-CYM5541-Gi1/β1/γ2
17.65Single7F58THIQ7F58-MC4-THIQ-Gs/β1/γ2
17.65Single7M8W15r-Methyl-Prostaglandin D27M8W-DP2-15r-Methyl-Prostaglandin D2-Na
17.65Single7PX4PSB-21137PX4-A2A-PSB-2113
17.65Single7TUYGSK682753A7TUY-GPR183-GSK682753A
17.65Single7XTQR3997XTQ-GPBA-R399-Gs/β1/γ2
17.65Single8I2GCompound 7163408I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
17.65Single8I9LC3a anaphylatoxin8I9L-C3aB-C3a anaphylatoxin-Go/β1/γ2
17.65Single8ID6Oleic acid8ID6-FFA4-Oleic acid-Gi1/β1/γ2
17.65Single8IYHMK68928IYH-HCA2-MK6892-Go/β1/γ2
17.65Single8JLPRalmitaront8JLP-TA1-Ralmitaront-Gs/β1/γ2
17.65Single8JSRAnamorelin8JSR-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single8JT6(R)-IHCH-71798JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2
17.65Single8JXVClozapine8JXV-H4-Clozapine-Gi1/β1/γ2
17.65Single8JXWVUF68848JXW-H4-VUF6884-Gi1/β1/γ2
17.65Single8JZPC5A anaphylatoxin8JZP-C5a1-C5A anaphylatoxin-Go/β1/γ2
17.65Single8WJXADP8WJX-P2Y1-ADP-chim(Gs-CtGq)/β1/γ2
17.65Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
17.65Single8X16Piclidenoson8X16-A3A-Piclidenoson-Gi1/β1/γ2
17.65Single8X79MRE-2698X79-I2-MRE-269-Gs/β1/γ2
17.65Single8YH6Namodenoson8YH6-A3A-Namodenoson-Gi1/β1/γ2
17.65Single8ZR5Firuglipel8ZR5-GPR119-Firuglipel-Gs/β1/γ2
17.65Single8ZW0PGD28ZW0-DP1-PGD2-Gs/β1/γ2
17.65Single8ZWFJR14a8ZWF-C3aB-JR14a
17.65Single9AS9RS130-1809AS9-5-HT2A-RS130-180
17.65Single9ASARS130-1809ASA-5-HT2A-RS130-180-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Single9IJDCarazolol9IJD-β3-Carazolol-chim(NtGi1-Gs)/β1/γ2
17.65Single9UY3Anamorelin9UY3-Ghrelin-Anamorelin-chim(NtGi1-Gs-CtGq)/β1/γ2
17.65Consensusbeta2_onOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
17.65Consensusbeta2_on_gpOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2
17.65Consensusgi_5htOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8W8B-5-HT1A-SEP-363856-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E32-5-HT1D-Serotonin-Gi1/β1/γ2 7XTA-5-HT4-Serotonin-Gi1/β1/γ2 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 7X5H-5-HT5A-5-CT-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 7EXD-5-HT1F-Lasmiditan-Gi1/β1/γ2 7UM6-5-HT5A-Lisuride-chim(NtGi1-Go)/β1/γ2
17.65Consensusgs_adrenergicOrthosteric Ligand7DHI-β2-Salbutamol-Gs/β1/γ2 7XJI-β3-Solabegron-Gs/β1/γ2 7JJO-β1-Isoprenaline-Gs/β1/γ2 6NI3-β2-BI167107-Gs/β1/γ2 8DCR-β1-Dobutamine-Gs/β1/γ2 7XJH-β3-Isoproterenol-Gs/β1/γ2 7DH5-β3-Mirabegron-Gs/β1/γ2
17.65Consensusm1_on_gpOrthosteric Ligand6OIJ-M1-Iperoxo-chim(NtGi1L-G11)/β1/γ2
17.65Consensustachykinin_offOrthosteric Ligandnk1_off
17.50Single7DW9AVP7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.50Single7F4HAfamelanotide7F4H-MC1-Afamelanotide-chim(NtGi1-Gs)/β1/γ2
17.50Single7KH0AVP7KH0-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.50Single7T10Somatostatin-147T10-SST2-Somatostatin-14-Gi3/β1/γ2
17.50Single7XK8Neuromedin-U-257XK8-NMUR2-Neuromedin-U-25-Gi1/β1/γ2
17.50Single8WSTPro-MCH8WST-MCH2-Pro-MCH-chim(NtGi1L-Gs-CtGq)/β1/γ2
17.50Single8X8LCortistatin8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2
17.50Consensusgs_vasop-oxyOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.50Consensustachykinin_onOrthosteric Ligandnk1_on nk2_on nk3_on
17.50Consensusv2_onOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.50Consensusv2_on_gpOrthosteric Ligand7DW9-V2-AVP-chim(NtGi1-Gs)/β1/γ2
17.50Consensusvasop-oxy_onOrthosteric Ligandv2_on
17.50Consensusvasop-oxy_on_gpOrthosteric Ligandv2_on_gp
17.24Single3OE6IT1t3OE6-CXCR4-IT1t
17.24Single5WKTOctyl-Beta-D-Glucopyranoside5WKT-Rhodopsin-Octyl-β-D-Glucopyranoside-Gt(CT)
17.24Single8GGFConstrained Epinephrine8GGF-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
17.24Single8GH1Constrained Epinephrine8GH1-β2-Constrained Epinephrine
17.24Single8J6QBeta-Hydroxybutyrate8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
17.24Single8POKHistamine8POK-H2-Histamine-Gs/β1/γ2
17.24Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
17.24Single8X9UMetenolone8X9U-ADGRD1-Metenolone-chim(NtGi1-Gs)/β1/γ2
17.24Single9IV15alpha-DHT9IV1-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
17.24Consensush2_on_gpOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
17.14Single4XEENeurotensin4XEE-NTS1-Neurotensin
17.14Single4XESNeurotensin4XES-NTS1-Neurotensin
17.14Single6AK3Dinoprostone IPGE26AK3-EP3-Dinoprostone IPGE2
17.14Single6CM4Risperidone6CM4-D2-Risperidone
17.14Single6DRYMethylergonovine6DRY-5-HT2B-Methylergonovine
17.14Single6IIURamatroban6IIU-TXA2-Ramatroban
17.14Single6VMSBromoergocryptine6VMS-D2-Bromoergocryptine-Gi1/β1/γ2
17.14Single6YVRNTS8-136YVR-NTS1-NTS8-13
17.14Single6ZG4HTL00099366ZG4-M1-HTL0009936
17.14Single7L1VPubChem 1554910097L1V-OX2-PubChem 155491009-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single7XMTJ-21567XMT-SST4-J-2156-Gi1/β1/γ2
17.14Single7XW5ML1097XW5-TSH-TSH-ML109-Gs/β1/γ2
17.14Single7XZ5Lysophosphatidylcholine7XZ5-GPR119-Lysophosphatidylcholine-Gs/β1/γ2
17.14Single7Y66BM2137Y66-C5a1-BM213-Gi1/β1/γ2
17.14Single7YMJTamsulosin7YMJ-Alpha1A-Tamsulosin
17.14Single8IQ6Latanoprost8IQ6-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single8IYWGSK2560738IYW-HCA2-GSK256073-Go/β1/γ2
17.14Single8J6DEP1418J6D-C3aB-EP141-Go/β1/γ2
17.14Single8JD3JNJ-404118138JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
17.14Single8JJPChemerin8JJP-CML2-Chemerin-Gi1/β1/γ2
17.14Single8JPCNeurotensin-(8-13)8JPC-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
17.14Single8JWY2-1188JWY-A2A-2-118
17.14Single8JWZAB9288JWZ-A2A-AB928-Na
17.14Single8T3QDocosa-4,7,10,13,16,19-Hexaenoic acid8T3Q-FFA4-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.14Single8W1VPubChem 1717162658W1V-β2-PubChem 171716265
17.14Single8XJNCloprosetnol8XJN-TXA2-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
17.14Single8XYIVUF106618XYI-CXCR3-VUF10661
17.14Single9GGGI-BOP9GGG-TXA2-I-BOP-chim(NtGi2L-Gs-CtGq)/β1/γ2
17.14Single9L3WRetinoic acid receptor responder protein 29L3W-CML1-Retinoic acid receptor responder protein 2-Gi1/β1/γ2
17.14Consensus5ht1a_onOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
17.14Consensus5ht1a_on_gpOrthosteric Ligand8FYT-5-HT1A-LSD-Gi1/β1/γ1 8FYX-5-HT1A-Buspirone-Gi1/β1/γ1 8JSP-5-HT1A-Ulotaront-Gi1/β1/γ2 8JT6-5-HT1A-(R)-IHCH-7179-Gi1/β1/γ2 7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2 7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2 8FY8-5-HT1A-5-MeO-DMT-Gi1/β1/γ1 8FYE-5-HT1A-4-F,5-MeO-PyrT-Gi1/β1/γ1 8FYL-5-HT1A-Vilazodone-Gi1/β1/γ1
17.14Consensusalpha1_offOrthosteric Ligandalpha1a_off
17.14Consensusalpha1a_offOrthosteric Ligand7YMJ-Alpha1A-Tamsulosin
17.14Consensusbeta_onOrthosteric Ligandbeta1_on beta2_on beta3_on
17.14Consensusbeta_on_gpOrthosteric Ligandbeta1_on_gp beta2_on_gp beta3_on_gp
17.14Consensuscxcr_onOrthosteric Ligandcxcr3_on cxcr4_on cxcr1_on cxcr2_on
17.14Consensusgi_muscarinicOrthosteric Ligand8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2 7TRS-M4-Acetylcholine-Gi1/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2
17.14Consensusm4_onOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
17.14Consensusm4_on_gpOrthosteric Ligand7TRS-M4-Acetylcholine-Gi1/β1/γ2 7V6A-M4-PubChem 9864275-Gi1/β1/γ2 8E9X-M4-2-Deoxycytidine-chim(NtGi1-Go)/β1/γ2 7TRK-M4-Iperoxo-Gi1/β1/γ2
17.14Consensusnk1_offOrthosteric Ligand6HLP-NK1-Netupitant 6HLO-NK1-Aprepitant 6HLL-NK1-CP99994 6E59-NK1-L-760735
17.14Consensusorexin_onOrthosteric Ligandox2_on
17.07Single7F6IKallidin7F6I-BK2-Kallidin-Gq/β1/γ2
17.07Single7F9YGhrelin-287F9Y-Ghrelin-Ghrelin-28-chim(NtGi1-Gs-CtGq)/β1/γ2
17.07Single7VL9CCL15(26-92)7VL9-CCR1-CCL15(26-92)-Gi1/β1/γ2
17.07Single7X9CPancreatic Hormone7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
17.07Single7XV3Lysophosphatidylserine7XV3-GPR174-Lysophosphatidylserine-chim(NtGi1-Gs)/β1/γ2
17.07Single8HNKCXCL118HNK-CXCR3-CXCL11-Gi1/β1/γ2
17.07Single8WWMMCH8WWM-MCH1-MCH-Gi1/β1/γ2
17.02Single7X9ANeuropeptide-Y7X9A-Y1-Neuropeptide-Y-Gi1/β1/γ2
16.67Single3AYMAll-trans-Retinal3AYM-Rhodopsin-All-trans-Retinal
16.67Single3PBLEticlopride3PBL-D3-Eticlopride
16.67Single4BUONeurotensin4BUO-NTS1-Neurotensin
16.67Single4NC3Ergotamine4NC3-5-HT2B-Ergotamine
16.67Single5TUDErgotamine5TUD-5-HT2B-Ergotamine
16.67Single6H7LDobutamine6H7L-β1-Dobutamine
16.67Single6IBLArformoterol6IBL-β1-Arformoterol
16.67Single6K1QIRL25006K1Q-ETB-IRL2500
16.67Single6LI0C176LI0-GPR52-C17
16.67Single6TKOArformoterol6TKO-β1-Arformoterol-Arrestin2
16.67Single7D76Beclomethasone7D76-ADGRG3-Beclomethasone-Go/β1/γ2
16.67Single7SK3CXCL127SK3-ACKR3-CXCL12
16.67Single7W3ZGastrin Releasing Peptide7W3Z-BB2-Gastrin Releasing Peptide-chim(NtGi1L-Gq)/β1/γ2
16.67Single7XKFBeta-Hydroxyandrosterone7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
16.67Single7XT9Serotonin7XT9-5-HT4-Serotonin-Gs/β1/γ2
16.67Single7XTASerotonin7XTA-5-HT4-Serotonin-Gi1/β1/γ2
16.67Single7YFCHistamine7YFC-H4-Histamine-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single7YFDImetit7YFD-H4-Imetit-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8DPFLorcaserin8DPF-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8EF6Morphine8EF6-μ-Morphine-Gi1/β1/γ2
16.67Single8GGYConstrained Epinephrine8GGY-β2-Constrained Epinephrine
16.67Single8H2GNiacin8H2G-HCA2-Niacin-Gi1/β1/γ2
16.67Single8HN8Histamine8HN8-H4-Histamine-Gi1/β1/γ2
16.67Single8JLOUlotaront8JLO-TA1-Ulotaront-Gs/β1/γ2
16.67Single8K2XCXCL108K2X-CXCR3-CXCL10-Gi1/β1/γ2
16.67Single8K5BNiacin8K5B-HCA2-Niacin
16.67Single8UO3Constrained Epinephrine8UO3-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
16.67Single8W89PEA8W89-TA1-PEA-chim(NtGi1L-Gs)/β1/γ2
16.67Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Single8X2KOleic monoethanolamide8X2K-GPR3-Oleic monoethanolamide-chim(NtGi1-Gs)/β1/γ2
16.67Single8XGSMetastin8XGS-Kiss1-Metastin-chim(NtGi1-Gq)/β1/γ2
16.67Single8XJKCloprosetnol8XJK-FP-alpha-Cloprosetnol-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8XJOU466198XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single8YKWSuccinic acid8YKW-Succinate-Succinic acid-Gi1/β1/γ1
16.67Single8ZX4Lysophosphatidylinositol 8ZX4-GPR55-Lysophosphatidylinositol-chim(NtGi1-G13)/β1/γ2
16.67Single9AS2DMT9AS2-5-HT2A-DMT-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Single9B9Y7DY9B9Y-CB1-7DY
16.67Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
16.67Single9CGJC6-Quino9CGJ-δ-C6-Quino-Gi1/β1/γ2
16.67Single9EPRRetinal9EPR-Rhodopsin-Retinal-Gi1/β1/γ2
16.67Single9IJEEpinephrine9IJE-β3-Epinephrine-chim(NtGi1-Gs)/β1/γ2
16.67Single9IQTNiacin9IQT-HCA2-Niacin-Gi1/β1/γ2
16.67Consensus5ht4_onOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
16.67Consensus5ht4_on_gpOrthosteric Ligand7XTA-5-HT4-Serotonin-Gi1/β1/γ2
16.67Consensusbeta1_onOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
16.67Consensusbeta1_on_gpOrthosteric Ligand8DCR-β1-Dobutamine-Gs/β1/γ2 7S0F-β1-Isoprenaline-Gi1/β1/γ2
16.67Consensuscck_onOrthosteric Ligandccka_on cckb_on
16.67Consensuscck_on_gpOrthosteric Ligandccka_on_gp cckb_on_gp
16.67Consensuschemerin_onOrthosteric Ligandcml1_on
16.67Consensusd3_offOrthosteric Ligand3PBL-D3-Eticlopride
16.67Consensusgal2_onOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Consensusgal2_on_gpOrthosteric Ligand7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2 7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.67Consensush4_onOrthosteric Ligand8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2 8JXX-H4-Clobenpropit-Gi1/β1/γ2
16.67Consensusnpy4_onOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
16.67Consensusnpy4_on_gpOrthosteric Ligand7X9C-Y4-Pancreatic Hormone-Gi1/β1/γ2
16.67Consensusnucleotide_on_gpOrthosteric Ligandadenosine_on_gp p2y_on_gp
16.67Consensusorexin_on_gpOrthosteric Ligandox2_on_gp
16.67Consensusprostanoid_offOrthosteric Ligandep_off dp_off
16.67Consensusprostanoid_onOrthosteric Ligandtp_on fp-alpha_on
16.67Consensusprostanoid_on_gpOrthosteric Ligandtp_on_gp fp-alpha_on_gp
16.67Consensustp_onOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.67Consensustp_on_gpOrthosteric Ligand8XJO-TXA2-U46619-chim(NtGi1-Gs-CtGq)/β1/γ2
16.28Single8W8WAlpha-MSH8W8W-MC3-α-MSH-Ca-Gs/β1/γ2
16.28Single8W8XBeta-MSH8W8X-MC3-β-MSH-Ca-Gs/β1/γ2
16.28Consensusp2y10_on_gpOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
16.22Single5VBLApelin mimetic peptide agonist5VBL-Apelin-Apelin mimetic peptide agonist
16.22Single6XBJCholesterol6XBJ-SMO-Cholesterol-Gi1/β1/γ2
16.22Single7F2OBradykinin7F2O-BK2-Bradykinin-chim(NtGi1-Gs-CtGq)/β1/γ2
16.22Single7F8WGastrin-177F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
16.22Single8F7REndomorphin8F7R-μ-Endomorphin-Gi1/β1/γ2
16.22Single8IA7Cholecystokinin-88IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2
16.22Single8XZFWN5618XZF-Apelin-WN561-Gi1/β1/γ2
16.22Single9EAJNanobody AT2099EAJ-AT1-Nanobody AT209
16.22Single9JF4PD1683689JF4-BB1-PD168368
16.22Single9MD1Buspirone9MD1-5-HT1A-Buspirone-Gz/β1/γ2
16.13Single2PED9-cis-Retinal2PED-Rhodopsin-9-cis-Retinal
16.13Single2Z7311-cis-Retinal2Z73-Rhodopsin-11-cis-Retinal
16.13Single3AYN9-cis-Retinal3AYN-Rhodopsin-9-cis-Retinal
16.13Single3ODUIT1t3ODU-CXCR4-IT1t
16.13Single3VG9ZM-2413853VG9-A2A-ZM-241385-Antibody
16.13Single4S0VSuvorexant4S0V-OX2-Suvorexant
16.13Single5K2DZM-2413855K2D-A2A-ZM-241385-Na
16.13Single5OLOTozadenant5OLO-A2A-Tozadenant-Na
16.13Single5WS3EMPA5WS3-OX2-EMPA
16.13Single6AKXA4R6AKX-CCR5-A4R
16.13Single6AKYMaraviroc6AKY-CCR5-Maraviroc
16.13Single6JZHZM-2413856JZH-A2A-ZM-241385-Na
16.13Single6KUYPubChem 1457046436KUY-α2a-PubChem 145704643
16.13Single6ME2Ramelteon6ME2-MT1-Ramelteon
16.13Single6OYAAll-trans-Retinal6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
16.13Single6PS7ZM-2413856PS7-A2A-ZM-241385-Na
16.13Single6TPJSuvorexant6TPJ-OX2-Suvorexant
16.13Single7BR3Elagolix7BR3-GnRH1-Elagolix
16.13Single7DHRIsoprenaline7DHR-β2-Isoprenaline-Gs/β1/γ2
16.13Single7F1ODopamine7F1O-D1-Dopamine-GDP; Mg-Gs/β1/γ2
16.13Single7LCJDanuglipron7LCJ-GLP-1-Danuglipron
16.13Single7LD4Adenosine7LD4-A1-Adenosine-Gi2/β1/γ2
16.13Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
16.13Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
16.13Single7T6SPubChem 247763417T6S-FPR2-ALX-PubChem 24776341-Gi1/β1/γ2
16.13Single7T8XAcetylcholine7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
16.13Single7T90Acetylcholine7T90-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
16.13Single7T96Acetylcholine7T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
16.13Single7TUZ7-alpha,25-dihydroxycholesterol7TUZ-GPR183-7-α,25-dihydroxycholesterol-Gi1/β1/γ2
16.13Single7VDLCortistatin-147VDL-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
16.13Single7VIHCBP-3077VIH-S1P1-CBP-307-Gi1/β1/γ2
16.13Single7VVOPTH7VVO-PTH1-PTH-Gs/β1/γ2
16.13Single7X5H5-CT7X5H-5-HT5A-5-CT-Gi1/β1/γ2
16.13Single7XRRLemborexant7XRR-OX2-Lemborexant
16.13Single7XT8Serotonin7XT8-5-HT4-Serotonin-Gs/β1/γ2
16.13Single7YM8Oxymetazoline7YM8-Alpha1A-Oxymetazoline-chim(Gs-CtGq)
16.13Single8DWGML3828DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
16.13Single8GGWConstrained Epinephrine8GGW-β2-Constrained Epinephrine
16.13Single8GGZConstrained Epinephrine8GGZ-β2-Constrained Epinephrine
16.13Single8GNGIstradefylline8GNG-A2A-Istradefylline
16.13Single8HOCImetit8HOC-H4-Imetit-Gi1/β1/γ2
16.13Single8IJBAcipimox8IJB-HCA2-Acipimox-Gi1/β1/γ2
16.13Single8IW4Spermidine8IW4-TA9-Spermidine-chim(NtGi1-Gs)/β1/γ2
16.13Single8IWESpermidine8IWE-TA9-Spermidine
16.13Single8RW0Istradefylline8RW0-A2A-Istradefylline-Na
16.13Single8UNSConstrained Epinephrine8UNS-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.13Single8UNTConstrained Epinephrine8UNT-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.13Single8UNXConstrained Epinephrine8UNX-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
16.13Single8WC3SEP-3638568WC3-TA1-SEP-363856-chim(NtGi1-Gs)/β1/γ2
16.13Single8YNAImmepip8YNA-H4-Immepip-Gi1/β1/γ2
16.13Single8YYWAlpha-ketoglutarate8YYW-Oxoglutarate-α-ketoglutarate-α-ketoglutarate-chim(Gi1-CtGq)/β1/γ2
16.13Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
16.13Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
16.13Single9EBHAdenosine9EBH-A3A-Adenosine-Gi1/β1/γ2
16.13Single9H2XA1IR19H2X-A2A-A1IR1-Na
16.13Single9MQJIsoquinuclidine9MQJ-μ-Isoquinuclidine
16.13Consensus5ht1e_onOrthosteric Ligand7E33-5-HT1E-BRL-54443-Gi1/β1/γ2 8UGY-5-HT1E-Mianserin-Gi1/β1/γ1 8UH3-5-HT1E-Setiptiline-Gi1/β1/γ1
16.13Consensus5ht_onOrthosteric Ligand5ht1_on 5ht2_on 5ht4_on 5ht5_on 5ht6_on 5ht7_on
16.13Consensusa1_onOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
16.13Consensusa1_on_gpOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2
16.13Consensusalpha2_offOrthosteric Ligandalpha2c_off
16.13Consensusangiotensin_offOrthosteric Ligandat1_off
16.13Consensusgnrh1_offOrthosteric Ligand7BR3-GnRH1-Elagolix
16.13Consensusgs_5htOrthosteric Ligand7XTC-5-HT7-5-CT-Gs/β1/γ2 7XTB-5-HT6-Serotonin-Gs/β1/γ2 8JLZ-5-HT6-ST1936-Gs/β1/γ2 7XT8-5-HT4-Serotonin-Gs/β1/γ2
16.13Consensushistamine_onOrthosteric Ligandh1_on h2_on h3_on h4_on
16.13Consensushistamine_on_gpOrthosteric Ligandh1_on_gp h2_on_gp h3_on_gp h4_on_gp
16.13Consensusm2_onOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
16.13Consensusm2_on_gpOrthosteric Ligand7T8X-M2-Acetylcholine-chim(NtGi1-Go)/β1/γ2
16.13Consensusorexin_offOrthosteric Ligandox2_off ox1_off
16.13Consensusox1_offOrthosteric Ligand6TP6-OX1-Filorexant 6TP4-OX1-ACT-462206 6V9S-OX1-GTPL11403 6TOT-OX1-Lemborexant 6TP3-OX1-Nemorexant 6TQ6-OX1-PubChem 145714283 6TQ9-OX1-SB-408124 4ZJC-OX1-SB-674042 4ZJ8-OX1-Suvorexant 6TOD-OX1-EMPA-Na 6TOS-OX1-GSK1059865-Na 6TQ4-OX1-PubChem 16046844-Na
16.13Consensusox2_offOrthosteric Ligand5WQC-OX2-EMPA 6TPN-OX2-HTL6641 7XRR-OX2-Lemborexant 6TPJ-OX2-Suvorexant
16.13Consensusrhodopsin_on_gpOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
16.13Consensussensory_offonOrthosteric Ligandsensory_off sensory_on
16.13Consensussensory_offon_gpOrthosteric Ligandsensory_on_gp sensory_on
15.91Single7VGXNeuropeptide-Y7VGX-Y1-Neuropeptide-Y-Gi1/β1/γ2
15.91Single8KGGLPS8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
15.79Single7F54Afamelanotide7F54-MC4-Afamelanotide-Gs/β1/γ2
15.79Single7F8XNN90567F8X-CCKA-NN9056
15.79Single7L0RNeurotensin7L0R-NTS1-Neurotensin-Gi1/β1/γ1
15.79Single7XAUOctreotide7XAU-SST2-Octreotide-Gi1/β1/γ2
15.79Single8F7XNociceptin8F7X-NOP-Nociceptin-Gi1/β1/γ2
15.79Single8INRAlpha-MSH8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.79Single8IZBLysophosphatidylserine8IZB-GPR174-Lysophosphatidylserine-Gs/β1/γ2
15.79Single8KIGSHU91198KIG-MC3-SHU9119-Ca
15.79Single8U4OCXCL128U4O-CXCR4-CXCL12-Gi1/β1/γ2
15.79Single8WKYPG-9348WKY-MC4-PG-934
15.79Single8WZ2Orexigenic Neuropeptide QRFP8WZ2-QRFP-Orexigenic Neuropeptide QRFP-chim(NtGi1L-Gs-CtGq)/β1/γ2
15.79Single8XBHS3E-LysoPS8XBH-GPR34-S3E-LysoPS-Gi1/β1/γ2
15.79Single9J0IUDP-Glucuronic acid9J0I-P2Y14-UDP-Glucuronic acid-Gi1/β1/γ2
15.79Single9M4TSilodosin9M4T-Alpha1A-Silodosin
15.79Consensuschemokine_onOrthosteric Ligandccr_on cxcr_on
15.79Consensuscxcr4_onOrthosteric Ligand8K3Z-CXCR4-CXCL12-Gi1/β1/γ1
15.79Consensusgi_nucleotideOrthosteric Ligandgi_adenosine gi_p2y
15.79Consensusmc4_onOrthosteric Ligand7AUE-MC4-Setmelanotide-chim(NtGi1L-Gs)/β1/γ2 7F58-MC4-THIQ-Gs/β1/γ2 7F54-MC4-Afamelanotide-Gs/β1/γ2 7F53-MC4-α-MSH-Gs/β1/γ2 7F55-MC4-Bremelanotide-Gs/β1/γ2
15.79Consensusnop_onOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
15.79Consensusnop_on_gpOrthosteric Ligand8F7X-NOP-Nociceptin-Gi1/β1/γ2
15.79Consensussomatostatin_offOrthosteric Ligandsst2_off
15.79Consensussst5_onOrthosteric Ligand8X8L-SST5-Cortistatin-chim(NtGi1-Gs-CtGi1)/β1/γ2 8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
15.62Single1F8811-cis-Retinal1F88-Rhodopsin-11-cis-Retinal
15.62Single4DKLBeta-Funaltrexamine4DKL-μ-β-Funaltrexamine
15.62Single4MBSMaraviroc4MBS-CCR5-Maraviroc
15.62Single4MQTIperoxo4MQT-M2-Iperoxo-LY2119620
15.62Single4ZJCSB-6740424ZJC-OX1-SB-674042
15.62Single5IU4ZM-2413855IU4-A2A-ZM-241385-Na
15.62Single5IUBQ274563445IUB-A2A-Q27456344-Na
15.62Single5K2CZM-2413855K2C-A2A-ZM-241385-Na
15.62Single5NLXZM-2413855NLX-A2A-ZM-241385-Na
15.62Single5NM4ZM-2413855NM4-A2A-ZM-241385-Na
15.62Single5UVIZM-2413855UVI-A2A-ZM-241385
15.62Single6FKAPubChem 1324730376FKA-Rhodopsin-PubChem 132473037
15.62Single6IQLL7458706IQL-D4-L745870
15.62Single6K41Dexmedetomidine6K41-α2b-Dexmedetomidine-Go/β1/γ2
15.62Single6ME32-Phenylmelatonin6ME3-MT1-2-Phenylmelatonin
15.62Single6MH8ZM-2413856MH8-A2A-ZM-241385
15.62Single6PELCitronellol6PEL-Rhodopsin-Citronellol-Gt(CT)
15.62Single6PS82-Phenylmelatonin6PS8-MT1-2-Phenylmelatonin
15.62Single6TP3Nemorexant6TP3-OX1-Nemorexant
15.62Single6V9SGTPL114036V9S-OX1-GTPL11403
15.62Single6WH4Methiothepin6WH4-5-HT2A-Methiothepin
15.62Single6ZG9GSK10347026ZG9-M1-GSK1034702
15.62Single7AROLUF58337ARO-A2A-LUF5833-Na
15.62Single7C2EPubChem 1490507997C2E-GLP-1-PubChem 149050799-Gs/β1/γ2
15.62Single7CKZDopamine7CKZ-D1-Dopamine-Mevidalen-Gs/β1/γ2
15.62Single7CMUPramipexole7CMU-D3-Pramipexole-Gi1/β1/γ2
15.62Single7CMVPD1289077CMV-D3-PD128907-Gi1/β1/γ2
15.62Single7E33BRL-544437E33-5-HT1E-BRL-54443-Gi1/β1/γ2
15.62Single7EJADexmedetomidine7EJA-α2a-Dexmedetomidine-Go/β1/γ2
15.62Single7F0TDopamine7F0T-D1-Dopamine-Gs/β1/γ2
15.62Single7F61PF-036547467F61-H3-PF-03654746
15.62Single7RANPubChem 1645758477RAN-5-HT2A-PubChem 164575847-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.62Single7T94Acetylcholine7T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
15.62Single7TRSAcetylcholine7TRS-M4-Acetylcholine-Gi1/β1/γ2
15.62Single7UL3Famotidine7UL3-H2-Famotidine
15.62Single7UM7Methylergometrine7UM7-5-HT5A-Methylergometrine-chim(NtGi1-Go)/β1/γ2
15.62Single7VUGJNJ-635330547VUG-GPR139-JNJ-63533054-Gi1/β1/γ2
15.62Single7WC9PubChem 1624213647WC9-5-HT2A-PubChem 162421364
15.62Single7XOVSR1461317XOV-CCKA-SR146131-Gs/β1/γ2
15.62Single7XXH2MeSADP7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.62Single8FCZ11-cis-Retinal8FCZ-Rhodopsin-11-cis-Retinal
15.62Single8GEDConstrained Epinephrine8GED-β2-Constrained Epinephrine-Gs/β1/γ2
15.62Single8GG5Constrained Epinephrine8GG5-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.62Single8HNMVUF112228HNM-CXCR3-VUF11222-Gi1/β1/γ2
15.62Single8IHKAcifran8IHK-HCA3-Acifran
15.62Single8JEI3-nitro-4-(propylamino)benzoic acid8JEI-HCAR3-3-nitro-4-(propylamino)benzoic acid-Gi1/β1/γ2
15.62Single8JERAcipimox8JER-HCA2-Acipimox-Go/β1/γ2
15.62Single8K9LDamgo8K9L-μ-Damgo-BMS-986122-Gi3/β1/γ1
15.62Single8RLNLUF58348RLN-A2A-LUF5834
15.62Single8RWCStilSwitch28RWC-A2A-StilSwitch2-Na
15.62Single8RWDStilSwitch38RWD-A2A-StilSwitch3-Na
15.62Single8RWIStilSwitch28RWI-A2A-StilSwitch2-Na
15.62Single8U02L-Dopamine8U02-D2-L-Dopamine-Go/β1/γ2
15.62Single8UNMConstrained Epinephrine8UNM-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.62Single8UNWConstrained Epinephrine8UNW-β2-Constrained Epinephrine-GTP-Gs/β1/γ2
15.62Single8V6UPubChem 1713924568V6U-5-HT2A-PubChem 171392456-chim(NtGi2-Gs-CtGq)/β1/γ2
15.62Single8W8BSEP-3638568W8B-5-HT1A-SEP-363856-Gi1/β1/γ2
15.62Single8Y53MK50468Y53-BB3-MK5046-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single8Y62C16:0 Ceramide8Y62-FPR2-ALX-C16:0 Ceramide-Gi1/β1/γ2
15.62Single8Y6YGLPG09748Y6Y-FFA2-GLPG0974
15.62Single8YH2Adenosine8YH2-A3A-Adenosine-Gi1/β1/γ2
15.62Single8YN3Histamine8YN3-H2-Histamine-Gs/β1/γ2
15.62Single8ZMGPimavanserin8ZMG-5-HT2A-Pimavanserin
15.62Single9ARXSerotonin9ARX-5-HT2A-Serotonin
15.62Single9AS5Mescaline9AS5-5-HT2A-Mescaline
15.62Single9AS6Mescaline9AS6-5-HT2A-Mescaline-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single9BA0A1AKN9BA0-CB1-A1AKN
15.62Single9CBLEpinephrine9CBL-α2a-Epinephrine-Gi1/β1/γ2
15.62Single9JFUNE52-QQ579JFU-GPR4-NE52-QQ57
15.62Single9JH3CMF-0199JH3-Apelin-CMF-019-Gi1/β1/γ2
15.62Single9JMDAzithromycin9JMD-Motilin-Azithromycin-chim(Gs-CtGq)/β1/γ2
15.62Single9K0KUTP9K0K-P2Y4-UTP-chim(NtGi1-Gs-CtGq)/β1/γ2
15.62Single9MQIIsoquinuclidine9MQI-μ-Isoquinuclidine
15.62Consensus5ht2a_offOrthosteric Ligand6A94-5-HT2A-Zotepine 6A93-5-HT2A-Risperidone 7VOD-5-HT2A-Cariprazine 7WC8-5-HT2A-Lumateperone 8JT8-5-HT2A-(R)-IHCH-7179
15.62Consensusadenosine_onOrthosteric Liganda1_on a2_on a3_on
15.62Consensusd3_onOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
15.62Consensusd3_on_gpOrthosteric Ligand7CMV-D3-PD128907-Gi1/β1/γ2 8IRT-D3-Rotigotine-Gi1/β1/γ2 7CMU-D3-Pramipexole-Gi1/β1/γ2
15.62Consensusgi_adenosineOrthosteric Ligand7LD4-A1-Adenosine-Gi2/β1/γ2 8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
15.62Consensusgrh_offOrthosteric Ligandgnrh1_off
15.62Consensusnop_offOrthosteric Ligand4EA3-NOP-PubChem 10296561 5DHG-NOP-C-35 5DHH-NOP-SB-612111
15.62Consensusnucleotide_offOrthosteric Ligandadenosine_off p2y_off
15.62Consensusopsins_offOrthosteric Ligandrhodopsin_off
15.62Consensusp2y1_on_gpOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
15.62Consensussensory_offOrthosteric Ligandopsins_off
15.38Single7EZKCholecystokinin-87EZK-CCKA-Cholecystokinin-8-chim(NtGi1-Gs)/β1/γ2
15.38Single7F1QMIP-1a7F1Q-CCR5-MIP-1a-Gi1/β1/γ2
15.38Single7RMISubstance-P7RMI-NK1-Substance-P-chim(Gs-CtGq)/β1/γ2
15.38Single7SK5CXCL127SK5-ACKR3-CXCL12
15.38Single7WJ5Somatostatin-147WJ5-SST2-Somatostatin-14-Gi1/β1/γ2
15.38Single8IBVMotilin8IBV-Motilin-Motilin-chim(NtGi1-Gs-CtGq)/β1/γ2
15.38Single8KH5Lysophosphatidylserine8KH5-GPR174-Lysophosphatidylserine-Gs/β1/γ2
15.38Single8WSSPro-MCH8WSS-MCH1-Pro-MCH-Gi1/β1/γ1
15.38Single9EAINanobody AT2099EAI-AT1-Losartan-Nanobody AT209
15.38Single9IQSMuscarinic toxin 39IQS-M4-Muscarinic toxin 3
15.38Single9J0FNADH9J0F-P2Y14-NADH-Gi1/β1/γ2
15.38Consensuscckb_onOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.38Consensusmc5_onOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
15.38Consensustachykinin_on_gpOrthosteric Ligandnk1_on_gp nk2_on_gp nk3_on_gp
15.15Single1HZX11-cis-Retinal1HZX-Rhodopsin-11-cis-Retinal
15.15Single4EJ4Naltrindole4EJ4-δ-Naltrindole
15.15Single4QKX35V4QKX-β2-35V
15.15Single4X1HNonyl-Beta-D-Glucopyranoside4X1H-Rhodopsin-Nonyl-β-D-Glucopyranoside-Gt(CT)
15.15Single5DHGC-355DHG-NOP-C-35
15.15Single5DHHSB-6121115DHH-NOP-SB-612111
15.15Single5NDDAZ8838; Na5NDD-PAR2-AZ8838; Na
15.15Single5UENDU1725UEN-A1-DU172
15.15Single5UIGCmpd-15UIG-A2A-Cmpd-1
15.15Single6D27CAY104716D27-DP2-CAY10471
15.15Single6DRXLisuride6DRX-5-HT2B-Lisuride
15.15Single6DRZMethysergide6DRZ-5-HT2B-Methysergide
15.15Single6FK7PubChem 1324730346FK7-Rhodopsin-PubChem 132473034
15.15Single6FKCPubChem 1324730396FKC-Rhodopsin-PubChem 132473039
15.15Single6GPSMK08126GPS-CCR2-MK0812
15.15Single6K42Dexmedetomidine6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
15.15Single6LPJZM-2413856LPJ-A2A-ZM-241385-Na
15.15Single6LPKZM-2413856LPK-A2A-ZM-241385-Na
15.15Single6WHADB139486WHA-5-HT2A-DB13948-chim(NtGi2L-Gs-CtGq)/β1/γ2
15.15Single6X1ADanuglipron6X1A-GLP-1-Danuglipron-Gs/β1/γ2
15.15Single6Z4VNTS8-136Z4V-NTS1-NTS8-13
15.15Single7BU7BI1671077BU7-β1-BI167107
15.15Single7CFMP3957CFM-GPBA-P395-Gs/β1/γ2
15.15Single7DB6Ramelteon7DB6-MT1-Ramelteon-Gi1/β1/γ2
15.15Single7FIHOrg435537FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
15.15Single7NA8PubChem 1780247NA8-Ghrelin-PubChem 178024-Gi1/β1/γ2
15.15Single7SQOTAK-9257SQO-OX2-TAK-925-Gi1/β1/γ2
15.15Single7T2GMitragynine Pseudoindoxyl7T2G-μ-Mitragynine Pseudoindoxyl-Gi1/β1/γ2
15.15Single7VKTLTB47VKT-BLT1-LTB4-Gi1/β1/γ2
15.15Single7WC8Lumateperone7WC8-5-HT2A-Lumateperone
15.15Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
15.15Single8EFQDamgo8EFQ-μ-Damgo-Gi1/β1/γ2
15.15Single8IHJAcifran8IHJ-HCA3-Acifran-Gi1/β1/γ2
15.15Single8IRTRotigotine8IRT-D3-Rotigotine-Gi1/β1/γ2
15.15Single8JD0NAM5638JD0-mGlu2; mGlu3-Glutamate-NAM563
15.15Single8JT8(R)-IHCH-71798JT8-5-HT2A-(R)-IHCH-7179
15.15Single8RW7StilSwitch18RW7-A2A-StilSwitch1-Na
15.15Single8RWXStilSwitch38RWX-A2A-StilSwitch3-Na
15.15Single8UWLLisuride8UWL-5-HT2A-Lisuride-chim(NtGi2-Gs-CtGq)/β1/γ2
15.15Single8WC7ZH86678WC7-TA1-ZH8667-chim(NtGi1-Gs)/β1/γ2
15.15Single8X17Namodenoson8X17-A3A-Namodenoson-Gi1/β1/γ2
15.15Single9IYAONO-97105319IYA-GPR55-ONO-9710531
15.15Single9PQD(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole9PQD-α2a-(6m)-1-methyl-6-(1,2,5,6-tetrahydropyridin-3-yl)-1h-indole
15.15Consensus5ht2b_offOrthosteric Ligand6DRZ-5-HT2B-Methysergide
15.15Consensusa3_onOrthosteric Liganda3a_on
15.15Consensusalpha2_onOrthosteric Ligandalpha2b_on
15.15Consensusalpha2_on_gpOrthosteric Ligandalpha2b_on_gp
15.15Consensusalpha2b_onOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
15.15Consensusalpha2b_on_gpOrthosteric Ligand6K42-α2b-Dexmedetomidine-Gi1/β1/γ2
15.15Consensusblt1_onOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
15.15Consensusblt1_on_gpOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
15.15Consensusblt_onOrthosteric Ligandblt1_on
15.15Consensusblt_on_gpOrthosteric Ligandblt1_on_gp
15.15Consensuscck_offOrthosteric Ligandccka_off
15.15Consensusccka_offOrthosteric Ligand7F8Y-CCKA-Devazepide 7F8U-CCKA-Lintitript
15.15Consensusccr2_offOrthosteric Ligand6GPS-CCR2-MK0812
15.15Consensusdop_offOrthosteric Ligand4EJ4-δ-Naltrindole
15.15Consensusgi_histamineOrthosteric Ligand8JXX-H4-Clobenpropit-Gi1/β1/γ2 8JXV-H4-Clozapine-Gi1/β1/γ2 8YUU-H3-Histamine-Gi1/β1/γ1 8HN8-H4-Histamine-Gi1/β1/γ2 8HOC-H4-Imetit-Gi1/β1/γ2 8JXW-H4-VUF6884-Gi1/β1/γ2
15.15Consensusgi_leukotrieneOrthosteric Ligand7VKT-BLT1-LTB4-Gi1/β1/γ2
15.15Consensusgi_orexinOrthosteric Ligand7SQO-OX2-TAK-925-Gi1/β1/γ2
15.15Consensusgq_amineOrthosteric Ligandgq_muscarinic gq_histamine
15.15Consensusleukotriene_onOrthosteric Ligandblt_on
15.15Consensusleukotriene_on_gpOrthosteric Ligandblt_on_gp
15.15Consensusmuscarinic_onOrthosteric Ligandm2_on m3_on m4_on m1_on
15.15Consensusmuscarinic_on_gpOrthosteric Ligandm2_on_gp m3_on_gp m4_on_gp m1_on_gp
15.00Single6MEOEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MEO-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
15.00Single7F4DAlpha-MSH7F4D-MC1-α-MSH-chim(NtGi1-Gs)/β1/γ2
15.00Consensuscckb_on_gpOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7F8V-CCKB-Gastrin-17-Gi2/β1/γ2
15.00Consensusmc3_onOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
15.00Consensusmc3_on_gpOrthosteric Ligand8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
14.71Single6GPXMK08126GPX-CCR2-MK0812
14.71Single6LUQHaloperidol6LUQ-D2-Haloperidol
14.71Single6OIKIperoxo6OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
14.71Single7EUOfMLF7EUO-FPR1-ALX-fMLF-Gi1/β1/γ2
14.71Single7VFXfMLF7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
14.71Single7VOEAripiprazole7VOE-5-HT2A-Aripiprazole
14.71Single7VV4Cortistatin-147VV4-MRGPRX2-Cortistatin-14
14.71Single7WC6LSD7WC6-5-HT2A-LSD
14.71Single8HNLPS3724248HNL-CXCR3-PS372424-Gi1/β1/γ2
14.71Single8X0BVU04244658X0B-mGlu5; mGlu5-Quisqualate-VU0424465
14.71Single8X0CVU04244658X0C-mGlu5; mGlu5-Quisqualate-VU0424465
14.71Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
14.71Single8X0DVU04244658X0D-mGlu5; mGlu5-Quisqualate-VU0424465
14.71Single8XYKVUF106618XYK-CXCR3-VUF10661-Go/β1/γ2
14.71Single8YH0NECA8YH0-A3A-NECA-Gi1/β1/γ2
14.71Single8ZVZBW245C8ZVZ-DP1-BW245C-Gs/β1/γ2
14.71Single8ZYTNeurotensin peptide 8-138ZYT-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
14.71Single9GE2ML1849GE2-GPR55-ML184-chim(NtGi1-G13)/β1/γ2
14.71Single9HAPTolvaptan9HAP-V2-Tolvaptan
14.71Consensusa3_on_gpOrthosteric Liganda3a_on_gp
14.71Consensusa3a_onOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.71Consensusa3a_on_gpOrthosteric Ligand8X17-A3A-Namodenoson-Gi1/β1/γ2 8X16-A3A-Piclidenoson-Gi1/β1/γ2
14.71Consensusfpr1-alx_onOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
14.71Consensusfpr1-alx_on_gpOrthosteric Ligand7VFX-FPR1-ALX-fMLF-Gi1/β1/γ2
14.71Consensusnucleotide_onOrthosteric Ligandadenosine_on p2y_on
14.63Single5WB2CX3CL1.355WB2-US28-CX3CL1.35
14.63Single6METEnvelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd46MET-CCR5-Envelope Glycoprotein Gp160; T-Cell Surface Glycoprotein Cd4
14.63Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
14.63Single8IEDA1LYA8IED-GPR156-A1LYA-Go/β1/γ2
14.63Consensusmc5_on_gpOrthosteric Ligand8INR-MC5-α-MSH-Ca-chim(NtGi1-Gs)/β1/γ2 8IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
14.63Consensusneuromedin-u_onOrthosteric Ligandnmur1_on nmur2_on
14.29Single3ZEVNeurotensin3ZEV-NTS1-Neurotensin
14.29Single4BV0Neurotensin4BV0-NTS1-Neurotensin
14.29Single6E59L-7607356E59-NK1-L-760735
14.29Single7E2ZAripiprazole7E2Z-5-HT1A-Aripiprazole-Gi1/β1/γ2
14.29Single7F1TMIP-1a7F1T-CCR5-MIP-1a
14.29Single7L0PNeurotensin7L0P-NTS1-Neurotensin-Gi1/β1/γ1
14.29Single7L0QNeurotensin7L0Q-NTS1-Neurotensin-Gi1/β1/γ1
14.29Single7P2L4YI7P2L-mGlu5-4YI
14.29Single7S8MCortistatin-147S8M-MRGPRX2-Cortistatin-14-Gi1/β1/γ2
14.29Single7T9NDPPC7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
14.29Single7XBDGalanin7XBD-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7XJLSpexin7XJL-GAL2-Spexin-chim(NtGi2L-Gs-CtGq)/β1/γ2
14.29Single7XKEBeta-Hydroxyandrosterone7XKE-ADGRG2-β-Hydroxyandrosterone-chim(NtGi1-Gs)/β1/γ2
14.29Single7Y24Octreotide7Y24-SST2-Octreotide-Go/β1/γ2
14.29Single7Y67C089 peptide7Y67-C5a1-C089 peptide-Gi1/β1/γ2
14.29Single8EFLSR170188EFL-μ-SR17018-Gi1/β1/γ2
14.29Single8FN1Neurotensin/Neuromedin-N8FN1-NTS1-Neurotensin/Neuromedin-N-chim(NtGi1-Go)/β1/γ2
14.29Single8IODPG-9018IOD-MC5-PG-901-Ca-chim(NtGi1-Gs)/β1/γ2
14.29Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
14.29Single8VVEnorBNI8VVE-κ-norBNI-Gi1/β1/γ2
14.29Single8XBIS3E-LysoPS8XBI-GPR34-S3E-LysoPS
14.29Single8XIPPasireotide8XIP-SST1-Pasireotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
14.29Single8XJMLatanoprost8XJM-FP-alpha-Latanoprost-chim(NtGi2-Gs-CtGq)/β1/γ2
14.29Single8XQTCholesterol8XQT-TAS2R14-Cholesterol-Gi1/β1/γ1
14.29Single8YNTSNAP-948478YNT-MCH1-SNAP-94847
14.29Consensuscyslt1_offOrthosteric Ligand6RZ5-CysLT1-Zafirlukast-Na 6RZ4-CysLT1-Pranlukast-Na
14.29Consensusneuromedin-u_on_gpOrthosteric Ligandnmur1_on_gp nmur2_on_gp
14.29Consensusneurotensin_onOrthosteric Ligandnts1_on
14.29Consensusnpy_offOrthosteric Ligandnpy1_off npy2_off
14.29Consensusnts1_onOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
14.29Consensusp2y10_onOrthosteric Ligand8KGG-P2Y10-LPS-chim(NtGi2-G13)/β1/γ2
13.89Single4GRVNeurotensin-(8-13)4GRV-NTS1-Neurotensin-(8-13)
13.89Single4PXZ2MeSADP4PXZ-P2Y12-2MeSADP
13.89Single4PY02MeSATP4PY0-P2Y12-2MeSATP
13.89Single5TZYMK8666; AP85TZY-FFA1-MK8666; AP8
13.89Single5X33BIIL2605X33-BLT1-BIIL260
13.89Single6OSAJMV4496OSA-NTS1-JMV449-Gi1/β1/γ2
13.89Single6XBLCholesterol6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
13.89Single7L0SNeurotensin7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.89Single7XJKGalanin7XJK-GAL2-Galanin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.89Single7XW6ML1097XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
13.89Single7XW9TRH7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.89Single8GCPPGE28GCP-EP4-PGE2-Gi1/β1/γ2
13.89Single8HK2C3a anaphylatoxin8HK2-C3aB-C3a anaphylatoxin-Gi1/β1/γ2
13.89Single8JPBNeurotensin-(8-13)8JPB-NTS1-Neurotensin-(8-13)-SBI-553; GDP; Mg-Gq; GRK2
13.89Single8U26Protachykinin-18U26-NK1-Protachykinin-1-Gs/β1/γ2
13.89Single8X8NOctreotide8X8N-SST5-Octreotide-chim(NtGi1-Gs-CtGi1)/β1/γ2
13.89Single9AU0BW245C9AU0-DP1-BW245C-Gs/β1/γ2
13.89Consensusffa2_on_gpOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
13.89Consensusgalanin_onOrthosteric Ligandgal2_on gal1_on
13.89Consensusgalanin_on_gpOrthosteric Ligandgal2_on_gp gal1_on_gp
13.89Consensusgi_neurotensinOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.89Consensusneurotensin_on_gpOrthosteric Ligandnts1_on_gp
13.89Consensusnts1_on_gpOrthosteric Ligand6OSA-NTS1-JMV449-Gi1/β1/γ2 7L0S-NTS1-Neurotensin-Gi1/β1/γ1
13.89Consensustrh_onOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.89Consensustrh_on_gpOrthosteric Ligand7XW9-TRH-TRH-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.79Single3OE8IT1t3OE8-CXCR4-IT1t
13.79Single6TQ9SB-4081246TQ9-OX1-SB-408124
13.79Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
13.79Single8A2OTheophylline8A2O-A2A-Theophylline-Na
13.79Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
13.79Single9CHUNoradrenaline9CHU-β2-Noradrenaline
13.79Consensusgs_histamineOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
13.79Consensush2_onOrthosteric Ligand8POK-H2-Histamine-Gs/β1/γ2
13.79Consensusopsins_onOrthosteric Ligandrhodopsin_on opsin1lw_on
13.79Consensussensory_onOrthosteric Ligandopsins_on
13.51Single4RWSvMIP-II4RWS-CXCR4-vMIP-II
13.51Single5CGDHTL142425CGD-mGlu5-HTL14242
13.51Single7EZHCholecystokinin-87EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
13.51Single7EZMCholecystokinin-87EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2
13.51Single7MBYCholecystokinin-87MBY-CCKA-Cholecystokinin-8-chim(NtGi1L-Gs-CtGq)/β1/γ2
13.51Single7PIUSetmelanotide7PIU-MC4-Setmelanotide-Gs/β1/γ2
13.51Single8FN0Neurotensin/Neuromedin-N8FN0-NTS1-Neurotensin/Neuromedin-N-SBI-553-chim(NtGi1-Go)/β1/γ2
13.51Single8HN1Toxin AdTx18HN1-Alpha1A-Toxin AdTx1
13.51Single8IULLatanoprost8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.51Single8JPFNeurotensin8JPF-NTS1-Neurotensin-SBI-553
13.51Single8K4OCXCL18K4O-KSHV-CXCL1-Gi1/β1/γ1
13.51Single8XVJMacitentan8XVJ-ETA-Macitentan
13.51Single8XVUCXCL28XVU-CXCR2-CXCL2
13.51Single8XXHCXCL28XXH-CXCR2-CXCL2-Go/β1/γ2
13.51Single8ZPLHF511168ZPL-CXCR4-HF51116
13.51Single9GG5U466199GG5-TXA2-U46619-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.51Consensusccka_onOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
13.51Consensusccka_on_gpOrthosteric Ligand7EZH-CCKA-Cholecystokinin-8-Gi1/β1/γ2
13.33Single2J4Y11-cis-Retinal2J4Y-Rhodopsin-11-cis-Retinal
13.33Single6FUFAll-trans-Retinal6FUF-Rhodopsin-All-trans-Retinal-Go
13.33Single6ME5Agomelatine6ME5-MT1-Agomelatine
13.33Single7D77Hydrocortisone7D77-ADGRG3-Hydrocortisone-Go/β1/γ2
13.33Single7EJKOxymetazoline7EJK-α2a-Oxymetazoline-Go/β1/γ2
13.33Single7MT8All-trans-Retinal7MT8-Rhodopsin-All-trans-Retinal-GRK1
13.33Single7MT9All-trans-Retinal7MT9-Rhodopsin-All-trans-Retinal-GRK1
13.33Single7MTAAll-trans-Retinal7MTA-Rhodopsin-All-trans-Retinal-GRK1
13.33Single8DPILorcaserin8DPI-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.33Single8F76Propanoic acid8F76-OR51E2-Propanoic acid-Gs/β1/γ2
13.33Single8ITFDMCHA8ITF-TA9-DMCHA-chim(NtGi1-Gs)/β1/γ2
13.33Single8IW72-Phenylethylamine8IW7-TA9-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
13.33Single8JEF(3S)-3-hydroxyoctanoic acid8JEF-HCA3-(3S)-3-hydroxyoctanoic acid-Gi1/β1/γ2
13.33Single8JRVGlucagon8JRV-Glucagon-Glucagon-Arrestin2
13.33Single8JXTHistamine8JXT-H4-Histamine-PO4-Gi1/β1/γ2
13.33Single8WC62-Phenylethylamine8WC6-TA1-2-Phenylethylamine-chim(NtGi1-Gs)/β1/γ2
13.33Single8WC9ZH86518WC9-TA1-ZH8651-chim(NtGi1-Gs-CtGq)/β1/γ2
13.33Single8Y63C20:0 Ceramide8Y63-FPR2-ALX-C20:0 Ceramide-Gi1/β1/γ2
13.33Single8YN9Histamine8YN9-H4-Histamine-Gi1/β1/γ2
13.33Single8YUUHistamine8YUU-H3-Histamine-Gi1/β1/γ1
13.33Single9JHJC18:0 Ceramide9JHJ-FPR2-ALX-C18:0 Ceramide-Gi1/β1/γ2
13.33Single9LRCHistamine9LRC-H4-Histamine
13.33Single9LREHistamine9LRE-H4-Histamine-Gi1/β1/γ2
13.33Consensush3_onOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
13.33Consensush3_on_gpOrthosteric Ligand8YUU-H3-Histamine-Gi1/β1/γ1
13.33Consensusopsins_on_gpOrthosteric Ligandrhodopsin_on_gp opsin1lw_on_gp
13.33Consensusrhodopsin_onOrthosteric Ligand6OYA-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
13.33Consensussensory_on_gpOrthosteric Ligandopsins_on_gp
13.16Single7CX2PGE27CX2-EP2-PGE2-Gs/β1/γ2
13.16Single7S8LCortistatin-147S8L-MRGPRX2-Cortistatin-14-chim(NtGi2L-Gs-CtGq)/β1/γ2
13.16Single7T11Octreotide7T11-SST2-Octreotide-Gi3/β1/γ2
13.16Single7XN9L-054,5227XN9-SST2-L-054,522
13.16Single8GDAL9026888GDA-EP4-L902688-Gs/β1/γ2
13.16Single8IQ4Carboprost8IQ4-FP-alpha-Carboprost-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single8IUMTafluprost acid8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Single8J22TUG-13758J22-FFA2-TUG-1375-Gi1/β1/γ2
13.16Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
13.16Consensusgq_cckOrthosteric Ligand8IA7-CCKB-Cholecystokinin-8-chim(NtGi1L-Gq)/β1/γ2 7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2 7EZM-CCKA-Cholecystokinin-8-chim(NtGsL-Gq)/β1/γ2 7F8W-CCKB-Gastrin-17-chim(NtGsL-Gq)/β1/γ2
13.16Consensusnmur1_onOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
13.16Consensussst2_onOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
13.16Consensussst2_on_gpOrthosteric Ligand7WIC-SST2-Somatostatin-14-Gi1/β1/γ2 7WIG-SST2-L-054,264-Gi1/β1/γ2 7YAE-SST2-Octreotide-Gi1/β1/γ2 7YAC-SST2-Paltusotine-Gi1/β1/γ2
12.90Single1U1911-cis-Retinal1U19-Rhodopsin-11-cis-Retinal
12.90Single2G87All-trans-Retinal2G87-Rhodopsin-All-trans-Retinal
12.90Single2I3511-cis-Retinal2I35-Rhodopsin-11-cis-Retinal
12.90Single6FK6PubChem 1324730336FK6-Rhodopsin-PubChem 132473033
12.90Single6HLLCP999946HLL-NK1-CP99994
12.90Single6PGSGeraniol6PGS-Rhodopsin-Geraniol-Gt(CT)
12.90Single6QNOAll-trans-Retinal6QNO-Rhodopsin-All-trans-Retinal-Gi1/β1/γ1
12.90Single6TP4ACT-4622066TP4-OX1-ACT-462206
12.90Single6TQ4PubChem 160468446TQ4-OX1-PubChem 16046844-Na
12.90Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
12.90Single7T96LY21196207T96-M2-Acetylcholine-LY2119620-Go/β1/γ2
12.90Single7TRPLY20332987TRP-M4-Iperoxo-LY2033298-Gi1/β1/γ2
12.90Single7V68Iperoxo7V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
12.90Single7VUIJNJ-635330547VUI-GPR139-JNJ-63533054-GTP-chim(Gs-CtGq)/β1/γ2
12.90Single7XTBSerotonin7XTB-5-HT6-Serotonin-Gs/β1/γ2
12.90Single7YS6Serotonin7YS6-5-HT6-Serotonin-chim(NtGi1-Gs)/β1/γ2
12.90Single8HSCFab0468HSC-GPR20-Fab046-Gi1/β1/γ2
12.90Single8IHIAcifran8IHI-HCA2-Acifran-Gi1/β1/γ2
12.90Single8RWHStilSwitch28RWH-A2A-StilSwitch2-Na
12.90Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
12.90Single8U4RREGN7663-Fab8U4R-CXCR4-REGN7663-Fab
12.90Single8UO4Constrained Epinephrine8UO4-β2-Constrained Epinephrine-GTP; Mg-Gs/β1/γ2
12.90Single8YH3N-methyladenosine8YH3-A3A-N-methyladenosine-Gi1/β1/γ2
12.90Single8YN4Histamine8YN4-H2-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.90Single8YN5Histamine8YN5-H3-Histamine-Gi1/β1/γ2
12.90Single8YN6Imetit8YN6-H3-Imetit-Gi1/β1/γ2
12.90Single8YN7Immethridine8YN7-H3-Immethridine-Go/β1/γ2
12.90Single8ZX5AM2518ZX5-GPR55-AM251-chim(NtGi1-G13)/β1/γ2
12.90Single9AS7Psilocin9AS7-5-HT2A-Psilocin
12.90Single9IXJHistamine9IXJ-H2-Histamine-Gs/β1/γ2
12.82Single7NA7Ghrelin-277NA7-Ghrelin-Ghrelin-27-Gi1/β1/γ2
12.82Single7W53Neuromedin-U-257W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.82Single7WICSomatostatin-147WIC-SST2-Somatostatin-14-Gi1/β1/γ2
12.82Single7XMRSomatostatin-147XMR-SST2-Somatostatin-14-Gi1/β1/γ2
12.82Single8IEBA1LYA8IEB-GPR156-A1LYA
12.82Single8IEIA1LYA8IEI-GPR156-A1LYA
12.82Single8IEIA1LYA8IEI-GPR156-A1LYA
12.82Single8IEPA1LYA8IEP-GPR156-A1LYA
12.82Single8IEPA1LYA8IEP-GPR156-A1LYA
12.82Consensusnmur1_on_gpOrthosteric Ligand7W53-NMUR1-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single1GZM11-cis-Retinal1GZM-Rhodopsin-11-cis-Retinal
12.50Single3C9L11-cis-Retinal3C9L-Rhodopsin-11-cis-Retinal
12.50Single3PWHZM-2413853PWH-A2A-ZM-241385
12.50Single4BWBNeurotensin4BWB-NTS1-Neurotensin
12.50Single4MQTLY21196204MQT-M2-Iperoxo-LY2119620
12.50Single5OLHVipadenant5OLH-A2A-Vipadenant-Na
12.50Single5OLVLUAA410635OLV-A2A-LUAA41063-Na
12.50Single5ZKQABT-4915ZKQ-PAF-ABT-491
12.50Single6D9HAdenosine6D9H-A1-Adenosine-Gi2/β1/γ2
12.50Single6LFOInterleukin-86LFO-CXCR2-Interleukin-8-Gi1/β1/γ2
12.50Single6ME9Ramelteon6ME9-MT2-Ramelteon
12.50Single6RNKNF-56-EJ406RNK-Succinate-NF-56-EJ40
12.50Single6TODEMPA6TOD-OX1-EMPA-Na
12.50Single6TQ6PubChem 1457142836TQ6-OX1-PubChem 145714283
12.50Single7EJ0L-Norepinephrine7EJ0-α2a-L-Norepinephrine-Go/β1/γ2
12.50Single7F8ULintitript7F8U-CCKA-Lintitript
12.50Single7F8YDevazepide7F8Y-CCKA-Devazepide
12.50Single7S8PMS471347S8P-MRGPRX4-MS47134-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.50Single7SRSLSD7SRS-5-HT2B-LSD-Arrestin2
12.50Single7W0MPubChem 1227019087W0M-Apelin-PubChem 122701908-Gi1/β1/γ2
12.50Single7X2CFenoldopam7X2C-D1-Fenoldopam-Fenoldopam-Gs/β1/γ2
12.50Single7X2FDopamine7X2F-D1-Dopamine-Mevidalen-Gs/β1/γ2
12.50Single7XJJGalanin7XJJ-GAL1-Galanin-Go/β1/γ2
12.50Single8FYXBuspirone8FYX-5-HT1A-Buspirone-Gi1/β1/γ1
12.50Single8H8JLodoxamide8H8J-GPR35-Lodoxamide-Ca-chim(NtGi1L-G13)/β1/γ2
12.50Single8HDPAdenosine8HDP-A2B-Adenosine-Gs/β1/γ2
12.50Single8HMPC178HMP-GPR52-C17-Gs/β1/γ2
12.50Single8IEBA1LYA8IEB-GPR156-A1LYA
12.50Single8IOCGamma-MSH8IOC-MC3-γ-MSH-Ca-chim(NtGi1-Gs)/β1/γ2
12.50Single8J6LNiacin8J6L-HCA2-Niacin-Gi1/β1/γ2
12.50Single8JBHSubstance-P8JBH-NK3-Substance-P-chim(NtGi1-Gs-CtGq)/β1/γ2
12.50Single8RVWStilSwitch38RVW-A2A-StilSwitch3-Na
12.50Single8RW4AzoSwitch28RW4-A2A-AzoSwitch2-Na
12.50Single8RWEStilSwitch48RWE-A2A-StilSwitch4-Na
12.50Single8TZQL-Dopamine8TZQ-D2-L-Dopamine-Go/β1/γ2
12.50Single8U4PAMD31008U4P-CXCR4-AMD3100-Gi1/β1/γ2
12.50Single8UTDMK19038UTD-HCA2-MK1903-Gi1/β1/γ2
12.50Single8XXVIndomethacin8XXV-DP2-Indomethacin-A1D5Q-Gi1/β1/γ2
12.50Single8YUTAmthamine8YUT-H2-Amthamine-Gs/β1/γ2
12.50Single8YUVImmepip8YUV-H3-Immepip-Gi1/β1/γ2
12.50Single9FUPIstradefylline9FUP-A2A-Istradefylline-Na
12.50Single9IK8SST analogue9IK8-SST1-SST analogue-Gi1/β1/γ2
12.50Single9IQVMuscarinic toxin 39IQV-Alpha1A-Muscarinic toxin 3
12.50Single9LRBHistamine9LRB-H1-Histamine-Gs/β1/γ2
12.50Consensuscxcr1_onOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
12.50Consensusgq_histamineOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
12.50Consensush1_on_gpOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
12.50Consensusp2y1_onOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
12.50Consensuspaf_offOrthosteric Ligand5ZKQ-PAF-ABT-491
12.50Consensusrhodopsin_offOrthosteric Ligand1U19-Rhodopsin-11-cis-Retinal 2PED-Rhodopsin-9-cis-Retinal 5TE5-Rhodopsin-20-Methanoretinal
12.20Single7W55Neuromedin-U-257W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Single7XOUCholecystokinin-87XOU-CCKA-Cholecystokinin-8-Gs/β1/γ2
12.20Single8K6MNeuropeptide-Y8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
12.20Consensusnmur2_onOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Consensusnmur2_on_gpOrthosteric Ligand7W55-NMUR2-Neuromedin-U-25-chim(NtGi1-Gs-CtGq)/β1/γ2
12.20Consensusnpy1_onOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
12.20Consensusnpy1_on_gpOrthosteric Ligand8K6M-Y1-Neuropeptide-Y-Gi2/β1/γ1
12.12Single3OAX11-cis-Retinal3OAX-Rhodopsin-11-cis-Retinal
12.12Single3REYXAC3REY-A2A-XAC
12.12Single3RZECidoxepin3RZE-H1-Cidoxepin
12.12Single4N6HNaltrindole4N6H-δ-Naltrindole-Na
12.12Single6FK8PubChem 1324730356FK8-Rhodopsin-PubChem 132473035
12.12Single6U1NLY21196206U1N-M2-LY2119620-Arrestin2
12.12Single6VI4JDTic6VI4-κ-JDTic
12.12Single6WJCMuscarinic toxin 76WJC-M1-Atropine-Muscarinic toxin 7
12.12Single6ZDVChromone 5d6ZDV-A2A-Chromone 5d-Na
12.12Single6ZFZ77-LH-28-16ZFZ-M1-77-LH-28-1
12.12Single7F1ZDopamine7F1Z-D1-Dopamine-GDP-Gs/β1/γ2
12.12Single7F24Dopamine7F24-D1-Dopamine-GDP-Gs/β1/γ2
12.12Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
12.12Single7T94LY21196207T94-M2-Acetylcholine-LY2119620-chim(NtGi1-Go)/β1/γ2
12.12Single7UTZDPPC7UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
12.12Single7WVUfMLF7WVU-FPR1-ALX-fMLF-Gi1/β1/γ2
12.12Single7ZBC11-cis-Retinal7ZBC-Rhodopsin-11-cis-Retinal
12.12Single7ZBE11-cis-Retinal7ZBE-Rhodopsin-11-cis-Retinal
12.12Single8DPGPsilocin8DPG-5-HT2C-Psilocin-chim(NtGi2L-Gs-CtGq)/β1/γ2
12.12Single8H4LDoconexent8H4L-FFA4-Doconexent-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single8K2WAMG4878K2W-CXCR3-AMG487
12.12Single8K4SDCA-3P8K4S-MRGPRX4-DCA-3P-chim(NtGi1L-Gs-CtGq)/β1/γ2
12.12Single8X7ATreprostinil8X7A-I2-Treprostinil-Gs/β1/γ2
12.12Single8Y45ADL58598Y45-δ-ADL5859-Gi2/β1/γ2
12.12Single8ZPMAMD0708ZPM-CXCR4-AMD070
12.12Single8ZPNAMD31008ZPN-CXCR4-AMD3100
12.12Single9AS3LSD9AS3-5-HT2A-LSD
12.12Single9AS4LSD9AS4-5-HT2A-LSD-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single9K0XATP9K0X-P2Y2-ATP-chim(NtGi1-Gs-CtGq)/β1/γ2
12.12Single9K20ATP9K20-P2Y2-ATP-chim(NtGi1-Go)/β1/γ2
12.12Consensuscxcr2_onOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
12.12Consensuscxcr3_offOrthosteric Ligand8K2W-CXCR3-AMG487
11.90Single7W57Neuromedin-S7W57-NMUR2-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
11.76Single4QIMANTA XV4QIM-SMO-ANTA XV
11.76Single5T04Neurotensin5T04-NTS1-Neurotensin
11.76Single6ORVTT-OAD26ORV-GLP-1-TT-OAD2-Gs/β1/γ2
11.76Single6Z10PubChem 1545855546Z10-Succinate-PubChem 154585554
11.76Single7PP1Selatogrel7PP1-P2Y12-Selatogrel
11.76Single7SCGFH2107SCG-μ-FH210-Gi1/β1/γ2
11.76Single7TRQVU04671547TRQ-M4-Iperoxo-VU0467154-Gi1/β1/γ2
11.76Single7WQ3Galanin7WQ3-GAL1-Galanin-Gi1/β1/γ2
11.76Single8EJKTAK-8758EJK-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
11.76Single8IC0Interleukin-88IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.76Single8KEXDCA-3P8KEX-MRGPRX4-DCA-3P
11.76Single8KFYZK-7563268KFY-CCR8-ZK-756326-Gi1/β1/γ2
11.76Single8XJLPGF2-alpha8XJL-FP-alpha-PGF2-α-chim(NtGi2-Gs-CtGq)/β1/γ2
11.76Single8YH5Riboprine8YH5-A3A-Riboprine-Gi1/β1/γ2
11.76Single8ZYYNeurotensin peptide 8-138ZYY-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
11.76Single9JGKBalovaptan9JGK-5-HT2B-Balovaptan
11.76Consensusalicarboxylic_offOrthosteric Ligandsuccinate_off
11.76Consensuscxcr1_on_gpOrthosteric Ligand8IC0-CXCR1-Interleukin-8-Gi1/β1/γ2
11.76Consensusgal1_onOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
11.76Consensusgal1_on_gpOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
11.76Consensusgi_galaninOrthosteric Ligand7WQ3-GAL1-Galanin-Gi1/β1/γ2
11.76Consensussuccinate_offOrthosteric Ligand6RNK-Succinate-NF-56-EJ40 6Z10-Succinate-PubChem 154585554
11.43Single4JKVTaladegib4JKV-SMO-Taladegib
11.43Single4PHUFasiglifam4PHU-FFA1-Fasiglifam
11.43Single5CGCHTL142425CGC-mGlu5-HTL14242
11.43Single5T1ABMS-6815T1A-CCR2-BMS-681-PubChem 12093170
11.43Single5YHLPubChem 1351213525YHL-EP4-PubChem 135121352
11.43Single5YWYONO-AE3-2085YWY-EP4-ONO-AE3-208
11.43Single6LFMInterleukin-86LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
11.43Single6M9TMisoprostol-FA6M9T-EP3-Misoprostol-FA
11.43Single6RZ4Pranlukast6RZ4-CysLT1-Pranlukast-Na
11.43Single7WIGL-054,2647WIG-SST2-L-054,264-Gi1/β1/γ2
11.43Single8GD9Rivenprost8GD9-EP4-Rivenprost-Gs/β1/γ2
11.43Single8GDCPGE28GDC-EP3-PGE2-Gi1/β1/γ2
11.43Single9HC04YI9HC0-mGlu5-4YI
11.43Consensusadgrg2_onOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.43Consensusadgrg2_on_gpOrthosteric Ligand7WUI-ADGRG2-IP15-chim(NtGi1-Gs)/β1/γ2 7WUQ-ADGRG2-Gs/β1/γ2 7XKF-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
11.43Consensuscxcr2_on_gpOrthosteric Ligand6LFM-CXCR2-Interleukin-8-Gi1/β1/γ2
11.43Consensuscyslt_offOrthosteric Ligandcyslt2_off cyslt1_off
11.43Consensusep4_offOrthosteric Ligand5YWY-EP4-ONO-AE3-208 5YHL-EP4-PubChem 135121352
11.43Consensusep_offOrthosteric Ligandep4_off
11.11Single4OO9Mavoglurant4OO9-mGlu5-Mavoglurant
11.11Single5TZRMK86665TZR-FFA1-MK8666
11.11Single5V56TC1145V56-SMO-TC114
11.11Single5V57TC1145V57-SMO-TC114
11.11Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
11.11Single6RZ5Zafirlukast6RZ5-CysLT1-Zafirlukast-Na
11.11Single7R0CAVP7R0C-V2-AVP-Arrestin2
11.11Single7XOWGastrin7XOW-CCKB-Gastrin-chim(NtGi1-Gq)/β1/γ2
11.11Single8FMZNeurotensin/Neuromedin-N8FMZ-NTS1-Neurotensin/Neuromedin-N-chim(NtGi2L-Gs-CtGq)/β1/γ2
11.11Single8GDBPGE28GDB-EP4-PGE2-Gs/β1/γ2
11.11Single8IUKPGF2-alpha8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2
11.11Single8TAOCDPPB8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
11.11Single8X0FVU04244658X0F-mGlu5; mGlu5-Quisqualate-VU0424465
11.11Single9IK9SST analogue9IK9-SST1-SST analogue-Gi1/β1/γ2
11.11Single9ITELPA9ITE-LPA6-LPA-chim(NtGi2-G13)/β1/γ2
11.11Consensusffa2_onOrthosteric Ligand8J22-FFA2-TUG-1375-Gi1/β1/γ2
11.11Consensusffa_onOrthosteric Ligandffa2_on ffa3_on
11.11Consensusffa_on_gpOrthosteric Ligandffa2_on_gp ffa3_on_gp
11.11Consensusgi_ffaOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2 8J22-FFA2-TUG-1375-Gi1/β1/γ2
11.11Consensusnpy1_offOrthosteric Ligand5ZBH-Y1-BMS-193885 5ZBQ-Y1-UR-MK-299
10.81Single3VW7Vorapaxar; Na3VW7-PAR1-Vorapaxar; Na
10.81Single4N4WSANT-14N4W-SMO-SANT-1
10.81Single7F55Bremelanotide7F55-MC4-Bremelanotide-Gs/β1/γ2
10.81Single7L1UOrexin7L1U-OX2-Orexin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single7WQ4Galanin7WQ4-GAL2-Galanin-chim(NtGi1-Gs-CtGq)/β1/γ2
10.81Single8WRBLysophosphatidylserine8WRB-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
10.81Single8XQJJN2418XQJ-Apelin-JN241
10.81Single8XWMCXCL68XWM-CXCR2-CXCL6
10.81Single8XX3CXCL38XX3-CXCR2-CXCL3-Go/β1/γ2
10.81Single8Y6WTUG-13758Y6W-FFA2-TUG-1375-4-CMTB-Gi1/β1/γ2
10.81Single9BJKNAM9BJK-μ-Naloxone-NAM
10.71Single8GEJConstrained Epinephrine8GEJ-β2-Constrained Epinephrine-Gs/β1/γ2
10.71Single8WCBCyclohexylammonium Ion8WCB-TA1-Cyclohexylammonium Ion-chim(NtGi1-Gs-CtGq)/β1/γ2
10.71Single8WCCCyclohexylammonium Ion8WCC-TA1-Cyclohexylammonium Ion
10.53Single6UP7Neurotensin6UP7-NTS1-Neurotensin-Arrestin2
10.53Single7CX4Evatanepag7CX4-EP2-Evatanepag-Gs/β1/γ2
10.53Single7D7MDinoprostone7D7M-EP4-Dinoprostone-Gs/β1/γ1
10.53Single8XBES3E-LysoPS8XBE-GPR34-S3E-LysoPS-Gi1/β1/γ1
10.53Single8XWFCXCL38XWF-CXCR2-CXCL3
10.53Single9M1HProstaglandin E29M1H-EP1-Prostaglandin E2-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Consensusfp-alpha_onOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
10.53Consensusfp-alpha_on_gpOrthosteric Ligand8IUK-FP-alpha-PGF2-α-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUL-FP-alpha-Latanoprost-chim(NtGi1-Gs-CtGq)/β1/γ2 8IUM-FP-alpha-Tafluprost acid-chim(NtGi1-Gs-CtGq)/β1/γ2
10.34Single3PXOAll-trans-Retinal3PXO-Rhodopsin-All-trans-Retinal
10.34Single5DYSAll-trans-Retinal5DYS-Rhodopsin-All-trans-Retinal
10.34Single5MZJTheophylline5MZJ-A2A-Theophylline-Na
10.34Single7XKDBeta-Hydroxyandrosterone7XKD-ADGRG2-β-Hydroxyandrosterone-Gs/β1/γ2
10.34Single8HQMNPGLY8HQM-GPR132-NPGLY-Gi1/β1/γ2
10.34Single8HS2Fab0468HS2-GPR20-Fab046
10.34Single8HVINOX-6-78HVI-GPR132-NOX-6-7-Gi1/β1/γ2
10.34Single8PWNTheophylline8PWN-A2A-Theophylline
10.34Single8X9S5alpha-DHT8X9S-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
10.34Single9IV25alpha-DHT9IV2-ADGRD1-5α-DHT-chim(NtGi1-Gs)/β1/γ2
10.26Single6KNMJN241-96KNM-Apelin-JN241-9
10.26Single6OS9JMV4496OS9-NTS1-JMV449-Gi1/β1/γ2
10.26Single6RZ6ONO-25703666RZ6-CysLT2-ONO-2570366
10.26Single7YAEOctreotide7YAE-SST2-Octreotide-Gi1/β1/γ2
10.26Single8SAI1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine8SAI-GPR34-1-Oleoyl-2-Hydroxy-Sn-Glycero-3-Phospho-L-Serine-Gi1/β1/γ2
10.26Single8XQJJN2418XQJ-Apelin-JN241
10.26Single8XX6CXCL88XX6-CXCR2-CXCL8-Go/β1/γ2
10.26Single8Z74Agonistic antibody8Z74-Apelin-Agonistic antibody
10.26Single9ITBLPA9ITB-LPA6-LPA-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single9JH6C20:0 Ceramide9JH6-CysLT2-C20:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
10.26Single9NS9TUG-13759NS9-FFA2-TUG-1375-Compound 187-Gi1/β1/γ2
10.26Consensuskiss1_onOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.26Consensuskisspeptin_onOrthosteric Ligandkiss1_on
10.00Single2HPYAll-trans-Retinal2HPY-Rhodopsin-All-trans-Retinal
10.00Single3RFMCaffeine3RFM-A2A-Caffeine
10.00Single6OY9All-trans-Retinal6OY9-Rhodopsin-All-trans-Retinal-Gt/β1/γ1
10.00Single6RZ8ONO-20803656RZ8-CysLT2-ONO-2080365
10.00Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
10.00Single7CX3Taprenepag7CX3-EP2-Taprenepag-Gs/β1/γ2
10.00Single7MTBAll-trans-Retinal7MTB-Rhodopsin-All-trans-Retinal-GRK1
10.00Single7W56Neuromedin-S7W56-NMUR1-Neuromedin-S-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8DPHLorcaserin8DPH-5-HT2C-Lorcaserin-chim(NtGi2L-Gs-CtGq)/β1/γ2
10.00Single8GEIConstrained Epinephrine8GEI-β2-Constrained Epinephrine-Gs/β1/γ2
10.00Single8IWM2-Phenylethylamine8IWM-TA9-2-Phenylethylamine
10.00Single8WC5Tetramethylammonium Ion8WC5-TA1-Tetramethylammonium Ion-chim(NtGi1-Gs)/β1/γ2
10.00Single8XOFLys058XOF-GPR30-Lys05-chim(NtGi1-Gs-CtGq)/β1/γ2
10.00Single8XWNCXCL88XWN-CXCR2-CXCL8
10.00Single8Y02Retinal8Y02-OPN1SW-Retinal-Gi1/β1/γ2
10.00Single8ZBJSomatostatin-148ZBJ-SST5-Somatostatin-14-Gi1/β1/γ2
10.00Single8ZCJPasireotide8ZCJ-SST5-Pasireotide-Gi1/β1/γ1
10.00Single8ZJDKisspeptin-108ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.00Single9EE9Adenosine9EE9-A2A-Adenosine-Gs/β1/γ2
10.00Consensusgq_kisspeptinOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.00Consensuskiss1_on_gpOrthosteric Ligand8ZJD-Kiss1-Kisspeptin-10-chim(NtGi1-Gq)/β1/γ1
10.00Consensuskisspeptin_on_gpOrthosteric Ligandkiss1_on_gp
10.00Consensusp2y_offOrthosteric Ligandp2y1_off
9.76Single9IQRMuscarinic toxin 39IQR-α2a-Muscarinic toxin 3
9.68Single3C9M11-cis-Retinal3C9M-Rhodopsin-11-cis-Retinal
9.68Single3PQRAll-trans-Retinal3PQR-Rhodopsin-All-trans-Retinal-Gt(CT)
9.68Single3UZAGTPL92363UZA-A2A-GTPL9236
9.68Single4XNWMRS25004XNW-P2Y1-MRS2500
9.68Single6FK9PubChem 1324730366FK9-Rhodopsin-PubChem 132473036
9.68Single6OIKLY21196206OIK-M2-Iperoxo-LY2119620-chim(NtGi1-Go)/β1/γ2
9.68Single7F23Dopamine7F23-D1-Dopamine-GDP-Gs/β1/γ2
9.68Single8EITDoconexent8EIT-FFA1-Doconexent-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.68Single8IU2Retinal8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
9.68Single8J21Butyric acid8J21-FFA3-Butyric acid-Gi1/β1/γ2
9.68Single8J24Acetic acid8J24-FFA2-Acetic acid-Gi1/β1/γ2
9.68Consensus5ht2_onOrthosteric Ligand5ht2b_on
9.68Consensus5ht2b_onOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.68Consensusffa3_onOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
9.68Consensusffa3_on_gpOrthosteric Ligand8J21-FFA3-Butyric acid-Gi1/β1/γ2
9.68Consensusgi_opsinsOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
9.68Consensusgi_sensoryOrthosteric Ligandgi_opsins
9.68Consensusopsin1lw_onOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
9.68Consensusopsin1lw_on_gpOrthosteric Ligand8IU2-Opsin1LW-Retinal-Gi1/β1/γ2
9.68Consensusp2y1_offOrthosteric Ligand4XNW-P2Y1-MRS2500
9.38Single1L9H11-cis-Retinal1L9H-Rhodopsin-11-cis-Retinal
9.38Single4O9RCyclopamine4O9R-SMO-Cyclopamine
9.38Single5L7IVismodegib5L7I-SMO-Vismodegib
9.38Single5TE520-Methanoretinal5TE5-Rhodopsin-20-Methanoretinal
9.38Single6I9K9-cis-Retinal6I9K-Rhodopsin-9-cis-Retinal
9.38Single6PH7Nerol6PH7-Rhodopsin-Nerol-Gt(CT)
9.38Single7DFLHistamine7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
9.38Single7E2YSerotonin7E2Y-5-HT1A-Serotonin-Gi1/β1/γ2
9.38Single7SRQLSD7SRQ-5-HT2B-LSD
9.38Single8A2PLUAA470708A2P-A2A-LUAA47070-Na
9.38Single8JILNiacin8JIL-HCA2-Niacin-Gi1/β1/γ2
9.38Single8YKDDehydroepiandrosterone8YKD-ADGRG2-Dehydroepiandrosterone-chim(NtGi1-Gs)/β1/γ2
9.38Single8YN2Histamine8YN2-H1-Histamine-chim(NtGi1L-Gs-CtGq)/β1/γ2
9.38Single9IZDCHBA9IZD-HCA1-CHBA-Gi1/β1/γ2
9.38Single9LMPNE52-QQ579LMP-GPR4-NE52-QQ57
9.38Consensusadgrg_onOrthosteric Ligandadgrg2_on adgrg4_on
9.38Consensusadgrg_on_gpOrthosteric Ligandadgrg2_on_gp adgrg4_on_gp
9.38Consensusgq_nucleotideOrthosteric Ligandgq_p2y
9.38Consensusgq_p2yOrthosteric Ligand7XXH-P2Y1-2MeSADP-chim(NtGi1-G11)/β1/γ2
9.38Consensush1_onOrthosteric Ligand7DFL-H1-Histamine-chim(NtGi1L-Gq)/β1/γ2
9.09Single4QINSAG1.54QIN-SMO-SAG1.5
9.09Single6DS0Ly2660976DS0-5-HT2B-Ly266097
9.09Single6FKBPubChem 1324730386FKB-Rhodopsin-PubChem 132473038
9.09Single6O3CSAG21k6O3C-SMO-SAG21k-Cholesterol
9.09Single6WWZCCL206WWZ-CCR6-CCL20-Go/β1/γ2
9.09Single6ZA8RTI-3a6ZA8-NTS1-RTI-3a
9.09Single7LJDDopamine7LJD-D1-Dopamine-Mevidalen-Gs/β1/γ1
9.09Single7SRRLSD7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single7VUJJNJ-635330547VUJ-GPR139-JNJ-63533054-GDP-chim(Gs-CtGq)/β1/γ2
9.09Single8A6CAll-trans-Retinal8A6C-Rhodopsin-All-trans-Retinal
9.09Single8A6DAll-trans-Retinal8A6D-Rhodopsin-All-trans-Retinal
9.09Single8A6EAll-trans-Retinal8A6E-Rhodopsin-All-trans-Retinal
9.09Single8DWHPubChem 1390305318DWH-MRGPRX1-PubChem 139030531-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8J20Valeric acid8J20-FFA3-Valeric acid-AR420626-Gi1/β1/γ2
9.09Single8T3SButyric acid8T3S-FFA2-Butyric acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8T3VDocosa-4,7,10,13,16,19-Hexaenoic acid8T3V-FFA1-Docosa-4,7,10,13,16,19-Hexaenoic acid-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Single8U4SREGN7663-Fab8U4S-CXCR4-REGN7663-Fab
9.09Single8U4TREGN7663-Fab8U4T-CXCR4-REGN7663-Fab
9.09Single8U8FPalmitic Acid8U8F-GPR3-Palmitic Acid-Gs/β1/γ2
9.09Consensus5ht2_on_gpOrthosteric Ligand5ht2b_on_gp
9.09Consensus5ht2b_on_gpOrthosteric Ligand7SRR-5-HT2B-LSD-chim(NtGi2L-Gs-CtGq)/β1/γ2
9.09Consensusccr6_onOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
9.09Consensusccr6_on_gpOrthosteric Ligand6WWZ-CCR6-CCL20-Go/β1/γ2
8.82Single6FFIMMPEP6FFI-mGlu5-MMPEP
8.82Single6TPKRetosiban6TPK-OT-Retosiban
8.82Single6XBLSAG6XBL-SMO-SAG-Cholesterol-Gi1/β1/γ2
8.82Single7BB6AVP7BB6-V2-AVP-Gs/β1/γ2
8.82Single7VODCariprazine7VOD-5-HT2A-Cariprazine
8.82Single7ZI0SAG7ZI0-SMO-SAG-Cholesterol
8.82Single8HQN9-S-HODE8HQN-GPR132-9-S-HODE-Gi1/β1/γ2
8.82Single8JD6VU03647708JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
8.82Single8K4NVF08K4N-GPR34-VF0-Gi1/β1/γ2
8.82Single8YRGFospropofol8YRG-MRGPRX4-Fospropofol-chim(NtGi1-Gs-CtGq)/β1/γ2
8.82Single9DQJEP-39459DQJ-MRGPRD-EP-3945-chim(NtGi1-Gs-CtGq)/β1/γ2
8.82Single9K1DButanoic acid9K1D-FFA2-Butanoic acid-Gi1/β1/γ2
8.82Single9LRDHistamine9LRD-H1-Histamine-Gi1/β1/γ2
8.82Consensusot_offOrthosteric Ligand6TPK-OT-Retosiban
8.82Consensusvasop-oxy_offOrthosteric Ligandot_off
8.57Single6FFHFenobam6FFH-mGlu5-Fenobam
8.57Single6XBM5LWE6XBM-SMO-5LWE-Gi1/β1/γ2
8.57Single7SK8CXCL127SK8-ACKR3-CXCL12-CCX662
8.57Single8GCML9026888GCM-EP4-L902688-Gi1/β1/γ2
8.57Single8XBGS3E-LysoPS8XBG-GPR34-S3E-LysoPS
8.57Single8ZBEOctreotide8ZBE-SST5-Octreotide-Gi1/β1/γ1
8.57Single9IMATalquetamab9IMA-GPRC5D-Talquetamab
8.33Single4NTJAZD12834NTJ-P2Y12-AZD1283
8.33Single5ZBQUR-MK-2995ZBQ-Y1-UR-MK-299
8.33Single6XBKCholesterol6XBK-SMO-Cholesterol-Gi1/β1/γ2
8.33Single6Z4QSR142948A6Z4Q-NTS1-SR142948A
8.33Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
8.33Single7VV0PAMP-127VV0-MRGPRX2-PAMP-12
8.33Single7Y26Octreotide7Y26-SST2-Octreotide-chim(NtGi2L-Gs-CtGq)/β1/γ2
8.33Single8EJCTAK-8758EJC-FFA1-TAK-875-chim(NtGi1L-Gs-CtGq)/β1/γ2
8.33Single8IZ4Lysophosphatidylserine8IZ4-GPR34-Lysophosphatidylserine-Gi1/β1/γ2
8.33Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
8.33Single8T6JCDPPB8T6J-mGlu5; mGlu5-CDPPB
8.33Single8TH4AT118-L Nanobody8TH4-AT1-Losartan-AT118-L Nanobody
8.33Single9DQHEP-28259DQH-MRGPRD-EP-2825-chim(NtGi1-Gs-CtGq)/β1/γ2
8.33Single9EAHNanobody AT2099EAH-AT1-Olmesartan-Nanobody AT209
8.11Single5ZBHBMS-1938855ZBH-Y1-BMS-193885
8.11Single6Z8NSRI-98296Z8N-NTS1-SRI-9829
8.11Single7SK7CXCL127SK7-ACKR3-CXCL12-CCX662
8.11Single7XAVLanreotide7XAV-SST2-Lanreotide-Gi1/β1/γ2
8.11Single7XWONeurokinin-A7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
8.11Single8JBGNeurokinin-B8JBG-NK3-Neurokinin-B-chim(NtGi1-Gs-CtGq)/β1/γ2
8.11Single8JD5JNJ-40411813; ADX881788JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
8.11Single8XX7CXCL58XX7-CXCR2-CXCL5-Go/β1/γ2
8.11Consensusnk2_on_gpOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
8.11Consensusp2y12_onOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
7.89Single6RZ7ONO-25703666RZ7-CysLT2-ONO-2570366
7.89Single7XXI2MeSADP7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
7.89Single8DWCProenkephalin-A8DWC-MRGPRX1-Proenkephalin-A-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.89Single8H0QGastrin Releasing Peptide8H0Q-BB2-Gastrin Releasing Peptide-chim(NtGi1-Gs-CtGq)/β1/γ2
7.89Single8XWACXCL18XWA-CXCR2-CXCL1
7.89Single8XWSCXCL58XWS-CXCR2-CXCL5
7.89Single9CM3TUG-13759CM3-FFA2-TUG-1375-Compound 187-chim(NtGi1L-Gs-CtGq)/β1/γ2
7.89Consensusgi_p2yOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
7.89Consensusp2y12_on_gpOrthosteric Ligand7XXI-P2Y12-2MeSADP-Gi2/β1/γ2
7.69Single6RZ9ONO-27703726RZ9-CysLT2-ONO-2770372
7.69Single7QVMOxytocin7QVM-OT-Oxytocin-chim(NtGi1-Go-CtGq)/β1/γ2
7.69Single8XWVCXCL18XWV-CXCR2-CXCL1-Go/β1/γ2
7.69Consensuscyslt2_offOrthosteric Ligand6RZ7-CysLT2-ONO-2570366 6RZ8-CysLT2-ONO-2080365 6RZ9-CysLT2-ONO-2770372
7.69Consensusnk2_onOrthosteric Ligand7XWO-NK2-Neurokinin-A-chim(NtGi1-Gs-CtGq)/β1/γ2
7.50Single9CM7TUG-13759CM7-FFA2-TUG-1375-AZ-1729-Gi1/β1/γ2
7.32Single7VLACCL15(27-92)7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.32Single8DWGProenkephalin-A8DWG-MRGPRX1-Proenkephalin-A-ML382-chim(NtGi2L-Gs-CtGq)/β1/γ2
7.32Consensusccr1_onOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.32Consensusccr1_on_gpOrthosteric Ligand7VLA-CCR1-CCL15(27-92)-Gi1/β1/γ2
7.14Single8K6OPro-neuropeptide-Y8K6O-Y1-Pro-neuropeptide-Y-Gi2/β1/γ1
6.90Single4A4MAll-trans-Retinal4A4M-Rhodopsin-All-trans-Retinal-Gt(CT)
6.90Single5EN0All-trans-Retinal5EN0-Rhodopsin-All-trans-Retinal-Gt(CT)
6.90Single5MZPCaffeine5MZP-A2A-Caffeine-Na
6.67Single7V68LY21196207V68-M4-Iperoxo-LY2119620-Gi1/β1/γ2
6.67Single7WC4Serotonin7WC4-5-HT2A-Serotonin
6.45Single6OT025(S)-Epoxycholesterol6OT0-SMO-25(S)-Epoxycholesterol-Gi1/β1/γ2
6.45Single8U4QREGN7663-Fab8U4Q-CXCR4-REGN7663-Fab-Gi1/β1/γ2
6.25Single2ZIY11-cis-Retinal2ZIY-Rhodopsin-11-cis-Retinal
6.25Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
6.25Single6PWCNeurotensin6PWC-NTS1-Neurotensin-Arrestin2
6.25Single7WC5Psilocin7WC5-5-HT2A-Psilocin
6.06Single7VDHC48/807VDH-MRGPRX2-C48/80-Gi1/β1/γ2
6.06Single8FX5Xanomeline8FX5-M4-Xanomeline-Xanomeline-Gi1/β1/γ2
6.06Single9E7RGB889E7R-PAR2-GB88-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.88Single4K5YCP-3763954K5Y-CRF1-CP-376395
5.88Single7VV5C48/807VV5-MRGPRX2-C48/80-Gi1/β1/γ2
5.88Single8XXXCXCL68XXX-CXCR2-CXCL6-Go/β1/γ2
5.71Single6ZINSR486926ZIN-NTS1-SR48692
5.71Single7VV6C48/807VV6-MRGPRX2-C48/80
5.71Single9IXXLTD49IXX-CysLT2-LTD4-chim(NtGi1-Gs-CtGq)/β1/γ2
5.56Single4Z9GCP-3763954Z9G-CRF1-CP-376395
5.56Single8GTIBMK-C2058GTI-CRF1-BMK-C205
5.56Single8TH3AT118-H Nanobody8TH3-AT1-AT118-H Nanobody
5.41Single6Z4SSR486926Z4S-NTS1-SR48692
5.41Single8GTGBMK-I1528GTG-CRF1-BMK-I152
5.41Single8JGGBAM8-228JGG-MRGPRX1-BAM8-22-Gi1/β1/γ2
5.26Single8JGFBAM8-228JGF-MRGPRX1-BAM8-22-chim(NtGi1-Gs-CtGq)/β1/γ2
5.26Single9CLWTUG-13759CLW-FFA2-TUG-1375-4-CMTB-chim(NtGi1L-Gs-CtGq)/β1/γ2
5.13Single8GTMBMK-C2038GTM-CRF1-BMK-C203
3.70Single6D32Cyclopamine6D32-SMO-Cyclopamine-Cyclopamine
3.70Single6D35Cholesterol6D35-SMO-Cholesterol
3.70Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
3.70Single6N51Quisqualate6N51-mGlu5; mGlu5-Quisqualate
3.70Single6UO8SKF975416UO8-GABAB1, GABAB2-SKF97541-GS39783
3.70Single6UO9SKF975416UO9-GABAB1, GABAB2-SKF97541
3.70Single6W2XPubChem 53110426W2X-GABAB1, GABAB2-PubChem 5311042
3.70Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
3.70Single6W2YPubChem 53110426W2Y-GABAB1; GABAB1-PubChem 5311042
3.70Single7C7QBaclofen7C7Q-GABAB1, GABAB2-Baclofen-BHFF
3.70Single7C7SCGP546267C7S-GABAB1, GABAB2-CGP54626
3.70Single7CUMCGP546267CUM-GABAB1, GABAB2-CGP54626
3.70Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.70Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.70Single7DD5Ca7DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.70Single7DD5Ca; Ca; Tryptophan; NPS-21437DD5-CaS-Ca-Ca; Ca; Tryptophan; NPS-2143
3.70Single7DGEQuisqualate7DGE-mGlu1; mGlu1-Quisqualate
3.70Single7DTTCa7DTT-CaS-Ca-Ca
3.70Single7DTTCa7DTT-CaS-Ca-Ca
3.70Single7DTUTryptophan7DTU-CaS-Tryptophan
3.70Single7DTUTryptophan7DTU-CaS-Tryptophan
3.70Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
3.70Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
3.70Single7DTVCa7DTV-CaS-Ca-Ca; Tryptophan
3.70Single7DTVCa; Tryptophan7DTV-CaS-Ca-Ca; Tryptophan
3.70Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.70Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.70Single7E6TCa7E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.70Single7E6TCa; Ca; Cyclomethyltryptophan; PO47E6T-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.70Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
3.70Single7E9GEglumetad7E9G-mGlu2; mGlu2-Eglumetad-JNJ-40411813-Gi1/β1/γ2
3.70Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
3.70Single7E9HPhosphoserine7E9H-mGlu4; mGlu4-Phosphoserine-Gi3/β1/γ2
3.70Single7EB2Baclofen7EB2-GABAB2; GABAB1-Baclofen-rac-BHFF-Gi1/β1/γ2
3.70Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
3.70Single7EPBEglumetad7EPB-mGlu2; mGlu2-Eglumetad
3.70Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
3.70Single7FD8Quisqualate7FD8-mGlu5; mGlu5-Quisqualate
3.70Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
3.70Single7FD9LY3414957FD9-mGlu5; mGlu5-LY341495
3.70Single7FIHhCG7FIH-LH-hCG-Org43553-chim(NtGi1-Gs)/β1/γ2
3.70Single7FIIhCG7FII-LH-hCG-chim(NtGi1-Gs)/β1/γ2
3.70Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.70Single7M3ECa; Ca; Tryptophan; NPS-21437M3E-CaS-Ca; Ca; Tryptophan; NPS-2143
3.70Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
3.70Single7M3FCa; Ca; Tryptophan; Cinacalcet; PO47M3F-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4
3.70Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.70Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.70Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.70Single7M3GCa; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO47M3G-CaS-Ca; Ca; Tryptophan; Evocalcet; Etelcalcetide; PO4
3.70Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
3.70Single7MTQLY3414957MTQ-mGlu2; mGlu2-LY341495
3.70Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
3.70Single7MTRGlutamate7MTR-mGlu2; mGlu2-Glutamate-ADX55164
3.70Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
3.70Single7MTSGlutamate7MTS-mGlu2; mGlu2-Glutamate-ADX55164-Gi1/β1/γ2
3.70Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.70Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.70Single7SILCa7SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.70Single7SILCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO47SIL-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4
3.70Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.70Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.70Single7SIMCa7SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.70Single7SIMCa; Ca; Cyclomethyltryptophan; PO47SIM-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; PO4
3.70Single7T9NM22 Fab7T9N-TSH-M22 Fab-DPPC-Gs/β1/γ2
3.70Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
3.70Single7WI6LY3414957WI6-mGlu3; mGlu3-LY341495
3.70Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
3.70Single7WI8LY3414957WI8-mGlu3; mGlu3-LY341495
3.70Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
3.70Single7WIHLY27941937WIH-mGlu3; mGlu3-LY2794193
3.70Single7XW6M22 Fab7XW6-TSH-M22 Fab-ML109-Gs/β1/γ2
3.70Single7XW7K1-707XW7-TSH-K1-70
3.70Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
3.70Single8JCULY3414958JCU-mGlu2; mGlu3-LY341495
3.70Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
3.70Single8JCVLY3414958JCV-mGlu2; mGlu3-LY341495
3.70Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
3.70Single8JCWLY3414958JCW-mGlu2; mGlu3-LY341495
3.70Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
3.70Single8JCXLY3414958JCX-mGlu2; mGlu3-LY341495
3.70Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
3.70Single8JCYLY3414958JCY-mGlu2; mGlu3-LY341495
3.70Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
3.70Single8JCZLY3414958JCZ-mGlu2; mGlu3-LY341495
3.70Single8JD0Glutamate8JD0-mGlu2; mGlu3-Glutamate-NAM563
3.70Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
3.70Single8JD1Glutamate8JD1-mGlu2; mGlu3-Glutamate
3.70Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
3.70Single8JD2Glutamate8JD2-mGlu2; mGlu3-Glutamate
3.70Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
3.70Single8JD3Glutamate8JD3-mGlu2; mGlu3-Glutamate-JNJ-40411813-Gi1/β1/γ2
3.70Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
3.70Single8JD4Glutamate8JD4-mGlu2; mGlu4-Glutamate
3.70Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.70Single8JD5Glutamate8JD5-mGlu2; mGlu4-Glutamate-JNJ-40411813; ADX88178-Gi1/β1/γ2
3.70Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.70Single8JD6Phosphoserine8JD6-mGlu4; mGlu4-Phosphoserine-VU0364770-Gi3/β1/γ2
3.70Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.70Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.70Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
3.70Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
3.70Single8T7HQuisqualate8T7H-mGlu5; mGlu5-Quisqualate
3.70Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
3.70Single8T8MQuisqualate8T8M-mGlu5; mGlu5-Quisqualate
3.70Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.70Single8TAOQuisqualate8TAO-mGlu5; mGlu5-Quisqualate-CDPPB
3.70Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
3.70Single8TQBCa; PAM VU60233268TQB-mGlu3; mGlu3-Ca; PAM VU6023326-Ca
3.70Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
3.70Single8TR0LY3414958TR0-mGlu3; mGlu3-LY341495
3.70Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
3.70Single8TR2Ca; LY3792688TR2-mGlu3; mGlu3-Ca; LY379268-Ca
3.70Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
3.70Single8TRCLY3414958TRC-mGlu3; mGlu3-LY341495
3.70Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
3.70Single8TRDLY3414958TRD-mGlu3; mGlu3-LY341495
3.70Single8WG9(2S)-2-amino-4-phosphonobutanoic acid8WG9-mGlu4; mGlu2-(2S)-2-amino-4-phosphonobutanoic acid
3.70Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
3.70Single8WGBGlutammate8WGB-mGlu4; mGlu2-Glutammate-VU0155041-Gi3/β1/γ2
3.70Single8WGCLY3792688WGC-mGlu4; mGlu2-LY379268
3.70Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
3.70Single8WGDWAG; WA68WGD-mGlu4; mGlu2-WAG; WA6
3.70Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.70Single8WPGTryptophan; Cinacalcet; PO4; Ca8WPG-CaS-Tryptophan; Cinacalcet; PO4; Ca
3.70Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single8WPUTryptophan; Cinacalcet; PO4; Ca8WPU-CaS-Tryptophan; Cinacalcet; PO4; Ca-chim(NtGi2L-Gs-CtGq)/β1/γ2
3.70Single8WVXNorrin8WVX-LGR4-Norrin
3.70Single8WVYNorrin8WVY-LGR4-Norrin
3.70Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.70Single8X0BQuisqualate8X0B-mGlu5; mGlu5-Quisqualate-VU0424465
3.70Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.70Single8X0CQuisqualate8X0C-mGlu5; mGlu5-Quisqualate-VU0424465
3.70Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.70Single8X0DQuisqualate8X0D-mGlu5; mGlu5-Quisqualate-VU0424465
3.70Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
3.70Single8X0EQuisqualate8X0E-mGlu5; mGlu5-Quisqualate
3.70Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.70Single8X0FQuisqualate8X0F-mGlu5; mGlu5-Quisqualate-VU0424465
3.70Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
3.70Single8X0GQuisqualate8X0G-mGlu5; mGlu5-Quisqualate
3.70Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
3.70Single8X0HQuisqualate8X0H-mGlu5; mGlu5-Quisqualate
3.70Single8XUMR-spondin-28XUM-LGR4-R-spondin-2
3.70Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.70Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.70Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.70Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.70Single9AVLCa9AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.70Single9AVLCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVL-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi3/β2/γ2
3.70Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single9AXFCa9AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single9AXFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AXF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.70Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.70Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.70Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.70Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.70Single9C1PCa9C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.70Single9C1PCa; Tryptophan; '6218; PO49C1P-CaS-Ca-Ca; Tryptophan; '6218; PO4
3.70Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.70Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.70Single9C2FCa9C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.70Single9C2FCa; Ca; Tryptophan; '54149; PO49C2F-CaS-Ca-Ca; Ca; Tryptophan; '54149; PO4
3.70Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
3.70Single9II2Glutamate9II2-mGlu3; mGlu3-Glutamate-Arrestin2
3.70Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
3.70Single9II3Glutamate9II3-mGlu3; mGlu3-Glutamate-Arrestin2
3.70Single9KHHNorrin9KHH-LGR4-Norrin
3.70Single9S37NB219S37-LGR4-NB21
3.70Single9UTBSucralose9UTB-TAS1R2; TAS1R3-Sucralose
3.57Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.57Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.57Single7DD6Ca7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.57Single7DD6Ca; Ca; Tryptophan7DD6-CaS-Ca-Ca; Ca; Tryptophan
3.57Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.57Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.57Single7DD7Ca7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.57Single7DD7Ca; Ca; Tryptophan; Evocalcet7DD7-CaS-Ca-Ca; Ca; Tryptophan; Evocalcet
3.57Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.57Single8SZFCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZF-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine
3.57Single9ASBCa9ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9ASBCa; Ca; Cyclomethyltryptophan; 9IG; PO49ASB-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs-CtGq)/β1/γ2
3.57Single9AVGCa9AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.57Single9AVGCa; Ca; Cyclomethyltryptophan; 9IG; PO49AVG-CaS-Ca-Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-chim(NtGi1-Gs)/β1/γ2
3.57Single9AYFCa9AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.57Single9AYFCa; Ca; Ca; Cyclomethyltryptophan; 9IG; PO49AYF-CaS-Ca-Ca; Ca; Ca; Cyclomethyltryptophan; 9IG; PO4-Gi1/β1/γ2
3.57Consensusclass-b2_onOrthosteric Ligandadgrg_on adgrf_on adgrl_on adgre_on adgrd_on
3.57Consensusclass-b2_on_gpOrthosteric Ligandadgrg_on_gp adgrf_on_gp adgrl_on_gp adgre_on_gp adgrd_on_gp
3.45Single7KNUCalcitonin gene-related peptide-17KNU-CT Like-Calcitonin gene-related peptide-1-RAMP1
3.45Single7T9MCS-17 Antibody7T9M-TSH-CS-17 Antibody
3.45Single8SZGCa; Ca; Tryptophan; Cinacalcet; PO4; Spermine8SZG-CaS-Ca; Ca; Tryptophan; Cinacalcet; PO4; Spermine-chim(NtGi1-Gq)/β1/γ2
3.45Single8TLMAnti-murine CCR8 antibody8TLM-CCR8-Anti-murine CCR8 antibody
3.33Single6O3CCholesterol6O3C-SMO-SAG21k-Cholesterol
3.33Single7FIGhCG7FIG-LH-hCG-chim(NtGi1L-Gs)/β1/γ2
3.33Single7UTZTR14027UTZ-TSH-TR1402-DPPC-Gs/β1/γ2
3.33Single7XW5TSH7XW5-TSH-TSH-ML109-Gs/β1/γ2
3.33Single7ZI0Cholesterol7ZI0-SMO-SAG-Cholesterol
3.23Single5L7DCholesterol5L7D-SMO-Cholesterol
3.23Single6VCBLSN31604406VCB-GLP-1-GLP-1-LSN3160440-Gs/β1/γ2
3.23Single7T9ITSH7T9I-TSH-TSH-Gs/β1/γ2
3.23Single8I2GGlycoprotein hormones alpha chain8I2G-FSH-Glycoprotein hormones α chain-Compound 716340-Gs/β1/γ2
3.12Single7VDMSubstance-P7VDM-MRGPRX2-Substance-P-Gi1/β1/γ2
3.12Single9IVMLSN33188399IVM-GLP-1-GLP-1 (Truncated)-LSN3318839-chim(NtGi1-Gs)/β2/γ2
3.03Single7V6APubChem 98642757V6A-M4-PubChem 9864275-Gi1/β1/γ2
3.03Single8J6QCompound 9n8J6Q-HCA2-β-Hydroxybutyrate-Compound 9n-Gi1/β1/γ2
3.03Single8JPSCCL78JPS-ACKR1-CCL7
2.94Single7S8NR-Zinc-35737S8N-MRGPRX2-R-Zinc-3573-chim(NtGi2L-Gs-CtGq)/β1/γ2
2.94Single7S8OR-Zinc-35737S8O-MRGPRX2-R-Zinc-3573-Gi1/β1/γ2
2.94Single7UL2SR486927UL2-NTS1-SR48692-Na
2.94Single8J6PCompound 9n8J6P-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
2.94Single8JHYCompound 9n8JHY-HCA2-Compound 9n-Gi1/β1/γ2
2.94Single8JIICompound 9n8JII-HCA2-Niacin-Compound 9n-Gi1/β1/γ2
2.94Single8ZYUNeurotensin peptide 8-138ZYU-NTS1-Neurotensin peptide 8-13-SBI-553-Arrestin2
2.94Consensusneurotensin_offOrthosteric Ligandnts1_off
2.94Consensusnts1_offOrthosteric Ligand7UL2-NTS1-SR48692-Na
2.86Single6C1QNDT95137276C1Q-C5a1-PMX53-NDT9513727
2.78Single8HJ5PubChem 1390305318HJ5-MRGPRX1-PubChem 139030531-chim(NtGi1-Gs-CtGq)/β1/γ2
2.78Single8IYXYL-3658IYX-GPR34-YL-365
2.44Single9JH5C16:0 Ceramide9JH5-CysLT2-C16:0 Ceramide-chim(NtGi1-Gs-CtGq)/β1/γ2
2.33Single8XFTR-spondin-28XFT-LGR4-R-spondin-2-ZNRF3
2.33Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.22Single8WVUR-spondin-18WVU-LGR4-R-spondin-1-RNF43
2.22Single8Y69R-spondin-28Y69-LGR4-R-spondin-2-ZNRF3
2.17Single8XFPR-spondin-28XFP-LGR4-R-spondin-2-ZNRF3
2.04Single8XFSR-spondin-28XFS-LGR4-R-spondin-2-ZNRF3

Consensus Members
Id Members
crf2_on_gp 7TS0-CRF2-Urocortin-chim(NtGi1L-Go)/β1/γ2
crf1_on_gp 6PB0-CRF1-Urocortin-chim(NtGi1-Gs)/β1/γ2
6P9X-CRF1-Corticoliberin-Gs/β1/γ2
Net Summary
Imin 2.8875
Number of Linked Nodes 877
Number of Links 1055
Number of Hubs 169
Number of Links mediated by Hubs 653
Number of Communities 23
Number of Nodes involved in Communities 212
Number of Links involved in Communities 318
Path Summary
Number Of Nodes in MetaPath 100
Number Of Links MetaPath 99
Number of Shortest Paths 943327
Length Of Smallest Path 3
Average Path Length 30.4928
Length of Longest Path 68
Minimum Path Strength 0.34375
Average Path Strength 5.52709
Maximum Path Strength 22.4013
Minimum Path Correlation 0.7
Average Path Correlation 0.972227
Maximum Path Correlation 1
Minimum % Of Corr. Nodes 1.75439
Average % Of Corr. Nodes 42.9042
Maximum % Of Corr. Nodes 100
Minimum Path Hubs % 0
Average Path Hubs % 50.0668
Maximum Path Hubs % 100

Details about the values in these tables can be found in the corresponding documentation page .

This network is also present in following consensuses:
IdComponents
class-b1_on_gpglucagon_on_gp
vip-pacap_on_gp
pth_on_gp
crf_on_gp
calcitonin_on_gp



You can download a compressed (zip) file with structure(s), 3D outputs (as PyMol and VMD scripts) and numerical data files (as csv and plain text files).

Download crf_on_gp.zip



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